Target Pair Drug Name
EGFR3 --- HER2 N-[4-(4-Benzyloxy-3-chloro-phenylamino)-3-cyano-7-ethoxy-quinolin-6-yl]-2-dimethylaminomethyl-acrylamide Drug Info
PI3K gamma --- PI3K delta CHEMBL1645108 Drug Info
VEGFR2 --- VEGFR1 N-(3,4-dimethoxyphenyl)-1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazole-5-carboxamide Drug Info
H3 --- SERT 4-(3,4-dichlorophenyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine Drug Info
EGFR3 --- HER2 N-[4-(3-Chloro-4-fluoro-phenylamino)-quinazolin-6-yl]-acrylamide Drug Info
PI3K gamma --- PI3K delta (R)-2-(3-benzylmorpholino)-5,5-dimethyl-5,6-dihydrobenzo[d]thiazol-7(4H)-one Drug Info
VEGFR2 --- VEGFR1 N-(3,4-dichlorophenyl)-1-methyl-4-(pyridin-4-ylmethylamino)-1H-pyrazole-5-carboxamide Drug Info
H3 --- SERT 4-(7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinolin-4-yl)benzonitrile Drug Info
EGFR3 --- HER2 4-(3-bromophenylamino)-6,7-dihydroxyquinoline-3-carbonitrile Drug Info
PI3K gamma --- PI3K delta 6,6-dimethyl-2-(6-phenyl-2,3-dihydrobenzo[b][1,4]oxazin-4-yl)-6,7-dihydrothiazolo[5,4-c]pyridin-4(5H)-one Drug Info
VEGFR2 --- VEGFR1 N-(4-isopropylphenyl)-4-(2-(isoxazol-4-yl)ethyl)thiazole-5-carboxamide Drug Info
H3 --- SERT N-ethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine Drug Info
EGFR3 --- HER2 3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6-methylpyrimidin-5-yl)-2-fluoro-N-(2-(pyrrolidin-1-yl)ethyl)acrylamide Drug Info
PKCA --- NPKC delta 2-{2,6-Dihydroxy-4-[(3R,4R)-2-(4-hydroxy-benzoylamino)-cyclopentyloxymethyl]-benzoyl}-3-hydroxy-benzoic acid Drug Info
VEGFR2 --- VEGFR1 2-(1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl)-N-(pyridin-4-ylmethyl)aniline Drug Info
HDAC1 --- HD6 (S)-benzyl 1-(2-(4-methoxyphenyl)thiazol-4-yl)-5-(sulfamoylamino)pentylcarbamate Drug Info
EGFR3 --- HER2 N-(4-(o-tolylamino)quinazolin-6-yl)acrylamide Drug Info
PKCA --- NPKC delta 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3R,4R)-3-(4-hydroxy-benzoylamino)-1-(toluene-4-sulfonyl)-azepan-4-yl ester Drug Info
VEGFR2 --- VEGFR1 1-[3-(4-Methyl-piperazin-1-yl)-propyl]-4-(3-thiophen-3-yl-pyrazolo[1,5-a]pyrimidin-6-yl)-1H-pyridin-2-one Drug Info
HDAC1 --- HD6 N-hydroxy-3-(3-(1-(2-(piperidin-1-yl)ethyl)-1H-benzo[d]imidazol-2-yl)phenyl)acrylamide Drug Info
EGFR3 --- HER2 (3R,5S)-5-((4-(3-chloro-4-(6-fluoroquinolin-4-yloxy)phenylamino)thieno[3,2-d]pyrimidin-6-yl)ethynyl)pyrrolidin-3-yl morpholine-4-carboxylate Drug Info
PKCA --- NPKC delta 4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (1R,2R)-2-(4-hydroxy-benzoylamino)-4-methanesulfonyl-cyclopentyl ester Drug Info
VEGFR2 --- VEGFR1 1-(3-Piperidin-1-yl-propyl)-3-(5-thiophen-3-yl-pyridin-3-yl)-1H-indole Drug Info
HDAC1 --- HD6 N1-hydroxy-N8-(4-((2R,4S,6R)-4-phenyl-6-((pyridin-4-ylthio)methyl)-1,3-dioxan-2-yl)phenyl)octanediamide Drug Info
EGFR3 --- HER2 CHEMBL258282 Drug Info
PKCA --- NPKCtheta 3-(5-(4-(2-hydroxy-2-methylpropanoyl)piperazin-1-yl)-2-(trifluoromethyl)phenyl)-4-(1H-indol-3-yl)-1H-pyrrole-2,5-dione Drug Info
VEGFR2 --- VEGFR1 3-Chloro-N-(2,4-dichloro-benzoyl)-4-fluoro-benzenesulfonamide Drug Info
HDAC1 --- HD6 N-hydroxy-3-(3-(1-phenyl-1H-benzo[d]imidazol-2-yl)phenyl)acrylamide Drug Info
EGFR3 --- HER2 SID85267487 Drug Info
PPAR gamma --- LXRalpha 2-(5-((3-(8-(trifluoromethyl)quinolin-4-yl)phenyl)methylamino)naphthalen-1-yl)acetic acid Drug Info
HDAC1 --- HD6 Ethyl 2-oxo-2-(4-{[(1-phenyl-methanoyl)-amino]-methyl}-phenyl)-ethyl trithiocarbonate Drug Info
EGFR3 --- HER2 N4-(3-bromophenyl)-N6-methylquinazoline-4,6-diamine Drug Info
PPAR gamma --- PPAR delta 5-methyl-2-(3-(6-methyl-1H-indol-1-ylsulfonyl)benzamido)benzoic acid Drug Info
HDAC1 --- HD6 N-hydroxy-3-(3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)acrylamide Drug Info
EGFR3 --- MCSF (6,7-Dimethyl-quinazolin-4-yl)-methyl-m-tolyl-amine; hydrochloride Drug Info
PPAR gamma --- PPAR delta (R)-3-{(S)-4-[(E)-5-(4-{5-[4-(2-Carboxy-2-ethoxy-ethyl)-phenoxy]-3-methyl-pent-3-en-1-ynyl}-phenyl)-3-methyl-pent-2-en-4-ynyloxy]-phenyl}-2-ethoxy-propionic acid Drug Info
HDAC1 --- HDAC2 N-hydroxy-7-(5-(4-methoxyphenyl)oxazol-2-yl)heptanamide Drug Info
Erbeta --- ER 4-[1-(1-Methyl-butyl)-1,7a-dihydro-pyrrolo[2,1,5-cd]indolizin-2-yl]-phenol Drug Info
PPAR gamma --- PPAR delta 3-(1-((2-(3,5-dimethoxyphenyl)-5-methyloxazol-4-yl)methyl)-1H-indol-5-yl)-2-ethoxypropanoic acid Drug Info
HDAC1 --- HDAC2 6-Methoxy-1H-indole-2-carboxylic acid (6-hydroxycarbamoyl-hexyl)-amide Drug Info
Erbeta --- ER 4-[4-(2-hexahydro-1-pyridinylethoxy)phenyl]-3-phenyl-(3S,4R)-3,4-dihydro-2H-7-chromenol Drug Info
PPAR gamma --- PPAR delta (S)-3-{4-[3,3-Bis-(4-furan-2-yl-phenyl)-allyloxy]-phenyl}-2-ethoxy-propionic acid Drug Info
HDAC1 --- HDAC2 4-(3-(3,4-Dimethoxyphenyl)propanamido)-N-hydroxybenzamide Drug Info
Erbeta --- ER (2S,3S)-3-(4-Hydroxy-phenyl)-2-[4-(2-piperidin-1-yl-ethoxy)-phenyl]-chroman-4-one Drug Info
PPAR gamma --- PPAR delta 4-{4-[3-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-propoxy]-phenyl}-butyric acid Drug Info
HDAC1 --- HDAC2 Thailandepsin B Drug Info
Erbeta --- ER 4-hydroxy-N-(4-hydroxyphenyl)-N-(3,3,3-trifluoropropyl)benzenesulfonamide Drug Info
PPAR gamma --- PPAR delta 3-{2-Methyl-4-[4-methyl-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-phenyl}-propionic acid Drug Info
HDAC1 --- HDAC4 (R)-N2-hydroxy-N5-(1-phenylethyl)thiophene-2,5-dicarboxamide Drug Info
Erbeta --- ER (3aS,4R,9bR)-2,2-difluoro-4-(4-hydroxyphenyl)-1,2,3,3a,4,9b-hexahydrocyclopenta[c]chromen-8-ol Drug Info

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