TTD_Target_ID	Target_Name	TTD_Drug_ID	Drug_Name	Drug_Highest_Status	Drug_PubchemID	Molecular_Formula	Molecular_Weight	Canonical_SMILES	Activity	Binder_Type
T71266	RAC-gamma serine/threonine-protein kinase	B4CH0F	1-(1-{[4-(3-Phenylquinoxalin-2-yl)phenyl]methyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one	Investigative	9871034	C33H29N5O	511.6	C1CN(CCC1N2C3=CC=CC=C3NC2=O)CC4=CC=C(C=C4)C5=NC6=CC=CC=C6N=C5C7=CC=CC=C7	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	B5SQ2I	1-{1-[(4-{5-[(4-Hydroxyphenyl)methyl]-6-oxo-3-phenyl-1,6-dihydropyrazin-2-yl}phenyl)methyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one	Investigative	23647019	C36H33N5O3	583.7	C1CN(CCC1N2C3=CC=CC=C3NC2=O)CC4=CC=C(C=C4)C5=C(N=C(C(=O)N5)CC6=CC=C(C=C6)O)C7=CC=CC=C7	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	B6QAR1	1-[1-({4-[7-(2-Methyl-2H-1,2,3,4-tetrazol-5-yl)-3-phenylquinoxalin-2-yl]phenyl}methyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one	Investigative	21103119	C35H31N9O	593.7	CN1N=C(N=N1)C2=CC3=C(C=C2)N=C(C(=N3)C4=CC=C(C=C4)CN5CCC(CC5)N6C7=CC=CC=C7NC6=O)C8=CC=CC=C8	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	B9CSY0	1-(1-{[4-(6-Oxo-3-phenyl-1,6-dihydropyrazin-2-yl)phenyl]methyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one	Investigative	10174144	C29H27N5O2	477.6	C1CN(CCC1N2C3=CC=CC=C3NC2=O)CC4=CC=C(C=C4)C5=C(N=CC(=O)N5)C6=CC=CC=C6	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	BB51ZY	2-(4-{[4-(2-Oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]methyl}phenyl)-3-phenylquinoxaline-6-carboxylic acid	Investigative	21103197	C34H29N5O3	555.6	C1CN(CCC1N2C3=CC=CC=C3NC2=O)CC4=CC=C(C=C4)C5=NC6=C(C=C(C=C6)C(=O)O)N=C5C7=CC=CC=C7	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	BE18UC	1-{1-[(4-{6-[(4-Hydroxyphenyl)methyl]-5-oxo-3-phenyl-4,5-dihydropyrazin-2-yl}phenyl)methyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one	Investigative	23647018	C36H33N5O3	583.7	C1CN(CCC1N2C3=CC=CC=C3NC2=O)CC4=CC=C(C=C4)C5=C(NC(=O)C(=N5)CC6=CC=C(C=C6)O)C7=CC=CC=C7	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	BIPT98	1-(1-{[4-(6-Methyl-5-oxo-3-phenyl-4,5-dihydropyrazin-2-yl)phenyl]methyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one	Investigative	10289038	C30H29N5O2	491.6	CC1=NC(=C(NC1=O)C2=CC=CC=C2)C3=CC=C(C=C3)CN4CCC(CC4)N5C6=CC=CC=C6NC5=O	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	BM2CH5	N-[[4-[2-(2-Aminopyridin-3-yl)-6-phenylimidazo[4,5-b]pyridin-3-yl]phenyl]methyl]benzamide	Investigative	58345169	C31H24N6O	496.6	C1=CC=C(C=C1)C2=CC3=C(N=C2)N(C(=N3)C4=C(N=CC=C4)N)C5=CC=C(C=C5)CNC(=O)C6=CC=CC=C6	IC50 ~ 100000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	BM4Z6O	N-[[4-[2-(2-Aminopyridin-3-yl)-6-cyclopentylimidazo[4,5-b]pyridin-3-yl]phenyl]methyl]benzamide	Investigative	58345019	C30H28N6O	488.6	C1CCC(C1)C2=CC3=C(N=C2)N(C(=N3)C4=C(N=CC=C4)N)C5=CC=C(C=C5)CNC(=O)C6=CC=CC=C6	IC50 ~ 100000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	BN78XR	1-[1-({4-[6-(2-Methyl-2H-1,2,3,4-tetrazol-5-yl)-3-phenylquinoxalin-2-yl]phenyl}methyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one	Investigative	21103111	C35H31N9O	593.7	CN1N=C(N=N1)C2=CC3=C(C=C2)N=C(C(=N3)C4=CC=CC=C4)C5=CC=C(C=C5)CN6CCC(CC6)N7C8=CC=CC=C8NC7=O	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	BP65OT	1-(1-{[4-(6-Benzyl-5-oxo-3-phenyl-4,5-dihydropyrazin-2-yl)phenyl]methyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one	Investigative	23647016	C36H33N5O2	567.7	C1CN(CCC1N2C3=CC=CC=C3NC2=O)CC4=CC=C(C=C4)C5=C(NC(=O)C(=N5)CC6=CC=CC=C6)C7=CC=CC=C7	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	BSF0J3	1-(1-{[4-(5-Oxo-3-phenyl-4,5-dihydropyrazin-2-yl)phenyl]methyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one	Investigative	10152003	C29H27N5O2	477.6	C1CN(CCC1N2C3=CC=CC=C3NC2=O)CC4=CC=C(C=C4)C5=C(NC(=O)C=N5)C6=CC=CC=C6	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	BTB2X5	1-[1-({4-[6-(Butan-2-yl)-5-oxo-3-phenyl-4,5-dihydropyrazin-2-yl]phenyl}methyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one	Investigative	10128689	C33H35N5O2	533.7	CCC(C)C1=NC(=C(NC1=O)C2=CC=CC=C2)C3=CC=C(C=C3)CN4CCC(CC4)N5C6=CC=CC=C6NC5=O	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	BU3JF8	1-[1-({4-[5-(Butan-2-yl)-6-oxo-3-phenyl-1,6-dihydropyrazin-2-yl]phenyl}methyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one	Investigative	10152760	C33H35N5O2	533.7	CCC(C)C1=NC(=C(NC1=O)C2=CC=C(C=C2)CN3CCC(CC3)N4C5=CC=CC=C5NC4=O)C6=CC=CC=C6	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	BUTQ49	1-[1-({4-[6-(2-Methylpropyl)-5-oxo-3-phenyl-4,5-dihydropyrazin-2-yl]phenyl}methyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one	Investigative	10218178	C33H35N5O2	533.7	CC(C)CC1=NC(=C(NC1=O)C2=CC=CC=C2)C3=CC=C(C=C3)CN4CCC(CC4)N5C6=CC=CC=C6NC5=O	IC50 ~ 50000 nM	Poor binder
T71266	RAC-gamma serine/threonine-protein kinase	BYHV64	2-[4-(3-Phenylquinoxalin-2-yl)phenyl]propan-2-amine	Investigative	9819282	C23H21N3	339.4	CC(C)(C1=CC=C(C=C1)C2=NC3=CC=CC=C3N=C2C4=CC=CC=C4)N	IC50 ~ 50000 nM	Poor binder