TTD_Target_ID	Target_Name	TTD_Drug_ID	Drug_Name	Drug_Highest_Status	Drug_PubchemID	Molecular_Formula	Molecular_Weight	Canonical_SMILES	Activity	Binder_Type
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B15ZRE	Butyrolactone I 3-sulfate	Investigative	24861908	C24H24O10S	504.5	CC(=CCC1=C(C=CC(=C1)C[C@@]2(C(=C(C(=O)O2)OS(=O)(=O)O)C3=CC=C(C=C3)O)C(=O)OC)O)C	IC50 ~ 100000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B1BK5M	1-(3,4-Dichlorophenyl)-4-(3,5-dihydroxybenzylidene)pyrazolidine-3,5-dione	Investigative	44592358	C16H10Cl2N2O4	365.2	C1=CC(=C(C=C1N2C(=O)/C(=C/C3=CC(=CC(=C3)O)O)/C(=O)N2)Cl)Cl	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B24QYZ	1-(3,4-Dichlorophenyl)-4-(2,4-dimethoxybenzylidene)pyrazolidine-3,5-dione	Investigative	44592356	C18H14Cl2N2O4	393.2	COC1=CC(=C(C=C1)/C=C/2\\C(=O)NN(C2=O)C3=CC(=C(C=C3)Cl)Cl)OC	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B2X9CW	2-[2-[[4-[(3-Carboxy-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)amino]-2-methyl-4-oxobutan-2-yl]amino]-2-oxoethyl]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid	Investigative	57403741	C23H26N2O6S2	490.6	CC(C)(CC(=O)NC1=C(C2=C(S1)CCC2)C(=O)O)NC(=O)CC3=C(C4=C(S3)CCC4)C(=O)O	IC50 = 88130 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B4K2DG	4-(2,3-Dichlorobenzylidene)-1-(4-methoxyphenyl)pyrazolidine-3,5-dione	Investigative	44592500	C17H12Cl2N2O3	363.2	COC1=CC=C(C=C1)N2C(=O)/C(=C/C3=C(C(=CC=C3)Cl)Cl)/C(=O)N2	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B5CI2B	(4E)-4-Benzylidene-1-(3,4-dichlorophenyl)pyrazolidine-3,5-dione	Investigative	748299	C16H10Cl2N2O2	333.2	C1=CC=C(C=C1)/C=C/2\\C(=O)NN(C2=O)C3=CC(=C(C=C3)Cl)Cl	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B5IEV7	2-(3-Methoxyphenyl)-N-[(4-methylphenyl)methyl]pyrimidin-4-amine	Investigative	44820599	C19H19N3O	305.4	CC1=CC=C(C=C1)CNC2=NC(=NC=C2)C3=CC(=CC=C3)OC	IC50 = 65400 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B61JSG	1-(6-Oxospiro[1,3,4,10b-tetrahydropyrido[2,1-a]isoindole-2,2'-1,3-dioxolane]-10-yl)-3-pyrazin-2-ylurea	Investigative	67134967	C19H19N5O4	381.4	C1CN2C(CC13OCCO3)C4=C(C2=O)C=CC=C4NC(=O)NC5=NC=CN=C5	IC50 = 93000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B6MQ2W	4-(3-Hydroxy-4-methoxybenzylidene)-1-(4-methoxyphenyl)pyrazolidine-3,5-dione	Investigative	44591835	C18H16N2O5	340.3	COC1=CC=C(C=C1)N2C(=O)/C(=C/C3=CC(=C(C=C3)OC)O)/C(=O)N2	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B7ML4P	4-(2,6-Dichlorobenzylidene)-1-(3,4-dichlorophenyl)pyrazolidine-3,5-dione	Investigative	44592360	C16H8Cl4N2O2	402.1	C1=CC(=C(C(=C1)Cl)/C=C/2\\C(=O)NN(C2=O)C3=CC(=C(C=C3)Cl)Cl)Cl	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B9ACL4	1-(3,4-Dichlorophenyl)-4-(2-methoxybenzylidene)pyrazolidine-3,5-dione	Investigative	44592293	C17H12Cl2N2O3	363.2	COC1=CC=CC=C1/C=C/2\\C(=O)NN(C2=O)C3=CC(=C(C=C3)Cl)Cl	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B9TWO6	1-(3,4-Dichlorophenyl)-4-(3-methoxybenzylidene)pyrazolidine-3,5-dione	Investigative	44592292	C17H12Cl2N2O3	363.2	COC1=CC=CC(=C1)/C=C/2\\C(=O)NN(C2=O)C3=CC(=C(C=C3)Cl)Cl	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	B9XHD0	1-(3,4-Dichlorophenyl)-4-(3-hydroxy-4-methoxybenzylidene)pyrazolidine-3,5-dione	Investigative	44592329	C17H12Cl2N2O4	379.2	COC1=C(C=C(C=C1)/C=C/2\\C(=O)NN(C2=O)C3=CC(=C(C=C3)Cl)Cl)O	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BA0JQ8	1-(3,4-Dichlorophenyl)-4-(4-hydroxy-3,5-dimethoxybenzylidene)pyrazolidine-3,5-dione	Investigative	29961826	C18H14Cl2N2O5	409.2	COC1=CC(=CC(=C1O)OC)/C=C/2\\C(=O)NN(C2=O)C3=CC(=C(C=C3)Cl)Cl	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BC52VB	1-(3,4-Dichlorophenyl)-4-(4-methoxybenzylidene)pyrazolidine-3,5-dione	Investigative	1270516	C17H12Cl2N2O3	363.2	COC1=CC=C(C=C1)/C=C/2\\C(=O)NN(C2=O)C3=CC(=C(C=C3)Cl)Cl	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BCN70Y	1-(3,4-Dichlorophenyl)-4-(2-fluorobenzylidene)pyrazolidine-3,5-dione	Investigative	44592328	C16H9Cl2FN2O2	351.2	C1=CC=C(C(=C1)/C=C/2\\C(=O)NN(C2=O)C3=CC(=C(C=C3)Cl)Cl)F	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BI62LT	1-(3,4-Dichlorophenyl)-4-(2-nitrobenzylidene)pyrazolidine-3,5-dione	Investigative	44592326	C16H9Cl2N3O4	378.2	C1=CC=C(C(=C1)/C=C/2\\C(=O)NN(C2=O)C3=CC(=C(C=C3)Cl)Cl)[N+](=O)[O-]	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BJE04N	4-(4-(3-Hydroxy-4-methoxybenzylidene)-3,5-dioxopyrazolidin-1-yl)benzonitrile	Investigative	44592496	C18H13N3O4	335.3	COC1=C(C=C(C=C1)/C=C/2\\C(=O)NN(C2=O)C3=CC=C(C=C3)C#N)O	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BK6DP9	1-(3,4-Dichlorophenyl)-4-(3,4-dimethoxybenzylidene)pyrazolidine-3,5-dione	Investigative	1350361	C18H14Cl2N2O4	393.2	COC1=C(C=C(C=C1)/C=C/2\\C(=O)NN(C2=O)C3=CC(=C(C=C3)Cl)Cl)OC	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BK9A1N	1-(6-Oxospiro[1,3,4,10b-tetrahydropyrido[2,1-a]isoindole-2,2'-1,3-dioxolane]-10-yl)-3-pyridin-2-ylurea	Investigative	67134733	C20H20N4O4	380.4	C1CN2C(CC13OCCO3)C4=C(C2=O)C=CC=C4NC(=O)NC5=CC=CC=N5	IC50 = 80000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BR3LB6	4-(2-Methoxybenzylidene)-1-(4-methoxyphenyl)pyrazolidine-3,5-dione	Investigative	44592497	C18H16N2O4	324.3	COC1=CC=C(C=C1)N2C(=O)/C(=C/C3=CC=CC=C3OC)/C(=O)N2	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BR4NY1	4-(3,5-Dihydroxybenzylidene)-1-(4-methoxyphenyl)pyrazolidine-3,5-dione	Investigative	44591834	C17H14N2O5	326.3	COC1=CC=C(C=C1)N2C(=O)/C(=C/C3=CC(=CC(=C3)O)O)/C(=O)N2	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BR76SB	(4Z)-2-Anilino-4-benzylidene-1H-imidazol-5-one	Investigative	135604653	C16H13N3O	263.29	C1=CC=C(C=C1)/C=C\\2/C(=O)NC(=N2)NC3=CC=CC=C3	IC50 ~ 100000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BRFC35	4-(2-Fluorobenzylidene)-1-(4-methoxyphenyl)pyrazolidine-3,5-dione	Investigative	44592499	C17H13FN2O3	312.29	COC1=CC=C(C=C1)N2C(=O)/C(=C/C3=CC=CC=C3F)/C(=O)N2	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BTCL04	4-(4-Hydroxy-3,5-dimethoxybenzylidene)-1-(4-methoxyphenyl)pyrazolidine-3,5-dione	Investigative	44591837	C19H18N2O6	370.4	COC1=CC=C(C=C1)N2C(=O)/C(=C/C3=CC(=C(C(=C3)OC)O)OC)/C(=O)N2	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BTG0S3	1-(4-Fluorophenyl)-4-(2-methoxybenzylidene)pyrazolidine-3,5-dione	Investigative	705248	C17H13FN2O3	312.29	COC1=CC=CC=C1/C=C/2\\C(=O)NN(C2=O)C3=CC=C(C=C3)F	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BU91PH	4-(3,5-Dimethoxybenzylidene)-1-(4-methoxyphenyl)pyrazolidine-3,5-dione	Investigative	44591833	C19H18N2O5	354.4	COC1=CC=C(C=C1)N2C(=O)/C(=C/C3=CC(=CC(=C3)OC)OC)/C(=O)N2	IC50 ~ 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BUA03Z	CID 67284258	Investigative	67284258	C17H15N5O3	337.33	C1CN2C(CC1=O)C3=C(C2=O)C=CC=C3NC(=O)NC4=NC=CN=C4	IC50 = 50000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BVI90B	Chembl4276946	Investigative	134611886	C12H11Cl2N3O	284.14	CC1=NN(C(=C1C2=CC(=C(C=C2)Cl)Cl)N)C(=O)C	IC50 ~ 100000 nM	Poor binder
T92803	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	BY1A4Q	4-(3-Methoxybenzylidene)-1-(4-methoxyphenyl)pyrazolidine-3,5-dione	Investigative	44592498	C18H16N2O4	324.3	COC1=CC=C(C=C1)N2C(=O)/C(=C/C3=CC(=CC=C3)OC)/C(=O)N2	IC50 ~ 50000 nM	Poor binder