TTD_Target_ID Target_Name TTD_Drug_ID Drug_Name Drug_Highest_Status Drug_PubchemID Molecular_Formula Molecular_Weight Canonical_SMILES Activity Binder_Type T35940 ERK activator kinase 1 BU67WQ 6-[[(3R)-Piperidin-3-yl]methoxy]-2H-isoquinolin-1-one Investigative 57652534 C15H18N2O2 258.32 C1C[C@H](CNC1)COC2=CC3=C(C=C2)C(=O)NC=C3 IC50 = 491000 nM Non binder T35940 ERK activator kinase 1 BXJ45V 3-Amino-1H-indazole-4-carbonitrile Investigative 54016394 C8H6N4 158.16 C1=CC(=C2C(=C1)NN=C2N)C#N IC50 = 300000 nM Non binder