TTD_Target_ID	Target_Name	TTD_Drug_ID	Drug_Name	Drug_Highest_Status	Drug_PubchemID	Molecular_Formula	Molecular_Weight	Canonical_SMILES	Activity	Binder_Type
T58921	Peroxisome proliferator-activated receptor gamma	D07XGR	Fenofibrate	Approved	3339	C20H21ClO4	360.8	CC(C)OC(=O)C(C)(C)OC1=CC=C(C=C1)C(=O)C2=CC=C(C=C2)Cl	EC50 = 300000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	D0J5DC	Clofibrate	Approved	2796	C12H15ClO3	242.7	CCOC(=O)C(C)(C)OC1=CC=C(C=C1)Cl	EC50 ~ 500000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B04NKM	2-[(1S)-5-[3-[4-(4,5,6,7-Tetrahydro-1,3-benzothiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110489	C27H29NO4S	463.6	C1CCC2=C(C1)N=C(S2)C3=CC=C(C=C3)OCCCOC4=CC5=C(C=C4)[C@@H](CC5)CC(=O)O	EC50 = 3467368.5 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B0I4HU	2-[(1S)-5-(3-{2-Methoxy-4-[4-(trifluoromethyl)-1,3-thiazol-2-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110487	C25H24F3NO5S	507.5	COC1=C(C=CC(=C1)C2=NC(=CS2)C(F)(F)F)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 3090295.43 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B0O1AZ	(2S)-2-[(2-Benzoylcyclohexen-1-yl)amino]-3-(4-phenylmethoxyphenyl)propanoic acid	Investigative	10527748	C29H29NO4	455.5	C1CCC(=C(C1)C(=O)C2=CC=CC=C2)N[C@@H](CC3=CC=C(C=C3)OCC4=CC=CC=C4)C(=O)O	Ki = 147570653.3 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B0S7RC	Chembl4171403	Investigative	142738569	C17H14BrNO2	344.2	C1=CC(=CC(=C1)Br)C2=CC3=C(N2)C=CC(=C3)CCC(=O)O	EC50 = 236400 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B14NRX	Methyl 2-(1-(4-chlorobenzoyl)-2-methyl-5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-1H-indol-3-yl)acetate	Investigative	54580445	C31H27ClN2O5	543	CC1=C(C2=C(N1C(=O)C3=CC=C(C=C3)Cl)C=CC(=C2)OCCC4=C(OC(=N4)C5=CC=CC=C5)C)CC(=O)OC	EC50 = 620000000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B1EWL2	2-[(1S)-5-[3-[2-Methoxy-4-(4-methyl-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110484	C25H27NO5S	453.6	CC1=CSC(=N1)C2=CC(=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O)OC	EC50 = 1047128.55 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B2GUZ8	2-(5-(2-(2-(Biphenyl-4-yl)-5-methyloxazol-4-yl)ethoxy)-1-(4-chlorobenzoyl)-2-methyl-1H-indol-3-yl)acetic acid	Investigative	54581456	C36H29ClN2O5	605.1	CC1=C(C2=C(N1C(=O)C3=CC=C(C=C3)Cl)C=CC(=C2)OCCC4=C(OC(=N4)C5=CC=C(C=C5)C6=CC=CC=C6)C)CC(=O)O	EC50 = 40000000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B31FTE	3-[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-[2-(2-phenylacetyl)anilino]propanoic acid	Investigative	10721363	C33H31N3O5	549.6	CN(CCOC1=CC=C(C=C1)CC(C(=O)O)NC2=CC=CC=C2C(=O)CC3=CC=CC=C3)C4=NC5=CC=CC=C5O4	Ki = 118032063.6 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B32PMY	2-[(1S)-5-[3-(2,4-Dimethylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110424	C22H26O4	354.4	CC1=CC(=C(C=C1)OCCCOC2=CC3=C(C=C2)[C@@H](CC3)CC(=O)O)C	EC50 = 467735.14 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B38OKU	2-[4-(3-{[(1S)-1-(Carboxymethyl)-2,3-dihydro-1H-inden-5-yl]oxy}propoxy)phenyl]-4-methyl-1,3-thiazole-5-carboxylic acid	Investigative	10434749	C25H25NO6S	467.5	CC1=C(SC(=N1)C2=CC=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O)C(=O)O	EC50 = 3235936.57 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B3D9AQ	2-[(1S)-5-[3-(4-Cyano-2-propylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110425	C24H27NO4	393.5	CCCC1=C(C=CC(=C1)C#N)OCCCOC2=CC3=C(C=C2)[C@@H](CC3)CC(=O)O	EC50 = 1778279.41 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B3FXK5	2-[(1S)-5-(3-{2-Methyl-4-[3-(trifluoromethyl)-1,2,4-thiadiazol-5-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	11755396	C24H23F3N2O4S	492.5	CC1=C(C=CC(=C1)C2=NC(=NS2)C(F)(F)F)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 6456542.29 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B4T3RV	3-[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-(2-benzoylphenoxy)propanoic acid	Investigative	10578273	C32H28N2O6	536.6	CN(CCOC1=CC=C(C=C1)CC(C(=O)O)OC2=CC=CC=C2C(=O)C3=CC=CC=C3)C4=NC5=CC=CC=C5O4	Ki = 133659551.7 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B58ARF	2-[(1S)-5-[3-[4-(1H-Indol-6-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110438	C28H27NO4	441.5	C1CC2=C([C@@H]1CC(=O)O)C=CC(=C2)OCCCOC3=CC=C(C=C3)C4=CC5=C(C=C4)C=CN5	EC50 = 1380384.26 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B5EH6P	2-[(1S)-5-[3-[4-(4,5-Dimethyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	11754345	C26H29NO5S	467.6	CC1=C(SC(=N1)C2=CC(=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O)OC)C	EC50 = 30902954.33 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B5Z4RJ	2-[4-(3-{[(1S)-1-(Carboxymethyl)-2,3-dihydro-1h-inden-5-yl]oxy}propoxy)-3-methoxyphenyl]-4-methyl-1,3-thiazole-5-carboxylic acid	Investigative	16110532	C26H27NO7S	497.6	CC1=C(SC(=N1)C2=CC(=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O)OC)C(=O)O	EC50 = 1000000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B69OPB	2-[(1S)-5-[3-[4-(4-Ethyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10254028	C26H29NO5S	467.6	CCC1=CSC(=N1)C2=CC(=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O)OC	EC50 = 15488166.19 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B6YWA3	3-[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-[(9,10-dioxoanthracen-1-yl)amino]propanoic acid	Investigative	10578809	C33H27N3O6	561.6	CN(CCOC1=CC=C(C=C1)CC(C(=O)O)NC2=CC=CC3=C2C(=O)C4=CC=CC=C4C3=O)C5=NC6=CC=CC=C6O5	Ki = 120781383.5 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B74YCS	2-[(1S)-5-[3-[2-Propyl-4-(trifluoromethyl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic Acid	Investigative	10455681	C24H27F3O4	436.5	CCCC1=C(C=CC(=C1)C(F)(F)F)OCCCOC2=CC3=C(C=C2)[C@@H](CC3)CC(=O)O	EC50 = 3311311.21 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B78JHL	(2S)-2-(2-Benzoylanilino)-3-[4-[(6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydrochromen-2-yl)methoxy]phenyl]propanoic acid	Investigative	10745789	C36H37NO6	579.7	CC1=C(C2=C(CCC(O2)(C)COC3=CC=C(C=C3)C[C@@H](C(=O)O)NC4=CC=CC=C4C(=O)C5=CC=CC=C5)C(=C1O)C)C	Ki = 120781383.5 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B7CY2E	1-[4-[2-(Benzenesulfonamido)ethyl]phenyl]sulfonyl-3-(4-methoxyphenyl)thiourea	Investigative	44565167	C22H23N3O5S3	505.6	COC1=CC=C(C=C1)NC(=S)NS(=O)(=O)C2=CC=C(C=C2)CCNS(=O)(=O)C3=CC=CC=C3	IC50 = 1000000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B7EIO6	2-[(1S)-5-{3-[4-(Pyridin-3-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110439	C25H25NO4	403.5	C1CC2=C([C@@H]1CC(=O)O)C=CC(=C2)OCCCOC3=CC=C(C=C3)C4=CN=CC=C4	EC50 = 1819700.86 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B7JIA6	2-[(1S)-5-[3-[2-Methoxy-4-(4-methoxy-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110534	C25H27NO6S	469.6	COC1=C(C=CC(=C1)C2=NC(=CS2)OC)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 14791083.88 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B7KFL3	(2S)-2-(4-Benzoylanilino)-3-(4-phenylmethoxyphenyl)propanoic acid	Investigative	44364361	C29H25NO4	451.5	C1=CC=C(C=C1)COC2=CC=C(C=C2)C[C@@H](C(=O)O)NC3=CC=C(C=C3)C(=O)C4=CC=CC=C4	Ki = 169824365.3 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B7N2RE	Methyl 2-(5-(2-(2-(biphenyl-4-yl)-5-methyloxazol-4-yl)ethoxy)-1-(4-chlorobenzoyl)-2-methyl-1H-indol-3-yl)acetate	Investigative	44224204	C37H31ClN2O5	619.1	CC1=C(C2=C(N1C(=O)C3=CC=C(C=C3)Cl)C=CC(=C2)OCCC4=C(OC(=N4)C5=CC=C(C=C5)C6=CC=CC=C6)C)CC(=O)OC	EC50 = 20000000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B7NJ2B	2-[(1S)-5-[3-[4-(5-Acetyl-4-methyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10074505	C27H29NO6S	495.6	CC1=C(SC(=N1)C2=CC(=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O)OC)C(=O)C	EC50 = 20417379.45 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B7O6CT	3-[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-(2-benzoylphenyl)sulfanylpropanoic acid	Investigative	10506906	C32H28N2O5S	552.6	CN(CCOC1=CC=C(C=C1)CC(C(=O)O)SC2=CC=CC=C2C(=O)C3=CC=CC=C3)C4=NC5=CC=CC=C5O4	Ki = 132129563.4 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B7QTX9	2-[(1S)-5-[3-[4-(4-Ethyl-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110485	C25H27NO4S	437.6	CCC1=CSC(=N1)C2=CC=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 1148153.62 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B7SHP9	2-[(1S)-5-{3-[4-(Pyrimidin-5-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110441	C24H24N2O4	404.5	C1CC2=C([C@@H]1CC(=O)O)C=CC(=C2)OCCCOC3=CC=C(C=C3)C4=CN=CN=C4	EC50 = 1047128.55 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B7TMD6	2-(1-(4-Chlorobenzoyl)-2-methyl-5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-1H-indol-3-yl)acetic acid	Investigative	54584409	C30H25ClN2O5	529	CC1=C(C2=C(N1C(=O)C3=CC=C(C=C3)Cl)C=CC(=C2)OCCC4=C(OC(=N4)C5=CC=CC=C5)C)CC(=O)O	EC50 = 1230000000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B7XUQ8	2-[(1S)-5-(3-{4-[5-(Trifluoromethyl)pyridin-2-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110444	C26H24F3NO4	471.5	C1CC2=C([C@@H]1CC(=O)O)C=CC(=C2)OCCCOC3=CC=C(C=C3)C4=NC=C(C=C4)C(F)(F)F	EC50 = 562341.33 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B8HK7E	2-[(1S)-5-[3-(4-Methoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110420	C21H24O5	356.4	COC1=CC=C(C=C1)OCCCOC2=CC3=C(C=C2)[C@@H](CC3)CC(=O)O	EC50 = 338844.16 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	B8PS7E	2-[(1S)-5-[3-[4-(4-Ethoxy-5-methyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10481007	C27H31NO6S	497.6	CCOC1=C(SC(=N1)C2=CC(=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O)OC)C	EC50 = 5754399.37 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BA7J5K	2-[[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]methyl]-3-(2-benzoylphenyl)propanoic acid	Investigative	10673872	C33H30N2O5	534.6	CN(CCOC1=CC=C(C=C1)CC(CC2=CC=CC=C2C(=O)C3=CC=CC=C3)C(=O)O)C4=NC5=CC=CC=C5O4	Ki = 132739445.8 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BA98XI	2-[(1S)-5-[3-(2-Propylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110516	C23H28O4	368.5	CCCC1=CC=CC=C1OCCCOC2=CC3=C(C=C2)[C@@H](CC3)CC(=O)O	EC50 = 660693.45 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BBE54U	2-[(1S)-5-[3-(2-Ethoxy-4-methylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110518	C23H28O5	384.5	CCOC1=C(C=CC(=C1)C)OCCCOC2=CC3=C(C=C2)[C@@H](CC3)CC(=O)O	EC50 = 812830.52 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BCBO93	2-[(1S)-5-[3-[4-(2,4-Dimethoxypyrimidin-5-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110442	C26H28N2O6	464.5	COC1=NC(=NC=C1C2=CC=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O)OC	EC50 = 3388441.56 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BD90WK	2-[(1S)-5-[3-(2-Methoxy-4-methylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110426	C22H26O5	370.4	CC1=CC(=C(C=C1)OCCCOC2=CC3=C(C=C2)[C@@H](CC3)CC(=O)O)OC	EC50 = 602559.59 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BDC2J3	3-(((6-((5-Cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid	Investigative	49862248	C28H22Cl2F3N3O4	592.4	CN(CC1=CC(=CC=C1)C(=O)O)C2=C(N=C(C=C2)OCC3=C(ON=C3C4=C(C=CC=C4Cl)Cl)C5CC5)C(F)(F)F	EC50 = 1450000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BDLO05	2-[(1S)-5-[3-[4-(4-Ethoxy-5-ethyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110535	C28H33NO6S	511.6	CCC1=C(N=C(S1)C2=CC(=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O)OC)OCC	EC50 = 5623413.25 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BDPT96	2-[(1S)-5-[3-[4-(4-Ethoxy-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110493	C25H27NO5S	453.6	CCOC1=CSC(=N1)C2=CC=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 1348962.88 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BE47UQ	(2S)-2-(2-Benzoylanilino)-3-[4-[(1-methylcyclohexyl)methoxy]phenyl]propanoic acid	Investigative	10624243	C30H33NO4	471.6	CC1(CCCCC1)COC2=CC=C(C=C2)C[C@@H](C(=O)O)NC3=CC=CC=C3C(=O)C4=CC=CC=C4	Ki = 137404197.5 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BE7OH8	2-[(1S)-5-(3-{2-Methoxy-4-[4-(propan-2-yloxy)-1,3-thiazol-2-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10323599	C27H31NO6S	497.6	CC(C)OC1=CSC(=N1)C2=CC(=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O)OC	EC50 = 22908676.53 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BGC5Q1	(2S)-2-(2-Benzoylanilino)-3-(4-phenylmethoxyphenyl)propanoic acid	Investigative	44364575	C29H25NO4	451.5	C1=CC=C(C=C1)COC2=CC=C(C=C2)C[C@@H](C(=O)O)NC3=CC=CC=C3C(=O)C4=CC=CC=C4	Ki = 164058977.3 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BGNF12	2-[(1S)-5-[3-[4-(4-Tert-butyl-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	11755968	C30H37NO4S	507.7	CCCC1=C(C=CC(=C1)C2=NC(=CS2)C(C)(C)C)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 56234132.52 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BHIX30	2-[(1S)-5-[3-(4-Ethyl-2-methoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110517	C23H28O5	384.5	CCC1=CC(=C(C=C1)OCCCOC2=CC3=C(C=C2)[C@@H](CC3)CC(=O)O)OC	EC50 = 616595 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BI9UC7	2-[(1S)-5-[3-[4-(1,3-Benzothiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10005763	C28H27NO5S	489.6	COC1=C(C=CC(=C1)C2=NC3=CC=CC=C3S2)OCCCOC4=CC5=C(C=C4)[C@@H](CC5)CC(=O)O	EC50 = 4677351.41 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BIC8Y1	2-[(1S)-5-[3-[4-(4-Methoxypyridin-3-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110440	C26H27NO5	433.5	COC1=C(C=NC=C1)C2=CC=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 2089296.13 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BIVQ15	2-[(1S)-5-[3-[4-(Furan-3-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110437	C24H24O5	392.4	C1CC2=C([C@@H]1CC(=O)O)C=CC(=C2)OCCCOC3=CC=C(C=C3)C4=COC=C4	EC50 = 245470.89 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BIY15P	3-(2,3,10,11-Tetramethoxy-1,4-dihydroisoquinolino[2,1-b]isoquinolin-7-ium-8-yl)propanoic acid	Investigative	53249102	C24H26NO6+	424.5	COC1=C(CC2=C(C1)C=C[N+]3=C2C=C4C=C(C(=CC4=C3CCC(=O)O)OC)OC)OC	EC50 = 220000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BJH76Q	(S)-3-[4-[2-[Methyl(benzoxazol-2-yl)amino]ethoxy]phenyl]-2-[(2-benzoylphenyl)amino]propionic acid	Investigative	10186986	C32H29N3O5	535.6	CN(CCOC1=CC=C(C=C1)C[C@@H](C(=O)O)NC2=CC=CC=C2C(=O)C3=CC=CC=C3)C4=NC5=CC=CC=C5O4	Ki = 112201845.4 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BK8E6C	2-[(1S)-5-[3-[4-(4,5-Dimethyl-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10003213	C25H27NO4S	437.6	CC1=C(SC(=N1)C2=CC=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O)C	EC50 = 3630780.55 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BKJ69N	2-[(1S)-5-[3-(4-{4H,5H,6H-Cyclopenta[d][1,3]thiazol-2-yl}-2-methoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10457843	C27H29NO5S	479.6	COC1=C(C=CC(=C1)C2=NC3=C(S2)CCC3)OCCCOC4=CC5=C(C=C4)[C@@H](CC5)CC(=O)O	EC50 = 8709635.9 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BKY9R0	2-[(1S)-5-[3-[2-Methoxy-4-(1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110483	C24H25NO5S	439.5	COC1=C(C=CC(=C1)C2=NC=CS2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 2691534.8 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BMS79G	2-(4-(Benzyloxy)-2-(2,6-dichlorophenylamino)phenyl)acetic acid	Investigative	54582468	C21H17Cl2NO3	402.3	C1=CC=C(C=C1)COC2=CC(=C(C=C2)CC(=O)O)NC3=C(C=CC=C3Cl)Cl	EC50 = 6030000000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BO07WK	2-[(1S)-5-[3-[4-(4-Ethoxy-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10480923	C28H33NO5S	495.6	CCCC1=C(C=CC(=C1)C2=NC(=CS2)OCC)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 24547089.16 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BO1D7R	(2S)-2-(2-Benzoylanilino)-3-[4-[2-(5-ethylpyridin-2-yl)ethoxy]phenyl]propanoic acid	Investigative	10648889	C31H30N2O4	494.6	CCC1=CN=C(C=C1)CCOC2=CC=C(C=C2)C[C@@H](C(=O)O)NC3=CC=CC=C3C(=O)C4=CC=CC=C4	Ki = 122179966 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BO25AD	2-[(1S)-5-(3-{2-Propyl-4-[4-(trifluoromethyl)-1,3-thiazol-2-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10075336	C27H28F3NO4S	519.6	CCCC1=C(C=CC(=C1)C2=NC(=CS2)C(F)(F)F)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 18197008.59 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BP8QR6	2-[(1S)-5-(3-{4-[5-(Dimethylcarbamoyl)-4-methyl-1,3-thiazol-2-yl]-2-propylphenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10347115	C30H36N2O5S	536.7	CCCC1=C(C=CC(=C1)C2=NC(=C(S2)C(=O)N(C)C)C)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 50118723.36 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BPC9I7	2-[2-(Benzenesulfonyl)anilino]-3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]propanoic acid	Investigative	10626890	C31H29N3O6S	571.6	CN(CCOC1=CC=C(C=C1)CC(C(=O)O)NC2=CC=CC=C2S(=O)(=O)C3=CC=CC=C3)C4=NC5=CC=CC=C5O4	Ki = 147570653.3 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BPOD17	2-[(1S)-5-[3-[4-(4-Methoxy-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic Acid	Investigative	10455871	C24H25NO5S	439.5	COC1=CSC(=N1)C2=CC=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 3388441.56 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BPZ3Y7	2-[(1S)-5-[3-(4-{4H,5H,6H-Cyclopenta[d][1,3]thiazol-2-yl}-2-propylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10323352	C29H33NO4S	491.6	CCCC1=C(C=CC(=C1)C2=NC3=C(S2)CCC3)OCCCOC4=CC5=C(C=C4)[C@@H](CC5)CC(=O)O	EC50 = 10715193.05 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BQB0F8	(2S)-3-[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-(2-phenoxyanilino)propanoic acid	Investigative	54584463	C31H29N3O5	523.6	CN(CCOC1=CC=C(C=C1)C[C@@H](C(=O)O)NC2=CC=CC=C2OC3=CC=CC=C3)C4=NC5=CC=CC=C5O4	Ki = 118850222.7 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BS6A1U	2-[(1S)-5-[3-(4-Ethoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110421	C22H26O5	370.4	CCOC1=CC=C(C=C1)OCCCOC2=CC3=C(C=C2)[C@@H](CC3)CC(=O)O	EC50 = 1071519.31 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BS71JU	2-[(1S)-5-[3-[4-(5-Acetyl-4-methyl-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10074964	C29H33NO5S	507.6	CCCC1=C(C=CC(=C1)C2=NC(=C(S2)C(=O)C)C)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 58884365.54 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BS86NI	2-[(1S)-5-(3-{4-[4-(Propan-2-yloxy)-1,3-thiazol-2-yl]-2-propylphenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110494	C29H35NO5S	509.7	CCCC1=C(C=CC(=C1)C2=NC(=CS2)OC(C)C)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 22387211.39 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BTOS83	2-[(1S)-5-{3-[4-(6-Methylpyridin-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110443	C26H27NO4	417.5	CC1=NC(=CC=C1)C2=CC=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 1819700.86 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BUVM01	2-[(1S)-5-[3-[4-(4-Ethoxy-5-methyl-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10075041	C29H35NO5S	509.7	CCCC1=C(C=CC(=C1)C2=NC(=C(S2)C)OCC)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 29512092.27 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BWCG72	2-[N-(2-Phenylmethoxyethyl)-4-[(2,4,6-trioxo-1,3-diazinan-5-ylidene)methyl]anilino]ethyl acetate	Investigative	127036555	C24H25N3O6	451.5	CC(=O)OCCN(CCOCC1=CC=CC=C1)C2=CC=C(C=C2)C=C3C(=O)NC(=O)NC3=O	IC50 > 200000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BWG96H	3-[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-[(9-oxofluoren-1-yl)amino]propanoic acid	Investigative	10816129	C32H27N3O5	533.6	CN(CCOC1=CC=C(C=C1)CC(C(=O)O)NC2=CC=CC3=C2C(=O)C4=CC=CC=C34)C5=NC6=CC=CC=C6O5	Ki = 141579378 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BX1F6B	2-[4-(3-{[(1S)-1-(Carboxymethyl)-2,3-dihydro-1h-inden-5-yl]oxy}propoxy)-3-propylphenyl]-4-(hydroxymethyl)-1,3-thiazole-5-carboxylic acid	Investigative	16110492	C28H31NO7S	525.6	CCCC1=C(C=CC(=C1)C2=NC(=C(S2)C(=O)O)CO)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 1148153.62 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BX2JF1	2-[(1S)-5-[3-[4-(5-Acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110525	C26H27NO5S	465.6	CC1=C(SC(=N1)C2=CC=C(C=C2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O)C(=O)C	EC50 = 2089296.13 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BX4Y2N	2-[(1S)-5-{3-[4-(Thiophen-3-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110436	C24H24O4S	408.5	C1CC2=C([C@@H]1CC(=O)O)C=CC(=C2)OCCCOC3=CC=C(C=C3)C4=CSC=C4	EC50 = 1548816.62 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BXC67Q	2-[(1S)-5-[3-(2-Methoxy-4-{5H,6H,7H-pyrano[2,3-d][1,3]thiazol-2-yl}phenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110524	C27H29NO6S	495.6	COC1=C(C=CC(=C1)C2=NC3=C(S2)CCCO3)OCCCOC4=CC5=C(C=C4)[C@@H](CC5)CC(=O)O	EC50 = 5623413.25 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BY0AD5	2-[(1S)-5-[3-(4-Cyano-2-methoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110427	C22H23NO5	381.4	COC1=C(C=CC(=C1)C#N)OCCCOC2=CC3=C(C=C2)[C@@H](CC3)CC(=O)O	EC50 = 1445439.77 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BY13US	2-[(1S)-5-[3-[4-(Trifluoromethoxy)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110512	C21H21F3O5	410.4	C1CC2=C([C@@H]1CC(=O)O)C=CC(=C2)OCCCOC3=CC=C(C=C3)OC(F)(F)F	EC50 = 1000000 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BY3LJ8	((1S)-5-{3-[4-(4-Ethyl-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl)acetic acid	Investigative	16110486	C28H33NO4S	479.6	CCCC1=C(C=CC(=C1)C2=NC(=CS2)CC)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 22387211.39 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BY8OL9	2-[(1S)-5-[3-(2-Propyl-4-{5H,6H,7H-pyrano[2,3-d][1,3]thiazol-2-yl}phenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110490	C29H33NO5S	507.6	CCCC1=C(C=CC(=C1)C2=NC3=C(S2)CCCO3)OCCCOC4=CC5=C(C=C4)[C@@H](CC5)CC(=O)O	EC50 = 23988329.19 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BY9RN8	2-[(1S)-5-{3-[4-(1H-1,2,4-Triazol-1-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110428	C22H23N3O4	393.4	C1CC2=C([C@@H]1CC(=O)O)C=CC(=C2)OCCCOC3=CC=C(C=C3)N4C=NC=N4	EC50 = 1819700.86 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BZ1I8H	2-[(1S)-5-[3-[2-Methoxy-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10368444	C28H31NO5S	493.6	COC1=C(C=CC(=C1)C2=NC3=C(S2)CCCC3)OCCCOC4=CC5=C(C=C4)[C@@H](CC5)CC(=O)O	EC50 = 12022644.35 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BZ2M3K	2-[4-(3-{[(1S)-1-(Carboxymethyl)-2,3-dihydro-1H-inden-5-yl]oxy}propoxy)-3-propylphenyl]-4-methyl-1,3-thiazole-5-carboxylic acid	Investigative	10075037	C28H31NO6S	509.6	CCCC1=C(C=CC(=C1)C2=NC(=C(S2)C(=O)O)C)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 4265795.19 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BZ3X9L	2-[(1S)-5-[3-[2-Propyl-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	10458842	C30H35NO4S	505.7	CCCC1=C(C=CC(=C1)C2=NC3=C(S2)CCCC3)OCCCOC4=CC5=C(C=C4)[C@@H](CC5)CC(=O)O	EC50 = 85113803.82 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	BZ82YL	2-[(1S)-5-[3-[2-Propyl-4-(1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid	Investigative	16110482	C26H29NO4S	451.6	CCCC1=C(C=CC(=C1)C2=NC=CS2)OCCCOC3=CC4=C(C=C3)[C@@H](CC4)CC(=O)O	EC50 = 20892961.31 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	D04DYM	GW1929	Investigative	6518171	C30H29N3O4	495.6	CN(CCOC1=CC=C(C=C1)C[C@@H](C(=O)O)NC2=CC=CC=C2C(=O)C3=CC=CC=C3)C4=CC=CC=N4	Ki = 113240036.3 nM	Non binder
T58921	Peroxisome proliferator-activated receptor gamma	D06RRD	Fibrates	Investigative	2797	C10H11ClO3	214.64	CC(C)(C(=O)O)OC1=CC=C(C=C1)Cl	EC50 > 300000 nM	Non binder