TTD_Target_ID Target_Name TTD_Drug_ID Drug_Name Drug_Highest_Status Drug_PubchemID Molecular_Formula Molecular_Weight Canonical_SMILES Activity Binder_Type T66665 Prostaglandin G/H synthase 2 D0KP0U PMID26394986-Compound-22 Patented 2662 C17H14F3N3O2S 381.4 CC1=CC=C(C=C1)C2=CC(=NN2C3=CC=C(C=C3)S(=O)(=O)N)C(F)(F)F IC50 = 390000 nM Non binder T66665 Prostaglandin G/H synthase 2 B0UJI7 4,6-Dimethyl-2-[3-oxo-3-(4-phenylpiperazin-1-yl)propyl]-[1,2]thiazolo[5,4-b]pyridin-3-one Investigative 134134738 C21H24N4O2S 396.5 CC1=CC(=NC2=C1C(=O)N(S2)CCC(=O)N3CCN(CC3)C4=CC=CC=C4)C IC50 = 281838.29 nM Non binder T66665 Prostaglandin G/H synthase 2 B0YKS9 N-(Cyclohexylmethyl)-2-(4-methylsulfonylphenyl)-6-(trifluoromethyl)pyrimidin-4-amine Investigative 44456666 C19H22F3N3O2S 413.5 CS(=O)(=O)C1=CC=C(C=C1)C2=NC(=CC(=N2)NCC3CCCCC3)C(F)(F)F IC50 = 675678.34 nM Non binder T66665 Prostaglandin G/H synthase 2 B1OWF8 2,3-Diphenylthiophene Investigative 2801736 C16H12S 236.3 C1=CC=C(C=C1)C2=C(SC=C2)C3=CC=CC=C3 IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 B1YWX4 1-Tert-Butyloxycarbonyl-2-bromo-4-(4-fluorophenyl)-5-(4-methylsulfonylphenyl)pyrrole Investigative 10097252 C22H21BrFNO4S 494.4 CC(C)(C)OC(=O)N1C(=CC(=C1C2=CC=C(C=C2)S(=O)(=O)C)C3=CC=C(C=C3)F)Br IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 B2ENM1 (2-Methylsulfanylphenyl) 2-bromoacetate Investigative 10563335 C9H9BrO2S 261.14 CSC1=CC=CC=C1OC(=O)CBr IC50 = 510000 nM Non binder T66665 Prostaglandin G/H synthase 2 B2LR1U N'-[(E)-(4-Oxo-4H-chromen-3-yl)methylidene]benzenecarbohydrazide Investigative 9559931 C17H12N2O3 292.29 C1=CC=C(C=C1)C(=O)N/N=C/C2=COC3=CC=CC=C3C2=O IC50 = 802320 nM Non binder T66665 Prostaglandin G/H synthase 2 B2R3UD 4-[4-(Benzylamino)-6-(trifluoromethyl)pyrimidin-2-yl]benzenesulfonamide Investigative 44456801 C18H15F3N4O2S 408.4 C1=CC=C(C=C1)CNC2=NC(=NC(=C2)C(F)(F)F)C3=CC=C(C=C3)S(=O)(=O)N IC50 = 300303.23 nM Non binder T66665 Prostaglandin G/H synthase 2 B3O7KQ 5-Chloro-3-(4-ethylphenyl)-2-[4-(methanesulfonyl)phenyl]-4H-pyran-4-one Investigative 44309929 C20H17ClO4S 388.9 CCC1=CC=C(C=C1)C2=C(OC=C(C2=O)Cl)C3=CC=C(C=C3)S(=O)(=O)C IC50 = 720111.92 nM Non binder T66665 Prostaglandin G/H synthase 2 B3S2QY 2-Benzyl-4''-methanesulfonyl-biphenyl Investigative 44384330 C20H18O2S 322.4 CS(=O)(=O)C1=CC=C(C=C1)C2=CC=CC=C2CC3=CC=CC=C3 IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 B3Z2MD Sodium;2-[4-[(2-oxocyclopentyl)methyl]-3-phenylphenyl]propanoate Investigative 56665210 C21H21NaO3 344.4 CC(C1=CC(=C(C=C1)CC2CCCC2=O)C3=CC=CC=C3)C(=O)[O-].[Na+] IC50 = 290000 nM Non binder T66665 Prostaglandin G/H synthase 2 B4DCG1 1-[5-Bromo-3-(4-fluorophenyl)-2-(4-methylsulfonylphenyl)pyrrol-1-yl]ethanone Investigative 10071673 C19H15BrFNO3S 436.3 CC(=O)N1C(=CC(=C1C2=CC=C(C=C2)S(=O)(=O)C)C3=CC=C(C=C3)F)Br IC50 = 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 B58HMR 4,6-Dimethyl-2-[4-oxo-4-(4-phenylpiperazin-1-yl)butyl]-[1,2]thiazolo[5,4-b]pyridin-3-one Investigative 134147676 C22H26N4O2S 410.5 CC1=CC(=NC2=C1C(=O)N(S2)CCCC(=O)N3CCN(CC3)C4=CC=CC=C4)C IC50 = 389045.14 nM Non binder T66665 Prostaglandin G/H synthase 2 B5DQG7 4-[(4,6-Dimethyl-[1,2]thiazolo[5,4-b]pyridin-3-yl)oxy]butanoic acid Investigative 134141655 C12H14N2O3S 266.32 CC1=CC(=NC2=C1C(=NS2)OCCCC(=O)O)C IC50 = 245470.89 nM Non binder T66665 Prostaglandin G/H synthase 2 B5I3RX 4-(4''-Methanesulfonyl-biphenyl-2-yl)-pyridine Investigative 44383014 C18H15NO2S 309.4 CS(=O)(=O)C1=CC=C(C=C1)C2=CC=CC=C2C3=CC=NC=C3 IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 B5JP4S Sodium;2-[2-(4-methylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate Investigative 56668670 C22H23NaO3 358.4 CC1=CC=C(C=C1)C2=C(C=CC(=C2)CC3CCCC3=O)C(C)C(=O)[O-].[Na+] IC50 = 540000 nM Non binder T66665 Prostaglandin G/H synthase 2 B5SB2E Arenarioside Investigative 44584310 C34H44O19 756.7 C[C@H]1[C@@H]([C@H]([C@H](C(O1)O[C@@H]2[C@H]([C@@H](O[C@@H]([C@H]2OC(=O)/C=C/C3=CC(=C(C=C3)O)O)CO[C@H]4[C@@H]([C@H]([C@@H](CO4)O)O)O)OCCC5=CC(=C(C=C5)O)O)O)O)O)O IC50 = 600000 nM Non binder T66665 Prostaglandin G/H synthase 2 B61BNA [2-[3-[3-Fluoro-5-(4-methoxyoxan-4-yl)phenoxy]propyl]-8-methoxy-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]-(3-fluorophenyl)methanone;hydrochloride Investigative 46906735 C34H37ClF2N2O5 627.1 COC1=CC2=C(C=C1)N(C3=C2CN(CC3)CCCOC4=CC(=CC(=C4)C5(CCOCC5)OC)F)C(=O)C6=CC(=CC=C6)F.Cl IC50 = 357200 nM Non binder T66665 Prostaglandin G/H synthase 2 B63QJT 3-(2,3-Dihydro-1,4-benzodioxin-5-yl)-2-(4-methylphenyl)sulfonyl-5-(trifluoromethyl)-3,4-dihydropyrazole Investigative 118706122 C19H17F3N2O4S 426.4 CC1=CC=C(C=C1)S(=O)(=O)N2C(CC(=N2)C(F)(F)F)C3=C4C(=CC=C3)OCCO4 IC50 > 500000 nM Non binder T66665 Prostaglandin G/H synthase 2 B6V0ZS 2-Ethoxy-6-pentadecylbenzyl 5-nitro-1H-benzimidazole-2-yl sulfide Investigative 44373312 C31H45N3O3S 539.8 CCCCCCCCCCCCCCCC1=C(C(=CC=C1)OCC)CSC2=NC3=C(N2)C=C(C=C3)[N+](=O)[O-] IC50 = 384000 nM Non binder T66665 Prostaglandin G/H synthase 2 B71LJO 2-[3-[4-(3-Chlorophenyl)piperazin-1-yl]-3-oxopropyl]-4,6-dimethyl-[1,2]thiazolo[5,4-b]pyridin-3-one Investigative 134154144 C21H23ClN4O2S 431 CC1=CC(=NC2=C1C(=O)N(S2)CCC(=O)N3CCN(CC3)C4=CC(=CC=C4)Cl)C IC50 = 295120.92 nM Non binder T66665 Prostaglandin G/H synthase 2 B79PZH 2-(4-Methylsulfonylphenyl)-N-(3-thiophen-2-ylpropyl)-6-(trifluoromethyl)pyrimidin-4-amine Investigative 76315140 C19H18F3N3O2S2 441.5 CS(=O)(=O)C1=CC=C(C=C1)C2=NC(=CC(=N2)NCCCC3=CC=CS3)C(F)(F)F IC50 = 826456.5 nM Non binder T66665 Prostaglandin G/H synthase 2 B91HQM 5-Chloro-3-(4-chlorophenyl)-2-(4-methylsulfonylphenyl)pyran-4-one Investigative 44309825 C18H12Cl2O4S 395.3 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C(=O)C(=CO2)Cl)C3=CC=C(C=C3)Cl IC50 = 936052.05 nM Non binder T66665 Prostaglandin G/H synthase 2 B93RBW Sodium;2-[2-(4-methoxyphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate Investigative 56675535 C22H23NaO4 374.4 CC(C1=C(C=C(C=C1)CC2CCCC2=O)C3=CC=C(C=C3)OC)C(=O)[O-].[Na+] IC50 = 430000 nM Non binder T66665 Prostaglandin G/H synthase 2 B9J5HW 3-(4-Methylsulfonylphenyl)-4-phenylbenzoic acid Investigative 44384436 C20H16O4S 352.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C=CC(=C2)C(=O)O)C3=CC=CC=C3 IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 B9VK4M [1-(4-Methanesulfonyl-phenyl)-2-pyridin-3-yl-1H-imidazol-4-yl]-methanol Investigative 10830211 C16H15N3O3S 329.4 CS(=O)(=O)C1=CC=C(C=C1)N2C=C(N=C2C3=CN=CC=C3)CO IC50 = 934000 nM Non binder T66665 Prostaglandin G/H synthase 2 BB78JV 2-[4-(Methylsulfonyl)phenyl]-3-(4-fluorophenyl)-5-(trifluoroacetyl)-1H-pyrrole Investigative 10431739 C19H13F4NO3S 411.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C=C(N2)C(=O)C(F)(F)F)C3=CC=C(C=C3)F IC50 = 298200 nM Non binder T66665 Prostaglandin G/H synthase 2 BDC5S7 5-Chloro-3-(4-fluorophenyl)-2-(4-methylsulfonylphenyl)pyran-4-thione Investigative 44309745 C18H12ClFO3S2 394.9 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C(=S)C(=CO2)Cl)C3=CC=C(C=C3)F IC50 = 835795.45 nM Non binder T66665 Prostaglandin G/H synthase 2 BE9TN6 4,6-Dimethyl-2-[1-oxo-1-(4-phenylpiperazin-1-yl)butan-2-yl]-[1,2]thiazolo[5,4-b]pyridin-3-one Investigative 134152691 C22H26N4O2S 410.5 CCC(C(=O)N1CCN(CC1)C2=CC=CC=C2)N3C(=O)C4=C(S3)N=C(C=C4C)C IC50 = 251188.64 nM Non binder T66665 Prostaglandin G/H synthase 2 BET3Q7 3-(4-Hydroxy-phenyl)-4-(4-methanesulfonyl-phenyl)-5H-furan-2-one Investigative 10359269 C17H14O5S 330.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C(=O)OC2)C3=CC=C(C=C3)O IC50 > 250000 nM Non binder T66665 Prostaglandin G/H synthase 2 BF5GM3 7,8-Dichloro-2-(trifluoromethyl)-2H-chromene-3-carboxylic Acid Investigative 9818254 C11H5Cl2F3O3 313.05 C1=CC(=C(C2=C1C=C(C(O2)C(F)(F)F)C(=O)O)Cl)Cl IC50 = 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 BF78TK 2-[[2-Anilinoethyl(methyl)amino]methyl]-4,6-dimethyl-[1,2]thiazolo[5,4-b]pyridin-3-one Investigative 11544686 C18H22N4OS 342.5 CC1=CC(=NC2=C1C(=O)N(S2)CN(C)CCNC3=CC=CC=C3)C IC50 = 494300 nM Non binder T66665 Prostaglandin G/H synthase 2 BG8D0L 4-(4,6-Dimethyl-3-oxo-[1,2]thiazolo[5,4-b]pyridin-2-yl)butanoic acid Investigative 134135733 C12H14N2O3S 266.32 CC1=CC(=NC2=C1C(=O)N(S2)CCCC(=O)O)C IC50 = 269153.48 nM Non binder T66665 Prostaglandin G/H synthase 2 BHQ86P 5-Chloro-2-(4-methylsulfonylcyclohexyl)-3-(3-methylthiophen-1-ium-1-yl)pyran-4-one Investigative 53323460 C17H20ClO4S2+ 387.9 CC1=C[S+](C=C1)C2=C(OC=C(C2=O)Cl)C3CCC(CC3)S(=O)(=O)C IC50 = 736037.6 nM Non binder T66665 Prostaglandin G/H synthase 2 BJ72WC 2-(Methylthio)phenol, trifluoroacetate Investigative 10847385 C9H7F3O2S 236.21 CSC1=CC=CC=C1OC(=O)C(F)(F)F IC50 = 260000 nM Non binder T66665 Prostaglandin G/H synthase 2 BJV7O4 (2S)-2-[[(2S)-2-[[(2S)-2-[(4-Fluorobenzoyl)amino]-3-(1H-indol-3-yl)propanoyl]amino]-4-methylsulfanylbutanoyl]amino]butanedioic acid Investigative 57393171 C27H29FN4O7S 572.6 CSCC[C@@H](C(=O)N[C@@H](CC(=O)O)C(=O)O)NC(=O)[C@H](CC1=CNC2=CC=CC=C21)NC(=O)C3=CC=C(C=C3)F IC50 = 450000 nM Non binder T66665 Prostaglandin G/H synthase 2 BKCM19 2-[1-(4-Chlorobenzoyl)-2-phenylindol-3-yl]acetic acid Investigative 57393522 C23H16ClNO3 389.8 C1=CC=C(C=C1)C2=C(C3=CC=CC=C3N2C(=O)C4=CC=C(C=C4)Cl)CC(=O)O IC50 > 400000 nM Non binder T66665 Prostaglandin G/H synthase 2 BL2CU0 2-[3-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-3-oxopropyl]-4,6-dimethyl-[1,2]thiazolo[5,4-b]pyridin-3-one Investigative 134143054 C22H25N3O4S 427.5 CC1=CC(=NC2=C1C(=O)N(S2)CCC(=O)N3CCC4=CC(=C(C=C4C3)OC)OC)C IC50 = 288403.15 nM Non binder T66665 Prostaglandin G/H synthase 2 BLH4M6 2-[(4,6-Dimethyl-[1,2]thiazolo[5,4-b]pyridin-3-yl)oxy]propanoic acid Investigative 134138298 C11H12N2O3S 252.29 CC1=CC(=NC2=C1C(=NS2)OC(C)C(=O)O)C IC50 = 218776.16 nM Non binder T66665 Prostaglandin G/H synthase 2 BLKV17 4-Methyl-N''-((4-oxo-4H-chromen-3-yl)methylene)benzenesulfonohydrazide Investigative 9644405 C17H14N2O4S 342.4 CC1=CC=C(C=C1)S(=O)(=O)N/N=C/C2=COC3=CC=CC=C3C2=O IC50 = 203690 nM Non binder T66665 Prostaglandin G/H synthase 2 BM7BG4 [(2R,3R,4R,5R,6R)-2-[[(2S,3S)-3,4-Dihydroxy-4-(hydroxymethyl)oxolan-2-yl]oxymethyl]-6-[2-(3,4-dihydroxyphenyl)ethoxy]-5-hydroxy-4-[(2R,3S,4S,5S,6R)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxyoxan-3-yl] (E)-3-(3,4-dihydroxyphenyl)prop-2-enoate Investigative 44429859 C34H44O19 756.7 C[C@@H]1[C@H]([C@@H]([C@@H]([C@H](O1)O[C@@H]2[C@H]([C@@H](O[C@@H]([C@H]2OC(=O)/C=C/C3=CC(=C(C=C3)O)O)CO[C@@H]4[C@H](C(CO4)(CO)O)O)OCCC5=CC(=C(C=C5)O)O)O)O)O)O IC50 = 490000 nM Non binder T66665 Prostaglandin G/H synthase 2 BM7LQ0 Acetic acid 2-benzylsulfanyl-phenyl ester Investigative 9834940 C15H14O2S 258.3 CC(=O)OC1=CC=CC=C1SCC2=CC=CC=C2 IC50 = 250000 nM Non binder T66665 Prostaglandin G/H synthase 2 BO4DI5 (2S)-2-[[(2S)-2-[[(2S)-2-[(4-Fluorobenzoyl)amino]-3-phenylpropanoyl]amino]-4-methylsulfanylbutanoyl]amino]butanedioic acid Investigative 57391400 C25H28FN3O7S 533.6 CSCC[C@@H](C(=O)N[C@@H](CC(=O)O)C(=O)O)NC(=O)[C@H](CC1=CC=CC=C1)NC(=O)C2=CC=C(C=C2)F IC50 = 450000 nM Non binder T66665 Prostaglandin G/H synthase 2 BOA98P 3-[5-(4-Fluoro-phenyl)-4-(4-methanesulfonyl-phenyl)-thiophen-2-yl]-propionic acid Investigative 44330273 C20H17FO4S2 404.5 CS(=O)(=O)C1=CC=C(C=C1)C2=C(SC(=C2)CCC(=O)O)C3=CC=C(C=C3)F IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 BOHT35 (2S)-2-[[(2S)-2-[[(2S)-2-[(4-Fluorobenzoyl)amino]-3-(4-hydroxyphenyl)propanoyl]amino]-4-methylsulfanylbutanoyl]amino]pentanedioic acid Investigative 57400090 C26H30FN3O8S 563.6 CSCC[C@@H](C(=O)N[C@@H](CCC(=O)O)C(=O)O)NC(=O)[C@H](CC1=CC=C(C=C1)O)NC(=O)C2=CC=C(C=C2)F IC50 = 500000 nM Non binder T66665 Prostaglandin G/H synthase 2 BOM70P 2-[(4-Cyclohexylpiperazin-1-yl)methyl]-4,6-dimethyl-[1,2]thiazolo[5,4-b]pyridin-3-one Investigative 24848656 C19H28N4OS 360.5 CC1=CC(=NC2=C1C(=O)N(S2)CN3CCN(CC3)C4CCCCC4)C IC50 = 245470.89 nM Non binder T66665 Prostaglandin G/H synthase 2 BP3OQ7 N-[3-(1-Methylpyrrol-2-yl)propyl]-2-(4-methylsulfonylphenyl)-6-(trifluoromethyl)pyrimidin-4-amine Investigative 76326065 C20H21F3N4O2S 438.5 CN1C=CC=C1CCCNC2=NC(=NC(=C2)C(F)(F)F)C3=CC=C(C=C3)S(=O)(=O)C IC50 = 251258.06 nM Non binder T66665 Prostaglandin G/H synthase 2 BP9F3H 5-(4''-Methanesulfonyl-biphenyl-2-yl)-pyrimidine Investigative 44383556 C17H14N2O2S 310.4 CS(=O)(=O)C1=CC=C(C=C1)C2=CC=CC=C2C3=CN=CN=C3 IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 BPY42U 2-(4-Methylsulfonylphenyl)-6-(trifluoromethyl)-N-[[4-(trifluoromethyl)phenyl]methyl]pyrimidin-4-amine Investigative 44456739 C20H15F6N3O2S 475.4 CS(=O)(=O)C1=CC=C(C=C1)C2=NC(=CC(=N2)NCC3=CC=C(C=C3)C(F)(F)F)C(F)(F)F IC50 = 520834.81 nM Non binder T66665 Prostaglandin G/H synthase 2 BQ8P0W 3,4-Bis-(4-methanesulfonyl-phenyl)-thiophene Investigative 44330531 C18H16O4S3 392.5 CS(=O)(=O)C1=CC=C(C=C1)C2=CSC=C2C3=CC=C(C=C3)S(=O)(=O)C IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 BQM6J4 (2S)-2-[[(2S)-2-[[(2S)-2-[(4-Fluorobenzoyl)amino]-3-(1H-indol-3-yl)propanoyl]amino]-4-methylsulfanylbutanoyl]amino]pentanedioic acid Investigative 57400089 C28H31FN4O7S 586.6 CSCC[C@@H](C(=O)N[C@@H](CCC(=O)O)C(=O)O)NC(=O)[C@H](CC1=CNC2=CC=CC=C21)NC(=O)C3=CC=C(C=C3)F IC50 = 350000 nM Non binder T66665 Prostaglandin G/H synthase 2 BR3JF7 2-(4-Methanesulfonyl-phenyl)-3-phenyl-pyrazine Investigative 44384383 C17H14N2O2S 310.4 CS(=O)(=O)C1=CC=C(C=C1)C2=NC=CN=C2C3=CC=CC=C3 IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 BR5F4S 4-[4-(Furan-2-ylmethylamino)-6-(trifluoromethyl)pyrimidin-2-yl]benzenesulfonamide Investigative 44456716 C16H13F3N4O3S 398.4 C1=COC(=C1)CNC2=NC(=NC(=C2)C(F)(F)F)C3=CC=C(C=C3)S(=O)(=O)N IC50 = 358426.41 nM Non binder T66665 Prostaglandin G/H synthase 2 BR8Z4X 2-[1-(4-Chlorobenzoyl)-2-ethylindol-3-yl]acetic acid Investigative 53249089 C19H16ClNO3 341.8 CCC1=C(C2=CC=CC=C2N1C(=O)C3=CC=C(C=C3)Cl)CC(=O)O IC50 > 400000 nM Non binder T66665 Prostaglandin G/H synthase 2 BRCU27 N-[(3-Methylphenyl)methyl]-2-(4-methylsulfonylphenyl)-6-(trifluoromethyl)pyrimidin-4-amine Investigative 44456798 C20H18F3N3O2S 421.4 CC1=CC(=CC=C1)CNC2=NC(=NC(=C2)C(F)(F)F)C3=CC=C(C=C3)S(=O)(=O)C IC50 = 518143.44 nM Non binder T66665 Prostaglandin G/H synthase 2 BS16FD Sodium;2-[2-iodo-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate Investigative 56668663 C15H16INaO3 394.18 CC(C1=C(C=C(C=C1)CC2CCCC2=O)I)C(=O)[O-].[Na+] IC50 = 540000 nM Non binder T66665 Prostaglandin G/H synthase 2 BSY6G9 2-(4''-Methanesulfonyl-biphenyl-2-yl)-pyridine Investigative 44383449 C18H15NO2S 309.4 CS(=O)(=O)C1=CC=C(C=C1)C2=CC=CC=C2C3=CC=CC=N3 IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 BTP1R2 N-Sinapoyl Serotonin Investigative 46892801 C21H22N2O5 382.4 COC1=CC(=CC(=C1O)OC)/C=C/C(=O)NCCC2=CNC3=C2C=C(C=C3)O IC50 > 400000 nM Non binder T66665 Prostaglandin G/H synthase 2 BU2XW4 2-[2-[4-(3-Chlorophenyl)piperazin-1-yl]-2-oxoethyl]-4,6-dimethyl-[1,2]thiazolo[5,4-b]pyridin-3-one Investigative 20876816 C20H21ClN4O2S 416.9 CC1=CC(=NC2=C1C(=O)N(S2)CC(=O)N3CCN(CC3)C4=CC(=CC=C4)Cl)C IC50 = 407380.28 nM Non binder T66665 Prostaglandin G/H synthase 2 BULG50 2-Acetoxyphenyl methyl sulfide Investigative 470258 C9H10O2S 182.24 CC(=O)OC1=CC=CC=C1SC IC50 = 250000 nM Non binder T66665 Prostaglandin G/H synthase 2 BV4EF1 2-Methylthiophenyl chloroacetate Investigative 10536723 C9H9ClO2S 216.68 CSC1=CC=CC=C1OC(=O)CCl IC50 = 360000 nM Non binder T66665 Prostaglandin G/H synthase 2 BVD6P0 Trp-Tyr-Asp Investigative 57398427 C24H26N4O7 482.5 C1=CC=C2C(=C1)C(=CN2)C[C@@H](C(=O)N[C@@H](CC3=CC=C(C=C3)O)C(=O)N[C@@H](CC(=O)O)C(=O)O)N IC50 = 700000 nM Non binder T66665 Prostaglandin G/H synthase 2 BVI13H 2-(4-Methanesulfonyl-phenyl)-3-phenyl-pyridine Investigative 44384384 C18H15NO2S 309.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C=CC=N2)C3=CC=CC=C3 IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 BVQ8X4 2-Hydroxy-5-[(E)-2-(4-hydroxyphenyl)ethenyl]benzoic Acid Investigative 11637444 C15H12O4 256.25 C1=CC(=CC=C1/C=C/C2=CC(=C(C=C2)O)C(=O)O)O IC50 > 500000 nM Non binder T66665 Prostaglandin G/H synthase 2 BVR52F 4-(4-Methylsulfonylphenyl)-3-phenylaniline Investigative 44384325 C19H17NO2S 323.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C=C(C=C2)N)C3=CC=CC=C3 IC50 = 254000 nM Non binder T66665 Prostaglandin G/H synthase 2 BY2T9H 2-[4-(Methylsulfonyl)phenyl]-3-(4-fluorophenyl)-4,5-diiodo-1H-pyrrole Investigative 10076665 C17H12FI2NO2S 567.2 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C(=C(N2)I)I)C3=CC=C(C=C3)F IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 BY9I6F Sodium;2-[3-(4-methylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate Investigative 56665212 C22H23NaO3 358.4 CC1=CC=C(C=C1)C2=C(C=CC(=C2)C(C)C(=O)[O-])CC3CCCC3=O.[Na+] IC50 = 420000 nM Non binder T66665 Prostaglandin G/H synthase 2 BZ0J2R (2E,5E)-5-[(3-Chlorophenyl)methylidene]-2-(1,3-thiazol-2-ylimino)-1,3-thiazolidin-4-one Investigative 135783304 C13H8ClN3OS2 321.8 C1=CC(=CC(=C1)Cl)/C=C/2\\C(=O)N/C(=N\\C3=NC=CS3)/S2 IC50 = 262000 nM Non binder T66665 Prostaglandin G/H synthase 2 BZ7P4R N-(5-Aminopyridin-2-yl)-4-(trifluoromethyl)benzamide Investigative 24752865 C13H10F3N3O 281.23 C1=CC(=CC=C1C(=O)NC2=NC=C(C=C2)N)C(F)(F)F IC50 = 210000 nM Non binder T66665 Prostaglandin G/H synthase 2 BZ8K2P (E)-3-[5-(4-Fluoro-phenyl)-4-(4-methanesulfonyl-phenyl)-thiophen-2-yl]-acrylic acid ethyl ester Investigative 44330483 C22H19FO4S2 430.5 CCOC(=O)/C=C/C1=CC(=C(S1)C2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)C IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 BZQ29K 1-Methyl-4-[2-(4-methylsulfonylphenyl)phenyl]-3,6-dihydro-2H-pyridine Investigative 15485951 C19H21NO2S 327.4 CN1CCC(=CC1)C2=CC=CC=C2C3=CC=C(C=C3)S(=O)(=O)C IC50 > 300000 nM Non binder T66665 Prostaglandin G/H synthase 2 D0F6CD SEROTONIN Investigative 5202 C10H12N2O 176.21 C1=CC2=C(C=C1O)C(=CN2)CCN IC50 > 400000 nM Non binder T66665 Prostaglandin G/H synthase 2 D0PJ3M cinnamaldehyde Investigative 637511 C9H8O 132.16 C1=CC=C(C=C1)/C=C/C=O IC50 = 245000 nM Non binder