TTD_Target_ID	Target_Name	TTD_Drug_ID	Drug_Name	Drug_Highest_Status	Drug_PubchemID	Molecular_Formula	Molecular_Weight	Canonical_SMILES	Activity	Binder_Type
T76685	Cannabinoid receptor 1	B0GA6S	N-[2-(4-Fluorophenyl)ethyl]-8-hydroxy-7-methoxy-2-oxo-6-pentyl-1H-quinoline-3-carboxamide	Investigative	56679805	C24H27FN2O4	426.5	CCCCCC1=C(C(=C2C(=C1)C=C(C(=O)N2)C(=O)NCCC3=CC=C(C=C3)F)O)OC	Ki = 2398000 nM	Non binder
T76685	Cannabinoid receptor 1	B4D2UC	N-[2-(4-Fluorophenyl)ethyl]-8-hydroxy-7-methoxy-1-methyl-2-oxo-6-pentylquinoline-3-carboxamide	Investigative	56669651	C25H29FN2O4	440.5	CCCCCC1=C(C(=C2C(=C1)C=C(C(=O)N2C)C(=O)NCCC3=CC=C(C=C3)F)O)OC	Ki = 864000 nM	Non binder
T76685	Cannabinoid receptor 1	B4R9JT	4-[[2-(Oxan-4-ylmethylcarbamoyl)pyridin-3-yl]carbamoyl]naphthalene-1-carboxylic acid	Investigative	58973328	C24H23N3O5	433.5	C1COCCC1CNC(=O)C2=C(C=CC=N2)NC(=O)C3=CC=C(C4=CC=CC=C43)C(=O)O	IC50 > 10000000 nM	Non binder
T76685	Cannabinoid receptor 1	B6XA4B	CID 23555598	Investigative	23555598	C22H23FN2O4	398.4	CCCOC1=C(C=CC2=C1NC(=O)C(=C2)C(=O)NCCC3=CC=C(C=C3)F)OC	Ki = 336000 nM	Non binder
T76685	Cannabinoid receptor 1	BA4RP8	(4-Fluoronaphthalen-1-yl)-(2-methyl-1-propylindol-3-yl)methanone	Investigative	71454235	C23H20FNO	345.4	CCCN1C(=C(C2=CC=CC=C21)C(=O)C3=CC=C(C4=CC=CC=C43)F)C	EC50 = 268000 nM	Non binder
T76685	Cannabinoid receptor 1	BE9MZ8	N-(3-Tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-(4-chlorophenylsulfonyl)-2-methylpropanamide	Investigative	25181481	C18H24ClN3O3S	397.9	CC(C)(C)C1=NN(C(=C1)NC(=O)C(C)(C)S(=O)(=O)C2=CC=C(C=C2)Cl)C	EC50 = 223000 nM	Non binder
T76685	Cannabinoid receptor 1	BFX82N	N-(Cyclobutylmethyl)-3-[[4-(methylsulfonylmethyl)naphthalene-1-carbonyl]amino]pyridine-2-carboxamide	Investigative	71545855	C24H25N3O4S	451.5	CS(=O)(=O)CC1=CC=C(C2=CC=CC=C12)C(=O)NC3=C(N=CC=C3)C(=O)NCC4CCC4	IC50 = 240000 nM	Non binder
T76685	Cannabinoid receptor 1	BJ0GD9	N-(4-Chloro-3-(trifluoromethyl)phenyl)-2-(4-chlorophenylsulfonyl)-2-methylpropanamide	Investigative	25181480	C17H14Cl2F3NO3S	440.3	CC(C)(C(=O)NC1=CC(=C(C=C1)Cl)C(F)(F)F)S(=O)(=O)C2=CC=C(C=C2)Cl	EC50 = 700000 nM	Non binder
T76685	Cannabinoid receptor 1	BQ2BN7	2-[2-Methyl-6-(4-methyl-piperazin-1-yl)-9-(tetrahydro-pyran-4-yl)-9h-purin-8-yl]-benzonitrile hydrochloride salt	Investigative	67427023	C23H28ClN7O	454	CC1=NC2=C(C(=N1)N3CCN(CC3)C)N=C(N2C4CCOCC4)C5=CC=CC=C5C#N.Cl	EC50 > 1000000 nM	Non binder