TTD_Target_ID Target_Name TTD_Drug_ID Drug_Name Drug_Highest_Status Drug_PubchemID Molecular_Formula Molecular_Weight Canonical_SMILES Activity Binder_Type T66665 Prostaglandin G/H synthase 2 D00IBN Piroxicam Approved 54676228 C15H13N3O4S 331.3 CN1C(=C(C2=CC=CC=C2S1(=O)=O)O)C(=O)NC3=CC=CC=N3 IC50 = 89125.09 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0GY5Z Aspirin Approved 2244 C9H8O4 180.16 CC(=O)OC1=CC=CC=C1C(=O)O Ki = 52000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0U5QK Acetaminophen Approved 1983 C8H9NO2 151.16 CC(=O)NC1=CC=C(C=C1)O IC50 = 141000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D00QOF ORG-13011 Phase 2 44473151 C38H43N3O4S 637.8 CCOC1=NC=C(C=C1)C2=CC=C(C=C2)CN3C4=C(C=C(C=C4)OCC5=NC=C(C=C5)C)C(=C3CC(C)(C)C(=O)O)SC(C)(C)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D05FGR R-flurbiprofen Phase 2 92337 C15H13FO2 244.26 C[C@H](C1=CC(=C(C=C1)C2=CC=CC=C2)F)C(=O)O IC50 = 123000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0DK4I PMID26560530-Compound-24 Patented 4534 C18H22O4 302.4 CC(CC1=CC(=C(C=C1)O)O)C(C)CC2=CC(=C(C=C2)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0M6LX N-(naphthylamino)-benzoate derivative 1 Patented 56851703 C17H12N2O4 308.29 C1=CC=C2C(=C1)C(=CC=C2[N+](=O)[O-])NC3=CC=CC(=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0O4QB EUGENOL Patented 3314 C10H12O2 164.2 COC1=C(C=CC(=C1)CC=C)O IC50 = 129000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0SG9Q US9388139, 12 Patented 60194756 C20H20Cl2N2O2 391.3 CC(C)(C)C1=NN(C(C1)C2=C(C=C(C=C2)Cl)Cl)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D07HBI ZD-2138 Discontinued in Phase 2 132306 C23H24FNO4 397.4 CN1C2=C(C=CC1=O)C=C(C=C2)COC3=CC(=CC(=C3)C4(CCOCC4)OC)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0K2ER MK-886 Discontinued in Phase 2 3651377 C27H34ClNO2S 472.1 CC(C)C1=CC2=C(C=C1)N(C(=C2SC(C)(C)C)CC(C)(C)C(=O)O)CC3=CC=C(C=C3)Cl IC50 = 58000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B01YEX [(1S,2S,6R,10S,11R,13S,14R,15R)-1,6-Dihydroxy-8-(hydroxymethyl)-4,12,12,15-tetramethyl-14-[(E)-2-methylbut-2-enoyl]oxy-5,9-dioxo-13-tetracyclo[8.5.0.02,6.011,13]pentadeca-3,7-dienyl] 2-methylbutanoate Investigative 118727931 C30H40O9 544.6 CCC(C)C(=O)O[C@@]12[C@@H](C1(C)C)[C@@H]3C(=O)C(=C[C@]4([C@H]([C@]3([C@@H]([C@H]2OC(=O)/C(=C/C)/C)C)O)C=C(C4=O)C)O)CO IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B02SYO (Z)-4-Amino-4-(5-chlorofuran-2-yl)-3-phenylbut-3-en-2-one Investigative 71682135 C14H12ClNO2 261.7 CC(=O)/C(=C(/C1=CC=C(O1)Cl)\\N)/C2=CC=CC=C2 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B05EOI 4-(4-(Methylsulfonyl)phenyl)-5-phenyl-3H-1,2-dithiol-3-one Investigative 44564048 C16H12O3S3 348.5 CS(=O)(=O)C1=CC=C(C=C1)C2=C(SSC2=O)C3=CC=CC=C3 IC50 = 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B08WRE 3-Amino-N-[3-(trifluoromethyl)phenyl]benzamide Investigative 2317371 C14H11F3N2O 280.24 C1=CC(=CC(=C1)N)C(=O)NC2=CC=CC(=C2)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B09SVN 3-Amino-N-[2-(trifluoromethyl)phenyl]benzamide Investigative 20115449 C14H11F3N2O 280.24 C1=CC=C(C(=C1)C(F)(F)F)NC(=O)C2=CC(=CC=C2)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0A7ZF 1-Methyl-2-guanidino-5-[(Z)-3,5-di-tert-butyl-4-hydroxybenzylidene]-2-imidazolin-4-one Investigative 11726707 C20H29N5O2 371.5 CC(C)(C)C1=CC(=CC(=C1O)C(C)(C)C)/C=C\\2/C(=O)N=C(N2C)N=C(N)N IC50 = 81000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0AO4Z (1E,4E)-1,5-Bis(4-pyrrolidin-1-ylphenyl)penta-1,4-dien-3-one Investigative 88749792 C25H28N2O 372.5 C1CN(CC1)C2=CC=C(C=C2)/C=C/C(=O)/C=C/C3=CC=C(C=C3)N4CCCC4 IC50 = 69820 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0CF9Z 4,5-Bis(4-hydroxyphenyl)-3H-1,2-dithiole-3-thione Investigative 136036210 C15H10O2S3 318.4 C1=CC(=CC=C1C2=C(SSC2=S)C3=CC=C(C=C3)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0D8ZC 2,6-Di-tert-butyl-4-(5-methoxy-1,2,4-thiadiazol-3-yl)phenol Investigative 135474341 C17H24N2O2S 320.5 CC(C)(C)C1=CC(=CC(=C1O)C(C)(C)C)C2=NSC(=N2)OC IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0ERO2 N-[(2-Methylphenyl)methyl]-2-(4-methylsulfonylphenyl)-6-(trifluoromethyl)pyrimidin-4-amine Investigative 44456799 C20H18F3N3O2S 421.4 CC1=CC=CC=C1CNC2=NC(=NC(=C2)C(F)(F)F)C3=CC=C(C=C3)S(=O)(=O)C IC50 = 174827.6 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0FLY1 2-[3-(4-Methoxyphenyl)-1-phenylpyrazol-4-yl]-5-phenyl-1,3,4-oxadiazole Investigative 46934257 C24H18N4O2 394.4 COC1=CC=C(C=C1)C2=NN(C=C2C3=NN=C(O3)C4=CC=CC=C4)C5=CC=CC=C5 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0HX8R 2-(6-Chloro-9H-carbazol-2-yl)-propionic acid 2-nitrooxy-ethyl ester Investigative 44587411 C17H15ClN2O5 362.8 CC(C1=CC2=C(C=C1)C3=C(N2)C=CC(=C3)Cl)C(=O)OCCO[N+](=O)[O-] IC50 = 65000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0L9CV Chembl4282434 Investigative 145979761 C23H16FNO4S 421.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(ON=C2C3=CC=C(C=C3)F)C(=O)C4=CC=CC=C4 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0PK3Z Chembl4173747 Investigative 138542656 C30H36N2O11 600.6 COC1=CC=C(C=C1)C2=C(ON=C2C3=CC=C(C=C3)OC)CC(=O)NCCCCC(=O)OC[C@@H]4[C@@H]([C@@H]([C@H](C(O4)O)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0TJ4F N-(Methylsulfonyl)-N-(3-(4-(2-(pyrrolidin-1-yl)ethoxy)phenoxy)-phenyl)methanesulfonamide Investigative 49805305 C20H26N2O6S2 454.6 CS(=O)(=O)N(C1=CC(=CC=C1)OC2=CC=C(C=C2)OCCN3CCCC3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0TS3K 2-(4-Fluoro-phenyl)-5-methanesulfonyl-3-(4-methanesulfonyl-phenyl)-thiophene Investigative 44330530 C18H15FO4S3 410.5 CS(=O)(=O)C1=CC=C(C=C1)C2=C(SC(=C2)S(=O)(=O)C)C3=CC=C(C=C3)F IC50 = 200000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0U2PZ N-(3-Phenylsulfinyl-4-pyridinyl)trifluoromethanesulfonamide Investigative 11256603 C12H9F3N2O3S2 350.3 C1=CC=C(C=C1)S(=O)C2=C(C=CN=C2)NS(=O)(=O)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B0XE2U [3-[2-Fluoro-4-(1-hydroxypropan-2-yl)phenyl]phenyl] N-hexylcarbamate Investigative 73054809 C22H28FNO3 373.5 CCCCCCNC(=O)OC1=CC=CC(=C1)C2=C(C=C(C=C2)C(C)CO)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B13XFG 2-[6-Chloro-9-(methylcarbamoyl)carbazol-2-yl]propanoic acid Investigative 71457026 C17H15ClN2O3 330.8 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)NC)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B14FJB 3-Mesityl-4-phenyl-5-methylisoxazole Investigative 11231244 C19H19NO 277.4 CC1=CC(=C(C(=C1)C)C2=NOC(=C2C3=CC=CC=C3)C)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B14JLX 2-(6-Chloro-9-methyl-9H-carbazol-2-yl)propanoic acid Investigative 71462406 C16H14ClNO2 287.74 CC(C1=CC2=C(C=C1)C3=C(N2C)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B17GID 4-[3-(2-Bromophenyl)-5-tert-butyl-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548447 C20H21BrN2O2 401.3 CC(C)(C)C1=NN(C(C1)C2=CC=CC=C2Br)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B17LIW 4-[5-Tert-butyl-3-(2-fluorophenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548633 C20H21FN2O2 340.4 CC(C)(C)C1=NN(C(C1)C2=CC=CC=C2F)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1BCO8 4-(2-(4-Fluorophenyl)-1H-pyrrol-1-yl)-N-methylbenzenesulfonamide Investigative 10520447 C17H15FN2O2S 330.4 CNS(=O)(=O)C1=CC=C(C=C1)N2C=CC=C2C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1FH9Q N-Caffeoyl serotonin Investigative 16659826 C19H18N2O4 338.4 C1=CC(=C(C=C1/C=C/C(=O)NCCC2=CNC3=C2C=C(C=C3)O)O)O Ki = 65500 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1GC2Y 2-(Benzenesulfonyl)-3-(1,3-benzodioxol-4-yl)-5-(trifluoromethyl)-3,4-dihydropyrazole Investigative 118706117 C17H13F3N2O4S 398.4 C1C(N(N=C1C(F)(F)F)S(=O)(=O)C2=CC=CC=C2)C3=C4C(=CC=C3)OCO4 IC50 = 60980 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1H2QN trans-AUCB Investigative 16038368 C24H32N2O4 412.5 C1CC(CCC1NC(=O)NC23CC4CC(C2)CC(C4)C3)OC5=CC=C(C=C5)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1H3QL 2-(4-Fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-5-phenylsulfanyl-thiophene Investigative 44330495 C23H17FO2S3 440.6 CS(=O)(=O)C1=CC=C(C=C1)C2=C(SC(=C2)SC3=CC=CC=C3)C4=CC=C(C=C4)F IC50 = 66000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1I9MY Chembl4278979 Investigative 145980296 C18H14FNO5S 375.4 COC(=O)C1=C(C(=NO1)C2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1JL3E 2-(4-Chlorophenyl)-4-(methylsulfonylmethyl)-1-(4-methylsulfonylphenyl)imidazole Investigative 10670044 C18H17ClN2O4S2 424.9 CS(=O)(=O)CC1=CN(C(=N1)C2=CC=C(C=C2)Cl)C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1L9XT 3,5-Diphenyl-1,2-oxazole-4-carboxylic acid Investigative 13804275 C16H11NO3 265.26 C1=CC=C(C=C1)C2=C(C(=NO2)C3=CC=CC=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1N7AP 2-[6-Chloro-9-[(2-methoxyphenyl)methyl]carbazol-2-yl]propanoic acid Investigative 71458882 C23H20ClNO3 393.9 CC(C1=CC2=C(C=C1)C3=C(N2CC4=CC=CC=C4OC)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1NG7J Chembl4173674 Investigative 145949529 C20H19ClN6O2 410.9 C1COCC(=O)N1C2=CC=C(C=C2)NC3=NC(=NC(=N3)NCC4=CC=CC=C4)Cl IC50 = 60000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1QF5G (3E,5E)-3,5-Bis[(4-pyrrolidin-1-ylphenyl)methylidene]piperidin-4-one Investigative 118706207 C27H31N3O 413.6 C1CN(CC1)C2=CC=C(C=C2)/C=C\\3/C(=O)/C(=C/C4=CC=C(C=C4)N5CCCC5)/CNC3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1TKH3 4-[(3E,6E,9E,12E)-Pentadeca-3,6,9,12-tetraenyl]sulfanylbutanoic acid Investigative 44584307 C19H30O2S 322.5 CC/C=C/C/C=C/C/C=C/C/C=C/CCSCCCC(=O)O IC50 = 120000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1W5SP 4-[5-Tert-butyl-3-(3-chlorophenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 68308827 C20H21ClN2O2 356.8 CC(C)(C)C1=NN(C(C1)C2=CC(=CC=C2)Cl)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1WLV8 N-[4-(4-Chloroanilino)phenyl]-4-hydroxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728408 C21H16ClN3O4S 441.9 C1=CC=C2C(=C1)C(=C(NS2(=O)=O)C(=O)NC3=CC=C(C=C3)NC4=CC=C(C=C4)Cl)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1XKC6 [2-[3-[3-Fluoro-5-(4-methoxyoxan-4-yl)phenoxy]propyl]-8-methoxy-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]-(4-fluorophenyl)methanone;hydrochloride Investigative 46845030 C34H37ClF2N2O5 627.1 COC1=CC2=C(C=C1)N(C3=C2CN(CC3)CCCOC4=CC(=CC(=C4)C5(CCOCC5)OC)F)C(=O)C6=CC=C(C=C6)F.Cl IC50 = 53600 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1XMA7 2-Bromo-4-(4-fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-thiophene Investigative 44330429 C17H12BrFO2S2 411.3 CS(=O)(=O)C1=CC=C(C=C1)C2=C(SC=C2C3=CC=C(C=C3)F)Br IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B1ZP8A Acetic acid 2-ethylsulfanyl-phenyl ester Investigative 9813036 C10H12O2S 196.27 CCSC1=CC=CC=C1OC(=O)C IC50 = 200000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B21EIN 2-[4-[3-(Benzylcarbamoyloxy)phenyl]-3-fluorophenyl]propanoic acid Investigative 73054547 C23H20FNO4 393.4 CC(C1=CC(=C(C=C1)C2=CC(=CC=C2)OC(=O)NCC3=CC=CC=C3)F)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B26CVM 4-Methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide Investigative 743974 C16H19NO3S 305.4 CC1=CC(=C(C(=C1)C)NS(=O)(=O)C2=CC=C(C=C2)OC)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B26LDF 4-[[2-(4-Fluorophenyl)-4-oxo-1,3-thiazolidin-3-yl]amino]benzenesulfonamide Investigative 70691164 C15H14FN3O3S2 367.4 C1C(=O)N(C(S1)C2=CC=C(C=C2)F)NC3=CC=C(C=C3)S(=O)(=O)N IC50 = 63000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B26WTR 4-(4-Cyclohexyl-2-methyl-oxazol-5-yl)-2-methoxy-benzenesulfonamide Investigative 11002614 C17H22N2O4S 350.4 CC1=NC(=C(O1)C2=CC(=C(C=C2)S(=O)(=O)N)OC)C3CCCCC3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B28FJT Methyl 5-(4-fluorophenyl)-1-(4-sulfamoylphenyl)pyrazole-3-carboxylate Investigative 10738225 C17H14FN3O4S 375.4 COC(=O)C1=NN(C(=C1)C2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)N IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B28LDQ Schembl20646331 Investigative 137412863 C18H12F8O3S 460.3 C1=CC=C(C=C1)CC2=CC(=CC3=C2OC(C(=C3)C(=O)O)C(F)(F)F)S(F)(F)(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B29MZO N-[3-(3-Bromo-4-hydroxyanilino)pyridin-4-yl]-1,1,1-trifluoromethanesulfonamide Investigative 76310403 C12H9BrF3N3O3S 412.18 C1=CC(=C(C=C1NC2=C(C=CN=C2)NS(=O)(=O)C(F)(F)F)Br)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2BC7E 3-[4-Methyl-1-(4-methylsulfonylphenyl)imidazol-2-yl]pyridine Investigative 10663006 C16H15N3O2S 313.4 CC1=CN(C(=N1)C2=CN=CC=C2)C3=CC=C(C=C3)S(=O)(=O)C IC50 = 79000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2BTZ5 (2R,3R)-6-[(E)-2-Carboxyethenyl]-2-(3,4-dihydroxyphenyl)-2,3-dihydro-1,4-benzodioxine-3-carboxylic acid Investigative 57395427 C18H14O8 358.3 C1=CC2=C(C=C1/C=C/C(=O)O)O[C@H]([C@H](O2)C3=CC(=C(C=C3)O)O)C(=O)O IC50 = 52600 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2C0ZE Methyl (2S)-4-methyl-2-[[2-[[(2S)-3-methyl-2-(phenylmethoxycarbonylamino)butanoyl]amino]acetyl]amino]pentanoate Investigative 127043218 C22H33N3O6 435.5 CC(C)C[C@@H](C(=O)OC)NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)OCC1=CC=CC=C1 IC50 = 56000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2CDW6 4-(4-(2-(Pyrrolidin-1-yl)ethoxy)phenoxy)aniline Investigative 49805303 C18H22N2O2 298.4 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=C(C=C3)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2EC1Z 1,2-Dihydro-7-methoxy-3-(2,3,4-trimethoxyphenyl)-naphthalene Investigative 23627031 C20H22O4 326.4 COC1=CC2=C(C=C1)C=C(CC2)C3=C(C(=C(C=C3)OC)OC)OC IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2ETU0 5-[(5-Anilino-1,3,4-thiadiazol-2-yl)methyl]-3-methyl-7-[(4-nitrophenyl)methyl]-[1,2]oxazolo[4,5-d]pyridazin-4-one Investigative 70689657 C22H17N7O4S 475.5 CC1=NOC2=C1C(=O)N(N=C2CC3=CC=C(C=C3)[N+](=O)[O-])CC4=NN=C(S4)NC5=CC=CC=C5 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2IO8D 3-(4-(2-(Pyrrolidin-1-yl)ethoxy)phenoxy)aniline Investigative 49805302 C18H22N2O2 298.4 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=CC(=C3)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2J3WI 2-[1-(4-Chloro-benzoyl)-5-methoxy-1H-indol-3-yl]-N-phenethyl-acetamide Investigative 10718261 C26H23ClN2O3 446.9 COC1=CC2=C(C=C1)N(C=C2CC(=O)NCCC3=CC=CC=C3)C(=O)C4=CC=C(C=C4)Cl IC50 ~ 66000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2K1DI 8-(4-Carboxyphenyl)-6-chloro-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid Investigative 53316515 C18H10ClF3O5 398.7 C1=CC(=CC=C1C2=CC(=CC3=C2OC(C(=C3)C(=O)O)C(F)(F)F)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2M7LF 1-(4-Fluorophenyl)-2-(4-methylsulfonylphenyl)-5-(trifluoromethyl)pyrrole Investigative 10809969 C18H13F4NO2S 383.4 CS(=O)(=O)C1=CC=C(C=C1)C2=CC=C(N2C3=CC=C(C=C3)F)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2O8NX 2-(Benzenesulfonyl)-3-naphthalen-1-yl-5-(trifluoromethyl)-3,4-dihydropyrazole Investigative 118706112 C20H15F3N2O2S 404.4 C1C(N(N=C1C(F)(F)F)S(=O)(=O)C2=CC=CC=C2)C3=CC=CC4=CC=CC=C43 IC50 = 67130 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2PUG6 6-Chloro-7-((2,6-dimethylpiperidin-1-yl)methyl)-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid Investigative 53319287 C19H21ClF3NO3 403.8 CC1CCCC(N1CC2=C(C=C3C=C(C(OC3=C2)C(F)(F)F)C(=O)O)Cl)C IC50 = 62200 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2Q4FY 2-(2,6-Dichloro-3-methylphenylamino)benzohydroxamic acid 4-nitrobenzyl ester Investigative 11744262 C21H17Cl2N3O4 446.3 CC1=C(C(=C(C=C1)Cl)NC2=CC=CC=C2C(=O)NOCC3=CC=C(C=C3)[N+](=O)[O-])Cl IC50 = 66000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2QM5E Indomethacin derivative, 21 Investigative 10505250 C27H27BrN2O2 491.4 CC1=C(C2=C(N1CC3=CC=C(C=C3)Br)C=CC(=C2)OC)CC(=O)NCCC4=CC=CC=C4 IC50 ~ 66000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2TON8 2-[3-Fluoro-4-[2-(hexylcarbamoyloxy)phenyl]phenyl]propanoic acid Investigative 73055091 C22H26FNO4 387.4 CCCCCCNC(=O)OC1=CC=CC=C1C2=C(C=C(C=C2)C(C)C(=O)O)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2UI8R 4-(4-Fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-1H-pyrazole Investigative 15380227 C16H13FN2O2S 316.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C=NN2)C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2V4YX N-[3-(3-Chlorophenoxy)-4-pyridinyl]trifluoromethanesulfonamide Investigative 11291135 C12H8ClF3N2O3S 352.72 C1=CC(=CC(=C1)Cl)OC2=C(C=CN=C2)NS(=O)(=O)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2WEG7 3-(5-Chlorofuran-2-Yl)-5-Methyl-4-Phenyl-1,2-Oxazole Investigative 10355223 C14H10ClNO2 259.69 CC1=C(C(=NO1)C2=CC=C(O2)Cl)C3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2X8PC (2E)-2-[(4-Pyrrolidin-1-ylphenyl)methylidene]-3,4-dihydronaphthalen-1-one Investigative 90645132 C21H21NO 303.4 C1CCN(C1)C2=CC=C(C=C2)/C=C/3\\CCC4=CC=CC=C4C3=O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B2XCZ4 (E)-3-(4-Methylsulfonylphenyl)-2-[3-(4-propan-2-yloxyphenyl)phenyl]prop-2-enoic acid Investigative 76309082 C25H24O5S 436.5 CC(C)OC1=CC=C(C=C1)C2=CC(=CC=C2)/C(=C\\C3=CC=C(C=C3)S(=O)(=O)C)/C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B37TYH 4-[[4-Oxo-2-[4-(trifluoromethyl)phenyl]-1,3-thiazolidin-3-yl]amino]benzenesulfonamide Investigative 70689055 C16H14F3N3O3S2 417.4 C1C(=O)N(C(S1)C2=CC=C(C=C2)C(F)(F)F)NC3=CC=C(C=C3)S(=O)(=O)N IC50 = 51800 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3CLD7 4-[5-(4-Hydroxy-phenyl)-3-trifluoromethyl-pyrazol-1-yl]-benzenesulfonamide Investigative 135532444 C16H12F3N3O3S 383.3 C1=CC(=CC=C1C2=CC(=NN2C3=CC=C(C=C3)S(=O)(=O)N)C(F)(F)F)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3CXD5 4-Amino-N-[3-(trifluoromethyl)phenyl]benzamide Investigative 2756535 C14H11F3N2O 280.24 C1=CC(=CC(=C1)NC(=O)C2=CC=C(C=C2)N)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3F0NS 4-[5-(4-Methoxyphenyl)tetrazol-1-yl]benzenesulfonamide Investigative 57390392 C14H13N5O3S 331.35 COC1=CC=C(C=C1)C2=NN=NN2C3=CC=C(C=C3)S(=O)(=O)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3H6NO 4-(5-Tert-butyl-3-phenyl-3,4-dihydropyrazol-2-yl)benzoic acid Investigative 68292820 C20H22N2O2 322.4 CC(C)(C)C1=NN(C(C1)C2=CC=CC=C2)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3KW9B 6-(4-Methanesulfonyl-phenyl)-5-phenyl-2-trifluoromethyl-thiazolo[3,2-b][1,2,4]triazole Investigative 44371442 C18H12F3N3O2S2 423.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(SC3=NC(=NN23)C(F)(F)F)C4=CC=CC=C4 IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3L9PX 2-Phenylethyl 2-{1-[(4-bromophenyl)methyl]-5-methoxy-2-methyl-1H-indol-3-yl}acetate Investigative 10648828 C27H26BrNO3 492.4 CC1=C(C2=C(N1CC3=CC=C(C=C3)Br)C=CC(=C2)OC)CC(=O)OCCC4=CC=CC=C4 IC50 ~ 66000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3LT5J 4-(4-(2-(Pyrrolidin-1-yl)ethoxy)phenoxy)pyridine Investigative 49805050 C17H20N2O2 284.35 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=NC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3MEY9 2-(4-(2-(Pyrrolidin-1-yl)ethoxy)phenoxy)pyrazine Investigative 49805055 C16H19N3O2 285.34 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=NC=CN=C3 IC50 = 61600 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3NCX5 5-Amino-N-[4-(trifluoromethyl)phenyl]pyridine-2-carboxamide Investigative 24854032 C13H10F3N3O 281.23 C1=CC(=CC=C1C(F)(F)F)NC(=O)C2=NC=C(C=C2)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3OUB7 1-(4-Methylsulfonylphenyl)-5-(4-nitrophenyl)tetrazole Investigative 57402675 C14H11N5O4S 345.34 CS(=O)(=O)C1=CC=C(C=C1)N2C(=NN=N2)C3=CC=C(C=C3)[N+](=O)[O-] IC50 = 69000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3QB0G 2,6-Bis(4-(pyrrolidin-1-yl)benzylidene)cyclohexanone Investigative 118706205 C28H32N2O 412.6 C1CN(CC1)C2=CC=C(C=C2)/C=C\\3/C(=O)/C(=C/C4=CC=C(C=C4)N5CCCC5)/CCC3 IC50 = 54320 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3QN4W (7-Tert-Butyl-3,3-dimethyl-2,3-dihydro-benzofuran-5-yl)-(4,5-dihydro-pyrazol-1-yl)-amine Investigative 44344893 C17H25N3O 287.4 CC1(COC2=C1C=C(C=C2C(C)(C)C)NN3CCC=N3)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B3S2RA 2-[6-Chloro-9-(4-fluorobenzoyl)carbazol-2-yl]propanoic acid Investigative 71457021 C22H15ClFNO3 395.8 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)C4=CC=C(C=C4)F)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B40XZF 5-(4-(Methylsulfonyl)phenyl)-1-phenyl-1H-tetrazole Investigative 53320894 C14H12N4O2S 300.34 CS(=O)(=O)C1=CC=C(C=C1)C2=NN=NN2C3=CC=CC=C3 IC50 = 200000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B42DXU 3,3-Dimethyl-5-[pyrrolizino(imino)methyl]-7-tert-butyl-2,3-dihydrobenzofuran Investigative 10637982 C19H28N2O 300.4 CC1(COC2=C1C=C(C=C2C(C)(C)C)C(=N)N3CCCC3)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B42HPU 1-(4-Chlorophenyl)-5-(4-(methylsulfonyl)phenyl)-1H-tetrazole Investigative 53318243 C14H11ClN4O2S 334.8 CS(=O)(=O)C1=CC=C(C=C1)C2=NN=NN2C3=CC=C(C=C3)Cl IC50 = 110000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B43SPG Clematichinenoside C Investigative 49799271 C70H114O34 1499.6 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H](O[C@H]([C@@H]([C@H]2O)O)OC[C@@H]3[C@H]([C@@H]([C@H]([C@@H](O3)OC(=O)[C@@]45CC[C@@]6(C(=CC[C@H]7[C@]6(CC[C@@H]8[C@@]7(CC[C@@H](C8(C)C)O[C@H]9[C@@H]([C@H]([C@H](CO9)O)O)O[C@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)C)O)O[C@H]1[C@@H]([C@@H]([C@@H](CO1)O[C@H]1[C@@H]([C@H]([C@@H]([C@H](O1)CO)O)O)O)O)O)O)C)C)[C@@H]4CC(CC5)(C)C)C)O)O)O)CO)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B43WXO 4-[5-(4-Fluorophenyl)tetrazol-1-yl]benzenesulfonamide Investigative 57392194 C13H10FN5O2S 319.32 C1=CC(=CC=C1C2=NN=NN2C3=CC=C(C=C3)S(=O)(=O)N)F IC50 = 56000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B45HNP US9271961, Bmt 4-90 Investigative 124222779 C14H12N2O5 288.25 COC1=CC(=C(C=C1)[N+](=O)[O-])NC2=CC=CC=C2C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B47SGK Mofezolac Investigative 4237 C19H17NO5 339.3 COC1=CC=C(C=C1)C2=C(ON=C2C3=CC=C(C=C3)OC)CC(=O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4A8KI 4-(3-Methoxy-5-phenyl-pyrazol-1-yl)-benzenesulfonamide Investigative 10853804 C16H15N3O3S 329.4 COC1=NN(C(=C1)C2=CC=CC=C2)C3=CC=C(C=C3)S(=O)(=O)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4BH3D 12-O-Tiglylphorbol-13-isobutyrate Investigative 73350378 C29H40O8 516.6 C/C=C(\\C)/C(=O)O[C@@H]1[C@H]([C@]2([C@@H](C=C(C[C@]3([C@H]2C=C(C3=O)C)O)CO)[C@H]4[C@@]1(C4(C)C)OC(=O)C(C)C)O)C IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4EW3S N-Methyl-N-(2-(4-(2-(pyrrolidin-1-yl)ethoxy)phenoxy)phenyl)methanesulfonamide Investigative 49805307 C20H26N2O4S 390.5 CN(C1=CC=CC=C1OC2=CC=C(C=C2)OCCN3CCCC3)S(=O)(=O)C IC50 = 92000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4FC8U 6-Chloro-7-((isopropyl(methyl)amino)methyl)-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid Investigative 53325872 C16H17ClF3NO3 363.76 CC(C)N(C)CC1=C(C=C2C=C(C(OC2=C1)C(F)(F)F)C(=O)O)Cl IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4FCR7 N-[4-[(Z)-2-Cyclohexyl-1,2-diphenylethenyl]phenyl]methanesulfonamide Investigative 76312773 C27H29NO2S 431.6 CS(=O)(=O)NC1=CC=C(C=C1)/C(=C(/C2CCCCC2)\\C3=CC=CC=C3)/C4=CC=CC=C4 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4G6MU [1-(4-Chloro-benzoyl)-5-methoxy-1H-indol-3-yl]-acetic acid phenethyl ester Investigative 10599548 C26H22ClNO4 447.9 COC1=CC2=C(C=C1)N(C=C2CC(=O)OCCC3=CC=CC=C3)C(=O)C4=CC=C(C=C4)Cl IC50 ~ 66000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4HB0K 4-[2-(4-Fluoro-phenyl)-pyrrol-1-yl]-N,N-dimethyl-benzenesulfonamide Investigative 10688810 C18H17FN2O2S 344.4 CN(C)S(=O)(=O)C1=CC=C(C=C1)N2C=CC=C2C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4I6QF 5-(2-Acetoxy-phenylsulfanyl)-pentanoic acid Investigative 10516041 C13H16O4S 268.33 CC(=O)OC1=CC=CC=C1SCCCCC(=O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4K9MD N-(3-Aminopyridin-2-yl)-3-(trifluoromethyl)benzamide Investigative 24853947 C13H10F3N3O 281.23 C1=CC(=CC(=C1)C(F)(F)F)C(=O)NC2=C(C=CC=N2)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4N1UE 1-Allyl-4-(4-fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-1H-pyrazole Investigative 44307569 C19H17FN2O2S 356.4 CS(=O)(=O)C1=CC=C(C=C1)C2=NN(C=C2C3=CC=C(C=C3)F)CC=C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4OFC8 N-(4-Amino-2-pyridyl)-4-(trifluoromethyl)benzamide Investigative 24854030 C13H10F3N3O 281.23 C1=CC(=CC=C1C(=O)NC2=NC=CC(=C2)N)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4QC2Z Methyl 2-[3-fluoro-4-[3-(hexylcarbamoyloxy)phenyl]phenyl]propanoate Investigative 90036171 C23H28FNO4 401.5 CCCCCCNC(=O)OC1=CC=CC(=C1)C2=C(C=C(C=C2)C(C)C(=O)OC)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4SK0Y [2-[3-[3-Fluoro-5-(4-methoxyoxan-4-yl)phenoxy]propyl]-8-methoxy-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]-phenylmethanone;hydrochloride Investigative 46906729 C34H38ClFN2O5 609.1 COC1=CC2=C(C=C1)N(C3=C2CN(CC3)CCCOC4=CC(=CC(=C4)C5(CCOCC5)OC)F)C(=O)C6=CC=CC=C6.Cl IC50 = 78300 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4TJI8 3,4-Bis-(4-methylsulfanyl-phenyl)-thiophene Investigative 44330563 C18H16S3 328.5 CSC1=CC=C(C=C1)C2=CSC=C2C3=CC=C(C=C3)SC IC50 = 101000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4WH0S (R)-Carprofen Investigative 6997572 C15H12ClNO2 273.71 C[C@H](C1=CC2=C(C=C1)C3=C(N2)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4YQ8G (2E,6Z)-2,6-Bis[[4-(dimethylamino)-2-nitrophenyl]methylidene]cyclohexan-1-one Investigative 90645116 C24H26N4O5 450.5 CN(C)C1=CC(=C(C=C1)/C=C/2\\CCC/C(=C/C3=C(C=C(C=C3)N(C)C)[N+](=O)[O-])/C2=O)[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B4ZBX9 3-Morpholin-4-ylpropyl 3-(5-chlorofuran-2-yl)-4-phenyl-1,2-oxazole-5-carboxylate Investigative 57780770 C21H21ClN2O5 416.9 C1COCCN1CCCOC(=O)C2=C(C(=NO2)C3=CC=C(O3)Cl)C4=CC=CC=C4 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B51GHP 2-[6-Chloro-9-(1,3-thiazole-4-carbonyl)carbazol-2-yl]propanoic acid Investigative 71458879 C19H13ClN2O3S 384.8 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)C4=CSC=N4)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B52ZWH 5-Chloro-3-(3-fluoro-4-phenylphenyl)-2-(4-methylsulfonylphenyl)pyran-4-one Investigative 44310048 C24H16ClFO4S 454.9 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C(=O)C(=CO2)Cl)C3=CC(=C(C=C3)C4=CC=CC=C4)F IC50 = 87902.25 nM Poor binder T66665 Prostaglandin G/H synthase 2 B53FJE 2-(4-Fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-spiro[4.5]dec-2-ene Investigative 10810080 C23H25FO2S 384.5 CS(=O)(=O)C1=CC=C(C=C1)C2=C(CC3(C2)CCCCC3)C4=CC=C(C=C4)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B57GXV 2-(4-Methylphenyl)sulfonyl-3-naphthalen-1-yl-5-(trifluoromethyl)-3,4-dihydropyrazole Investigative 118706118 C21H17F3N2O2S 418.4 CC1=CC=C(C=C1)S(=O)(=O)N2C(CC(=N2)C(F)(F)F)C3=CC=CC4=CC=CC=C43 IC50 = 89070 nM Poor binder T66665 Prostaglandin G/H synthase 2 B5A6BG 3-(4-Methoxy-2-nitroanilino)benzoic acid Investigative 43358934 C14H12N2O5 288.25 COC1=CC(=C(C=C1)NC2=CC=CC(=C2)C(=O)O)[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B5FX1D 4-[3-(4-Methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]benzenesulfonamide Investigative 2950007 C22H21N3O3S 407.5 COC1=CC=C(C=C1)C2CC(=NN2C3=CC=C(C=C3)S(=O)(=O)N)C4=CC=CC=C4 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B5G4CO N-(2-Aminophenyl)-4-(trifluoromethyl)benzamide Investigative 572427 C14H11F3N2O 280.24 C1=CC=C(C(=C1)N)NC(=O)C2=CC=C(C=C2)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B5I4XW Ketorolac tromethamine Investigative 84003 C19H24N2O6 376.4 C1CN2C(=CC=C2C(=O)C3=CC=CC=C3)C1C(=O)O.C(C(CO)(CO)N)O IC50 = 60500 nM Poor binder T66665 Prostaglandin G/H synthase 2 B5KGW2 3-Amino-N-[4-(trifluoromethyl)phenyl]benzamide Investigative 13609513 C14H11F3N2O 280.24 C1=CC(=CC(=C1)N)C(=O)NC2=CC=C(C=C2)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B5MJ8Q 4-[5-Tert-butyl-3-(4-chlorophenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 68292588 C20H21ClN2O2 356.8 CC(C)(C)C1=NN(C(C1)C2=CC=C(C=C2)Cl)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B5Q7AT 2-(6-Chloro-9H-carbazol-2-yl)-N-(2-hydroxyethyl)propanamide Investigative 16415139 C17H17ClN2O2 316.8 CC(C1=CC2=C(C=C1)C3=C(N2)C=CC(=C3)Cl)C(=O)NCCO IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B5SX3M 5-Methyl-4-phenyl-3-(2,4,6-trimethoxy-phenyl)-isoxazole Investigative 11301795 C19H19NO4 325.4 CC1=C(C(=NO1)C2=C(C=C(C=C2OC)OC)OC)C3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B5V9FC 4-[3-(4-Methanesulfonyl-phenyl)-thiophen-2-yl]-phenol Investigative 44330592 C17H14O3S2 330.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(SC=C2)C3=CC=C(C=C3)O IC50 = 86000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B5W0LS 4-[(3R,3Ar,6R,6aR)-6-(4-hydroxy-3-methoxyphenyl)-1,3,3a,4,6,6a-hexahydrofuro[3,4-c]furan-3-yl]-2-methoxyphenol Investigative 12309637 C20H22O6 358.4 COC1=C(C=CC(=C1)[C@H]2[C@H]3CO[C@H]([C@H]3CO2)C4=CC(=C(C=C4)O)OC)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B5Y3TI [(2S,3R,4S,5S,6R)-6-[[(2R,3R,4R,5S,6R)-3,4-Dihydroxy-6-(hydroxymethyl)-5-[(2S,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxyoxan-2-yl]oxymethyl]-3,4,5-trihydroxyoxan-2-yl] (4aS,6aR,6aS,6bR,8aR,9R,10S,12aR,14bS)-10-[(2S,3R,4S,5S)-3-[(2S,3R,4R,5S,6S)-4-[(2S,3R,4S,5R)-5-[(2R,3R,4R,5S,6R)-3,4-dihydroxy-6-(hydroxymethyl)-5-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyoxan-2-yl]oxy-3,4-dihydroxyoxan-2-yl]oxy-3,5-dihydroxy-6-methyloxan-2-yl]oxy-4,5-dihydroxyoxan-2-yl]oxy-9-(hydroxymethyl)-2,2,6a,6b,9,12a-hexamethyl-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylate Investigative 49799273 C76H124O40 1677.8 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H](O[C@H]([C@@H]([C@H]2O)O)OC[C@@H]3[C@H]([C@@H]([C@H]([C@@H](O3)OC(=O)[C@@]45CC[C@@]6(C(=CC[C@H]7[C@]6(CC[C@@H]8[C@@]7(CC[C@@H]([C@@]8(C)CO)O[C@H]9[C@@H]([C@H]([C@H](CO9)O)O)O[C@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)C)O)O[C@H]1[C@@H]([C@@H]([C@@H](CO1)O[C@H]1[C@@H]([C@H]([C@@H]([C@H](O1)CO)O[C@H]1[C@@H]([C@H]([C@@H]([C@H](O1)CO)O)O)O)O)O)O)O)O)C)C)[C@@H]4CC(CC5)(C)C)C)O)O)O)CO)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B5Y4WD Chembl4278833 Investigative 145981172 C18H14FNO4S 359.4 CC(=O)C1=C(C(=NO1)C2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B60SWZ N-[4-(3,4-Dichlorophenyl)phenyl]-4-hydroxy-1,1-dioxo-3,4-dihydro-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 46880352 C21H16Cl2N2O4S 463.3 C1=CC=C2C(=C1)C(C(NS2(=O)=O)C(=O)NC3=CC=C(C=C3)C4=CC(=C(C=C4)Cl)Cl)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B62HPJ 2-[6-Chloro-9-[(4-chlorophenyl)methyl]carbazol-2-yl]propanoic acid Investigative 71453516 C22H17Cl2NO2 398.3 CC(C1=CC2=C(C=C1)C3=C(N2CC4=CC=C(C=C4)Cl)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B64JTA 4-[3-(3-Bromophenyl)-5-tert-butyl-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548631 C20H21BrN2O2 401.3 CC(C)(C)C1=NN(C(C1)C2=CC(=CC=C2)Br)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B67FMY 4-[5-(4-Nitrophenyl)tetrazol-1-yl]benzenesulfonamide Investigative 57399159 C13H10N6O4S 346.32 C1=CC(=CC=C1C2=NN=NN2C3=CC=C(C=C3)S(=O)(=O)N)[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B6BWH4 (2S)-2-[[(2S)-2-[(4-Fluorobenzoyl)amino]-3-(4-hydroxyphenyl)propanoyl]amino]butanedioic acid Investigative 57393176 C20H19FN2O7 418.4 C1=CC(=CC=C1C[C@@H](C(=O)N[C@@H](CC(=O)O)C(=O)O)NC(=O)C2=CC=C(C=C2)F)O IC50 = 110000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B6ME9Q N,N-Dimethyl-12-(S-valinoyl)-13-acetyl-4r-4-deoxyphorbol Investigative 11526431 C29H43NO7 517.7 C[C@@H]1[C@H]([C@@]2([C@@H](C2(C)C)[C@H]3[C@]1([C@@H]4C=C(C(=O)[C@@H]4CC(=C3)CO)C)O)OC(=O)C)OC(=O)[C@H](C(C)C)N(C)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B6N4MR Chembl4279921 Investigative 145982141 C16H12FNO3S 317.3 CS(=O)(=O)C1=CC=C(C=C1)C2=CC(=NO2)C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B6OPT3 4-Chloro-5-(4-chlorophenyl)-1-(4-sulfamoylphenyl)pyrazole-3-carboxylic Acid Investigative 11795928 C16H11Cl2N3O4S 412.2 C1=CC(=CC=C1C2=C(C(=NN2C3=CC=C(C=C3)S(=O)(=O)N)C(=O)O)Cl)Cl IC50 = 70000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B6S5QU N-(3-Phenylsulfonyl-4-pyridinyl)trifluoromethanesulfonamide Investigative 11382984 C12H9F3N2O4S2 366.3 C1=CC=C(C=C1)S(=O)(=O)C2=C(C=CN=C2)NS(=O)(=O)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B6U7KM 1-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl)-4-methyl-1H-imidazole Investigative 10568417 C17H15FN2O2S 330.4 CC1=CN(C(=N1)C2=CC=C(C=C2)S(=O)(=O)C)C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B6V3XK 1-(5-Chloro-1,3-benzoxazol-2-yl)-N-cyclopentylpiperidine-4-carboxamide Investigative 71520910 C18H22ClN3O2 347.8 C1CCC(C1)NC(=O)C2CCN(CC2)C3=NC4=C(O3)C=CC(=C4)Cl IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B6VRJ1 2-[4-(Methylsulfonyl)phenyl]-3-(4-fluorophenyl)-1H-pyrrole-5-carbonitrile Investigative 10449908 C18H13FN2O2S 340.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C=C(N2)C#N)C3=CC=C(C=C3)F IC50 = 64400 nM Poor binder T66665 Prostaglandin G/H synthase 2 B6WX8C N-(4-Aminophenyl)-3-(trifluoromethyl)benzamide Investigative 18543182 C14H11F3N2O 280.24 C1=CC(=CC(=C1)C(F)(F)F)C(=O)NC2=CC=C(C=C2)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B6XGT4 N-(3,4-Dimethoxyphenyl)-1-(4-methoxyphenyl)-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazole-3-carboxamide Investigative 90654429 C27H28N4O7 520.5 COC1=CC=C(C=C1)N2C(=NC(=N2)C(=O)NC3=CC(=C(C=C3)OC)OC)C4=CC(=C(C(=C4)OC)OC)OC IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B6YRO1 Sodium;2-[2-(4-methylsulfanylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate Investigative 56672143 C22H23NaO3S 390.5 CC(C1=C(C=C(C=C1)CC2CCCC2=O)C3=CC=C(C=C3)SC)C(=O)[O-].[Na+] IC50 = 150000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B6ZDE5 (5Z)-2-[1-(6-Methoxynaphthalen-2-yl)ethyl]-5-[(4-phenylphenyl)methylidene]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one Investigative 118729078 C30H23N3O2S 489.6 CC(C1=CC2=C(C=C1)C=C(C=C2)OC)C3=NN4C(=O)/C(=C/C5=CC=C(C=C5)C6=CC=CC=C6)/SC4=N3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B71CQZ 4-Phenyl-5-methyl-3-(5-methylfuran-2-yl)isoxazole Investigative 44194811 C15H13NO2 239.27 CC1=CC=C(O1)C2=NOC(=C2C3=CC=CC=C3)C IC50 = 68200 nM Poor binder T66665 Prostaglandin G/H synthase 2 B72LPH 1-[1-[(2-Chlorophenyl)methyl]-2-oxopyridin-3-yl]-3-(3-ethylphenyl)urea Investigative 52946883 C21H20ClN3O2 381.9 CCC1=CC(=CC=C1)NC(=O)NC2=CC=CN(C2=O)CC3=CC=CC=C3Cl Ki ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B73AJR (3E,5E)-3,5-Bis[(4-pyrrolidin-1-ylphenyl)methylidene]oxan-4-one Investigative 118706206 C27H30N2O2 414.5 C1CN(CC1)C2=CC=C(C=C2)/C=C\\3/C(=O)/C(=C/C4=CC=C(C=C4)N5CCCC5)/COC3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B73XWZ 5-(4-Methylphenyl)-1-(4-methylsulfonylphenyl)tetrazole Investigative 57399160 C15H14N4O2S 314.4 CC1=CC=C(C=C1)C2=NN=NN2C3=CC=C(C=C3)S(=O)(=O)C IC50 = 87000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B75MIO (-)-Epiafzelechin Investigative 443639 C15H14O5 274.27 C1[C@H]([C@H](OC2=CC(=CC(=C21)O)O)C3=CC=C(C=C3)O)O IC50 = 69700 nM Poor binder T66665 Prostaglandin G/H synthase 2 B75WEK Huzhangoside B Investigative 49799269 C64H104O29 1337.5 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H](O[C@H]([C@@H]([C@H]2O)O)OC[C@@H]3[C@H]([C@@H]([C@H]([C@@H](O3)OC(=O)[C@@]45CC[C@@]6(C(=CC[C@H]7[C@]6(CC[C@@H]8[C@@]7(CC[C@@H](C8(C)C)O[C@H]9[C@@H]([C@H]([C@H](CO9)O)O)O[C@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)C)O)O[C@H]1[C@@H]([C@@H]([C@@H](CO1)O)O)O)O)C)C)[C@@H]4CC(CC5)(C)C)C)O)O)O)CO)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B79TIS 4-(2-(4-(Methylsulfonyl)phenyl)-1-phenylbut-1-enyl)phenol Investigative 11485761 C23H22O3S 378.5 CC/C(=C(\\C1=CC=CC=C1)/C2=CC=C(C=C2)O)/C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B79YHC 4-Methyl-3-[1-(4-methylsulfonylphenyl)-4-(trifluoromethyl)imidazol-2-yl]pyridine Investigative 10571870 C17H14F3N3O2S 381.4 CC1=C(C=NC=C1)C2=NC(=CN2C3=CC=C(C=C3)S(=O)(=O)C)C(F)(F)F IC50 = 54000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7C9XS 3-(5-Chlorofuran-2-yl)-4-(2-fluorophenyl)-5-methyl-1,2-oxazole Investigative 44194812 C14H9ClFNO2 277.68 CC1=C(C(=NO1)C2=CC=C(O2)Cl)C3=CC=CC=C3F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7DE4X N-[4-(4-Chlorophenoxy)phenyl]-4-hydroxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728407 C21H15ClN2O5S 442.9 C1=CC=C2C(=C1)C(=C(NS2(=O)=O)C(=O)NC3=CC=C(C=C3)OC4=CC=C(C=C4)Cl)O IC50 = 70000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7F0AP Methyl 3-(5-chlorofuran-2-yl)-5-phenyl-1,2-oxazole-4-carboxylate Investigative 57780779 C15H10ClNO4 303.69 COC(=O)C1=C(ON=C1C2=CC=C(O2)Cl)C3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7H9JQ 4-[5-(4-Fluoro-phenyl)-3-trifluoromethyl-pyrazol-1-yl]-N-methyl-benzenesulfonamide Investigative 10834744 C17H13F4N3O2S 399.4 CNS(=O)(=O)C1=CC=C(C=C1)N2C(=CC(=N2)C(F)(F)F)C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7HJC0 Mulberrin Investigative 5481958 C25H26O6 422.5 CC(=CCC1=C2C(=C(C=C1O)O)C(=O)C(=C(O2)C3=C(C=C(C=C3)O)O)CC=C(C)C)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7IZV6 (S)-Methyl 2-(2-(((benzyloxy)carbonyl)amino)-3-methylbutanamido)acetate Investigative 12951906 C16H22N2O5 322.36 CC(C)[C@@H](C(=O)NCC(=O)OC)NC(=O)OCC1=CC=CC=C1 IC50 = 75000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7JB2W N-(4-Chlorophenyl)-1-(4-methoxyphenyl)-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazole-3-carboxamide Investigative 90654428 C25H23ClN4O5 494.9 COC1=CC=C(C=C1)N2C(=NC(=N2)C(=O)NC3=CC=C(C=C3)Cl)C4=CC(=C(C(=C4)OC)OC)OC IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7LO6I 3-[5-Tert-butyl-3-(4-chlorophenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548444 C20H21ClN2O2 356.8 CC(C)(C)C1=NN(C(C1)C2=CC=C(C=C2)Cl)C3=CC=CC(=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7ML3F N-(Methylsulfonyl)-N-(2-(4-(2-(pyrrolidin-1-yl)ethoxy)phenoxy)phenyl)methanesulfonamide Investigative 49805304 C20H26N2O6S2 454.6 CS(=O)(=O)N(C1=CC=CC=C1OC2=CC=C(C=C2)OCCN3CCCC3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7MV3Q [3-(5-Chlorofuran-2-yl)-4-phenylisoxazol-5-yl]carboxylic acid Investigative 57780765 C14H8ClNO4 289.67 C1=CC=C(C=C1)C2=C(ON=C2C3=CC=C(O3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7NMA6 2-[4-(Methylsulfonyl)phenyl]-3-(4-fluorophenyl)pyrazine Investigative 10735037 C17H13FN2O2S 328.4 CS(=O)(=O)C1=CC=C(C=C1)C2=NC=CN=C2C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7P6VC Chembl4281362 Investigative 145982402 C15H11FN2O3S 318.3 C1=CC(=CC=C1C2=NOC(=C2)C3=CC=C(C=C3)S(=O)(=O)N)F IC50 = 81200 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7XQO0 3-Bromo-2-chloro-4-(4-fluorophenyl)-5-(4-methylsulfonylphenyl)-1H-pyrrole Investigative 10342564 C17H12BrClFNO2S 428.7 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C(=C(N2)Cl)Br)C3=CC=C(C=C3)F IC50 = 88000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7ZG0N 3-(4-Fluorophenyl)-5-iodo-2-(4-methylsulfonylphenyl)-1H-pyrrole Investigative 11743998 C17H13FINO2S 441.3 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C=C(N2)I)C3=CC=C(C=C3)F IC50 = 92300 nM Poor binder T66665 Prostaglandin G/H synthase 2 B7ZGJ8 2-[3-Fluoro-4-(3-isopropylphenyl)phenyl]propanoic acid Investigative 44336320 C18H19FO2 286.3 CC(C)C1=CC=CC(=C1)C2=C(C=C(C=C2)C(C)C(=O)O)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B82QYA 2-(9-Benzoyl-6-chlorocarbazol-2-yl)propanoic acid Investigative 71458884 C22H16ClNO3 377.8 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)C4=CC=CC=C4)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B82VUK 1-(5-Chloro-1,3-benzoxazol-2-yl)-N-[(1S,2S)-2-phenylmethoxycyclopentyl]piperidine-4-carboxamide Investigative 71720415 C25H28ClN3O3 454 C1C[C@@H]([C@H](C1)OCC2=CC=CC=C2)NC(=O)C3CCN(CC3)C4=NC5=C(O4)C=CC(=C5)Cl IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B87WOC N-(2-Aminophenyl)-3-(trifluoromethyl)benzamide Investigative 572426 C14H11F3N2O 280.24 C1=CC=C(C(=C1)N)NC(=O)C2=CC(=CC=C2)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B89HPQ Chembl4160466 Investigative 145957891 C23H24ClN7O2 465.9 C1CN(CCN1C2=CC=CC=C2)C3=NC(=NC(=N3)NC4=CC=C(C=C4)N5CCOCC5=O)Cl IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8AC1J 4-[5-Tert-butyl-3-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548266 C21H24N2O3 352.4 CC(C)(C)C1=NN(C(C1)C2=CC=C(C=C2)OC)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8AV3F 2-(4-Oxo-4H-1-benzopyran-3-ylmethyleneamino)benzoic acid Investigative 44582833 C17H11NO4 293.27 C1=CC=C2C(=C1)C(=O)C(=CO2)C=NC3=CC=CC=C3C(=O)O IC50 = 65720 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8CQB3 (+)-3,4,3',4'-Tetrahydroxy-9,7'alpha-epoxy-7alpha,9'-lactone Investigative 16681478 C18H16O7 344.3 C1[C@H]2[C@@H]([C@H](O1)C3=CC(=C(C=C3)O)O)C(=O)O[C@@H]2C4=CC(=C(C=C4)O)O IC50 = 90200 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8D3MA 4-Amino-N-[2-(trifluoromethyl)phenyl]benzamide Investigative 8566717 C14H11F3N2O 280.24 C1=CC=C(C(=C1)C(F)(F)F)NC(=O)C2=CC=C(C=C2)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8FR2U 1-(4-Methoxyphenyl)-N-methyl-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazole-3-carboxamide Investigative 90654426 C20H22N4O5 398.4 CNC(=O)C1=NN(C(=N1)C2=CC(=C(C(=C2)OC)OC)OC)C3=CC=C(C=C3)OC IC50 = 68200 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8FWA5 5-(4-Methoxyphenyl)-1-(4-methylsulfonylphenyl)tetrazole Investigative 57393944 C15H14N4O3S 330.4 COC1=CC=C(C=C1)C2=NN=NN2C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8JFB1 N-[4-(3,4-Dichlorophenyl)phenyl]-4-hydroxy-6-methoxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728423 C22H16Cl2N2O5S 491.3 COC1=CC2=C(C=C1)S(=O)(=O)NC(=C2O)C(=O)NC3=CC=C(C=C3)C4=CC(=C(C=C4)Cl)Cl IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8JV9Y 2-[6-Chloro-9-[(4-chlorophenyl)carbamoyl]carbazol-2-yl]propanoic acid Investigative 71453517 C22H16Cl2N2O3 427.3 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)NC4=CC=C(C=C4)Cl)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8LN2Z 2-Amino-N-[4-(trifluoromethyl)phenyl]benzamide Investigative 10564674 C14H11F3N2O 280.24 C1=CC=C(C(=C1)C(=O)NC2=CC=C(C=C2)C(F)(F)F)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8MJ1R 2-[4-[3-(Cyclobutylcarbamoyloxy)phenyl]-3-fluorophenyl]propanoic acid Investigative 90035911 C20H20FNO4 357.4 CC(C1=CC(=C(C=C1)C2=CC(=CC=C2)OC(=O)NC3CCC3)F)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8MSW5 2-(4-Fluoro-phenyl)-1-(3-methanesulfonyl-phenyl)-1H-pyrrole Investigative 10710438 C17H14FNO2S 315.4 CS(=O)(=O)C1=CC=CC(=C1)N2C=CC=C2C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8NAC4 2-[3-(Methoxymethyl)phenyl]-1-(4-methylsulfonylphenyl)-4-(trifluoromethyl)imidazole Investigative 10669268 C19H17F3N2O3S 410.4 COCC1=CC(=CC=C1)C2=NC(=CN2C3=CC=C(C=C3)S(=O)(=O)C)C(F)(F)F IC50 = 68100 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8NHC9 4-Hydroxy-N-[4-(4-methylphenyl)phenyl]-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728428 C22H18N2O4S 406.5 CC1=CC=C(C=C1)C2=CC=C(C=C2)NC(=O)C3=C(C4=CC=CC=C4S(=O)(=O)N3)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8PD7R 4-[3-(5-Chloro-furan-2-yl)-5-methyl-isoxazol-4-yl]-benzenesulfonamide Investigative 11382191 C14H11ClN2O4S 338.8 CC1=C(C(=NO1)C2=CC=C(O2)Cl)C3=CC=C(C=C3)S(=O)(=O)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8QYV1 1-(3-Chloro-4-methanesulfonyl-phenyl)-2-(4-fluoro-phenyl)-1H-pyrrole Investigative 10665504 C17H13ClFNO2S 349.8 CS(=O)(=O)C1=C(C=C(C=C1)N2C=CC=C2C3=CC=C(C=C3)F)Cl IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8SGL7 4-[2-[4-(Methylsulfonyl)phenyl]-1-cyclopentenyl]benzonitrile Investigative 10448879 C19H17NO2S 323.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(CCC2)C3=CC=C(C=C3)C#N IC50 = 77900 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8V2LE 2-[3-Fluoro-5-(trifluoromethyl)phenyl]-1-(4-methylsulfonylphenyl)-4-(trifluoromethyl)imidazole Investigative 10742264 C18H11F7N2O2S 452.3 CS(=O)(=O)C1=CC=C(C=C1)N2C=C(N=C2C3=CC(=CC(=C3)F)C(F)(F)F)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8WD3T Chembl4173819 Investigative 145951867 C20H19ClN6O2 410.9 CC1=CC=C(C=C1)NC2=NC(=NC(=N2)Cl)NC3=CC=C(C=C3)N4CCOCC4=O IC50 = 70000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8X3PM 2-[3-Fluoro-4-[3-(4-phenylbutylcarbamoyloxy)phenyl]phenyl]propanoic acid Investigative 73055093 C26H26FNO4 435.5 CC(C1=CC(=C(C=C1)C2=CC(=CC=C2)OC(=O)NCCCCC3=CC=CC=C3)F)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B8YRG4 4-[2-[3-(Trifluoromethyl)-4-fluorophenyl]-1-cyclopentenyl]-1-(methylsulfonyl)benzene Investigative 10786241 C19H16F4O2S 384.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(CCC2)C3=CC(=C(C=C3)F)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B90AZM 1-(2-(4-(2-(Methylsulfonyl)phenoxy)phenoxy)ethyl)pyrrolidine Investigative 49805051 C19H23NO4S 361.5 CS(=O)(=O)C1=CC=CC=C1OC2=CC=C(C=C2)OCCN3CCCC3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B93JUR 5-Acetyl-2-(3-carboxyanilino)benzoic acid Investigative 56964583 C16H13NO5 299.28 CC(=O)C1=CC(=C(C=C1)NC2=CC=CC(=C2)C(=O)O)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B96MIJ 7-Benzyl-5-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]methyl]-3-methyl-[1,2]oxazolo[4,5-d]pyridazin-4-one Investigative 70695977 C18H18N6O2S 382.4 CCNC1=NN=C(S1)CN2C(=O)C3=C(C(=N2)CC4=CC=CC=C4)ON=C3C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9BQK0 2-[4-(Methylsulfonyl)phenyl]-3-(4-fluorophenyl)-5-(methylsulfonyl)-1H-pyrrole Investigative 10000662 C18H16FNO4S2 393.5 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C=C(N2)S(=O)(=O)C)C3=CC=C(C=C3)F IC50 = 92300 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9CB4P 4-[5-Tert-butyl-3-(4-nitrophenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548267 C20H21N3O4 367.4 CC(C)(C)C1=NN(C(C1)C2=CC=C(C=C2)[N+](=O)[O-])C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9DB2V 2-[2-(4-Methylsulfonylphenyl)phenyl]quinoline Investigative 21223977 C22H17NO2S 359.4 CS(=O)(=O)C1=CC=C(C=C1)C2=CC=CC=C2C3=NC4=CC=CC=C4C=C3 IC50 = 57000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9EKJ4 1,2,3,4-Tetrafluoro-5-(4-fluorophenyl)-6-(4-methylsulfonylphenyl)benzene Investigative 11795129 C19H11F5O2S 398.3 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C(=C(C(=C2F)F)F)F)C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9EU3P Methyl 3-(5-chlorofuran-2-yl)-4-phenyl-1,2-oxazole-5-carboxylate Investigative 57780764 C15H10ClNO4 303.69 COC(=O)C1=C(C(=NO1)C2=CC=C(O2)Cl)C3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9EW6L 4-[5-(2-Methoxyphenyl)-3-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548445 C24H22N2O4 402.4 COC1=CC=C(C=C1)C2CC(=NN2C3=CC=C(C=C3)C(=O)O)C4=CC=CC=C4OC IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9EYG5 6-Chloro-8-(4-fluorophenyl)-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid Investigative 53316516 C17H9ClF4O3 372.7 C1=CC(=CC=C1C2=CC(=CC3=C2OC(C(=C3)C(=O)O)C(F)(F)F)Cl)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9F0DI 2-[3-(4-Bromophenyl)-1-phenylpyrazol-4-yl]-5-(4-chlorophenyl)-1,3,4-oxadiazole Investigative 90643444 C23H14BrClN4O 477.7 C1=CC=C(C=C1)N2C=C(C(=N2)C3=CC=C(C=C3)Br)C4=NN=C(O4)C5=CC=C(C=C5)Cl IC50 = 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9G0DM 2-[3-[3-Fluoro-5-(4-methoxyoxan-4-yl)phenoxy]propyl]-8-methoxy-5-[(4-methylsulfonylphenyl)methyl]-3,4-dihydro-1H-pyrido[4,3-b]indole;hydrochloride Investigative 46845034 C35H42ClFN2O6S 673.2 COC1=CC2=C(C=C1)N(C3=C2CN(CC3)CCCOC4=CC(=CC(=C4)C5(CCOCC5)OC)F)CC6=CC=C(C=C6)S(=O)(=O)C.Cl IC50 = 109200 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9HJV1 3-Fluoro-4-[3-(hexylcarbamoyloxy)phenyl]benzoic acid Investigative 127029897 C20H22FNO4 359.4 CCCCCCNC(=O)OC1=CC=CC(=C1)C2=C(C=C(C=C2)C(=O)O)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9I8KU 4-[5-(3-Methoxyphenyl)-3-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 68293474 C24H22N2O4 402.4 COC1=CC=C(C=C1)C2CC(=NN2C3=CC=C(C=C3)C(=O)O)C4=CC(=CC=C4)OC IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9LCQ3 2-(1-((1-(Difluoromethyl)-6-oxo-1,2,5,6-tetrahydropyridin-3-yl)methyl)-5-methoxy-2-methyl-1H-indol-3-yl)acetic acid Investigative 52946122 C19H20F2N2O4 378.4 CC1=C(C2=C(N1CC3=CCC(=O)N(C3)C(F)F)C=CC(=C2)OC)CC(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9MJ1F 1-(4-Fluoro-benzyl)-2-(4-methanesulfonyl-phenyl)-5-methyl-1H-pyrrole Investigative 10688742 C19H18FNO2S 343.4 CC1=CC=C(N1CC2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9NG5C 4-[5-Tert-butyl-3-(2-chlorophenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548632 C20H21ClN2O2 356.8 CC(C)(C)C1=NN(C(C1)C2=CC=CC=C2Cl)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9PBS0 [2-[3-[3-Fluoro-5-(4-methoxyoxan-4-yl)phenoxy]propyl]-8-methoxy-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]-(2,4,6-trichlorophenyl)methanone;hydrochloride Investigative 46906737 C34H35Cl4FN2O5 712.5 COC1=CC2=C(C=C1)N(C3=C2CN(CC3)CCCOC4=CC(=CC(=C4)C5(CCOCC5)OC)F)C(=O)C6=C(C=C(C=C6Cl)Cl)Cl.Cl IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9PO4E 1-[2,6-Ditert-butyl-4-[(Z)-2-(4-methylsulfonylphenyl)-1-phenylhex-1-enyl]phenyl]ethanone Investigative 76327240 C35H44O3S 544.8 CCCC/C(=C(\\C1=CC=CC=C1)/C2=CC(=C(C(=C2)C(C)(C)C)C(=O)C)C(C)(C)C)/C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9R3XB 3-[3-(Pentafluoro-lambda6-sulfanyl)anilino]benzoic acid Investigative 122192741 C13H10F5NO2S 339.28 C1=CC(=CC(=C1)NC2=CC(=CC=C2)S(F)(F)(F)(F)F)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9YD2X 1-(4-Methanesulfonyl-phenyl)-2-(2-methoxy-phenyl)-4-trifluoromethyl-1H-imidazole Investigative 10596883 C18H15F3N2O3S 396.4 COC1=CC=CC=C1C2=NC(=CN2C3=CC=C(C=C3)S(=O)(=O)C)C(F)(F)F IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 B9YWK4 N-Hydroxyethanesulfonamide Investigative 78363 C2H7NO3S 125.15 CCS(=O)(=O)NO IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BA0KH5 [2-[3-[3-Fluoro-5-(4-methoxyoxan-4-yl)phenoxy]propyl]-8-methoxy-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]-(2-fluorophenyl)methanone;hydrochloride Investigative 46906733 C34H37ClF2N2O5 627.1 COC1=CC2=C(C=C1)N(C3=C2CN(CC3)CCCOC4=CC(=CC(=C4)C5(CCOCC5)OC)F)C(=O)C6=CC=CC=C6F.Cl IC50 = 126000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BA37NI 2-{[2-Nitro-5-(trifluoromethyl)phenyl]amino}benzoic acid Investigative 45117711 C14H9F3N2O4 326.23 C1=CC=C(C(=C1)C(=O)O)NC2=C(C=CC(=C2)C(F)(F)F)[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BA7GZ2 2-(2,6-Dichloro-3-methylphenylamino)benzohydroxamic acid benzyl ester Investigative 24825638 C21H18Cl2N2O2 401.3 CC1=C(C(=C(C=C1)Cl)NC2=CC=CC=C2C(=O)NOCC3=CC=CC=C3)Cl IC50 = 66000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BABX61 6-Methoxy-2-(trifluoromethyl)-2H-chromene-3-carboxylic Acid Investigative 9965352 C12H9F3O4 274.19 COC1=CC2=C(C=C1)OC(C(=C2)C(=O)O)C(F)(F)F IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BAL2J3 4-[5-Tert-butyl-2-(4-carboxyphenyl)-3,4-dihydropyrazol-3-yl]-3-methoxybenzoic acid Investigative 129012347 C22H24N2O5 396.4 CC(C)(C)C1=NN(C(C1)C2=C(C=C(C=C2)C(=O)O)OC)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BAMX25 (2S)-2-[[(2S)-2-[(4-Fluorobenzoyl)amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-hydroxypropanoic acid Investigative 57391410 C19H19FN2O6 390.4 C1=CC(=CC=C1C[C@@H](C(=O)N[C@@H](CO)C(=O)O)NC(=O)C2=CC=C(C=C2)F)O IC50 = 140000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BAZ69R 6-Chloro-5-ethoxy-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid Investigative 53323225 C13H10ClF3O4 322.66 CCOC1=C(C=CC2=C1C=C(C(O2)C(F)(F)F)C(=O)O)Cl IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BB0M4S 4-[5-(2,5-Dichlorophenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzenesulfonamide Investigative 10526904 C16H10Cl2F3N3O2S 436.2 C1=CC(=CC=C1N2C(=CC(=N2)C(F)(F)F)C3=C(C=CC(=C3)Cl)Cl)S(=O)(=O)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BB34NM 3-[1-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-1H-pyrrol-2-yl]-propionic acid Investigative 10524261 C20H18FNO4S 387.4 CS(=O)(=O)C1=CC=C(C=C1)C2=CC=C(N2C3=CC=C(C=C3)F)CCC(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BB3EZ7 3-Methoxyacetaminophen Investigative 3080594 C9H11NO3 181.19 CC(=O)NC1=CC(=C(C=C1)O)OC IC50 = 138000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BB3Y7L 3-(4-(Methylsulfonyl)phenyl)-5-phenyl-4,5-dihydro-1H-pyrazole-1-carbothioamide Investigative 50906487 C17H17N3O2S2 359.5 CS(=O)(=O)C1=CC=C(C=C1)C2=NN(C(C2)C3=CC=CC=C3)C(=S)N IC50 = 50310 nM Poor binder T66665 Prostaglandin G/H synthase 2 BB4I2P (R)-2-[4-((1S,2R)-2-Hydroxy-cyclopentylmethyl)-phenyl]-propionic acid Investigative 13148390 C15H20O3 248.32 C[C@H](C1=CC=C(C=C1)C[C@@H]2CCC[C@H]2O)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BB6L0K 2-[6-Chloro-9-[(3-methoxyphenyl)methyl]carbazol-2-yl]propanoic acid Investigative 16098419 C23H20ClNO3 393.9 CC(C1=CC2=C(C=C1)C3=C(N2CC4=CC(=CC=C4)OC)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BB8HN9 1-[4,4-Diethyl-2-(4-methylsulfonylphenyl)-1-cyclopentenyl]-4-fluorobenzene Investigative 10022177 C22H25FO2S 372.5 CCC1(CC(=C(C1)C2=CC=C(C=C2)S(=O)(=O)C)C3=CC=C(C=C3)F)CC IC50 = 65000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BBQ83Y N-(3-Chloro-2-methylphenyl)-2-(2-oxochromen-4-yl)oxypropanamide Investigative 71462077 C19H16ClNO4 357.8 CC1=C(C=CC=C1Cl)NC(=O)C(C)OC2=CC(=O)OC3=CC=CC=C32 IC50 = 74910 nM Poor binder T66665 Prostaglandin G/H synthase 2 BC1QE2 [4,5-Bis(4-methoxyphenyl)-2-thiazolyl]-(4-methyl-1-piperazinyl)methanone Investigative 196841 C23H25N3O3S 423.5 CN1CCN(CC1)C(=O)C2=NC(=C(S2)C3=CC=C(C=C3)OC)C4=CC=C(C=C4)OC IC50 = 65000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BC20IJ 1,1,1-Trifluoro-N-[3-(4-hydroxyanilino)pyridin-4-yl]methanesulfonamide Investigative 76314063 C12H10F3N3O3S 333.29 C1=CC(=CC=C1NC2=C(C=CN=C2)NS(=O)(=O)C(F)(F)F)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BC2S1J 2-[(E)-3-(4-Pyrrolidin-1-ylphenyl)prop-2-enoyl]-3,4-dihydro-2H-naphthalen-1-one Investigative 90645133 C23H23NO2 345.4 C1CCN(C1)C2=CC=C(C=C2)/C=C/C(=O)C3CCC4=CC=CC=C4C3=O IC50 = 61230 nM Poor binder T66665 Prostaglandin G/H synthase 2 BC3G8X 4-[5-(4-Chlorophenyl)tetrazol-1-yl]benzenesulfonamide Investigative 57399158 C13H10ClN5O2S 335.77 C1=CC(=CC=C1C2=NN=NN2C3=CC=C(C=C3)S(=O)(=O)N)Cl IC50 = 62000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BC4N0Y 2-(1-(1-(Difluoromethyl)-2-oxo-1,2-dihydropyridine-4-carbonyl)-5-methoxy-2-methyl-1H-indol-3-yl)acetic acid Investigative 49765093 C19H16F2N2O5 390.3 CC1=C(C2=C(N1C(=O)C3=CC(=O)N(C=C3)C(F)F)C=CC(=C2)OC)CC(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BC4ZL5 6-[(2-Acetoxyphenyl)thio]hexanoic acid Investigative 9921835 C14H18O4S 282.36 CC(=O)OC1=CC=CC=C1SCCCCCC(=O)O IC50 = 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BC6UH3 1H-Pyrrole, 2-methyl-5-[4-(methylsulfonyl)phenyl]- Investigative 10799759 C12H13NO2S 235.3 CC1=CC=C(N1)C2=CC=C(C=C2)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BC82MP (R)-6-Chloro-7,8-dimethyl-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid Investigative 52948912 C13H10ClF3O3 306.66 CC1=C(C=C2C=C([C@@H](OC2=C1C)C(F)(F)F)C(=O)O)Cl IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BC91TJ (2E,5E)-2,5-Bis[[4-(dimethylamino)-2-nitrophenyl]methylidene]cyclopentan-1-one Investigative 90645122 C23H24N4O5 436.5 CN(C1=CC(=C(C=C1)/C=C\\2/C(=O)/C(=C/C3=C(C=C(C=C3)N(C)C)[N+](=O)[O-])/CC2)[N+](=O)[O-])C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BCDG20 1-(Carboxymethyl)-3,5-diphenyl-2-methylbenzene Investigative 10040599 C21H18O2 302.4 CC1=C(C=C(C=C1C2=CC=CC=C2)C3=CC=CC=C3)CC(=O)O IC50 = 120000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BCJ3Q4 2-(5,6-Dihydro-9-hydroxy-2-methyl-2,6-methano-2H-1-benzoxocin-4-yl)-5a,10a-dihydro-1,3,8,10a-tetrahydroxy-5a-(3-methyl-2-butenyl)-11H-benzofuro[3,2-b][1]benzopyran-11-one Investigative 44559963 C33H30O9 570.6 CC(=CCC12C3=C(C=C(C=C3)O)OC1(C(=O)C4=C(O2)C=C(C(=C4O)C5=CC6(CC(C5)C7=C(O6)C=C(C=C7)O)C)O)O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BCJ61T Sodium;2-[4-[(2-oxocyclopentyl)methyl]-3-[4-(trifluoromethoxy)phenyl]phenyl]propanoate Investigative 56675533 C22H20F3NaO4 428.4 CC(C1=CC(=C(C=C1)CC2CCCC2=O)C3=CC=C(C=C3)OC(F)(F)F)C(=O)[O-].[Na+] IC50 = 72000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BCO04V N-[4-(2,3-Dimethylphenyl)phenyl]-4-hydroxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728417 C23H20N2O4S 420.5 CC1=C(C(=CC=C1)C2=CC=C(C=C2)NC(=O)C3=C(C4=CC=CC=C4S(=O)(=O)N3)O)C IC50 = 94700 nM Poor binder T66665 Prostaglandin G/H synthase 2 BCOB05 2-[6-Chloro-9-(hexylcarbamoyl)carbazol-2-yl]propanoic acid Investigative 71458883 C22H25ClN2O3 400.9 CCCCCCNC(=O)N1C2=C(C=C(C=C2)Cl)C3=C1C=C(C=C3)C(C)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BCS4L6 Ciwujianoside C3 Investigative 21626481 C53H86O21 1059.2 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H](O[C@H]([C@@H]([C@H]2O)O)OC[C@@H]3[C@H]([C@@H]([C@H]([C@@H](O3)OC(=O)[C@@]45CC[C@@]6(C(=CC[C@H]7[C@]6(CC[C@@H]8[C@@]7(CC[C@@H](C8(C)C)O[C@H]9[C@@H]([C@H]([C@H](CO9)O)O)O)C)C)[C@@H]4CC(CC5)(C)C)C)O)O)O)CO)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BCS64T 2-Ethyl-1-(4-fluorophenyl)-5-(4-methylsulfonylphenyl)pyrrole Investigative 10807315 C19H18FNO2S 343.4 CCC1=CC=C(N1C2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BCW57P N-[(5-Bromo-8-hydroxy-7-quinolinyl)-thiophen-2-ylmethyl]acetamide Investigative 44460175 C16H13BrN2O2S 377.3 CC(=O)NC(C1=CC=CS1)C2=CC(=C3C=CC=NC3=C2O)Br IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BD25RC 2-(4-Tert-Butylphenyl)-4-(4-fluorophenyl)-5-[4-(methylsulfonyl)phenyl]thiazole Investigative 44271105 C26H24FNO2S2 465.6 CC(C)(C)C1=CC=C(C=C1)C2=NC(=C(S2)C3=CC=C(C=C3)S(=O)(=O)C)C4=CC=C(C=C4)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BD27MZ 1-(2-(4-(4-(Methylsulfonyl)-2-nitrophenoxy)phenoxy)ethyl)pyrrolidine Investigative 49805054 C19H22N2O6S 406.5 CS(=O)(=O)C1=CC(=C(C=C1)OC2=CC=C(C=C2)OCCN3CCCC3)[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BD2UY4 1-(2-(4-(4-Nitrophenoxy)phenoxy)ethyl)pyrrolidine Investigative 49804919 C18H20N2O4 328.4 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=C(C=C3)[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BD5Q3N 4-(4-Fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-5-trifluoromethyl-1H-pyrazole Investigative 15380222 C17H12F4N2O2S 384.3 CS(=O)(=O)C1=CC=C(C=C1)C2=NNC(=C2C3=CC=C(C=C3)F)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BD8I2Z 2-Phenyl-4-cyclohexyl-5-[4-(methylsulfonyl)phenyl]oxazole Investigative 22624559 C22H23NO3S 381.5 CS(=O)(=O)C1=CC=C(C=C1)C2=C(N=C(O2)C3=CC=CC=C3)C4CCCCC4 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BD8PK7 4-Methyl-2-[5-(2-methylphenyl)-1H-pyrazol-3-yl]phenol Investigative 775994 C17H16N2O 264.32 CC1=CC(=C(C=C1)O)C2=NNC(=C2)C3=CC=CC=C3C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BDC07X N-[2-Cyano-4-(trifluoromethyl)phenyl]-2-(2-oxochromen-4-yl)oxypropanamide Investigative 71460385 C20H13F3N2O4 402.3 CC(C(=O)NC1=C(C=C(C=C1)C(F)(F)F)C#N)OC2=CC(=O)OC3=CC=CC=C32 IC50 = 50250 nM Poor binder T66665 Prostaglandin G/H synthase 2 BDE9W0 3-Nitrooxypropyl 3-(5-chlorofuran-2-yl)-4-phenyl-1,2-oxazole-5-carboxylate Investigative 57780777 C17H13ClN2O7 392.7 C1=CC=C(C=C1)C2=C(ON=C2C3=CC=C(O3)Cl)C(=O)OCCCO[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BDJ0F2 4-[2-Oxo-4-(4-sulfamoyl-phenyl)-oxazol-3-yl]-benzoic acid Investigative 10808453 C16H12N2O6S 360.3 C1=CC(=CC=C1C2=COC(=O)N2C3=CC=C(C=C3)C(=O)O)S(=O)(=O)N IC50 = 59000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BDP45T 1-[2-(4-Phenoxyphenoxy)ethyl]pyrrolidine Investigative 9993978 C18H21NO2 283.4 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BDU3J9 (2R)-2-[6-Chloro-9-(4-chlorobenzoyl)carbazol-2-yl]propanoic acid Investigative 71449872 C22H15Cl2NO3 412.3 C[C@H](C1=CC2=C(C=C1)C3=C(N2C(=O)C4=CC=C(C=C4)Cl)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BE41BL 4-[5-(4-Fluoro-phenyl)-3-trifluoromethyl-pyrazol-1-yl]-N,N-dimethyl-benzenesulfonamide Investigative 10549657 C18H15F4N3O2S 413.4 CN(C)S(=O)(=O)C1=CC=C(C=C1)N2C(=CC(=N2)C(F)(F)F)C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BE4T2Y 2-[6-Chloro-9-(4-chlorophenyl)sulfonylcarbazol-2-yl]propanoic acid Investigative 16098411 C21H15Cl2NO4S 448.3 CC(C1=CC2=C(C=C1)C3=C(N2S(=O)(=O)C4=CC=C(C=C4)Cl)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BE50XS 1-(4-Methylsulfonylphenyl)-5-[4-(trifluoromethyl)phenyl]tetrazole Investigative 57393945 C15H11F3N4O2S 368.3 CS(=O)(=O)C1=CC=C(C=C1)N2C(=NN=N2)C3=CC=C(C=C3)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BE7GR5 2-(2,6-Dichloro-3-methyl-phenylamino)-N-isopropoxy-benzamide Investigative 44365785 C18H20Cl2N2O2 367.3 CC1=C(C(=C(C=C1)Cl)NC2=CC=CC=C2C(=O)NOC(C)(C)C)Cl IC50 = 66000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BE7PD5 1-(2-(4-(2,4-Dinitrophenoxy)phenoxy)ethyl)pyrrolidine Investigative 49804920 C18H19N3O6 373.4 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=C(C=C(C=C3)[N+](=O)[O-])[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BEL35F 3-[2-(4-Methylsulfonylphenyl)phenyl]pyridine Investigative 21223973 C18H15NO2S 309.4 CS(=O)(=O)C1=CC=C(C=C1)C2=CC=CC=C2C3=CN=CC=C3 IC50 = 87000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BEM15W 2-(1-(1-(Difluoromethyl)-6-oxo-1,2,5,6-tetrahydropyridine-3-carbonyl)-5-methoxy-2-methyl-1H-indol-3-yl)acetic acid Investigative 52941574 C19H18F2N2O5 392.4 CC1=C(C2=C(N1C(=O)C3=CCC(=O)N(C3)C(F)F)C=CC(=C2)OC)CC(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BEMZ75 4-[5-Tert-butyl-3-(4-chlorophenyl)-3,4-dihydropyrazol-2-yl]benzenesulfonic acid Investigative 66548636 C19H21ClN2O3S 392.9 CC(C)(C)C1=NN(C(C1)C2=CC=C(C=C2)Cl)C3=CC=C(C=C3)S(=O)(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BEV83K (5Z)-2-[1-(6-Methoxynaphthalen-2-yl)ethyl]-5-(naphthalen-1-ylmethylidene)-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one Investigative 118729079 C28H21N3O2S 463.6 CC(C1=CC2=C(C=C1)C=C(C=C2)OC)C3=NN4C(=O)/C(=C/C5=CC=CC6=CC=CC=C65)/SC4=N3 IC50 = 68200 nM Poor binder T66665 Prostaglandin G/H synthase 2 BEVP95 5-(4-(Methylsulfonyl)phenyl)-4-phenyl-3H-1,2-dithiole-3-thione Investigative 11175990 C16H12O2S4 364.5 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C(=S)SS2)C3=CC=CC=C3 IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BF0B3H N-[4-(3-Chlorophenyl)phenyl]-4-hydroxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728411 C21H15ClN2O4S 426.9 C1=CC=C2C(=C1)C(=C(NS2(=O)=O)C(=O)NC3=CC=C(C=C3)C4=CC(=CC=C4)Cl)O IC50 = 74700 nM Poor binder T66665 Prostaglandin G/H synthase 2 BF41IZ 2-[4-[3-(Cyclopentylcarbamoyloxy)phenyl]-3-fluorophenyl]propanoic acid Investigative 73054543 C21H22FNO4 371.4 CC(C1=CC(=C(C=C1)C2=CC(=CC=C2)OC(=O)NC3CCCC3)F)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BF4GR7 4-[3-Difluoromethyl-5-(2,5-dimethyl-phenyl)-pyrazol-1-yl]-benzenesulfonamide Investigative 10643308 C18H17F2N3O2S 377.4 CC1=CC(=C(C=C1)C)C2=CC(=NN2C3=CC=C(C=C3)S(=O)(=O)N)C(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BFN8I4 (5Z)-2-[1-(6-Methoxynaphthalen-2-yl)ethyl]-5-[(4-propan-2-ylphenyl)methylidene]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one Investigative 118729071 C27H25N3O2S 455.6 CC(C)C1=CC=C(C=C1)/C=C\\2/C(=O)N3C(=NC(=N3)C(C)C4=CC5=C(C=C4)C=C(C=C5)OC)S2 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BFO4C7 Chembl4169332 Investigative 145955075 C15H15ClN8O3 390.78 C1COCC(=O)N1C2=CC=C(C=C2)NC3=NC(=NC(=N3)Cl)OCCN=[N+]=[N-] IC50 = 75000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BFU91R 2,4,6-Trimethyl-3-(5-methyl-4-phenyl-isoxazol-3-yl)-benzenesulfonamide Investigative 11302745 C19H20N2O3S 356.4 CC1=CC(=C(C(=C1C2=NOC(=C2C3=CC=CC=C3)C)C)S(=O)(=O)N)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BFV74L p-Terphenyl Investigative 7115 C18H14 230.3 C1=CC=C(C=C1)C2=CC=C(C=C2)C3=CC=CC=C3 IC50 = 144000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BFX1O9 4-(4-Chlorophenyl)-5-p-tolyl-3H-1,2-dithiole-3-thione Investigative 44564507 C16H11ClS3 334.9 CC1=CC=C(C=C1)C2=C(C(=S)SS2)C3=CC=C(C=C3)Cl IC50 = 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BG0XT2 [(1S,2S,6R,10S,11R,13S,14R,15R)-14-Acetyloxy-1,6-dihydroxy-8-(hydroxymethyl)-4,12,12,15-tetramethyl-5,9-dioxo-13-tetracyclo[8.5.0.02,6.011,13]pentadeca-3,7-dienyl] 2-methylbutanoate Investigative 118727933 C27H36O9 504.6 CCC(C)C(=O)O[C@@]12[C@@H](C1(C)C)[C@@H]3C(=O)C(=C[C@]4([C@H]([C@]3([C@@H]([C@H]2OC(=O)C)C)O)C=C(C4=O)C)O)CO IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BG2A9V 3-[1-(3-Chloro-phenoxy)-2,2,2-trifluoro-ethyl]-1-(4-fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-methyl-1H-pyrrole Investigative 10816219 C26H20ClF4NO3S 538 CC1=C(C=C(N1C2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)C)C(C(F)(F)F)OC4=CC(=CC=C4)Cl IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BG8CK2 4-[2-(3,4,5-Trifluorophenyl)-1-cyclopentenyl]-1-(methylsulfonyl)benzene Investigative 10641720 C18H15F3O2S 352.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(CCC2)C3=CC(=C(C(=C3)F)F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BG8ZO2 2-(2-Chloro-6-methyl-phenyl)-1-(4-methanesulfonyl-phenyl)-4-trifluoromethyl-1H-imidazole Investigative 10645484 C18H14ClF3N2O2S 414.8 CC1=C(C(=CC=C1)Cl)C2=NC(=CN2C3=CC=C(C=C3)S(=O)(=O)C)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BGCZ96 3-(4-Methylsulfonylphenyl)-4-phenylphenol Investigative 15871996 C19H16O3S 324.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C=CC(=C2)O)C3=CC=CC=C3 IC50 = 147000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BGI7H3 6-Chloro-7-((2,5-dimethylpyrrolidin-1-yl)methyl)-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid Investigative 53323226 C18H19ClF3NO3 389.8 CC1CCC(N1CC2=C(C=C3C=C(C(OC3=C2)C(F)(F)F)C(=O)O)Cl)C IC50 = 96000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BGJ2B9 2-[4-[3-(Cyclohexylmethylcarbamoyloxy)phenyl]-3-fluorophenyl]propanoic acid Investigative 73054545 C23H26FNO4 399.5 CC(C1=CC(=C(C=C1)C2=CC(=CC=C2)OC(=O)NCC3CCCCC3)F)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BGJ53O 4-[5-(Difluoromethyl)-2-(4-sulfamoylphenyl)pyrazol-3-yl]benzamide Investigative 10715523 C17H14F2N4O3S 392.4 C1=CC(=CC=C1C2=CC(=NN2C3=CC=C(C=C3)S(=O)(=O)N)C(F)F)C(=O)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BGMO76 N-[4-(3,4-Dichlorophenyl)phenyl]-4,6-dihydroxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728424 C21H14Cl2N2O5S 477.3 C1=CC(=CC=C1C2=CC(=C(C=C2)Cl)Cl)NC(=O)C3=C(C4=C(C=CC(=C4)O)S(=O)(=O)N3)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BGP49B 1-(2-(4-(4-(Trifluoromethyl)phenoxy)phenoxy)ethyl)pyrrolidine Investigative 49805177 C19H20F3NO2 351.4 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=C(C=C3)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BGQ01J 2-[6-Chloro-9-(octylcarbamoyl)carbazol-2-yl]propanoic acid Investigative 71449873 C24H29ClN2O3 428.9 CCCCCCCCNC(=O)N1C2=C(C=C(C=C2)Cl)C3=C1C=C(C=C3)C(C)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BGQ3F1 6-Chloro-7-(diisopropylamino)-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid Investigative 53320186 C17H19ClF3NO3 377.8 CC(C)N(C1=C(C=C2C=C(C(OC2=C1)C(F)(F)F)C(=O)O)Cl)C(C)C IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BGR5K1 4-Amino-N-[5-(trifluoromethyl)pyridin-2-yl]benzamide Investigative 24854031 C13H10F3N3O 281.23 C1=CC(=CC=C1C(=O)NC2=NC=C(C=C2)C(F)(F)F)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BGY4M8 N-[3-(3,5-Dimethylanilino)pyridin-4-yl]methanesulfonamide Investigative 76335832 C14H17N3O2S 291.37 CC1=CC(=CC(=C1)NC2=C(C=CN=C2)NS(=O)(=O)C)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BH32JZ (2R)-2-[4-[[(1R,2S)-2-Hydroxycyclopentyl]methyl]phenyl]propanoic acid Investigative 13148391 C15H20O3 248.32 C[C@H](C1=CC=C(C=C1)C[C@H]2CCC[C@@H]2O)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BH53MB 4-[5-(4-Fluorophenyl)-4-propyl-3-(trifluoromethyl)pyrazol-1-yl]benzenesulfonamide Investigative 10717364 C19H17F4N3O2S 427.4 CCCC1=C(N(N=C1C(F)(F)F)C2=CC=C(C=C2)S(=O)(=O)N)C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BH57JZ 3-(5-Chlorofuran-2-yl)-4-phenyl-5-(trifluoromethyl)-1,2-oxazole Investigative 44194814 C14H7ClF3NO2 313.66 C1=CC=C(C=C1)C2=C(ON=C2C3=CC=C(O3)Cl)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BH71VQ 2-[6-Chloro-9-(cyclohexylcarbamoyl)carbazol-2-yl]propanoic acid Investigative 71453518 C22H23ClN2O3 398.9 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)NC4CCCCC4)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BH9C3M 2-{4-[4-Chloro-1-(4-(methylsulfonyl)phenyl)-1H-imidazol-5-yl]-2-fluorophenoxy}ethanol Investigative 16125427 C18H16ClFN2O4S 410.8 CS(=O)(=O)C1=CC=C(C=C1)N2C=NC(=C2C3=CC(=C(C=C3)OCCO)F)Cl IC50 = 56000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BHB71Y [1-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-methyl-1H-pyrrol-3-ylmethyl]-dimethyl-amine Investigative 10738921 C21H23FN2O2S 386.5 CC1=C(C=C(N1C2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)C)CN(C)C IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BHBD92 N-(3-Anilinopyridin-4-yl)-N-cyclopropylsulfonylcyclopropanesulfonamide Investigative 76317623 C17H19N3O4S2 393.5 C1CC1S(=O)(=O)N(C2=C(C=NC=C2)NC3=CC=CC=C3)S(=O)(=O)C4CC4 IC50 = 56760 nM Poor binder T66665 Prostaglandin G/H synthase 2 BHC31I 1,4-Benzodioxan-6-ylacetic acid Investigative 87020 C10H10O4 194.18 C1COC2=C(O1)C=CC(=C2)CC(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BHIO47 2,6-Di-tert-butyl-4-(5-propylsulfanyl-[1,3,4]thiadiazol-2-yl)-phenol Investigative 135503854 C19H28N2OS2 364.6 CCCSC1=NN=C(S1)C2=CC(=C(C(=C2)C(C)(C)C)O)C(C)(C)C IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BHL71Y 2-(9-Benzyl-6-chlorocarbazol-2-yl)propanoic acid Investigative 71458880 C22H18ClNO2 363.8 CC(C1=CC2=C(C=C1)C3=C(N2CC4=CC=CC=C4)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BHLF89 2-(6-Chloro-9H-carbazole-2-yl)propionic acid methyl ester Investigative 14049818 C16H14ClNO2 287.74 CC(C1=CC2=C(C=C1)C3=C(N2)C=CC(=C3)Cl)C(=O)OC IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BHQ0N6 3-(1,3-Benzodioxol-4-yl)-2-(4-methylphenyl)sulfonyl-5-(trifluoromethyl)-3,4-dihydropyrazole Investigative 118706123 C18H15F3N2O4S 412.4 CC1=CC=C(C=C1)S(=O)(=O)N2C(CC(=N2)C(F)(F)F)C3=C4C(=CC=C3)OCO4 IC50 = 57360 nM Poor binder T66665 Prostaglandin G/H synthase 2 BHS07O Methyl 3-[(4-nitronaphthalen-1-yl)amino]benzoate Investigative 70911877 C18H14N2O4 322.3 COC(=O)C1=CC(=CC=C1)NC2=CC=C(C3=CC=CC=C32)[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BHU2X5 (E)-2-[3-(2,4-Difluorophenyl)phenyl]-3-(4-methylsulfonylphenyl)prop-2-enoic acid Investigative 76316303 C22H16F2O4S 414.4 CS(=O)(=O)C1=CC=C(C=C1)/C=C(\\C2=CC=CC(=C2)C3=C(C=C(C=C3)F)F)/C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BHY3C0 (2R)-2-[6-Chloro-9-(1,3-oxazole-4-carbonyl)carbazol-2-yl]propanoic acid Investigative 71457024 C19H13ClN2O4 368.8 C[C@H](C1=CC2=C(C=C1)C3=C(N2C(=O)C4=COC=N4)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BHYC34 (2S)-2-[[(2S)-2-[(4-Fluorobenzoyl)amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-hydroxypropanoic acid Investigative 57394899 C21H20FN3O5 413.4 C1=CC=C2C(=C1)C(=CN2)C[C@@H](C(=O)N[C@@H](CO)C(=O)O)NC(=O)C3=CC=C(C=C3)F IC50 = 200000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BI3R0K Acetic acid 2-(4-cyano-butylsulfanyl)-phenyl ester Investigative 10848242 C13H15NO2S 249.33 CC(=O)OC1=CC=CC=C1SCCCCC#N IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BI85SU 2-[3-Fluoro-4-[3-(propylcarbamoyloxy)phenyl]phenyl]propanoic acid Investigative 90036150 C19H20FNO4 345.4 CCCNC(=O)OC1=CC=CC(=C1)C2=C(C=C(C=C2)C(C)C(=O)O)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BI8E6T 4-[5-Tert-butyl-3-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 68291773 C21H24N2O2 336.4 CC1=CC=C(C=C1)C2CC(=NN2C3=CC=C(C=C3)C(=O)O)C(C)(C)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BI93DJ 2-Amino-N-[2-(trifluoromethyl)phenyl]benzamide Investigative 5080393 C14H11F3N2O 280.24 C1=CC=C(C(=C1)C(=O)NC2=CC=CC=C2C(F)(F)F)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BI98CZ 4-[3-(Difluoromethyl)-5-(4-methylsulfonylphenyl)pyrazol-1-yl]benzenesulfonamide Investigative 11796738 C17H15F2N3O4S2 427.4 CS(=O)(=O)C1=CC=C(C=C1)C2=CC(=NN2C3=CC=C(C=C3)S(=O)(=O)N)C(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BI9F1Z 4-[5-Tert-butyl-3-(4-ethoxyphenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548448 C22H26N2O3 366.5 CCOC1=CC=C(C=C1)C2CC(=NN2C3=CC=C(C=C3)C(=O)O)C(C)(C)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BIEW03 2-[3-Fluoro-4-[3-(2-phenylethylcarbamoyloxy)phenyl]phenyl]propanoic acid Investigative 73054548 C24H22FNO4 407.4 CC(C1=CC(=C(C=C1)C2=CC(=CC=C2)OC(=O)NCCC3=CC=CC=C3)F)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BIF8Y2 N-(3-Cyclopentylamino-4-pyridinyl)methanesulfonamide Investigative 44473651 C11H17N3O2S 255.34 CS(=O)(=O)NC1=C(C=NC=C1)NC2CCCC2 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BIH3Y1 Chembl4290080 Investigative 145989313 C19H21NO3SSi 371.5 C[Si](C)(C)C1=C(ON=C1C2=CC=CC=C2)C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BIM75L Meclofenamic acid derivative, 27 Investigative 10409583 C22H20Cl2N2O2 415.3 CC1=C(C(=C(C=C1)Cl)NC2=CC=CC=C2C(=O)NCCOC3=CC=CC=C3)Cl IC50 = 66000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BINJ79 2-[6-Chloro-9-[(4-cyanophenyl)methyl]carbazol-2-yl]propanoic acid Investigative 71457025 C23H17ClN2O2 388.8 CC(C1=CC2=C(C=C1)C3=C(N2CC4=CC=C(C=C4)C#N)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BIPY25 N-(3-Aminopyridin-2-yl)-4-(trifluoromethyl)benzamide Investigative 24853950 C13H10F3N3O 281.23 C1=CC(=C(N=C1)NC(=O)C2=CC=C(C=C2)C(F)(F)F)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BIRD47 N-[4-(3,4-Dimethylphenyl)phenyl]-4-hydroxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728429 C23H20N2O4S 420.5 CC1=C(C=C(C=C1)C2=CC=C(C=C2)NC(=O)C3=C(C4=CC=CC=C4S(=O)(=O)N3)O)C IC50 ~ 57700 nM Poor binder T66665 Prostaglandin G/H synthase 2 BIV25M 2-Fluoro-1-methoxy-4-[2-(4-methylsulfonylphenyl)phenyl]benzene Investigative 10546170 C20H17FO3S 356.4 COC1=C(C=C(C=C1)C2=CC=CC=C2C3=CC=C(C=C3)S(=O)(=O)C)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BIV78W 2,4,6-Trimethyl-3-[5-methyl-4-(4-sulfamoyl-phenyl)-isoxazol-3-yl]-benzenesulfonamide Investigative 11487377 C19H21N3O5S2 435.5 CC1=CC(=C(C(=C1C2=NOC(=C2C3=CC=C(C=C3)S(=O)(=O)N)C)C)S(=O)(=O)N)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BIWU85 5-[(5-Anilino-1,3,4-thiadiazol-2-yl)methyl]-7-[(4-methoxyphenyl)methyl]-3-methyl-[1,2]oxazolo[4,5-d]pyridazin-4-one Investigative 70687599 C23H20N6O3S 460.5 CC1=NOC2=C1C(=O)N(N=C2CC3=CC=C(C=C3)OC)CC4=NN=C(S4)NC5=CC=CC=C5 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BIX5H6 1,5-Diphenyl-3-trifluoromethyl-1H-pyrazole Investigative 10424186 C16H11F3N2 288.27 C1=CC=C(C=C1)C2=CC(=NN2C3=CC=CC=C3)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJ0G8A 2-[3-Fluoro-4-[3-(2-methylpropylcarbamoyloxy)phenyl]phenyl]propanoic acid Investigative 73054544 C20H22FNO4 359.4 CC(C)CNC(=O)OC1=CC=CC(=C1)C2=C(C=C(C=C2)C(C)C(=O)O)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJ0OZ2 5-[[5-(Ethylamino)-1,3,4-thiadiazol-2-yl]methyl]-7-[(4-methoxyphenyl)methyl]-3-methyl-[1,2]oxazolo[4,5-d]pyridazin-4-one Investigative 70693860 C19H20N6O3S 412.5 CCNC1=NN=C(S1)CN2C(=O)C3=C(C(=N2)CC4=CC=C(C=C4)OC)ON=C3C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJ0Y1Z 2-(Phenylacetyloxy)Ethanesulfonylhydroxamic Acid Investigative 51351150 C10H13NO5S 259.279 C1=CC=C(C=C1)CC(=O)OCCS(=O)(=O)NO IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJ24DB 2-(4-Chlorophenyl)-3-(4-methylsulfonylanilino)-1,3-thiazolidin-4-one Investigative 70689056 C16H15ClN2O3S2 382.9 CS(=O)(=O)C1=CC=C(C=C1)NN2C(SCC2=O)C3=CC=C(C=C3)Cl IC50 = 121700 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJ27AZ Sodium;2-[4-[(2-oxocyclopentyl)methyl]-2-phenylphenyl]propanoate Investigative 56665216 C21H21NaO3 344.4 CC(C1=C(C=C(C=C1)CC2CCCC2=O)C3=CC=CC=C3)C(=O)[O-].[Na+] IC50 = 70000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJ3VO6 4-(4-Methanesulfonyl-phenyl)-3-phenyl-5H-[1,2]oxathiole 2-oxide Investigative 11450459 C16H14O4S2 334.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(S(=O)OC2)C3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJ4D1F 3-Methyl-4-(4-fluorophenyl)-5-[4-(methylsulfonyl)phenyl]isoxazole Investigative 10947517 C17H14FNO3S 331.4 CC1=NOC(=C1C2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJ4FV3 Hederasaponin B Investigative 21626480 C59H96O25 1205.4 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H](O[C@H]([C@@H]([C@H]2O)O)OC[C@@H]3[C@H]([C@@H]([C@H]([C@@H](O3)OC(=O)[C@@]45CC[C@@]6(C(=CC[C@H]7[C@]6(CC[C@@H]8[C@@]7(CC[C@@H](C8(C)C)O[C@H]9[C@@H]([C@H]([C@H](CO9)O)O)O[C@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)C)O)O)O)C)C)[C@@H]4CC(CC5)(C)C)C)O)O)O)CO)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJ95GE 4-[5-Tert-butyl-3-(3-fluorophenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548634 C20H21FN2O2 340.4 CC(C)(C)C1=NN(C(C1)C2=CC(=CC=C2)F)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJ9FO6 Chembl4160157 Investigative 145960574 C22H23ClN6O5S 519 CC1=CC=C(C=C1)S(=O)(=O)NCCOC2=NC(=NC(=N2)NC3=CC=C(C=C3)N4CCOCC4=O)Cl IC50 = 80000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJAG15 N-(4-(4-(2-(Pyrrolidin-1-yl)ethoxy)phenoxy)phenyl)methanesulfonamide Investigative 49805306 C19H24N2O4S 376.5 CS(=O)(=O)NC1=CC=C(C=C1)OC2=CC=C(C=C2)OCCN3CCCC3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJBH34 2-Pyridinecarboxylic acid, 6-((5-chloro-2-((4-chloro-2-fluorophenyl)methoxy)phenyl)methyl)-, sodium salt Investigative 23696973 C20H13Cl2FNNaO3 428.2 C1=CC(=NC(=C1)C(=O)[O-])CC2=C(C=CC(=C2)Cl)OCC3=C(C=C(C=C3)Cl)F.[Na+] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJM3H2 7-Benzyl-3-methyl-5-[(4-phenyl-5-sulfanylidene-1H-1,2,4-triazol-3-yl)methyl]-[1,2]oxazolo[4,5-d]pyridazin-4-one Investigative 70681274 C22H18N6O2S 430.5 CC1=NOC2=C1C(=O)N(N=C2CC3=CC=CC=C3)CC4=NNC(=S)N4C5=CC=CC=C5 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BJON65 [2-[3-[3-Fluoro-5-(4-methoxyoxan-4-yl)phenoxy]propyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]-phenylmethanone;hydrochloride Investigative 46906731 C33H36ClFN2O4 579.1 COC1(CCOCC1)C2=CC(=CC(=C2)F)OCCCN3CCC4=C(C3)C5=CC=CC=C5N4C(=O)C6=CC=CC=C6.Cl IC50 = 101900 nM Poor binder T66665 Prostaglandin G/H synthase 2 BK0ZF6 5-Methyl-3-(oxolan-2-yl)-4-phenyl-1,2-oxazole Investigative 44194816 C14H15NO2 229.27 CC1=C(C(=NO1)C2CCCO2)C3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BK1Y5E 2-(5-Fluoro-2-methyl-phenyl)-1-(4-methanesulfonyl-phenyl)-4-trifluoromethyl-1H-imidazole Investigative 10810863 C18H14F4N2O2S 398.4 CC1=C(C=C(C=C1)F)C2=NC(=CN2C3=CC=C(C=C3)S(=O)(=O)C)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BK4I2Z 2-(6-Chloro-9-hexylsulfonylcarbazol-2-yl)propanoic acid Investigative 71460692 C21H24ClNO4S 421.9 CCCCCCS(=O)(=O)N1C2=C(C=C(C=C2)Cl)C3=C1C=C(C=C3)C(C)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BK5JL2 (3E,5E)-1-Benzyl-3,5-bis[(4-pyrrolidin-1-ylphenyl)methylidene]piperidin-4-one Investigative 118706209 C34H37N3O 503.7 C1CN(CC1)C2=CC=C(C=C2)/C=C\\3/C(=O)/C(=C/C4=CC=C(C=C4)N5CCCC5)/CN(C3)CC6=CC=CC=C6 IC50 = 57220 nM Poor binder T66665 Prostaglandin G/H synthase 2 BK5O4P 4-[4-Chloro-5-[3-fluoro-4-(3-hydroxypropoxy)phenyl]imidazol-1-yl]benzenesulfonamide Investigative 16125422 C18H17ClFN3O4S 425.9 C1=CC(=CC=C1N2C=NC(=C2C3=CC(=C(C=C3)OCCCO)F)Cl)S(=O)(=O)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BK70EO Methyl 3,5-diphenyl-4-isoxazolecarboxylate Investigative 827480 C17H13NO3 279.29 COC(=O)C1=C(ON=C1C2=CC=CC=C2)C3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BK7D2P (2E)-2-[(4-Pyrrolidin-1-ylphenyl)methylidene]-3H-inden-1-one Investigative 38864639 C20H19NO 289.4 C1CCN(C1)C2=CC=C(C=C2)/C=C/3\\CC4=CC=CC=C4C3=O IC50 = 54640 nM Poor binder T66665 Prostaglandin G/H synthase 2 BKD8E4 4-[2-(5-Methoxypyridin-3-yl)-4-(trifluoromethyl)imidazol-1-yl]benzenesulfonamide Investigative 10524898 C16H13F3N4O3S 398.4 COC1=CN=CC(=C1)C2=NC(=CN2C3=CC=C(C=C3)S(=O)(=O)N)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BKGP69 2,2,2-Trifluoro-1-[4-[5-(4-fluorophenyl)-3-(trifluoromethyl)pyrazol-1-yl]phenyl]ethanone Investigative 10621114 C18H9F7N2O 402.3 C1=CC(=CC=C1C2=CC(=NN2C3=CC=C(C=C3)C(=O)C(F)(F)F)C(F)(F)F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BKGY62 3-[4-(Pentafluoro-lambda6-sulfanyl)anilino]benzoic acid Investigative 122192742 C13H10F5NO2S 339.28 C1=CC(=CC(=C1)NC2=CC=C(C=C2)S(F)(F)(F)(F)F)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BKL09N 2-(9H-Carbazol-2-yl)propanoic acid Investigative 13771052 C15H13NO2 239.27 CC(C1=CC2=C(C=C1)C3=CC=CC=C3N2)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BKL7W1 Disodium;4-[2-(1-carboxylatoethyl)-5-[(2-oxocyclopentyl)methyl]phenyl]benzoate Investigative 56672145 C22H20Na2O5 410.4 CC(C1=C(C=C(C=C1)CC2CCCC2=O)C3=CC=C(C=C3)C(=O)[O-])C(=O)[O-].[Na+].[Na+] IC50 = 76000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BL1I0Q 4-Hydroxy-1,1-dioxo-N-(4-phenylphenyl)-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728413 C21H16N2O4S 392.4 C1=CC=C(C=C1)C2=CC=C(C=C2)NC(=O)C3=C(C4=CC=CC=C4S(=O)(=O)N3)O IC50 = 92600 nM Poor binder T66665 Prostaglandin G/H synthase 2 BL2KA0 N-[3-(3-Methoxyphenylamino)-4-pyridinyl]methanesulfonamide Investigative 44473494 C13H15N3O3S 293.34 COC1=CC=CC(=C1)NC2=C(C=CN=C2)NS(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BL4GQ6 3-(4-Methylsulfonylphenyl)-4-phenylaniline Investigative 44384324 C19H17NO2S 323.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C=CC(=C2)N)C3=CC=CC=C3 IC50 = 194000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BL6J8Z 2-(4-Mesylphenyl)-3-(4-fluorophenyl)-5-nitro-1H-pyrrole Investigative 10316456 C17H13FN2O4S 360.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C=C(N2)[N+](=O)[O-])C3=CC=C(C=C3)F IC50 = 63000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BL6WH2 N-(4-Bromophenyl)-1-(4-methoxyphenyl)-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazole-3-carboxamide Investigative 90654427 C25H23BrN4O5 539.4 COC1=CC=C(C=C1)N2C(=NC(=N2)C(=O)NC3=CC=C(C=C3)Br)C4=CC(=C(C(=C4)OC)OC)OC IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BLB75T Acetic acid 2-phenethylsulfanyl-phenyl ester Investigative 9900153 C16H16O2S 272.4 CC(=O)OC1=CC=CC=C1SCCC2=CC=CC=C2 IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BLH03C 4-[5-(4-Fluorophenyl)-3-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548637 C23H19FN2O3 390.4 COC1=CC=C(C=C1)C2CC(=NN2C3=CC=C(C=C3)C(=O)O)C4=CC=C(C=C4)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BLYX03 N-(3-Phenylsulfonyl-4-pyridinyl)methanesulfonamide Investigative 11415723 C12H12N2O4S2 312.4 CS(=O)(=O)NC1=C(C=NC=C1)S(=O)(=O)C2=CC=CC=C2 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BM0QB7 N-[3-(3-Ethylphenylamino)-4-pyridinyl]methanesulfonamide Investigative 44475683 C14H17N3O2S 291.37 CCC1=CC(=CC=C1)NC2=C(C=CN=C2)NS(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BM0U2Z Sanggenon D Investigative 9987332 C40H36O12 708.7 CC1=C[C@@H]([C@H]([C@@H](C1)C2=C(C=C(C=C2)O)O)C(=O)C3=C(C=C(C=C3)O)O)C4=C(C5=C(C=C4O)OC6(C7=C(C=C(C=C7)O)OC6(C5=O)CC=C(C)C)O)O IC50 = 73000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BM4O2L 2-[6-Chloro-9-(4-methoxybenzoyl)carbazol-2-yl]propanoic acid Investigative 71451683 C23H18ClNO4 407.8 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)C4=CC=C(C=C4)OC)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BM56JK [2'-[(Cyclopropanecarbonyl-ethyl-amino)-methyl]-4'-(6-ethoxy-pyridin-3-yl)-6-methoxy-biphenyl-3-yl]-acetic acid sodium salt Investigative 50901657 C29H31N2NaO5 510.6 CCN(CC1=C(C=CC(=C1)C2=CN=C(C=C2)OCC)C3=C(C=CC(=C3)CC(=O)[O-])OC)C(=O)C4CC4.[Na+] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BM71EY 4-(4-Fluorophenyl)-5-(4-methylsulfonylphenyl)dithiole-3-thione Investigative 11474526 C16H11FO2S4 382.5 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C(=S)SS2)C3=CC=C(C=C3)F IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BM72KB 5-(4-Fluorophenyl)-1-(4-nitrophenyl)-3-(trifluoromethyl)pyrazole Investigative 11792223 C16H9F4N3O2 351.25 C1=CC(=CC=C1C2=CC(=NN2C3=CC=C(C=C3)[N+](=O)[O-])C(F)(F)F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BM8J3Y 3-Oxaheneicosa-5,9,12,15,18-pentaenoic acid Investigative 44584287 C20H30O3 318.4 CC/C=C/C/C=C/C/C=C/C/C=C/CC/C=C/COCC(=O)O IC50 = 180000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BM9ZJ0 3-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl)-5-thiocyanato-1H-pyrrole Investigative 10474426 C18H13FN2O2S2 372.4 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C=C(N2)SC#N)C3=CC=C(C=C3)F IC50 = 72000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BMC5S8 2-(4-Methylphenyl)sulfonyl-3-naphthalen-2-yl-5-(trifluoromethyl)-3,4-dihydropyrazole Investigative 118706119 C21H17F3N2O2S 418.4 CC1=CC=C(C=C1)S(=O)(=O)N2C(CC(=N2)C(F)(F)F)C3=CC4=CC=CC=C4C=C3 IC50 = 95380 nM Poor binder T66665 Prostaglandin G/H synthase 2 BMO3U7 4-[5-(4-Methylphenyl)tetrazol-1-yl]benzenesulfonamide Investigative 57393943 C14H13N5O2S 315.35 CC1=CC=C(C=C1)C2=NN=NN2C3=CC=C(C=C3)S(=O)(=O)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BMZX93 4-[3-(4-Methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 5181298 C23H20N2O3 372.4 COC1=CC=C(C=C1)C2CC(=NN2C3=CC=C(C=C3)C(=O)O)C4=CC=CC=C4 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BN08DI 1-(4-Methanesulfonyl-phenyl)-2-pyridin-3-yl-1H-imidazole-4-carboxylic acid ethyl ester Investigative 10499452 C18H17N3O4S 371.4 CCOC(=O)C1=CN(C(=N1)C2=CN=CC=C2)C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BN1V8Y 2-(6-Chloro-9H-carbazol-2-yl)-N-phenylpropanamide Investigative 71451686 C21H17ClN2O 348.8 CC(C1=CC2=C(C=C1)C3=C(N2)C=CC(=C3)Cl)C(=O)NC4=CC=CC=C4 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BN1XG8 1-Isopropyl-2-(4-methanesulfonyl-phenyl)-5-methyl-1H-pyrrole Investigative 10660176 C15H19NO2S 277.4 CC1=CC=C(N1C(C)C)C2=CC=C(C=C2)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BN69AX 2-(4-Chlorophenyl)-1-(4-methylsulfonylphenyl)imidazole-4-carboxylic Acid Investigative 11793960 C17H13ClN2O4S 376.8 CS(=O)(=O)C1=CC=C(C=C1)N2C=C(N=C2C3=CC=C(C=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BN6S8B N-(4-Aminophenyl)-4-(trifluoromethyl)benzamide Investigative 24689970 C14H11F3N2O 280.24 C1=CC(=CC=C1C(=O)NC2=CC=C(C=C2)N)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BN7I6K N-(2-Aminophenyl)-2-(trifluoromethyl)benzamide Investigative 16774693 C14H11F3N2O 280.24 C1=CC=C(C(=C1)C(=O)NC2=CC=CC=C2N)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BN7S1I Pallidol Investigative 484757 C28H22O6 454.5 C1=CC(=CC=C1[C@H]2[C@H]3[C@H]([C@@H](C4=C3C=C(C=C4O)O)C5=CC=C(C=C5)O)C6=C2C(=CC(=C6)O)O)O IC50 = 80000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BN8FW2 [2-(4-Chlorophenyl)-1-(4-methylsulfonylphenyl)imidazol-4-yl]methanamine Investigative 10594776 C17H16ClN3O2S 361.8 CS(=O)(=O)C1=CC=C(C=C1)N2C=C(N=C2C3=CC=C(C=C3)Cl)CN IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BNB68G Chembl4170326 Investigative 145954463 C20H24O5 344.4 CC(C)CC(=O)OC/C(=C/CC1=C(C=CC2=C1OC(=O)C=C2)OC)/C IC50 = 56400 nM Poor binder T66665 Prostaglandin G/H synthase 2 BNC4I7 5-(4-Chlorophenyl)-4-p-tolyl-3H-1,2-dithiole-3-thione Investigative 44564506 C16H11ClS3 334.9 CC1=CC=C(C=C1)C2=C(SSC2=S)C3=CC=C(C=C3)Cl IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BND25B 3-Nitro-2-(4-(2-(pyrrolidin-1-yl)ethoxy)phenoxy)pyridine Investigative 49805174 C17H19N3O4 329.35 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=C(C=CC=N3)[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BNJX08 4-[5-(4-Fluoro-phenyl)-pyrazol-1-yl]-benzenesulfonamide Investigative 10852952 C15H12FN3O2S 317.3 C1=CC(=CC=C1C2=CC=NN2C3=CC=C(C=C3)S(=O)(=O)N)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BNO9C4 (8-Methoxy-1,2,3,4-tetrahydropyrido[4,3-b]indol-5-yl)-phenylmethanone;hydrochloride Investigative 46906687 C19H19ClN2O2 342.8 COC1=CC2=C(C=C1)N(C3=C2CNCC3)C(=O)C4=CC=CC=C4.Cl IC50 = 87600 nM Poor binder T66665 Prostaglandin G/H synthase 2 BNX5L6 4-[5-(4-Ethylsulfanyl-phenyl)-3-trifluoromethyl-pyrazol-1-yl]-2-hydroxymethyl-benzenesulfonamide Investigative 44364510 C19H18F3N3O3S2 457.5 CCSC1=CC=C(C=C1)C2=CC(=NN2C3=CC(=C(C=C3)S(=O)(=O)N)CO)C(F)(F)F IC50 = 51200 nM Poor binder T66665 Prostaglandin G/H synthase 2 BO1GS0 5-Methanesulfonyl-1-(4-methoxy-benzyl)-1H-indole-2-carboxylic acid methyl ester Investigative 11025137 C19H19NO5S 373.4 COC1=CC=C(C=C1)CN2C3=C(C=C(C=C3)S(=O)(=O)C)C=C2C(=O)OC IC50 = 51300 nM Poor binder T66665 Prostaglandin G/H synthase 2 BO6Z7H 2-(2-Oxochromen-4-yl)oxy-N-pyridin-4-ylpropanamide Investigative 71451368 C17H14N2O4 310.3 CC(C(=O)NC1=CC=NC=C1)OC2=CC(=O)OC3=CC=CC=C32 IC50 = 52390 nM Poor binder T66665 Prostaglandin G/H synthase 2 BO76YP 3-(3-Chloro-2,4,6-trimethoxy-phenyl)-5-methyl-4-phenyl-isoxazole Investigative 11382825 C19H18ClNO4 359.8 CC1=C(C(=NO1)C2=C(C(=C(C=C2OC)OC)Cl)OC)C3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BO8V3Z (Z)-4-Amino-4-(furan-2-yl)-3-phenylbut-3-en-2-one Investigative 71682136 C14H13NO2 227.26 CC(=O)/C(=C(/C1=CC=CO1)\\N)/C2=CC=CC=C2 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BOAN10 2-[6-Chloro-9-(2-chlorobenzoyl)carbazol-2-yl]propanoic acid Investigative 71451684 C22H15Cl2NO3 412.3 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)C4=CC=CC=C4Cl)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BOEP86 3-(3,4-Dimethoxyphenyl)-1,2-dihydronaphthalene Investigative 11608668 C18H18O2 266.3 COC1=C(C=C(C=C1)C2=CC3=CC=CC=C3CC2)OC IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BOH89M Clematichinenoside B Investigative 49799272 C70H114O35 1515.6 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H](O[C@H]([C@@H]([C@H]2O)O)OC[C@@H]3[C@H]([C@@H]([C@H]([C@@H](O3)OC(=O)[C@@]45CC[C@@]6(C(=CC[C@H]7[C@]6(CC[C@@H]8[C@@]7(CC[C@@H]([C@@]8(C)CO)O[C@H]9[C@@H]([C@H]([C@H](CO9)O)O)O[C@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)C)O)O[C@H]1[C@@H]([C@@H]([C@@H](CO1)O[C@H]1[C@@H]([C@H]([C@@H]([C@H](O1)CO)O)O)O)O)O)O)C)C)[C@@H]4CC(CC5)(C)C)C)O)O)O)CO)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BOK1Y4 2-[4-[3-(Butylcarbamoyloxy)phenyl]-3-fluorophenyl]propanoic acid Investigative 73054805 C20H22FNO4 359.4 CCCCNC(=O)OC1=CC=CC(=C1)C2=C(C=C(C=C2)C(C)C(=O)O)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BOL0Z6 2-[6-Chloro-9-(1H-imidazole-5-carbonyl)carbazol-2-yl]propanoic acid Investigative 71457023 C19H14ClN3O3 367.8 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)C4=CN=CN4)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BOQL75 Acetic acid 2-(5-acetoxy-pentylsulfanyl)-phenyl ester Investigative 9857378 C15H20O4S 296.4 CC(=O)OCCCCCSC1=CC=CC=C1OC(=O)C IC50 = 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BORW68 N-(3',4'-Dichloro[1,1'-biphenyl]-4-yl)-4-hydroxy-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide Investigative 54728414 C21H14Cl2N2O4S 461.3 C1=CC=C2C(=C1)C(=C(NS2(=O)=O)C(=O)NC3=CC=C(C=C3)C4=CC(=C(C=C4)Cl)Cl)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BOS73C Z-Val-Gly-OH Investigative 7005167 C15H20N2O5 308.33 CC(C)[C@@H](C(=O)NCC(=O)O)NC(=O)OCC1=CC=CC=C1 IC50 = 55000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BOVD92 Benzenesulfonamide,4-(3-methyl-5-phenyl-1h-pyrazol-1-yl)- Investigative 10710312 C16H15N3O2S 313.4 CC1=NN(C(=C1)C2=CC=CC=C2)C3=CC=C(C=C3)S(=O)(=O)N IC50 = 62800 nM Poor binder T66665 Prostaglandin G/H synthase 2 BP34KB (4-Bromophenyl)-[2-[3-[3-fluoro-5-(4-methoxyoxan-4-yl)phenoxy]propyl]-8-methoxy-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]methanone;hydrochloride Investigative 46906739 C34H37BrClFN2O5 688 COC1=CC2=C(C=C1)N(C3=C2CN(CC3)CCCOC4=CC(=CC(=C4)C5(CCOCC5)OC)F)C(=O)C6=CC=C(C=C6)Br.Cl IC50 = 85400 nM Poor binder T66665 Prostaglandin G/H synthase 2 BP4LE1 4-[5-[4-(Trifluoromethyl)phenyl]tetrazol-1-yl]benzenesulfonamide Investigative 57397474 C14H10F3N5O2S 369.32 C1=CC(=CC=C1C2=NN=NN2C3=CC=C(C=C3)S(=O)(=O)N)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BP59JX (2S)-2-[[(2R)-2-[[(2S)-2-[(4-Fluorobenzoyl)amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-sulfanylpropanoyl]amino]-3-hydroxypropanoic acid Investigative 57384031 C24H25FN4O6S 516.5 C1=CC=C2C(=C1)C(=CN2)C[C@@H](C(=O)N[C@@H](CS)C(=O)N[C@@H](CO)C(=O)O)NC(=O)C3=CC=C(C=C3)F IC50 = 85000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BP6V7T 2-[1-(4-Chlorobenzoyl)-5-methoxy-2-methylindol-3-yl]ethyl N-(3-nitrooxypropylsulfamoyl)carbamate Investigative 11854079 C23H25ClN4O9S 569 CC1=C(C2=C(N1C(=O)C3=CC=C(C=C3)Cl)C=CC(=C2)OC)CCOC(=O)NS(=O)(=O)NCCCO[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BP81OK 2-[9-(Butylcarbamoyl)-6-chlorocarbazol-2-yl]propanoic acid Investigative 71460693 C20H21ClN2O3 372.8 CCCCNC(=O)N1C2=C(C=C(C=C2)Cl)C3=C1C=C(C=C3)C(C)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BPC7B6 2-(9-Acetyl-6-chlorocarbazol-2-yl)propanoic acid Investigative 71449874 C17H14ClNO3 315.7 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)C)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BPI5B4 2-{[(3'',4''-Dichloro-biphenyl-4-ylcarbamoyl)-methyl]-sulfamoyl}-benzoic acid Investigative 46880353 C21H16Cl2N2O5S 479.3 C1=CC=C(C(=C1)C(=O)O)S(=O)(=O)NCC(=O)NC2=CC=C(C=C2)C3=CC(=C(C=C3)Cl)Cl IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BPK47W N-[3-(2-Methoxyphenylamino)-4-pyridinyl]methanesulfonamide Investigative 44475684 C13H15N3O3S 293.34 COC1=CC=CC=C1NC2=C(C=CN=C2)NS(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BPK9C4 3-(5-Chlorofuran-2-yl)-4-phenyl-5-hydroxymethylisoxazole Investigative 57780767 C14H10ClNO3 275.68 C1=CC=C(C=C1)C2=C(ON=C2C3=CC=C(O3)Cl)CO IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BPO09B (3E,5E)-1-Methyl-3,5-bis[(4-pyrrolidin-1-ylphenyl)methylidene]piperidin-4-one Investigative 118706208 C28H33N3O 427.6 CN1C/C(=C\\C2=CC=C(C=C2)N3CCCC3)/C(=O)/C(=C/C4=CC=C(C=C4)N5CCCC5)/C1 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BPO7C9 1-(2-(4-(4-(Methylsulfonyl)phenoxy)phenoxy)ethyl)pyrrolidine Investigative 49805053 C19H23NO4S 361.5 CS(=O)(=O)C1=CC=C(C=C1)OC2=CC=C(C=C2)OCCN3CCCC3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BPTS73 4-[3-(3-Nitrophenyl)-5-propan-2-yl-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 129012346 C19H19N3O4 353.4 CC(C)C1=NN(C(C1)C2=CC(=CC=C2)[N+](=O)[O-])C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BPU19E Kazinol B Investigative 480869 C25H28O4 392.5 CC(=CCC1=C(C=C2C=CC(OC2=C1O)(C)C)[C@@H]3CCC4=C(O3)C=C(C=C4)O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BPX7S1 2-[1-(4-Chlorobenzoyl)-5-methoxy-2-methylindol-3-yl]ethyl N-(3-nitrooxypropyl)carbamate Investigative 11854078 C23H24ClN3O7 489.9 CC1=C(C2=C(N1C(=O)C3=CC=C(C=C3)Cl)C=CC(=C2)OC)CCOC(=O)NCCCO[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BPZ0Y6 1-(2-(4-(4-Fluorophenoxy)phenoxy)ethyl)pyrrolidine Investigative 18678268 C18H20FNO2 301.4 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BQ2B5D (2S)-2-[4-[[(1S,2R)-2-Hydroxycyclopentyl]methyl]phenyl]propanoic acid Investigative 13148392 C15H20O3 248.32 C[C@@H](C1=CC=C(C=C1)C[C@@H]2CCC[C@H]2O)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BQ4Z3E 2-[4-(Methylsulfonyl)phenyl]-3-(4-fluorophenyl)-1-methyl-4,5-dibromo-1H-pyrrole Investigative 9982906 C18H14Br2FNO2S 487.2 CN1C(=C(C(=C1Br)Br)C2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)C IC50 = 55670 nM Poor binder T66665 Prostaglandin G/H synthase 2 BQ61WT 1-(2-(4-(4-Bromophenoxy)phenoxy)ethyl)pyrrolidine Investigative 49805179 C18H20BrNO2 362.3 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=C(C=C3)Br IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BQ7D8R Bromoloxoprofen Investigative 49837500 C15H16BrNaO3 347.18 CC(C1=C(C=C(C=C1)CC2CCCC2=O)Br)C(=O)[O-].[Na+] IC50 = 65000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BQ7T1O Cussonoside B Investigative 169187 C48H78O17 927.1 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H](O[C@H]([C@@H]([C@H]2O)O)OC[C@@H]3[C@H]([C@@H]([C@H]([C@@H](O3)OC(=O)[C@@]45CC[C@@]6(C(=CC[C@H]7[C@]6(CC[C@@H]8[C@@]7(CC[C@@H](C8(C)C)O)C)C)[C@@H]4CC(CC5)(C)C)C)O)O)O)CO)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BQB0D7 3-(4-Tert-butylanilino)benzoic acid Investigative 53316889 C17H19NO2 269.34 CC(C)(C)C1=CC=C(C=C1)NC2=CC=CC(=C2)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BQE8C2 2,3-Dichloro-4-(4-fluorophenyl)-5-(4-methylsulfonylphenyl)-1H-pyrrole Investigative 11740714 C17H12Cl2FNO2S 384.3 CS(=O)(=O)C1=CC=C(C=C1)C2=C(C(=C(N2)Cl)Cl)C3=CC=C(C=C3)F IC50 = 69000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BQFK50 2-[6-Chloro-9-[hexyl(methyl)carbamoyl]carbazol-2-yl]propanoic acid Investigative 71460694 C23H27ClN2O3 414.9 CCCCCCN(C)C(=O)N1C2=C(C=C(C=C2)Cl)C3=C1C=C(C=C3)C(C)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BQS7L0 1-(4-Methanesulfonyl-phenyl)-2-phenyl-1H-imidazole Investigative 10804032 C16H14N2O2S 298.4 CS(=O)(=O)C1=CC=C(C=C1)N2C=CN=C2C3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BQU6F9 (4-Fluoro-2-(4-(methylsulfonyl)phenyl)but-1-ene-1,1-diyl)dibenzene Investigative 49864438 C23H21FO2S 380.5 CS(=O)(=O)C1=CC=C(C=C1)C(=C(C2=CC=CC=C2)C3=CC=CC=C3)CCF IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BR0CT9 N-[3-(3,5-Dichlorophenoxy)-4-pyridinyl]trifluoromethanesulfonamide Investigative 11463338 C12H7Cl2F3N2O3S 387.2 C1=CN=CC(=C1NS(=O)(=O)C(F)(F)F)OC2=CC(=CC(=C2)Cl)Cl IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BR13WD N-[4-[5-(4-Fluorophenyl)-3-(trifluoromethyl)pyrazol-1-yl]phenyl]methanesulfonamide Investigative 10524951 C17H13F4N3O2S 399.4 CS(=O)(=O)NC1=CC=C(C=C1)N2C(=CC(=N2)C(F)(F)F)C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BR14AI 4-[2-(4-Methylpyridin-3-yl)-4-(trifluoromethyl)imidazol-1-yl]benzenesulfonamide Investigative 10714907 C16H13F3N4O2S 382.4 CC1=C(C=NC=C1)C2=NC(=CN2C3=CC=C(C=C3)S(=O)(=O)N)C(F)(F)F IC50 = 51000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BR2GD9 4-[5-Pyridin-4-yl-3-(trifluoromethyl)pyrazol-1-yl]benzenesulfonamide Investigative 10666704 C15H11F3N4O2S 368.3 C1=CC(=CC=C1N2C(=CC(=N2)C(F)(F)F)C3=CC=NC=C3)S(=O)(=O)N IC50 = 64700 nM Poor binder T66665 Prostaglandin G/H synthase 2 BR2K7S 12-O-[3-Methyl-2-butenoyl]-4-deoxyphorbol 13-acetate Investigative 44583798 C29H41NO7 515.6 C[C@@H]1[C@H]([C@@]2([C@@H](C2(C)C)[C@H]3[C@]1([C@@H]4C=C(C(=O)[C@@H]4CC(=C3)CO)C)O)OC(=O)C)OC(=O)C(=C(C)C)N(C)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BR3KO2 Norartocarpetin Investigative 5481970 C15H10O6 286.24 C1=CC(=C(C=C1O)O)C2=CC(=O)C3=C(C=C(C=C3O2)O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BR53MX 2-(4-Fluorophenyl)-1-[4-(methylsulfonyl)phenyl]-5-methyl-1H-pyrrole Investigative 10830212 C18H16FNO2S 329.4 CC1=CC=C(N1C2=CC=C(C=C2)S(=O)(=O)C)C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BR6E4B Epicatechin-(4beta-8)-epiafzelechin Investigative 14015948 C30H26O11 562.5 C1[C@H]([C@H](OC2=C1C(=CC(=C2[C@@H]3[C@H]([C@H](OC4=CC(=CC(=C34)O)O)C5=CC(=C(C=C5)O)O)O)O)O)C6=CC=C(C=C6)O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BR8UP2 2-[4-[3-(Ethylcarbamoyloxy)phenyl]-3-fluorophenyl]propanoic acid Investigative 90036448 C18H18FNO4 331.3 CCNC(=O)OC1=CC=CC(=C1)C2=C(C=C(C=C2)C(C)C(=O)O)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BRA05V 2-[6-Chloro-9-(3,4-dichlorobenzoyl)carbazol-2-yl]propanoic acid Investigative 71460691 C22H14Cl3NO3 446.7 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)C4=CC(=C(C=C4)Cl)Cl)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BRAF14 Loxoprofen Investigative 3965 C15H18O3 246.3 CC(C1=CC=C(C=C1)CC2CCCC2=O)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BRC17J N-[4-(2,4-Dichlorophenyl)phenyl]-4-hydroxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728416 C21H14Cl2N2O4S 461.3 C1=CC=C2C(=C1)C(=C(NS2(=O)=O)C(=O)NC3=CC=C(C=C3)C4=C(C=C(C=C4)Cl)Cl)O IC50 ~ 74800 nM Poor binder T66665 Prostaglandin G/H synthase 2 BRG31Y 2-(4-Methylsulfinylphenyl)-1-(4-methylsulfonylphenyl)-4-(trifluoromethyl)imidazole Investigative 10574542 C18H15F3N2O3S2 428.5 CS(=O)C1=CC=C(C=C1)C2=NC(=CN2C3=CC=C(C=C3)S(=O)(=O)C)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BRH36X 4-[5-(3,4-Dimethoxyphenyl)-3-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 68292453 C25H24N2O5 432.5 COC1=CC=C(C=C1)C2CC(=NN2C3=CC=C(C=C3)C(=O)O)C4=CC(=C(C=C4)OC)OC IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BRI78N 4-[5-Tert-butyl-3-(3,4-dichlorophenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548446 C20H20Cl2N2O2 391.3 CC(C)(C)C1=NN(C(C1)C2=CC(=C(C=C2)Cl)Cl)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BRI89U 2-Amino-N-[3-(trifluoromethyl)phenyl]benzamide Investigative 1517275 C14H11F3N2O 280.24 C1=CC=C(C(=C1)C(=O)NC2=CC=CC(=C2)C(F)(F)F)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BRJI73 2-(2-Chlorophenyl)-4-(2,5-difluorophenyl)-5-[4-(methylsulfonyl)phenyl]thiazole Investigative 44271141 C22H14ClF2NO2S2 461.9 CS(=O)(=O)C1=CC=C(C=C1)C2=C(N=C(S2)C3=CC=CC=C3Cl)C4=C(C=CC(=C4)F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BRJP30 2-(4-(2-(Pyrrolidin-1-yl)ethoxy)phenoxy)pyridine Investigative 49805049 C17H20N2O2 284.35 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=CC=N3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BS1WG4 5-Acetoxymethyl-3-(5-chlorofuran-2-yl)-4-phenylisoxazole Investigative 57780766 C16H12ClNO4 317.72 CC(=O)OCC1=C(C(=NO1)C2=CC=C(O2)Cl)C3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BS38CE 2-[6-Chloro-9-(4-chlorobenzoyl)carbazol-2-yl]propanoic acid Investigative 71460695 C22H15Cl2NO3 412.3 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)C4=CC=C(C=C4)Cl)C=CC(=C3)Cl)C(=O)O IC50 = 72300 nM Poor binder T66665 Prostaglandin G/H synthase 2 BS3C5Y 2-(4-Chlorophenyl)-N,N-diethyl-1-(4-methylsulfonylphenyl)imidazole-4-carboxamide Investigative 10526696 C21H22ClN3O3S 431.9 CCN(CC)C(=O)C1=CN(C(=N1)C2=CC=C(C=C2)Cl)C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BS62OW 5-(4-Fluoro-phenyl)-1-(4-sulfamoyl-phenyl)-1H-pyrazole-3-carboxylic acid amide Investigative 12080914 C16H13FN4O3S 360.4 C1=CC(=CC=C1C2=CC(=NN2C3=CC=C(C=C3)S(=O)(=O)N)C(=O)N)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BS74ZD 1-Butyl-2-(4-methanesulfonyl-phenyl)-5-methyl-1H-pyrrole Investigative 10541610 C16H21NO2S 291.4 CCCCN1C(=CC=C1C2=CC=C(C=C2)S(=O)(=O)C)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BS95HZ Kizuta Saponin K12 Investigative 49799268 C59H96O26 1221.4 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H](O[C@H]([C@@H]([C@H]2O)O)OC[C@@H]3[C@H]([C@@H]([C@H]([C@@H](O3)OC(=O)[C@@]45CC[C@@]6(C(=CC[C@H]7[C@]6(CC[C@@H]8[C@@]7(CC[C@@H](C8(C)CO)O[C@H]9[C@@H]([C@H]([C@H](CO9)O)O)O[C@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)C)O)O)O)C)C)[C@@H]4CC(CC5)(C)C)C)O)O)O)CO)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BS9AN7 4-[5-Tert-butyl-3-(4-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 66548270 C20H22N2O3 338.4 CC(C)(C)C1=NN(C(C1)C2=CC=C(C=C2)O)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BSG98J 1-(2-(4-(3-(Methylsulfonyl)phenoxy)phenoxy)ethyl)pyrrolidine Investigative 49805052 C19H23NO4S 361.5 CS(=O)(=O)C1=CC=CC(=C1)OC2=CC=C(C=C2)OCCN3CCCC3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BSJ3U6 [(1R,2R,6R,10S,11R,13S,14R,15R)-1,14-Dihydroxy-8-(hydroxymethyl)-4,12,12,15-tetramethyl-5-oxo-13-tetracyclo[8.5.0.02,6.011,13]pentadeca-3,8-dienyl] 2-methylbutanoate Investigative 118727932 C25H36O6 432.5 CCC(C)C(=O)O[C@@]12[C@@H](C1(C)C)[C@@H]3C=C(C[C@@H]4[C@H]([C@]3([C@@H]([C@H]2O)C)O)C=C(C4=O)C)CO IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BSJ98I (R)-8-Methyl-6-(trifluoromethoxy)-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid Investigative 52942694 C13H8F6O4 342.19 CC1=CC(=CC2=C1O[C@H](C(=C2)C(=O)O)C(F)(F)F)OC(F)(F)F IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BSN3U4 Huzhangoside D Investigative 49799270 C64H104O30 1353.5 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H](O[C@H]([C@@H]([C@H]2O)O)OC[C@@H]3[C@H]([C@@H]([C@H]([C@@H](O3)OC(=O)[C@@]45CC[C@@]6(C(=CC[C@H]7[C@]6(CC[C@@H]8[C@@]7(CC[C@@H]([C@@]8(C)CO)O[C@H]9[C@@H]([C@H]([C@H](CO9)O)O)O[C@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)C)O)O[C@H]1[C@@H]([C@@H]([C@@H](CO1)O)O)O)O)C)C)[C@@H]4CC(CC5)(C)C)C)O)O)O)CO)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BSU3M4 [(1S,2S,6R,10S,11R,13S,14R,15R)-1,6-Dihydroxy-8-(hydroxymethyl)-4,12,12,15-tetramethyl-14-[(E)-2-methylbut-2-enoyl]oxy-5-oxo-13-tetracyclo[8.5.0.02,6.011,13]pentadeca-3,8-dienyl] 2-methylbutanoate Investigative 20675009 C30H42O8 530.6 CCC(C)C(=O)O[C@@]12[C@@H](C1(C)C)[C@@H]3C=C(C[C@]4([C@H]([C@]3([C@@H]([C@H]2OC(=O)/C(=C/C)/C)C)O)C=C(C4=O)C)O)CO IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BSUD29 Chembl4177170 Investigative 145971990 C15H17ClN6O3 364.79 C1COCC(=O)N1C2=CC=C(C=C2)NC3=NC(=NC(=N3)Cl)OCCN IC50 = 90000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BSZO92 5-(1,2-Dihydro-3-naphthalenyl)-1,3-benzodioxole Investigative 44424403 C17H14O2 250.29 C1CC(=CC2=CC=CC=C21)C3=CC4=C(C=C3)OCO4 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BT1PH7 1-(2-(4-(3-Nitrophenoxy)phenoxy)ethyl)pyrrolidine Investigative 49804918 C18H20N2O4 328.4 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=CC(=C3)[N+](=O)[O-] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BT2I6O (2E)-2-[[4-(Diethoxymethyl)phenyl]methylidene]-3,4-dihydronaphthalen-1-one Investigative 90645114 C22H24O3 336.4 CCOC(C1=CC=C(C=C1)/C=C/2\\CCC3=CC=CC=C3C2=O)OCC IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BT5J8V (4-Chlorophenyl)-[2-[3-[3-fluoro-5-(4-methoxyoxan-4-yl)phenoxy]propyl]-8-methoxy-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]methanone;hydrochloride Investigative 46845032 C34H37Cl2FN2O5 643.6 COC1=CC2=C(C=C1)N(C3=C2CN(CC3)CCCOC4=CC(=CC(=C4)C5(CCOCC5)OC)F)C(=O)C6=CC=C(C=C6)Cl.Cl IC50 = 197900 nM Poor binder T66665 Prostaglandin G/H synthase 2 BTDC57 4-(4-(Methylsulfonyl)phenyl)-5-p-tolyl-3H-1,2-dithiole-3-thione Investigative 44564000 C17H14O2S4 378.6 CC1=CC=C(C=C1)C2=C(C(=S)SS2)C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BTF70K N-(3-Aminophenyl)-3-(trifluoromethyl)benzamide Investigative 20117519 C14H11F3N2O 280.24 C1=CC(=CC(=C1)C(F)(F)F)C(=O)NC2=CC=CC(=C2)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BTJ51W Acetic acid 2-(3-propoxy-propylsulfanyl)-phenyl ester Investigative 10778330 C14H20O3S 268.37 CCCOCCCSC1=CC=CC=C1OC(=O)C IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BTKQ54 N-[4-[2-(3,4-Dichlorophenyl)ethyl]phenyl]-4-hydroxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728405 C23H18Cl2N2O4S 489.4 C1=CC=C2C(=C1)C(=C(NS2(=O)=O)C(=O)NC3=CC=C(C=C3)CCC4=CC(=C(C=C4)Cl)Cl)O IC50 ~ 68000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BTM8U5 N-(5-Aminopyridin-2-yl)-3-(trifluoromethyl)benzamide Investigative 24853949 C13H10F3N3O 281.23 C1=CC(=CC(=C1)C(F)(F)F)C(=O)NC2=NC=C(C=C2)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BU02PO Chembl4279197 Investigative 145978940 C19H20FNO3SSi 389.5 C[Si](C)(C)C1=C(ON=C1C2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BU15YB 1-(4-Methylsulfonylphenyl)-2-thiophen-3-yl-4-(trifluoromethyl)imidazole Investigative 10619274 C15H11F3N2O2S2 372.4 CS(=O)(=O)C1=CC=C(C=C1)N2C=C(N=C2C3=CSC=C3)C(F)(F)F IC50 = 51000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BU3P6F 2-[6-Chloro-9-[(4-methoxyphenyl)methyl]carbazol-2-yl]propanoic acid Investigative 71458881 C23H20ClNO3 393.9 CC(C1=CC2=C(C=C1)C3=C(N2CC4=CC=C(C=C4)OC)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BU4V3N 2-[3-[4-(3-Chlorophenyl)piperazin-1-yl]-3-oxopropyl]-1,2-benzothiazol-3-one Investigative 134154737 C20H20ClN3O2S 401.9 C1CN(CCN1C2=CC(=CC=C2)Cl)C(=O)CCN3C(=O)C4=CC=CC=C4S3 IC50 = 128824.96 nM Poor binder T66665 Prostaglandin G/H synthase 2 BU51GK (2S)-2-[[(2S)-2-[[(2S)-2-[(4-Fluorobenzoyl)amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-hydroxypropanoic acid Investigative 57401899 C30H29FN4O7 576.6 C1=CC=C2C(=C1)C(=CN2)C[C@@H](C(=O)N[C@@H](CO)C(=O)O)NC(=O)[C@H](CC3=CC=C(C=C3)O)NC(=O)C4=CC=C(C=C4)F IC50 = 180000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BU7V6A Chembl4175569 Investigative 145972167 C17H19ClN6O3 390.8 C1COCCN1C2=NC(=NC(=N2)NC3=CC=C(C=C3)N4CCOCC4=O)Cl IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BU91HB 4-[1-(4-Methylsulfonylphenyl)-4-(trifluoromethyl)imidazol-2-yl]pyridine Investigative 10570970 C16H12F3N3O2S 367.3 CS(=O)(=O)C1=CC=C(C=C1)N2C=C(N=C2C3=CC=NC=C3)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BU9K3G 2-[3-Fluoro-4-[3-(propan-2-ylcarbamoyloxy)phenyl]phenyl]propanoic acid Investigative 90036900 C19H20FNO4 345.4 CC(C)NC(=O)OC1=CC=CC(=C1)C2=C(C=C(C=C2)C(C)C(=O)O)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BU9Y8E 1-(2-(4-(4-Chlorophenoxy)phenoxy)ethyl)pyrrolidine Investigative 49805178 C18H20ClNO2 317.8 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=C(C=C3)Cl IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BUC5N8 4-(1-Morpholin-4-yl-1-oxopropan-2-yl)oxychromen-2-one Investigative 71454915 C16H17NO5 303.31 CC(C(=O)N1CCOCC1)OC2=CC(=O)OC3=CC=CC=C32 IC50 = 69940 nM Poor binder T66665 Prostaglandin G/H synthase 2 BUC86H US9271961, Bmt 3-224 Investigative 124222778 C16H13NO5 299.28 CC(=O)C1=CC(=C(C=C1)C(=O)O)NC2=CC=CC=C2C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BUCX40 3-(4-Acetylanilino)benzoic acid Investigative 11184397 C15H13NO3 255.27 CC(=O)C1=CC=C(C=C1)NC2=CC=CC(=C2)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BUD95L 2-(2,6-Dichloro-3-methYlphenyl)amino-N-methoxybenzamide Investigative 19815165 C15H14Cl2N2O2 325.2 CC1=C(C(=C(C=C1)Cl)NC2=CC=CC=C2C(=O)NOC)Cl IC50 = 55000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BV0N7C [1-[4-[5-Chloro-3-(4-methylsulfonylphenyl)imidazol-4-yl]-2-fluorophenoxy]-3-nitrooxypropan-2-yl] nitrate Investigative 16125491 C19H16ClFN4O9S 530.9 CS(=O)(=O)C1=CC=C(C=C1)N2C=NC(=C2C3=CC(=C(C=C3)OCC(CO[N+](=O)[O-])O[N+](=O)[O-])F)Cl IC50 = 76000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BV3H1X 1-(2-(4-(3-(Trifluoromethyl)phenoxy)phenoxy)ethyl)pyrrolidine Investigative 49805176 C19H20F3NO2 351.4 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=CC(=C3)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BV9G7Y 2-[4-[3-(Cyclopropylcarbamoyloxy)phenyl]-3-fluorophenyl]propanoic acid Investigative 90036800 C19H18FNO4 343.3 CC(C1=CC(=C(C=C1)C2=CC(=CC=C2)OC(=O)NC3CC3)F)C(=O)O IC50 = 74300 nM Poor binder T66665 Prostaglandin G/H synthase 2 BVA4F8 3-[(4-Bromophenyl)Amino]Benzoic Acid Investigative 53316888 C13H10BrNO2 292.13 C1=CC(=CC(=C1)NC2=CC=C(C=C2)Br)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BVB6W2 (3E,5E)-1-Benzyl-3,5-bis[[4-(diethoxymethyl)phenyl]methylidene]piperidin-4-one Investigative 90645110 C36H43NO5 569.7 CCOC(OCC)C1=CC=C(C=C1)/C=C\\2/C(=O)/C(=C/C3=CC=C(C=C3)C(OCC)OCC)/CN(C2)CC4=CC=CC=C4 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BVB93O Acetic acid 2-(5-hydroxy-pentylsulfanyl)-phenyl ester Investigative 10729633 C13H18O3S 254.35 CC(=O)OC1=CC=CC=C1SCCCCCO IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BVDT20 Acetic acid 2-propylsulfanyl-phenyl ester Investigative 9813147 C11H14O2S 210.29 CCCSC1=CC=CC=C1OC(=O)C IC50 = 66000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BVF8E1 N-(4-Aminopyridin-2-yl)-3-(trifluoromethyl)benzamide Investigative 24853948 C13H10F3N3O 281.23 C1=CC(=CC(=C1)C(F)(F)F)C(=O)NC2=NC=CC(=C2)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BVHZ43 1,3-Dichloro-5-[4,5-difluoro-2-(4-methylsulfonylphenyl)phenyl]-2-methoxybenzene Investigative 10789363 C20H14Cl2F2O3S 443.3 COC1=C(C=C(C=C1Cl)C2=CC(=C(C=C2C3=CC=C(C=C3)S(=O)(=O)C)F)F)Cl IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BVL5C1 N-[3-(4-Chlorobenzoyl)phenyl]-4-hydroxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728410 C22H15ClN2O5S 454.9 C1=CC=C2C(=C1)C(=C(NS2(=O)=O)C(=O)NC3=CC=CC(=C3)C(=O)C4=CC=C(C=C4)Cl)O IC50 = 95300 nM Poor binder T66665 Prostaglandin G/H synthase 2 BVUM70 4-[3-(4-Bromophenyl)-5-tert-butyl-3,4-dihydropyrazol-2-yl]benzoic acid Investigative 68293323 C20H21BrN2O2 401.3 CC(C)(C)C1=NN(C(C1)C2=CC=C(C=C2)Br)C3=CC=C(C=C3)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BW0SJ1 1-(4-Benzenesulfonyl-phenyl)-2-(4-fluoro-phenyl)-1H-pyrrole Investigative 10762141 C22H16FNO2S 377.4 C1=CC=C(C=C1)S(=O)(=O)C2=CC=C(C=C2)N3C=CC=C3C4=CC=C(C=C4)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BW1K2S 4-(4-(Methylsulfonyl)phenyl)-5-phenyl-3H-1,2-dithiole-3-thione Investigative 44563999 C16H12O2S4 364.5 CS(=O)(=O)C1=CC=C(C=C1)C2=C(SSC2=S)C3=CC=CC=C3 IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BW28IU 3-[2-Oxo-4-(4-sulfamoyl-phenyl)-oxazol-3-yl]-benzoic acid Investigative 10666215 C16H12N2O6S 360.3 C1=CC(=CC(=C1)N2C(=COC2=O)C3=CC=C(C=C3)S(=O)(=O)N)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BW5V2F 4-[(4-Oxo-2-phenyl-1,3-thiazolidin-3-yl)amino]benzenesulfonamide Investigative 70695366 C15H15N3O3S2 349.4 C1C(=O)N(C(S1)C2=CC=CC=C2)NC3=CC=C(C=C3)S(=O)(=O)N IC50 = 78200 nM Poor binder T66665 Prostaglandin G/H synthase 2 BW9Y2D Clematiunicinoside E Investigative 11994185 C76H124O39 1661.8 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H](O[C@H]([C@@H]([C@H]2O)O)OC[C@@H]3[C@H]([C@@H]([C@H]([C@@H](O3)OC(=O)[C@@]45CC[C@@]6(C(=CC[C@H]7[C@]6(CC[C@@H]8[C@@]7(CC[C@@H](C8(C)C)O[C@H]9[C@@H]([C@H]([C@H](CO9)O)O)O[C@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)C)O)O[C@H]1[C@@H]([C@@H]([C@@H](CO1)O[C@H]1[C@@H]([C@H]([C@@H]([C@H](O1)CO)O[C@H]1[C@@H]([C@H]([C@@H]([C@H](O1)CO)O)O)O)O)O)O)O)O)C)C)[C@@H]4CC(CC5)(C)C)C)O)O)O)CO)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BWI75Z 2-[3-(4-Bromophenyl)-1-phenylpyrazol-4-yl]-5-phenyl-1,3,4-oxadiazole Investigative 46934255 C23H15BrN4O 443.3 C1=CC=C(C=C1)C2=NN=C(O2)C3=CN(N=C3C4=CC=C(C=C4)Br)C5=CC=CC=C5 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BWK64U Cussonoside A Investigative 171596 C48H78O18 943.1 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H](O[C@H]([C@@H]([C@H]2O)O)OC[C@@H]3[C@H]([C@@H]([C@H]([C@@H](O3)OC(=O)[C@@]45CC[C@@]6(C(=CC[C@H]7[C@]6(CC[C@@H]8[C@@]7(CC[C@@H]([C@@]8(C)CO)O)C)C)[C@@H]4CC(CC5)(C)C)C)O)O)O)CO)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BWKQ39 (3R,4S)-4-(4-Methanesulfonyl-phenyl)-3-phenyl-dihydro-furan-2-one Investigative 44323830 C17H16O4S 316.4 CS(=O)(=O)C1=CC=C(C=C1)[C@H]2COC(=O)[C@H]2C3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BWM30K 3-(5-Chlorofuran-2-yl)-5-phenyl-1,2-oxazole-4-carboxylic acid Investigative 57780772 C14H8ClNO4 289.67 C1=CC=C(C=C1)C2=C(C(=NO2)C3=CC=C(O3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BWOH67 2-[4-(Methylsulfonyl)phenyl]-3-(4-fluorophenyl)naphthalene Investigative 10762072 C23H17FO2S 376.4 CS(=O)(=O)C1=CC=C(C=C1)C2=CC3=CC=CC=C3C=C2C4=CC=C(C=C4)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BWUG40 1-(5-Chloro-1,3-benzoxazol-2-yl)-N-[(1S,2R)-2-phenylmethoxycyclopentyl]piperidine-4-carboxamide Investigative 71521226 C25H28ClN3O3 454 C1C[C@@H]([C@@H](C1)OCC2=CC=CC=C2)NC(=O)C3CCN(CC3)C4=NC5=C(O4)C=CC(=C5)Cl IC50 = 76600 nM Poor binder T66665 Prostaglandin G/H synthase 2 BX1Y8W 2-(4-Chlorophenyl)-5-[3-(4-methylphenyl)-1-phenylpyrazol-4-yl]-1,3,4-oxadiazole Investigative 90643446 C24H17ClN4O 412.9 CC1=CC=C(C=C1)C2=NN(C=C2C3=NN=C(O3)C4=CC=C(C=C4)Cl)C5=CC=CC=C5 IC50 = 58000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BX29JL 3-Methyl-7-[(4-nitrophenyl)methyl]-5-[(4-phenyl-5-sulfanylidene-1H-1,2,4-triazol-3-yl)methyl]-[1,2]oxazolo[4,5-d]pyridazin-4-one Investigative 70687604 C22H17N7O4S 475.5 CC1=NOC2=C1C(=O)N(N=C2CC3=CC=C(C=C3)[N+](=O)[O-])CC4=NNC(=S)N4C5=CC=CC=C5 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BX38TG 3-{4-[4-Chloro-1-(4-(methylsulfonyl)phenyl)-1H-imidazol-5-yl]-2-fluorophenoxy}propan-1-ol Investigative 16125428 C19H18ClFN2O4S 424.9 CS(=O)(=O)C1=CC=C(C=C1)N2C=NC(=C2C3=CC(=C(C=C3)OCCCO)F)Cl IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BX4I2F 3-((4-(Trifluoromethyl)Phenyl)Amino)Benzoic Acid Investigative 51346826 C14H10F3NO2 281.23 C1=CC(=CC(=C1)NC2=CC=C(C=C2)C(F)(F)F)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BX5MA2 2-[3-(4-Methylphenyl)-1-phenylpyrazol-4-yl]-5-pyridin-4-yl-1,3,4-oxadiazole Investigative 90643445 C23H17N5O 379.4 CC1=CC=C(C=C1)C2=NN(C=C2C3=NN=C(O3)C4=CC=NC=C4)C5=CC=CC=C5 IC50 = 53000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BX5R7G 2-Methyl-4-phenyl-5-[4-(methylsulfonyl)phenyl]-4-isoxazoline Investigative 10947004 C17H17NO3S 315.4 CN1CC(=C(O1)C2=CC=C(C=C2)S(=O)(=O)C)C3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BX7T9L 4-[3-(3-Chloro-2,4,6-trimethoxy-phenyl)-5-methyl-isoxazol-4-yl]-benzenesulfonamide Investigative 11316581 C19H19ClN2O6S 438.9 CC1=C(C(=NO1)C2=C(C(=C(C=C2OC)OC)Cl)OC)C3=CC=C(C=C3)S(=O)(=O)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BX9Z2M Cauloside D Investigative 21630094 C53H86O22 1075.2 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H](O[C@H]([C@@H]([C@H]2O)O)OC[C@@H]3[C@H]([C@@H]([C@H]([C@@H](O3)OC(=O)[C@@]45CC[C@@]6(C(=CC[C@H]7[C@]6(CC[C@@H]8[C@@]7(CC[C@@H]([C@@]8(C)CO)O[C@H]9[C@@H]([C@H]([C@H](CO9)O)O)O)C)C)[C@@H]4CC(CC5)(C)C)C)O)O)O)CO)O)O)O IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BXAM45 2-[6-Chloro-9-(3-chlorobenzoyl)carbazol-2-yl]propanoic acid Investigative 71455230 C22H15Cl2NO3 412.3 CC(C1=CC2=C(C=C1)C3=C(N2C(=O)C4=CC(=CC=C4)Cl)C=CC(=C3)Cl)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BXD7Q8 N-[3-(2-Ethylphenylamino)-4-pyridinyl]methanesulfonamide Investigative 44473492 C14H17N3O2S 291.37 CCC1=CC=CC=C1NC2=C(C=CN=C2)NS(=O)(=O)C IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BXH3D6 N-[3-(3,5-Dichlorophenoxy)-4-pyridinyl]methanesulfonamide Investigative 11302033 C12H10Cl2N2O3S 333.2 CS(=O)(=O)NC1=C(C=NC=C1)OC2=CC(=CC(=C2)Cl)Cl IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BXK6Z8 N-(3-Aminophenyl)-4-(trifluoromethyl)benzamide Investigative 24695790 C14H11F3N2O 280.24 C1=CC(=CC(=C1)NC(=O)C2=CC=C(C=C2)C(F)(F)F)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BXMZ29 2-(6-Chloro-9-hexoxycarbonylcarbazol-2-yl)propanoic acid Investigative 71453519 C22H24ClNO4 401.9 CCCCCCOC(=O)N1C2=C(C=C(C=C2)Cl)C3=C1C=C(C=C3)C(C)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BY0B9N 2-(Cyanoamino)-5-(3,5-di-tert-butyl-4-hydroxybenzylidene)thiazol-4(5H)-one Investigative 135430565 C19H23N3O2S 357.5 CC(C)(C)C1=CC(=CC(=C1O)C(C)(C)C)/C=C\\2/C(=O)NC(=NC#N)S2 IC50 = 55000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BY0H7X 2-[4,5-Difluoro-2-(4-methylsulfonylphenyl)phenyl]-5-methylpyridine Investigative 10522463 C19H15F2NO2S 359.4 CC1=CN=C(C=C1)C2=CC(=C(C=C2C3=CC=C(C=C3)S(=O)(=O)C)F)F IC50 = 52300 nM Poor binder T66665 Prostaglandin G/H synthase 2 BY54XT 3-[5-(4-Fluoro-phenyl)-4-(4-methanesulfonyl-phenyl)-thiophen-2-yl]-propionic acid ethyl ester Investigative 44330480 C22H21FO4S2 432.5 CCOC(=O)CCC1=CC(=C(S1)C2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)C IC50 = 130000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BY57WS (2E,5Z)-5-[(3,5-Ditert-butyl-4-hydroxyphenyl)methylidene]-2-ethoxyimino-1,3-oxazolidin-4-one Investigative 135506078 C20H28N2O4 360.4 CCO/N=C/1\\NC(=O)/C(=C/C2=CC(=C(C(=C2)C(C)(C)C)O)C(C)(C)C)/O1 IC50 = 79000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BY5UJ2 2-(4-Chlorophenyl)-5-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]-1,3,4-oxadiazole Investigative 90643447 C24H17ClN4O2 428.9 COC1=CC=C(C=C1)C2=NN(C=C2C3=NN=C(O3)C4=CC=C(C=C4)Cl)C5=CC=CC=C5 IC50 = 67000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BY68CN Osthole Investigative 10228 C15H16O3 244.28 CC(=CCC1=C(C=CC2=C1OC(=O)C=C2)OC)C IC50 = 81100 nM Poor binder T66665 Prostaglandin G/H synthase 2 BY7AD6 3-[2-Nitro-4-(trifluoromethyl)anilino]benzoic acid Investigative 4763963 C14H9F3N2O4 326.23 C1=CC(=CC(=C1)NC2=C(C=C(C=C2)C(F)(F)F)[N+](=O)[O-])C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BYAV26 4-Amino-N-(4-trifluoromethylphenyl)benzamide Investigative 13609518 C14H11F3N2O 280.24 C1=CC(=CC=C1C(=O)NC2=CC=C(C=C2)C(F)(F)F)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BYD0P5 N-[3-Chloro-4-(4-chlorobenzoyl)phenyl]-4-hydroxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide Investigative 54728409 C22H14Cl2N2O5S 489.3 C1=CC=C2C(=C1)C(=C(NS2(=O)=O)C(=O)NC3=CC(=C(C=C3)C(=O)C4=CC=C(C=C4)Cl)Cl)O IC50 = 95600 nM Poor binder T66665 Prostaglandin G/H synthase 2 BYKL39 2-[4-(Pentafluoro-lambda6-sulfanyl)anilino]benzoic acid Investigative 122192743 C13H10F5NO2S 339.28 C1=CC=C(C(=C1)C(=O)O)NC2=CC=C(C=C2)S(F)(F)(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BYL3T9 2-[4-[3-(Cyclohexylcarbamoyloxy)phenyl]-3-fluorophenyl]propanoic acid Investigative 73054542 C22H24FNO4 385.4 CC(C1=CC(=C(C=C1)C2=CC(=CC=C2)OC(=O)NC3CCCCC3)F)C(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BYN29G Chembl4167707 Investigative 145955705 C22H20ClFN6O4 486.9 C1COCC(=O)N1C2=CC=C(C=C2)NC3=NC(=NC(=N3)Cl)OCCNC(=O)C4=CC=CC=C4F IC50 = 70000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BYU27W 2-[3-Fluoro-4-[4-(hexylcarbamoyloxy)phenyl]phenyl]propanoic acid Investigative 127031160 C22H26FNO4 387.4 CCCCCCNC(=O)OC1=CC=C(C=C1)C2=C(C=C(C=C2)C(C)C(=O)O)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BZ04AL Morusin Investigative 5281671 C25H24O6 420.5 CC(=CCC1=C(OC2=C(C1=O)C(=CC3=C2C=CC(O3)(C)C)O)C4=C(C=C(C=C4)O)O)C IC50 = 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BZ0PV1 4-[5-Tert-butyl-3-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]benzenesulfonic acid Investigative 88930915 C19H21FN2O3S 376.4 CC(C)(C)C1=NN(C(C1)C2=CC=C(C=C2)F)C3=CC=C(C=C3)S(=O)(=O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BZ0U4E N-(3-Aminophenyl)-2-(trifluoromethyl)benzamide Investigative 16774950 C14H11F3N2O 280.24 C1=CC=C(C(=C1)C(=O)NC2=CC=CC(=C2)N)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BZ3M6H 2-(4-(2-(Pyrrolidin-1-yl)ethoxy)phenoxy)aniline Investigative 49805180 C18H22N2O2 298.4 C1CCN(C1)CCOC2=CC=C(C=C2)OC3=CC=CC=C3N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BZ3O2L 1-(4-Ethanesulfonyl-phenyl)-2-(4-fluoro-phenyl)-1H-pyrrole Investigative 10664116 C18H16FNO2S 329.4 CCS(=O)(=O)C1=CC=C(C=C1)N2C=CC=C2C3=CC=C(C=C3)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BZ97PY [3-(2-Fluoro-4-methylphenyl)phenyl] N-hexylcarbamate Investigative 127033540 C20H24FNO2 329.4 CCCCCCNC(=O)OC1=CC=CC(=C1)C2=C(C=C(C=C2)C)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BZB16W 2-(Benzenesulfonyl)-3-naphthalen-2-yl-5-(trifluoromethyl)-3,4-dihydropyrazole Investigative 118706113 C20H15F3N2O2S 404.4 C1C(N(N=C1C(F)(F)F)S(=O)(=O)C2=CC=CC=C2)C3=CC4=CC=CC=C4C=C3 IC50 = 173600 nM Poor binder T66665 Prostaglandin G/H synthase 2 BZI80J 5-(4-Fluorophenyl)-1-(4-sulfamoylphenyl)pyrazole-3-carboxylic Acid Investigative 10666285 C16H12FN3O4S 361.3 C1=CC(=CC=C1C2=CC(=NN2C3=CC=C(C=C3)S(=O)(=O)N)C(=O)O)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BZLV20 [(1S,2S,6R,10S,11R,13S,14R,15R)-14-Acetyloxy-1,6-dihydroxy-8-(hydroxymethyl)-4,12,12,15-tetramethyl-5-oxo-13-tetracyclo[8.5.0.02,6.011,13]pentadeca-3,8-dienyl] 2-methylpropanoate Investigative 118727929 C26H36O8 476.6 C[C@@H]1[C@H]([C@@]2([C@@H](C2(C)C)[C@H]3[C@]1([C@@H]4C=C(C(=O)[C@]4(CC(=C3)CO)O)C)O)OC(=O)C(C)C)OC(=O)C IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 BZQ31A N-(4-Aminophenyl)-2-(trifluoromethyl)benzamide Investigative 16777326 C14H11F3N2O 280.24 C1=CC=C(C(=C1)C(=O)NC2=CC=C(C=C2)N)C(F)(F)F IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D00VHS 4-(5-(4-Hydroxyphenyl)isothiazol-4-yl)phenol Investigative 136036233 C15H11NO2S 269.3 . IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D00XIX 5-(4-Chlorophenyl)-4-p-tolyl-3H-1,2-dithiol-3-one Investigative 44564003 C16H11ClOS2 318.8 CC1=CC=C(C=C1)C2=C(SSC2=O)C3=CC=C(C=C3)Cl IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D01PBO (+)-3,3'-bisdemethyltanegool Investigative 44423052 C18H20O7 348.3 C1[C@@H]([C@H]([C@H](O1)C2=CC(=C(C=C2)O)O)CO)[C@@H](C3=CC(=C(C=C3)O)O)O IC50 = 73900 nM Poor binder T66665 Prostaglandin G/H synthase 2 D03NMM AM-643 Investigative 46843035 C36H39N4NaO4S 646.8 CC1=CN=C(C=C1)COC2=CC3=C(C=C2)N(C(=C3SC(C)(C)C)CC(C)(C)C(=O)[O-])CC4=CC=C(C=C4)C5=NC=C(C=N5)OC.[Na+] IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D03TLR 5-(4-Chlorophenyl)-4-p-tolylisothiazole Investigative 44564454 C16H12ClNS 285.8 CC1=CC=C(C=C1)C2=C(SN=C2)C3=CC=C(C=C3)Cl IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D05QOR SCOPOLETIN Investigative 5280460 C10H8O4 192.17 COC1=C(C=C2C(=C1)C=CC(=O)O2)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D06TPF PYROGALLOL Investigative 1057 C6H6O3 126.11 C1=CC(=C(C(=C1)O)O)O IC50 = 144000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D06YGF Caffeic acid phenethyl ester Investigative 5281787 C17H16O4 284.31 C1=CC=C(C=C1)CCOC(=O)/C=C/C2=CC(=C(C=C2)O)O IC50 = 82000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D06ZRX OXYRESVERATROL Investigative 5281717 C14H12O4 244.24 C1=CC(=C(C=C1O)O)/C=C/C2=CC(=CC(=C2)O)O IC50 = 109000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D07LUJ URSOLIC ACID Investigative 64945 C30H48O3 456.7 C[C@@H]1CC[C@@]2(CC[C@@]3(C(=CC[C@H]4[C@]3(CC[C@@H]5[C@@]4(CC[C@@H](C5(C)C)O)C)C)[C@@H]2[C@H]1C)C)C(=O)O IC50 = 86000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D07OAV 5-(2-1H-indenyl)-1,3-benzodioxole Investigative 44424411 C16H12O2 236.26 C1C2=CC=CC=C2C=C1C3=CC4=C(C=C3)OCO4 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D08RCQ 5-(4-Methoxyphenyl)-4-p-tolylisothiazole Investigative 44564416 C17H15NOS 281.4 CC1=CC=C(C=C1)C2=C(SN=C2)C3=CC=C(C=C3)OC IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0E0RW ISOSCOPOLETIN Investigative 69894 C10H8O4 192.17 COC1=C(C=C2C=CC(=O)OC2=C1)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0G3TK KAEMPFEROL Investigative 5280863 C15H10O6 286.24 C1=CC(=CC=C1C2=C(C(=O)C3=C(C=C(C=C3O2)O)O)O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0G7RA 4-(4-Chlorophenyl)-5-p-tolyl-3H-1,2-dithiol-3-one Investigative 44564004 C16H11ClOS2 318.8 CC1=CC=C(C=C1)C2=C(C(=O)SS2)C3=CC=C(C=C3)Cl IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0L6TP N-(3-phenoxy-4-pyridinyl)propanesulfonamide Investigative 11277773 C14H16N2O3S 292.36 CCCS(=O)(=O)NC1=C(C=NC=C1)OC2=CC=CC=C2 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0M5MI SC-560 Investigative 4306515 C17H12ClF3N2O 352.7 COC1=CC=C(C=C1)N2C(=CC(=N2)C(F)(F)F)C3=CC=C(C=C3)Cl IC50 = 74900 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0N7OP 2-(2-methoxyphenyl)-1H-indene Investigative 44424412 C16H14O 222.28 COC1=CC=CC=C1C2=CC3=CC=CC=C3C2 IC50 = 62300 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0N7XM (-)-3,3'-bisdemethylpinoresinol Investigative 24992964 C18H18O6 330.3 C1[C@@H]2[C@@H](CO[C@H]2C3=CC(=C(C=C3)O)O)[C@@H](O1)C4=CC(=C(C=C4)O)O IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0NH1E Org-231295 Investigative 1383884 C20H22N2O3 338.4 C1CCC(CC1)NC(=O)OC2=CC=CC(=C2)C3=CC(=CC=C3)C(=O)N IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0PQ3Q 4-(4-Chlorophenyl)-5-(4-methoxyphenyl)isothiazole Investigative 44564458 C16H12ClNOS 301.8 COC1=CC=C(C=C1)C2=C(C=NS2)C3=CC=C(C=C3)Cl IC50 ~ 50000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0SJ2Q OLEANOLIC_ACID Investigative 10494 C30H48O3 456.7 C[C@]12CC[C@@H](C([C@@H]1CC[C@@]3([C@@H]2CC=C4[C@]3(CC[C@@]5([C@H]4CC(CC5)(C)C)C(=O)O)C)C)(C)C)O IC50 = 87000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0V7AA CATECHIN Investigative 9064 C15H14O6 290.27 C1[C@@H]([C@H](OC2=CC(=CC(=C21)O)O)C3=CC(=C(C=C3)O)O)O IC50 = 93300 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0V9EN 3,4-Dihydroxycinnamic Acid Investigative 689043 C9H8O4 180.16 C1=CC(=C(C=C1/C=C/C(=O)O)O)O IC50 = 129700 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0VF6F N-(3-phenoxypyridin-4-yl)methanesulfonamide Investigative 10244543 C12H12N2O3S 264.3 CS(=O)(=O)NC1=C(C=NC=C1)OC2=CC=CC=C2 IC50 ~ 100000 nM Poor binder T66665 Prostaglandin G/H synthase 2 D0Y1YR gingerol Investigative 442793 C17H26O4 294.4 CCCCC[C@@H](CC(=O)CCC1=CC(=C(C=C1)O)OC)O IC50 = 125000 nM Poor binder