TTD_Target_ID	Target_Name	TTD_Drug_ID	Drug_Name	Drug_Highest_Status	Drug_PubchemID	Molecular_Formula	Molecular_Weight	Canonical_SMILES	Activity	Binder_Type
T86399	Bromodomain-containing protein 2	B1J5EV	5-[4-[(Dimethylamino)methyl]-2,5-dimethoxyphenyl]-1,3,6-trimethylpyridin-2-one	Investigative	127048256	C19H26N2O3	330.4	CC1=CC(=C(N(C1=O)C)C)C2=C(C=C(C(=C2)OC)CN(C)C)OC	IC50 = 59555 nM	Poor binder
T86399	Bromodomain-containing protein 2	B1Y9EC	8-[4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl]-6-methylpyrido[4,3-d]pyrimidin-5-one	Investigative	127051087	C19H22N4O3	354.4	CN1C=C(C2=NC=NC=C2C1=O)C3=CC(=C(C(=C3)OC)CN(C)C)OC	IC50 ~ 100000 nM	Poor binder
T86399	Bromodomain-containing protein 2	B2HE4W	4-[4-[(Dimethylamino)methyl]-3,5-Dimethoxy-Phenyl]-2-Methyl-2,7-Naphthyridin-1-One	Investigative	118796358	C20H23N3O3	353.4	CN1C=C(C2=C(C1=O)C=NC=C2)C3=CC(=C(C(=C3)OC)CN(C)C)OC	IC50 ~ 100000 nM	Poor binder
T86399	Bromodomain-containing protein 2	B4CZF3	(cis)-1-Acetyl-2-methyl-6-[4-(1-piperidinylmethyl)phenyl]-1,2,3,4-tetrahydro-4-quinolinamine	Investigative	67195867	C24H31N3O	377.5	C[C@H]1C[C@H](C2=C(N1C(=O)C)C=CC(=C2)C3=CC=C(C=C3)CN4CCCCC4)N	IC50 = 50118.72 nM	Poor binder
T86399	Bromodomain-containing protein 2	B4MX5P	3-Butyl-8-[(6-Butyl-5,7-Dimethyl-[1,2,4]triazolo[1,5-A]pyrimidin-2-Yl)sulfanylmethyl]-7-Ethyl-Purine-2,6-Dione	Investigative	60498769	C23H32N8O2S	484.6	CCCCC1=C(N2C(=NC(=N2)SCC3=NC4=C(N3CC)C(=O)NC(=O)N4CCCC)N=C1C)C	IC50 = 59000 nM	Poor binder
T86399	Bromodomain-containing protein 2	B7C4JV	4-{4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl}-2-methyl-1,2-dihydroisoquinolin-1-one	Investigative	119098889	C21H24N2O3	352.4	CN1C=C(C2=CC=CC=C2C1=O)C3=CC(=C(C(=C3)OC)CN(C)C)OC	IC50 = 50857 nM	Poor binder
T86399	Bromodomain-containing protein 2	BA69TQ	4-[(E)-2-(2,4-Dimethoxyphenyl)-3-(4-methoxyphenyl)prop-2-enoyl]-1,3-dihydroquinoxalin-2-one	Investigative	122180904	C26H24N2O5	444.5	COC1=CC=C(C=C1)/C=C(\\C2=C(C=C(C=C2)OC)OC)/C(=O)N3CC(=O)NC4=CC=CC=C43	IC50 ~ 50000 nM	Poor binder
T86399	Bromodomain-containing protein 2	BATC31	7-Methoxy-4-[(E)-3-(4-methoxyphenyl)-2-phenylprop-2-enoyl]-1,3-dihydroquinoxalin-2-one	Investigative	122180900	C25H22N2O4	414.5	COC1=CC=C(C=C1)/C=C(\\C2=CC=CC=C2)/C(=O)N3CC(=O)NC4=C3C=CC(=C4)OC	IC50 ~ 50000 nM	Poor binder
T86399	Bromodomain-containing protein 2	BD2L5V	Ethyl N-[(4S)-1-methyl-6-phenyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]carbamate	Investigative	72703043	C20H19N5O2	361.4	CCOC(=O)N[C@@H]1C2=NN=C(N2C3=CC=CC=C3C(=N1)C4=CC=CC=C4)C	IC50 = 100000 nM	Poor binder
T86399	Bromodomain-containing protein 2	BDI85R	4-[4-[(Dimethylamino)methyl]-2,5-Dimethoxy-Phenyl]-2-Methyl-2,7-Naphthyridin-1-One	Investigative	117072549	C20H23N3O3	353.4	CN1C=C(C2=C(C1=O)C=NC=C2)C3=C(C=C(C(=C3)OC)CN(C)C)OC	IC50 ~ 100000 nM	Poor binder
T86399	Bromodomain-containing protein 2	BGH61F	4-[(E)-2-(3,4-Dimethylphenyl)-3-(4-methoxyphenyl)prop-2-enoyl]-1,3-dihydroquinoxalin-2-one	Investigative	122180895	C26H24N2O3	412.5	CC1=C(C=C(C=C1)/C(=C\\C2=CC=C(C=C2)OC)/C(=O)N3CC(=O)NC4=CC=CC=C43)C	IC50 ~ 50000 nM	Poor binder
T86399	Bromodomain-containing protein 2	BH1NI5	2-(4-Hydroxy-3,5-Dimethylphenyl)-7-Methyl-5,6,7,8-Tetrahydropyrido[4',3':4,5]thieno[2,3-D]pyrimidin-4(3h)-One	Investigative	135567026	C18H19N3O2S	341.4	CC1=CC(=CC(=C1O)C)C2=NC3=C(C4=C(S3)CN(CC4)C)C(=O)N2	IC50 ~ 100000 nM	Poor binder
T86399	Bromodomain-containing protein 2	BKUG12	5-[4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl]-7-methyl-1,7-naphthyridin-8-one	Investigative	127051726	C20H23N3O3	353.4	CN1C=C(C2=C(C1=O)N=CC=C2)C3=CC(=C(C(=C3)OC)CN(C)C)OC	IC50 ~ 100000 nM	Poor binder
T86399	Bromodomain-containing protein 2	BOR93S	4-[4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl]-2-methyl-2,6-naphthyridin-1-one	Investigative	127051727	C20H23N3O3	353.4	CN1C=C(C2=C(C1=O)C=CN=C2)C3=CC(=C(C(=C3)OC)CN(C)C)OC	IC50 ~ 100000 nM	Poor binder
T86399	Bromodomain-containing protein 2	BTPG20	8-[4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl]-6-methyl-1,6-naphthyridin-5-one	Investigative	127052023	C20H23N3O3	353.4	CN1C=C(C2=C(C1=O)C=CC=N2)C3=CC(=C(C(=C3)OC)CN(C)C)OC	IC50 ~ 100000 nM	Poor binder