TTD Target ID TTD Drug/Compound ID Pubchem CID Activity T34562 CANH78 17280 IC50 = 3270000 nM T34562 C27IRS 197934 IC50 = 1280000 nM T34562 CBJ36Y 639433 IC50 = 564130 nM T34562 CF2BD8 907361 IC50 = 21370 nM T34562 C5NQG3 940069 IC50 = 31410 nM T34562 CJGB43 941230 IC50 = 40000 nM T34562 CEX1K9 10243765 IC50 = 19050 nM T34562 C5I4SX 10402002 IC50 = 28980 nM T34562 C2JY8F 15388819 IC50 = 3000 nM T34562 C8G9AL 16756850 IC50 > 10000 nM T34562 C0SDW6 127025482 Ki = 2390 nM T34562 CK7L8U 127027355 IC50 = 23700 nM T34562 CH6ON2 127027684 IC50 = 625710 nM T34562 C7ST9X 127028306 IC50 = 317310 nM T34562 CN86IR 127028327 IC50 = 3333300 nM T34562 CHU16M 127028328 IC50 = 2064200 nM T34562 CV03TZ 127028660 IC50 = 237500 nM T34562 CBE6M2 127028661 IC50 = 627000 nM T34562 C5P3GA 127029548 IC50 = 8760 nM T34562 C1ZP4G 130431469 IC50 > 10000 nM T34562 CMA35H 130431481 IC50 > 10000 nM T34562 D0S9LT 12793 IC50 = 3250000 nM T34562 D0T0YI 378 IC50 = 18500000 nM T25464 D06OMK 445643 IC50 = 14.8 nM T25464 D0G7UX 5284373 IC50 = 183 nM T25464 C12CHL 4470793 Ki > 300000 nM T25464 C6YF5L 9918081 Ki > 3000 nM T25464 CC30ZA 10305301 Ki > 200000 nM T25464 C9TQ7U 11105029 IC50 = 2.8 nM T25464 C7WJF0 15546641 IC50 = 7.2 nM T25464 CU2A6K 44306123 IC50 = 7.32 nM T25464 C7WNM2 44306124 IC50 = 4.17 nM T25464 C86EOZ 44306135 IC50 = 8.65 nM T25464 C8T5NI 44306145 IC50 = 14 nM T25464 CUH17I 44306155 IC50 = 8.7 nM T25464 C6OQ4D 44306156 IC50 = 5.85 nM T25464 CN58YR 44306157 IC50 = 7.25 nM T25464 C8N7QZ 44306253 IC50 = 4.93 nM T25464 CD8O6N 44306280 IC50 = 7.91 nM T25464 C68IRQ 44306324 IC50 = 3.96 nM T25464 CBI4S6 44373943 IC50 > 5000 nM T25464 CQX6L4 44374010 IC50 = 348 nM T25464 C4I9DK 44374019 IC50 = 742 nM T25464 CBH09L 44374020 IC50 = 363 nM T25464 C89QDY 44374110 IC50 = 890 nM T25464 CQ65HS 44374127 IC50 > 5000 nM T25464 CJ9G7T 44374128 IC50 = 1539 nM T25464 C4XI8B 44374132 IC50 = 581 nM T25464 CYO20C 44374169 IC50 = 636 nM T25464 C1G6CI 44374400 IC50 = 840 nM T25464 CS30FH 49863381 IC50 = 140 nM T25464 C3YI2V 49863382 IC50 = 89 nM T25464 CS48JU 49863383 IC50 = 49 nM T71367 D0E3TC 44259 IC50 = 0.57 nM T71367 D00SDR 90054634 IC50 = 330 nM T71367 D0HK8C 90054733 IC50 = 121 nM T71367 D0L2FW 90054621 IC50 = 546 nM T71367 CA3C5S 3685259 IC50 < 5000 nM T71367 CACS26 11561968 Ki > 1000 nM T71367 CU0E8O 11690457 Ki > 1000 nM T71367 CJ21EH 13626914 IC50 = 94 nM T71367 C5VPH9 16129448 IC50 = 892 nM T71367 CGD89T 27126517 IC50 = 861 nM T71367 CC71QJ 27666048 IC50 > 100000 nM T71367 C61HBG 45102725 IC50 = 4200 nM T71367 CLS29B 46872626 IC50 > 10000 nM T71367 C5BZV3 57958821 IC50 = 381 nM T71367 C1MR8Q 60097495 IC50 > 1000 nM T71367 C37NKO 67129970 IC50 > 10000 nM T71367 CK80LJ 67130050 IC50 = 9430 nM T71367 CV63UL 67240318 IC50 > 10000 nM T71367 C7GRV2 68755406 IC50 > 10000 nM T71367 C7D2UQ 69463478 IC50 = 189 nM T71367 CVIA91 71553085 IC50 = 120 nM T71367 C1TR3O 71553152 IC50 = 2480 nM T71367 CDJY72 71568837 IC50 = 1600 nM T71367 C8CAG7 71578921 IC50 > 10000 nM T71367 C6P5YH 71657853 IC50 = 1.4 nM T71367 CKRS82 71678791 IC50 = 18 nM T71367 C7ROZ1 71679297 IC50 = 46 nM T71367 C9JTE7 71679299 IC50 = 16 nM T71367 C9RQW2 71679784 IC50 = 32 nM T71367 CHR3P5 71679785 IC50 = 15 nM T71367 CK1HR0 71679949 IC50 = 41 nM T71367 CF7R0Y 71682057 IC50 = 8000 nM T71367 CZM67T 72703518 IC50 = 150 nM T71367 C84AEF 72705109 IC50 = 77 nM T71367 CBK47T 72705487 IC50 = 132 nM T71367 CVF5P0 73603034 IC50 = 5700 nM T71367 C3SJQ2 76336279 IC50 > 100000 nM T71367 CI6NL9 77068235 IC50 = 8 nM T71367 C7RO1U 86703926 IC50 = 60 nM T71367 C97DVA 89729987 IC50 = 401 nM T71367 C2O4JR 89730033 IC50 = 3.5 nM T71367 C4UY2V 89730039 IC50 = 1.6 nM T71367 CB7Y0S 89730041 IC50 = 3.7 nM T71367 CQM98T 89730047 IC50 = 3.7 nM T71367 CC97QK 90054623 IC50 = 689 nM T71367 C93YPW 90054630 IC50 = 1700 nM T71367 CX0WH7 90054720 IC50 = 297 nM T71367 C9CRM6 90054726 IC50 = 423 nM T71367 CJX51L 90054730 IC50 = 225 nM T71367 CRF7M2 90054734 IC50 = 387 nM T71367 CEO7I0 90054986 IC50 = 58 nM T71367 CIZ2T6 90055028 IC50 = 351 nM T71367 C3ZV1C 90655985 IC50 = 5840 nM T71367 CE9KY0 90655986 IC50 = 2120 nM T71367 C6JIP7 91664348 IC50 = 4000 nM T71367 C18QYF 105539853 IC50 = 19.95 nM T71367 CBZ59D 118701008 IC50 = 3.7 nM T71367 C9CUL3 118711764 IC50 = 1600 nM T71367 CZH6E4 118711841 IC50 = 150 nM T71367 CYL46R 118711842 IC50 = 70 nM T71367 C2OK7E 118711843 IC50 = 710 nM T71367 CR8B9H 118711844 IC50 = 160 nM T71367 C5VDI0 118711845 IC50 = 840 nM T71367 C92TDH 118711846 IC50 = 300 nM T71367 C37IZJ 118711847 IC50 = 640 nM T71367 C8XFB1 118711848 IC50 = 130 nM T71367 COM51H 118711849 IC50 = 180 nM T71367 C7CB6W 118711850 IC50 = 10 nM T71367 CPNM74 118711851 IC50 = 70 nM T71367 C48DCS 118711852 IC50 = 10 nM T71367 CX8CL3 118711853 IC50 = 11000 nM T71367 CZV53F 118711854 IC50 = 19000 nM T71367 C2LT9G 118711855 IC50 = 37000 nM T71367 C0VBS5 118711856 IC50 = 7000 nM T71367 C0IJF5 118711857 IC50 = 23000 nM T71367 C7JV3C 118711858 IC50 = 3000 nM T71367 C4LJ6U 118711859 IC50 = 10000 nM T71367 C0QDO9 118711860 IC50 = 6000 nM T71367 CK0W1O 118711861 IC50 = 1000 nM T71367 C9XBL5 118711862 IC50 = 2000 nM T71367 CT3IS4 118711863 IC50 = 2000 nM T71367 C26EOM 118711864 IC50 = 1000 nM T71367 C9AGI1 118711865 IC50 = 2000 nM T71367 C2SQ6P 118711866 IC50 = 2000 nM T71367 C5GPJ9 118711891 IC50 = 2000 nM T71367 C76KYO 118711892 IC50 = 6000 nM T71367 CKBQ72 118711893 IC50 = 3000 nM T71367 CEU0S4 118711894 IC50 = 5000 nM T71367 CK63ES 118711895 IC50 = 10000 nM T71367 C92ZJE 118711896 IC50 = 8000 nM T71367 C2JA8B 127025153 IC50 = 600 nM T71367 CVUE54 127025154 IC50 = 84 nM T71367 C6W1UY 127025155 IC50 = 64 nM T71367 CLIP96 127026999 IC50 = 96 nM T71367 CEBO19 127027293 IC50 = 46 nM T71367 C5CUO0 127027294 IC50 = 248 nM T71367 CYS8L4 127027295 IC50 = 270 nM T71367 C39LPD 127027304 IC50 = 20 nM T71367 C3E7FZ 127028834 IC50 = 410 nM T71367 CJX04U 127029806 IC50 = 1509 nM T71367 CWVN31 127029807 IC50 = 1722 nM T71367 C9TZ7D 127034994 IC50 = 48 nM T71367 CE7M4J 127036775 IC50 = 14.9 nM T71367 CP89UZ 127036952 IC50 = 13 nM T71367 CX3Z7Q 134136970 IC50 > 100000 nM T71367 C82XFJ 134139661 IC50 > 100000 nM T71367 CKB1J9 134144378 IC50 = 44000 nM T71367 COF17E 134147249 IC50 = 5600 nM T71367 C60OFR 134154014 IC50 > 100000 nM T71367 CY4D8I 135566504 Ki = 812.4 nM T71367 CG3UZ1 135927974 Ki > 1000 nM T71367 CWGA76 137530158 IC50 = 12.59 nM T71367 CI1E8V 137634241 IC50 > 10000 nM T71367 C2E4DP 139592531 IC50 = 158.49 nM T71367 CZ7YS0 146027031 IC50 = 19.95 nM T71367 C2MD1Q 155513187 IC50 > 10000 nM T71367 CE7TI4 155521619 IC50 = 7943.28 nM T71367 CPW4H0 155531070 IC50 = 19952.62 nM T71367 CONB81 155557716 IC50 = 3981.07 nM T71367 D0NY6U 86703914 IC50 = 17 nM T71367 D0O6OH 71553154 IC50 = 18 nM T86928 D04AIT 5280445 IC50 = 500 nM T86928 D0K8KX 5280343 IC50 = 550 nM T86928 D0R3JB 4212 IC50 = 660 nM T86928 D09JEJ 24748573 IC50 = 3 nM T86928 D0B9BU 6918454 EC50 = 100 nM T86928 D0WS1V 448991 IC50 > 10000 nM T86928 C2OAV0 7328982 EC50 = 1600 nM T86928 CQVZ16 44123806 IC50 = 710 nM T86928 C1O6NR 44123807 IC50 = 480 nM T86928 C91MBN 44123808 IC50 = 820 nM T86928 CX08MT 44590715 IC50 = 2610 nM T86928 CVK4W9 44590746 IC50 = 2600 nM T86928 CO1UP9 44590747 IC50 = 5870 nM T86928 C3QRL8 44590749 IC50 = 2500 nM T86928 C4MY0L 44590794 IC50 = 8600 nM T86928 CLPU05 44590795 IC50 = 1520 nM T86928 C1CQS8 44590796 IC50 = 1100 nM T86928 C1MR8Q 60097495 IC50 > 10000 nM T86928 CPL8X0 139593287 EC50 = 6000 nM T86928 C7UNX2 145991479 IC50 < 1000 nM T86928 C2MD1Q 155513187 IC50 > 10000 nM T86928 C4PL1X 155536605 IC50 = 45100 nM T86928 CT9D0Q 155547691 IC50 = 18230 nM T86928 C2G8TU 155550182 IC50 = 1650 nM T86928 C1ACW9 155552233 IC50 = 8070 nM T86928 CDXK27 155562302 IC50 = 850 nM T86928 C6ICJ5 155562508 IC50 = 21990 nM T86928 CV74OB 155566389 IC50 = 4400 nM T86928 CGSU30 155566872 IC50 = 17750 nM T86928 D00RIX 5280443 IC50 = 800 nM T86928 D00YEV 5281605 IC50 = 10000 nM T86928 D01UYI 5281607 IC50 = 9000 nM T86928 D02DML 5281707 IC50 = 200 nM T86928 D07OAT 456214 IC50 > 10000 nM T86928 D0CP3M 5149739 IC50 = 930 nM T86928 D0G3TK 5280863 IC50 = 400 nM T86928 D0LH4L 10154 IC50 = 700 nM T86928 D0MF5Y 5281614 IC50 = 350 nM T86928 D0NJ4H 5281670 IC50 = 10000 nM T86928 D0O1YH 1694 IC50 = 1600 nM T86928 D0T3PW 5281672 IC50 = 900 nM T59102 D00STL 644241 IC50 = 71 nM T59102 D01PZD 5329098 IC50 = 68 nM T59102 D03ZBT 11626560 IC50 > 1000 nM T59102 D07POC 176870 IC50 = 12200 nM T59102 D08CDI 208908 IC50 = 8500 nM T59102 D09GDD 11167602 IC50 = 1.5 nM T59102 D09KTS 24821094 IC50 > 1000 nM T59102 D0AZ3C 5291 IC50 = 72 nM T59102 D0E6XR 3062316 Ki < 10 nM T59102 D0G6QF 3081361 IC50 = 1100 nM T59102 D0H0EQ 24826799 IC50 = 1.2 nM T59102 D0J9ZR 4477 IC50 > 100000 nM T59102 D0R0MW 5329102 IC50 = 2 nM T59102 D0W5HK 216239 IC50 = 37 nM T59102 D00UZR 5330286 IC50 > 10000 nM T59102 D02UFQ 11620908 IC50 > 10000 nM T59102 D03AND 11656518 IC50 = 6 nM T59102 D08HOM 46207586 IC50 = 3 nM T59102 D0A1AQ 5329099 IC50 = 50 nM T59102 D0D1GF 42642645 IC50 = 9.4 nM T59102 D0E3TC 44259 IC50 = 0.6 nM T59102 D0HS5V 11234052 IC50 > 6000 nM T59102 D0M0XB 10302451 IC50 > 5000 nM T59102 D0M9QZ 11485656 IC50 = 60 nM T59102 D0O0LS 25141092 IC50 > 10000 nM T59102 D0O6WV 24794418 IC50 > 500 nM T59102 D0P6DJ 151194 IC50 = 490 nM T59102 D0T2ER 24767976 IC50 = 13 nM T59102 D0Z6MT 16662431 IC50 = 4 nM T59102 D03BNU 59604787 IC50 > 3500 nM T59102 D0JY1I 42613483 IC50 = 3900 nM T59102 D06GBK 2048 IC50 = 6200 nM T59102 D0H4GI 10275001 IC50 = 406 nM T59102 D0IT6Q 3038522 IC50 = 26 nM T59102 D0L5YF 5329032 IC50 = 3400 nM T59102 D0T3ME 156422 IC50 = 6200 nM T59102 C63WLY 89644 IC50 > 10 ug.mL-1 T59102 C5JE2Z 104860 IC50 = 7.6 ug.mL-1 T59102 C6Y9CV 151193 IC50 = 490 nM T59102 CI1NA5 159926 IC50 > 10 ug.mL-1 T59102 CYBA43 177458 IC50 > 10 ug.mL-1 T59102 C32HFB 396514 IC50 = 2000 nM T59102 C4MNG8 445840 IC50 = 5000 nM T59102 C75EDQ 644355 IC50 = 100 nM T59102 C5HPF3 644356 IC50 = 20 nM T59102 C9D7UY 727518 IC50 > 100000 nM T59102 CXB5A2 964113 IC50 > 100000 nM T59102 CDB17F 1538822 IC50 = 24200 nM T59102 CZ2B4M 2358462 IC50 > 100000 nM T59102 CXA1L7 2365265 IC50 > 100000 nM T59102 CEF62M 2379240 IC50 = 33100 nM T59102 CKT64G 2396126 IC50 > 10000 nM T59102 CFVK40 3008950 IC50 > 50000 nM T59102 CD8UW1 3008956 IC50 = 17000 nM T59102 CCD93P 3008957 IC50 > 50000 nM T59102 CU64VM 3008958 IC50 > 50000 nM T59102 C8F0KM 3008959 IC50 > 50000 nM T59102 CV8R9Z 3008960 IC50 > 50000 nM T59102 C8EZ6O 3008961 IC50 > 50000 nM T59102 CX95SU 3008962 IC50 = 8900 nM T59102 C9B2MN 3008963 IC50 > 50000 nM T59102 C9E7BW 3008964 IC50 > 50000 nM T59102 CGK91Q 3008965 IC50 = 14700 nM T59102 CCN9D5 3142817 IC50 = 1000 nM T59102 CY28LS 5293755 IC50 > 100000 nM T59102 CFW19M 5329009 IC50 = 3000 nM T59102 C9I7WT 5329100 IC50 = 60 nM T59102 CMWB28 5329101 IC50 = 17 nM T59102 CGX50J 5329104 IC50 = 5 nM T59102 C2VX0H 5329105 IC50 = 0.5 nM T59102 CK71MQ 5329106 IC50 = 1 nM T59102 CL0Q4S 5329107 IC50 = 3 nM T59102 C6YRH8 5329108 IC50 = 2 nM T59102 CFP59Y 5329109 IC50 = 1 nM T59102 C0JW3Y 5329134 IC50 = 2110 nM T59102 CO7J2A 5329135 IC50 = 620 nM T59102 CQ4TP5 5329136 IC50 = 8290 nM T59102 CXQC42 5329137 IC50 = 11300 nM T59102 CT94JS 5329138 IC50 = 140 nM T59102 CNH06M 5329139 IC50 = 4190 nM T59102 CRY4Z2 5329140 IC50 = 5980 nM T59102 CAPE50 5329141 IC50 = 1400 nM T59102 CFU58A 5329142 IC50 = 160 nM T59102 C5Q8XK 5329143 IC50 = 170 nM T59102 C8PX4D 5329144 IC50 = 650 nM T59102 C6USQ5 5329145 IC50 = 2780 nM T59102 C56LWT 5329146 IC50 = 3650 nM T59102 CZ16MN 5329147 IC50 = 1210 nM T59102 CAN16I 5329148 IC50 = 1530 nM T59102 CG4NC2 5329149 IC50 = 550 nM T59102 CIW70H 5329150 IC50 = 110 nM T59102 C5FT6A 5329151 IC50 = 230 nM T59102 CB0N4L 5329152 IC50 = 940 nM T59102 COFP24 5329153 IC50 = 680 nM T59102 CGWD98 5329154 IC50 = 5460 nM T59102 C4PD0K 5329156 IC50 = 11500 nM T59102 C0RWT8 5329157 IC50 = 1030 nM T59102 C3MU5S 5329158 IC50 = 3460 nM T59102 CN6O4R 5329159 IC50 = 70600 nM T59102 CG68DI 5329160 IC50 > 100000 nM T59102 CYR7V0 5329161 IC50 = 13900 nM T59102 C9BXE2 5329162 IC50 = 94010 nM T59102 CY4V5Z 5329163 IC50 = 240 nM T59102 CI64YA 5329164 IC50 = 4 nM T59102 C2ZV0O 5329165 IC50 < 780 nM T59102 CAB53L 5329166 IC50 = 20 nM T59102 CTW9R8 5329167 IC50 = 19300 nM T59102 C8A3TJ 5329168 IC50 = 40 nM T59102 CVTD82 5329169 IC50 = 680 nM T59102 CQ5WK1 5329170 IC50 = 870 nM T59102 CNC9T7 5329171 IC50 = 5430 nM T59102 C6L0UW 5329229 IC50 > 20000 nM T59102 C1DBV6 5329230 IC50 > 20000 nM T59102 CLKM80 5329231 IC50 > 20000 nM T59102 CTQ18A 5329232 IC50 > 100000 nM T59102 CM5KG6 5329233 IC50 > 20000 nM T59102 CQG6R2 5329234 IC50 > 20000 nM T59102 CJ3A9I 5329235 IC50 > 100000 nM T59102 CPS7X1 5329236 IC50 > 100000 nM T59102 CAN60T 5329237 IC50 > 20000 nM T59102 CY15JP 5329238 IC50 > 20000 nM T59102 C41UBI 5329239 IC50 > 20000 nM T59102 C6VQ9F 5329240 IC50 > 20000 nM T59102 C8WS5K 5329241 IC50 > 20000 nM T59102 CI26UN 5329242 IC50 > 20000 nM T59102 C6PJ2R 5329243 IC50 > 20000 nM T59102 C0OKB7 5329244 IC50 = 20000 nM T59102 C78ZNL 5329245 IC50 > 20000 nM T59102 CWL5S4 5329246 IC50 = 20000 nM T59102 C4X3OE 5329248 IC50 = 5620 nM T59102 CK8FH6 5329249 IC50 > 20000 nM T59102 CN5B6C 5329250 IC50 > 20000 nM T59102 CQ0B6E 5329251 IC50 > 10000 nM T59102 C4KO3N 5329252 IC50 > 100000 nM T59102 C6MZF8 5329253 IC50 > 20000 nM T59102 C9NBG7 5330546 IC50 = 70 nM T59102 CS3A8F 5331081 IC50 > 20000 nM T59102 CG4W8K 5331082 IC50 > 20000 nM T59102 CD4C2A 5331083 IC50 > 20000 nM T59102 C6AT8V 5331084 IC50 > 20000 nM T59102 CJVS23 5331085 IC50 > 20000 nM T59102 CZ29FN 5331086 IC50 > 20000 nM T59102 CYL78A 5331087 IC50 > 20000 nM T59102 CJ87XR 5331088 IC50 = 2100 nM T59102 CFB3K7 5331089 IC50 = 18000 nM T59102 C9WY1O 5331090 IC50 > 20000 nM T59102 C9ZK3D 5331091 IC50 > 20000 nM T59102 C6RJC8 5331092 IC50 = 1100 nM T59102 C0IOY8 5331093 IC50 = 1400 nM T59102 CMD08O 5331094 IC50 = 1100 nM T59102 CDQ3M7 5359485 IC50 = 0.89 ug.mL-1 T59102 C54BYP 5360741 IC50 = 1.8 ug.mL-1 T59102 CD65JT 5427216 IC50 > 100000 nM T59102 CPB95V 5427224 IC50 > 100000 nM T59102 C61NCL 5482344 IC50 = 1800 nM T59102 CDK3J0 5703619 IC50 = 0.4 nM T59102 CA6L5V 5707304 IC50 > 100000 nM T59102 C43YGE 5713379 IC50 > 100000 nM T59102 CT8U7I 5874584 IC50 = 8390 nM T59102 CM8LW9 6036100 IC50 > 100000 nM T59102 C6L5HS 6419386 IC50 = 2800 nM T59102 C3CQW0 6419387 IC50 = 1000 nM T59102 CWOA63 6419388 IC50 = 2000 nM T59102 CZVU64 6419389 IC50 = 1400 nM T59102 C9FN4B 6419390 IC50 = 800 nM T59102 CN53YW 6419391 IC50 = 4000 nM T59102 C17NWJ 6419392 IC50 = 600 nM T59102 C13IRC 6419393 IC50 = 2000 nM T59102 C4FLE9 6419394 IC50 = 800 nM T59102 C4GHT0 6419395 IC50 = 4000 nM T59102 C8SAQ1 6419396 IC50 > 10000 nM T59102 CP71CL 6419397 IC50 > 10000 nM T59102 CQ3S8L 6450842 IC50 = 3700 nM T59102 C2N0IR 6477203 IC50 = 12800 nM T59102 CW5YJ2 6536705 IC50 > 100000 nM T59102 C2OL7K 9796455 IC50 = 353 nM T59102 CI80BK 9803350 IC50 = 2500 nM T59102 C9TAL6 9826308 IC50 = 160 nM T59102 CWVH12 9828619 IC50 = 50 nM T59102 CX10KR 9828962 IC50 = 170 nM T59102 CE5X8J 9844744 IC50 = 490 nM T59102 CSAY10 9845576 IC50 = 1500 nM T59102 C6A9HS 9871170 IC50 = 97 nM T59102 C3CI1J 9872659 IC50 = 20 nM T59102 CUZ07T 9884745 IC50 > 100000 nM T59102 CHF7G5 9890746 IC50 = 90 nM T59102 CXA5C8 9893493 IC50 > 2000 nM T59102 CZ25GL 9894619 IC50 = 70 nM T59102 C3EUB4 9911005 IC50 = 240 nM T59102 C24JTF 9911313 IC50 = 13300 nM T59102 C1Y3MH 9915808 IC50 = 90 nM T59102 C6HP3L 9948410 IC50 > 100000 nM T59102 C7T9DJ 9950440 IC50 > 30000 nM T59102 CO4N3Q 9995374 IC50 > 100000 nM T59102 C5WF7J 10007113 IC50 = 300 nM T59102 CY90DN 10023010 IC50 = 5 nM T59102 CJ95HR 10041745 IC50 = 12 nM T59102 CG57EC 10047098 IC50 = 13400 nM T59102 CUJR40 10062694 EC50 = 6 nM T59102 C1JUF8 10073832 IC50 > 2000 nM T59102 CIV15Q 10113978 IC50 = 84 nM T59102 C5WCL2 10117540 IC50 = 216 nM T59102 C5KHX2 10118413 IC50 = 50 nM T59102 C46DHW 10119600 IC50 = 230 nM T59102 CRNC72 10120038 IC50 = 90 nM T59102 C4VW8P 10121424 IC50 = 40 nM T59102 CYQ01B 10121530 IC50 = 30 nM T59102 CR5D2N 10121709 IC50 = 1 nM T59102 C5X7LQ 10121737 IC50 = 20 nM T59102 C3XW0Y 10122339 IC50 = 2.4 nM T59102 C6IA4L 10143909 IC50 = 77 nM T59102 C7X5LY 10145209 IC50 = 110 nM T59102 CL89XT 10165712 IC50 = 2 nM T59102 C76XOL 10166902 IC50 = 10 nM T59102 C1Y7HR 10167597 IC50 = 36 nM T59102 CR5Y7O 10168074 IC50 = 0.4 nM T59102 CJH54G 10186893 IC50 = 1430 nM T59102 C3ER4N 10187285 IC50 < 4 nM T59102 CM26BU 10187537 IC50 = 140 nM T59102 CA03YO 10187699 IC50 = 1010 nM T59102 CUG37L 10187829 IC50 = 335 nM T59102 C8T7RC 10188599 IC50 = 265 nM T59102 C6FB3Q 10188863 IC50 = 5040 nM T59102 C0N3HC 10189022 IC50 = 50 nM T59102 C6G2RK 10189131 IC50 = 20 nM T59102 CD4C9B 10207679 IC50 = 70 nM T59102 CZU79W 10208916 IC50 = 320 nM T59102 C4G2AD 10209993 IC50 = 9 nM T59102 CZJ78I 10210309 IC50 = 145 nM T59102 CBFZ09 10210632 IC50 = 99 nM T59102 C5YCN2 10215023 IC50 = 66000 nM T59102 C95ZXY 10226609 IC50 = 800 nM T59102 CB83CI 10228726 IC50 = 10 nM T59102 C18DRH 10229841 IC50 = 710 nM T59102 CD7J3O 10231458 IC50 = 20 nM T59102 CL9N2E 10231519 IC50 = 100 nM T59102 CAE03L 10231813 IC50 < 4 nM T59102 CPD6Z9 10236164 IC50 > 100000 nM T59102 CX15BI 10246728 IC50 = 3 nM T59102 C1WL8B 10251852 IC50 > 500000 nM T59102 CH30RC 10253133 IC50 = 1400 nM T59102 CBI47E 10264222 IC50 > 100000 nM T59102 C6DC8Q 10275163 IC50 = 3300 nM T59102 CD2IE3 10278606 IC50 = 920 nM T59102 CH5DQ0 10280082 IC50 = 140 nM T59102 C65JZS 10296462 IC50 = 1250 nM T59102 CVO54Z 10300451 IC50 > 20000 nM T59102 C63DPY 10301981 IC50 = 10 nM T59102 CO90LX 10302121 IC50 = 216 nM T59102 CC4G8B 10302519 IC50 < 4 nM T59102 C2T3WU 10302586 IC50 = 168 nM T59102 C4FP8M 10303591 IC50 < 4 nM T59102 C5CBF9 10320381 IC50 = 6600 nM T59102 C97YDQ 10344304 IC50 = 510 nM T59102 CZV0G7 10359698 IC50 = 16 nM T59102 CQB9H7 10389422 IC50 = 11000 nM T59102 CLAX64 10413508 IC50 = 11000 nM T59102 CQ43JU 10426229 IC50 = 17500 nM T59102 CU8JP3 10432698 IC50 = 1100 nM T59102 C95LYF 10457505 IC50 = 530 nM T59102 C7PLI5 10478569 IC50 > 2000 nM T59102 CJ5M1D 10482445 IC50 = 8000 nM T59102 CJWH60 10489322 IC50 > 100000 nM T59102 C5SVT4 10537949 IC50 > 100000 nM T59102 CGAW17 10562306 IC50 = 85400 nM T59102 C6AJI9 10562777 IC50 = 25500 nM T59102 CE5L6D 10587839 IC50 > 100000 nM T59102 CM8N6L 10593765 IC50 = 24500 nM T59102 CI30LZ 10613858 IC50 > 100000 nM T59102 CH6Z3L 10635478 IC50 = 65500 nM T59102 CB97UD 10636005 IC50 > 100000 nM T59102 C2UWA0 10658651 IC50 = 41700 nM T59102 C5L0IX 10663368 IC50 > 100000 nM T59102 C9Z7XH 10663503 IC50 = 49900 nM T59102 CH1G6P 10682457 IC50 > 100000 nM T59102 C54UAK 10728035 IC50 = 2800 nM T59102 CXSH91 10753550 IC50 = 18200 nM T59102 CVPW04 10755069 IC50 > 100000 nM T59102 C3WR0Q 10779668 IC50 > 100000 nM T59102 CF5T1H 10783444 IC50 > 100000 nM T59102 CX1DH7 10862508 IC50 = 6720 nM T59102 CU8P7M 10862866 IC50 = 2000 nM T59102 C54VTR 10863323 IC50 = 720 nM T59102 C43CLE 10863395 IC50 = 440 nM T59102 CD8M0L 10863993 IC50 = 8180 nM T59102 C71JKT 10873266 IC50 > 30000 nM T59102 C16FCD 10874104 IC50 = 18200 nM T59102 CY7E1M 10874618 IC50 = 160 nM T59102 CU92JA 10875187 IC50 = 1.4 nM T59102 CSTP13 10875630 IC50 = 26 nM T59102 C6QV1L 10885200 IC50 = 9420 nM T59102 C8TDN1 10885583 IC50 = 2210 nM T59102 C70PLZ 10885776 IC50 = 6500 nM T59102 CI4XR0 10885830 IC50 = 20 nM T59102 CRN57U 10895433 IC50 = 2570 nM T59102 CJSX79 10896366 IC50 = 4690 nM T59102 C0BN9J 10896386 IC50 = 150 nM T59102 CJ4P5T 10905857 IC50 = 850 nM T59102 CM5IA4 10906467 IC50 = 210 nM T59102 CO21NS 10907015 IC50 = 80 nM T59102 CB0MK5 10907225 IC50 = 150 nM T59102 C2IOU4 10907383 IC50 = 2810 nM T59102 CC3P6X 10907564 IC50 = 520 nM T59102 CJUI34 10917610 IC50 = 510 nM T59102 CCB49T 10917872 IC50 = 1040 nM T59102 C4WJ2T 10918068 IC50 = 715 nM T59102 C62LQW 10918358 IC50 = 290 nM T59102 C4OX0I 10918469 IC50 = 662 nM T59102 CS0BJ5 10928229 IC50 = 110 nM T59102 C1DS2G 10929540 IC50 = 440 nM T59102 C7MTO0 10929814 IC50 = 2970 nM T59102 CY0J9W 10951558 IC50 = 53 nM T59102 CJE7Y2 10961232 IC50 > 10000 nM T59102 C94GTN 10963029 IC50 = 5000 nM T59102 CBT4S3 10963044 IC50 = 29 nM T59102 CAC02X 10963192 IC50 = 500 nM T59102 CKD72X 10972606 IC50 = 9210 nM T59102 CL89QG 10973305 IC50 = 100 nM T59102 CPY51V 10983215 IC50 = 30 nM T59102 CCN5F8 10984279 IC50 = 3230 nM T59102 C9ELG2 10984685 IC50 = 222 nM T59102 CAP7E6 10995060 IC50 = 305 nM T59102 CB5AD7 11004892 IC50 = 230 nM T59102 C53QCD 11006148 IC50 = 177 nM T59102 C0LK2Q 11006502 IC50 = 494 nM T59102 CC87FE 11015336 IC50 = 1210 nM T59102 C71TOQ 11015640 IC50 > 30000 nM T59102 CY3B6O 11015880 IC50 = 330 nM T59102 C4F8ZN 11026804 IC50 > 30000 nM T59102 CDQ0H4 11027671 IC50 = 178 nM T59102 C59LQM 11027750 IC50 = 100 nM T59102 C4GLS2 11036639 IC50 = 11100 nM T59102 C9NYE2 11037955 IC50 = 290 nM T59102 CT5V2C 11039013 IC50 = 813 nM T59102 CL3FG7 11039428 IC50 = 0.4 nM T59102 CJ05CL 11048367 IC50 = 80 nM T59102 CWVC81 11049206 IC50 = 2310 nM T59102 C5V9DI 11049316 IC50 = 5590 nM T59102 CD9GY6 11049581 IC50 = 1260 nM T59102 C04QKG 11069972 IC50 = 2060 nM T59102 CXDA03 11070177 IC50 > 30000 nM T59102 CB7ND4 11071122 IC50 = 290 nM T59102 C0HM8T 11071223 IC50 = 160 nM T59102 CYG8V1 11071546 IC50 = 335 nM T59102 CV4R8X 11081103 IC50 = 740 nM T59102 CM04HI 11081393 IC50 = 60 nM T59102 CKX3Z5 11081446 IC50 = 220 nM T59102 C4G2AF 11091152 IC50 = 5360 nM T59102 CEB97L 11112669 IC50 = 1260 nM T59102 C4YUN5 11112927 IC50 > 30000 nM T59102 CQDC05 11113190 IC50 = 190 nM T59102 CYH21N 11113218 IC50 > 30000 nM T59102 CDZ80M 11114435 IC50 = 582 nM T59102 C5MAN7 11124388 IC50 = 300 nM T59102 C6HQ2L 11133954 IC50 = 480 nM T59102 CM9QT3 11143981 IC50 = 9960 nM T59102 C9KES6 11144730 IC50 = 790 nM T59102 CTJ9U3 11145086 IC50 = 1410 nM T59102 CU5DO2 11145515 IC50 = 20 nM T59102 C0D8CT 11155618 IC50 = 180 nM T59102 C7CNO9 11156466 IC50 = 100 nM T59102 CMJ31L 11156812 IC50 = 20 nM T59102 CBDS75 11157185 IC50 = 90 nM T59102 CP16ND 11168221 IC50 = 80 nM T59102 CL8Y4F 11177747 IC50 = 270 nM T59102 CWIT81 11178110 IC50 = 150 nM T59102 CCAG52 11179181 IC50 = 70 nM T59102 CK7B4X 11190431 IC50 > 30000 nM T59102 CBG94A 11191231 IC50 = 40 nM T59102 C7BHE0 11200526 IC50 = 4590 nM T59102 C09YIQ 11202821 IC50 > 30000 nM T59102 C65JPE 11212551 IC50 > 30000 nM T59102 C50JAG 11223943 IC50 = 1440 nM T59102 CN6BC7 11226164 IC50 > 30000 nM T59102 C87WCG 11226298 IC50 = 1390 nM T59102 CYA59I 11235645 IC50 > 30000 nM T59102 C0E1ML 11236566 IC50 = 140 nM T59102 C1QAS6 11237612 IC50 = 190 nM T59102 CH2VD7 11245435 IC50 > 30000 nM T59102 CGL6R0 11249274 IC50 = 200 nM T59102 CUV15L 11249319 IC50 > 30000 nM T59102 CKRA10 11258984 IC50 > 10000 nM T59102 C9F6KW 11260252 IC50 = 180 nM T59102 CC93YJ 11260253 IC50 > 30000 nM T59102 C6ZD4C 11270126 IC50 > 30000 nM T59102 CKI25P 11272815 IC50 = 70 nM T59102 CJW65Q 11273677 IC50 > 30000 nM T59102 C3IU8T 11281396 IC50 = 1300 nM T59102 C28XHQ 11282038 IC50 = 620 nM T59102 CZX0K9 11283270 IC50 = 550 nM T59102 C9I8AN 11293184 IC50 > 30000 nM T59102 C7I9TG 11293913 IC50 = 310 nM T59102 CIXK95 11295243 IC50 = 640 nM T59102 CYFT17 11295612 IC50 = 780 nM T59102 CNF7V4 11304951 IC50 > 30000 nM T59102 CVCE09 11305002 IC50 = 2700 nM T59102 CEN1J8 11306433 IC50 > 30000 nM T59102 C5PW1K 11306478 IC50 > 30000 nM T59102 CJ3N8G 11316908 IC50 > 30000 nM T59102 C41RWG 11318423 IC50 = 330 nM T59102 CVQ1Y0 11318736 IC50 = 20 nM T59102 C9G4YJ 11325945 IC50 > 30000 nM T59102 C2WKC3 11330812 IC50 > 30000 nM T59102 C15ZLJ 11340108 IC50 = 100 nM T59102 C4ICB0 11341503 IC50 = 650 nM T59102 C9K3LZ 11350308 IC50 = 1540 nM T59102 CV3K6Q 11351606 IC50 > 10000 nM T59102 C1LT5J 11352217 IC50 > 30000 nM T59102 CU18NY 11352407 IC50 = 3260 nM T59102 C24LHS 11353568 IC50 = 21000 nM T59102 C1UD0O 11372879 IC50 > 30000 nM T59102 CM4UY7 11373369 IC50 = 170 nM T59102 C25ZCN 11374110 IC50 = 130 nM T59102 C6EGP9 11374800 IC50 = 90 nM T59102 C8TLG4 11396174 IC50 = 380 nM T59102 CL19HT 11397589 IC50 = 810 nM T59102 C41NOY 11409644 IC50 = 80 nM T59102 CEG81P 11419763 IC50 = 130 nM T59102 C9IQP7 11419787 IC50 > 30000 nM T59102 C3NBZ9 11420151 IC50 = 6080 nM T59102 CMAI17 11420386 IC50 = 10200 nM T59102 CREQ51 11429654 IC50 = 96 nM T59102 CVQC06 11429694 IC50 > 30000 nM T59102 C9WEH6 11432198 IC50 = 60 nM T59102 C7AI2V 11432911 IC50 > 2000 nM T59102 C17WNX 11443611 IC50 = 90 nM T59102 C3SKT6 11443633 IC50 = 80 nM T59102 COF7Z1 11443718 IC50 > 30000 nM T59102 C6I2ER 11455034 IC50 = 100 nM T59102 CX5L2B 11464443 IC50 = 10300 nM T59102 CD3P4Q 11465678 IC50 = 390 nM T59102 CT34RJ 11466063 IC50 = 290 nM T59102 C6M9NC 11477626 IC50 > 2000 nM T59102 CEB29T 11490006 IC50 > 30000 nM T59102 C46JFZ 11494322 IC50 = 33 nM T59102 C9K8RE 11496022 IC50 = 137 nM T59102 CY72AM 11496228 IC50 = 659 nM T59102 C5UEK0 11510816 IC50 = 110 nM T59102 CG3BZ9 11517980 IC50 = 4 nM T59102 CFQ42U 11525980 IC50 = 23 nM T59102 CL7X4Q 11530963 IC50 = 1867 nM T59102 CID2P7 11536421 IC50 = 54 nM T59102 C6IOJ4 11546085 IC50 = 310 nM T59102 CF28TK 11565353 IC50 = 217 nM T59102 CZ1H0X 11569258 IC50 = 5500 nM T59102 CRL95F 11569396 IC50 = 1 nM T59102 CO9KP5 11583459 IC50 > 10000 nM T59102 CB91RQ 11589811 IC50 = 40 nM T59102 CM65QP 11590120 IC50 = 3 nM T59102 C69FYK 11604142 Ki = 200 nM T59102 CEG5W8 11608830 IC50 = 9 nM T59102 C8IKG5 11616255 IC50 = 458 nM T59102 CCB3X0 11617740 IC50 = 6220 nM T59102 CSM62L 11626920 IC50 = 31 nM T59102 CK34LS 11632737 IC50 = 200 nM T59102 C7W3TE 11633427 IC50 = 10 nM T59102 C5R6DG 11634086 IC50 > 800 nM T59102 C8V0YT 11639969 IC50 = 1200 nM T59102 CZM9K1 11675974 IC50 = 410 nM T59102 C3M1CF 11682291 IC50 = 5420 nM T59102 CCX2F5 11682611 IC50 = 0.4 nM T59102 C8AEX7 11687971 IC50 = 151900 nM T59102 CHG14R 11688408 IC50 = 55 nM T59102 CZY05V 11719421 IC50 = 6 nM T59102 CUB2N6 11719537 IC50 = 5 nM T59102 C9P0VD 11729539 IC50 = 550 nM T59102 CBL38T 11730367 IC50 = 260 nM T59102 C4PE0D 11730369 IC50 = 1140 nM T59102 C3DVE0 11730809 IC50 = 370 nM T59102 CCQO28 11731042 IC50 = 871 nM T59102 C23STH 11731130 IC50 = 601 nM T59102 CSLC27 11731197 IC50 = 50 nM T59102 C5NLG6 11732326 IC50 = 3180 nM T59102 CU54IA 11732691 IC50 > 30000 nM T59102 C2M7ZD 11733137 IC50 = 1240 nM T59102 C67FZJ 11734285 IC50 = 400 nM T59102 CT49LJ 11734851 IC50 = 12 nM T59102 CU9BR4 11749848 IC50 > 30000 nM T59102 C0QV3M 11752083 IC50 = 10900 nM T59102 CAS0V7 11752632 IC50 = 290 nM T59102 CP7AH3 11755812 IC50 = 7700 nM T59102 CRW2H3 11762328 IC50 = 21600 nM T59102 CRI64Z 11762329 IC50 = 1200 nM T59102 CJI7T6 11763085 IC50 = 76 nM T59102 C61QXW 11785508 IC50 > 30000 nM T59102 CEOH20 11813259 IC50 = 943 nM T59102 C89SNG 11813434 IC50 > 30000 nM T59102 C4V8PJ 11813761 IC50 = 110 nM T59102 C1CI6M 11826385 IC50 = 440 nM T59102 CEUB71 11826832 IC50 = 1470 nM T59102 C9EV8H 11827121 IC50 = 3110 nM T59102 C72RZN 11827714 IC50 = 720 nM T59102 C14MZC 11827841 IC50 = 6750 nM T59102 CDZ1I3 11989153 IC50 = 637 nM T59102 CM50UH 12000646 EC50 = 170 nM T59102 CI39TK 12004372 IC50 = 10700 nM T59102 CDGF78 15282555 IC50 = 3300 nM T59102 C7LB4I 15949613 IC50 = 96 nM T59102 C9TU1O 16046126 IC50 > 1000 nM T59102 CW2XK6 16050925 IC50 = 110 nM T59102 C9JK2M 16059071 IC50 > 2000 nM T59102 CW6UJ9 16059338 IC50 > 1000 nM T59102 CH7MS6 16059729 IC50 > 42000 nM T59102 CFKE48 16064750 IC50 = 1 nM T59102 CQG45C 16109001 IC50 = 1940 nM T59102 C5VPH9 16129448 IC50 = 5270 nM T59102 C0V8FB 16730091 IC50 = 2 nM T59102 CA24TE 16730092 IC50 = 5 nM T59102 CGX61W 22041319 IC50 = 10 nM T59102 CYP32E 22707343 IC50 = 540 nM T59102 CFO6J5 22707344 IC50 = 10700 nM T59102 CWXO86 22707354 IC50 = 1320 nM T59102 C8JD2X 22707384 IC50 > 750 nM T59102 CAG61Z 22707433 IC50 = 2880 nM T59102 C20RYA 22707442 IC50 = 1380 nM T59102 CNR0O7 22707450 IC50 = 5160 nM T59102 CEOV57 22707452 IC50 > 100 nM T59102 CPO51J 22707462 IC50 = 6250 nM T59102 CGR94W 22707466 IC50 = 500 nM T59102 C3H1VE 22707498 IC50 = 1160 nM T59102 CDI35F 22707517 IC50 > 30000 nM T59102 C6MBW9 22707526 IC50 = 970 nM T59102 CQ3TW0 22707568 IC50 = 29700 nM T59102 CB29GC 22707603 IC50 = 350 nM T59102 C2UO3S 22707619 IC50 > 30000 nM T59102 CM5R8B 22707669 IC50 = 1120 nM T59102 C7G6NJ 22707741 IC50 = 5170 nM T59102 C9QLP0 23133323 IC50 = 1100 nM T59102 CG12OL 23518511 IC50 > 20000 nM T59102 CRX0Q6 23625758 IC50 = 780 nM T59102 C2RV3U 24180608 IC50 > 30000 nM T59102 C3X1WH 24742411 IC50 = 2 nM T59102 CS78XJ 24742412 IC50 = 3 nM T59102 C2KA6G 24742584 IC50 = 4 nM T59102 CN9GC8 24742586 IC50 = 10 nM T59102 CHU49V 24757938 IC50 < 1 nM T59102 C0D2PA 24758868 IC50 = 20 nM T59102 C3K5YO 24758982 IC50 = 7 nM T59102 CYU0Z8 24758983 IC50 = 6 nM T59102 CJL67N 24759089 IC50 = 4 nM T59102 C2APK8 24759090 IC50 = 9 nM T59102 C5CRF6 24759091 IC50 = 6 nM T59102 CA8U7X 24759094 IC50 = 4 nM T59102 CRB89L 24759205 IC50 = 1 nM T59102 C13JUP 24759314 IC50 = 5 nM T59102 CCPS81 24764502 IC50 > 35000 nM T59102 C9B2TF 24880043 IC50 = 150 nM T59102 CFK2B9 24882503 IC50 = 1400 nM T59102 C43HWQ 24883287 IC50 > 10000 nM T59102 C8DA5Q 24883334 IC50 > 10000 nM T59102 C4V9GH 24894117 IC50 = 11000 nM T59102 CJH19T 24894883 IC50 = 45000 nM T59102 CB5TP8 24894992 IC50 = 38000 nM T59102 CF4N9X 24895100 IC50 = 40000 nM T59102 CY8L7E 24896769 IC50 > 10000 nM T59102 CN13JF 24899915 IC50 = 1.3 ug.mL-1 T59102 CBWR97 24899916 IC50 = 1.8 ug.mL-1 T59102 C9F2JD 24899917 IC50 > 10 ug.mL-1 T59102 C64MTI 24900160 IC50 = 5.8 ug.mL-1 T59102 CO2I6Q 24900161 IC50 > 10 ug.mL-1 T59102 C5FD1A 24937369 IC50 = 5300 nM T59102 C4KG0Y 25022599 IC50 > 1000 nM T59102 CRO0Y8 25022735 IC50 = 90000 nM T59102 C72AJM 25022736 IC50 > 500000 nM T59102 CQ27UI 25113814 IC50 = 10 nM T59102 C2IHY0 25114266 IC50 = 5 nM T59102 CP8S9W 25116064 IC50 = 11 nM T59102 CTV54O 25123227 IC50 = 14 nM T59102 C1IYN7 25127854 IC50 = 5.9 nM T59102 CKD14B 25127856 IC50 = 19 nM T59102 CJBX60 25128180 IC50 = 8.3 nM T59102 CC5SD9 25128181 IC50 = 21 nM T59102 CIG4H0 25178539 IC50 = 4200 nM T59102 C4GI6J 25178540 IC50 = 6700 nM T59102 CL0Z1F 25181502 IC50 = 830 nM T59102 COB9G8 25181586 IC50 = 2800 nM T59102 C8YLD6 25194331 IC50 = 5 nM T59102 CXC9B3 25194865 IC50 = 9 nM T59102 C1I0VS 25194866 IC50 = 3 nM T59102 C9OZN3 25194867 IC50 = 30 nM T59102 C6FGQ1 25206346 IC50 = 91 nM T59102 CXNW87 25207322 IC50 = 8 nM T59102 C8IJB9 25218207 IC50 = 40300 nM T59102 C2TXC6 25218656 IC50 > 2000 nM T59102 CVM13K 42596931 IC50 = 100 nM T59102 CU53WB 42596953 IC50 = 2500 nM T59102 C7GIQ3 42625508 IC50 = 4600 nM T59102 CVZ83M 42625582 IC50 = 2700 nM T59102 C5MD9E 42625892 IC50 = 7300 nM T59102 CJ5U1X 42639664 IC50 = 6.4 ug.mL-1 T59102 CEL61X 44229839 IC50 > 10000 nM T59102 C4NWP5 44246325 IC50 > 200000 nM T59102 C2EW0I 44246326 IC50 = 118000 nM T59102 CSD8T0 44246327 IC50 > 200000 nM T59102 CMKF08 44246328 IC50 > 200000 nM T59102 CAO87V 44246329 IC50 > 200000 nM T59102 CLU2V3 44246330 IC50 = 17400 nM T59102 CHZ6Q1 44269004 IC50 = 10 nM T59102 CY6WC0 44299236 IC50 = 13000 nM T59102 C3RG0C 44299304 IC50 = 2300 nM T59102 CJM26I 44299321 IC50 = 4700 nM T59102 C9UGL3 44299325 IC50 = 10000 nM T59102 CJEZ96 44299338 IC50 = 9000 nM T59102 C8XGN5 44299339 IC50 = 5100 nM T59102 CNH34G 44299354 IC50 = 5600 nM T59102 C82MSD 44299360 IC50 = 18000 nM T59102 CSY8A3 44321301 IC50 > 100000 nM T59102 CCG2M5 44321317 IC50 = 60400 nM T59102 CY9ED1 44321395 IC50 > 100000 nM T59102 C5U1CR 44321686 IC50 > 10000 nM T59102 CETY53 44321717 IC50 = 66000 nM T59102 CV60ME 44321734 IC50 = 13800 nM T59102 C61OFE 44332377 IC50 > 1000 nM T59102 CI2NP3 44332378 IC50 = 160 nM T59102 CHKA01 44332616 IC50 = 820 nM T59102 CYAU21 44349046 IC50 = 409 nM T59102 CWFI13 44349291 IC50 = 564 nM T59102 C18OEK 44349292 IC50 = 50 nM T59102 C8XZ0Q 44349293 IC50 = 292 nM T59102 CYV2D7 44368815 IC50 = 357 nM T59102 CG6NE0 44394479 IC50 = 450 nM T59102 C6QL8A 44394480 IC50 = 970 nM T59102 C1BQ6T 44394484 IC50 = 240 nM T59102 CZ10CS 44394568 IC50 = 3590 nM T59102 CUF85K 44394571 IC50 = 400 nM T59102 CHO52Q 44394593 IC50 = 1010 nM T59102 CHCY97 44394612 IC50 = 2930 nM T59102 C7AB5H 44394617 IC50 = 350 nM T59102 C8M2PH 44394619 IC50 = 90 nM T59102 C58FRU 44394632 IC50 = 460 nM T59102 CB5S0R 44394633 IC50 = 220 nM T59102 CGLU71 44394634 IC50 = 10 nM T59102 CDU4J7 44394635 IC50 = 10 nM T59102 C4ZS5C 44394664 IC50 = 1150 nM T59102 C4ADU7 44394665 IC50 = 1400 nM T59102 C79BHS 44394670 IC50 = 180 nM T59102 CM0GF2 44394673 IC50 = 920 nM T59102 CF31RW 44394679 IC50 = 5 nM T59102 C53PUJ 44394680 IC50 = 280 nM T59102 C2JT4Q 44394704 IC50 = 770 nM T59102 C15GEC 44394709 IC50 = 1060 nM T59102 C6AEU0 44394722 IC50 = 5 nM T59102 C1GNQ7 44394737 IC50 = 4090 nM T59102 C2OAX3 44394745 IC50 = 510 nM T59102 C9RBN1 44394760 IC50 = 20 nM T59102 C6SRC1 44394772 IC50 = 1540 nM T59102 C70JWY 44394773 IC50 = 430 nM T59102 CPT6I0 44394781 IC50 = 3760 nM T59102 CLDS93 44394803 IC50 = 420 nM T59102 C81CTG 44394822 IC50 = 70 nM T59102 CRA0U1 44394842 IC50 = 2000 nM T59102 C0O8HG 44394845 IC50 = 630 nM T59102 C5PD3W 44394846 IC50 = 3090 nM T59102 C97CVT 44394847 IC50 = 100 nM T59102 CLT7U8 44394848 IC50 = 550 nM T59102 CD4U9G 44394849 IC50 = 590 nM T59102 CH8D0U 44394850 IC50 = 3420 nM T59102 CGOD34 44394853 IC50 = 2370 nM T59102 C6QNI1 44394865 IC50 = 80 nM T59102 CE8HO9 44394869 IC50 = 60 nM T59102 C43HND 44394870 IC50 = 100 nM T59102 C1L0SE 44394874 IC50 = 31700 nM T59102 CSE64J 44394875 IC50 = 370 nM T59102 C0XSD5 44394876 IC50 = 800 nM T59102 CW1QA3 44394898 IC50 = 13400 nM T59102 CFC1S9 44394899 IC50 = 160 nM T59102 C6GFO1 44394903 IC50 = 2130 nM T59102 CARP42 44394904 IC50 = 5190 nM T59102 CCT0R3 44394905 IC50 = 100 nM T59102 C8VJ2E 44405089 IC50 = 17 nM T59102 C8K4AL 44407237 IC50 > 50000 nM T59102 CUA18B 44407238 IC50 = 7600 nM T59102 C04HFE 44407248 IC50 > 50000 nM T59102 CR3O1C 44407275 IC50 = 15900 nM T59102 C70BFV 44407276 IC50 = 10200 nM T59102 CMH7W6 44407277 IC50 = 8700 nM T59102 C8W5YG 44447872 IC50 = 6 nM T59102 CUB12D 44449577 IC50 = 389 nM T59102 C3ZBV8 44450546 IC50 = 920 nM T59102 CLK0W7 44453682 IC50 > 1000 nM T59102 C0LY6E 44552561 IC50 = 6100 nM T59102 C7KRU3 44552562 EC50 = 2000 nM T59102 CYV71I 44555430 IC50 = 12.3 nM T59102 CJ1X9V 44565013 IC50 > 10000 nM T59102 CN2Q3D 44565014 IC50 = 1100 nM T59102 CM2GN3 44565015 IC50 > 10000 nM T59102 CV91YE 44572385 IC50 = 2600 nM T59102 C3CB2K 44572429 IC50 = 7800 nM T59102 CM2Q8J 44572430 IC50 = 5200 nM T59102 CAN4B0 44572431 IC50 = 1100 nM T59102 CMAT21 44572489 IC50 = 71000 nM T59102 CU1SY9 44572490 IC50 = 8700 nM T59102 CSD74G 44572491 IC50 = 13000 nM T59102 CA9WO3 44572537 IC50 = 47000 nM T59102 C06SLW 44572538 IC50 = 28000 nM T59102 CY8TG3 44572539 IC50 = 11000 nM T59102 C1JR4C 44572540 IC50 = 40000 nM T59102 CZ0PA9 44572581 IC50 = 2100 nM T59102 CD9VR5 44572582 IC50 = 13000 nM T59102 CG5UK0 44572584 IC50 = 11000 nM T59102 CMX32U 44572633 IC50 = 6200 nM T59102 C5WOE2 44586449 IC50 = 11800 nM T59102 C0VF8M 44586450 IC50 > 50000 nM T59102 C4K7NP 44586451 IC50 > 50000 nM T59102 C1JNR5 44586452 IC50 = 13700 nM T59102 C6T8UP 44586490 IC50 > 500000 nM T59102 CU95NI 44586526 IC50 = 100400 nM T59102 CBK9R3 44586527 IC50 > 500000 nM T59102 CA18IW 44586528 IC50 > 500000 nM T59102 C0YSZ2 44586577 IC50 = 77400 nM T59102 C8M5KI 44611919 IC50 = 22.8 nM T59102 C4KWJ3 45379956 IC50 > 50000 nM T59102 C2CU0B 45380067 IC50 > 50000 nM T59102 C6E2SC 45482700 IC50 > 10000 nM T59102 CZXH74 45482750 IC50 > 10000 nM T59102 CNI92D 46182735 IC50 = 230 nM T59102 CUA97D 46209401 IC50 = 120 nM T59102 C8YPN0 46225596 IC50 > 10000 nM T59102 C34JTS 46225597 IC50 = 5100 nM T59102 CGD73B 46225598 IC50 = 9100 nM T59102 C3E0PU 46225599 IC50 = 10000 nM T59102 CRDY89 46225610 IC50 = 3600 nM T59102 C0JMT8 46225611 IC50 > 10000 nM T59102 CF0D5J 46225612 IC50 = 1400 nM T59102 CFVO38 46225632 IC50 = 8700 nM T59102 CLZ1O6 46225634 IC50 = 4400 nM T59102 C07VDX 46225635 IC50 = 3800 nM T59102 CT70DX 46225640 IC50 = 7900 nM T59102 CJUF68 46225641 IC50 = 7700 nM T59102 C6AJ5N 46225647 IC50 = 3400 nM T59102 C2WCV1 46225648 IC50 = 9900 nM T59102 CBS96A 46225649 IC50 > 10000 nM T59102 C38BFC 46225657 IC50 = 2100 nM T59102 CD0A6F 46225658 IC50 > 10000 nM T59102 C1B3KS 46225663 IC50 = 2100 nM T59102 CU46XI 46225664 IC50 = 8000 nM T59102 CO3HS2 46225665 IC50 > 10000 nM T59102 C2UV1S 46225666 IC50 = 8200 nM T59102 CX5B1G 46225667 IC50 = 9200 nM T59102 C2Q9OH 46225668 IC50 > 10000 nM T59102 CM14FH 46225680 IC50 > 10000 nM T59102 CQS96E 46225681 IC50 > 10000 nM T59102 CJIK35 46225682 IC50 = 3800 nM T59102 C8S4QA 46225688 IC50 = 6700 nM T59102 C2P9QO 46228508 IC50 = 1550 nM T59102 C6E5PY 46228822 IC50 = 7490 nM T59102 C3T8AM 46228951 IC50 = 2390 nM T59102 CYZV41 46231219 IC50 = 2667 nM T59102 C7J5UP 46231220 IC50 = 858 nM T59102 CC96GZ 46231221 IC50 = 900 nM T59102 C9H4YO 46233889 IC50 = 49 nM T59102 CRT34L 46235770 IC50 = 27 nM T59102 CFR1C6 46845026 IC50 > 300000 nM T59102 C7NUY3 46847552 IC50 > 1000 nM T59102 CE3WH9 46865125 IC50 > 200000 nM T59102 C45LYT 46865445 IC50 > 200000 nM T59102 C1XEY4 46866615 IC50 > 200000 nM T59102 CF6K3E 46866616 IC50 > 200000 nM T59102 CA57MX 46886970 IC50 = 24600 nM T59102 CRGH62 46886971 IC50 = 183100 nM T59102 C68AGR 46886972 IC50 > 300000 nM T59102 CP32GW 46886973 IC50 > 300000 nM T59102 C48JWD 46886974 IC50 > 300000 nM T59102 C7H3MD 46887038 IC50 = 174900 nM T59102 C40NOR 46887039 IC50 = 43000 nM T59102 C7I4SB 46887074 IC50 = 182000 nM T59102 CI5QX2 46887110 IC50 = 171300 nM T59102 C0Q7NG 46887111 IC50 = 220400 nM T59102 CU15AN 46887112 IC50 = 110100 nM T59102 CD90BV 46887113 IC50 = 142200 nM T59102 CH3O9K 46887255 IC50 = 8500 nM T59102 C7NUT3 46887298 IC50 > 500000 nM T59102 CWV65D 46887299 IC50 > 500000 nM T59102 CH5BZ6 46887300 IC50 = 192400 nM T59102 C20UCB 46887348 IC50 > 500000 nM T59102 C0KEG5 46887349 IC50 > 500000 nM T59102 CY59RB 46887397 IC50 = 104200 nM T59102 C0WYM1 46898022 IC50 = 10000 nM T59102 CB92VU 46912443 IC50 = 2800 nM T59102 CU6HC7 46912444 IC50 = 34800 nM T59102 C8A4KU 46912445 IC50 > 500000 nM T59102 CNOS56 46912446 IC50 = 1300 nM T59102 CV38NE 46912546 IC50 > 500000 nM T59102 CQLT07 46913878 IC50 < 1000 nM T59102 CHSF07 49806372 IC50 > 1000 nM T59102 CVS85M 49831162 IC50 = 58 nM T59102 CR58WT 49840391 IC50 = 3 nM T59102 CA2J6U 49840467 IC50 = 13 nM T59102 CB0S2P 49842666 IC50 = 9200 nM T59102 C0NA9U 49842670 IC50 > 100000 nM T59102 CAI20B 49842778 IC50 = 21000 nM T59102 CRA74I 49842779 IC50 = 42000 nM T59102 CF91RS 49843531 IC50 > 10000 nM T59102 CE7D2J 49855568 IC50 = 3300 nM T59102 CFD9P3 49855569 IC50 = 1100 nM T59102 C1AU5N 49855758 IC50 = 2300 nM T59102 CIFK93 49855759 IC50 = 4000 nM T59102 CK48OJ 49855760 IC50 = 2300 nM T59102 CZI3M1 49855761 IC50 = 3900 nM T59102 CRPZ58 49855949 IC50 = 2500 nM T59102 CTU0K3 49855950 IC50 = 2700 nM T59102 CF85NL 49855951 IC50 = 4700 nM T59102 CF7YS9 49855952 IC50 = 1000 nM T59102 CJU38G 49855953 IC50 = 1800 nM T59102 CD2K4R 50908681 Ki > 1000000 nM T59102 C2Y6QS 50938552 IC50 > 10000 nM T59102 C9NYP4 51036677 IC50 > 10000 nM T59102 C4WRY3 51037112 IC50 > 10000 nM T59102 CRI28Z 51037948 IC50 > 10000 nM T59102 C4R7IM 52941368 IC50 = 71700 nM T59102 C7BY6M 52942956 IC50 > 200000 nM T59102 CA62KU 52944152 IC50 = 88200 nM T59102 CQV34K 52945403 IC50 > 200000 nM T59102 C97XZA 52946619 IC50 > 200000 nM T59102 CE0X5U 52947574 IC50 = 348000 nM T59102 CD9S4I 52947801 IC50 > 200000 nM T59102 CA6IL3 52947802 IC50 > 200000 nM T59102 C2KAJ4 52948634 IC50 > 500000 nM T59102 C0A1GQ 52949915 IC50 > 500000 nM T59102 C09SDH 53257410 IC50 > 10000 nM T59102 CZY0J7 53323592 IC50 > 100000 nM T59102 CNPM14 53341082 IC50 > 3000 nM T59102 C0SWH5 53348216 IC50 > 40000 nM T59102 CBK9Q6 53357848 IC50 > 10000 nM T59102 C8NA4L 53384644 IC50 > 30000 nM T59102 CVG90B 53389651 IC50 > 10000 nM T59102 C0JMY7 54673975 IC50 = 50500 nM T59102 C8AB1J 54759606 Ki = 19 nM T59102 CQ17GA 56640518 IC50 > 200000 nM T59102 CG20VK 56640520 IC50 > 200000 nM T59102 CZ9C8M 56640588 IC50 > 200000 nM T59102 CH0D7P 56640590 IC50 > 200000 nM T59102 C9DX3J 56649281 IC50 = 26 nM T59102 CR50TJ 56835147 IC50 = 2788 nM T59102 CI5ZJ7 56835161 IC50 > 100000 nM T59102 C2ML5S 56837168 IC50 = 518 nM T59102 CCW89V 56932477 IC50 = 185 nM T59102 CR3FK5 56932525 IC50 = 8 nM T59102 CY36EG 56945171 IC50 = 49 nM T59102 C4OG7H 56945172 IC50 = 93 nM T59102 CH0QA3 56945173 IC50 = 190 nM T59102 CM0NQ5 56945174 IC50 = 1100 nM T59102 CXKF03 56945175 IC50 = 550 nM T59102 CE07AQ 56945176 IC50 = 1600 nM T59102 CU86KC 56945272 IC50 = 23 nM T59102 C9SX7F 56945273 IC50 = 27 nM T59102 CG7VH5 56945274 IC50 = 72 nM T59102 C6WU4V 56945277 IC50 = 19 nM T59102 C7U9SL 56951304 IC50 > 50000 nM T59102 C0GQ9I 56951305 IC50 > 300000 nM T59102 C5YT6A 56951306 IC50 = 8920 nM T59102 CB03EH 56951307 IC50 = 193200 nM T59102 CP58NG 56954518 IC50 = 5 nM T59102 CAK91L 56955954 IC50 > 3600 nM T59102 C4YFJ5 57384105 IC50 = 1500 nM T59102 CV9RW5 57384106 IC50 = 1800 nM T59102 C4WE9B 57391179 IC50 = 10 nM T59102 CY10TP 57391180 IC50 = 6 nM T59102 CR4T2Y 57391283 IC50 = 129100 nM T59102 CU3DM9 57391295 IC50 > 1000 nM T59102 CBL74E 57392425 IC50 = 44300 nM T59102 CU7J9C 57393063 IC50 = 2 nM T59102 CD4HS3 57393074 IC50 = 9 nM T59102 CS60KL 57393075 IC50 > 2000 nM T59102 CWMT98 57394785 IC50 > 1000 nM T59102 CG18LI 57394786 IC50 = 34200 nM T59102 CEDP89 57394787 IC50 = 129300 nM T59102 C9PY4Q 57394798 IC50 = 10 nM T59102 C3F9VS 57394799 IC50 = 700 nM T59102 CP6W4C 57394879 IC50 > 500000 nM T59102 CVR13L 57394880 IC50 > 500000 nM T59102 CA4Q3Y 57395925 IC50 = 145900 nM T59102 C4CN6V 57396453 IC50 = 10 nM T59102 CCT58R 57396454 IC50 > 200 nM T59102 CXA5Z9 57396541 IC50 = 2 nM T59102 CPAH35 57396542 IC50 = 4 nM T59102 CUGP85 57396545 IC50 = 212400 nM T59102 CY8U1Q 57396557 IC50 = 0.9 nM T59102 CBUP96 57396646 IC50 = 159600 nM T59102 CWV96N 57398329 IC50 = 3 nM T59102 C8K1WJ 57398330 IC50 = 0.3 nM T59102 CXJ68F 57398331 IC50 = 229600 nM T59102 CBK02S 57399984 IC50 = 1 nM T59102 CNU4I7 57399985 IC50 = 2 nM T59102 CD9KF3 57399986 IC50 = 2 nM T59102 C0BA7P 57401686 IC50 = 20 nM T59102 CH56JP 57401785 IC50 = 3 nM T59102 C7YMG1 57401804 IC50 = 300 nM T59102 C20ZAX 57401805 IC50 = 4 nM T59102 C15YQW 57401806 IC50 = 20 nM T59102 CY5TJ9 57401807 IC50 = 4 nM T59102 C4L0SA 57401808 IC50 = 0.4 nM T59102 C4J0OD 57403506 IC50 = 0.8 nM T59102 CN0M3Z 57403518 IC50 = 300 nM T59102 CZSM95 57412684 IC50 > 10000 nM T59102 CN53XW 57428969 IC50 = 57.3 nM T59102 CE59QS 57505507 IC50 = 5.5 nM T59102 C8P6RD 57505528 IC50 = 15 nM T59102 C8R4FE 57991377 IC50 = 125.4 nM T59102 CH7L5N 58172700 IC50 = 768.4 nM T59102 C4V7FY 58191950 IC50 = 16000 nM T59102 CPCA29 58191961 IC50 = 70000 nM T59102 C7HF1L 58191965 IC50 = 7200 nM T59102 C8LWY9 58191997 IC50 = 28000 nM T59102 C4IBV1 59375998 IC50 = 12.7 nM T59102 CV8Q2D 59376002 IC50 = 89.9 nM T59102 CL3ND8 59376009 IC50 = 7.6 nM T59102 CC2AF9 59376012 IC50 = 19.4 nM T59102 CR7CG3 59376014 IC50 = 22.7 nM T59102 C60RIS 59376021 IC50 = 41.6 nM T59102 CT3Q5G 59376025 IC50 = 21.3 nM T59102 C97YSI 59376026 IC50 = 64.8 nM T59102 CEH5X6 59376027 IC50 = 40.1 nM T59102 C79EBT 59376032 IC50 = 40.7 nM T59102 C06DNI 59376037 IC50 = 12.1 nM T59102 C0XM7N 59376046 IC50 = 118.4 nM T59102 C70WCP 59376053 IC50 = 15.6 nM T59102 C5IHG9 59376058 IC50 = 18 nM T59102 CTK90V 59376059 IC50 = 260.3 nM T59102 C7ZY5I 59376061 IC50 = 101.4 nM T59102 CFT69X 59376062 IC50 = 70.3 nM T59102 C7D0BF 59376072 IC50 = 13.2 nM T59102 CD0RP7 59376074 IC50 = 62.1 nM T59102 C3HXC7 59376075 IC50 = 19.3 nM T59102 CAY6H8 59376079 IC50 = 13.3 nM T59102 CCX2W0 59376082 IC50 = 160.6 nM T59102 CLH49Z 59790029 IC50 = 1 nM T59102 C9QRX3 60098131 IC50 = 310 nM T59102 CSZA16 60155724 IC50 > 3600 nM T59102 CU79HD 60202383 IC50 = 243 nM T59102 C9ZCT2 62705065 IC50 > 1000 nM T59102 CK6WO0 66552478 IC50 < 10000 nM T59102 C37NKO 67129970 IC50 > 10000 nM T59102 CK80LJ 67130050 IC50 > 10000 nM T59102 CA63QI 67219716 IC50 > 5000 nM T59102 CV63UL 67240318 IC50 > 10000 nM T59102 C7GRV2 68755406 IC50 > 10000 nM T59102 CCS20X 69063773 IC50 = 3 nM T59102 CEB12M 70681395 IC50 = 3 nM T59102 CH27DE 70681409 IC50 = 2 nM T59102 CN29RI 70681410 IC50 = 5 nM T59102 CG93IE 70683519 IC50 = 0.3 nM T59102 CXSN14 70685622 IC50 = 6 nM T59102 CL24MP 70687766 IC50 = 0.2 nM T59102 C51DHN 70689791 IC50 = 3 nM T59102 C6ITV3 70689792 IC50 = 0.9 nM T59102 CMLY63 70689816 IC50 = 0.5 nM T59102 C08ASR 70689830 IC50 = 4 nM T59102 C4TF3G 70691955 IC50 = 5 nM T59102 CTWD94 70691956 IC50 = 50 nM T59102 CIK5N2 70691957 IC50 = 10 nM T59102 C8RZP3 70691958 IC50 = 5 nM T59102 C0XRC9 70691981 IC50 = 3 nM T59102 C9RT8C 70693982 IC50 = 0.7 nM T59102 C2X1KJ 70694006 IC50 = 0.4 nM T59102 C54VLD 70694007 IC50 = 0.2 nM T59102 C6O3SM 70696108 IC50 = 50 nM T59102 CEBO91 71452977 IC50 > 10000 nM T59102 C9DIK2 71512060 IC50 = 2102 nM T59102 C6HF8S 71521082 IC50 = 35400 nM T59102 C9Z3AI 71521083 IC50 > 5000 nM T59102 C5OBF0 71525245 IC50 > 500000 nM T59102 CJX73B 71525246 IC50 > 500000 nM T59102 CCN90I 71525247 IC50 = 331500 nM T59102 CY6JA9 71525248 IC50 > 500000 nM T59102 CGQJ60 71525249 IC50 > 500000 nM T59102 CMKD15 71525283 IC50 = 89700 nM T59102 C3OJ6R 71525284 IC50 > 500000 nM T59102 CP5Q2U 71525285 IC50 = 430100 nM T59102 CZ8N0J 71525286 IC50 > 500000 nM T59102 CG31MI 71525287 IC50 > 500000 nM T59102 CRX81Q 71575642 IC50 = 408 nM T59102 CGK76E 71583411 IC50 > 200000 nM T59102 CB5WX0 71583412 IC50 > 200000 nM T59102 CI8K3T 71583527 IC50 = 196200 nM T59102 C6FGI0 71583528 IC50 > 200000 nM T59102 C3QGE7 71583529 IC50 = 172200 nM T59102 CS9HX7 71583530 IC50 = 70600 nM T59102 CQTZ32 71583531 IC50 > 200000 nM T59102 C0G5RS 71583532 IC50 > 200000 nM T59102 CVEY46 71583533 IC50 = 170800 nM T59102 CX6TR7 71583634 IC50 > 200000 nM T59102 CR15QP 71583635 IC50 = 196200 nM T59102 CZ31PU 71583657 IC50 > 10000 nM T59102 CU1IL6 71741204 IC50 > 100000 nM T59102 CN1GA3 71741327 IC50 > 100000 nM T59102 COS5D7 71741328 IC50 > 100000 nM T59102 C8PWZ0 71741329 IC50 > 100000 nM T59102 CT4XR9 71741332 IC50 > 50000 nM T59102 C4Q6FE 71815105 IC50 = 86.9 nM T59102 CJ9OX6 71815106 IC50 = 176.7 nM T59102 CCKL45 72191698 IC50 = 395.7 nM T59102 C60TUV 72737208 IC50 > 10000 nM T59102 CJ3WA6 72737404 IC50 > 10000 nM T59102 C8SIL6 73349435 IC50 = 1.42 nM T59102 CVNW01 73386831 IC50 > 1000 nM T59102 C2PAK9 73438493 IC50 = 1055 nM T59102 CBAT06 76071144 IC50 = 1083 nM T59102 CH8W7D 77461036 IC50 > 1000 nM T59102 CA65HB 78319164 IC50 = 20 nM T59102 CCJ43A 86302281 IC50 > 10000 nM T59102 CB5NJ4 86302541 IC50 = 4.6 nM T59102 CPG3A5 86302574 IC50 > 30000 nM T59102 C08WGI 86566799 IC50 = 16.3 nM T59102 C5S3YB 90645165 IC50 = 92.3 nM T59102 C6Q4DH 90645475 IC50 = 29.9 nM T59102 C89HTB 90645476 IC50 = 56.5 nM T59102 C9ASG1 90645478 IC50 = 27.1 nM T59102 COY53U 90645479 IC50 = 16.2 nM T59102 C48OSQ 90645480 IC50 = 23.1 nM T59102 CL8GW5 90645481 IC50 = 66.1 nM T59102 CL7SC6 90645482 IC50 = 28.3 nM T59102 CI3OD6 90645484 IC50 = 63.5 nM T59102 CX29IY 90655145 IC50 > 10000 nM T59102 C96DTL 90682879 IC50 = 21.9 nM T59102 CI97DL 102431709 IC50 = 19000 nM T59102 C09MIG 102431710 IC50 = 1500 nM T59102 C5HRO7 102431711 IC50 = 1400 nM T59102 CTGP06 117996541 IC50 > 10000 nM T59102 CY7BI2 118706214 IC50 > 10000 nM T59102 C2IN3C 118710236 IC50 = 8.1 nM T59102 CF2YR1 118710237 IC50 = 1.54 nM T59102 C4AHL2 118711367 IC50 = 5800 nM T59102 C46QUT 118717614 IC50 > 200000 nM T59102 CJC34Y 118717615 IC50 > 200000 nM T59102 CFEP93 118717616 IC50 > 200000 nM T59102 CEC4H0 118717617 IC50 > 200000 nM T59102 CU2TG3 118717618 IC50 > 200000 nM T59102 C5OL0W 118717619 IC50 > 200000 nM T59102 C3KLI5 118723185 IC50 = 500 nM T59102 C5UZ9X 118723186 IC50 = 4000 nM T59102 C3XV6L 118723187 IC50 > 100000 nM T59102 CLD41J 118723188 IC50 > 100000 nM T59102 C0H9YD 118723189 IC50 = 5000 nM T59102 CP8FW0 118723190 IC50 = 13000 nM T59102 CCV0H1 118723191 IC50 = 13000 nM T59102 C1J7QE 118723192 IC50 = 12000 nM T59102 CMHV05 118723193 IC50 = 32000 nM T59102 CRQY80 118723194 IC50 = 300 nM T59102 CVZM84 118723195 IC50 = 1000 nM T59102 CP8Z6I 118723196 IC50 = 14000 nM T59102 CI6HB3 118723197 IC50 = 56000 nM T59102 CVGE25 118723198 IC50 = 2000 nM T59102 C78BAF 118723199 IC50 = 9000 nM T59102 C02HAD 118723200 IC50 = 3000 nM T59102 CDAN63 118723201 IC50 = 26000 nM T59102 CL6T5K 118723202 IC50 = 1000 nM T59102 CDQ92V 118723203 IC50 = 8000 nM T59102 CV0B6M 118723204 IC50 = 2000 nM T59102 CX4E1N 118723205 IC50 = 1000 nM T59102 C8BU5O 118723206 IC50 = 2000 nM T59102 C2G1TN 118723207 IC50 = 7000 nM T59102 C1JO0D 118723208 IC50 = 22000 nM T59102 CYXF26 118723209 IC50 = 31000 nM T59102 C7JYP8 118723210 IC50 = 800 nM T59102 CV6HJ8 118723211 IC50 = 5000 nM T59102 CI6QA2 118723212 IC50 = 100 nM T59102 C3XKJ9 118723213 IC50 = 2000 nM T59102 CU1B5W 118723214 IC50 = 19000 nM T59102 CD5HK1 118723215 IC50 = 8000 nM T59102 CU06YS 118723216 IC50 > 100000 nM T59102 CWYF91 118729842 IC50 = 40.4 nM T59102 CR54XL 118729843 IC50 = 66.1 nM T59102 CF3X9J 118729844 IC50 = 166.3 nM T59102 CT3Q6C 118729845 IC50 = 50.1 nM T59102 C1QWK6 118729846 IC50 = 24.6 nM T59102 CWUA61 118729847 IC50 = 25 nM T59102 C63CDP 118729848 IC50 = 73.2 nM T59102 C1WB7L 118729849 IC50 = 198 nM T59102 C8A7ZT 118729850 IC50 = 58.2 nM T59102 C9WDF4 118729851 IC50 = 84 nM T59102 CT08EZ 118729852 IC50 = 132 nM T59102 C08KEM 122179540 IC50 = 2000 nM T59102 CG0RP7 122179547 IC50 = 2200 nM T59102 C1A0SQ 122179548 IC50 = 4600 nM T59102 C4X7SD 122192466 IC50 = 1982 nM T59102 CNX0Q2 122193763 IC50 = 850 nM T59102 CWV0C3 122193764 IC50 = 2120 nM T59102 CSG98Y 122193765 IC50 = 2820 nM T59102 CCLQ75 122193769 IC50 = 320 nM T59102 CXDR48 122193770 IC50 = 570 nM T59102 CPA8C5 122193773 IC50 = 2300 nM T59102 CY30FL 123752658 IC50 = 5.5 nM T59102 C8KXV1 127025843 IC50 > 1000 nM T59102 C1XD6R 127029809 IC50 = 526.5 nM T59102 CI1E5W 127029864 IC50 = 4.57 nM T59102 CKS28E 127034802 IC50 = 64.2 nM T59102 CKX40V 127037812 IC50 = 223.9 nM T59102 C70RUP 127038480 IC50 > 10000 nM T59102 C3WCN8 127041777 IC50 > 10000 nM T59102 CC58IQ 127043948 IC50 = 120 nM T59102 CHK16Q 127045929 IC50 > 1000 nM T59102 CY3J0C 127047591 IC50 > 1000 nM T59102 CF5D2Y 129318936 IC50 = 6115 nM T59102 C0FM1R 130196825 IC50 = 392 nM T59102 CUO0C5 132156633 IC50 > 10000 nM T59102 C6OMB1 132204257 IC50 = 606 nM T59102 C6ROQ3 132546210 IC50 = 80 nM T59102 CJ04HZ 132585195 IC50 < 1 nM T59102 CERS64 132937256 IC50 = 26197 nM T59102 CN9SD7 132942957 IC50 = 51.4 nM T59102 CMP2S9 132942958 IC50 = 62.2 nM T59102 CN35SO 134146628 IC50 > 1000 nM T59102 CIK38Q 134229735 IC50 = 63.4 nM T59102 CYL5V1 134694986 IC50 > 30000 nM T59102 CLCO61 135398510 EC50 = 51 nM T59102 CN5T7W 135400982 IC50 = 12 nM T59102 CVJ07T 135402853 IC50 = 70 nM T59102 CBK6I2 135407156 IC50 = 30 nM T59102 CMVS34 135410282 IC50 = 10 nM T59102 CUT52Q 135421574 IC50 = 19000 nM T59102 CK9D4A 135428921 IC50 = 4500 nM T59102 C8X5SV 135433815 IC50 = 20 nM T59102 CNZ04G 135453357 IC50 = 4 nM T59102 CS63IO 135476717 IC50 = 65 nM T59102 C2MAC7 135536640 IC50 > 100000 nM T59102 CW08GF 135674125 IC50 = 70 nM T59102 CLS64T 135674129 IC50 = 0.9 nM T59102 C54ABM 135674133 IC50 = 0.3 nM T59102 CM7YH4 135674136 IC50 = 5 nM T59102 C1WSO7 135674140 IC50 = 130 nM T59102 CA0Y7V 135674142 IC50 = 5 nM T59102 CM90FP 135674144 IC50 = 0.9 nM T59102 C3CP1X 135674147 IC50 = 0.3 nM T59102 CBSV42 135674149 IC50 = 5 nM T59102 C1NTB0 135674153 IC50 = 2 nM T59102 CID0W9 135674167 IC50 = 0.1 nM T59102 C1DL9J 135674173 IC50 = 30 nM T59102 CO89UX 135674193 IC50 = 8 nM T59102 C2H3XB 135926086 IC50 = 2 nM T59102 C7BES6 135926087 IC50 = 2 nM T59102 CNTK81 135926088 IC50 = 7 nM T59102 CQ64OH 135926089 IC50 = 39 nM T59102 CXG7O4 135926090 IC50 = 0.1 nM T59102 CN4FG3 135926091 IC50 = 14 nM T59102 C7NZU3 135926094 IC50 > 25000 nM T59102 CL6HQ4 135926104 IC50 = 1 nM T59102 CE37KQ 135926113 IC50 = 0.7 nM T59102 C1ZRT7 135926114 IC50 = 1 nM T59102 CU5W2V 135926115 IC50 = 7 nM T59102 C1D3EW 135926116 IC50 = 0.6 nM T59102 C2PAV1 135971426 IC50 = 10000 nM T59102 CHA4N2 136013680 IC50 > 10 nM T59102 CLN6Y8 136026516 IC50 > 100000 nM T59102 CG1R7B 136087060 IC50 = 7000 nM T59102 C5QZ4H 136126664 IC50 = 1100 nM T59102 CB8RX0 136126665 IC50 = 0.2 nM T59102 CZ7EX0 136183413 IC50 = 3200 nM T59102 CDT7E4 136211077 IC50 > 1000 nM T59102 C9RE8D 136215817 IC50 = 530.6 nM T59102 C1YUD0 136219394 IC50 > 10 nM T59102 CIU8W3 136254389 IC50 > 10 nM T59102 C35MBU 136299423 IC50 = 45 nM T59102 C0W8KA 136299435 IC50 = 4.3 nM T59102 C5G4ES 136299436 IC50 = 3.2 nM T59102 C83OXU 137007054 IC50 = 12000 nM T59102 CCM42D 137249694 IC50 = 14.3 nM T59102 C25ERN 137631967 IC50 = 1 nM T59102 CFUY16 137633842 IC50 > 200000 nM T59102 CNX0F9 137634126 IC50 = 106.2 nM T59102 CHC70D 137634143 IC50 = 3.26 nM T59102 CI1E8V 137634241 IC50 = 5190 nM T59102 C85WBP 137634338 IC50 = 9 nM T59102 CAD3C5 137634686 IC50 = 45.52 nM T59102 CS23KQ 137635618 IC50 = 90100 nM T59102 C5JD9N 137635898 IC50 = 10.3 nM T59102 CK5Y3P 137635915 IC50 = 65.24 nM T59102 C06JRX 137637094 IC50 > 10 nM T59102 CU24QC 137638448 IC50 = 90.3 nM T59102 CO9D4W 137639407 IC50 = 31.36 nM T59102 C3UBE2 137639638 IC50 > 200 nM T59102 CU8YX6 137643005 IC50 = 58200 nM T59102 C2T6FV 137644825 IC50 = 29.79 nM T59102 C1DK0P 137651391 IC50 = 1 nM T59102 C5F3LP 137651946 IC50 = 83.17 nM T59102 CQUY83 137652218 IC50 > 200000 nM T59102 C9JT1N 137655519 IC50 = 60500 nM T59102 C9TEU1 137655771 IC50 = 27.11 nM T59102 CKVO51 137657233 IC50 = 30.2 nM T59102 CV5H3Z 137657932 IC50 > 100 nM T59102 CQMB10 137658515 IC50 = 197 nM T59102 C7IVT9 137658762 IC50 > 200 nM T59102 CQE9M4 137661156 IC50 = 67.85 nM T59102 CM0N3T 137661420 IC50 = 7.2 nM T59102 CT43IF 137661858 IC50 = 8.1 nM T59102 CIWG23 138393067 IC50 = 88 nM T59102 C07EKN 138454794 IC50 = 2075 nM T59102 C5LQU9 138479230 IC50 = 673.6 nM T59102 CSRI06 138547901 IC50 > 1000 nM T59102 CUXO19 138617501 IC50 > 1000 nM T59102 C6AK0N 139030518 IC50 = 97 nM T59102 C34CKN 141523354 IC50 = 19.46 nM T59102 CB3Z1W 145949428 IC50 = 180 nM T59102 CCM27G 145949662 IC50 = 64.6 nM T59102 CVJS01 145949677 IC50 = 12 nM T59102 CWQA26 145949916 IC50 = 34.3 nM T59102 CYF32C 145950953 IC50 = 15 nM T59102 CRXJ25 145951211 IC50 = 91 nM T59102 C4LBC0 145951650 IC50 = 116.2 nM T59102 CR9LH4 145952520 IC50 = 92.7 nM T59102 CC72WG 145953067 IC50 = 7800 nM T59102 C60XZR 145953297 IC50 = 19 nM T59102 CSLC73 145953358 IC50 = 44.2 nM T59102 CAL30B 145953560 IC50 = 15 nM T59102 C0V8SM 145954139 IC50 = 25 nM T59102 CDRQ06 145955547 IC50 = 45.5 nM T59102 C8VN1Y 145955561 IC50 = 27 nM T59102 C2O9XD 145955651 IC50 = 91.7 nM T59102 C1IX5N 145956333 IC50 = 22 nM T59102 C6ZNJ1 145956488 IC50 = 34 nM T59102 CLZH04 145956490 IC50 = 39 nM T59102 C5VSC7 145956704 IC50 = 177 nM T59102 CY69RH 145956768 IC50 = 49.2 nM T59102 CIW0V9 145956964 IC50 = 241.6 nM T59102 CB74GR 145957221 IC50 = 24 nM T59102 CB1MI9 145957910 IC50 = 4.5 nM T59102 CS47UF 145958497 IC50 = 14 nM T59102 CRVO52 145960991 IC50 > 500 nM T59102 CV4M1Z 145961849 IC50 = 60.7 nM T59102 C9PKU6 145963750 IC50 = 5.3 nM T59102 CTUF34 145966712 IC50 = 111 nM T59102 C4OD9Q 145967187 IC50 = 214.5 nM T59102 CNVT54 145971746 IC50 = 61 nM T59102 C3Q4XM 145972183 IC50 = 13 nM T59102 C71ZJX 145972445 IC50 = 135.1 nM T59102 CG8R0P 145972697 IC50 = 1.5 nM T59102 C74TYP 145975351 IC50 = 482.1 nM T59102 CCS92I 145982511 IC50 = 510 nM T59102 CWE21T 145982588 IC50 = 3250 nM T59102 CC12YA 145982666 IC50 = 57.8 nM T59102 CF4BO8 145982785 IC50 = 28.9 nM T59102 CM6ZS7 145982824 IC50 = 63 nM T59102 CZ3CG9 145982825 IC50 = 1260 nM T59102 CF28AU 145983389 IC50 = 42.6 nM T59102 CRL19G 145983447 IC50 = 40 nM T59102 C48UZH 145983504 IC50 = 2230 nM T59102 C8BZC5 145983753 IC50 = 20 nM T59102 CD5L8O 145983778 IC50 > 200 nM T59102 CNK7I9 145984104 IC50 = 3520 nM T59102 C4C2OM 145984258 IC50 = 8 nM T59102 C9DHL3 145984282 IC50 = 3780 nM T59102 CVT02P 145984555 IC50 = 20 nM T59102 CHW8E5 145984671 IC50 = 1230 nM T59102 CYG42V 145984818 IC50 > 200 nM T59102 CFS7D5 145984941 IC50 > 200 nM T59102 C05IMJ 145984942 IC50 = 38.9 nM T59102 C9Q5VI 145985608 IC50 = 820 nM T59102 CA2TW8 145985737 IC50 = 290 nM T59102 CS9C8J 145986155 IC50 > 200 nM T59102 C1Y5MO 145987062 IC50 = 1.81 nM T59102 CI85EU 145998085 IC50 = 1013 nM T59102 C2MD1Q 155513187 IC50 > 10000 nM T59102 C86HPW 155518524 IC50 = 81000 nM T59102 CU6Z5O 155520650 IC50 = 150 nM T59102 CY6NE1 155523855 IC50 = 100 nM T59102 CRP7Q6 155525519 IC50 = 110 nM T59102 CTD5R7 155528337 IC50 = 450 nM T59102 CLEJ03 155529517 IC50 = 230 nM T59102 CS69CA 155532132 IC50 = 25.3 nM T59102 C3NZO0 155533789 IC50 = 90 nM T59102 C2DJ0A 155534253 IC50 = 2010 nM T59102 C37RFQ 155534994 IC50 = 1590 nM T59102 CE46SL 155540854 IC50 > 30000 nM T59102 C5O4JM 155540856 IC50 > 30000 nM T59102 C7SF2C 155547229 IC50 = 356 nM T59102 C6URZ7 155550475 IC50 = 1820 nM T59102 CGVU70 155554426 IC50 > 30000 nM T59102 CUA73V 155555832 IC50 = 330 nM T59102 C8L6PM 155561965 IC50 = 3790 nM T59102 C81JZW 155563388 IC50 = 390 nM T59102 CM23DI 155565660 IC50 = 1290 nM T59102 CK10HA 155568167 IC50 = 3640 nM T59102 CBWO68 49800164 IC50 = 28 nM T59102 D00ATA 5908088 IC50 = 12000 nM T59102 D00GVV 5329155 IC50 = 920 nM T59102 D02BXJ 46864270 IC50 = 2.6 nM T59102 D04FNY 25195216 IC50 = 40 nM T59102 D05NKG 16760286 IC50 = 316.23 nM T59102 D05WTI 11550535 IC50 = 317 nM T59102 D06QWO 14824655 IC50 > 10 ug.mL-1 T59102 D07IHM 9823787 IC50 > 10000 nM T59102 D07OSK 6419834 IC50 = 4000 nM T59102 D09HVH 135566652 IC50 > 10 nM T59102 D09LPL 5329103 IC50 = 3 nM T59102 D09QBA 23378546 IC50 > 10000 nM T59102 D09TNR 9850161 IC50 = 69 nM T59102 D0A1CM 5281855 IC50 = 1300 nM T59102 D0A4XJ 5289418 IC50 = 510 nM T59102 D0BW4G 10907042 IC50 = 130 nM T59102 D0C2GE 67161540 IC50 = 1.3 nM T59102 D0D6MH 11617559 IC50 > 10000 nM T59102 D0EE6A 6398883 IC50 = 640 nM T59102 D0G3SZ 6918469 IC50 = 5.9 ug.mL-1 T59102 D0H1OK 11562302 Ki = 2090 nM T59102 D0HE0E 5941540 IC50 = 5100 nM T59102 D0I3XZ 11601743 IC50 = 171 nM T59102 D0L3FK 5289419 IC50 > 10000 nM T59102 D0M4QA 56935577 IC50 = 10.1 nM T59102 D0R2WK 16038120 IC50 = 3220 nM T59102 D0U3WQ 9817165 IC50 = 90 nM T59102 D0UN9O 3385203 IC50 = 1000 nM T59102 D0X1RH 16051023 IC50 = 420 nM T59102 D0XS9E 5330535 IC50 = 90 nM T59102 D0YE1X 9927943 IC50 = 30 nM T59102 D0YZ7H 9797370 IC50 = 3 nM T59102 D0Z7TM 22273644 IC50 > 2000 nM T85272 D03DAP 3356 IC50 = 209000 nM T85272 D04OSE 4485 IC50 = 96000 nM T85272 D08YIN 1727 IC50 = 89000 nM T85272 D0OB1J 39186 IC50 = 144000 nM T85272 D0U5CE 1548943 IC50 = 29000 nM T85272 D0K9IF 71666749 IC50 > 30000 nM T85272 C29SPL 5867 EC50 = 33000 nM T85272 C6HA8E 5388709 IC50 > 30000 nM T85272 C8W2QA 6439099 IC50 > 30000 nM T85272 C8NM2I 11538313 EC50 = 7000 nM T85272 CA5W9R 11618060 EC50 = 1200 nM T85272 CLT3Z7 11695929 EC50 = 1700 nM T85272 CW9V0Y 13088125 EC50 = 6000 nM T85272 C8JA3E 13703975 EC50 = 4300 nM T85272 C91QFN 25019282 IC50 = 2660 nM T85272 CQSZ72 90675942 IC50 > 30000 nM T85272 CTBD74 90675943 IC50 > 30000 nM T85272 CM12LR 102597975 IC50 > 30000 nM T85272 CQJ49Y 122187245 IC50 = 0.0067 nM T85272 CSW57U 122187246 IC50 = 0.0077 nM T85272 C98BUE 122187247 IC50 = 0.0034 nM T85272 CVT7A6 122187248 IC50 = 0.0027 nM T85272 CI9ZH1 122187249 IC50 = 0.0078 nM T85272 CHJ75V 122187250 IC50 = 0.0095 nM T85272 C20TPX 122187251 IC50 = 0.0028 nM T85272 CQ17ZP 122187252 IC50 = 0.011 nM T85272 C2XUA5 122187253 IC50 = 0.308 nM T85272 CQTJ57 122187272 IC50 = 0.0078 nM T85272 CX2YG6 122187273 IC50 = 0.0181 nM T85272 C4CLN5 122187274 IC50 > 3.333 nM T85272 CF5M8V 122187275 IC50 = 0.49 nM T85272 C24MEW 122187276 IC50 > 3.333 nM T85272 CI7VL5 122187277 IC50 > 3.333 nM T85272 COX2P3 122187278 IC50 = 0.014 nM T85272 CY9RL0 122187279 IC50 = 0.02 nM T85272 CT5B4D 122187280 IC50 = 0.028 nM T85272 C42SZA 122187281 IC50 = 1.8 nM T85272 C6S3XG 122187282 IC50 = 0.0018 nM T85272 C0YG3Z 122187283 IC50 = 0.0057 nM T85272 C1F5PE 122187284 IC50 = 0.0023 nM T85272 C26VHJ 122187285 IC50 = 0.0049 nM T85272 C24JCI 122187286 IC50 = 0.0083 nM T85272 CW4SU9 122187287 IC50 = 0.001 nM T85272 CT0GS6 122187288 IC50 = 0.007 nM T85272 CCO3Y2 122187289 IC50 = 3.279 nM T85272 C1ENW4 122187290 IC50 = 0.046 nM T85272 CFH36G 122187291 IC50 = 0.0172 nM T85272 C3CY5N 122187292 IC50 = 0.004 nM T85272 CY69QI 122187293 IC50 = 0.0027 nM T85272 C05WQZ 122187294 IC50 = 0.003 nM T85272 C1LW9V 122187295 IC50 = 0.0195 nM T85272 CBMT85 122187296 IC50 = 0.0018 nM T85272 C8AKN9 122187297 IC50 = 0.0154 nM T85272 CDM71F 122187298 IC50 = 0.055 nM T85272 CCM08N 122187299 IC50 = 0.0038 nM T85272 C7V2TW 122187300 IC50 = 0.0028 nM T85272 C81QSJ 122187301 IC50 > 3.333 nM T85272 C1IPG9 122187302 IC50 = 0.0324 nM T85272 C0RE2W 122187303 IC50 > 3.333 nM T85272 C9JDM3 122187304 IC50 > 3.333 nM T85272 C5QXR6 122187305 IC50 = 0.0087 nM T85272 C50RMQ 122187306 IC50 = 0.0018 nM T85272 C5Z9PU 122187307 IC50 = 0.07 nM T85272 CT0V4W 122187308 IC50 > 3.333 nM T85272 CX06CZ 122187309 IC50 = 0.008 nM T85272 CK9T7F 122187310 IC50 = 0.59 nM T85272 CC2LE0 122187311 IC50 = 0.0036 nM T85272 CS34VD 122187312 IC50 = 0.002 nM T85272 CIU9T5 122187313 IC50 = 0.0031 nM T85272 CS8QW7 122187314 IC50 = 0.0042 nM T85272 CID97N 122187315 IC50 = 0.458 nM T85272 CZ08GP 122187316 IC50 = 0.0026 nM T85272 C0P6IC 122187317 IC50 > 3.333 nM T85272 CY7M0F 122187318 IC50 = 0.005 nM T85272 CQZK10 122187319 IC50 = 0.0033 nM T85272 C62FDT 122187320 IC50 = 0.0024 nM T85272 C3QZY1 122187321 IC50 = 0.0044 nM T85272 C8B4YL 122187322 IC50 = 0.005 nM T85272 CWV12K 122187323 IC50 = 0.0527 nM T85272 CWVP15 122187324 IC50 = 2.342 nM T85272 CEW35A 122187325 IC50 = 0.0017 nM T85272 CP43GQ 122187326 IC50 = 0.0021 nM T85272 CH46BC 122187327 IC50 = 0.04 nM T85272 C6KW2B 122187328 IC50 = 0.004 nM T85272 C87MGD 122187329 IC50 = 0.0028 nM T85272 C0U9QN 122187330 IC50 = 0.0335 nM T85272 CH4G1L 122187331 IC50 = 0.075 nM T85272 C4ZR9M 122187332 IC50 = 0.266 nM T85272 CM8A1Y 122187333 IC50 = 0.174 nM T85272 CU3IE9 122187334 IC50 = 0.005 nM T85272 CYN12K 122187335 IC50 = 0.0051 nM T85272 CDE52G 122187336 IC50 = 0.74 nM T85272 CZH25J 122187337 IC50 = 0.011 nM T85272 CQP1R4 122187338 IC50 = 0.6 nM T85272 C3QS0A 122187339 IC50 = 9.5 nM T85272 CAFO71 122187340 IC50 = 0.015 nM T85272 CNYJ15 122187341 IC50 = 29.26 nM T85272 CY62QW 122187342 IC50 = 13.22 nM T85272 CCV2G0 122187343 IC50 > 33.33 nM T85272 C0Z8JH 122187344 IC50 = 0.014 nM T85272 CVT8Z7 122187345 IC50 = 0.847 nM T85272 C2YI7W 122187346 IC50 = 0.214 nM T85272 CO7MU2 122187445 IC50 = 0.002 nM T85272 C8QN9Z 122187446 IC50 = 0.0068 nM T85272 C09YUX 122187447 IC50 = 0.005 nM T85272 C8I6TF 122187448 IC50 = 0.0022 nM T85272 CR68ZK 122187449 IC50 = 0.0035 nM T85272 CTY96B 122187450 IC50 = 0.0053 nM T85272 C4WG0M 122187451 IC50 = 0.0182 nM T85272 CLS4H7 122187452 IC50 = 0.0014 nM T85272 CM23CQ 122187453 IC50 = 0.76 nM T85272 CJF8X1 122187454 IC50 > 3.333 nM T85272 C54PSK 122187455 IC50 = 0.005 nM T85272 CGS5Q1 122187456 IC50 = 0.0014 nM T85272 CW0MH4 122187457 IC50 = 0.0011 nM T85272 CXAV52 122187458 IC50 = 0.0034 nM T85272 C3D8EQ 122187459 IC50 = 0.446 nM T85272 CBUT59 122187460 IC50 = 0.005 nM T85272 C1XL3M 122187461 IC50 = 0.004 nM T85272 CBS95M 122187462 IC50 = 0.005 nM T85272 CY79JC 122187463 IC50 = 0.0037 nM T85272 CAY0P4 122187464 IC50 = 0.006 nM T85272 CRQ98D 122187465 IC50 = 0.006 nM T85272 CXP98T 122187466 IC50 = 0.0042 nM T85272 C5TJU8 122187467 IC50 > 3.333 nM T85272 CP7C2I 122187468 IC50 = 0.028 nM T85272 CKC0L8 122187469 IC50 = 0.305 nM T85272 CV3T2C 122187470 IC50 = 0.011 nM T85272 CN5OQ2 122187471 IC50 = 0.0009 nM T85272 CI0J4A 122187472 IC50 = 0.0274 nM T85272 CM14KC 122187473 IC50 = 0.0157 nM T85272 COFI26 122187474 IC50 = 0.0489 nM T85272 CTXG58 122187475 IC50 = 0.0102 nM T85272 CZWG59 122187476 IC50 > 3.333 nM T85272 C1TVY5 122187477 IC50 = 0.0033 nM T85272 CS6FK8 122187478 IC50 > 3.333 nM T85272 CJC21F 122187479 IC50 = 0.0262 nM T85272 C3ZE4Y 122187480 IC50 > 3.333 nM T85272 CS0U8H 122187481 IC50 > 3.333 nM T85272 CY0NV5 122187482 IC50 = 0.0091 nM T85272 C8SHE5 122187483 IC50 = 1.018 nM T85272 CHYI14 122187484 IC50 = 2.42 nM T85272 CEH14V 122187485 IC50 > 3.333 nM T85272 CG98KU 122187486 IC50 = 0.0032 nM T85272 C3P8WN 122187487 IC50 = 0.0061 nM T85272 C9MJ2K 122187488 IC50 = 0.0061 nM T85272 C7J0YH 122187489 IC50 = 0.0044 nM T85272 C4NYT7 122187490 IC50 = 0.04 nM T85272 CMT25I 122187491 IC50 = 0.0015 nM T85272 CQEV80 122187492 IC50 = 0.0076 nM T85272 CY07HP 122187493 IC50 = 1.2 nM T85272 CD0EU3 122187494 IC50 = 0.0256 nM T85272 CQZ0R1 122187495 IC50 = 0.032 nM T85272 CZU4N2 122187496 IC50 = 0.0073 nM T85272 CITK91 122187497 IC50 = 0.0059 nM T85272 C69JKA 122187498 IC50 = 0.0042 nM T85272 C6R5CY 122187499 IC50 = 0.029 nM T85272 CM87YE 122187500 IC50 = 0.0045 nM T85272 CP4GJ7 122187501 IC50 = 0.051 nM T85272 CB14ES 122187502 IC50 = 0.004 nM T85272 CEGB98 122187503 IC50 = 0.042 nM T85272 CU61JG 137651545 IC50 = 13000 nM T85272 CW9P6A 145964460 IC50 > 30000 nM T85272 CQR49Z 145965116 IC50 > 30000 nM T85272 CR6L2G 145967358 IC50 > 30000 nM T85272 CHXE25 145978207 IC50 > 30000 nM T85272 D06PZZ 5413 IC50 = 30000 nM T85272 D08BMM 6312649 IC50 > 30000 nM T85272 D0R9CF 11302540 IC50 = 250 nM T96736 CR57DL 50803848 IC50 = 35000 nM T96736 CP79TH 52931882 IC50 = 2580 nM T96736 CPE79U 52931883 IC50 = 3280 nM T96736 C9LGO3 52931939 IC50 = 2620 nM T96736 C92SRX 52931998 IC50 = 1510 nM T96736 C5F1IT 52932001 IC50 = 2050 nM T96736 CWFG81 52932003 IC50 = 1680 nM T96736 C65DNB 52932059 IC50 = 1240 nM T96736 C06LVX 53363853 IC50 = 2090 nM T96736 C3QGZ1 53364100 IC50 = 3000 nM T96736 CXYI14 71681394 IC50 = 9200 nM T96736 COBN97 71681395 IC50 = 10000 nM T96736 CR5BQ2 71681396 IC50 = 31000 nM T96736 C6E8TM 71681562 IC50 = 9900 nM T96736 C7ITA6 71681563 IC50 = 27000 nM T96736 C9KP1U 71681564 IC50 = 26000 nM T96736 CE6P5O 71681565 IC50 = 33000 nM T96736 CH4F1V 71681566 IC50 = 33000 nM T96736 CA2GQ5 71681720 IC50 = 35000 nM T96736 CP8UN5 71681721 IC50 = 43000 nM T96736 C6O8VG 71681722 IC50 = 51000 nM T96736 C3WU8P 71681723 IC50 = 67000 nM T96736 CA68PI 71681724 IC50 = 78000 nM T96736 C0TKW7 71682046 IC50 = 1500 nM T96736 CGJ18W 71682047 IC50 = 1600 nM T96736 CGMO97 71682048 IC50 = 2300 nM T96736 C4QA6W 71682049 IC50 = 5600 nM T96736 CY63JH 71682050 IC50 = 6100 nM T96736 C2QH9Y 71682204 IC50 = 8100 nM T96736 CS45BO 71682205 IC50 = 11000 nM T96736 CE87JT 71682206 IC50 = 12000 nM T96736 C5KR2M 71682207 IC50 = 12000 nM T96736 CKG6I5 71682208 IC50 = 26000 nM T96736 C4MDP1 71682354 IC50 = 30000 nM T96736 C1H9AY 71682355 IC50 = 32000 nM T96736 CB9J7C 71682356 IC50 = 32000 nM T96736 C0X4DB 71682357 IC50 = 66000 nM T96736 CPQ8K0 71682358 IC50 = 76000 nM T96736 CM82DF 71682662 IC50 = 21000 nM T96736 C5XR3L 71682663 IC50 = 7400 nM T96736 C96MSZ 71682815 IC50 = 10000 nM T96736 C0IE1G 73349029 IC50 = 4700 nM T96736 D0I3KR 71681561 IC50 = 5300 nM T96736 D0Y9BU 46190808 IC50 = 9800 nM T86808 CL2Q6J 44178077 IC50 > 100000 nM T86808 C0BQC4 44586265 IC50 = 2200 nM T86808 C2IML9 58580486 IC50 = 460 nM T86808 D0K1NM 20541332 IC50 > 100000 nM T55398 D0OB0F 5328940 IC50 = 574 nM T55398 D03LWG 53235510 IC50 > 10000 nM T55398 D07EHV 44814409 IC50 > 10000 nM T55398 D07NUL 118414016 IC50 = 2 nM T55398 D0E3TC 44259 IC50 = 4.21 nM T55398 D0T3ME 156422 IC50 > 30000 nM T55398 CGEW10 1247796 IC50 = 2200 nM T55398 CJ3U9Y 2728161 IC50 = 55000 nM T55398 CF6WI5 2824236 IC50 = 2800 nM T55398 C1KY3I 4455946 IC50 = 12000 nM T55398 CRC65X 9863786 IC50 > 30000 nM T55398 C5UG6X 10114595 Ki = 0.48 nM T55398 C8K9HL 10142476 Ki = 0.42 nM T55398 C4RNU9 10184123 Ki = 0.5 nM T55398 CN37YZ 10207985 Ki = 0.34 nM T55398 C8BHJ3 10226185 Ki = 8.2 nM T55398 C78SMB 10227510 Ki = 2.8 nM T55398 CXN06I 10227557 Ki = 2.8 nM T55398 C0SR5Y 10278151 Ki = 0.7 nM T55398 CBOP58 11293798 Ki > 10000 nM T55398 C26BZX 11362471 Ki > 10000 nM T55398 CWXB93 11397177 Ki > 10000 nM T55398 CTG83F 11539329 Ki > 9900 nM T55398 CACS26 11561968 Ki > 4000 nM T55398 CMIL86 11590363 Ki > 9900 nM T55398 C9T6SC 11640926 Ki > 9900 nM T55398 CU0E8O 11690457 Ki = 1900 nM T55398 CB0AP2 11705863 Ki > 4000 nM T55398 CE2VU0 11987888 Ki = 1.2 nM T55398 CFPW41 16007116 Ki > 9900 nM T55398 CST43D 21899140 Ki = 6.5 nM T55398 CM4F0B 21899142 Ki = 1.3 nM T55398 CT46EH 21899147 IC50 = 8000 nM T55398 C7YG1N 24759534 IC50 = 210 nM T55398 CIN29Y 24801862 IC50 = 400 nM T55398 CZ12SD 24801863 IC50 = 3000 nM T55398 CZJ9P4 24857834 IC50 = 70 nM T55398 C3E5XY 24857850 IC50 = 420 nM T55398 CLZ23U 24951610 IC50 = 1100 nM T55398 C2KY1G 25094210 IC50 = 167 nM T55398 CGT1W6 25144294 IC50 = 56 nM T55398 CU7VR0 25144732 IC50 = 8 nM T55398 C6BWZ8 25145145 IC50 = 1000 nM T55398 CA75YC 25169380 IC50 = 6 nM T55398 CC3BU0 25169381 IC50 = 4 nM T55398 CFB65H 25169382 IC50 = 6 nM T55398 CRXS80 25169384 IC50 = 9 nM T55398 CC71QJ 27666048 IC50 > 100000 nM T55398 CTA08W 41420877 IC50 = 2000 nM T55398 CO6HU7 44178069 IC50 = 1142 nM T55398 C8KNA3 44219632 Ki > 4000 nM T55398 C0VIX4 44219633 Ki = 2300 nM T55398 CZH6G2 44412152 IC50 > 30000 nM T55398 C1OQP6 44412156 IC50 = 1500 nM T55398 CJR94S 44412164 IC50 > 30000 nM T55398 COZ5X9 44412166 IC50 = 25000 nM T55398 CU7Q3F 44412167 IC50 = 4000 nM T55398 CU0T2G 44412174 IC50 = 1000 nM T55398 C0V4FU 44412178 IC50 = 550 nM T55398 CIF5C1 44412201 IC50 = 1000 nM T55398 CCY3L4 44412220 IC50 = 20000 nM T55398 CR7Y9K 44412242 IC50 = 30000 nM T55398 C4UOZ2 44412243 IC50 = 6000 nM T55398 CGJ61S 44412251 Ki = 4500 nM T55398 C18ZMY 44412252 IC50 = 800 nM T55398 CM6X1B 44412253 IC50 = 2000 nM T55398 C6TN3O 44412266 IC50 = 1000 nM T55398 CD2W6N 44412267 IC50 = 2000 nM T55398 CRB74Z 44412281 IC50 = 400 nM T55398 C0R2LO 44412325 IC50 = 30000 nM T55398 CA0MI2 44412326 IC50 = 400 nM T55398 CH7M4G 44412327 IC50 = 1000 nM T55398 C35CLR 44412343 IC50 = 150 nM T55398 C7XE0D 44412352 IC50 = 4000 nM T55398 CUV9B8 44412391 IC50 = 6500 nM T55398 CH6F7D 44412392 IC50 = 2000 nM T55398 CG3LU0 44412407 IC50 = 30000 nM T55398 CZ16BF 44412434 IC50 = 4000 nM T55398 CA48QG 44412435 IC50 = 3000 nM T55398 C20AUC 44412442 IC50 = 500 nM T55398 C6N1MJ 44412480 IC50 = 3000 nM T55398 C6O0TZ 44412492 IC50 = 6500 nM T55398 CRK51G 44448764 IC50 = 39 nM T55398 CKI6S2 44448795 IC50 = 6900 nM T55398 C1HB0N 44448797 IC50 = 313 nM T55398 C7GA2S 44448798 IC50 = 3030 nM T55398 CTGL39 44448828 IC50 = 225 nM T55398 CSAH90 44448865 IC50 = 1300 nM T55398 CDWX21 44448867 IC50 = 914 nM T55398 CXV8T5 44448904 IC50 = 497 nM T55398 C3DP0G 44448905 IC50 = 8100 nM T55398 CAQ4T1 44448906 IC50 = 433 nM T55398 CO7Y6K 44448908 IC50 = 1134 nM T55398 COY50K 44448910 IC50 = 1085 nM T55398 CL28QE 44448912 IC50 = 10 nM T55398 CVQ74G 44448939 IC50 = 49 nM T55398 CIUF03 44448940 IC50 = 1156 nM T55398 C28SLH 44448941 IC50 = 5 nM T55398 C47GQS 44448942 IC50 = 263 nM T55398 CCV97Y 44448943 IC50 = 166 nM T55398 CHCN76 44448970 IC50 = 2 nM T55398 C3YM1B 44448971 IC50 = 63 nM T55398 C4S5TP 44448972 IC50 = 112 nM T55398 CV5F0Q 44448973 IC50 = 7 nM T55398 CX8PM6 44448975 IC50 = 3 nM T55398 CH61MQ 44449000 IC50 = 8 nM T55398 C3C2TM 44449002 IC50 = 181 nM T55398 CT3B1M 44449003 IC50 = 208 nM T55398 CE07NB 44449025 IC50 = 15 nM T55398 C5X0LI 44449050 IC50 = 1 nM T55398 CZ3V1X 44449078 IC50 = 35 nM T55398 C0SQE3 44449102 IC50 = 216 nM T55398 CK6E5J 44449122 IC50 = 95 nM T55398 CT7U9G 44449126 IC50 = 7 nM T55398 C37YOA 44449160 IC50 = 487 nM T55398 CXL76B 44449162 IC50 = 535 nM T55398 CSRC92 44449189 IC50 = 1880 nM T55398 CQ5I9D 44449190 IC50 = 126 nM T55398 C3DU4B 44449218 IC50 = 19 nM T55398 C64YUV 44449221 IC50 = 545 nM T55398 C1G4DC 44449335 IC50 = 710 nM T55398 C0CR1V 44449336 IC50 = 660 nM T55398 C1W9XR 44449364 IC50 = 1600 nM T55398 CMC7U0 44449365 IC50 > 10000 nM T55398 C2DCP7 44449366 IC50 > 10000 nM T55398 CP6R3S 44449367 IC50 > 10000 nM T55398 C6IHR2 44449391 IC50 = 3400 nM T55398 CJ68ZB 44449392 IC50 = 160 nM T55398 CZJ8U5 44449393 IC50 = 350 nM T55398 CZYR60 44449394 IC50 = 1200 nM T55398 C2SO6L 44449424 IC50 > 10000 nM T55398 CEGF72 44449425 IC50 > 10000 nM T55398 CBA80K 44449426 IC50 = 700 nM T55398 CUY8W6 44449427 IC50 = 2800 nM T55398 CRWG12 44449486 IC50 = 2400 nM T55398 CF0V1N 44449548 IC50 = 3700 nM T55398 C24SWN 44449549 IC50 = 8900 nM T55398 CD6XC0 44449584 IC50 = 4800 nM T55398 C9TR0X 44449617 IC50 = 1000 nM T55398 C3V7EY 44449647 IC50 = 800 nM T55398 CWB60J 44449650 IC50 > 10000 nM T55398 C6DHC9 44450171 IC50 = 7300 nM T55398 C3DQJ6 44450195 IC50 = 7200 nM T55398 CYH6P3 44520205 IC50 = 340 nM T55398 COV31Z 44586245 IC50 = 200 nM T55398 CE3V0Z 44586278 IC50 = 1189 nM T55398 CC5W9J 44586319 IC50 = 456 nM T55398 C8WPI5 44586320 IC50 = 1934 nM T55398 CZI08B 46175395 IC50 = 170 nM T55398 C35UQP 46175482 IC50 = 240 nM T55398 CF0OV6 46175578 IC50 = 1060 nM T55398 CRC37F 46176531 IC50 > 20000 nM T55398 CY3HW5 46224684 IC50 > 10000 nM T55398 COTJ39 46863083 IC50 = 1100 nM T55398 CLS29B 46872626 IC50 > 10000 nM T55398 C1Q8AW 49824621 Ki = 38.5 nM T55398 CAZQ43 51003133 IC50 = 380 nM T55398 CC24GM 52913874 IC50 = 21 nM T55398 CXA03W 52920796 IC50 = 640 nM T55398 CEQN27 52936621 Ki > 1000 nM T55398 C6OTY5 53251320 IC50 = 26000 nM T55398 CE8OY2 53317913 IC50 = 8 nM T55398 C0SWH5 53348216 IC50 > 40000 nM T55398 C8ZRE3 53356518 IC50 > 50000 nM T55398 C8NA4L 53384644 IC50 > 30000 nM T55398 C1XS2J 54760383 IC50 > 10000 nM T55398 C5KR6N 56595558 Ki = 43 nM T55398 COI9U2 56595687 Ki = 420 nM T55398 C2AM6B 56595688 Ki = 1200 nM T55398 CFY2I4 56595689 Ki = 160 nM T55398 CAM8E1 56595690 Ki = 440 nM T55398 CN5EV7 56595691 Ki = 36 nM T55398 C6ET0W 56595693 Ki = 78 nM T55398 CTR10F 56658543 Ki = 340 nM T55398 C9MJG4 56929824 IC50 = 430 nM T55398 C0UDY9 57401151 IC50 = 7500 nM T55398 COY07J 57519810 IC50 <= 5000 nM T55398 C0PA3D 57519811 Ki = 50 nM T55398 CO75VX 58056108 Ki = 1.7 nM T55398 CSN35V 58056134 Ki = 790 nM T55398 C8CG6L 58056265 Ki = 52 nM T55398 CVQ2U4 58056270 Ki = 610 nM T55398 C8GFI0 58056341 Ki = 2 nM T55398 C9MIL7 58450666 IC50 = 1800 nM T55398 C9HUB2 58570982 IC50 = 240 nM T55398 C6BPR2 58985201 IC50 > 30000 nM T55398 CT3EW2 59292007 IC50 > 1000 nM T55398 CP9A8T 59503659 IC50 = 1219 nM T55398 C1MA6J 59503711 IC50 = 1423 nM T55398 CX29EU 59503744 IC50 = 873 nM T55398 CXJ63M 59603829 IC50 = 64 nM T55398 CQEU96 59603842 IC50 = 23 nM T55398 COH62U 60097413 IC50 > 10000 nM T55398 C1MR8Q 60097495 IC50 > 10000 nM T55398 CK6WO0 66552478 IC50 < 10000 nM T55398 CUF20T 66554581 IC50 = 80 nM T55398 CZ92KC 66554752 IC50 = 2100 nM T55398 CF7RQ2 66554923 IC50 = 280 nM T55398 CMS6L3 66554926 IC50 = 180 nM T55398 CU1DM5 66555095 IC50 = 220 nM T55398 CVQW04 66555265 IC50 = 59 nM T55398 C53YWX 66555955 IC50 = 99 nM T55398 CSL0F3 66555956 IC50 = 170 nM T55398 COS5Q9 66555957 IC50 = 44 nM T55398 C7N3DE 66557142 IC50 < 100 nM T55398 C08DXU 66557143 IC50 < 100 nM T55398 COU2C4 66664636 Ki = 8 nM T55398 CV63UL 67240318 IC50 > 10000 nM T55398 C80HMA 68115414 IC50 = 1500 nM T55398 CW23JE 68241353 IC50 = 470 nM T55398 CK9E0Y 68327832 IC50 = 7 nM T55398 CU26SP 68327847 IC50 = 150 nM T55398 CPG75C 68327866 IC50 = 85 nM T55398 CE41YS 68327879 IC50 = 180 nM T55398 CA47UH 68328137 IC50 = 410 nM T55398 C5Z7QJ 68328146 IC50 = 2400 nM T55398 C8OAS6 68328387 IC50 = 27 nM T55398 C3QE9V 68328415 IC50 = 390 nM T55398 CI4HV8 68328491 IC50 = 2 nM T55398 C9HZG1 68328492 IC50 = 40 nM T55398 CC6F8D 68328504 IC50 = 47 nM T55398 C43RXO 68328520 IC50 = 310 nM T55398 CB2OM0 68328789 IC50 = 61 nM T55398 CRM6L5 68357884 IC50 = 5 nM T55398 CZG9X7 68357894 IC50 = 13 nM T55398 C2B1TC 68357902 IC50 = 370 nM T55398 CYI75G 68678653 IC50 = 24400 nM T55398 C5DGR9 69036886 IC50 = 10000 nM T55398 CV0QP3 70947961 Ki = 11 nM T55398 CKT60L 71455860 Ki > 9900 nM T55398 C6T1LM 71506869 IC50 < 50 nM T55398 CE5XR2 71612615 IC50 = 1.8 nM T55398 C5RZ7I 72709739 IC50 = 100 nM T55398 CV3I1N 72943654 IC50 < 100 nM T55398 CIT2V7 72945768 IC50 = 100 nM T55398 CX1UE8 72945946 IC50 = 100 nM T55398 CM94EG 72945952 IC50 > 30000 nM T55398 CZNM96 73053607 IC50 < 100 nM T55398 C25UCH 73053622 IC50 < 100 nM T55398 C1RO3T 73053624 IC50 < 100 nM T55398 CX75YR 73352604 IC50 = 3.981 nM T55398 C8JTD0 73442848 IC50 = 138 nM T55398 CE5CX0 73442898 IC50 = 300 nM T55398 COU3K5 73669498 IC50 = 113 nM T55398 CS2QC6 73669499 IC50 = 204 nM T55398 C7LER5 73669500 IC50 = 3452 nM T55398 C5C4SU 73669664 IC50 = 1140 nM T55398 CF0C4R 73669837 IC50 = 42000 nM T55398 CYO3D1 73669840 IC50 = 2570 nM T55398 C0FH9Y 73670011 IC50 = 1000 nM T55398 C5WLK7 73670169 IC50 = 410 nM T55398 CTG6S3 73670172 IC50 = 333000 nM T55398 C40BHZ 73670173 IC50 = 228000 nM T55398 CJKB83 73670174 IC50 = 11 nM T55398 CF42WG 73670176 IC50 = 4700 nM T55398 C62MPO 73670344 IC50 = 1081000 nM T55398 CW1VG7 73670345 IC50 = 3012000 nM T55398 CJF7Y5 73670346 IC50 = 104 nM T55398 CZU1A0 73670347 IC50 = 24 nM T55398 CCUH57 73670348 IC50 = 16 nM T55398 C82COK 73670350 IC50 = 18 nM T55398 CD23NU 73670513 IC50 = 6000 nM T55398 C1LPW5 73670673 IC50 = 1000 nM T55398 CLO61M 73670847 IC50 = 89 nM T55398 C6T4WZ 73670848 IC50 = 94 nM T55398 CF7TD8 73670850 IC50 = 530 nM T55398 CT3L4F 73670851 IC50 = 932 nM T55398 CN4B8K 75202037 IC50 = 1.5 nM T55398 CFL54M 75204288 IC50 = 1.8 nM T55398 CYJ4C6 76955703 IC50 < 100 nM T55398 CSH9R0 77847460 IC50 < 100 nM T55398 CQ2SU8 78673832 IC50 > 30000 nM T55398 CE0W9R 78673833 IC50 > 30000 nM T55398 C1HW4B 89735655 IC50 = 3000 nM T55398 C89YHN 90134560 IC50 = 5.3 nM T55398 C2CY5A 90154381 IC50 = 3.6 nM T55398 CGTN69 90154630 IC50 = 1.9 nM T55398 C5S0DF 90154917 IC50 = 3.5 nM T55398 CZTM62 90155093 IC50 = 5.6 nM T55398 CAL0O9 90155375 IC50 = 13 nM T55398 CI5GF8 90155577 IC50 = 300 nM T55398 CSC20O 90271946 IC50 = 20 nM T55398 CWA46G 90271957 IC50 < 100 nM T55398 CC1S2P 90272141 IC50 = 71 nM T55398 CM2LJ5 90275527 IC50 = 2400 nM T55398 CNX5V4 91844450 IC50 = 1193000 nM T55398 C0Y8ZK 91933875 IC50 > 1000 nM T55398 CA1K0F 91938073 IC50 = 1.3 nM T55398 CAU45T 91971978 IC50 > 30000 nM T55398 C0YSX8 117826679 IC50 = 4300 nM T55398 CWA8X7 117871492 IC50 = 2197 nM T55398 CI40BM 117871555 IC50 = 3649 nM T55398 CU1V7Y 117871558 IC50 = 187 nM T55398 CQ6E2O 117871721 IC50 > 20000 nM T55398 CTS35E 117871724 IC50 = 3452 nM T55398 CE7X1L 117871750 IC50 = 212 nM T55398 C6MG7L 117871760 IC50 = 730 nM T55398 C0A4XC 117871929 IC50 = 74 nM T55398 CV4B2W 117871992 IC50 = 307 nM T55398 CY60JR 117872182 IC50 = 401 nM T55398 C3VJ0I 117872205 IC50 = 542 nM T55398 CY5JF0 117872250 IC50 = 187 nM T55398 COIM28 117872315 IC50 = 190 nM T55398 C7PM6F 117872316 IC50 = 1100 nM T55398 C63OVX 117872321 IC50 = 653 nM T55398 CT4AZ2 117872334 IC50 = 1100 nM T55398 C6X8VS 117872368 IC50 = 191 nM T55398 CR0JN8 117872469 IC50 = 128 nM T55398 CBOI97 117872492 IC50 = 478 nM T55398 CO6BH7 117872621 IC50 = 1449 nM T55398 CD8J9G 117872890 IC50 = 1605 nM T55398 CQ5S7L 117872990 IC50 = 285 nM T55398 CD6EA9 117873013 IC50 = 2677 nM T55398 C9OA4U 117873033 IC50 = 101 nM T55398 CL6QV4 117873045 IC50 = 261 nM T55398 CDO5I6 117873092 IC50 = 106 nM T55398 CP89EY 117873164 IC50 = 2 nM T55398 C8QB3S 117873179 IC50 = 1582 nM T55398 CWG60S 117873194 IC50 = 2725 nM T55398 CT3B6F 117873210 IC50 = 683 nM T55398 C08YAE 117885624 IC50 = 12 nM T55398 C2V1RC 117885639 IC50 = 830 nM T55398 CS9J3N 117885675 IC50 = 155 nM T55398 CJ8I7U 117885678 IC50 = 12 nM T55398 CK1A0N 117885680 IC50 = 11900 nM T55398 CYP9O7 117885688 IC50 = 12 nM T55398 C4ECT8 117885692 IC50 = 2107 nM T55398 CYN4S1 117885705 IC50 = 3 nM T55398 C2ABD1 117885712 IC50 = 852 nM T55398 CF6UT1 117885715 IC50 = 373 nM T55398 C3VN9K 117885730 IC50 = 7 nM T55398 CZ8P4J 117885751 IC50 = 4 nM T55398 C9R3WU 117885753 IC50 = 6008 nM T55398 C1HND8 117885755 IC50 = 9510 nM T55398 CS72RV 117885758 IC50 = 216 nM T55398 C6Z3NJ 117885766 IC50 = 44 nM T55398 CKU6S4 117885912 IC50 = 8 nM T55398 C1E2DK 118072831 IC50 < 100 nM T55398 C1ZR5E 118173110 IC50 = 33 nM T55398 CV5Q9X 118388894 IC50 = 4381 nM T55398 CT9RU4 118413945 IC50 = 1.3 nM T55398 C36CUE 118414094 IC50 = 0.5 nM T55398 C69QWZ 118414114 IC50 = 29.5 nM T55398 C7J6RO 118414128 IC50 = 4.8 nM T55398 CLWJ18 118414336 IC50 = 7.6 nM T55398 CSQV50 118414357 IC50 = 840 nM T55398 CUJ9O2 118414389 IC50 = 0.1 nM T55398 CF2D3K 118414391 IC50 = 2836 nM T55398 C5XRA6 118414397 IC50 = 23.9 nM T55398 CHL38K 118414437 IC50 = 5.9 nM T55398 CFM20Z 118414536 IC50 = 0.3 nM T55398 CW3IC5 118414671 IC50 = 4.6 nM T55398 C3N5SA 118414693 IC50 = 12.1 nM T55398 CIH2O7 118414733 IC50 = 3.7 nM T55398 C51HAN 118414780 IC50 = 2.7 nM T55398 C0O3SN 118424414 IC50 = 2.4 nM T55398 CUN8Y5 118424424 IC50 = 0.6 nM T55398 COH1T4 118453721 IC50 = 6 nM T55398 CR7DJ0 118453722 IC50 = 55 nM T55398 CK1Z7I 118462026 IC50 = 4 nM T55398 COB6M3 118475320 IC50 = 2 nM T55398 CX2GE1 118475349 IC50 = 250 nM T55398 CZBA29 118641364 IC50 <= 100 nM T55398 CX58DI 118716791 IC50 > 30000 nM T55398 CD9X2B 118716796 IC50 > 30000 nM T55398 C2YJ0O 118716797 IC50 > 30000 nM T55398 CL3UO9 118716798 IC50 > 30000 nM T55398 C71BAM 118716799 IC50 > 30000 nM T55398 CU4EL6 118716806 IC50 > 30000 nM T55398 C5FK7T 118719435 IC50 = 0.36 nM T55398 CA2NJ8 118719437 IC50 = 0.24 nM T55398 CEFG28 118719438 IC50 = 2.8 nM T55398 CL1N2T 118719440 IC50 = 0.32 nM T55398 CCJ0X7 118719442 IC50 = 2.6 nM T55398 CJ2IZ0 118719443 IC50 = 2.2 nM T55398 CIV1H2 118719446 IC50 <= 100 nM T55398 CHT6K9 118728811 Ki > 4000 nM T55398 CUA3Y2 118728812 Ki > 4000 nM T55398 CDQ78G 118728813 Ki > 4000 nM T55398 CZ6XL7 118728814 Ki > 4000 nM T55398 CMO67K 118728815 Ki > 4000 nM T55398 CR2M0Q 118728816 Ki > 4000 nM T55398 C62SCL 118728817 Ki > 4000 nM T55398 CSB30C 118728819 Ki > 4000 nM T55398 CV7XU8 118728820 Ki = 2700 nM T55398 C3J1EX 118728821 Ki > 4000 nM T55398 CIWB78 118728822 Ki > 4000 nM T55398 CP18SE 118728823 Ki = 3300 nM T55398 CM42CA 118728824 Ki > 4000 nM T55398 C9Q7CL 118728825 Ki > 4000 nM T55398 CCR3S0 118728826 Ki > 4000 nM T55398 CNJK97 118729800 IC50 > 20000 nM T55398 C14CYV 118729801 IC50 = 5190 nM T55398 CNP64R 118729802 IC50 > 20000 nM T55398 CP3U7F 118729803 IC50 = 6850 nM T55398 CQ4Z2H 118729804 IC50 > 20000 nM T55398 CQ92UP 118729805 IC50 > 20000 nM T55398 CX9BS1 118729806 IC50 > 20000 nM T55398 C7WFP3 118729807 IC50 > 20000 nM T55398 C3MUB5 118729808 IC50 > 20000 nM T55398 CHDF03 118729809 IC50 > 20000 nM T55398 C6AW4N 118729810 IC50 > 20000 nM T55398 CBWY74 118729811 IC50 = 1140 nM T55398 CN1KS6 118729812 IC50 > 20000 nM T55398 C36BLM 118729813 IC50 = 403000 nM T55398 C4R1EI 121254788 IC50 = 10 nM T55398 C0XU9Y 121255032 IC50 = 7400 nM T55398 CNQ6Z2 121255052 IC50 = 16 nM T55398 CS64MC 121255054 IC50 = 300 nM T55398 CM1W3K 121255069 IC50 = 16 nM T55398 CYDF91 121255074 IC50 = 9 nM T55398 CDQ48W 121255075 IC50 = 19 nM T55398 CZTX30 121256083 IC50 = 12 nM T55398 CJY83B 121258892 IC50 = 17 nM T55398 CTPB07 121262387 IC50 = 32 nM T55398 CUL6H1 121262551 IC50 = 35 nM T55398 C7X1BQ 121493987 IC50 = 38 nM T55398 C30ILY 122180370 IC50 = 690 nM T55398 CK6YL8 122181591 IC50 = 110 nM T55398 CZFT46 122181592 IC50 = 150 nM T55398 COJ93A 122181593 IC50 = 9200 nM T55398 C3EN9U 122181594 IC50 = 2 nM T55398 CWL8R2 122181623 IC50 = 95 nM T55398 CJD5F2 122181624 IC50 = 20 nM T55398 C8C5TR 122181625 IC50 = 8 nM T55398 CT2BY5 122181626 IC50 = 0.3 nM T55398 CYEG26 122181627 IC50 = 14 nM T55398 C06BWF 122181628 IC50 = 6 nM T55398 CEN5P0 122181629 IC50 = 0.8 nM T55398 C6W4PS 122181630 IC50 = 0.3 nM T55398 C1Z0EK 122181631 IC50 = 0.2 nM T55398 CY4HG7 122181632 IC50 = 2 nM T55398 CW74UE 122181633 IC50 = 6 nM T55398 CV87TR 122181634 IC50 = 62 nM T55398 C92TUX 122181635 IC50 = 160 nM T55398 CSD5U0 122181636 IC50 = 480 nM T55398 CC3FS4 122181637 IC50 = 21 nM T55398 CD83YT 122181638 IC50 = 4 nM T55398 CVQ7H5 122181639 IC50 = 10 nM T55398 CTD2I5 122181640 IC50 = 1 nM T55398 CKJU62 122181641 IC50 = 23 nM T55398 CMQ2R0 122181642 IC50 = 13 nM T55398 C4WZR2 122181643 IC50 = 3 nM T55398 CF2LI0 122181644 IC50 = 3 nM T55398 CMZ95X 122181645 IC50 = 1 nM T55398 CFU63N 122181674 IC50 = 0.5 nM T55398 CF7OC2 122181675 IC50 = 0.5 nM T55398 C76RQM 122181676 IC50 = 6 nM T55398 C8D3JG 122184715 IC50 = 11 nM T55398 C0BLW3 122184716 IC50 = 647 nM T55398 CAQ71B 122191866 IC50 = 470 nM T55398 CO6S2E 122196062 IC50 = 40 nM T55398 C8R7FJ 122196063 IC50 = 5 nM T55398 CJA40H 122196064 IC50 = 1 nM T55398 CV85FQ 122196065 IC50 = 10 nM T55398 CBW67H 122196066 IC50 = 1 nM T55398 C7W5QA 122196067 IC50 = 0.2 nM T55398 CS6AP9 122196068 IC50 = 38 nM T55398 CJO8V9 122196168 IC50 = 3 nM T55398 CVI2P6 122196169 IC50 < 0.5 nM T55398 CO72HB 122196170 IC50 = 2 nM T55398 CA6BO3 122196171 IC50 = 1 nM T55398 CU2XL4 122196172 IC50 = 0.8 nM T55398 CZ3W8X 122196173 IC50 < 0.5 nM T55398 CB21TD 122196174 IC50 = 24 nM T55398 C51YFU 122196175 IC50 = 0.9 nM T55398 CX07CU 122196176 IC50 = 0.4 nM T55398 C2HLK9 122196177 IC50 = 0.2 nM T55398 C84DQM 122196178 IC50 = 0.7 nM T55398 C0DO3U 122196179 IC50 < 0.5 nM T55398 CYMK98 122196180 IC50 = 1 nM T55398 CQ1OM7 122196181 IC50 = 1 nM T55398 CLFH30 122196246 IC50 = 7 nM T55398 C5Z2FM 122196247 IC50 = 25 nM T55398 CTX0M5 122196248 IC50 = 12 nM T55398 C43LHP 122196249 IC50 = 0.4 nM T55398 C6QZE1 123917405 IC50 = 2400 nM T55398 CZEV34 125479776 IC50 = 1200 nM T55398 CR3A1O 125495464 IC50 = 15 nM T55398 CGU28T 126573669 IC50 = 121 nM T55398 C2T8ZA 126573681 IC50 = 146 nM T55398 C4S5LR 126622195 IC50 = 0.2 nM T55398 CH4C5O 126961337 IC50 = 58 nM T55398 CAGL14 126970816 IC50 = 71.9 nM T55398 C31ZLG 127034634 Ki = 7.8 nM T55398 CX3YO4 127034635 Ki = 11 nM T55398 CUS38N 127034643 IC50 = 150 nM T55398 C1C4UV 127034834 Ki = 3.8 nM T55398 CZ7H8F 127035289 Ki = 1.6 nM T55398 CZD87E 127037084 IC50 = 465 nM T55398 CB9Z0V 127038973 IC50 = 234 nM T55398 C1KH4L 129284027 Ki = 30 nM T55398 C6RGX5 129284078 Ki = 2.1 nM T55398 C9VL8H 129284112 Ki = 7.4 nM T55398 CWF79O 129284190 Ki = 14 nM T55398 CBJ6X9 129284195 IC50 = 0.38 nM T55398 C3VK4I 129284254 Ki = 7.3 nM T55398 C4VS8P 129284274 Ki = 35 nM T55398 CK2IL4 129284334 IC50 = 0.19 nM T55398 C96LDG 129284345 Ki = 5.1 nM T55398 CN8WZ2 129284370 Ki = 80 nM T55398 C8VNP1 129284385 IC50 = 7.2 nM T55398 CWA5R2 129284395 Ki = 6.6 nM T55398 CR2YV6 129284442 IC50 = 3.6 nM T55398 C4MG6I 129284483 Ki = 1.1 nM T55398 C9W4CS 129284507 Ki = 6.1 nM T55398 CR94JT 129284517 Ki = 3.5 nM T55398 CF19RT 129284574 Ki = 15 nM T55398 CM2J9U 129284575 Ki = 13 nM T55398 C49BMA 129284616 Ki = 6.1 nM T55398 CO4QV7 129284658 Ki = 1.5 nM T55398 C43SGU 129284679 Ki = 31 nM T55398 CS71NJ 129284701 Ki = 34 nM T55398 CV25CZ 129284859 Ki = 3.2 nM T55398 CM23FX 129297015 Ki = 12 nM T55398 CQO83S 129297033 Ki = 10 nM T55398 C0Z5NP 129297518 Ki = 5.8 nM T55398 C2FU6N 129297531 IC50 = 1.2 nM T55398 CFSC56 129297811 Ki = 3.2 nM T55398 C4NG3W 129298165 IC50 = 0.16 nM T55398 CUOX69 129298210 IC50 = 0.081 nM T55398 CTA06R 129298213 IC50 = 0.32 nM T55398 C96KMC 129298275 Ki = 6.5 nM T55398 C8MXQ4 130274633 IC50 = 7 nM T55398 CK4N0V 130274681 IC50 = 122 nM T55398 C45OHZ 130275697 IC50 = 3 nM T55398 C18QMF 130275783 IC50 = 3 nM T55398 C3WG8E 130276452 IC50 = 8 nM T55398 C9WK5I 130276470 IC50 = 17 nM T55398 CXTZ19 131704459 IC50 = 10 nM T55398 C25WQI 131704460 IC50 > 10000 nM T55398 CY70JL 131839618 IC50 = 6 nM T55398 C4Z5MQ 131839619 IC50 = 5 nM T55398 C2W8TC 131839620 IC50 = 42 nM T55398 C0M7PT 131839621 IC50 = 2 nM T55398 CNF79T 133107904 IC50 = 4 nM T55398 CB0C4Y 133107905 IC50 = 69 nM T55398 CJ43BV 133107906 IC50 = 21.38 nM T55398 C2AN7T 134611886 IC50 > 100000 nM T55398 CY4D8I 135566504 Ki > 1000 nM T55398 C7PJ6X 135566704 IC50 > 30000 nM T55398 C6DP4U 135567024 IC50 = 25 nM T55398 CX3UR8 135567025 IC50 = 19 nM T55398 CPV59N 135685787 Ki = 1500 nM T55398 CG3UZ1 135927974 Ki > 1000 nM T55398 CF1PS8 135934877 Ki = 690 nM T55398 CTRL59 135976660 Ki = 1100 nM T55398 CU0SZ4 136074298 IC50 < 100 nM T55398 CDMS84 136074299 IC50 < 100 nM T55398 CSOR07 136074300 IC50 = 14 nM T55398 CQ84IZ 136180335 Ki > 4000 nM T55398 COLR97 136272332 IC50 = 1487 nM T55398 CS9Z2N 136272346 IC50 = 1688 nM T55398 CX48MU 136272376 IC50 = 11 nM T55398 CYUF15 136272377 IC50 = 78 nM T55398 CL6S3R 136272378 IC50 = 43 nM T55398 C6T7AE 136272379 IC50 = 135 nM T55398 C7Y1QZ 136272387 IC50 = 43 nM T55398 C2V7QH 136272388 IC50 = 27 nM T55398 CN49DR 136272389 IC50 = 490 nM T55398 C7XY1B 136272390 IC50 = 67 nM T55398 COQ3V4 136504460 IC50 = 972 nM T55398 CVPE08 136504461 IC50 = 2429 nM T55398 CB0M7Z 136504482 IC50 = 454 nM T55398 C7ZF1S 136508720 IC50 = 79 nM T55398 CY1Q8P 136508752 IC50 = 85 nM T55398 C5K8ED 136932639 IC50 = 565 nM T55398 C9DF2X 136932640 IC50 = 580 nM T55398 C9IS5M 136983815 IC50 = 121 nM T55398 C9V3KL 136983853 IC50 = 258 nM T55398 CHT7X2 136983871 IC50 = 352 nM T55398 C24BNM 136983876 IC50 = 635 nM T55398 C39FNY 136983894 IC50 = 36 nM T55398 CWL74T 136983918 IC50 = 354 nM T55398 CSJI86 136983949 IC50 = 620 nM T55398 C3R0PB 136984063 IC50 = 450 nM T55398 C5KN9F 136984064 IC50 = 100 nM T55398 CH3M4B 137083628 IC50 > 30000 nM T55398 CJA07O 137083629 IC50 > 30000 nM T55398 C9F8PX 137083630 IC50 = 579 nM T55398 C96CJQ 137348875 IC50 = 360 nM T55398 C8GD6Y 137367179 IC50 = 0.47 nM T55398 CT2FE0 137367190 IC50 = 0.11 nM T55398 C52UFH 137367200 Ki = 210 nM T55398 C3PBN7 137367378 IC50 = 0.026 nM T55398 CZ4VW3 137631374 IC50 = 21 nM T55398 C0U4AO 137631449 IC50 = 10 nM T55398 CN32XA 137631833 IC50 = 82 nM T55398 C90ELI 137631990 IC50 = 730 nM T55398 CSVD52 137632007 IC50 = 20 nM T55398 C0OWI4 137632095 IC50 = 3 nM T55398 CQU8G7 137632864 IC50 = 33 nM T55398 CZH08K 137633516 IC50 = 180 nM T55398 CC9IU4 137634304 IC50 = 5 nM T55398 CYEO71 137634466 IC50 = 5 nM T55398 CQR3H5 137634670 IC50 = 140 nM T55398 CXG74K 137635345 IC50 = 50 nM T55398 CY6TH8 137635761 IC50 = 4.571 nM T55398 CJE35M 137636090 IC50 = 20 nM T55398 C8Z9VW 137637011 IC50 = 3 nM T55398 C1KWC2 137637354 IC50 = 99 nM T55398 CPEI56 137637758 IC50 = 16 nM T55398 CE8AB3 137639678 IC50 = 400 nM T55398 CB6GD5 137639959 IC50 = 47 nM T55398 CB0JI5 137640711 IC50 = 2000 nM T55398 CO1MS6 137641896 IC50 = 14600 nM T55398 CY9QE7 137642189 IC50 = 4.786 nM T55398 CA9DE5 137642519 IC50 = 390 nM T55398 CP6K0U 137642747 IC50 = 120 nM T55398 C47KFJ 137642928 IC50 = 4 nM T55398 C1BK8H 137643835 IC50 = 9 nM T55398 CBA59R 137644862 IC50 = 1300 nM T55398 CP74MV 137644945 IC50 = 75 nM T55398 C7KHW3 137645090 IC50 = 410 nM T55398 CXIN67 137645231 IC50 = 58 nM T55398 C0GYU1 137646905 IC50 = 8 nM T55398 CGU2E5 137648767 IC50 = 840 nM T55398 CQHO93 137649163 IC50 = 3 nM T55398 CBY15N 137649190 IC50 = 56 nM T55398 CX8N6D 137650526 IC50 = 13 nM T55398 C98RIA 137651604 IC50 = 270 nM T55398 C0RUL8 137651621 IC50 = 10 nM T55398 CFX6Y3 137651671 IC50 = 13 nM T55398 C5NUY0 137651713 IC50 = 25 nM T55398 C7BJN4 137652293 IC50 = 170 nM T55398 C5CKI4 137652730 IC50 = 64 nM T55398 CAFG38 137653032 IC50 = 630.96 nM T55398 C8UGS4 137653281 IC50 = 50 nM T55398 CQT9B3 137653599 IC50 = 13 nM T55398 CS6RE8 137654629 IC50 = 50 nM T55398 CNIX25 137655529 IC50 = 1600 nM T55398 C27SVK 137656133 IC50 = 11 nM T55398 CR8Z9G 137656476 IC50 = 2087 nM T55398 CQ0GX8 137657147 IC50 = 40 nM T55398 CLW29O 137657406 IC50 = 9000 nM T55398 C49DOZ 137657630 IC50 = 19 nM T55398 CXS2U8 137658175 IC50 = 34 nM T55398 CO6XD2 137658443 IC50 = 22 nM T55398 CU0ST8 137659008 IC50 = 130 nM T55398 C6Z8YN 137659188 IC50 = 70 nM T55398 CB1XR5 137659870 IC50 = 4 nM T55398 CMZ36T 137659999 IC50 = 730 nM T55398 CK1B4W 137660846 IC50 = 6 nM T55398 CM23OE 137661767 IC50 = 44 nM T55398 CJ0G3C 138376590 Ki = 1.8 nM T55398 CX64WE 138620530 IC50 < 30 nM T55398 C2LHE0 138620547 IC50 < 30 nM T55398 CA63ML 138620560 IC50 < 30 nM T55398 CR0Y8I 138656676 IC50 < 30 nM T55398 CA1I4Y 138656977 IC50 < 30 nM T55398 C72APW 138727769 IC50 = 97.72 nM T55398 C5J2WV 138728749 IC50 = 94 nM T55398 CVU63L 139582016 IC50 = 37 nM T55398 C8PH9S 139582017 IC50 = 4 nM T55398 C45PVO 142501440 Ki = 22 nM T55398 CU12BZ 142501542 IC50 = 0.1 nM T55398 CV1KM9 145979754 IC50 = 77.62 nM T55398 CX05ZN 145979845 IC50 = 22 nM T55398 CY9X5Q 145979885 IC50 = 1190 nM T55398 C9N2XW 145980788 IC50 = 19.5 nM T55398 CNQ67H 145987089 IC50 = 207 nM T55398 C1N9LZ 145987466 IC50 = 446 nM T55398 C9O6WH 145987619 IC50 = 1530 nM T55398 C4QX5P 145987677 IC50 = 44.67 nM T55398 CYS4V9 145990152 IC50 = 234.42 nM T55398 C3T6XI 145991666 IC50 = 1770 nM T55398 CEL5Y6 145991871 IC50 = 738 nM T55398 CP15XW 145992518 IC50 = 33 nM T55398 CSHF19 145992913 IC50 = 602.56 nM T55398 C1N8CA 145993210 IC50 = 671 nM T55398 C12VLN 145993338 IC50 = 87.1 nM T55398 CE9PV2 145993467 IC50 > 10000 nM T55398 CT74QG 145993512 IC50 = 4073.8 nM T55398 C2B4VW 145993656 IC50 = 42 nM T55398 C5H2WU 145993757 IC50 = 16 nM T55398 CHT23F 145993921 IC50 = 804 nM T55398 C6PK4L 146483027 IC50 = 0.078 nM T55398 CMZ4J3 155510495 IC50 < 30 nM T55398 CHX57D 155511560 Ki = 95 nM T55398 CKB64L 155512869 IC50 = 69 nM T55398 C2MD1Q 155513187 IC50 > 10000 nM T55398 C93SNT 155514207 IC50 = 1 nM T55398 C17BHJ 155516763 IC50 = 0.022 nM T55398 C08VAM 155517957 IC50 = 2.5 nM T55398 C8UI7G 155520013 IC50 = 0.29 nM T55398 CCL0S9 155520435 IC50 = 0.099 nM T55398 C7YSD8 155522882 IC50 > 5000 nM T55398 C70GEI 155525183 IC50 > 5000 nM T55398 CWP05R 155527255 Ki = 1.7 nM T55398 CE2YX6 155527737 Ki = 290 nM T55398 CSGV07 155529499 Ki > 8400 nM T55398 CA83QP 155529897 IC50 > 5000 nM T55398 CGDE18 155530136 IC50 > 5000 nM T55398 CSJB85 155530835 Ki = 0.5 nM T55398 CWU8N1 155535119 IC50 = 38 nM T55398 CL5F3C 155537218 Ki = 0.5 nM T55398 CG4LQ2 155539650 Ki = 1.2 nM T55398 C29FDV 155542370 IC50 = 9 nM T55398 C8NOD0 155544794 Ki > 30000 nM T55398 CX9FM8 155548286 IC50 = 2.1 nM T55398 CSJ72Y 155549539 IC50 = 6 nM T55398 CR79JM 155549965 IC50 = 1 nM T55398 CN6O2U 155552158 IC50 > 5000 nM T55398 CM8O9G 155552851 Ki = 170 nM T55398 CWO25P 155555362 Ki = 26 nM T55398 C4Y6BV 155556454 Ki = 6.7 nM T55398 C0WUZ4 155556888 IC50 = 5 nM T55398 C8NMG3 155558108 IC50 > 5000 nM T55398 CWJ08R 155560232 Ki = 0.8 nM T55398 C4IP2Y 155561648 IC50 = 17 nM T55398 C0EBX7 155561943 IC50 = 279 nM T55398 C3D2GP 155562155 IC50 = 21 nM T55398 D00ERW 44444843 Ki > 9921 nM T55398 D00HVA 11624601 Ki > 9900 nM T55398 D02JIL 3572750 IC50 = 4000 nM T55398 D04CFM 86343751 Ki = 1 nM T55398 D04ZIV 58056241 IC50 = 1 nM T55398 D06HVH 54613583 IC50 > 10000 nM T55398 D06WGX 9549184 IC50 > 25000 nM T55398 D09JUD 44449334 IC50 = 20 nM T55398 D0I2FZ 11983295 IC50 = 200 nM T55398 D0J3LR 11634725 Ki > 4000 nM T55398 D0J8VR 25169383 IC50 = 1 nM T55398 D0LY5S 2635761 IC50 = 13600 nM T55398 D0ME9B 46868971 IC50 = 1800 nM T55398 D0Q3NG 11715520 Ki > 9900 nM T55398 D0S7IE 11658882 Ki > 9900 nM T55398 D0T2NE 58056092 IC50 = 8 nM T55398 D0Y2ZC 68115559 IC50 = 7.5 nM T66505 D03EDQ 24776445 IC50 = 5.1 nM T66505 D03LWG 53235510 Ki = 46.5 nM T66505 D04MXN 56846693 Ki = 187.8 nM T66505 D08FDX 24901704 Ki = 41.7 nM T66505 D09BNZ 24775005 Ki = 6 nM T66505 D09UMN 45100669 IC50 < 100 nM T66505 D0D1GF 42642645 Ki = 59.7 nM T66505 D0GD4Q 25027363 IC50 = 1.4 nM T66505 D0M9QZ 11485656 Ki = 87.6 nM T66505 C5V3DJ 1048811 Ki = 50.4 nM T66505 CBVR03 1139102 IC50 = 281 nM T66505 C5W4RP 1300425 IC50 = 89 nM T66505 C0MHW2 2270563 IC50 = 109 nM T66505 C80TKI 2952255 IC50 = 4.4 nM T66505 CFWS91 2953198 IC50 = 91 nM T66505 C1FQR3 3537781 IC50 = 13 nM T66505 CVOH96 3591787 IC50 > 2500 nM T66505 C0LY1H 4269048 Ki = 168.1 nM T66505 CB9I0U 5284329 IC50 = 1500 nM T66505 CK73QZ 6405276 IC50 = 13 nM T66505 CEA26I 6407374 IC50 = 19 nM T66505 C8UB6G 6878030 IC50 = 4.74 nM T66505 CR4Z0H 8440567 IC50 = 1860 nM T66505 C2MJB3 9869236 IC50 = 3420 nM T66505 CLH27B 10392802 IC50 = 140 nM T66505 C1IZR8 10951208 IC50 = 120 nM T66505 CL4BI2 11762419 IC50 = 7520 nM T66505 C2JYM1 18526613 IC50 = 1243 nM T66505 CKU1F2 20875737 IC50 > 5000 nM T66505 C4C9WL 22291085 IC50 = 450 nM T66505 CK6P2Z 24797888 IC50 = 170 nM T66505 CY69VQ 24797889 IC50 = 10 nM T66505 C16WVQ 24797980 IC50 = 240 nM T66505 CZ3EV7 24798071 IC50 = 120 nM T66505 CKYJ26 24905375 IC50 = 8 nM T66505 CN97YF 25065064 IC50 = 724 nM T66505 CEJT74 25065069 IC50 = 2261 nM T66505 CV3R7X 25065678 IC50 = 34 nM T66505 C24YFH 25065681 IC50 = 82 nM T66505 C0HPL9 25065893 IC50 = 185 nM T66505 CJ68BR 25065894 IC50 = 196 nM T66505 CC90KI 25066322 IC50 > 5000 nM T66505 C5UGO6 25066518 IC50 = 112 nM T66505 CGI08J 25066520 IC50 = 95 nM T66505 CYL6V4 25067132 IC50 = 391 nM T66505 CEA5R6 25181471 IC50 < 6 nM T66505 CVPH81 25210551 IC50 = 2700 nM T66505 CI6VC1 25211577 IC50 = 7 nM T66505 CUWT70 25211578 IC50 = 7 nM T66505 CJPE39 25211677 IC50 = 770 nM T66505 CJ0C6Z 25224531 IC50 = 16 nM T66505 C2GBS5 25224707 IC50 = 66 nM T66505 CNX9T4 25226761 IC50 = 1 nM T66505 CUL3B0 25226762 IC50 = 5.8 nM T66505 CCP60F 25226764 IC50 = 12 nM T66505 CC7GX8 25253556 IC50 < 12 nM T66505 C7WZY2 25255940 IC50 = 2.8 nM T66505 CR63VO 44186114 IC50 > 5000 nM T66505 CAU96H 44186115 IC50 = 59 nM T66505 C8I5FZ 44186181 IC50 = 217 nM T66505 CB7K3J 44186182 IC50 > 5000 nM T66505 CBQD07 44186183 IC50 > 5000 nM T66505 C8OLT2 44186184 IC50 = 401 nM T66505 C2EIF1 44186185 IC50 = 230 nM T66505 C9ROY5 44186310 IC50 = 306 nM T66505 CM4SK2 44186312 IC50 = 654 nM T66505 CB5US1 44186313 IC50 = 15 nM T66505 CGR97M 44186314 IC50 = 484 nM T66505 CQ58TU 44186375 IC50 = 67 nM T66505 CJD40V 44186376 IC50 = 21 nM T66505 C3QDF2 44186378 IC50 = 70 nM T66505 CS96ZI 44186429 IC50 = 103 nM T66505 C0L4ES 44186430 IC50 = 25 nM T66505 C1PTH6 44186431 IC50 = 2929 nM T66505 CM8H5Z 44186480 IC50 = 34 nM T66505 C31RVS 44186482 IC50 = 17 nM T66505 C8Z1DQ 44186485 IC50 > 5000 nM T66505 CQT23O 44186526 IC50 > 5000 nM T66505 C6BD5U 44250034 IC50 = 5 nM T66505 CZTH83 44250105 IC50 = 40 nM T66505 C8H9TQ 44395035 IC50 = 3200 nM T66505 C0T2GL 44395101 IC50 = 1100 nM T66505 CY9R4E 44395109 IC50 = 450 nM T66505 C0MT1L 44395257 IC50 > 3000 nM T66505 CF9IW1 44412191 IC50 = 78.4 nM T66505 C1NF9R 44463317 IC50 = 90 nM T66505 CT14KB 44464376 IC50 = 190 nM T66505 CE7J2C 44464620 IC50 = 107 nM T66505 CYJ02G 44464875 IC50 = 80 nM T66505 CYLN29 44517800 IC50 = 31 nM T66505 C3O7TI 44548374 IC50 = 44 nM T66505 C7CJM3 44548378 IC50 = 93 nM T66505 CY9M7W 44549004 IC50 = 40 nM T66505 CRT70E 44591268 IC50 = 30 nM T66505 CQE8H0 44591290 IC50 = 790 nM T66505 C7ZX3O 44591292 IC50 = 1150 nM T66505 C5VUK4 44591325 IC50 = 14 nM T66505 CF1E9T 44591326 IC50 = 340 nM T66505 CVB19K 44591344 IC50 = 32 nM T66505 CMR54E 44591345 IC50 = 55 nM T66505 CPW59G 44591346 IC50 = 210 nM T66505 CO31UZ 44591347 IC50 = 130 nM T66505 CZ2C0W 44610687 IC50 = 380 nM T66505 C4U9EN 44628220 IC50 = 3400 nM T66505 CKM92Y 44628222 IC50 = 2200 nM T66505 CO72KB 44628287 IC50 = 1100 nM T66505 C0YM5V 44628288 IC50 = 1500 nM T66505 CV9A3W 44628450 IC50 = 1200 nM T66505 CMA16F 44628452 IC50 = 1500 nM T66505 CAW8Y9 44628525 IC50 = 320 nM T66505 CK0G2O 44628528 IC50 = 1800 nM T66505 CZY63O 44628618 IC50 = 420 nM T66505 C62FGB 44628620 IC50 = 1300 nM T66505 CPG83O 44628898 IC50 > 2500 nM T66505 CS37ZL 44629065 IC50 = 790 nM T66505 CEX0I1 44629066 IC50 = 1000 nM T66505 CVS96Z 44629067 IC50 = 280 nM T66505 CL9N4Z 44629071 IC50 = 520 nM T66505 CER8Q0 44629155 IC50 = 470 nM T66505 C8XGK2 44629232 IC50 = 510 nM T66505 CDQ47G 44629236 IC50 = 700 nM T66505 CGW6U0 44629295 IC50 = 750 nM T66505 CX1QC4 44629366 IC50 > 2500 nM T66505 CE6B2G 45267515 IC50 = 130 nM T66505 CF8VX0 45267523 IC50 > 10000 nM T66505 CUW4Z0 45267528 IC50 = 70 nM T66505 C0Z3MB 45267540 IC50 = 1800 nM T66505 CUM1G5 45268389 IC50 = 10000 nM T66505 CYU5Q0 45268404 IC50 = 310 nM T66505 CC7H9M 45268408 IC50 = 200 nM T66505 C9VCH6 45268412 IC50 = 100 nM T66505 CS90AD 45269254 IC50 = 3000 nM T66505 CHCB29 45269261 IC50 = 900 nM T66505 CH3NB9 45269264 IC50 = 950 nM T66505 CD0FN3 45270098 IC50 = 1200 nM T66505 CI16LK 45270102 IC50 = 360 nM T66505 CKNH75 45270116 IC50 = 130 nM T66505 CH2F3N 45270117 IC50 > 25000 nM T66505 CRO2M3 45270118 IC50 = 6300 nM T66505 C3PTM6 45270935 IC50 = 720 nM T66505 CN2F0B 45270940 IC50 = 900 nM T66505 CI95MH 45270943 IC50 = 200 nM T66505 C29UPR 45270944 IC50 = 120 nM T66505 CDV71Y 45270956 IC50 = 1400 nM T66505 CGYD64 45271780 IC50 = 10000 nM T66505 CQ9K4Y 45271789 IC50 = 1300 nM T66505 CF12YU 45271790 IC50 = 1200 nM T66505 C2P1MF 45272645 IC50 = 10000 nM T66505 CL1S7X 45272649 IC50 = 10000 nM T66505 CL91PA 45272656 IC50 = 680 nM T66505 CGO7B5 45272667 IC50 > 10000 nM T66505 CB6S7D 45272668 IC50 = 1830 nM T66505 C3C1DS 45273570 IC50 = 330 nM T66505 CES8O2 45273586 IC50 = 150 nM T66505 C1B4AO 45273591 IC50 = 4500 nM T66505 CIQ7M3 45273599 IC50 = 340 nM T66505 CK7XM8 46871826 IC50 = 5.3 nM T66505 CP87LJ 46871827 IC50 = 2.2 nM T66505 CT8FV6 46890873 IC50 = 9.5 nM T66505 CXY13W 46890935 IC50 = 13 nM T66505 C1CIG5 46890990 IC50 = 5.3 nM T66505 CVBK65 46890991 IC50 = 17.3 nM T66505 CIZ8O7 46890992 IC50 = 5.2 nM T66505 C4GR0D 46891044 IC50 = 15 nM T66505 CMT7B2 46891045 IC50 = 10.8 nM T66505 CH1K0L 46891046 IC50 = 20 nM T66505 CY0T2V 46891103 IC50 = 212 nM T66505 CY0A3H 46891104 IC50 = 15 nM T66505 CRW3N1 46891105 IC50 = 20.3 nM T66505 C1V4PY 46891106 IC50 = 110 nM T66505 C2JRG0 46891162 IC50 = 213 nM T66505 C1PC7R 46891163 IC50 = 96 nM T66505 CK6RY3 46891164 IC50 = 3.2 nM T66505 CE46PC 46891165 IC50 = 7 nM T66505 C1JFY6 46891197 IC50 = 11.8 nM T66505 CHQ06G 46891198 IC50 = 3.6 nM T66505 CAYC57 46891199 IC50 = 0.7 nM T66505 CLD87G 46891200 IC50 = 0.4 nM T66505 CVK3A7 46891245 IC50 = 2.3 nM T66505 CQCN85 46891246 IC50 = 7.3 nM T66505 C0NF6E 46891247 IC50 = 10.1 nM T66505 CY89AF 46891248 IC50 = 2.7 nM T66505 C7D9UV 46891298 IC50 = 3.1 nM T66505 CH03ZS 46891299 IC50 = 5.2 nM T66505 CV6MN7 46891300 IC50 = 2340 nM T66505 C59RFZ 46891346 IC50 = 2700 nM T66505 C24DXJ 49840814 IC50 = 4 nM T66505 C2O7ZC 49862152 IC50 = 1870 nM T66505 C9AQO8 49862153 IC50 = 1690 nM T66505 C0AY1M 49862154 IC50 = 20 nM T66505 CSR2H4 49862176 IC50 = 12 nM T66505 CPNL82 49862194 IC50 > 5000 nM T66505 CN0V7S 49862195 IC50 > 5000 nM T66505 CFNZ30 49862196 IC50 = 333 nM T66505 C06TVH 49862197 IC50 = 105 nM T66505 C7H2NL 49862220 IC50 = 19 nM T66505 C0U7CJ 49862221 IC50 = 21 nM T66505 CIUH50 49862222 IC50 > 1000 nM T66505 CZ8GI9 49862236 IC50 = 64.7 nM T66505 C6OQV2 49862237 IC50 = 40.8 nM T66505 C6IW4Q 49862238 IC50 = 8.27 nM T66505 CP1YK8 49862269 IC50 = 3.3 nM T66505 C4HRQ3 49862270 IC50 = 4.8 nM T66505 CCL25Y 49862311 IC50 = 25 nM T66505 C16VMC 49862312 IC50 = 79 nM T66505 C7H5LT 49862313 IC50 = 57 nM T66505 C1J9KL 49862314 IC50 = 8.7 nM T66505 CI0Q6T 49862371 IC50 = 8 nM T66505 C8GS6K 49862372 IC50 > 1000 nM T66505 CB10HZ 49862373 IC50 > 1000 nM T66505 C4FYZ5 49862424 IC50 > 1000 nM T66505 C3QF1T 50768213 IC50 > 2500 nM T66505 CXN52T 50835422 IC50 = 63 nM T66505 CRZL59 53361076 IC50 = 13 nM T66505 C0CE7M 53387030 IC50 = 13 nM T66505 C1RHF7 53387681 IC50 = 5 nM T66505 CTY6C4 53484000 IC50 = 7.2 nM T66505 C13WTO 56658050 IC50 = 46 nM T66505 C8GZD4 56658051 IC50 = 2600 nM T66505 CT62BA 56658169 IC50 = 230 nM T66505 CJDL15 56658170 IC50 = 2000 nM T66505 C30TCQ 56658188 IC50 = 6.4 nM T66505 CV68SR 56658189 IC50 = 48 nM T66505 CL38IE 56658549 IC50 = 180 nM T66505 C4U7WK 56658550 IC50 = 4700 nM T66505 C0G4XL 56658551 IC50 > 2500 nM T66505 C7MBL0 56658552 IC50 > 2500 nM T66505 C75ITF 56658553 IC50 > 2500 nM T66505 C1SH5E 56658575 IC50 = 480 nM T66505 CV2EY4 56658696 IC50 > 2500 nM T66505 CA9KM7 56658697 IC50 = 480 nM T66505 CV6T7E 56658698 IC50 > 2500 nM T66505 CW72LF 56658699 IC50 > 2500 nM T66505 CCA76B 56661560 IC50 = 46 nM T66505 C4H3VZ 56661561 IC50 = 340 nM T66505 CRI23C 56661562 IC50 = 64 nM T66505 C43ICJ 56661679 IC50 = 72 nM T66505 C8D9PR 56662002 IC50 = 15000 nM T66505 C35SAR 56662003 IC50 = 620 nM T66505 CG2U1T 56662004 IC50 = 1000 nM T66505 C9BNK7 56662005 IC50 = 1900 nM T66505 CY26QZ 56662006 IC50 > 2500 nM T66505 CQ41MY 56662174 IC50 = 110 nM T66505 CB4W0O 56662175 IC50 > 2500 nM T66505 CVSD83 56662176 IC50 = 670 nM T66505 C8E5BX 56662793 IC50 = 18 nM T66505 C3PKE1 56663266 IC50 = 3000 nM T66505 CM2O8C 56664980 IC50 = 330 nM T66505 C92THJ 56664981 IC50 = 380 nM T66505 C1ME2L 56665113 IC50 = 37 nM T66505 CAY4Z3 56665494 IC50 = 640 nM T66505 CT9O7X 56665495 IC50 = 6000 nM T66505 CWCK98 56665496 IC50 > 2500 nM T66505 C41XMQ 56665497 IC50 = 2200 nM T66505 CG75HU 56665498 IC50 > 2500 nM T66505 CKA36R 56665499 IC50 > 2500 nM T66505 CKB71O 56665632 IC50 > 2500 nM T66505 CMJ13X 56666699 IC50 = 4600 nM T66505 CX4IC9 56668414 IC50 = 200 nM T66505 CX8Q5Y 56668540 IC50 = 13000 nM T66505 CUFX01 56668541 IC50 = 240 nM T66505 CF7LR5 56668542 IC50 = 32 nM T66505 CI4Q1R 56668557 IC50 = 49 nM T66505 C6KVX4 56668558 IC50 = 27 nM T66505 C2DR5K 56668559 IC50 = 27 nM T66505 CU19OY 56668560 IC50 = 93 nM T66505 CG6JS7 56668711 IC50 = 810 nM T66505 C8W4QB 56668923 IC50 > 2500 nM T66505 CP9U0G 56668924 IC50 = 1000 nM T66505 C02GYK 56668936 IC50 = 45 nM T66505 CMQS94 56669087 IC50 = 1900 nM T66505 C5W8BE 56669674 IC50 = 140 nM T66505 CQJ72G 56669675 IC50 = 100 nM T66505 C51HRV 56669676 IC50 = 15 nM T66505 CR9IJ2 56669677 IC50 = 21 nM T66505 C3IE7S 56671926 IC50 = 530 nM T66505 CYOA69 56671927 IC50 = 390 nM T66505 C5RFI6 56671928 IC50 = 19 nM T66505 CTL7J0 56671929 IC50 = 8 nM T66505 C68YBP 56672043 IC50 = 4900 nM T66505 C4XK3V 56672054 IC50 = 14 nM T66505 CVCW54 56672401 IC50 > 2500 nM T66505 C8CMQ3 56672402 IC50 = 1100 nM T66505 C67POD 56672403 IC50 > 2500 nM T66505 C60FCS 56672404 IC50 > 2500 nM T66505 CK8Y7L 56672544 IC50 = 490 nM T66505 CY8Q6Z 56672545 IC50 = 750 nM T66505 C9O6JQ 56672546 IC50 = 2900 nM T66505 CP0J8E 56672547 IC50 = 1300 nM T66505 COI7L2 56673182 IC50 = 1200 nM T66505 CI9QV5 56675303 IC50 = 790 nM T66505 CO4ND2 56675304 IC50 = 510 nM T66505 CKXE70 56675305 IC50 = 2700 nM T66505 CTE98L 56675306 IC50 = 17000 nM T66505 C5O7WK 56675307 IC50 = 290 nM T66505 CWI58T 56675308 IC50 = 15 nM T66505 CI06FK 56675419 IC50 = 6900 nM T66505 CJEA89 56675420 IC50 = 290 nM T66505 CK57CI 56675440 IC50 = 28 nM T66505 CM5UH2 56675441 IC50 = 33 nM T66505 CY6UA5 56675678 IC50 > 2500 nM T66505 C9C8FG 56675786 IC50 > 2500 nM T66505 CAI9O3 56675787 IC50 > 2500 nM T66505 CSA35C 56675788 IC50 > 2500 nM T66505 CMKQ61 56675800 IC50 = 1600 nM T66505 CK6GW1 56675801 IC50 = 350 nM T66505 CF2GB3 56675802 IC50 = 3 nM T66505 C6IU9P 56675925 IC50 > 2500 nM T66505 CF3R6A 56675926 IC50 = 1500 nM T66505 C04FDY 56675927 IC50 = 2500 nM T66505 C5I4KA 56676509 IC50 = 21 nM T66505 C6RVC4 56676510 IC50 = 230 nM T66505 C41FSK 56676511 IC50 = 19 nM T66505 CO9AX8 56678641 IC50 = 46 nM T66505 CBZ1S6 56678642 IC50 = 180 nM T66505 CL9V4G 56678643 IC50 = 360 nM T66505 CEI80K 56678644 IC50 = 15 nM T66505 CZ9LW6 56678777 IC50 = 79 nM T66505 CWMH38 56679102 IC50 > 2500 nM T66505 CKN39Z 56679103 IC50 > 2500 nM T66505 C0DV4W 56679122 IC50 = 1800 nM T66505 C07JIH 56679237 IC50 > 2500 nM T66505 CR19BZ 56679238 IC50 = 350 nM T66505 C3MI4V 56679239 IC50 = 1700 nM T66505 CC81YD 56679828 IC50 = 430 nM T66505 C03JCI 56679829 IC50 = 1400 nM T66505 CI6UC5 56680279 IC50 = 7800 nM T66505 CDR92Q 56680280 IC50 = 5100 nM T66505 C06HAF 56681960 IC50 = 370 nM T66505 CS30BK 56681961 IC50 = 16 nM T66505 C1Y0MO 56682216 IC50 = 30 nM T66505 CPRT14 56682402 IC50 = 2100 nM T66505 C07GSV 56682403 IC50 > 2500 nM T66505 CDH41P 56682417 IC50 = 760 nM T66505 CGCH03 56682418 IC50 = 25 nM T66505 C3F6TH 56682550 IC50 = 220 nM T66505 CH46PS 56682551 IC50 = 1400 nM T66505 C7BX5M 56682552 IC50 = 340 nM T66505 CN4RZ3 56682553 IC50 = 280 nM T66505 C3L5PZ 56682554 IC50 > 2500 nM T66505 C14GVW 56683156 IC50 = 140 nM T66505 CV85DJ 56683157 IC50 = 42 nM T66505 C6F7RL 56683158 IC50 = 12 nM T66505 C32GXL 56964691 IC50 = 24 nM T66505 C2Q8VL 56964692 IC50 = 41 nM T66505 C27ION 57326206 IC50 = 100 nM T66505 CRJ90X 57326301 IC50 = 180 nM T66505 CH96BW 57326302 IC50 = 820 nM T66505 CL8H5N 57326385 IC50 = 1100 nM T66505 C7SI0M 57326387 IC50 = 29 nM T66505 C61TYN 57326482 IC50 = 130 nM T66505 CF4X2S 57326483 IC50 = 520 nM T66505 CMI5L4 57326484 IC50 = 1800 nM T66505 C32LFE 67374618 IC50 < 16 nM T66505 C46VLA 67374621 EC50 = 15 nM T66505 CLKN38 67375395 IC50 < 19 nM T66505 C5BFR4 67378301 EC50 = 115 nM T66505 CKB37H 67379186 IC50 < 40 nM T66505 C8M9VH 67379418 EC50 = 28 nM T66505 C07NTU 68747277 IC50 = 42 nM T66505 CD9J0Y 68778068 EC50 = 30 nM T66505 CG16HX 68780878 EC50 = 7 nM T66505 CMGA79 70682196 EC50 = 27 nM T66505 CH0T3O 70684298 EC50 = 89 nM T66505 CTCF71 70688555 EC50 = 22 nM T66505 C1Y7FR 70688556 IC50 > 450 nM T66505 CNER46 70690618 EC50 = 21 nM T66505 CTYA67 70692760 EC50 = 8 nM T66505 CFYG52 70694242 IC50 = 110 nM T66505 C45SUB 70694800 EC50 = 17 nM T66505 C95IBJ 70694801 EC50 = 40 nM T66505 C2SWX1 70696850 EC50 = 29 nM T66505 CO58QT 71458712 Ki = 37.9 nM T66505 C0J3TE 76311001 IC50 = 300 nM T66505 C89CXE 76311004 IC50 = 40 nM T66505 CWZE58 76318208 IC50 = 100 nM T66505 C6H5MS 76848956 Ki = 30 nM T66505 C53NWC 86294818 IC50 = 87 nM T66505 CM0A5R 90286184 IC50 = 1800 nM T66505 CIU6F5 90286320 IC50 = 4100 nM T66505 CJ85YQ 90286388 IC50 > 10000 nM T66505 CW6BO1 90286529 IC50 = 910 nM T66505 C0YEV1 90286574 IC50 = 270 nM T66505 C89TEO 90299606 IC50 = 890 nM T66505 C5V3LH 90299611 IC50 = 350 nM T66505 C7LTZ2 90299612 IC50 = 300 nM T66505 C2UV3X 90299614 IC50 = 440 nM T66505 CZ1GP2 90299621 IC50 = 1300 nM T66505 CKD1F0 90299647 IC50 = 690 nM T66505 CFHB98 90644096 IC50 > 25000 nM T66505 CWK6N7 90656290 IC50 = 2700 nM T66505 CK2I6N 90656291 IC50 = 520 nM T66505 CRI41W 90656292 IC50 = 4100 nM T66505 CL29HQ 90656293 IC50 = 790 nM T66505 CD2PB6 90656294 IC50 > 10000 nM T66505 CS8TB7 90656295 IC50 > 10000 nM T66505 CWL3E0 90656296 IC50 = 550 nM T66505 CW7BV0 90656297 IC50 = 1200 nM T66505 CU4NV3 90656298 IC50 = 1500 nM T66505 CP36FA 90656299 IC50 = 420 nM T66505 C6F9NY 90656300 IC50 = 270 nM T66505 COK94Z 90656301 IC50 = 200 nM T66505 CRG6J5 90656302 IC50 = 380 nM T66505 CR4K2D 90656303 IC50 = 270 nM T66505 C9ZU3G 90656304 IC50 = 740 nM T66505 CI7F1H 90656305 IC50 = 960 nM T66505 CVH8R7 90656306 IC50 = 650 nM T66505 C9WDS7 97046899 Ki = 33 nM T66505 CM7LD8 122185868 IC50 = 5.6 nM T66505 CL0ZB6 122185870 IC50 = 10 nM T66505 C9CZ8G 127039132 IC50 = 19 nM T66505 CDVZ38 127039452 IC50 = 42 nM T66505 CILZ74 127048425 IC50 = 373 nM T66505 C0CF8P 127048730 IC50 = 294 nM T66505 C87LZN 127048731 IC50 = 315 nM T66505 C43IVQ 127048732 IC50 = 18 nM T66505 C38MXE 127048733 IC50 = 192 nM T66505 CS57TL 127048734 IC50 = 135 nM T66505 CDT1A0 127049057 IC50 = 352 nM T66505 C92DBP 127049409 IC50 = 326 nM T66505 C8NO0A 127051279 IC50 = 261 nM T66505 CWT20F 127052154 IC50 = 431 nM T66505 CKM9A3 127052181 IC50 = 217 nM T66505 CP7S9A 127052483 IC50 = 92 nM T66505 CCQ86W 127052484 IC50 = 213 nM T66505 C6LU2S 127052485 IC50 = 56 nM T66505 C2CA0W 127053107 IC50 = 456 nM T66505 C2SAG7 127053109 IC50 = 237 nM T66505 CXI0B3 132578555 IC50 > 10000 nM T66505 CY0BT9 136210502 IC50 = 290 nM T66505 CX67HE 136210503 IC50 = 370 nM T66505 CKP6L1 136210504 IC50 = 70 nM T66505 CL47YD 136210505 IC50 = 220 nM T66505 CE1US4 136210506 IC50 = 70 nM T66505 C7OW0J 136210508 IC50 = 160 nM T66505 CL4IW7 136210509 IC50 = 190 nM T66505 CDFZ95 136210510 IC50 = 33 nM T66505 CKS3V1 136210511 IC50 = 5 nM T66505 CKO48T 136210512 IC50 = 110 nM T66505 CE9OD5 136210517 IC50 = 900 nM T66505 CB7AI4 136210518 IC50 = 14 nM T66505 C0TI5R 136244207 IC50 = 640 nM T66505 C9C5MY 145958866 IC50 = 10 nM T66505 CJ8X4A 155515079 Ki = 55 nM T66505 COKI80 155515124 IC50 = 3.9 nM T66505 CTO9C8 155547338 IC50 = 18 nM T66505 CRG7H3 155549835 Ki = 45 nM T66505 C95DIM 155559226 Ki = 28 nM T66505 D03NPX 447077 Ki = 46.2 nM T66505 D05UKJ 442972 Ki = 12.7 nM T66505 D0R8DO 6404568 IC50 = 4237 nM T66505 D0S5OU 73729049 IC50 = 440 nM T41201 CGNU14 10408898 IC50 = 350 nM T41201 CZIY89 11081290 IC50 = 25 nM T41201 CQ4EM2 44344844 IC50 = 40 nM T41201 CCA3Z7 44344899 IC50 = 20 nM T41201 CTPO43 44345020 IC50 = 6 nM T41201 C5KH6G 44345023 IC50 = 5 nM T41201 CL6KF8 44345101 IC50 = 150 nM T41201 C6T5UV 44345102 IC50 = 45 nM T41201 CL32RO 44345105 IC50 = 10 nM T41201 C18KAP 44345106 IC50 = 100 nM T78319 CKUJ53 16217499 IC50 = 6700000 nM T78319 C5D3HE 30980948 IC50 = 14100000 nM T78319 CH8Z3J 73441667 IC50 = 3500000 nM T78319 CG0O3E 90655419 IC50 = 1320000 nM T78319 CR5MK9 90655420 IC50 = 108000 nM T78319 C3CNA9 90655421 IC50 = 65000 nM T78319 CF0EX8 90655422 IC50 = 48000 nM T78319 CGL84T 90655423 IC50 = 36000 nM T78319 D03EPY 7046 IC50 = 27000000 nM T43721 D02ENG 6918651 IC50 > 10000 nM T43721 D05WCI 11670435 IC50 > 10000 nM T43721 D0B5HF 44476893 IC50 > 10000 nM T43721 D0O1ZI 25006684 IC50 > 30000 nM T43721 D0R8IU 24946280 IC50 > 30000 nM T43721 D0T8QB 14982 IC50 = 0.4 nM T43721 D07EBU 135565424 IC50 > 10000 nM T43721 D07FHW 23725123 IC50 > 500000 nM T43721 CDM6C4 92730 IC50 = 400 nM T43721 C7JEN0 94320 IC50 = 750 nM T43721 C2O8KM 101788 IC50 = 490 nM T43721 CFG6D1 111253 IC50 = 329 nM T43721 C8UQT9 1484979 IC50 > 10000 nM T43721 C34FUY 2953793 Ki > 10000 nM T43721 C3B7LM 3146235 IC50 = 8900 nM T43721 CPT5Y6 6918663 IC50 > 200000 nM T43721 C84RBQ 9797661 IC50 > 4000 nM T43721 CY2K5B 9823394 IC50 = 4000 nM T43721 CHV1E3 9975108 IC50 > 4000 nM T43721 CSL50G 9975639 IC50 > 4000 nM T43721 CDZ92L 9998483 IC50 > 4000 nM T43721 CBUP07 10018475 IC50 = 1270 nM T43721 C0I6WB 10040175 IC50 = 3318 nM T43721 CU1W4M 10040176 IC50 = 2006 nM T43721 C4L0HV 10043410 IC50 > 4000 nM T43721 CA4SJ7 10064183 IC50 > 4000 nM T43721 C5LKO8 10085885 IC50 = 1035 nM T43721 CW6KU4 10250720 IC50 = 1300 nM T43721 CO0H7A 10250842 IC50 > 4000 nM T43721 COT1X3 10308303 IC50 > 4000 nM T43721 C2LWK5 10315044 IC50 > 4000 nM T43721 C0QH6L 10335644 IC50 > 4000 nM T43721 C7IUQ6 10335880 IC50 > 4000 nM T43721 CI64PJ 10340916 IC50 > 4000 nM T43721 CL5X6K 10355633 IC50 > 4000 nM T43721 CTLN27 10357519 IC50 > 4000 nM T43721 CTU13Q 10357992 IC50 = 503 nM T43721 CWKP54 10359991 IC50 > 4000 nM T43721 CEO4C7 10360107 IC50 = 613 nM T43721 CUL28X 10380007 IC50 < 4000 nM T43721 CF4NL2 10381554 IC50 = 216 nM T43721 CR4V3G 10402262 IC50 > 4000 nM T43721 C65EQT 10403095 IC50 = 1037 nM T43721 CV8K3E 10446474 IC50 = 4000 nM T43721 CQ9X4Y 10446475 IC50 > 4000 nM T43721 CYI70T 10447474 IC50 = 4000 nM T43721 CS06QG 10452320 IC50 > 100000 nM T43721 CA89WN 10470037 IC50 > 4000 nM T43721 C6LJI0 10473292 IC50 > 4000 nM T43721 CXH39G 10474399 IC50 > 4000 nM T43721 C0C6KD 11190936 IC50 = 122 nM T43721 CD3H7R 11232699 IC50 > 200000 nM T43721 C1PKI0 11257147 IC50 > 200000 nM T43721 CW1T5X 11259177 IC50 = 228 nM T43721 CH12WK 11278558 IC50 > 4000 nM T43721 CP9O5R 11280328 IC50 > 200000 nM T43721 CH85OD 11319723 IC50 = 2350 nM T43721 C8FQ9B 11375180 IC50 = 3950 nM T43721 CS0P1Q 11478969 IC50 = 280 nM T43721 CR4I9H 11484764 IC50 = 290 nM T43721 CN08AP 11495851 IC50 > 10000 nM T43721 CLT1Z9 11502804 IC50 = 6300 nM T43721 C76STL 11504178 IC50 = 21000 nM T43721 C19BYP 11505338 IC50 = 50000 nM T43721 CHW7L1 11510573 IC50 > 100000 nM T43721 CE40MU 11524868 IC50 = 550 nM T43721 C8NP4Y 11526147 IC50 = 3 nM T43721 CG1HB5 11533520 IC50 = 24000 nM T43721 CZE42S 11540388 IC50 = 13000 nM T43721 CN1A6F 11540493 IC50 > 100000 nM T43721 C3LVE2 11545617 IC50 = 30000 nM T43721 CD17CO 11551576 IC50 > 10000 nM T43721 CP8L9K 11552169 IC50 = 23000 nM T43721 CCT0Q7 11552781 IC50 = 18000 nM T43721 CA25ZF 11555218 IC50 = 34000 nM T43721 CJ58XB 11576524 IC50 = 25000 nM T43721 CKF3J6 11604308 IC50 = 16000 nM T43721 CGD7X9 11610822 IC50 = 12000 nM T43721 CDL39R 11613794 IC50 > 30000 nM T43721 C7KBZ4 11618761 IC50 = 5500 nM T43721 CW2XN3 11626362 IC50 = 85000 nM T43721 CXS05L 11627334 IC50 > 10000 nM T43721 CMF3U5 11634114 IC50 > 100000 nM T43721 CDL94B 11649095 IC50 > 100000 nM T43721 CX17LY 11654021 IC50 = 1800 nM T43721 C3B4SN 11655097 IC50 > 20000 nM T43721 C1DJ7W 11655188 IC50 = 26000 nM T43721 C1T6KE 11666874 IC50 = 8300 nM T43721 CFH6G5 11670914 IC50 = 20000 nM T43721 CU5TI1 11676805 IC50 > 100000 nM T43721 CJ13XD 11698697 IC50 = 5300 nM T43721 C26ITU 11699075 IC50 = 27000 nM T43721 CK8BF3 11705872 IC50 > 10000 nM T43721 C4D6YM 11712182 IC50 = 60000 nM T43721 C5AT6X 11722880 IC50 = 1961 nM T43721 CO32UM 11724534 IC50 = 1964 nM T43721 C6TPR1 11739354 IC50 > 4000 nM T43721 C4B5XT 11741200 IC50 > 4000 nM T43721 CB9WI2 11742158 IC50 > 4000 nM T43721 C37IRX 11771845 IC50 = 183 nM T43721 C2XW0P 11853305 IC50 = 6040 nM T43721 C4FKP2 13994830 IC50 > 1000000 nM T43721 CEYW48 15953464 IC50 = 2520 nM T43721 CY3A6Q 15987396 IC50 > 10000 nM T43721 C29ACV 15987476 IC50 > 10000 nM T43721 CS1XM4 16049788 IC50 = 100000 nM T43721 C2T4IM 16222378 IC50 = 30.4 nM T43721 C13TPH 16721119 IC50 > 10000 nM T43721 C2OJC1 16726072 IC50 > 10000 nM T43721 C69QUM 20724870 IC50 = 1174 nM T43721 C51LGI 20724898 IC50 > 4000 nM T43721 CP7JM8 20724899 IC50 > 4000 nM T43721 C31VAH 20724901 IC50 > 4000 nM T43721 CJU3T5 20724903 IC50 > 4000 nM T43721 CLX5A8 20724912 IC50 > 4000 nM T43721 CQ6CF3 20755069 IC50 > 4000 nM T43721 CTRD81 20755103 IC50 > 1000 nM T43721 CD1SR0 22591684 IC50 > 4000 nM T43721 CQ6AO5 22591709 IC50 = 7.5 nM T43721 CWF51V 22591726 IC50 > 4000 nM T43721 CEB47A 24744047 IC50 = 21200 nM T43721 CGR84K 24854349 IC50 > 500000 nM T43721 C6BV8N 24854350 IC50 > 500000 nM T43721 CEW31B 24856362 IC50 > 100000 nM T43721 C7QU2Z 24883422 IC50 = 10000 nM T43721 CLYS75 24889741 IC50 = 20 nM T43721 CVD4K7 24889906 IC50 = 15000 nM T43721 C6EFK9 24889907 IC50 > 30000 nM T43721 C5QD7L 24890069 IC50 = 1600 nM T43721 C9XUC0 24890070 IC50 = 1800 nM T43721 C3A9HI 24890073 IC50 = 90000 nM T43721 C6IHL0 24890239 IC50 = 23000 nM T43721 CEV27L 24895554 IC50 > 10000 nM T43721 C8LYV0 24895658 IC50 > 10000 nM T43721 C2QWU0 24895661 IC50 > 10000 nM T43721 C1G6DM 24895969 IC50 > 10 nM T43721 C59MRG 24896012 IC50 > 10 nM T43721 C6UYQ4 24948172 IC50 > 10000 nM T43721 CJL38O 25065024 IC50 > 10000 nM T43721 C8GR2K 25065025 IC50 = 510 nM T43721 CEMG39 25065027 IC50 > 10000 nM T43721 CB36SV 25065227 IC50 > 10000 nM T43721 C7YH6J 25065230 IC50 > 10000 nM T43721 C9EQ1D 25065231 IC50 > 10000 nM T43721 CU12CJ 25065232 IC50 = 10 nM T43721 CEQF65 25210659 IC50 > 100000 nM T43721 CU7E9B 25265683 IC50 > 10000 nM T43721 CMVE89 42603038 IC50 > 10000 nM T43721 C6VQM9 44143289 IC50 > 100000 nM T43721 CZ58CY 44143291 IC50 > 100000 nM T43721 C8X2ZV 44143292 IC50 > 100000 nM T43721 C1IA7U 44143299 IC50 > 100000 nM T43721 C63STN 44196869 IC50 = 31.2 nM T43721 C7YTM0 44197230 IC50 > 4000 nM T43721 CHA7J4 44250316 IC50 > 1000000 nM T43721 C9S2HX 44402393 IC50 > 200000 nM T43721 C8C2QJ 44402534 IC50 > 200000 nM T43721 CW7IP2 44402550 IC50 > 200000 nM T43721 C0NUI2 44402662 IC50 > 200000 nM T43721 C42FXZ 44418375 IC50 > 100000 nM T43721 CC93VQ 44418376 IC50 = 16000 nM T43721 CP9DO4 44418378 IC50 = 52000 nM T43721 CR7K6S 44418382 IC50 > 100000 nM T43721 C7B6GT 44418383 IC50 > 100000 nM T43721 C1Q8CH 44418384 IC50 > 100000 nM T43721 C7JNH9 44418385 IC50 = 100000 nM T43721 CB58SX 44418389 IC50 = 70000 nM T43721 CGKR51 44418390 IC50 = 49000 nM T43721 CQT37N 44418391 IC50 > 100000 nM T43721 CED27U 44418395 IC50 > 100000 nM T43721 C9L7BU 44418396 IC50 > 100000 nM T43721 C28DBM 44418400 IC50 > 100000 nM T43721 C1KD8E 44418401 IC50 > 100000 nM T43721 CT79UX 44418408 IC50 > 100000 nM T43721 C7RW1O 44418409 IC50 > 100000 nM T43721 C7WQD4 44418433 IC50 > 30000 nM T43721 CV87RE 44418434 IC50 > 30000 nM T43721 CK74ZJ 44418441 IC50 > 30000 nM T43721 C02AMZ 44418445 IC50 > 30000 nM T43721 C7YCN4 44418447 IC50 > 100000 nM T43721 C7AKJ2 44418450 IC50 > 100000 nM T43721 C90QWN 44418451 IC50 = 55000 nM T43721 CA2J1I 44418452 IC50 = 11000 nM T43721 CE1W9Y 44418456 IC50 = 90000 nM T43721 C7R3AT 44418457 IC50 > 100000 nM T43721 C4MVN6 44418458 IC50 = 15000 nM T43721 CXFR60 44418459 IC50 = 100000 nM T43721 CAW7Z2 44418817 IC50 > 100000 nM T43721 CC8ZR0 44418821 IC50 > 100000 nM T43721 CKX95Y 44418852 IC50 > 100000 nM T43721 CF56NG 44418856 IC50 = 56000 nM T43721 CGX84K 44418857 IC50 = 62000 nM T43721 CSP8W1 44419286 IC50 > 30000 nM T43721 CQH6X0 44419304 IC50 = 17000 nM T43721 CBI64W 44419309 IC50 = 14000 nM T43721 C6LOU9 44419313 IC50 = 630 nM T43721 C32WUT 44420153 IC50 > 10000 nM T43721 C14JQE 44420164 IC50 > 10000 nM T43721 C76RGZ 44420166 IC50 > 10000 nM T43721 CINJ57 44420180 IC50 > 10000 nM T43721 CWM5F9 44420181 IC50 > 10000 nM T43721 CLA82E 44420186 IC50 > 10000 nM T43721 C0ET3O 44420190 IC50 > 10000 nM T43721 C3JF5Z 44420196 IC50 > 10000 nM T43721 C64UQO 44420202 IC50 > 10000 nM T43721 CJI76N 44420207 IC50 > 10000 nM T43721 C0T6ML 44420212 IC50 > 10000 nM T43721 C5Y4UB 44420215 IC50 > 10000 nM T43721 C1NCR3 44420232 IC50 > 10000 nM T43721 CQ7B8C 44420233 IC50 > 10000 nM T43721 C0X3PE 44420237 IC50 > 10000 nM T43721 CO4S5M 44420238 IC50 > 10000 nM T43721 CV6P7Y 44420242 IC50 > 10000 nM T43721 C8IH5C 44420243 IC50 > 10000 nM T43721 CZG60J 44420244 IC50 = 50000 nM T43721 CN2B1J 44420246 IC50 > 10000 nM T43721 CG90VX 44420247 IC50 > 10000 nM T43721 C5PU7K 44420248 IC50 > 10000 nM T43721 C7KW0L 44420249 IC50 = 100000 nM T43721 CBL6K2 44420251 IC50 > 10000 nM T43721 CF9N4T 44420252 IC50 > 10000 nM T43721 CVX2Z3 44420253 IC50 > 10000 nM T43721 CX8IQ0 44420257 IC50 > 10000 nM T43721 CN3W4S 44420259 IC50 = 3600 nM T43721 C1YLR4 44420285 IC50 = 65000 nM T43721 CNRY91 44420288 IC50 > 10000 nM T43721 CF23SE 44420291 IC50 > 10000 nM T43721 CE7T4W 44420294 IC50 = 15000 nM T43721 CJ1O7N 44438556 IC50 = 17000 nM T43721 CH0K4M 44438559 IC50 = 3500 nM T43721 CXM65L 44438562 IC50 = 26000 nM T43721 CM01KY 44438566 IC50 = 20000 nM T43721 CFLP12 44438567 IC50 = 12000 nM T43721 CAW10E 44438568 IC50 = 25000 nM T43721 C3IK2C 44438569 IC50 > 100000 nM T43721 C43RLG 44438570 IC50 = 580 nM T43721 CM1Y7N 44438669 IC50 = 15000 nM T43721 CUE3I1 44438670 IC50 = 3300 nM T43721 CQM10L 44438671 IC50 = 15000 nM T43721 CB19EU 44438672 IC50 = 5400 nM T43721 CL4Y3J 44438673 IC50 = 17000 nM T43721 C7ON6I 44438675 IC50 = 65000 nM T43721 C5LN8W 44438676 IC50 > 100000 nM T43721 C8VI7M 44438677 IC50 > 100000 nM T43721 CV12KJ 44438678 IC50 = 21000 nM T43721 CBX9L4 44438679 IC50 = 59000 nM T43721 CF5YU4 44438681 IC50 > 100000 nM T43721 CJ2M3L 44438682 IC50 = 9000 nM T43721 CJB5H3 44443435 Ki > 10000 nM T43721 C3U1WZ 44448872 IC50 > 4000 nM T43721 CZ5A6G 44576636 IC50 > 4000 nM T43721 CHD6G5 44576637 IC50 > 4000 nM T43721 CK67LT 44576651 IC50 > 4000 nM T43721 C9JB2Y 44576672 IC50 > 4000 nM T43721 CMJ91U 44576707 IC50 > 4000 nM T43721 C8D1LU 44576749 IC50 > 4000 nM T43721 CKH1A8 44576750 IC50 > 4000 nM T43721 CN93WV 44576751 IC50 > 4000 nM T43721 CAH82I 44576752 IC50 > 4000 nM T43721 CK5S4W 44576802 IC50 > 4000 nM T43721 C9L3CP 44576803 IC50 > 4000 nM T43721 C2F5RM 44576804 IC50 > 4000 nM T43721 CK41XQ 44576805 IC50 > 4000 nM T43721 CO5YU9 44576846 IC50 > 4000 nM T43721 C4YIR7 44576873 IC50 > 4000 nM T43721 C2HW0I 44576875 IC50 > 4000 nM T43721 COQ7U4 44576945 IC50 > 4000 nM T43721 C18JAM 45269430 IC50 > 1000000 nM T43721 CGPF36 45270351 IC50 > 10000 nM T43721 C83OJH 45271081 IC50 > 1000000 nM T43721 C7O3DH 45271171 IC50 = 2487 nM T43721 CE07FS 45272366 IC50 > 10000 nM T43721 CK65BP 46213656 IC50 > 10000 nM T43721 CHI5S0 46216688 IC50 > 10000 nM T43721 CAX31B 46216689 IC50 > 10000 nM T43721 CN39HK 46229717 IC50 = 268 nM T43721 C4N8DB 46231719 IC50 > 10000 nM T43721 C4WT0Q 46231721 IC50 = 9000 nM T43721 CIX36V 46894126 IC50 = 2.9 nM T43721 CS13YQ 49846481 IC50 > 100000 nM T43721 C6W2XQ 49846838 IC50 > 100000 nM T43721 CA8N9P 52911994 IC50 > 30000 nM T43721 CICZ45 52918012 IC50 > 10000 nM T43721 C4X2WF 52939227 IC50 = 11 nM T43721 CQ6R0S 52939228 IC50 = 33 nM T43721 C1YRT3 52940913 IC50 = 4.9 nM T43721 CSXY62 52941059 IC50 = 7350 nM T43721 C8X4NE 52945350 IC50 = 61.1 nM T43721 CE3AQ9 52945888 IC50 = 458 nM T43721 CO7ZR1 52947102 IC50 = 8650 nM T43721 C2KHL7 52947144 IC50 = 14.5 nM T43721 CJI28A 52950107 IC50 = 2130 nM T43721 CSUK37 53322740 IC50 = 104 nM T43721 CQ7J8E 53322756 IC50 = 194 nM T43721 C6W3JM 53326660 IC50 = 17 nM T43721 CP91BU 53326661 IC50 = 45 nM T43721 C9H5YE 53361128 IC50 > 10000 nM T43721 CN93FS 54580118 IC50 > 4000 nM T43721 CF05VK 54580143 IC50 > 4000 nM T43721 C7FXV6 54580144 IC50 > 4000 nM T43721 C2M8XQ 54580210 IC50 > 4000 nM T43721 C4Q6MO 54580243 IC50 > 4000 nM T43721 CBX17R 54581094 IC50 > 4000 nM T43721 C8O9WK 54581095 IC50 > 4000 nM T43721 CM67RK 54581096 IC50 = 2300 nM T43721 C8ZDF3 54581137 IC50 > 4000 nM T43721 C14YRS 54581213 IC50 > 4000 nM T43721 CQ7GV2 54582134 IC50 > 4000 nM T43721 CZ1B6L 54582135 IC50 > 4000 nM T43721 C07KDH 54582136 IC50 = 3100 nM T43721 CK29GC 54582137 IC50 > 4000 nM T43721 CKGX19 54582164 IC50 > 4000 nM T43721 CWA6Q0 54582242 IC50 > 4000 nM T43721 C07LYE 54582261 IC50 > 4000 nM T43721 CP2N1C 54582262 IC50 > 4000 nM T43721 CM2QX4 54583079 IC50 > 4000 nM T43721 CMKQ26 54583080 IC50 > 4000 nM T43721 C2G7LK 54583125 IC50 > 4000 nM T43721 CL6Z9X 54583126 IC50 > 4000 nM T43721 CGM2W4 54583127 IC50 > 4000 nM T43721 CF42QY 54583128 IC50 > 4000 nM T43721 CWHS39 54583210 IC50 = 4000 nM T43721 CDK5V0 54583231 IC50 > 4000 nM T43721 C5V4DY 54583232 IC50 > 4000 nM T43721 C1JV9N 54583233 IC50 = 1600 nM T43721 CKA9L3 54583234 IC50 > 4000 nM T43721 CZ4YV3 54584081 IC50 > 4000 nM T43721 CHP62C 54584119 IC50 > 4000 nM T43721 CD2QO1 54584120 IC50 = 1300 nM T43721 CCT0B2 54584121 IC50 > 4000 nM T43721 C0VPS6 54584122 IC50 > 4000 nM T43721 C6P5XR 54584196 IC50 > 4000 nM T43721 CY2WM3 54584197 IC50 > 4000 nM T43721 CXNP26 54584198 IC50 > 4000 nM T43721 CWY83C 54584415 IC50 > 4000 nM T43721 CGD4N3 54585028 IC50 > 4000 nM T43721 C8NZ2B 54585029 IC50 > 4000 nM T43721 CHW48S 54585030 IC50 > 4000 nM T43721 CZ8R0S 54585053 IC50 > 4000 nM T43721 C04IZR 54585054 IC50 > 4000 nM T43721 C6GZB9 54585157 IC50 > 4000 nM T43721 C5SHO2 54585992 IC50 > 4000 nM T43721 CJA5Z6 54585993 IC50 > 4000 nM T43721 C4JTZ5 54585994 IC50 > 4000 nM T43721 CKF15E 54586030 IC50 > 4000 nM T43721 CT12RX 54586031 IC50 > 4000 nM T43721 CD6FC5 54586091 IC50 = 1300 nM T43721 CDG95F 54586092 IC50 > 4000 nM T43721 CJ8K1Y 54586966 IC50 > 4000 nM T43721 C51MDN 54586967 IC50 > 4000 nM T43721 CH2F8P 54586968 IC50 > 4000 nM T43721 C61ZTA 54586969 IC50 > 4000 nM T43721 C3Y6HF 54587012 IC50 > 4000 nM T43721 CUF68X 54587090 IC50 = 460 nM T43721 CI1PV5 54587121 IC50 > 4000 nM T43721 C6PSJ3 54587122 IC50 > 4000 nM T43721 C9D1UH 54587123 IC50 > 4000 nM T43721 C82TDJ 54587124 IC50 > 4000 nM T43721 CNQ41E 54590876 IC50 > 10000 nM T43721 C3IAB0 57392785 IC50 = 386 nM T43721 C4I9DE 57408764 IC50 > 100000 nM T43721 CM2DN9 57408765 IC50 = 400 nM T43721 CAI0P1 57418438 IC50 > 100000 nM T43721 C39SNL 57916360 IC50 > 30000 nM T43721 CG16CV 57916503 IC50 > 30000 nM T43721 CG1Y8Z 67464068 IC50 > 10000 nM T43721 CJL0P9 67468231 IC50 > 10000 nM T43721 CM80QX 70687773 EC50 = 2200 nM T43721 CZI43B 70691963 EC50 = 860 nM T43721 CQ5GB9 70691964 EC50 = 720 nM T43721 C3CAB4 71456572 IC50 = 2200 nM T43721 CU24OM 71458421 IC50 > 10000 nM T43721 C0D3IO 71511561 IC50 > 10 nM T43721 C4LAB0 72204152 IC50 = 2200 nM T43721 C17NBW 72204153 IC50 = 2410 nM T43721 CTN6U7 72204155 IC50 = 2690 nM T43721 C0N7EJ 72204340 IC50 = 5850 nM T43721 CS3TL6 72204534 IC50 = 4210 nM T43721 CA5KC4 72204732 IC50 = 6760 nM T43721 C2Q6YJ 72670421 IC50 = 4000 nM T43721 CYAJ36 73345978 IC50 = 1600 nM T43721 CG15WM 73352110 IC50 > 100000 nM T43721 CALM65 73352112 IC50 > 100000 nM T43721 C9WA7F 73353568 IC50 > 100000 nM T43721 CV72YC 73355069 IC50 > 100000 nM T43721 CGR3P5 73355072 IC50 = 228700 nM T43721 C15SEC 73356624 IC50 > 1000000 nM T43721 C2FOM5 73356626 IC50 = 700 nM T43721 CV70BR 73356628 IC50 > 1000000 nM T43721 CWC4Z5 73356629 IC50 > 100000 nM T43721 CPN65E 90643787 IC50 > 30000 nM T43721 CQ23WR 90667215 IC50 > 30000 nM T43721 CFSK10 101911911 IC50 = 25500 nM T43721 CO0H9S 101911912 IC50 = 40700 nM T43721 C91CLR 101911913 IC50 = 299600 nM T43721 C9RBA1 101911914 IC50 = 283600 nM T43721 CMOG09 101911915 IC50 = 11300 nM T43721 CMX6S5 118709259 IC50 > 10000 nM T43721 C7WYI8 127037831 IC50 > 1000000 nM T43721 CI5HA6 127037875 IC50 > 1000000 nM T43721 CP0JV9 127038197 IC50 > 1000000 nM T43721 C4E1LF 127040565 IC50 > 1000000 nM T43721 CTN4E7 127040566 IC50 > 1000000 nM T43721 CB67LT 127040901 IC50 > 1000000 nM T43721 C5P3KE 127040902 IC50 > 1000000 nM T43721 CT5Q1A 127040903 IC50 > 1000000 nM T43721 CW3FN4 127040904 IC50 > 1000000 nM T43721 C9EQX2 127040905 IC50 > 1000000 nM T43721 C32ADQ 127040906 IC50 > 1000000 nM T43721 CYNI06 127041808 IC50 > 1000000 nM T43721 C1ZUD5 127041809 IC50 > 1000000 nM T43721 CCU4H6 127041810 IC50 > 1000000 nM T43721 CZN2A0 127041811 IC50 > 1000000 nM T43721 CCKL17 127042099 IC50 > 1000000 nM T43721 C24EQS 127042100 IC50 > 1000000 nM T43721 CE64CI 127042101 IC50 > 1000000 nM T43721 COR6A5 127042102 IC50 > 1000000 nM T43721 CKM3I9 127042477 IC50 > 1000000 nM T43721 CMP75K 127042478 IC50 > 1000000 nM T43721 CMCP64 127042780 IC50 > 1000000 nM T43721 C4OUL9 127042781 IC50 > 1000000 nM T43721 CGWV92 132053849 IC50 < 100 nM T43721 CT05EL 135399889 IC50 > 10000 nM T43721 C02KAD 135440148 IC50 > 4000 nM T43721 CE0S3Y 135465949 IC50 > 4000 nM T43721 CM7A1J 135492551 IC50 > 4000 nM T43721 C98OIC 135611051 IC50 > 10000 nM T43721 CCQJ43 135611106 IC50 > 10000 nM T43721 C2K9OD 135611129 IC50 > 10000 nM T43721 C4YO9E 135612240 IC50 > 4000 nM T43721 C76MEG 135783319 IC50 > 10000 nM T43721 CMQ2L1 135783320 IC50 > 10000 nM T43721 CE6L4S 135783321 IC50 > 10000 nM T43721 CTAM34 135783322 IC50 > 10000 nM T43721 C7B3JV 135783325 IC50 > 10000 nM T43721 C59KXI 135783328 IC50 > 10000 nM T43721 CKB54L 135783329 IC50 > 10000 nM T43721 C7ZTC5 135783333 IC50 > 10000 nM T43721 C09UQY 135783334 IC50 > 10000 nM T43721 CL5F0J 135783335 IC50 > 10000 nM T43721 CA2ZD0 135857035 IC50 > 10000 nM T43721 CV64MY 135857036 IC50 > 10000 nM T43721 C6IYH3 135967877 IC50 = 35000 nM T43721 C0FO4G 135980568 IC50 = 15 nM T43721 CX3VU1 136000590 IC50 > 4000 nM T43721 CNQ25Z 136021384 IC50 > 10000 nM T43721 C7W4GE 136088954 IC50 > 4000 nM T43721 CT3RN8 136141565 IC50 = 11 nM T43721 CR74OZ 136188845 IC50 > 4000 nM T43721 CWJ0X4 137637923 IC50 = 6261 nM T43721 CDS86M 137656441 IC50 = 9582 nM T43721 C94RSY 137656587 IC50 > 10000 nM T43721 C0DHM9 145952000 IC50 = 100 nM T43721 CC91LF 145952333 IC50 < 100 nM T43721 CDT3Q6 145956314 IC50 = 1000 nM T43721 C09QUS 145958039 IC50 < 100 nM T43721 CV6Q5J 145960157 IC50 = 100 nM T43721 CMVS94 155512106 IC50 > 500000 nM T43721 C1F9PV 155515115 IC50 > 500000 nM T43721 CPO9M4 155520336 IC50 > 500000 nM T43721 CXOU89 155521135 IC50 > 500000 nM T43721 C8WNT0 155521284 IC50 > 500000 nM T43721 CN59WH 155525513 IC50 > 500000 nM T43721 C1D4WM 155537728 IC50 > 500000 nM T43721 CV5KQ0 155543491 IC50 > 500000 nM T43721 CKFU03 155545095 IC50 > 500000 nM T43721 CG19XT 155548236 IC50 > 500000 nM T43721 CB08IM 155548826 IC50 > 500000 nM T43721 C1GC0O 155553184 IC50 > 500000 nM T43721 CEM03Y 155556588 IC50 > 500000 nM T43721 C9E6AM 155561480 IC50 > 500000 nM T43721 COWH25 155562798 IC50 > 500000 nM T43721 CZT7P4 155567250 IC50 > 500000 nM T43721 D00PSW 3630776 IC50 > 3000 nM T43721 D00QOL 11673314 IC50 > 10000 nM T43721 D02KXX 586971 IC50 > 200000 nM T43721 D02WUU 15627039 IC50 > 200000 nM T43721 D03JWH 135450677 IC50 > 10000 nM T43721 D04WVV 10193044 IC50 > 4000 nM T43721 D0A4ZR 135950111 Ki > 10000 nM T43721 D0EU9W 16750524 IC50 > 200000 nM T43721 D0L4VR 636403 IC50 = 170 nM T43721 D0M4PP 4271571 IC50 > 200000 nM T43721 D0P7RN 1483401 IC50 > 200000 nM T43721 D0T3FW 44419251 IC50 > 10000 nM T43721 D0U8IF 10114 IC50 = 1.2 nM T09513 D0A3MV 448014 IC50 > 100000 nM T09513 CH20NR 403176 IC50 = 20 nM T09513 CNG96H 25210579 IC50 > 10000 nM T09513 CE1ZK6 54759168 IC50 > 10000 nM T09513 CL5IR0 135512024 IC50 = 7 nM T09513 D03YVL 5472558 IC50 = 25000 nM T09513 D0Y0ES 3707 IC50 = 100 nM T32880 D06VNK 1110 IC50 = 3000 nM T32880 D01SPD 69669724 IC50 = 280 nM T32880 D03GOO 444972 IC50 = 19000 nM T32880 D03YKE 11256664 IC50 = 591.4 nM T32880 D07KEH 23634441 IC50 = 29 nM T32880 D0N6CS 6914666 IC50 = 70 nM T32880 D00IKR 52912218 IC50 = 14000 nM T32880 D01XZT 24891734 IC50 = 650 nM T32880 D03TPE 97394 IC50 = 14000 nM T32880 D09NCT 53392492 IC50 = 83000 nM T32880 D0QI0J 134204791 IC50 = 15000 nM T32880 CWJ0U1 5312 IC50 = 18000 nM T32880 CMO39B 7493 Ki > 300000 nM T32880 CK23OU 76549 IC50 > 1000000 nM T32880 C8JBE5 94284 IC50 = 8500 nM T32880 C06WZQ 222878 IC50 > 100000 nM T32880 CBZ21G 231363 IC50 > 100000 nM T32880 COS62U 245007 IC50 > 100000 nM T32880 C0MHV8 252439 IC50 = 94000 nM T32880 C3OZ5L 919929 IC50 > 100000 nM T32880 C2OS3W 2238068 IC50 > 100000 nM T32880 CHV8N5 4666803 IC50 > 40000 nM T32880 CGP0X9 6914624 IC50 = 1400 nM T32880 CS7C1Z 8027170 IC50 = 12000 nM T32880 CYJ23Z 10470802 IC50 = 4800 nM T32880 CP76HX 11372202 IC50 = 2400 nM T32880 CM6Q3H 11788622 IC50 > 100000 nM T32880 CDM30S 13770962 IC50 > 1000000 nM T32880 CO03CL 14991438 IC50 = 95000 nM T32880 C9M2AL 16126655 IC50 = 190 nM T32880 CIU0N5 16126706 IC50 = 3900 nM T32880 CI45OC 16126774 IC50 = 3600 nM T32880 CX5VP0 18372521 IC50 = 5300 nM T32880 C52JUB 18372631 IC50 = 4400 nM T32880 CN2HO1 18632368 IC50 = 69700 nM T32880 CDSM62 20816892 IC50 = 4200 nM T32880 C20YQO 22122176 IC50 > 1000000 nM T32880 C92REF 22345738 IC50 = 398000 nM T32880 CCAM68 22959876 IC50 > 100000 nM T32880 CGE7Y9 23260762 IC50 > 1000000 nM T32880 CZ9X6U 24812792 IC50 = 3 nM T32880 CZ8WG7 24831508 IC50 = 22.2 nM T32880 CE9N0S 24891150 IC50 > 100000 nM T32880 CV17FS 24894050 IC50 = 21 nM T32880 C0R7YW 25105470 IC50 = 3 nM T32880 C9TN1M 25105471 IC50 = 3 nM T32880 C9CLE1 25138008 IC50 > 1000000 nM T32880 C8P4AV 25173259 IC50 = 185 nM T32880 C5PJZ9 25173339 IC50 = 44 nM T32880 CIM16Z 25173590 IC50 = 7.8 nM T32880 CP8D4L 25173666 IC50 = 140 nM T32880 CTNC06 25173744 IC50 = 52 nM T32880 C92CGK 25173747 IC50 = 30 nM T32880 C5YWM9 25173822 IC50 = 17 nM T32880 CIF90R 25173824 IC50 = 4.1 nM T32880 C3C0AO 25173900 IC50 = 11 nM T32880 C4TNI3 25206050 IC50 = 1500 nM T32880 CS6N9A 42639237 IC50 = 45500 nM T32880 C2AG1B 42639238 IC50 = 8600 nM T32880 C4LK0F 42639413 IC50 = 700 nM T32880 CY6M3D 42639898 IC50 = 1900 nM T32880 CDE5U3 44419123 IC50 = 46000 nM T32880 CFI5L3 44419124 IC50 = 39000 nM T32880 C0U8JS 44419131 IC50 = 15000 nM T32880 C0Y2EG 44419132 IC50 > 100000 nM T32880 CMD26E 44419133 IC50 = 20000 nM T32880 CLQ71X 44419139 IC50 = 4900 nM T32880 C7MYD0 44419140 IC50 = 6500 nM T32880 C0O3EP 44419147 IC50 = 15000 nM T32880 C5IQT0 44419154 IC50 = 18000 nM T32880 CO8HT3 44419159 IC50 = 15000 nM T32880 CGW2A6 44419160 IC50 = 7300 nM T32880 C6ZYP0 44419165 IC50 = 6800 nM T32880 CB1YA2 44419171 IC50 = 19000 nM T32880 C4QH8U 44419179 IC50 = 10000 nM T32880 CY4NW1 44419252 IC50 = 17000 nM T32880 C6T3AY 44419262 IC50 = 5000 nM T32880 C2FSX3 44419264 IC50 = 14200 nM T32880 C5M4KV 44419265 IC50 = 6800 nM T32880 CE5N3Y 44419266 IC50 = 4600 nM T32880 CQ0IJ2 44419267 IC50 = 7400 nM T32880 C38SEB 44419270 IC50 = 16000 nM T32880 C6OR8X 44419271 IC50 = 4400 nM T32880 C0CW1M 44419272 IC50 = 28700 nM T32880 CQ0A4B 44419273 IC50 = 6000 nM T32880 CVE69C 44419277 IC50 = 9700 nM T32880 C7UOR2 44419278 IC50 = 6100 nM T32880 C1H6FT 44419280 IC50 = 8100 nM T32880 CX43WB 44419281 IC50 = 5900 nM T32880 C0YGE2 44419282 IC50 = 14000 nM T32880 CNR45T 44419283 IC50 = 4100 nM T32880 CE5N6U 44419284 IC50 = 10000 nM T32880 C4UEG7 44419285 IC50 = 3200 nM T32880 CGSN20 44419287 IC50 = 7200 nM T32880 COR69J 44419288 IC50 = 6900 nM T32880 C6NXA4 44419290 IC50 = 5800 nM T32880 C3IW5O 44419297 IC50 = 19000 nM T32880 CAP3T5 44419302 IC50 = 24000 nM T32880 C2X1ZV 44419317 IC50 = 2700 nM T32880 CNV8A6 44419318 IC50 = 580 nM T32880 CS85EJ 44419319 IC50 = 1700 nM T32880 CI2M5C 44419320 IC50 = 2400 nM T32880 C0TIU7 44419321 IC50 = 2400 nM T32880 C1MOH2 44419325 IC50 = 1600 nM T32880 C7KUX4 44419326 IC50 = 1600 nM T32880 C37UJB 44419329 IC50 = 2100 nM T32880 C8SQT3 44419330 IC50 = 2900 nM T32880 C2GTJ8 44419333 IC50 = 1700 nM T32880 C96OKR 44419334 IC50 = 2800 nM T32880 CP42UL 44419336 IC50 = 12000 nM T32880 CPX3V9 44419342 IC50 = 24000 nM T32880 C0B9TD 44419346 IC50 > 100000 nM T32880 C5Z3XD 44462724 IC50 = 1.6 nM T32880 C3CST2 44462748 IC50 = 6.8 nM T32880 CR05QL 44469096 IC50 > 100000 nM T32880 C9MK8J 44469097 IC50 = 12589.25 nM T32880 CK6O8G 44469099 IC50 = 19952.62 nM T32880 CADR40 44469101 IC50 = 25118.86 nM T32880 CBSI48 44469229 IC50 = 50118.72 nM T32880 C4U5RZ 44478798 IC50 = 79.43 nM T32880 CR21XB 44478800 IC50 = 158.49 nM T32880 CXOU61 44481885 IC50 = 1000 nM T32880 CCGJ52 44482164 IC50 = 79.43 nM T32880 CIK17O 44482165 IC50 = 398.11 nM T32880 CBL07Q 44482167 IC50 = 398.11 nM T32880 C42FTP 44482169 IC50 = 316.23 nM T32880 CT15UI 44514766 IC50 = 2.1 nM T32880 CW9OQ6 44568201 IC50 = 72 nM T32880 CF9QX3 44568202 IC50 > 40000 nM T32880 CEQL05 44568203 IC50 > 40000 nM T32880 CVWD50 44568204 IC50 = 1300 nM T32880 CX8B7T 44568205 IC50 = 72 nM T32880 CJ12AH 44568206 IC50 = 98 nM T32880 CC4B5M 44568207 IC50 = 33 nM T32880 CU63MS 44568208 IC50 = 27 nM T32880 C69PMH 44568247 IC50 > 40000 nM T32880 C1M3GY 44568248 IC50 = 400 nM T32880 C3JLM8 44568249 IC50 = 410 nM T32880 CF1E4K 44568250 IC50 = 2300 nM T32880 CX2YE1 44568251 IC50 = 21 nM T32880 CO50XS 44568252 IC50 = 11 nM T32880 C43BDN 44568281 IC50 = 4400 nM T32880 CXR89P 44568282 IC50 = 1700 nM T32880 CVID82 44568283 IC50 > 40000 nM T32880 C9JGC4 44568284 IC50 = 600 nM T32880 CG62EN 44568285 IC50 = 50 nM T32880 CK3SI1 44579681 IC50 = 570 nM T32880 CDAN35 44579682 IC50 = 290 nM T32880 CL9O6W 44579683 IC50 = 320 nM T32880 C1OTW6 44579684 IC50 = 330 nM T32880 CE1KX7 44579685 IC50 = 400 nM T32880 CZF4B8 44579687 IC50 > 40000 nM T32880 C8A3XZ 44579730 IC50 = 2820 nM T32880 C6LQ9S 44579731 IC50 = 5540 nM T32880 CFN49B 44579732 IC50 = 66 nM T32880 CMI6G8 44579733 IC50 > 40000 nM T32880 CBVI46 44579734 IC50 = 730 nM T32880 CVD1W3 44591754 IC50 = 512 nM T32880 C3OL2Y 44591755 IC50 = 230000 nM T32880 C71GJA 44819566 IC50 > 400000 nM T32880 CKD8A7 44819735 IC50 > 400000 nM T32880 C1VH6I 45482712 IC50 = 78000 nM T32880 C0W6RQ 45482725 IC50 > 1000000 nM T32880 C34LSI 45482742 IC50 > 1000000 nM T32880 CK2R4F 45482768 IC50 > 1000000 nM T32880 CIU6F7 45482769 IC50 > 1000000 nM T32880 CJ7OS3 45482772 IC50 = 538000 nM T32880 CX42JP 45482778 IC50 > 1000000 nM T32880 C2HL7F 45486323 IC50 = 21 nM T32880 CUMF70 46899605 IC50 > 100000 nM T32880 C2DBN5 46899607 IC50 > 100000 nM T32880 C3G4QK 46899609 IC50 > 100000 nM T32880 CLK96Z 46899763 IC50 > 100000 nM T32880 CBOM64 46899765 IC50 > 100000 nM T32880 CA56RL 49831102 IC50 = 3 nM T32880 CU63QR 49847377 IC50 = 0.2 nM T32880 CZT4I8 49847378 IC50 = 0.2 nM T32880 CA72PE 49847379 IC50 = 1.6 nM T32880 CC23YW 49847498 IC50 = 55 nM T32880 CJ7H2B 49847753 IC50 = 3.4 nM T32880 C4V7EW 49848258 IC50 = 0.8 nM T32880 C4E2YF 49848485 IC50 = 13700 nM T32880 CWP7L0 49848519 IC50 = 427 nM T32880 CV0PU1 49848649 IC50 = 27 nM T32880 CP8TS6 49848895 IC50 = 0.4 nM T32880 C9COF5 49848896 IC50 = 0.5 nM T32880 CK0B1G 49848897 IC50 = 0.2 nM T32880 CP61VJ 49849002 IC50 = 0.2 nM T32880 C42SBF 49849005 IC50 = 4.3 nM T32880 CBM62Z 49849007 IC50 = 0.4 nM T32880 C05SEW 49849008 IC50 = 0.2 nM T32880 C78SAD 49849115 IC50 = 4.1 nM T32880 CF64IJ 49849120 IC50 = 0.2 nM T32880 CC9EB4 49849122 IC50 = 0.5 nM T32880 C2ORV5 49849123 IC50 = 5.4 nM T32880 CUJ4D6 49870967 IC50 = 100 nM T32880 CX8Z0D 50899320 IC50 = 120 nM T32880 C0HCX8 50916282 IC50 > 400000 nM T32880 C2QG8V 53318573 IC50 = 50118.72 nM T32880 C90UET 53319897 IC50 > 100000 nM T32880 CX7O4F 53319898 IC50 = 79432.82 nM T32880 CS3E2L 53493245 IC50 = 0.7 nM T32880 CRFI05 53493908 IC50 = 0.7 nM T32880 C68OFC 54681699 IC50 = 46 nM T32880 CJO04Q 54739165 IC50 < 50 nM T32880 CT0UM5 54741100 IC50 = 1.5 nM T32880 C28RDF 54746913 IC50 = 4.9 nM T32880 C35JDV 54746961 IC50 = 5.3 nM T32880 CDL06K 54746964 IC50 = 3.1 nM T32880 CK3GC9 54746970 IC50 < 10 nM T32880 C7Q4WV 54747815 IC50 < 10 nM T32880 C2TB1P 54747831 IC50 < 10 nM T32880 CZWR91 54747907 IC50 = 4.1 nM T32880 CT6MD1 54749350 IC50 = 0.65 nM T32880 C9OG0S 54749369 IC50 = 3 nM T32880 CU7S6Y 56656421 IC50 = 50 nM T32880 CMR1X3 56684140 IC50 > 1000000 nM T32880 CE26XI 56684141 IC50 > 1000000 nM T32880 CL8N7V 56964909 IC50 > 1000000 nM T32880 C34DJP 57384236 IC50 = 1.1 nM T32880 CEOC15 57384237 IC50 = 2 nM T32880 CY50WC 57384238 IC50 = 2.3 nM T32880 C7S0ZR 57384239 IC50 = 1.5 nM T32880 C2XN1G 57384481 IC50 = 1.6 nM T32880 CR73IZ 57384482 IC50 = 0.8 nM T32880 CR2M5H 57384483 IC50 = 0.5 nM T32880 CQ72HI 57384749 IC50 = 4.7 nM T32880 C68KGE 57384750 IC50 = 1.9 nM T32880 CA57BP 57384999 IC50 = 0.5012 nM T32880 C5OGF6 57385246 IC50 = 640 nM T32880 CJ8N5F 57385491 IC50 = 680 nM T32880 C2HXQ4 57385492 IC50 = 6600 nM T32880 CFB30C 57385493 IC50 = 2200 nM T32880 CE8A9F 57385494 IC50 = 1200 nM T32880 CHJ8G2 57385495 IC50 = 1000 nM T32880 CMSP14 57385496 IC50 = 7800 nM T32880 CB2Y1U 57385733 IC50 = 370 nM T32880 CH15PS 57385734 IC50 = 2600 nM T32880 CE40ZB 57385735 IC50 = 790 nM T32880 CKO54M 57385736 IC50 > 50000 nM T32880 C5XDF4 57385737 IC50 > 50000 nM T32880 CR7UN3 57385738 IC50 > 50000 nM T32880 C85XSW 57386006 IC50 > 50000 nM T32880 CUL23K 57386007 IC50 = 3040 nM T32880 CJTC03 57386008 IC50 = 440 nM T32880 C9THS0 57386009 IC50 = 15300 nM T32880 CV34YJ 57386010 IC50 > 50000 nM T32880 C0RKZ2 57386011 IC50 > 50000 nM T32880 COI01S 57386263 IC50 > 50000 nM T32880 CUF1Y0 57386264 IC50 = 3100 nM T32880 C2BJT0 57386265 IC50 = 840 nM T32880 CVZ19P 57386266 IC50 = 4700 nM T32880 C3SUV6 57386267 IC50 = 6000 nM T32880 CF0TG4 57386268 IC50 = 3.8 nM T32880 CCR1X8 57386520 IC50 = 98 nM T32880 CQ6JG3 57386521 IC50 = 31 nM T32880 CVK29R 57386523 IC50 = 2.1 nM T32880 C9S8MU 57386524 IC50 = 4.3 nM T32880 CMC8H6 57386782 IC50 = 0.4 nM T32880 CCT5D4 57386783 IC50 = 0.4 nM T32880 CC30XZ 57386784 IC50 = 5 nM T32880 C79BXP 57386785 IC50 = 0.8 nM T32880 CM6DV7 57387028 IC50 = 1 nM T32880 C0GS4F 57387282 IC50 = 0.6 nM T32880 C0TL9C 57387283 IC50 = 2.8 nM T32880 CRV2P5 57387539 IC50 = 0.2 nM T32880 CAU3G9 57387540 IC50 = 0.2 nM T32880 CL2AO8 57387541 IC50 = 0.4 nM T32880 C0XWL8 57387542 IC50 = 0.4 nM T32880 CC4DK0 57387775 IC50 = 1 nM T32880 C8DB9I 57387776 IC50 = 0.8 nM T32880 C2LZ8G 57387778 IC50 = 1200 nM T32880 CUN9V6 57388001 IC50 = 0.7 nM T32880 CV7W0P 57742961 IC50 = 65 nM T32880 CS6Z2D 57983461 IC50 < 100 nM T32880 C2DIK6 57983520 IC50 < 100 nM T32880 CCB65L 59603622 IC50 = 280 nM T32880 COL70Z 67049505 IC50 = 820 nM T32880 CKG14F 67049582 IC50 = 2500 nM T32880 CFM6H7 67049587 IC50 = 220 nM T32880 C3CU9D 67049655 IC50 = 7100 nM T32880 C7AJ1U 67049671 IC50 = 450 nM T32880 C2DPK9 67049808 EC50 = 4700 nM T32880 C3AP9U 67049854 IC50 = 1200 nM T32880 CB3HX6 67049905 IC50 = 1600 nM T32880 C5PM7A 67049973 EC50 = 14000 nM T32880 C4VG9Q 67050041 IC50 = 210 nM T32880 C6UHR9 67050359 IC50 = 730 nM T32880 C92WSG 67050361 EC50 = 13000 nM T32880 C7LBD8 67050367 IC50 = 850 nM T32880 C1N9OY 67050409 EC50 = 5800 nM T32880 C8VM6P 67283460 IC50 = 94 nM T32880 C5RGQ2 68392546 IC50 = 100 nM T32880 CKX41C 69674161 IC50 = 110 nM T32880 C4VU7J 70688210 IC50 = 4.9 nM T32880 CO7H3Q 71133989 IC50 = 2.3 nM T32880 CL3HT1 71449736 IC50 = 6300 nM T32880 CJH86V 71451542 IC50 > 100000 nM T32880 CH38AO 71453382 IC50 > 100000 nM T32880 C2U4AQ 71458738 IC50 = 14200 nM T32880 C1DYB4 71477196 IC50 = 17 nM T32880 C9XGE6 71537024 IC50 < 10 nM T32880 CK34XF 71538425 IC50 < 20 nM T32880 CX74LQ 71545631 IC50 = 18400 nM T32880 CP6WO8 71717922 IC50 = 20 nM T32880 C7Y8SB 71748680 IC50 = 15.85 nM T32880 CC7M4D 72204345 IC50 > 10000 nM T32880 CM41RB 72204346 IC50 > 10000 nM T32880 C9A4KH 72204347 IC50 > 10000 nM T32880 C5MZ7R 72204348 IC50 = 158.49 nM T32880 CA2C1U 72204349 IC50 = 199.53 nM T32880 C4JZ6C 72204350 IC50 = 794.33 nM T32880 CZFG12 72204539 IC50 = 630.96 nM T32880 C8PM1E 72204540 IC50 = 2.512 nM T32880 CT4X1K 72204541 IC50 = 1 nM T32880 CV4EJ6 72204542 IC50 = 79.43 nM T32880 C3X0TL 72204543 IC50 = 1995.26 nM T32880 CZF7R4 72204544 IC50 = 1258.93 nM T32880 CK63AC 72204738 IC50 = 3981.07 nM T32880 CGE63D 72204739 IC50 = 1000 nM T32880 CGR92Y 72204740 IC50 = 3162.28 nM T32880 CIBE51 72204741 IC50 = 398.11 nM T32880 C2C5QX 72204742 IC50 = 3162.28 nM T32880 C4JAC1 72204743 IC50 = 501.19 nM T32880 C3WV2R 72204920 IC50 = 1995.26 nM T32880 C4MO3I 72204921 IC50 = 630.96 nM T32880 C1E4BJ 72204922 IC50 = 7.943 nM T32880 CI0R2O 72204923 IC50 = 31.62 nM T32880 C40BFH 72204924 IC50 = 3.981 nM T32880 CB1G4W 72204925 IC50 = 25.12 nM T32880 C81AQS 72205106 IC50 = 39.81 nM T32880 CK5MI2 72205107 IC50 = 5.012 nM T32880 C35SGD 72205108 IC50 = 15.85 nM T32880 CI0ON6 72205109 IC50 = 50.12 nM T32880 C6LM0T 72205110 IC50 > 10000 nM T32880 CWJG76 72737642 IC50 = 14 nM T32880 C2UFG1 73052701 IC50 = 39 nM T32880 CW64KE 73052704 IC50 = 49 nM T32880 CZU9X4 73052863 IC50 = 13 nM T32880 C4XIZ8 73349624 IC50 = 12589.25 nM T32880 C68RKH 76310231 IC50 = 8500 nM T32880 C89AEL 76310612 IC50 = 0.7 nM T32880 CO1EN3 76317452 IC50 = 278000 nM T32880 CPE6U2 76335997 IC50 > 500000 nM T32880 C7K3JM 89812866 IC50 = 9400 nM T32880 CHVP04 92042841 IC50 = 61 nM T32880 C6NUD0 118718072 IC50 = 41800 nM T32880 CUR10H 118978237 IC50 = 5.8 nM T32880 CI5X2G 118978277 IC50 = 11 nM T32880 CH7WL3 118978299 IC50 = 20 nM T32880 C43IWX 118978308 IC50 = 22.9 nM T32880 C2LBH1 118978321 IC50 = 66 nM T32880 CB3I9Z 118978325 IC50 = 9 nM T32880 CWH4I0 118978339 IC50 = 19 nM T32880 C6XD3H 118978341 IC50 = 5.4 nM T32880 CJE6K4 118978367 IC50 = 7.3 nM T32880 CDBK07 118981498 IC50 = 2.6 nM T32880 CB23LS 118981525 IC50 = 10 nM T32880 C9F6RL 118981536 IC50 = 6.9 nM T32880 CF1E6T 118981546 IC50 = 6.8 nM T32880 C1ABC5 118981554 IC50 = 4.3 nM T32880 CR05OQ 118981555 IC50 = 4.2 nM T32880 CE9U5L 118981600 IC50 = 4 nM T32880 CO5XH7 118981638 IC50 = 4.9 nM T32880 CV84HB 118981731 IC50 = 4.4 nM T32880 CM3VL0 118981967 IC50 = 21 nM T32880 CW89CV 118982285 IC50 = 6.5 nM T32880 C51RST 121245332 IC50 = 3.8 nM T32880 C2LI6C 121245745 IC50 = 8.5 nM T32880 C69YAB 121246676 IC50 = 0.9 nM T32880 C27WIY 121246694 IC50 = 27 nM T32880 C0E7BZ 121246784 IC50 = 1.9 nM T32880 CH4O3R 121246791 IC50 = 1 nM T32880 C71YRT 121246805 IC50 = 5.4 nM T32880 CJU6X7 121246821 IC50 = 2 nM T32880 C1X3HT 121246837 IC50 = 6.1 nM T32880 C2UY6K 121246848 IC50 = 4.2 nM T32880 C5E0SB 121246859 IC50 = 1.8 nM T32880 CE3P9G 121246864 IC50 = 1.5 nM T32880 C6BIK2 121269752 IC50 = 0.62 nM T32880 C6H2YQ 122383780 IC50 = 96000 nM T32880 CT2UZ4 125377518 IC50 > 100000 nM T32880 C5NR3C 129027150 IC50 = 13700 nM T32880 CWO0V4 135566826 IC50 = 2800 nM T32880 CV9J3Z 135737442 IC50 = 195000 nM T32880 CSCH32 135871166 IC50 = 27500 nM T32880 C3Q9KJ 135871167 IC50 = 81000 nM T32880 CJIK12 135871172 IC50 = 2200 nM T32880 CWI9V2 135871182 IC50 = 2100 nM T32880 C39VQA 135871218 IC50 = 700 nM T32880 CF5TV8 135871220 IC50 = 3800 nM T32880 CD6QM3 135871221 IC50 = 800 nM T32880 C2G7XC 135871222 IC50 = 24000 nM T32880 CAJ08Y 135871235 IC50 = 400 nM T32880 C42ISC 135871238 IC50 = 1400 nM T32880 C9DPJ0 135871283 IC50 = 2000 nM T32880 CYVH90 135895253 IC50 = 8 nM T32880 CT57ZH 136069450 IC50 = 0.2 nM T32880 CFT9R3 136069453 IC50 = 0.6 nM T32880 CRPQ42 136069494 IC50 = 2.5 nM T32880 CK8Z3V 136069521 IC50 = 5 nM T32880 CPY1B2 136069522 IC50 = 31 nM T32880 CX0OM4 136069523 IC50 = 11 nM T32880 C6EU4D 136069524 IC50 = 76 nM T32880 CQA2Z1 136069531 IC50 = 9.3 nM T32880 CCH31A 136069532 IC50 = 0.9 nM T32880 CH8GV7 136069561 IC50 = 14 nM T32880 CQ1FS4 136069563 IC50 = 3.9 nM T32880 C97REI 136074309 IC50 = 6000 nM T32880 CN6X7E 136074310 IC50 = 13500 nM T32880 CLV1R6 136074312 IC50 = 5700 nM T32880 CY3Z2V 136074313 IC50 = 1200 nM T32880 CEJ1M9 136074314 IC50 = 3000 nM T32880 CR5IM8 136074315 IC50 = 3400 nM T32880 CX02WY 136074316 IC50 = 2400 nM T32880 CICS75 136074317 IC50 = 7300 nM T32880 CS9C0Q 136074318 IC50 = 3900 nM T32880 CQTB32 136205798 IC50 = 1.1 nM T32880 CV8QP3 136205832 IC50 = 0.2 nM T32880 CB93EM 136205833 IC50 = 0.6 nM T32880 CV1C5I 136986966 IC50 = 2600 nM T32880 CJNU29 137083353 IC50 = 12 nM T32880 C0F8XB 137150345 IC50 = 20 nM T32880 C5UFR2 138319689 IC50 = 62.23 nM T32880 C7RYB5 141508724 IC50 = 248 nM T32880 CI1DE9 141508725 IC50 = 280.6 nM T32880 C5PN8T 141508727 IC50 = 228.2 nM T32880 CE36KV 141508729 IC50 = 418.3 nM T32880 C29GLS 141508732 IC50 = 278.3 nM T32880 C8SW9L 141508738 IC50 = 75.82 nM T32880 C5NJS7 141508739 IC50 = 61.08 nM T32880 C0Q5YG 141508741 IC50 = 308.3 nM T32880 C4QT0G 141508742 IC50 = 759.4 nM T32880 C2XB9I 141508745 IC50 = 418.7 nM T32880 CLK1B4 141508746 IC50 = 419.3 nM T32880 CJ9O3L 141508747 IC50 = 77 nM T32880 CV6N8B 141508748 IC50 = 271 nM T32880 C5SIU2 141508749 IC50 = 67.58 nM T32880 C2JRM3 141508751 IC50 = 231.1 nM T32880 C3WIL6 141508752 IC50 = 375.4 nM T32880 CK2ST8 141508755 IC50 = 418.3 nM T32880 CG0FL4 141508765 IC50 = 52.84 nM T32880 CN8EK0 141508769 IC50 = 579.7 nM T32880 CVMW03 141617793 EC50 = 17000 nM T32880 C2ML4K 141740991 IC50 = 1.9 nM T32880 C15DMN 145955244 IC50 = 16000 nM T32880 CK41QM 145957905 IC50 = 650 nM T32880 CWU6S2 145958372 IC50 = 6500 nM T32880 C7SIP1 145960425 IC50 = 801.4 nM T32880 CID5Y8 145960662 IC50 = 2165 nM T32880 CC9A8D 145960865 IC50 = 3594 nM T32880 CZDC15 145961128 IC50 = 853.8 nM T32880 CVZ8E9 145961326 IC50 = 3086 nM T32880 CEJ90L 145961795 IC50 = 853.8 nM T32880 C9R1SO 145961819 IC50 = 69 nM T32880 CB62WJ 145961830 IC50 = 6995 nM T32880 C4C6NP 145962038 IC50 = 995.8 nM T32880 C2Y7SM 145962118 IC50 = 1507 nM T32880 C6D5GL 145962572 IC50 = 608.2 nM T32880 CPO03J 145962836 IC50 = 5527 nM T32880 CJS57A 145962965 IC50 = 2291 nM T32880 C6YJ5R 155539215 IC50 = 905 nM T32880 COL30E 155540589 IC50 = 63 nM T32880 C5MFJ8 155548449 IC50 = 143 nM T32880 CN7H9B 155554391 IC50 = 70 nM T32880 C0GU8Y 155559177 IC50 > 25000 nM T32880 CG7R3L 155559901 IC50 = 4.8 nM T32880 CGU0A2 155563031 IC50 > 25000 nM T32880 C32NYC 155565735 IC50 > 25000 nM T32880 D07IOY 10365 IC50 = 6100 nM T32880 D08IZY 3080614 Ki = 8000 nM T32880 D08JSE 45102710 IC50 = 100 nM T32880 D0B2WZ 15331 IC50 > 100000 nM T32880 D0R6GQ 1198 IC50 > 10000000 nM T32880 D0WA3E 54685215 IC50 = 22 nM T32880 D0X5US 459617 IC50 = 15000 nM T51487 D02YPG 667484 EC50 = 11000 nM T51487 D06ZII 969472 Ki = 50.1 nM T51487 D07JVL 3016 Ki = 16 nM T51487 D0D5GD 3373 Ki = 3.3 nM T51487 D0F0YZ 4737 IC50 = 1000000 nM T51487 D0L9GG 2118 EC50 = 37 nM T51487 D0T1WN 5732 IC50 = 14 nM T51487 D0A5MC 11712649 IC50 = 330 nM T51487 D0CH7C 57336276 Ki = 985 nM T51487 D0HO2T 23581869 Ki = 0.5 nM T51487 D0S4JK 24771867 IC50 = 490 nM T51487 D0Z9HW 23630026 Ki = 0.5 nM T51487 C7SZ9E 613843 IC50 > 10000 nM T51487 C12NWX 2729103 IC50 > 10000 nM T51487 CO61AF 2820320 IC50 > 10000 nM T51487 C59BWK 2820473 IC50 = 470 nM T51487 C1Z6YU 9821389 Ki = 71 nM T51487 CCX58U 9865233 Ki = 0.73 nM T51487 C1VRB9 9951530 EC50 = 56 nM T51487 CPC3U1 9971547 Ki = 362 nM T51487 CUT5W8 9976743 EC50 = 53 nM T51487 CUSM85 10221761 Ki = 1.3 nM T51487 CBQ4R7 10905261 EC50 = 36 nM T51487 C15NXT 10926766 EC50 = 266 nM T51487 CK1S7J 10927005 EC50 = 107 nM T51487 CWK02D 10936672 EC50 = 135 nM T51487 C09PCZ 10971225 EC50 = 92 nM T51487 CG9Z6N 10991911 EC50 = 17 nM T51487 C7DVK8 11014215 EC50 = 120 nM T51487 CJB1V2 11035207 EC50 = 258 nM T51487 C31EGD 11036467 EC50 = 81 nM T51487 CBV36I 11047145 EC50 = 127 nM T51487 C8B7TF 11067772 EC50 = 95 nM T51487 CNSA17 11143256 EC50 = 136 nM T51487 CCU8G9 11526006 IC50 = 150 nM T51487 CWO70Q 11673720 Ki = 15 nM T51487 CX7G9K 11759134 EC50 = 170 nM T51487 CL4XD0 11783674 EC50 = 18 nM T51487 CB9U0F 11825216 EC50 = 28 nM T51487 CTI32Y 15680235 EC50 < 100 nM T51487 C8SR4O 25187292 IC50 = 46 nM T51487 C6DBS4 25187295 IC50 = 50 nM T51487 CF1B8A 25188671 IC50 = 50 nM T51487 CW97NA 44273000 IC50 = 1 nM T51487 C5KV7A 44364531 EC50 = 208 nM T51487 CZK75V 44364548 EC50 = 118 nM T51487 C0FN6W 44364725 EC50 = 2200 nM T51487 CYE1R8 44364726 EC50 = 41 nM T51487 CE8F3Y 44364734 EC50 = 303 nM T51487 COH5G6 44364735 EC50 = 544 nM T51487 C2VHW7 44364747 EC50 = 133 nM T51487 CZL2P0 44364907 EC50 = 69 nM T51487 CCX08E 44364918 EC50 = 93 nM T51487 C6D3BI 44560284 EC50 = 250 nM T51487 C6J0GP 44561356 IC50 = 580 nM T51487 C9UW4V 44561357 IC50 = 580 nM T51487 CZR6A5 44561358 IC50 > 10000 nM T51487 C4IF7B 44561386 IC50 = 1000 nM T51487 C3GZU0 44576235 EC50 = 11000 nM T51487 C63IYQ 51003493 IC50 = 134 nM T51487 CP8IG3 53317278 IC50 = 64 nM T51487 CP9I6O 53319883 IC50 = 74 nM T51487 CO6P3V 53320033 IC50 = 242 nM T51487 CCZ98L 53321188 IC50 = 67 nM T51487 C8MZR1 53322513 IC50 = 157 nM T51487 CTG2S9 53322514 IC50 > 3000 nM T51487 C29ARN 53323855 IC50 = 1 nM T51487 CBGD06 53323856 IC50 = 94 nM T51487 C9DJP1 53326435 IC50 = 64 nM T51487 CBO9L1 60194848 IC50 = 120000 nM T51487 CU83BZ 60194849 IC50 = 3800 nM T51487 CQ91VU 118278442 Ki = 140 nM T51487 CH0D4J 130439777 Ki = 850 nM T51487 C56XBU 130439778 Ki = 55000 nM T51487 C9N8LW 130439889 Ki = 542 nM T51487 C89LNZ 136118605 IC50 = 479 nM T51487 D06SOQ 6918451 Ki = 0.88 nM T51487 D09IHE 6918583 Ki = 0.8 nM T51487 D0E7PY 11624499 Ki = 174 nM T51487 D0M4CP 5081 EC50 = 1.1 nM T51487 D0O9MG 5311203 Ki = 17 nM T52921 D04CRN 54841 IC50 > 5000 nM T52921 D0CS2F 3955 Ki > 10000 nM T52921 D0PG8O 5360515 Ki > 10000 nM T52921 D0U5FS 3396 Ki = 500 nM T52921 D03TBJ 11848225 Ki = 0.9 nM T52921 D0G2XE 6918468 IC50 = 2200 nM T52921 D0W4YO 16131448 Ki = 0.04898 nM T52921 D0M1YN 5311194 Ki = 0.403 nM T52921 D00ACC 9844019 Ki = 1.12 nM T52921 D08AWI 11430856 Ki > 2000 nM T52921 CBGO28 70419 Ki = 11 nM T52921 C3HB4V 416359 IC50 = 200 nM T52921 CQ6MW0 3655995 EC50 = 174 nM T52921 CLW4B1 5311340 Ki = 8.2 nM T52921 CD49UV 9797246 Ki = 133 nM T52921 CNO0W4 9799433 Ki = 5.22 nM T52921 CYR3O0 9802205 Ki = 50.7 nM T52921 CPG57N 9803475 Ki = 12.9 nM T52921 CX7DO4 9806799 Ki = 4.05 nM T52921 CK6GR9 9816910 IC50 > 5000 nM T52921 CE6NF9 9823363 IC50 = 1.3 nM T52921 C6LGX9 9824268 Ki = 82.4 nM T52921 C7TDX2 9824313 Ki = 46.7 nM T52921 C70KEP 9824565 Ki = 0.5 nM T52921 C06LIG 9825723 Ki = 2.3 nM T52921 CPK4X7 9836463 Ki = 1054 nM T52921 C6Y7NA 9844540 Ki = 2 nM T52921 C0F9RX 9845765 Ki = 7 nM T52921 C8M4HT 9846747 Ki = 2.2 nM T52921 CE2YQ9 9848110 Ki = 2 nM T52921 CKD2H4 9848990 Ki = 77 nM T52921 CLQ6Z8 9866158 Ki = 0.5 nM T52921 CEO0M2 9880173 Ki = 414 nM T52921 CPYK08 9887195 IC50 = 820 nM T52921 CV2G7M 9889948 Ki = 11.8 nM T52921 C1VM4H 9902583 Ki = 692 nM T52921 C5BC4P 9902874 Ki = 39 nM T52921 CX3CM8 9905428 Ki = 1.39 nM T52921 C2TE5X 9922658 Ki = 10 nM T52921 C4NJ0W 9923726 Ki = 125 nM T52921 CIUE54 9924406 Ki = 5.4 nM T52921 C5HN0J 9925137 Ki = 1.1 nM T52921 CZT2J0 9927928 Ki = 18.66 nM T52921 C2U8XH 9932834 Ki = 3.4 nM T52921 C9MK3B 9934232 Ki = 6.8 nM T52921 CUBQ95 9937777 Ki = 2.25 nM T52921 C4FD7V 9947044 Ki = 1.4 nM T52921 CG9ER5 9947155 Ki = 2297 nM T52921 COFT18 9951673 Ki = 4 nM T52921 C3GXH0 9954388 Ki = 5.6 nM T52921 CT8C2X 9958643 Ki = 1.8 nM T52921 CE3CJ4 9969865 Ki = 5102 nM T52921 CAGL19 9997843 Ki = 0.7 nM T52921 CL9QS0 10004950 IC50 = 19 nM T52921 C4N8YE 10020165 Ki = 6 nM T52921 C25DYT 10022859 Ki = 0.52 nM T52921 CFOK60 10042904 Ki = 3.96 nM T52921 CC60VS 10052051 Ki = 505 nM T52921 CV1OU6 10109140 Ki = 4.4 nM T52921 C7YCF1 10109899 Ki = 1 nM T52921 CJNE19 10110916 Ki = 225 nM T52921 C76MVA 10111186 Ki > 10000 nM T52921 CWEC34 10114637 Ki = 4461 nM T52921 C40BMF 10133108 Ki = 51 nM T52921 C2WZ9G 10133332 Ki = 1259 nM T52921 CP1SO7 10134077 Ki = 11 nM T52921 CEG0M4 10134217 Ki = 357 nM T52921 C3ZTU0 10137134 Ki = 225 nM T52921 C83KDV 10137876 Ki = 7.4 nM T52921 C8E9KP 10139672 Ki = 41 nM T52921 CQGE97 10150001 Ki = 94 nM T52921 C76SOW 10150260 Ki = 37 nM T52921 CRC46J 10154739 Ki = 634 nM T52921 CKN3A8 10154848 Ki = 410 nM T52921 CFIL01 10155966 Ki = 2.3 nM T52921 CIO6U3 10156336 Ki = 1239 nM T52921 CP53IB 10156591 Ki = 0.4 nM T52921 CI1U4Z 10156821 Ki = 7.5 nM T52921 CTO0N5 10158555 Ki = 31 nM T52921 CG51TX 10159203 Ki = 11 nM T52921 CWM2X6 10160920 Ki = 18 nM T52921 CB57JZ 10171862 Ki = 78 nM T52921 CDV15J 10172398 Ki = 58 nM T52921 CJN21A 10178311 Ki = 184 nM T52921 CHN4G6 10178563 Ki = 824 nM T52921 C5RO6K 10182346 Ki = 7114 nM T52921 CNZL85 10193971 Ki = 347 nM T52921 CN79QX 10194236 Ki = 31 nM T52921 CWC8L1 10199945 IC50 = 2.5 nM T52921 C12NGT 10199984 Ki = 3454 nM T52921 CH40KY 10202108 Ki = 437 nM T52921 CV1T7R 10202241 Ki > 10000 nM T52921 CYB0H9 10221539 IC50 = 3.3 nM T52921 CM27FK 10225083 Ki = 2 nM T52921 CZ0C5T 10252647 Ki = 66 nM T52921 CH54KF 10260917 EC50 = 0.1585 nM T52921 C8PL7B 10274330 Ki = 33 nM T52921 CR1HX2 10275388 Ki = 4358 nM T52921 CSO8D7 10276738 Ki = 0.38 nM T52921 CDP01X 10286440 Ki = 570 nM T52921 C1FE9H 10286996 Ki = 105 nM T52921 CJ14VU 10291377 Ki = 16 nM T52921 C61OKS 10292091 Ki = 111 nM T52921 CV0T3H 10301207 Ki = 1 nM T52921 C1ENR2 10323169 Ki = 2.3 nM T52921 CD09RQ 10338496 Ki = 110 nM T52921 C0G7RF 10362733 Ki = 4544 nM T52921 C59JAP 10363496 Ki = 2.2 nM T52921 CAYF18 10385808 Ki = 2.6 nM T52921 C95EWP 10395965 Ki = 27 nM T52921 CWK4O1 10406239 Ki = 0.1 nM T52921 CTA8Q0 10407144 Ki = 19.6 nM T52921 CX4TS2 10413540 Ki = 78 nM T52921 CYHC38 10430819 Ki = 0.5495 nM T52921 CZP0C7 10441529 EC50 = 0.302 nM T52921 CZ6I9V 10451761 IC50 = 6.8 nM T52921 CKMN08 10475466 Ki = 4.6 nM T52921 C1DI7F 10500922 Ki = 218 nM T52921 C90DEM 10504545 Ki = 6.8 nM T52921 CDK8W2 10548749 Ki = 5.8 nM T52921 C54EOA 10572810 Ki = 7.3 nM T52921 CD9JB5 10574643 Ki = 2.8 nM T52921 CQ74CO 10593778 Ki = 2.5 nM T52921 CZQ4J6 10596013 Ki = 79.9 nM T52921 CHV5D1 10601891 Ki = 15 nM T52921 CS84IW 10618605 Ki = 2.5 nM T52921 CPC52U 10646744 Ki = 7.2 nM T52921 C10KTE 10646745 Ki = 8.5 nM T52921 CH16SQ 10668903 Ki = 85.6 nM T52921 CMT48G 10669669 Ki = 20.4 nM T52921 CF7SX5 10669670 Ki = 13.2 nM T52921 CP25HJ 10669671 Ki = 37.3 nM T52921 CHC1I4 10697286 Ki = 15.3 nM T52921 C2RN9F 10713623 Ki = 10.2 nM T52921 C8XB3K 10714523 Ki = 1.4 nM T52921 CY36JZ 10715725 Ki = 88.5 nM T52921 CFH5N0 10715726 Ki = 121.2 nM T52921 C48PSE 10718869 Ki = 2.6 nM T52921 CN05WO 10763594 Ki = 0.39 nM T52921 CBC6U3 10765154 Ki = 1.8 nM T52921 CXF9R4 10766007 Ki = 1.8 nM T52921 CDJP34 10783436 IC50 = 6.8 nM T52921 CTR2I0 10788833 Ki = 6.5 nM T52921 CQS8K6 10789513 Ki = 1.8 nM T52921 C9SN6H 10831914 Ki = 369.3 nM T52921 CS3Y4G 10832076 IC50 = 5.9 nM T52921 CMVI50 10832445 Ki = 6.3 nM T52921 CPG23C 10836379 Ki = 20.7 nM T52921 C4IT2B 10837001 Ki = 3.3 nM T52921 C2QIL3 10876990 EC50 = 1 nM T52921 CWJL70 10905740 IC50 = 434 nM T52921 C4TSV6 10927662 Ki = 0.5248 nM T52921 C1TSN4 10928037 Ki = 0.7762 nM T52921 CT5UO7 10937810 Ki = 2.188 nM T52921 CU09AV 10937901 IC50 = 38 nM T52921 CVP6D3 10942284 EC50 = 0.2692 nM T52921 CN7XS4 10948527 IC50 = 340 nM T52921 CSLT97 10949380 IC50 = 283 nM T52921 C9FYG3 10950562 Ki = 1.66 nM T52921 CHK23I 10961428 Ki = 1.66 nM T52921 C2HP7F 10981761 IC50 = 758 nM T52921 C78FTE 10986100 EC50 = 63.1 nM T52921 C8Q6YE 11004121 Ki = 0.4467 nM T52921 CIR4E5 11007758 EC50 = 134.9 nM T52921 C0R2DW 11007770 EC50 = 31.62 nM T52921 C3V7LT 11014751 Ki = 0.6457 nM T52921 CY0S2I 11029698 EC50 = 257.04 nM T52921 CRP95V 11051525 EC50 = 0.2512 nM T52921 C9Z7BY 11115933 EC50 = 1.413 nM T52921 CDU0E5 11123873 Ki = 2.089 nM T52921 CU6PV0 11143820 IC50 = 97 nM T52921 C7HM0O 11152739 Ki = 3.5 nM T52921 C26ENL 11164004 Ki = 15.6 nM T52921 C62WBJ 11165726 Ki = 135 nM T52921 C4COM2 11170657 Ki = 0.05 nM T52921 C3TW2O 11187225 Ki = 4.5 nM T52921 C6EWJ9 11188910 Ki = 4.4 nM T52921 CUBX19 11189444 IC50 > 10000 nM T52921 CTKF50 11191683 IC50 = 5.5 nM T52921 CS5ET8 11212373 IC50 > 10000 nM T52921 C26MVG 11223982 IC50 > 10000 nM T52921 C4QT5Y 11233481 Ki = 15.5 nM T52921 CW1O5V 11256620 Ki = 12 nM T52921 CPBZ36 11274537 Ki > 5000 nM T52921 C4FRH7 11315651 Ki = 1.64 nM T52921 C5DBK1 11326750 Ki = 11 nM T52921 CJM7R5 11327115 Ki = 253 nM T52921 CW7SN4 11329662 Ki = 0.5012 nM T52921 CS1W7V 11338717 IC50 > 10000 nM T52921 CY0SV8 11349939 Ki > 10000 nM T52921 C6UZF7 11371415 Ki = 11.7 nM T52921 C4BZ1C 11372427 Ki = 4.3 nM T52921 CQC4G5 11372671 IC50 = 6150 nM T52921 CT6Z0B 11393860 Ki = 29.3 nM T52921 CGO58L 11406629 IC50 = 3700 nM T52921 CBJ0X5 11407510 IC50 > 10000 nM T52921 CU5GO6 11411841 IC50 = 25.2 nM T52921 CW0E4L 11418847 IC50 > 10000 nM T52921 C9KV1U 11451023 Ki = 5.64 nM T52921 C7UDE8 11461888 Ki = 7.49 nM T52921 CF6DQ2 11462727 Ki = 10 nM T52921 CKIQ83 11463791 IC50 > 10000 nM T52921 CC9TX5 11464294 IC50 > 10000 nM T52921 CMU9K5 11464846 Ki = 0.336 nM T52921 C3BA5F 11480038 Ki = 72 nM T52921 CVQ70S 11480201 Ki = 0.04 nM T52921 C41MEV 11511090 IC50 = 0.22 nM T52921 CZ4OM7 11516508 Ki = 2.2 nM T52921 C2N3BS 11523928 IC50 > 1000 nM T52921 CJE45X 11523929 IC50 > 1000 nM T52921 CL1O0H 11523972 IC50 = 350 nM T52921 CQ30PM 11525624 IC50 = 42 nM T52921 C8TZ9G 11544654 IC50 = 32 nM T52921 CS0B4G 11544795 Ki = 2.4 nM T52921 C3DG8U 11552010 Ki = 10.2 nM T52921 C10BUF 11559590 IC50 > 1000 nM T52921 C5ZR9W 11559820 IC50 = 540 nM T52921 CG6UM9 11561261 IC50 > 1000 nM T52921 CRX48F 11581029 Ki = 18.9 nM T52921 CA35LD 11583008 Ki = 4.6 nM T52921 CVA8L6 11583016 IC50 = 4 nM T52921 C1WBQ5 11597677 IC50 = 83 nM T52921 CY72UC 11602409 Ki = 8.5 nM T52921 C0AOU4 11603249 IC50 = 730 nM T52921 C38FTP 11619363 IC50 = 12 nM T52921 C8RKH0 11619553 IC50 = 8.3 nM T52921 C9WMX4 11624970 Ki = 29.8 nM T52921 C34OQC 11626062 Ki = 1.74 nM T52921 CF6R4S 11632761 IC50 > 1000 nM T52921 C4ZD1X 11633324 IC50 = 7.5 nM T52921 CIY0O4 11639705 IC50 > 1000 nM T52921 CFV5Q1 11661648 IC50 > 1000 nM T52921 CPN46U 11676849 IC50 = 580 nM T52921 C4ULQ7 11710187 IC50 = 23 nM T52921 CE0D1U 11743914 Ki = 116 nM T52921 CV8CF3 11749578 IC50 > 10000 nM T52921 CFRY36 11757207 Ki = 15 nM T52921 CED7I5 11761926 Ki = 0.6607 nM T52921 CCY92E 11768467 EC50 = 7.244 nM T52921 CG9HW8 11795019 Ki = 2.9 nM T52921 CN9M8E 11811722 IC50 = 2420 nM T52921 C8UE5W 11826819 Ki = 2.138 nM T52921 CS7W2V 11848793 Ki = 1.7 nM T52921 CJ34HP 11956520 Ki = 0.19 nM T52921 CA5ZX7 11956918 Ki = 9.4 nM T52921 C14RWU 11967729 EC50 = 10.96 nM T52921 CP1AZ0 11967746 EC50 = 26.3 nM T52921 CF01LM 12986253 Ki = 1.9 nM T52921 C63ASY 12986256 Ki = 120 nM T52921 CAW1M2 15512228 Ki = 0.52 nM T52921 C30CHU 15512229 Ki = 0.2512 nM T52921 C9B5OD 15512233 Ki = 39.81 nM T52921 CX6H8V 15512234 Ki = 1.259 nM T52921 CC5X0L 15512235 Ki = 3.981 nM T52921 CG0CS6 15512236 Ki = 15.85 nM T52921 C53KRM 15512237 Ki = 0.3162 nM T52921 CLA5K8 15512238 Ki = 3.981 nM T52921 C4I5TU 15512239 Ki = 10 nM T52921 CSX74V 15512240 Ki = 1.585 nM T52921 CET25R 15512241 Ki = 5.012 nM T52921 C23GHP 15512242 Ki = 100 nM T52921 C7CNY1 15512243 Ki = 1.585 nM T52921 CZA4J8 15541261 Ki = 23 nM T52921 CE18TP 15586319 Ki = 810 nM T52921 CD7K0Y 15965865 IC50 = 6000 nM T52921 CHN45W 15982524 IC50 = 510 nM T52921 CRX3U8 15982526 IC50 = 680 nM T52921 C6DW5M 15982528 IC50 > 10000 nM T52921 C7Z8OD 15982529 IC50 = 7400 nM T52921 CHO67K 15982530 IC50 = 600 nM T52921 C3B8AG 15982657 IC50 = 880 nM T52921 C4W6CK 15982658 IC50 = 140 nM T52921 CLWI08 15982659 IC50 = 10000 nM T52921 CV1G7O 15982660 IC50 = 83 nM T52921 CG3L8Z 15982661 IC50 = 120 nM T52921 CN64AP 15982791 IC50 = 320 nM T52921 C7KXO3 15982794 IC50 > 10000 nM T52921 CB1CR0 15982795 IC50 = 100 nM T52921 C0PKF1 15982796 IC50 = 10000 nM T52921 C3HL5F 15982797 IC50 = 820 nM T52921 CJY21D 15982932 IC50 > 10000 nM T52921 CJ6W1T 15982933 IC50 < 10000 nM T52921 CK97VS 15982935 IC50 = 250 nM T52921 C8TQ4B 15982937 IC50 = 900 nM T52921 C1PB8H 15982938 IC50 = 1120 nM T52921 CS46QG 15983062 IC50 = 800 nM T52921 CXJ61F 15983063 IC50 = 3600 nM T52921 CIG32A 15983065 IC50 = 10000 nM T52921 CG96OQ 15983067 IC50 = 2750 nM T52921 CA5GL7 16007142 Ki = 4 nM T52921 CDR71P 16043240 IC50 > 10000 nM T52921 C4H2NO 16061455 Ki = 6 nM T52921 C08RXS 16665915 Ki = 800 nM T52921 CS9FW1 16665917 Ki = 290 nM T52921 C1LX0I 16665918 Ki = 18 nM T52921 C6W9BJ 16733371 Ki = 6 nM T52921 C4ORI6 16739256 Ki = 15.1 nM T52921 C1MFJ2 16747695 Ki = 4.1 nM T52921 CG84KV 17858339 IC50 = 320 nM T52921 CWXD07 17858448 IC50 = 4.7 nM T52921 C8AZW7 18441735 IC50 = 15000 nM T52921 C1Y9FT 18782352 Ki = 0.9 nM T52921 CYUG80 18782376 Ki = 10.8 nM T52921 C46DPT 18782378 Ki = 2 nM T52921 C73DWV 18782384 Ki = 14.5 nM T52921 CHAI36 22272877 IC50 = 17 nM T52921 C5VSD6 22272900 IC50 = 17 nM T52921 CB5DY1 22272974 IC50 = 3.9 nM T52921 C1NU9M 22273044 IC50 = 2.1 nM T52921 CX3JY4 22273116 IC50 = 120 nM T52921 CRZ72H 22273255 IC50 = 3100 nM T52921 C8DF5U 22558157 Ki = 12 nM T52921 C1R5PV 22562132 Ki = 5670 nM T52921 CJ8OB0 22562135 Ki = 3592 nM T52921 C0GKU4 22562137 Ki = 20.4 nM T52921 CJ86RS 22725091 Ki = 10 nM T52921 CL7X2U 23383556 Ki = 0.4 nM T52921 COHN67 23383564 Ki = 0.5 nM T52921 C46ZSX 23542099 IC50 = 34 nM T52921 CVLY78 23542106 IC50 = 82 nM T52921 CB9MC8 24735827 Ki = 119 nM T52921 CWP85S 24776395 Ki = 3.1 nM T52921 CVD48X 24776396 Ki = 186 nM T52921 C3WDL8 24776397 Ki = 8.9 nM T52921 CXL4R0 24776398 Ki = 21 nM T52921 CR9I1S 24776399 Ki = 395 nM T52921 CQDJ35 24776400 Ki = 147 nM T52921 C6CX0Z 24776401 Ki = 6.6 nM T52921 CJH18I 24776402 Ki = 12 nM T52921 C27SGI 24776403 Ki = 26 nM T52921 CV5IG2 24776404 Ki = 51 nM T52921 CQ70IW 24776405 Ki = 81 nM T52921 CQ2P5J 24776406 Ki = 136 nM T52921 CYIV42 24776407 Ki = 4.7 nM T52921 CWB06Z 24776408 Ki = 23 nM T52921 C36WQO 24776409 Ki = 42 nM T52921 CUP2C6 24776410 Ki = 90 nM T52921 CC3W7E 24776411 Ki = 130 nM T52921 C3N6GE 24776412 Ki = 65 nM T52921 C2M6BR 24776413 Ki = 92 nM T52921 C8SXV9 24799146 Ki = 180 nM T52921 C1S2NC 24799325 Ki = 104 nM T52921 CLAU56 24799509 Ki = 100 nM T52921 C2VHP0 24799848 Ki = 545 nM T52921 C26ZYM 24800015 Ki = 260 nM T52921 CWV5F4 24800016 Ki = 740 nM T52921 CS01RL 24800107 Ki = 2.1 nM T52921 CL2WB0 24800108 Ki = 0.0858 nM T52921 CY89FP 24800188 Ki = 186 nM T52921 C13MJI 24822630 EC50 = 0.1 nM T52921 C6TWH4 24824635 EC50 = 88 nM T52921 CYM02E 24847114 IC50 = 15 nM T52921 C9O5NZ 24857819 IC50 = 0.65 nM T52921 CN0T1F 24857820 IC50 = 0.66 nM T52921 CS5D1K 24882570 IC50 = 0.033 nM T52921 CQ63PM 24894425 Ki = 17 nM T52921 C2EQR6 24894426 Ki = 0.47 nM T52921 CT9EZ4 24894428 Ki = 1.1 nM T52921 CN1E8M 24894430 Ki = 30 nM T52921 C9USO6 24894431 Ki = 58 nM T52921 C4IDR3 24894531 Ki = 11 nM T52921 CA8E4J 24894533 Ki = 21 nM T52921 C2AU5Y 24894647 Ki = 20 nM T52921 C8JL9I 24894652 Ki = 49 nM T52921 C6AZ9P 24894653 Ki = 25 nM T52921 CC6F9D 24894783 Ki = 51 nM T52921 CDLW86 25001412 Ki = 0.7244 nM T52921 CBIU48 25077447 EC50 = 4.37 nM T52921 CFB8G1 25077910 EC50 = 25 nM T52921 CHWB32 25082025 EC50 = 156 nM T52921 C2FPI9 25084159 EC50 = 22.3 nM T52921 C6HL3Q 25089553 EC50 = 0.1349 nM T52921 CP56DF 25089995 IC50 = 0.471 nM T52921 CF6RA5 25190572 Ki = 84 nM T52921 CPK5D7 25190573 Ki = 34 nM T52921 CON62K 25190574 Ki = 57 nM T52921 C6S3WN 25190575 Ki = 83 nM T52921 CF15AH 25190576 Ki = 53 nM T52921 CBN1Q0 25190577 Ki = 89 nM T52921 CKB72D 25190578 Ki = 234 nM T52921 CZR78G 25190579 Ki = 203 nM T52921 CF2JK0 25190580 Ki = 48.7 nM T52921 CE4R2X 25190581 Ki = 56 nM T52921 CYC6S0 25190582 Ki = 19.5 nM T52921 CE61QB 25190583 Ki = 18.5 nM T52921 C9V8MS 25190584 Ki = 26 nM T52921 C3UV5M 25190585 Ki = 47.8 nM T52921 CKFI42 25190586 Ki = 2.1 nM T52921 C5UQX3 25190587 Ki = 2.55 nM T52921 C5J2WE 25190588 Ki = 8.65 nM T52921 CX84WI 25190589 Ki = 5 nM T52921 C5RUI9 25190590 Ki = 3.5 nM T52921 CQY69C 25190591 Ki = 3.7 nM T52921 C8SEQ2 25190592 Ki = 12.1 nM T52921 C5BS7N 25190593 Ki = 2.15 nM T52921 CE19OU 25190594 Ki = 2.75 nM T52921 CP5ID6 25190595 Ki = 3.8 nM T52921 CO8E4G 25190596 Ki = 3.2 nM T52921 CX87HD 25190597 Ki = 8 nM T52921 CY6CV1 25190598 Ki = 2.3 nM T52921 CW5UP9 25190599 Ki = 0.8 nM T52921 C1C8VK 25190600 Ki = 0.7 nM T52921 CL7Q2F 25190601 Ki = 0.7 nM T52921 CD0H5U 25190602 Ki = 0.5 nM T52921 C8OWC0 25190603 Ki = 0.5 nM T52921 CH06YU 25190604 Ki = 0.6 nM T52921 CEJ25L 25190605 Ki = 0.5 nM T52921 CXD5R8 25190606 Ki = 1 nM T52921 CU6W8O 25190607 Ki = 5.4 nM T52921 CWJB54 25190608 Ki = 4.5 nM T52921 CMHS48 25190609 Ki = 1.7 nM T52921 CBL9S4 25190610 Ki = 2.1 nM T52921 CZ8Y6L 25190611 Ki = 1.6 nM T52921 CL9SN6 25190612 Ki = 1.4 nM T52921 C1MGY3 25190613 Ki = 0.9 nM T52921 CB1G6M 25190614 Ki = 0.9 nM T52921 CJLH27 25190615 Ki = 1 nM T52921 COE65V 25190616 Ki = 0.9 nM T52921 C30VGA 25190617 Ki = 1.5 nM T52921 CO7IV2 25190618 Ki = 0.8 nM T52921 C8Q7WV 25190619 Ki = 0.5 nM T52921 C0G4RJ 25190620 Ki = 6.7 nM T52921 C7X4IV 25190621 Ki = 1.4 nM T52921 CXG8O3 25190622 Ki = 0.5 nM T52921 CD5F6A 25190623 Ki = 0.4 nM T52921 CFUD47 25190624 Ki = 1.3 nM T52921 C15LIW 25190625 Ki = 0.7 nM T52921 C3LEW8 25190626 Ki = 3.6 nM T52921 CIDV61 25190627 Ki = 15.9 nM T52921 CAGS39 25190628 Ki = 1.8 nM T52921 CDS2E6 25190629 Ki = 0.6 nM T52921 CPW19O 25190630 Ki = 12.2 nM T52921 C0SBV7 25207946 Ki = 0.63 nM T52921 C21OJF 25207948 Ki = 0.3 nM T52921 C0P6CS 25207950 Ki = 0.18 nM T52921 CN9I8E 25208095 Ki = 0.2 nM T52921 C5OA1N 25208097 EC50 = 0.02512 nM T52921 C59IKP 25208099 Ki = 0.24 nM T52921 CUNA84 25208101 Ki = 0.15 nM T52921 C2WIG0 25208245 Ki = 0.22 nM T52921 CE4BI6 25208247 Ki = 1.7 nM T52921 CKNE16 25208249 Ki = 0.53 nM T52921 CB04CU 25235412 Ki = 20 nM T52921 CL2Z7J 42629117 EC50 = 14 nM T52921 CWJ2E3 43406622 IC50 > 1000 nM T52921 C49YRK 44143406 IC50 = 350 nM T52921 C3YMQ1 44143407 IC50 = 150 nM T52921 CBFR50 44143408 IC50 = 150 nM T52921 C4BOI0 44143409 IC50 = 75 nM T52921 CRL9K5 44143410 IC50 > 1000 nM T52921 CB4O2Y 44143411 IC50 > 1000 nM T52921 C0JS3Q 44143412 IC50 = 560 nM T52921 C6U7HP 44143413 IC50 = 28 nM T52921 C1TSC2 44143414 IC50 = 530 nM T52921 CAB3T9 44143415 IC50 = 37 nM T52921 CD26LJ 44143416 IC50 > 1000 nM T52921 CG3PW7 44143417 IC50 = 61 nM T52921 CB94OV 44143418 IC50 = 11 nM T52921 COP5W8 44143419 IC50 = 4 nM T52921 CY26BG 44143420 IC50 = 67 nM T52921 C8WLP6 44143421 IC50 = 270 nM T52921 C3S1PL 44143422 IC50 = 13 nM T52921 C05AWH 44143423 IC50 = 33 nM T52921 C4D0YQ 44143424 IC50 = 36 nM T52921 C5CR3I 44143425 IC50 = 72 nM T52921 CQE5U4 44143426 IC50 = 8.2 nM T52921 CZR49E 44143427 IC50 = 7.1 nM T52921 C63RXB 44143428 IC50 = 2.5 nM T52921 C8OH4S 44143429 IC50 = 4.5 nM T52921 CTE6S1 44143430 IC50 = 1.2 nM T52921 CL57VS 44143431 IC50 = 0.52 nM T52921 C2C5QW 44143432 IC50 = 0.72 nM T52921 C6GDL8 44143433 IC50 = 0.81 nM T52921 C3BNV0 44143434 IC50 = 5.7 nM T52921 CXV0B8 44143435 IC50 = 2 nM T52921 CN7HE0 44143436 IC50 = 38 nM T52921 C9CJN0 44143437 IC50 = 0.8 nM T52921 C6INT4 44143438 IC50 = 2.9 nM T52921 CJ46YA 44143439 IC50 = 23 nM T52921 CZ15CE 44143440 IC50 = 630 nM T52921 C0KB7Y 44143441 IC50 = 61 nM T52921 C3RF4I 44143442 IC50 = 27 nM T52921 CE20LQ 44143444 IC50 = 22 nM T52921 CFH9T2 44143445 IC50 = 21 nM T52921 C5NZM3 44143446 IC50 = 1.1 nM T52921 CGSW03 44143448 IC50 = 1.1 nM T52921 CBWD06 44143449 IC50 = 2.1 nM T52921 C2ST5N 44143450 IC50 = 1.4 nM T52921 CF4V5K 44143451 IC50 = 1 nM T52921 CL3R6D 44143452 IC50 = 4 nM T52921 C8IG1V 44143453 IC50 = 0.9 nM T52921 C2Q3DE 44143454 IC50 = 3.7 nM T52921 CZX75A 44143455 IC50 = 0.91 nM T52921 C02YJQ 44143456 IC50 = 1.1 nM T52921 CZV0C7 44143457 IC50 = 1.8 nM T52921 CPQ25W 44181744 Ki = 5 nM T52921 C2XE7Y 44189733 IC50 = 2.3 nM T52921 CGA8R1 44189735 IC50 = 1.9 nM T52921 C50FOG 44189834 IC50 = 2.3 nM T52921 CC63QX 44247589 Ki = 7 nM T52921 CP8Q5B 44248550 Ki = 7 nM T52921 CZNM65 44248674 Ki = 1 nM T52921 CIJF67 44248788 Ki = 272 nM T52921 C9G8KT 44248789 Ki = 34 nM T52921 C9JBR1 44248790 Ki = 22 nM T52921 C5YV0D 44248791 Ki = 14 nM T52921 C1CZ3M 44248792 Ki = 24 nM T52921 CDG15Z 44248915 Ki = 23 nM T52921 C5I7YZ 44248916 Ki = 29 nM T52921 C5T9AP 44248917 Ki = 467 nM T52921 CAY83B 44248918 Ki = 18 nM T52921 CL61MJ 44248919 Ki = 25 nM T52921 C2FLP9 44248920 Ki = 10 nM T52921 C6Q5ZF 44249045 Ki = 9 nM T52921 C0HWG8 44249046 Ki = 9 nM T52921 CHLS96 44249047 Ki = 5 nM T52921 CO4EA3 44249048 Ki = 69 nM T52921 CW6P4Y 44276782 Ki = 89 nM T52921 C9AF6B 44297435 Ki = 28.7 nM T52921 CNP5W1 44297519 Ki = 786 nM T52921 C52MGY 44297539 Ki = 0.49 nM T52921 C9UY4E 44297697 Ki = 535 nM T52921 C8F1ST 44297727 Ki = 189 nM T52921 C7ZYM4 44299404 Ki > 10000 nM T52921 CK6IY4 44315305 Ki = 10 nM T52921 CQ0OK5 44327446 EC50 = 0.7586 nM T52921 CAS38O 44332117 Ki = 4.67 nM T52921 CGZ9N2 44336905 Ki = 191 nM T52921 CYMH75 44337108 Ki = 420 nM T52921 CJ0I6Q 44337123 Ki = 64 nM T52921 CPOX86 44337129 Ki = 7222 nM T52921 CT78UG 44337131 Ki = 14 nM T52921 CO8Y5G 44337163 Ki = 745 nM T52921 CBJ01F 44337212 Ki = 49 nM T52921 C8IJM5 44337229 Ki = 26 nM T52921 C97YKG 44337230 Ki = 1062 nM T52921 C3B4WO 44337231 Ki = 1135 nM T52921 CU8IY3 44337232 Ki = 2532 nM T52921 C3M0QX 44337249 Ki = 680 nM T52921 C0MJL2 44337252 Ki = 1345 nM T52921 CB85KA 44337351 Ki = 94 nM T52921 CI13YG 44337357 Ki = 152 nM T52921 CW2FZ7 44337362 Ki = 198 nM T52921 CJ08FM 44337379 Ki = 30 nM T52921 CIP87K 44337437 Ki = 185 nM T52921 CR62KO 44337452 Ki = 79 nM T52921 C9CIP3 44337459 Ki = 3221 nM T52921 CFA2Q7 44337460 Ki = 684 nM T52921 CZP4K1 44337461 Ki = 2593 nM T52921 CF96JK 44337473 Ki = 367 nM T52921 CX87AS 44337513 Ki = 772 nM T52921 CP1VN3 44337550 Ki = 1016 nM T52921 CZ02BO 44337551 Ki = 34 nM T52921 CS9Z1O 44339374 Ki = 225 nM T52921 C73CSH 44339393 Ki = 153 nM T52921 CF08RA 44339398 Ki > 10000 nM T52921 CFNR91 44339423 Ki = 33 nM T52921 CW56BK 44339424 Ki = 12 nM T52921 C4POK5 44339425 Ki = 135 nM T52921 C03PDA 44339449 Ki = 692 nM T52921 CGI10R 44339450 Ki = 715 nM T52921 C7HIP9 44339463 Ki = 879 nM T52921 CQ24IT 44339491 Ki > 10000 nM T52921 CC1VG7 44339500 Ki = 234 nM T52921 C73QPW 44339504 Ki = 502 nM T52921 CABQ05 44339505 Ki = 1270 nM T52921 C7GRF4 44339525 Ki = 1194 nM T52921 CY85GQ 44339526 Ki = 6520 nM T52921 CZRJ83 44339528 Ki > 10000 nM T52921 CKP7R5 44339529 Ki > 10000 nM T52921 CAD1O4 44339530 Ki = 1106 nM T52921 CIZU20 44339531 Ki > 10000 nM T52921 C2LQO7 44339540 Ki = 307 nM T52921 C7E4MS 44339576 Ki = 47 nM T52921 C2PDT6 44339596 Ki = 102 nM T52921 C34DEN 44339684 Ki = 82 nM T52921 CO3C7M 44339695 Ki = 12 nM T52921 CGY16P 44339707 Ki = 827 nM T52921 CD9ZS8 44342270 IC50 = 1910 nM T52921 C4BK0O 44352743 EC50 = 439 nM T52921 CHX36W 44352744 EC50 = 286 nM T52921 C9RN1Y 44352745 IC50 = 2710 nM T52921 C1GZ8E 44352920 IC50 = 874 nM T52921 CD18TR 44366689 Ki = 2130 nM T52921 CYL95J 44366690 Ki = 35 nM T52921 C7IFR8 44366822 Ki = 34 nM T52921 CL1JV2 44366823 Ki = 44 nM T52921 CX7A3N 44388460 EC50 = 0.06607 nM T52921 CLV18K 44388461 EC50 = 0.1 nM T52921 CK95WL 44388462 EC50 = 0.06761 nM T52921 C5FA4H 44388465 EC50 = 0.4786 nM T52921 CBUS05 44388466 EC50 = 0.2399 nM T52921 CJG21X 44388467 EC50 = 0.2089 nM T52921 CZ7L6C 44388472 EC50 = 5.888 nM T52921 C4WRI8 44388474 EC50 = 0.4074 nM T52921 C5I7AN 44390989 Ki = 12 nM T52921 C2TP3J 44390999 Ki = 620 nM T52921 C9FBO3 44391012 Ki = 1115 nM T52921 C2W7BJ 44391023 Ki = 282 nM T52921 C4BF2U 44391031 Ki = 905 nM T52921 CF49QH 44391052 Ki = 32 nM T52921 C7A8DM 44391062 Ki = 10.8 nM T52921 CTA04B 44391063 Ki = 462 nM T52921 C1WGX6 44391067 Ki = 52 nM T52921 C8Y7OV 44391069 Ki = 218 nM T52921 CT8W3P 44391075 Ki = 1920 nM T52921 CY7OH0 44391079 Ki = 42 nM T52921 CPZ7L8 44391081 Ki = 28 nM T52921 CR5TN7 44391092 Ki = 37 nM T52921 C2DB4N 44391093 Ki = 768 nM T52921 CO2T5M 44391094 Ki = 14 nM T52921 CL79EO 44391099 Ki = 838 nM T52921 C3HTZ1 44391102 Ki = 509 nM T52921 CW76ZY 44391103 Ki = 24 nM T52921 CN1LD9 44391104 Ki = 38.2 nM T52921 CD3QV8 44391111 Ki = 60 nM T52921 CK2HV1 44391119 Ki = 113 nM T52921 C8RDV5 44391124 Ki = 3 nM T52921 C1UDL9 44391133 Ki = 20 nM T52921 CSV6X2 44391134 Ki = 25 nM T52921 CJ9MX1 44391137 Ki = 815 nM T52921 C18SDI 44391138 Ki = 126 nM T52921 C6ZF9E 44391155 Ki = 8.3 nM T52921 CY6T4F 44391156 Ki = 108 nM T52921 CJB0U8 44391157 Ki = 39 nM T52921 C5ZFX2 44394283 Ki = 231 nM T52921 COB70L 44394284 Ki = 40 nM T52921 C5BTZ1 44394320 Ki = 1878 nM T52921 C6DB4X 44394324 Ki = 28.7 nM T52921 C2OV9B 44394344 Ki = 46 nM T52921 C1Y3NV 44394345 Ki = 2614 nM T52921 CCR2U1 44394375 Ki = 83 nM T52921 CQ2O6J 44394381 Ki = 3.9 nM T52921 CTJ2I9 44394405 Ki = 63 nM T52921 CLFU54 44394419 Ki = 187 nM T52921 C0A1OW 44394487 Ki = 5 nM T52921 C61AXY 44394529 Ki = 9535 nM T52921 CRCV49 44394559 Ki = 609 nM T52921 C3YD8C 44395259 Ki > 10000 nM T52921 CR8AF5 44395265 Ki > 10000 nM T52921 CI7GR3 44395286 Ki = 149 nM T52921 CLB5E3 44395291 Ki > 10000 nM T52921 CEX0W2 44395306 Ki = 590 nM T52921 C69ACH 44395319 Ki > 10000 nM T52921 CQO0Y5 44395366 Ki > 10000 nM T52921 C0FUP2 44395387 Ki > 10000 nM T52921 C06LKH 44395410 Ki = 372 nM T52921 C7GP1E 44404646 IC50 = 290 nM T52921 CILB28 44404652 IC50 = 380 nM T52921 C38GAM 44404653 IC50 = 1310 nM T52921 CA58SU 44404670 IC50 = 120 nM T52921 C83PCH 44404679 IC50 = 100 nM T52921 CU0YX9 44404684 IC50 = 2400 nM T52921 CEJ7F8 44404689 IC50 = 2680 nM T52921 CD8M2R 44404693 IC50 = 710 nM T52921 C5X8YK 44404694 IC50 = 470 nM T52921 CODG94 44404695 IC50 = 150 nM T52921 CD79WM 44404698 IC50 = 450 nM T52921 C0BED6 44404699 IC50 = 37 nM T52921 CGA15Y 44404706 IC50 = 10000 nM T52921 C2NHS0 44404707 IC50 > 10000 nM T52921 CJCY60 44404711 IC50 = 1080 nM T52921 CK73OG 44404721 IC50 = 350 nM T52921 CNX5T8 44404731 IC50 = 180 nM T52921 CW9QG2 44406457 IC50 > 10000 nM T52921 CGN73V 44406458 IC50 > 10000 nM T52921 C0J7IK 44406489 IC50 = 6000 nM T52921 C5TIM4 44406497 IC50 = 1000 nM T52921 CBUR32 44406503 IC50 = 10000 nM T52921 C17FYG 44406538 IC50 = 15000 nM T52921 C07CNE 44406539 IC50 = 7000 nM T52921 C5DGV2 44406540 IC50 = 3850 nM T52921 C9Z0ET 44406541 IC50 > 10000 nM T52921 C1L8CG 44406543 IC50 = 10400 nM T52921 CP1OZ6 44406544 IC50 > 10000 nM T52921 CS04TK 44406550 IC50 = 5800 nM T52921 C8HRC9 44406551 IC50 = 15000 nM T52921 CSPE30 44406557 IC50 = 13400 nM T52921 CD7Y0Z 44406585 IC50 > 10000 nM T52921 CC15BY 44406587 IC50 = 10000 nM T52921 C1IM9R 44406603 IC50 = 1000 nM T52921 C3VE8N 44406604 IC50 = 1000 nM T52921 CCI5Z1 44406618 IC50 = 300 nM T52921 C7ES2W 44406621 IC50 = 130 nM T52921 C0SKT9 44406641 IC50 > 10000 nM T52921 C38ABN 44406682 IC50 > 10000 nM T52921 CZ65PF 44406685 IC50 > 10000 nM T52921 CWY76P 44406719 IC50 = 4000 nM T52921 CP5H7S 44406907 IC50 > 1000 nM T52921 CHKO45 44406969 IC50 > 1000 nM T52921 CV4C6R 44406970 IC50 > 1000 nM T52921 C7BNY9 44406975 IC50 > 1000 nM T52921 C0W1EN 44406978 IC50 > 1000 nM T52921 C5U7KF 44406979 IC50 > 1000 nM T52921 CM31XO 44406989 IC50 > 1000 nM T52921 CC0H4U 44406991 IC50 > 1000 nM T52921 CNP5V6 44406994 IC50 > 1000 nM T52921 C3BQ7S 44406995 IC50 > 1000 nM T52921 C92ZTH 44406996 IC50 > 1000 nM T52921 CN82CH 44406997 IC50 > 1000 nM T52921 CX20ZA 44406998 IC50 > 1000 nM T52921 CMRF31 44407013 IC50 = 630 nM T52921 C8RNE9 44407016 IC50 > 1000 nM T52921 CA2OD1 44407020 IC50 = 870 nM T52921 C0OB8F 44407023 IC50 > 1000 nM T52921 C21UFE 44407028 IC50 > 1000 nM T52921 C8GK1Q 44407036 IC50 > 1000 nM T52921 CGO7M0 44407037 IC50 > 1000 nM T52921 C4YW1C 44407038 IC50 > 1000 nM T52921 C4QT3D 44407040 IC50 > 1000 nM T52921 CK84HW 44407043 IC50 > 1000 nM T52921 CZ8D9R 44407044 IC50 = 30 nM T52921 C7QWZ5 44407048 IC50 = 360 nM T52921 CYJ04D 44407049 IC50 > 1000 nM T52921 CJ4A2W 44407050 IC50 > 1000 nM T52921 CU20IA 44407063 IC50 > 1000 nM T52921 C5PDG8 44407065 IC50 > 1000 nM T52921 CGAD30 44407066 IC50 > 1000 nM T52921 CT49JG 44407070 IC50 = 170 nM T52921 C9WJZ5 44407074 IC50 > 1000 nM T52921 CW2CP3 44407078 IC50 > 1000 nM T52921 CL9QK6 44407080 IC50 > 1000 nM T52921 C2S5NT 44407081 IC50 > 1000 nM T52921 C0QB6E 44407084 IC50 = 131 nM T52921 CLG4Y9 44407085 IC50 = 230 nM T52921 CPQ7H2 44407086 IC50 = 290 nM T52921 C0K7ZH 44407091 IC50 > 1000 nM T52921 CM8JK6 44407109 IC50 > 1000 nM T52921 C8R1QN 44407112 IC50 = 340 nM T52921 CEZ4I2 44407113 IC50 > 1000 nM T52921 CA3OW4 44407116 IC50 = 21 nM T52921 CLE6W9 44407119 IC50 > 1000 nM T52921 CK4NE2 44407129 IC50 = 50 nM T52921 CKUT49 44407133 IC50 = 24 nM T52921 COS85F 44407140 IC50 = 330 nM T52921 CAMX28 44407145 IC50 > 1000 nM T52921 CRP3D2 44407146 IC50 > 1000 nM T52921 CZO5R6 44407156 IC50 = 900 nM T52921 C2YME3 44413175 IC50 > 1000 nM T52921 CM7LE4 44413183 IC50 > 1000 nM T52921 C0M9TX 44413184 IC50 > 1000 nM T52921 CFJ64A 44413232 Ki = 970 nM T52921 CNFC81 44413248 Ki > 5000 nM T52921 C0V4FI 44413286 Ki = 550 nM T52921 CS7BI8 44413301 Ki = 81 nM T52921 C1NGS0 44413314 Ki = 94 nM T52921 C5J0BU 44413315 Ki > 5000 nM T52921 CH7E1C 44413329 Ki > 5000 nM T52921 C1OQ0L 44413330 Ki = 2 nM T52921 CKV5S0 44413361 Ki = 52 nM T52921 C5PHK7 44413362 Ki = 62 nM T52921 CSQZ28 44413379 Ki > 5000 nM T52921 CCU2B5 44413384 Ki = 660 nM T52921 CD5SZ9 44413385 Ki = 57 nM T52921 C7GE2K 44413395 Ki > 5000 nM T52921 CCK6Y5 44413396 Ki = 1650 nM T52921 C0FL8K 44413401 Ki = 3500 nM T52921 C6J3HP 44413402 Ki > 5000 nM T52921 CB2OJ9 44413408 Ki = 160 nM T52921 C82VJB 44413413 Ki > 5000 nM T52921 CP31JV 44413414 Ki = 820 nM T52921 C98OQG 44413423 Ki > 5000 nM T52921 CH0DS7 44413441 Ki = 710 nM T52921 CLSK72 44413442 Ki = 10 nM T52921 C6O2VL 44414730 IC50 > 10000 nM T52921 C5Z9VE 44414845 IC50 > 10000 nM T52921 C4LI9Q 44414865 IC50 > 10000 nM T52921 C10OMS 44426811 Ki = 9 nM T52921 C49KAS 44426813 Ki = 41 nM T52921 CJK6Y5 44426815 Ki = 4035 nM T52921 CJ5FC0 44426816 Ki = 295 nM T52921 C4TFP1 44426818 Ki = 1887 nM T52921 CP1Z5J 44426819 Ki = 10000 nM T52921 CP5V8D 44426821 Ki = 8183 nM T52921 C5L4SE 44426822 Ki = 214 nM T52921 C36SCP 44426823 Ki = 323 nM T52921 C72RXV 44426824 Ki = 35 nM T52921 C0S5TE 44426829 Ki = 12 nM T52921 CL1EG2 44426830 Ki = 357 nM T52921 CBFY73 44426831 Ki = 225 nM T52921 CFO9Q6 44426832 Ki = 0.6 nM T52921 C2NFA4 44426833 Ki = 26 nM T52921 COJ48Z 44426834 Ki = 132 nM T52921 CUD42S 44426835 Ki = 5 nM T52921 CKJ90O 44426836 Ki = 11 nM T52921 CZ4R6J 44426837 Ki = 125 nM T52921 CPDE73 44426838 Ki = 9 nM T52921 C53JGK 44426839 Ki = 6753 nM T52921 C7IJY0 44426840 Ki = 6 nM T52921 CJB90W 44426841 Ki = 42 nM T52921 C4Z1FX 44426842 Ki = 21 nM T52921 CK3B6E 44426843 Ki = 3 nM T52921 CD3TB8 44426844 Ki = 439 nM T52921 CF5OJ0 44430021 Ki = 1449 nM T52921 CUQ95Y 44430022 Ki = 16 nM T52921 CZA0E6 44430023 Ki = 1.6 nM T52921 CWX67P 44430033 Ki = 15 nM T52921 C40BHT 44430038 Ki = 0.4 nM T52921 C1QXR6 44430040 Ki = 0.7 nM T52921 CS6Y5Z 44430042 Ki = 0.5 nM T52921 C4CHV5 44430043 Ki = 1.1 nM T52921 CX9P5R 44430044 Ki = 0.5 nM T52921 CA51JN 44430045 Ki = 110 nM T52921 C2G9HQ 44430046 Ki = 674 nM T52921 C8PI4A 44430047 Ki = 9.6 nM T52921 CL1N4D 44430048 Ki = 4.6 nM T52921 C0AYM6 44430049 Ki = 5.5 nM T52921 CMJT74 44430050 Ki = 0.7 nM T52921 C4ZG6A 44430079 Ki = 2 nM T52921 CSNQ43 44430080 Ki = 12 nM T52921 CXV9J7 44430081 Ki = 5.9 nM T52921 CFHY18 44430083 Ki = 1.9 nM T52921 C6SBE1 44430084 Ki = 2.2 nM T52921 CXZ2D3 44430085 Ki = 0.9 nM T52921 CI4X3Z 44430087 Ki = 0.6 nM T52921 C8D0ZX 44431782 Ki = 1273 nM T52921 CT30KJ 44437601 Ki = 3 nM T52921 C1EHS4 44437602 Ki = 2 nM T52921 CX5O0J 44437604 Ki = 5 nM T52921 CWOJ02 44437605 Ki = 3 nM T52921 CK73VO 44437606 Ki = 3 nM T52921 CJ1ST3 44437610 Ki = 0.5 nM T52921 CFH6A5 44437613 Ki = 22 nM T52921 C0M9SC 44437615 Ki = 4 nM T52921 CFN8Z9 44437617 Ki = 6 nM T52921 CTK2S0 44437619 Ki = 1 nM T52921 C4PK1O 44437623 Ki = 5 nM T52921 CP4HR6 44437626 Ki = 4 nM T52921 CA5S2P 44437627 Ki = 46 nM T52921 CKEG06 44437628 Ki = 12 nM T52921 CT7V0O 44437629 Ki = 1595 nM T52921 C45ZTN 44437630 Ki = 10 nM T52921 CQKL94 44437636 Ki = 4 nM T52921 C43URV 44437637 Ki = 3 nM T52921 CJ8L4A 44437638 Ki = 2 nM T52921 CNBQ93 44437639 Ki = 5 nM T52921 C2AV5I 44437640 Ki = 19 nM T52921 CN3R5G 44437641 Ki = 29 nM T52921 C6NA9R 44437642 Ki = 20 nM T52921 CH5RW4 44437643 Ki = 155 nM T52921 C7RIC8 44437644 Ki = 15 nM T52921 C5IL8O 44437645 Ki = 20 nM T52921 CX1S4V 44437646 Ki = 12 nM T52921 CV19NL 44437647 Ki = 29 nM T52921 C02YET 44437648 Ki = 12 nM T52921 CJ2PH5 44437649 Ki = 3 nM T52921 CVH1I9 44437652 Ki = 23 nM T52921 C0ME9B 44437654 Ki = 2 nM T52921 CRKH10 44437656 Ki = 2 nM T52921 CZB4Q9 44438912 Ki = 61.2 nM T52921 CP85QV 44438914 Ki = 824 nM T52921 C7RD2E 44438916 Ki = 14 nM T52921 CNL30S 44438917 Ki = 3.2 nM T52921 C5D4NZ 44438920 Ki = 3.5 nM T52921 CA2LD5 44438921 Ki = 17 nM T52921 C6H7AD 44438922 Ki = 2.4 nM T52921 CRN3W4 44438961 Ki = 1.1 nM T52921 CGYD89 44438962 Ki = 1.5 nM T52921 CZ48KD 44438963 Ki = 36.5 nM T52921 C2EGK7 44438964 Ki = 10.8 nM T52921 COX57F 44438965 Ki = 9 nM T52921 C9S2HB 44438966 Ki = 11.5 nM T52921 C1HF6E 44438967 Ki = 140 nM T52921 C3L7SB 44438968 Ki = 9 nM T52921 CE63GK 44438971 Ki = 249 nM T52921 C8TVI4 44438974 Ki = 6.3 nM T52921 CPHS56 44438975 Ki = 250 nM T52921 CK3Z5G 44438978 Ki = 49 nM T52921 CPA4U5 44438983 Ki = 0.3 nM T52921 C2TKY5 44438988 Ki = 0.8 nM T52921 CL7WN5 44438993 Ki = 2.6 nM T52921 C0A2OM 44439000 Ki = 1.4 nM T52921 CMQA60 44439001 Ki = 8.4 nM T52921 CN4KX9 44449764 IC50 = 31 nM T52921 CWN0C3 44449766 IC50 = 78 nM T52921 CE97XC 44449767 IC50 = 180 nM T52921 C7NKJ3 44449771 IC50 = 140 nM T52921 CRO1B7 44449793 IC50 = 2900 nM T52921 CTMI71 44449822 IC50 = 63 nM T52921 CU6I5Y 44449823 IC50 > 10000 nM T52921 C8QE6N 44449850 IC50 = 8200 nM T52921 CH5MN1 44449851 IC50 = 910 nM T52921 CT39QP 44450085 IC50 = 1.8 nM T52921 C1SQ7M 44450086 IC50 = 20 nM T52921 CGN7O0 44450151 IC50 = 15 nM T52921 CS4DO9 44450180 IC50 = 240 nM T52921 CL5K3J 44450207 IC50 = 2900 nM T52921 CK41RX 44450208 IC50 = 140 nM T52921 CUR83O 44450209 IC50 = 380 nM T52921 C37FVM 44450210 IC50 = 55 nM T52921 CL78ZG 44451517 Ki = 3.548 nM T52921 CG2WD7 44451518 Ki = 21.88 nM T52921 CBK6R5 44451542 Ki = 3.89 nM T52921 CC36BM 44451543 Ki = 2.512 nM T52921 CKB0F9 44451569 Ki = 1.698 nM T52921 C2EJP0 44451572 Ki = 28.84 nM T52921 CYQ53B 44451573 Ki = 1174.9 nM T52921 CGJ3R8 44451592 Ki = 7.943 nM T52921 CAC1G4 44451593 Ki = 17.38 nM T52921 CV26FM 44451594 Ki = 4.898 nM T52921 CKRM60 44451595 Ki = 1.514 nM T52921 C4S0BF 44451619 Ki = 2.399 nM T52921 CAVN40 44451620 Ki = 912.01 nM T52921 C2NCL3 44451621 Ki = 1.202 nM T52921 CHPO59 44451647 Ki = 95.5 nM T52921 C70TSK 44451648 Ki = 11.75 nM T52921 CZ1R2D 44451649 Ki = 0.8913 nM T52921 C5UM1O 44451650 Ki = 1.995 nM T52921 CF4SX9 44451673 Ki = 37.15 nM T52921 C3O8ZP 44451696 Ki = 29.51 nM T52921 C7VLH3 44451724 Ki = 41.69 nM T52921 CYIP73 44451748 Ki = 1.862 nM T52921 C2IS4W 44451777 Ki = 4.898 nM T52921 CST06H 44451779 Ki = 3.311 nM T52921 C4C9TD 44451805 Ki = 4.169 nM T52921 C5RLP6 44451837 Ki = 3.715 nM T52921 CO01GQ 44451872 Ki = 5.888 nM T52921 C7KL9C 44451895 Ki = 9.55 nM T52921 C25JHV 44451918 Ki = 1.413 nM T52921 C4DL5C 44469677 IC50 > 10000 nM T52921 CFAZ41 44517710 IC50 = 5.6 nM T52921 C6T1UX 44551464 EC50 = 3.6 nM T52921 CC01KM 44561020 Ki = 3.7 nM T52921 CY14MD 44561518 Ki = 6 nM T52921 CPO2R3 44570675 Ki = 2.5 nM T52921 CNUJ50 44574003 IC50 = 38 nM T52921 C1T4QN 44574053 IC50 = 16 nM T52921 CW8DR7 44574393 Ki = 1571 nM T52921 C67IZG 44574538 Ki = 3 nM T52921 C5Q4HZ 44574539 Ki = 7.3 nM T52921 C74LHO 44574585 Ki = 2.7 nM T52921 CPL5V1 44574586 Ki = 5.2 nM T52921 C7K4PC 44574587 Ki = 13 nM T52921 C1JPH8 44574588 Ki = 1.9 nM T52921 CNCS12 44574629 Ki = 3.6 nM T52921 CJXE09 44574630 Ki = 14 nM T52921 C2FO5H 44574631 Ki = 3 nM T52921 C5YQ6B 44574632 Ki = 7.4 nM T52921 CD18EP 44574671 Ki = 385 nM T52921 CDS1G8 44574672 Ki = 8 nM T52921 C6ZMS9 44574705 Ki = 6 nM T52921 CDNP82 44574706 Ki = 3151 nM T52921 C13RZI 44574707 Ki = 100 nM T52921 CXQM01 44574708 Ki = 3 nM T52921 CW1GU7 44574743 Ki = 6 nM T52921 CL6UI1 44574744 Ki = 4 nM T52921 CKO8N4 44574745 Ki = 2 nM T52921 CLVU91 44574789 Ki = 11 nM T52921 C5JZK9 44574790 Ki = 5.3 nM T52921 CVZ6K3 44574848 Ki = 31 nM T52921 C1MWD8 44574849 Ki = 40 nM T52921 CA78KV 44574850 Ki = 22 nM T52921 CX1BL6 44574851 Ki = 285 nM T52921 C7YAD5 44574889 Ki = 678 nM T52921 CPH7D4 44574890 Ki = 4.9 nM T52921 CQL2E4 44574891 Ki = 7 nM T52921 C9C3ZJ 44574892 Ki = 10 nM T52921 CLG57R 44574958 Ki = 12 nM T52921 CLMH36 44574962 Ki = 8.2 nM T52921 CAW3R4 44574963 Ki = 11 nM T52921 CAWB12 44575043 Ki = 17 nM T52921 CZO5J4 44575091 Ki = 908 nM T52921 CI6Y7U 44575092 Ki = 142 nM T52921 CO26ZW 44576625 IC50 = 8 nM T52921 CSH8K2 44576626 IC50 = 59 nM T52921 CD0T5K 44576627 IC50 = 18 nM T52921 C4ZCX6 44576628 IC50 = 1.1 nM T52921 CR0LN1 44593575 Ki = 198 nM T52921 CTYR04 44593576 Ki = 19 nM T52921 CDPU87 44596170 EC50 = 94 nM T52921 C45PUQ 45102745 Ki = 0.7 nM T52921 CU8I6T 45263517 Ki = 0.7 nM T52921 CVDQ53 45265789 Ki = 23 nM T52921 C6VZM4 45267505 IC50 = 2.5 nM T52921 CA2MH1 45267506 IC50 = 33 nM T52921 CK16EZ 45267601 IC50 = 28 nM T52921 CR59UW 45267616 IC50 = 200 nM T52921 CY4UA3 45267639 IC50 > 1000 nM T52921 CA2O3N 45268153 Ki = 3 nM T52921 C4F6IO 45268355 IC50 = 4.3 nM T52921 CX3YO5 45268356 IC50 = 17 nM T52921 C7UG6Q 45268498 IC50 = 2.3 nM T52921 C8QG3U 45268503 IC50 = 160 nM T52921 C3YEJ9 45268504 IC50 = 33 nM T52921 C8BPX4 45269032 Ki = 2 nM T52921 CKC09D 45269228 IC50 = 210 nM T52921 CKZ35F 45269347 IC50 > 1000 nM T52921 C06ITN 45269349 IC50 > 1000 nM T52921 C78UOX 45269357 IC50 = 4.7 nM T52921 C4WT5J 45269358 IC50 = 1.4 nM T52921 C3I6YO 45269372 IC50 = 160 nM T52921 CSL62Z 45270082 IC50 = 6.4 nM T52921 C6PRX0 45270174 IC50 = 620 nM T52921 C6GRC1 45270175 IC50 > 1000 nM T52921 CA38NB 45270184 IC50 = 3.7 nM T52921 CVU53F 45270190 IC50 > 1000 nM T52921 CA3S7Q 45270196 IC50 = 530 nM T52921 CY79OE 45270202 IC50 = 540 nM T52921 CVP80J 45270203 IC50 = 500 nM T52921 CC5I8O 45270712 Ki = 71 nM T52921 CM5ZI0 45270907 IC50 = 2 nM T52921 C6P0AZ 45270917 IC50 = 13 nM T52921 CDT5G6 45270928 IC50 = 15 nM T52921 C8KS5V 45271014 IC50 = 850 nM T52921 C2G5XK 45271015 IC50 = 26 nM T52921 CO05CL 45271041 IC50 = 11 nM T52921 CU84PI 45271534 Ki = 2 nM T52921 CP6V4Q 45271862 IC50 = 520 nM T52921 CMGB49 45271885 IC50 = 190 nM T52921 CJGX41 45271896 IC50 > 1000 nM T52921 C6G9DQ 45271902 IC50 = 160 nM T52921 C1UOZ9 45272626 IC50 = 7.8 nM T52921 C0P6GI 45272729 IC50 > 1000 nM T52921 CL0Y5P 45272733 IC50 > 1000 nM T52921 C09HIZ 45272755 IC50 > 1000 nM T52921 CFU9R4 45273531 IC50 = 0.61 nM T52921 CX0N4V 45273537 IC50 = 3.1 nM T52921 CJNO02 45273546 IC50 = 1.4 nM T52921 C3ZPJ5 45273547 IC50 = 12 nM T52921 CGT48R 45273662 IC50 = 130 nM T52921 C91JXR 45273672 IC50 > 1000 nM T52921 C58HQB 45273679 IC50 = 4.5 nM T52921 CS0GA2 45273702 IC50 = 96 nM T52921 C3YHF0 46227961 EC50 = 135 nM T52921 C7LW1S 46227963 Ki = 4.2 nM T52921 C9L6WI 46227966 EC50 = 15 nM T52921 CA2P9C 46879475 Ki = 4082 nM T52921 CH45JY 46879476 Ki = 454 nM T52921 CS2V6N 46879477 Ki = 16 nM T52921 C6R8JO 46879478 Ki = 106 nM T52921 C9URN3 46879536 Ki = 21 nM T52921 C5PW9I 46879537 Ki = 11 nM T52921 CW2N7P 46879538 Ki = 2.9 nM T52921 CGJS91 46879539 Ki = 6.4 nM T52921 C08CHW 46879578 Ki = 28 nM T52921 CNF9D6 46879579 Ki = 2.3 nM T52921 C8UD2Z 46879580 Ki = 0.6 nM T52921 C9E8YP 46879581 Ki = 2.5 nM T52921 C9GB7O 46879627 Ki = 2152 nM T52921 C5VKU0 46879628 Ki = 227 nM T52921 CU2F0K 46879629 Ki = 111 nM T52921 CS7BP4 46879630 Ki = 295 nM T52921 C06NBW 46879667 Ki = 44 nM T52921 C0WY3K 46879668 Ki = 22 nM T52921 C5L7DB 46879669 Ki = 7.7 nM T52921 CSG31K 46879670 Ki = 5 nM T52921 C7P4UE 46879716 Ki = 7.1 nM T52921 CQSI16 46879992 Ki = 470 nM T52921 C16INW 46879993 Ki = 227 nM T52921 C9NR8Q 46880030 Ki = 35 nM T52921 C0O1PU 46880031 Ki = 15 nM T52921 CDY2L8 46880032 Ki = 0.2 nM T52921 CK01VS 46880033 Ki = 1.3 nM T52921 CFXU43 46880088 Ki = 62 nM T52921 CDM4C0 46880089 Ki = 5.2 nM T52921 CA8JU6 46880090 Ki = 5.5 nM T52921 C7LX9B 46880114 Ki = 4.7 nM T52921 CX7RS8 46880115 Ki = 253 nM T52921 C2VS0K 46880116 Ki = 3.5 nM T52921 C18JDU 46880117 Ki = 487 nM T52921 CHN70E 46880151 Ki = 2560 nM T52921 CI5D6H 46880152 Ki = 259 nM T52921 CF0ER7 46880153 Ki = 1118 nM T52921 CU8JO5 46880154 Ki = 471 nM T52921 CR35XL 46880155 Ki = 186 nM T52921 CI6ZA1 46880237 Ki = 29 nM T52921 CID57V 46880238 Ki = 2.7 nM T52921 CG6UO7 46880239 Ki = 18 nM T52921 C31BLP 46880240 Ki = 1050 nM T52921 C3T6NH 49843555 Ki = 1.438 nM T52921 C0TCI3 52915030 IC50 = 31.6 nM T52921 CK6GN5 52915031 IC50 = 28.1 nM T52921 CXF14W 52915032 IC50 = 32.7 nM T52921 CELZ30 52915143 IC50 = 98.9 nM T52921 CR57AK 52915144 IC50 = 308.9 nM T52921 CP29EV 52915145 IC50 = 186.2 nM T52921 C15YXV 52915146 IC50 = 208.6 nM T52921 C45JNG 52915147 IC50 = 141.9 nM T52921 COM38Z 52915266 IC50 = 146.5 nM T52921 COEU73 52915267 IC50 = 154.5 nM T52921 CZK59C 52915268 IC50 = 184.5 nM T52921 C27KOF 52915269 IC50 = 83 nM T52921 CQ71YX 52915270 IC50 = 1115.9 nM T52921 CH56XF 52915389 IC50 = 731.6 nM T52921 C02UBO 52915390 IC50 = 1217.8 nM T52921 CP2M6E 52915391 IC50 = 667.5 nM T52921 CPA43I 52915392 IC50 = 482.9 nM T52921 C5OA9H 52915393 IC50 = 304.6 nM T52921 CA3P2C 52915514 IC50 = 404.7 nM T52921 CK39TQ 52915515 IC50 = 159.6 nM T52921 C98UZW 52915516 IC50 = 799.8 nM T52921 CLAS61 52915517 IC50 = 206.9 nM T52921 C7FDE9 52915518 IC50 = 1106.7 nM T52921 C9YOD2 52915634 IC50 = 246.4 nM T52921 C1ZHF3 52915635 IC50 = 144 nM T52921 CZB67C 52915636 IC50 = 211.6 nM T52921 CE3IS2 52915637 IC50 = 152.9 nM T52921 C8F0TA 52916174 IC50 = 207.3 nM T52921 C4K3NO 52916266 IC50 = 115.7 nM T52921 CPV9S3 52916267 IC50 = 48 nM T52921 CXGN56 52916358 IC50 = 35.6 nM T52921 CO4Q6E 52916359 IC50 = 50.9 nM T52921 CM0KA5 52916360 IC50 = 83.3 nM T52921 CN8L4T 52916470 IC50 = 63.1 nM T52921 C96OUY 52916471 IC50 = 113.6 nM T52921 CC92WA 52916472 IC50 = 82.7 nM T52921 CG91EA 52916597 IC50 = 82.1 nM T52921 CYB6J8 52916598 IC50 = 76.5 nM T52921 CG1F9W 52916599 IC50 = 56.6 nM T52921 C7NO2D 52916712 IC50 = 76.2 nM T52921 CZ3K9S 52916713 IC50 = 71.7 nM T52921 CI32WO 52916714 IC50 = 30.1 nM T52921 C4FZT7 52951674 Ki = 0.231 nM T52921 CS4T2C 52951675 Ki = 0.101 nM T52921 C5VLO1 52951807 Ki = 0.106 nM T52921 CK7I1T 52951808 Ki = 0.137 nM T52921 C0UVH3 52951809 Ki = 0.09 nM T52921 C40BPO 52951810 Ki = 0.15 nM T52921 CF0L7D 52951938 Ki = 4.51 nM T52921 CDAN40 52951939 Ki = 17.1 nM T52921 C89QXK 52951940 Ki = 5.61 nM T52921 COVP24 52951941 Ki = 10.2 nM T52921 CR6B4G 52951942 Ki = 9.08 nM T52921 CSF4G7 52952043 Ki = 5.32 nM T52921 CTU43X 53316968 Ki = 4.54 nM T52921 CCOD69 53316969 Ki = 4.29 nM T52921 CI6CQ0 53319615 Ki = 0.15 nM T52921 C6SY4G 53319616 Ki = 80.5 nM T52921 C3PW1V 53319617 Ki = 4.29 nM T52921 C2EV1S 53322245 Ki = 0.96 nM T52921 C1L8IV 53322246 Ki > 250 nM T52921 C0MD2H 53324890 Ki = 0.73 nM T52921 C5E7LW 53325608 Ki = 4.29 nM T52921 CRZ76L 53326167 Ki = 6.56 nM T52921 CJ46YH 54580478 Ki = 58.88 nM T52921 C35VCH 54580479 Ki = 48.98 nM T52921 CED95R 54581495 Ki = 107.15 nM T52921 CW7FV5 54581497 Ki = 83.18 nM T52921 CWOA13 54583469 Ki > 10000 nM T52921 CE9OC2 54584439 Ki = 60.26 nM T52921 CA4XQ2 54584440 Ki = 1148.15 nM T52921 C8J5OH 54585395 Ki = 58.88 nM T52921 CM3A1U 54585396 Ki = 158.49 nM T52921 CYS7J8 54586351 Ki > 10000 nM T52921 CROS84 54756989 Ki = 18.5 nM T52921 C2ISE6 54756990 Ki = 22 nM T52921 CCN2E8 56658044 Ki = 16 nM T52921 C69VIF 56661555 Ki = 67.8 nM T52921 CDKP63 56664973 Ki = 8.46 nM T52921 C4QM3N 56668405 Ki = 237 nM T52921 CX8F2N 56681954 Ki = 133 nM T52921 C2A4MQ 56681955 Ki = 159 nM T52921 CQY16A 57391870 Ki > 10000 nM T52921 CI5H3N 58268566 Ki = 0.0916 nM T52921 C6Z9JF 58268629 Ki = 0.0892 nM T52921 C6G5TY 60154189 Ki = 7.37 nM T52921 C2ZG0F 60154190 Ki = 9.4 nM T52921 C8MS6N 60154191 Ki = 1.84 nM T52921 CW63KM 60154192 Ki = 5.16 nM T52921 C2QX6R 60154193 Ki > 10 nM T52921 CTCJ21 60154194 Ki > 10 nM T52921 CO4Q8V 60154195 Ki > 10 nM T52921 C80XNK 60154196 Ki > 10 nM T52921 CJ8DW1 60154197 Ki > 40 nM T52921 CD5R7A 60154198 Ki > 40 nM T52921 CY1U7F 60154199 Ki > 40 nM T52921 CXRV52 60154200 Ki = 0.396 nM T52921 CD46EJ 60154264 Ki = 0.114 nM T52921 C98XRD 66911347 Ki = 205 nM T52921 CZ63PG 66986460 Ki = 3.7 nM T52921 CF5I0R 68917692 Ki = 1.26 nM T52921 CPE62M 70682348 Ki > 250 nM T52921 C6KD9C 70682349 Ki > 250 nM T52921 C2PC8W 70682350 Ki > 250 nM T52921 C58AOU 70682351 Ki = 9.84 nM T52921 CH42QP 70682760 Ki = 0.194 nM T52921 C6G0SO 70684433 Ki = 11.6 nM T52921 CZ5B7A 70684434 Ki > 250 nM T52921 CLY56A 70684435 Ki > 250 nM T52921 C8U1PW 70684436 Ki = 13.6 nM T52921 C4ZU7H 70684841 Ki = 0.0902 nM T52921 C6DC8G 70684842 Ki = 0.0672 nM T52921 CWAL85 70686573 Ki > 250 nM T52921 CAFB10 70686574 Ki > 250 nM T52921 CZ6E9M 70686575 Ki > 250 nM T52921 CPD35T 70686907 Ki = 5.32 nM T52921 CI61FE 70688692 Ki > 250 nM T52921 C08OUK 70688693 Ki > 250 nM T52921 CMKZ80 70688694 Ki > 250 nM T52921 CLK7P0 70688695 Ki > 250 nM T52921 C8M4PI 70688696 Ki > 250 nM T52921 C3HAX5 70688697 Ki = 3.79 nM T52921 C7PNH3 70689062 Ki = 0.0373 nM T52921 CA3T1P 70689063 Ki = 0.127 nM T52921 CF7PZ4 70690755 Ki = 5.55 nM T52921 CMNL89 70690756 Ki = 128 nM T52921 CWB17N 70690757 Ki = 26.2 nM T52921 CX5VR6 70690758 Ki = 26.5 nM T52921 C8UYZ6 70690759 Ki > 250 nM T52921 CTB4I1 70690760 Ki = 0.96 nM T52921 CQJ6K3 70691171 Ki = 2.05 nM T52921 CEV6U7 70691173 Ki = 0.248 nM T52921 CY6E2Q 70691339 IC50 > 10000 nM T52921 C3E4FO 70692893 Ki = 101 nM T52921 CV61FR 70692894 Ki = 31.5 nM T52921 C05RKU 70692895 Ki = 286 nM T52921 CLM98A 70692896 Ki > 250 nM T52921 CU60IL 70694933 Ki > 250 nM T52921 CWO5F0 70695375 Ki = 0.169 nM T52921 CJ07AO 70696988 Ki > 250 nM T52921 C4Z0QA 70696990 Ki > 250 nM T52921 CV0P1X 70696991 Ki = 3.03 nM T52921 CFQ8Y9 70696992 Ki > 250 nM T52921 CTO0Y4 70697389 Ki = 0.458 nM T52921 CNE50L 70697390 Ki = 0.124 nM T52921 CG3U7F 70697391 Ki = 0.134 nM T52921 CEOQ43 71229805 Ki = 43.2 nM T52921 CJDR19 71230446 Ki = 44 nM T52921 CM0H5E 71454460 Ki = 22 nM T52921 CBEV63 71461579 Ki = 27.9 nM T52921 C0B7LC 71624265 Ki = 7.63 nM T52921 C7Q9VU 71624266 Ki = 15.26 nM T52921 CD9IO8 71624267 Ki = 212.8 nM T52921 CXZ6E1 71624268 Ki = 9.98 nM T52921 C0O6IR 71624269 Ki = 26.9 nM T52921 CW2G0T 71624270 Ki = 6.53 nM T52921 CBM1C8 71624387 Ki = 12.65 nM T52921 CML7K2 71624388 EC50 = 6.8 nM T52921 C1B9VM 71624389 Ki = 40.28 nM T52921 CWH6T3 72548703 IC50 = 0.98 nM T52921 CC6Q5R 72771081 Ki < 100 nM T52921 C7ZN1K 73345634 Ki = 0.05495 nM T52921 CN5S4A 73350483 Ki = 11.43 nM T52921 COS31U 73354624 Ki = 1700 nM T52921 CJQ25A 76309739 Ki = 4 nM T52921 CC01JG 76309740 Ki = 3 nM T52921 C69JCU 76313421 Ki = 31 nM T52921 CJR57Q 76313422 Ki = 401 nM T52921 CA4IN3 76313423 Ki = 16 nM T52921 CP3HV7 76313424 Ki = 10 nM T52921 CU56FN 76313425 Ki = 10 nM T52921 CPJ4N3 76313426 Ki = 36 nM T52921 C7LV2A 76313427 Ki = 13 nM T52921 CTN6G1 76316935 Ki = 15 nM T52921 C1AW8J 76316936 Ki = 22 nM T52921 CC2AG6 76316937 Ki = 17 nM T52921 CNAE72 76320663 Ki > 1000 nM T52921 CD0PC8 76320664 Ki > 1000 nM T52921 CF83DA 76320665 Ki = 6 nM T52921 C5W1XJ 76320666 Ki = 3 nM T52921 C0MI1G 76324308 Ki = 3 nM T52921 CI2A6W 76324309 Ki = 29 nM T52921 CT9XB8 76324310 Ki = 6 nM T52921 C4QM6R 76324311 Ki = 79 nM T52921 C6AY5S 76327872 Ki = 15 nM T52921 CCR5B1 76327873 Ki = 47 nM T52921 CL58DY 76327874 Ki = 9 nM T52921 CBVL29 76327875 Ki = 19 nM T52921 C64JDN 76327876 Ki = 7 nM T52921 C3G1LA 76327877 Ki = 42 nM T52921 CCN1M9 76331524 Ki = 75 nM T52921 CQ35XY 76331525 EC50 = 14 nM T52921 CDA37E 76335140 Ki = 72 nM T52921 CUZ30G 76335141 Ki = 122 nM T52921 CKZ7T2 76335142 Ki = 10 nM T52921 CQKT47 76335143 Ki = 10 nM T52921 C6K5RY 76335144 Ki = 10 nM T52921 CECO35 76335145 Ki = 12 nM T52921 CLH3X9 81689704 Ki = 80 nM T52921 CGH7J9 86279209 Ki = 3.16 nM T52921 C8HE3B 90306863 Ki = 4630 nM T52921 C1W9QL 90306885 Ki = 75 nM T52921 C1DOG7 90654745 Ki = 0.172 nM T52921 CX3WT1 90654746 Ki = 0.176 nM T52921 CC70MH 90654747 Ki = 0.145 nM T52921 C4ZQD5 90654748 Ki = 0.371 nM T52921 CBV23K 90654749 Ki = 0.114 nM T52921 C87NYV 90654750 Ki = 0.097 nM T52921 C20FOK 90654751 Ki = 0.105 nM T52921 CT91LC 90654752 Ki = 0.185 nM T52921 CT5U7G 90654753 Ki = 0.139 nM T52921 C42GMO 90654754 Ki = 0.0711 nM T52921 CBR5H7 90654755 Ki = 0.0954 nM T52921 C68VLU 90654756 Ki = 0.0648 nM T52921 C8GUX3 90654757 Ki = 0.122 nM T52921 C4Z6KQ 90654758 Ki = 0.0908 nM T52921 C13ACK 90654759 Ki = 0.0939 nM T52921 C7C5BM 90655970 Ki > 10000 nM T52921 CTV50C 90655971 Ki = 2.1 nM T52921 C1S5UB 90655972 Ki = 3.41 nM T52921 CV6A5T 90655973 Ki = 2.99 nM T52921 CL0D4Y 90655974 Ki = 8.63 nM T52921 C51CQN 90655975 Ki = 11.1 nM T52921 C2USA9 90655976 Ki = 76.6 nM T52921 CLKW80 90655977 Ki > 10000 nM T52921 C96DUE 90655978 EC50 = 72.2 nM T52921 C1N5QA 90655979 Ki > 10000 nM T52921 CK9FP8 90656664 Ki = 197 nM T52921 COGW86 90656666 Ki = 105 nM T52921 C9YKV8 90656667 Ki = 187 nM T52921 C3WLH8 90656668 Ki = 396 nM T52921 CP1ZW6 90663949 Ki > 5000 nM T52921 CZ9GL5 90663950 Ki = 45 nM T52921 CFK27M 90663951 Ki > 5000 nM T52921 CBT6F1 90663952 Ki > 5000 nM T52921 C1QAB3 90663953 Ki = 34 nM T52921 C07VRA 101341769 Ki = 39 nM T52921 C4VMI7 101354795 IC50 = 1.67 nM T52921 CBM3Q5 118662014 Ki = 68 nM T52921 CK8Y3E 118662042 Ki = 170 nM T52921 CS81PR 118662074 Ki = 0.8 nM T52921 C8AF6I 118662117 Ki = 29.5 nM T52921 CBJ16O 118662129 Ki = 1510 nM T52921 C4ZP0L 118662159 Ki = 1.6 nM T52921 CR6IU7 118662169 Ki = 2160 nM T52921 C7VE1O 118662183 Ki = 600 nM T52921 C1VR3B 118662189 Ki = 0.7 nM T52921 CG0R6H 118662291 Ki = 2.9 nM T52921 CI17PS 118662309 Ki = 5.8 nM T52921 CCIP14 118662342 Ki = 1.1 nM T52921 CB79UC 118662456 Ki = 2.3 nM T52921 C5LZ8I 118662460 Ki = 0.4 nM T52921 CM8TB4 118705898 Ki = 1300 nM T52921 C80UNO 118705899 Ki = 1500 nM T52921 C6RW0E 118705901 Ki = 880 nM T52921 C20RQZ 118711156 Ki = 1600 nM T52921 CV85YO 118711243 Ki = 5.4 nM T52921 CKUT03 118711485 Ki = 0.5 nM T52921 CI6BM7 118711486 Ki = 2 nM T52921 CMY0F1 118711490 Ki = 0.55 nM T52921 CMRV59 118711491 Ki = 1.1 nM T52921 CTVK82 118717442 IC50 = 1.39 nM T52921 CSIW96 118718262 Ki = 39 nM T52921 C4LM3W 118718263 Ki = 55 nM T52921 C2Q8YU 118718264 Ki = 116 nM T52921 C9BFP5 118718265 Ki = 5 nM T52921 CS14YZ 118718266 Ki = 7 nM T52921 CRBA23 118718267 Ki = 82 nM T52921 C4AS8L 118718268 Ki = 35 nM T52921 CP8I2K 118718269 Ki = 17 nM T52921 C6TGR8 118718270 Ki = 336 nM T52921 C3W1BL 118718271 Ki = 29 nM T52921 CPC23W 118718272 Ki = 24 nM T52921 C2Y4PK 118718273 Ki = 104 nM T52921 C8FC1Q 118718274 Ki = 4 nM T52921 C2BGR0 118718275 Ki = 27 nM T52921 CJZ1F7 118718276 Ki = 34 nM T52921 CCFR52 118718277 Ki = 15 nM T52921 C5O2VC 118718278 Ki = 58 nM T52921 CC0KE5 118718279 Ki = 7 nM T52921 CK1Q9B 118718280 Ki = 20 nM T52921 CB92OV 118718281 Ki = 50 nM T52921 CSK4N3 118718282 Ki = 173 nM T52921 CDBP05 118718283 Ki = 245 nM T52921 CDH69C 118718284 Ki = 670 nM T52921 CLRD02 118718285 Ki = 62 nM T52921 CYI4T2 118718286 Ki = 27 nM T52921 C2F8ZN 118718287 Ki = 99 nM T52921 CA9N0S 118718288 Ki = 11 nM T52921 CVT94Z 118718289 Ki = 6 nM T52921 C1RAX5 118718290 Ki = 10 nM T52921 CKNL94 118718291 Ki = 17 nM T52921 CKN54J 118718292 Ki = 20 nM T52921 CC6U5D 118718293 Ki = 210 nM T52921 C64JUV 118718294 Ki = 70 nM T52921 CICJ78 118718295 Ki = 68 nM T52921 CZMR06 118718296 Ki = 31 nM T52921 C92CER 118718297 Ki = 118 nM T52921 CP23YE 118718298 Ki = 50 nM T52921 COA69M 118718299 Ki = 39 nM T52921 CSW82H 118718300 Ki = 74 nM T52921 C2EGJ8 118718301 Ki = 11 nM T52921 CO5BV4 118718302 Ki = 12 nM T52921 CTF9L6 118722880 Ki = 7.4 nM T52921 CDI8J1 118722882 Ki = 0.5 nM T52921 C3T8YZ 118726261 IC50 = 61 nM T52921 C6I5HS 118726262 IC50 = 4.2 nM T52921 C10BIV 118726263 IC50 = 99.7 nM T52921 CA43CF 118726264 IC50 = 166 nM T52921 CLSG96 118726265 IC50 = 160 nM T52921 CYL40S 118726266 IC50 = 8 nM T52921 CPR0K2 118726267 IC50 = 14 nM T52921 CH9A3M 118726268 IC50 = 26 nM T52921 CEH89Y 118726269 IC50 = 3.9 nM T52921 CT7H2M 118726270 IC50 = 40.9 nM T52921 C1UD6R 118726271 IC50 = 8.8 nM T52921 CRK62Y 118726272 IC50 = 37 nM T52921 CF25IA 118726273 IC50 = 18 nM T52921 CQH1G3 118731120 Ki > 10000 nM T52921 CK0LH7 122179050 Ki = 97 nM T52921 CEY90C 122179051 Ki = 1270 nM T52921 CBP42W 122179052 EC50 = 14 nM T52921 CNCJ68 122179053 EC50 = 7.3 nM T52921 CY96XI 122179055 Ki = 820 nM T52921 C6LDU5 122179056 Ki = 240 nM T52921 C57GMN 122179057 Ki = 56 nM T52921 C0X6AF 122179058 Ki = 56 nM T52921 CS0B3O 122179059 Ki = 26 nM T52921 C09BYL 122179060 Ki = 47.8 nM T52921 CF83LN 122179061 Ki = 62.2 nM T52921 CC73XP 122179063 Ki = 571 nM T52921 C6YQM4 122179064 EC50 = 230 nM T52921 C9WF5T 122179567 EC50 = 323.59 nM T52921 CTA9E8 122179568 EC50 = 158.49 nM T52921 C35HVO 122179584 EC50 = 426.58 nM T52921 CF2W0K 122179586 EC50 = 208.93 nM T52921 CE3LH1 122179587 EC50 = 45.71 nM T52921 CAQ5B0 122409965 Ki = 0.53 nM T52921 C51MTO 124565311 Ki = 0.21 nM T52921 C1YEA7 127030671 Ki > 250 nM T52921 C1HO7F 127033703 Ki = 3.13 nM T52921 CB12AP 127033704 Ki > 250 nM T52921 C4NIU0 127034022 Ki = 5.65 nM T52921 C7ORD8 127034023 Ki = 5.55 nM T52921 CEWM81 127034292 Ki = 3.56 nM T52921 CBOC84 127034554 Ki = 18.1 nM T52921 CXMJ48 127043001 Ki = 27 nM T52921 CFU4H9 127043364 Ki = 47 nM T52921 C30BNK 127043559 Ki = 38 nM T52921 CCSZ68 127044528 Ki = 42 nM T52921 C1EHU5 129188443 Ki = 9.8 nM T52921 CD8FT9 129188454 Ki = 2.17 nM T52921 CC9Z0J 129188459 Ki = 10.3 nM T52921 CG57MT 134563466 Ki = 10.5 nM T52921 CE5RS7 134563496 Ki = 23.6 nM T52921 CAEY19 134563500 Ki = 216 nM T52921 C82SEF 134563650 Ki = 44.7 nM T52921 CC3HK6 134563655 Ki = 0.3 nM T52921 C4U9EM 134563691 Ki = 43.8 nM T52921 CFX37T 134563695 Ki = 129 nM T52921 CPEH72 134563698 Ki = 24.4 nM T52921 CR74XA 134563699 Ki = 31.8 nM T52921 C9PN6I 134578342 Ki = 15.9 nM T52921 CK62WY 134578456 Ki = 9.46 nM T52921 CN0C9Z 134578457 Ki = 1.47 nM T52921 C0HNI9 134578506 Ki = 64 nM T52921 C0JCQ2 134578518 Ki = 136 nM T52921 C1CH3X 135458466 IC50 = 199 nM T52921 CN14XB 136036819 Ki = 5.888 nM T52921 CL14DP 136043756 IC50 = 440 nM T52921 CC1N8P 136043758 IC50 > 1000 nM T52921 CUXY20 136043759 IC50 = 294 nM T52921 C7US0J 136043761 IC50 > 1000 nM T52921 CFLE34 136043762 IC50 > 1000 nM T52921 C0HPR7 136043764 IC50 > 1000 nM T52921 C9WN3S 136043765 IC50 = 580 nM T52921 CB5O8L 136043767 IC50 = 440 nM T52921 CW9HY3 136043768 IC50 > 1000 nM T52921 C8CTV4 136043771 IC50 = 140 nM T52921 CB36GF 136043772 IC50 > 1000 nM T52921 CIZ41F 136043774 IC50 > 1000 nM T52921 CKW90B 136043777 IC50 > 1000 nM T52921 CJL1Y8 136043778 IC50 > 1000 nM T52921 C5KZF8 136043779 IC50 = 58 nM T52921 C2LC8O 136043780 IC50 = 450 nM T52921 C9B0WD 136043781 IC50 = 568 nM T52921 CJM57B 136043782 IC50 = 233 nM T52921 C0A6NT 136043783 IC50 > 1000 nM T52921 C0QTA5 136043784 IC50 > 1000 nM T52921 CRGU10 136043785 IC50 > 1000 nM T52921 COL64J 136043786 IC50 = 120 nM T52921 CV5AJ0 136043787 IC50 > 1000 nM T52921 CH0VN9 136043788 IC50 = 62 nM T52921 C1GJE7 136043789 IC50 > 1000 nM T52921 CC8ZK4 136043790 IC50 = 210 nM T52921 C0QDL8 136043791 IC50 > 1000 nM T52921 CM2I3S 136043792 IC50 = 600 nM T52921 CZ6A5D 136043795 IC50 = 450 nM T52921 C24BXO 136043796 IC50 = 230 nM T52921 CQLF58 136043797 IC50 = 560 nM T52921 C9EF5P 136043798 IC50 > 1000 nM T52921 CEZ83O 136043799 IC50 > 1000 nM T52921 CFZX29 136043800 IC50 = 49 nM T52921 CVFX50 136043807 IC50 > 1000 nM T52921 C5TIE8 136043816 IC50 > 1000 nM T52921 C68CEZ 136043817 IC50 = 450 nM T52921 CCJ02K 136043818 IC50 > 1000 nM T52921 C06YGH 136043819 IC50 = 632 nM T52921 C1XV2U 136043820 IC50 > 1000 nM T52921 C53OLF 136043821 IC50 > 1000 nM T52921 C4NXF8 136043824 IC50 = 410 nM T52921 CX3H8P 146034954 EC50 = 72.44 nM T52921 C85LIH 146034955 EC50 = 7.244 nM T52921 CY5CL2 155521553 Ki = 20.9 nM T52921 CZ1V3B 155523994 IC50 = 0.63 nM T52921 CXH95L 155531153 Ki = 2.27 nM T52921 CTWG84 155533462 Ki = 2 nM T52921 C4RWI6 155536757 Ki = 27 nM T52921 CHJ59D 155537352 Ki = 15.5 nM T52921 C67WLH 155542684 Ki = 23.1 nM T52921 CU83VX 155544763 Ki = 11 nM T52921 CQ0GL3 155569552 Ki = 11 nM T52921 D00BIE 25084507 Ki = 0.34 nM T52921 D00HAJ 73347136 IC50 > 50000 nM T52921 D00LVW 44456141 IC50 = 3.42 nM T52921 D00XZH 44430025 Ki = 433 nM T52921 D00YCW 44426807 Ki = 19 nM T52921 D01CFO 44456028 IC50 = 7.42 nM T52921 D01MUV 10314141 Ki = 62 nM T52921 D01WMU 9820782 Ki = 4 nM T52921 D02NSY 10296561 Ki = 0.2399 nM T52921 D02TPK 44416445 IC50 = 0.0803 nM T52921 D02WBU 44456216 EC50 = 17.7 nM T52921 D03BVN 44456298 EC50 = 23.8 nM T52921 D03PTV 10022129 Ki = 59 nM T52921 D03UJW 22970051 Ki = 23 nM T52921 D04PUK 44426803 Ki = 613 nM T52921 D04WRO 44456337 IC50 = 218 nM T52921 D04ZQX 44426812 Ki = 18 nM T52921 D05NIE 44430036 Ki = 455 nM T52921 D05RII 44413409 Ki = 1140 nM T52921 D05YMD 44455999 IC50 = 21.3 nM T52921 D06MQG 44430018 Ki = 180 nM T52921 D06PHT 10269001 Ki = 13 nM T52921 D06PVO 44426806 Ki = 135 nM T52921 D06RSR 44456187 IC50 = 14.7 nM T52921 D07CIU 9924923 Ki = 55 nM T52921 D07FCB 9925737 Ki = 323 nM T52921 D07NMH 10093682 Ki = 51 nM T52921 D08BAW 44456185 IC50 = 1.86 nM T52921 D08DVV 44430026 Ki = 1147 nM T52921 D08IXN 5497186 Ki = 0.03 nM T52921 D08NDP 25080768 Ki = 0.1 nM T52921 D08QBS 44178080 IC50 = 4.6 nM T52921 D08QBU 44430029 Ki = 1667 nM T52921 D08TFY 10043439 Ki = 17 nM T52921 D08ZDP 44430014 Ki = 9155 nM T52921 D09BYD 20481138 Ki = 11 nM T52921 D09CTG 44416444 IC50 = 0.789 nM T52921 D09FJY 9863568 Ki = 2 nM T52921 D09KBQ 131534 Ki = 2151 nM T52921 D09LRO 44430008 Ki = 23 nM T52921 D09VRT 44426814 Ki = 16 nM T52921 D09XZM 10986104 IC50 = 3.03 nM T52921 D0A1XG 44416268 IC50 > 10000 nM T52921 D0A8NZ 44578000 Ki = 0.27 nM T52921 D0A8ZS 44456217 IC50 = 92.6 nM T52921 D0AC0A 10047612 Ki = 0.253 nM T52921 D0D0UP 10315818 Ki = 48 nM T52921 D0D9BB 10427620 Ki = 313 nM T52921 D0E3RQ 44416159 IC50 = 0.0464 nM T52921 D0F8AX 44430024 Ki = 376 nM T52921 D0F8CV 5462471 Ki > 10000 nM T52921 D0FF6S 16038374 IC50 > 10000 nM T52921 D0G4FA 10384734 Ki = 588 nM T52921 D0G7DF 44426827 Ki = 3 nM T52921 D0HN2M 44430609 Ki = 0.02818 nM T52921 D0IL9H 44430013 Ki = 1745 nM T52921 D0J5JO 44430009 Ki = 27 nM T52921 D0JH5D 44430007 Ki = 34 nM T52921 D0K2NY 44456101 IC50 = 5.67 nM T52921 D0L6QN 10070040 Ki = 24 nM T52921 D0L8YY 10066285 Ki = 5.7 nM T52921 D0M7TP 44456412 IC50 = 14.9 nM T52921 D0NE3U 5485199 IC50 > 10000 nM T52921 D0O7JV 44426810 Ki = 14 nM T52921 D0P3FP 44426808 Ki = 5 nM T52921 D0PN2C 44456140 IC50 = 2.81 nM T52921 D0PR2Q 44456220 EC50 = 27.6 nM T52921 D0Q2PO 25084509 Ki = 0.54 nM T52921 D0Q9TQ 10043898 Ki = 54 nM T52921 D0QH4A 10089987 Ki = 14 nM T52921 D0S2OA 10388166 Ki = 162 nM T52921 D0SE9S 9887077 Ki = 0.3 nM T52921 D0SN6V 44456299 EC50 = 46.5 nM T52921 D0T0GL 44456296 IC50 = 0.66 nM T52921 D0T4ZY 44426817 Ki = 134 nM T52921 D0T9KE 44430016 Ki = 85 nM T52921 D0TJ7R 97333 Ki = 1983 nM T52921 D0U6FM 44456339 IC50 = 21.7 nM T52921 D0V3OY 105104 Ki > 10000 nM T52921 D0VH3M 25088989 Ki = 0.83 nM T52921 D0W3VT 10091033 Ki = 24 nM T52921 D0W7CF 9963005 IC50 = 1.04 nM T52921 D0X4SX 10317947 Ki = 72 nM T52921 D0XX1Y 44426828 Ki = 53 nM T52921 D0Y0IE 44352919 EC50 = 1.97 nM T52921 D0Y2MT 44416158 IC50 = 11.6 nM T52921 D0Y4EW 6324645 EC50 = 0.3236 nM T52921 D0Y5LJ 10336926 Ki = 136 nM T52921 D0Y7KE 44430012 Ki = 1281 nM T52921 D0YM8F 25084510 Ki = 1.79 nM T52921 D0ZE2W 44430028 Ki = 2176 nM T98092 D02EEJ 6479267 Ki = 1.84 nM T98092 D0CE0O 11513676 Ki = 0.34 nM T98092 D0G7UX 5284373 Ki = 2.64 nM T98092 D0M2OY 53259809 Ki = 16800 nM T98092 D08MYL 6473876 Ki = 2.11 nM T98092 CY0Q4V 444384 IC50 = 2000000 nM T98092 CLYE08 497073 IC50 = 6000 nM T98092 C8SG7U 497075 IC50 > 10000000 nM T98092 CAWY91 497076 IC50 = 90000 nM T98092 CC9D3J 497077 IC50 > 10000000 nM T98092 CBMF04 497078 IC50 = 500000 nM T98092 C6KF5Y 1367020 IC50 = 580 nM T98092 CP61UY 2823177 IC50 = 920 nM T98092 CM6OW0 3190778 IC50 = 5.5 nM T98092 CDPT84 4128827 IC50 = 316 nM T98092 C7T6VH 4401642 IC50 = 14 nM T98092 CSQP36 5020377 IC50 = 303 nM T98092 CZ34OX 5116189 IC50 = 5500 nM T98092 C7DIT9 5493631 IC50 = 680000 nM T98092 C35VSF 5493632 IC50 = 1000000 nM T98092 CGN50H 5493634 IC50 = 260000 nM T98092 C8U3AT 5493635 IC50 = 115000 nM T98092 C5I2UC 5493638 IC50 = 280000 nM T98092 CNIC61 6475296 IC50 = 310 nM T98092 C8RA6C 6476061 IC50 = 11.1 nM T98092 CTXB32 6479257 IC50 = 3 nM T98092 CMH26D 6479258 IC50 = 47 nM T98092 C45EVU 6479259 IC50 = 15 nM T98092 CQ1X3C 6479260 IC50 = 61 nM T98092 C1YMW4 6479261 IC50 = 277 nM T98092 CAYZ53 6479262 IC50 = 97 nM T98092 CPCG74 6479263 IC50 = 128 nM T98092 C16CZK 6479264 IC50 = 19 nM T98092 CN1BF8 6479265 IC50 = 165 nM T98092 C8N4YK 6479266 IC50 = 110 nM T98092 CAGX82 6479268 IC50 = 6047 nM T98092 CM36KU 6479269 IC50 = 1572 nM T98092 CJWU53 6479270 IC50 = 882 nM T98092 CRV94O 6479271 IC50 = 959 nM T98092 C03LTJ 10034324 IC50 = 934 nM T98092 CODJ10 10626583 Ki = 795 nM T98092 CO9XA6 10819131 IC50 = 1500000 nM T98092 CF45ID 11516665 IC50 = 20 nM T98092 CGP87C 11531251 IC50 = 951 nM T98092 CSY31B 11559871 IC50 = 748 nM T98092 C6M1ZU 11567780 IC50 = 320 nM T98092 CJ27OG 11588606 IC50 = 140 nM T98092 CN8M2B 11617502 IC50 = 71 nM T98092 CS2Y6M 11631957 IC50 = 60 nM T98092 CX63ZC 11632684 IC50 = 60 nM T98092 CLP34W 11638938 IC50 = 592 nM T98092 CS3YJ8 11660364 IC50 = 640 nM T98092 C37WLM 11675245 IC50 = 528 nM T98092 C3SK8D 11703833 IC50 = 880 nM T98092 C2QN6F 11710570 IC50 = 1437 nM T98092 C73OMC 11717355 IC50 = 458 nM T98092 C89EKB 11718015 IC50 = 499 nM T98092 CUY92Q 13422114 IC50 = 130 nM T98092 CC6XY7 13578707 IC50 = 350 nM T98092 C8KA7W 20415061 IC50 = 460 nM T98092 C31GDL 24814873 IC50 = 14 nM T98092 C2ON4L 25044910 IC50 = 690 nM T98092 CY8HB6 25046022 IC50 = 330 nM T98092 CT2E3I 25098032 IC50 = 590 nM T98092 CK0P2Q 42630203 IC50 = 650 nM T98092 C69CNK 44248910 IC50 > 10000 nM T98092 C46XEC 44248911 IC50 = 103 nM T98092 CS6N9K 44248912 IC50 = 71.2 nM T98092 CHX9S4 44248913 IC50 = 159 nM T98092 CSDG42 44248914 IC50 > 10000 nM T98092 CJT1A8 44249039 IC50 = 364 nM T98092 CVW1T9 44249040 IC50 = 263 nM T98092 CNFI87 44249041 IC50 = 2.59 nM T98092 CW6LT7 44249042 IC50 = 1.52 nM T98092 C7U6PN 44249044 IC50 = 1910 nM T98092 C1HPV8 44249170 IC50 > 10000 nM T98092 CW4AU3 44249173 IC50 = 12.1 nM T98092 CKO3I0 44249174 IC50 > 10000 nM T98092 CL7M2J 44249303 IC50 = 620 nM T98092 C97JUQ 44249304 IC50 > 10000 nM T98092 C0SVJ1 44249305 IC50 = 31.6 nM T98092 CA3K2N 44249306 IC50 > 10000 nM T98092 CBEL85 44249307 IC50 = 370 nM T98092 C5M4VW 44249309 IC50 = 136 nM T98092 CR2K7N 44249310 IC50 > 10000 nM T98092 C57MCG 44249414 IC50 > 10000 nM T98092 CSJD94 44249415 IC50 > 10000 nM T98092 CER54N 44294512 IC50 = 2500000 nM T98092 CKYA61 44294584 IC50 = 850000 nM T98092 C4R1DL 44294708 IC50 > 10000000 nM T98092 CTE19D 44294709 IC50 > 10000000 nM T98092 CT5IJ4 44294814 IC50 = 2800000 nM T98092 C4GLS0 44294838 IC50 = 760000 nM T98092 C5EQ7U 44295020 IC50 = 1300000 nM T98092 CHI01J 44295050 IC50 = 1500000 nM T98092 CS5I9W 44295136 IC50 = 970000 nM T98092 COCG50 44295258 IC50 = 820000 nM T98092 CV7PD8 44341483 IC50 = 48 nM T98092 C5M1FB 44341507 IC50 = 256 nM T98092 CM9L8P 44365970 IC50 = 1500000 nM T98092 C50FPJ 44366040 IC50 = 2500000 nM T98092 C0JKL6 44366208 IC50 = 2600000 nM T98092 C98VGM 44366209 IC50 = 165000 nM T98092 C6PCZ9 44366232 IC50 = 850000 nM T98092 CRES48 44366233 IC50 = 325000 nM T98092 C7AQ3R 44366260 IC50 = 2100000 nM T98092 CS74HY 44366261 IC50 = 970000 nM T98092 CEH4W6 44366303 IC50 = 820000 nM T98092 CF3B2I 44366350 IC50 = 260000 nM T98092 C0I3BR 44366351 IC50 = 760000 nM T98092 C9HQ5S 44366390 IC50 = 2800000 nM T98092 CY89LF 44366391 IC50 = 1300000 nM T98092 CDJ21S 44366404 IC50 = 500000 nM T98092 CPW1A7 44366405 IC50 = 90000 nM T98092 C4SQ1N 44366450 IC50 = 280000 nM T98092 CUI2X6 44366451 IC50 = 6000 nM T98092 CMCP73 44366452 IC50 = 365000 nM T98092 C2LG1F 44366453 IC50 = 115000 nM T98092 C5Q4VN 44393426 Ki = 100 nM T98092 CP57YU 44393427 Ki = 75 nM T98092 CGX7M4 44393512 Ki = 10 nM T98092 CGP76Z 44393513 Ki = 24 nM T98092 CU0RC4 44393514 Ki = 18 nM T98092 CZAD42 44406917 IC50 = 4100 nM T98092 C0FLH5 44582698 IC50 = 740 nM T98092 C0ON5I 44582699 IC50 = 810 nM T98092 CW3R7N 44582757 IC50 = 740 nM T98092 CCV89D 44582780 IC50 = 880 nM T98092 CZM71K 44582804 IC50 = 600 nM T98092 CWF96D 44582805 IC50 = 450 nM T98092 CYN7C5 44582823 IC50 = 160 nM T98092 CW4P8K 44582824 IC50 = 450 nM T98092 CX94NI 45138814 IC50 = 2.4 nM T98092 CN72XD 45269870 IC50 > 10000 nM T98092 CS30FH 49863381 IC50 = 206 nM T98092 C3YI2V 49863382 IC50 = 950 nM T98092 CS48JU 49863383 IC50 = 4.75 nM T98092 CWI47U 50899161 IC50 = 26.6 nM T98092 CHN71J 52940634 IC50 = 31.2 nM T98092 CQ83LE 52940669 IC50 = 22.9 nM T98092 C2H0IK 52940670 IC50 = 46 nM T98092 CPKZ45 52940671 IC50 = 35.2 nM T98092 C7MA9P 52941831 IC50 = 9.12 nM T98092 CH9QA8 52941859 IC50 = 21.4 nM T98092 C97YWD 52945243 IC50 = 26.7 nM T98092 CE05IO 52945473 IC50 = 218 nM T98092 C43LWJ 52945496 IC50 = 140 nM T98092 C3BCG7 52946681 IC50 = 83.5 nM T98092 CR63JF 52946682 IC50 = 22.8 nM T98092 CH8TZ9 52946683 IC50 = 103 nM T98092 C7KW3U 52947912 IC50 = 23 nM T98092 C4KAU1 52947949 IC50 = 662 nM T98092 CGX04A 52947950 IC50 = 65.2 nM T98092 CS90AU 52952820 IC50 = 33.11 nM T98092 CBWK59 53321090 Ki = 106 nM T98092 CNS79R 53344622 IC50 = 2.7 nM T98092 CPD19A 53357115 IC50 = 350 nM T98092 CMYW90 53357116 IC50 = 630 nM T98092 C75LWY 53357117 IC50 = 500 nM T98092 C40GVQ 53357247 IC50 = 360 nM T98092 CC0Y1S 53357248 IC50 = 390 nM T98092 CPM2F7 53357386 IC50 = 330 nM T98092 COP18F 53357507 IC50 = 520 nM T98092 C4P3GC 53357508 IC50 = 420 nM T98092 C4O0YX 53357509 IC50 = 4.1 nM T98092 C96CAE 53357630 IC50 = 450 nM T98092 C8C9ZH 53358962 IC50 = 1.1 nM T98092 C3VJ0N 56668120 IC50 = 2000000 nM T98092 C30PVF 56675024 IC50 = 2600000 nM T98092 CFMP72 56678333 IC50 = 2100000 nM T98092 CFAY29 56678334 IC50 = 165000 nM T98092 CQB1I0 57384849 Ki = 14 nM T98092 CZK8P2 57384850 Ki = 65 nM T98092 CX67HU 57385085 Ki = 4 nM T98092 C6PXU0 57398046 IC50 = 4.9 nM T98092 C6ZK4A 67978739 Ki = 16 nM T98092 C6RT1L 71590783 IC50 = 740 nM T98092 CC0TY2 71590784 IC50 = 810 nM T98092 CH23LT 71596756 IC50 = 550 nM T98092 CZOT97 71596824 IC50 = 380 nM T98092 CC37ZO 71596825 IC50 = 330 nM T98092 C2IJ6X 71596826 IC50 = 460 nM T98092 CSE28O 73333514 Ki = 23 nM T98092 CDF54U 73333515 Ki = 10.7 nM T98092 CKS08Z 73333613 Ki = 12.4 nM T98092 C5FWY3 73333614 Ki = 43.9 nM T98092 C2LR7I 73333729 Ki = 11.8 nM T98092 CQH16I 73333730 Ki = 36.6 nM T98092 CRA39X 73333846 Ki = 57.7 nM T98092 C47PVY 73347049 IC50 = 680000 nM T98092 CKV1A9 73348786 IC50 = 2.3 nM T98092 CIXM26 73353051 IC50 = 16 nM T98092 C5J6GK 122437357 IC50 = 11.2 nM T98092 CUKL46 127038149 IC50 = 10000 nM T98092 CF7KS5 127038150 IC50 = 10000 nM T98092 C6HPE3 127038151 IC50 = 10000 nM T98092 CQC1L7 127038489 IC50 = 940 nM T98092 CI8EO6 127039060 IC50 = 10000 nM T98092 C7NW5Q 127039075 IC50 = 2760 nM T98092 CSU85H 127039831 IC50 = 10430 nM T98092 CA1P8V 127039832 IC50 = 10260 nM T98092 C2JQ4V 127039851 IC50 = 10000 nM T98092 C1DTR2 127039852 IC50 = 1220 nM T98092 CI03BD 127040172 IC50 = 10800 nM T98092 C0OTQ9 127040173 IC50 = 10000 nM T98092 CA75UB 127040174 IC50 = 10000 nM T98092 CC0GN1 127040175 IC50 = 10000 nM T98092 C8PI2G 127041686 IC50 = 10000 nM T98092 CS0EM4 127041788 IC50 = 10330 nM T98092 CE0KL8 127041789 IC50 = 10000 nM T98092 C35DGM 127042320 IC50 = 11620 nM T98092 C2VGI1 136220121 Ki = 64.7 nM T98092 C2ZA8L 137348679 Ki = 7 nM T98092 CY46VP 137637353 Ki = 4.3 nM T98092 D04PGW 6475368 IC50 = 166 nM T98092 D07ABJ 44358392 IC50 = 783 nM T98092 D07IQR 11639129 IC50 = 361 nM T98092 D0P6TX 3663276 IC50 = 754 nM T98092 D0X5JR 11574097 IC50 = 810 nM T52638 D03LWG 53235510 IC50 > 10000 nM T52638 D07EHV 44814409 IC50 > 10000 nM T52638 D0E3TC 44259 IC50 = 12100 nM T52638 C1ZPA9 1292979 IC50 = 623 nM T52638 C1XS2J 54760383 IC50 > 10000 nM T52638 CV63UL 67240318 IC50 > 10000 nM T52638 CM8LU3 122177129 IC50 = 420 nM T52638 CU5V7A 129318960 IC50 = 39 nM T52638 C38TVL 129318961 IC50 = 750 nM T52638 CX48MD 133080583 EC50 = 352 nM T52638 CTR4A0 135383414 IC50 = 95 nM T52638 C8MY4I 137632407 IC50 = 60 nM T52638 CTKX07 137635009 IC50 = 971 nM T52638 CLK3Y7 137635621 IC50 = 106 nM T52638 C0IMX2 137642056 Ki = 32.43 nM T52638 CVR5C8 137654407 IC50 = 2140 nM T52638 CLMT19 137660903 IC50 = 6 nM T52638 C2MD1Q 155513187 IC50 > 10000 nM T52638 D06HVH 54613583 IC50 > 10000 nM T56556 D00YZD 54726191 IC50 = 67000 nM T56556 D04AIT 5280445 IC50 = 8900 nM T56556 D07BSQ 5994 IC50 = 125892.54 nM T56556 D07POC 176870 IC50 = 50000 nM T56556 D09XZB 123631 IC50 = 1100 nM T56556 D0AZ3C 5291 IC50 = 4897.79 nM T56556 D0BP9C 193962 IC50 = 6000 nM T56556 D0J4JM 5770 IC50 = 12600 nM T56556 D0K8KX 5280343 EC50 = 30 nM T56556 D0OB1J 39186 IC50 = 851138.04 nM T56556 D0Q0PR 54675769 IC50 = 104000 nM T56556 D0R0FE 2520 EC50 = 900 nM T56556 D0R3JB 4212 IC50 = 903.8 nM T56556 D0T0KA 4474 IC50 = 16595.87 nM T56556 D01GFX 11640390 EC50 = 104 nM T56556 D02HTD 25167947 IC50 = 1400 nM T56556 D02QWY 24785538 IC50 = 10200 nM T56556 D0CE0O 11513676 IC50 = 2500 nM T56556 D0G7UX 5284373 EC50 = 1750 nM T56556 D0J1HB 23063810 IC50 = 65400 nM T56556 D0L4FS 5280961 IC50 = 6900 nM T56556 D00OWF 5280953 IC50 = 5080 nM T56556 D04RLX 148201 EC50 = 10 nM T56556 D09FGX 119373 IC50 = 400 nM T56556 D0Q7HO 4705 IC50 = 1730 nM T56556 C4DS3F 2361 IC50 = 6050 nM T56556 CQ9MW6 68077 IC50 = 17000 nM T56556 CJ65ZE 72344 IC50 = 4900 nM T56556 CSHM20 73201 IC50 = 8900 nM T56556 CI5UP7 88881 IC50 = 9200 nM T56556 C5ZCH7 97332 IC50 = 1880 nM T56556 CL97OF 97548 IC50 = 1280 nM T56556 CD8L6K 97696 IC50 = 7900 nM T56556 C6I9HU 97860 IC50 = 19000 nM T56556 C3NC7T 114429 IC50 = 11000 nM T56556 C8NLJ2 145659 IC50 = 8300 nM T56556 CNVB16 146013 IC50 = 1280 nM T56556 C4FEY6 147157 IC50 = 3400 nM T56556 C7E5NC 150893 IC50 = 1400 nM T56556 C4J5ZF 185617 IC50 = 10000 nM T56556 CRE67B 265724 IC50 = 1010 nM T56556 CABJ72 276138 IC50 = 1230 nM T56556 C1Q0WH 281852 IC50 = 1690 nM T56556 CPF26C 324081 IC50 = 10700 nM T56556 C4VJH5 324094 IC50 = 16600 nM T56556 CMC10D 324099 IC50 = 9000 nM T56556 CP5B4K 369597 IC50 = 4900 nM T56556 CKC6U2 369599 IC50 = 2800 nM T56556 CO6AM3 378567 IC50 = 17000 nM T56556 CA9IM5 396723 IC50 = 860 nM T56556 CVN3Z5 403923 IC50 = 451 nM T56556 C5YX1H 406017 IC50 = 30000 nM T56556 CHP8G0 406584 IC50 = 960 nM T56556 CWXZ47 406585 IC50 = 15000 nM T56556 CL6QB8 407032 IC50 = 4800 nM T56556 CC1Q8J 409920 IC50 = 6300 nM T56556 C3YG0Z 436659 IC50 > 20000 nM T56556 CWZ14N 468116 IC50 > 20000 nM T56556 CMT3P0 480764 IC50 = 3100 nM T56556 CL6E7C 609712 IC50 = 10000 nM T56556 C14NHZ 624831 IC50 = 12400 nM T56556 C34KNT 631171 IC50 = 2140 nM T56556 CSA18D 651672 IC50 = 940 nM T56556 C90LPE 688666 IC50 = 6500 nM T56556 CMR6U0 693195 IC50 = 2630 nM T56556 CH0DT9 693197 IC50 = 150 nM T56556 C1NZL9 693198 EC50 = 72 nM T56556 CW2U6N 698956 IC50 = 130 nM T56556 C19VMW 698960 EC50 = 72 nM T56556 C65SGT 712193 IC50 = 645 nM T56556 CH6MV7 715632 IC50 = 6380 nM T56556 C2NI7K 718862 IC50 = 890 nM T56556 CNS78D 719277 IC50 = 1150 nM T56556 CST9W8 719279 IC50 = 1480 nM T56556 CEC0X3 719282 IC50 = 2250 nM T56556 CRX4Q5 719284 IC50 = 1930 nM T56556 C6AKG9 735124 IC50 = 8120 nM T56556 C8OB6U 787509 EC50 = 50 nM T56556 C64RUF 877998 EC50 = 70 nM T56556 CXR0P5 917533 IC50 = 15800 nM T56556 C2X8PT 930478 IC50 = 108 nM T56556 CXQ4P8 1183964 IC50 = 944 nM T56556 CB31HC 1186125 IC50 = 362 nM T56556 CM42KO 1187243 IC50 = 107.15 nM T56556 CYT7E4 1214451 EC50 = 13 nM T56556 CCNX23 1361994 IC50 = 216 nM T56556 C35OEM 1413870 IC50 = 28900 nM T56556 CV7F8O 1418188 IC50 = 405 nM T56556 CAXQ59 1424290 IC50 = 2780 nM T56556 C2FL5J 1553837 IC50 = 250 nM T56556 C5RA6J 1566118 IC50 = 166 nM T56556 CQYO27 1597005 IC50 = 10700 nM T56556 C0M7DO 1696333 IC50 = 1340 nM T56556 COAE97 2176800 IC50 = 1060 nM T56556 C6ZFC1 2463411 IC50 = 791 nM T56556 CG3V9C 2549745 IC50 = 224 nM T56556 C2ZDU4 2562583 IC50 = 570 nM T56556 CFC30O 2789499 EC50 = 11 nM T56556 C01JRM 3034694 IC50 = 9300 nM T56556 C69NQO 3627000 EC50 = 58 nM T56556 C72VLI 4022553 IC50 = 196 nM T56556 C43JKM 4271896 IC50 = 3860 nM T56556 CHV3N6 4786429 IC50 = 360 nM T56556 CKG0Q7 4839583 IC50 = 724 nM T56556 CGKX02 4841865 IC50 = 1320 nM T56556 CN35MZ 4970131 IC50 = 11800 nM T56556 C8PN0C 5280682 IC50 = 680 nM T56556 CF6KZ2 5281677 IC50 = 17200 nM T56556 CQ9GX3 5320462 IC50 = 2000 nM T56556 C2TVO1 5328202 IC50 = 1980 nM T56556 C0O4SM 5332516 IC50 = 2630 nM T56556 CI6TE3 5348770 IC50 = 9230 nM T56556 CTO51S 5352005 IC50 = 540 nM T56556 CQL05G 5355469 IC50 = 3000 nM T56556 CTPE71 5355684 IC50 = 3280 nM T56556 CN8GP9 5355845 IC50 = 16200 nM T56556 C9T0DZ 5355846 IC50 = 10500 nM T56556 CW1UM5 5357488 IC50 = 2200 nM T56556 CU29TR 5373259 IC50 = 530 nM T56556 CV7Z2A 5373273 IC50 = 1060 nM T56556 CRW09S 5373997 IC50 = 3090 nM T56556 C09NZD 5380645 IC50 = 31020 nM T56556 C2KZF0 5476176 IC50 = 2400 nM T56556 CO17YB 5702790 IC50 = 1730 nM T56556 CI4U9Z 5711223 IC50 = 12050 nM T56556 CVF14X 5712116 IC50 = 4970 nM T56556 CCAT78 5723044 IC50 = 2190 nM T56556 CR51QS 5729243 IC50 = 22390 nM T56556 CG25KB 5729341 IC50 = 1950 nM T56556 CE0W8M 5730384 IC50 = 7800 nM T56556 CD18KY 5730712 EC50 = 2100 nM T56556 CA9WL4 5797184 IC50 = 18200 nM T56556 C7LKC3 5822497 IC50 = 10720 nM T56556 C29JCA 5909266 IC50 = 3320 nM T56556 CDLV62 5936200 IC50 = 2200 nM T56556 C9DB2C 5953849 IC50 = 850 nM T56556 CG82WY 5978982 IC50 = 2820 nM T56556 CFO1R0 6063342 IC50 = 1910 nM T56556 CP8O7I 6070899 IC50 = 1470 nM T56556 CMC06O 6123891 IC50 = 6440 nM T56556 C90ACD 6199559 IC50 = 9830 nM T56556 CYX45A 6213016 IC50 = 4910 nM T56556 CV91FR 6213967 EC50 = 1250 nM T56556 C6SZW5 6229071 IC50 = 7290 nM T56556 CU3X5P 6229072 IC50 = 9210 nM T56556 CFO9D1 6256073 IC50 = 8700 nM T56556 CX87NG 6475921 IC50 = 12300 nM T56556 COF72V 6919145 IC50 = 910 nM T56556 C0MGV7 7048595 IC50 = 3790 nM T56556 CNH60W 7946188 IC50 = 7220 nM T56556 C0O7PG 9109771 IC50 = 810 nM T56556 CLIG51 9281828 IC50 = 753 nM T56556 C1IPS5 9283400 EC50 = 85 nM T56556 C0D2SZ 9448204 IC50 = 4280 nM T56556 C4CF5U 9448550 EC50 = 512 nM T56556 C40XDF 9880195 EC50 = 14 nM T56556 CHI5S9 9975676 IC50 = 5910 nM T56556 C26IPN 10047854 IC50 = 5700 nM T56556 CY73KI 10322450 IC50 = 4 nM T56556 C7QYK3 10359377 IC50 = 830 nM T56556 C7Z8IW 10379829 IC50 = 4250 nM T56556 C0V5QI 10394010 IC50 = 11000 nM T56556 CT9MP2 10404096 IC50 = 3800 nM T56556 C36PIN 10407830 IC50 = 8190 nM T56556 C78HZG 10495050 IC50 = 6160 nM T56556 CR9SE7 10540319 IC50 = 6370 nM T56556 CEZ2B4 10612087 IC50 = 1940 nM T56556 CIOL78 10699195 IC50 = 16000 nM T56556 CF1UM5 10746774 IC50 = 29000 nM T56556 CI1RC8 10830017 IC50 = 9100 nM T56556 CT8PY0 10899903 IC50 > 20000 nM T56556 CDX92T 11210677 IC50 = 2460 nM T56556 CL1YX5 11246927 IC50 = 3620 nM T56556 C0SO6D 11312797 IC50 = 930 nM T56556 CL3YO1 11537442 IC50 = 700 nM T56556 C2C3WI 11957988 IC50 = 2089.3 nM T56556 C47ZJY 11996857 IC50 = 20000 nM T56556 CR3X7L 12388142 IC50 = 2890 nM T56556 C0KZQ2 12388145 IC50 = 5210 nM T56556 CS4YL1 12511782 IC50 = 2140 nM T56556 CRE67S 12753643 IC50 = 2580 nM T56556 CT24DO 13147509 IC50 = 920 nM T56556 C5VXB4 13147512 IC50 = 3550 nM T56556 C4GZ8Y 13168110 EC50 = 41 nM T56556 C5X4VH 13250463 IC50 > 20000 nM T56556 CM28RZ 13329020 IC50 = 424 nM T56556 C1U9IN 13707046 IC50 = 2890 nM T56556 C5DMA3 14034811 IC50 = 260 nM T56556 CRIH25 14259001 IC50 = 6600 nM T56556 CG0ZK1 14531326 EC50 = 900 nM T56556 C2LA5S 15556477 IC50 = 5680 nM T56556 CJ78CV 15648569 IC50 = 720 nM T56556 CJ5XV3 15965811 IC50 > 100000 nM T56556 C19FNV 15993184 EC50 = 12 nM T56556 CLD92G 15999199 EC50 = 4.7 nM T56556 C0A3IV 16092354 IC50 = 1190 nM T56556 C3TH4N 16092356 IC50 = 689 nM T56556 C7DW6Y 16092357 EC50 = 131 nM T56556 C7TBI5 16339054 IC50 = 15400 nM T56556 CMVW98 16618023 EC50 = 1310 nM T56556 CD04RW 16745324 IC50 = 2500 nM T56556 CN73EP 16805556 IC50 = 4790 nM T56556 CPOZ18 17375361 IC50 = 11200 nM T56556 CX06NR 17412108 IC50 = 16000 nM T56556 C5MOF7 17497142 IC50 = 10400 nM T56556 COG12F 17585222 IC50 = 8680 nM T56556 CPE15U 18004103 IC50 = 14500 nM T56556 CYSV63 19392346 IC50 = 60000 nM T56556 C3UT8G 20239593 IC50 = 170 nM T56556 CJ4Z1L 20646908 IC50 = 20900 nM T56556 C59FWO 20646970 IC50 = 51300 nM T56556 CIZV45 20646979 IC50 = 40000 nM T56556 CB7T2K 20963109 EC50 = 1.2 nM T56556 C2RQF6 21002393 IC50 = 1180 nM T56556 CB50QE 21418982 IC50 = 648 nM T56556 CCJ3M5 22004538 IC50 = 32400 nM T56556 CFI13S 22310708 IC50 = 420 nM T56556 CDQX04 22330280 IC50 = 462 nM T56556 C9IHU3 22330507 IC50 = 1990 nM T56556 C85SLA 23792651 IC50 = 8900 nM T56556 C7TOB4 23906108 IC50 = 1660 nM T56556 CU1G8A 23940255 IC50 = 87.1 nM T56556 CRCA82 23965087 EC50 = 21 nM T56556 CX2UF8 24016488 IC50 = 612 nM T56556 C2XB8M 24017959 IC50 = 183 nM T56556 C3ESV6 24178402 EC50 = 90000 nM T56556 C6AU1C 24204512 IC50 = 790 nM T56556 CU7LR8 24208774 IC50 = 458 nM T56556 CLY6U7 24626581 IC50 = 921 nM T56556 CCPS81 24764502 IC50 = 35000 nM T56556 CKW04J 24807980 EC50 = 7000 nM T56556 CJUW92 24807981 EC50 = 1500 nM T56556 CP8H2D 24807987 EC50 = 58000 nM T56556 C9T7BZ 24808155 EC50 = 75000 nM T56556 C9SMO0 24808156 EC50 = 120000 nM T56556 CW4EM8 24808157 EC50 = 150000 nM T56556 C7UV4H 24808344 EC50 = 500 nM T56556 C9F8CE 24826109 IC50 = 430 nM T56556 C9LXA0 24827935 IC50 = 350 nM T56556 C39SHG 24882446 IC50 = 23988.33 nM T56556 CF1JU8 24978503 IC50 = 230 nM T56556 C60EJI 25113688 EC50 = 73000 nM T56556 CS3ZN9 25195356 IC50 = 350 nM T56556 C2YA4G 25217469 IC50 = 1750 nM T56556 CM80XH 25222999 IC50 = 60 nM T56556 CSRV83 25223000 IC50 = 172 nM T56556 C26ZQR 25223001 IC50 = 632 nM T56556 C0S7AF 25223002 IC50 = 317 nM T56556 CZ4A5K 25223105 IC50 = 858 nM T56556 CKY89F 25223106 IC50 = 1990 nM T56556 CIJU21 25223199 IC50 = 119 nM T56556 CUZ5S9 25223200 IC50 = 183 nM T56556 C03FQV 25223201 IC50 = 552 nM T56556 C8S6UH 25223298 IC50 = 1015 nM T56556 CZQE36 25223299 IC50 = 977 nM T56556 C6O2ZR 25225119 EC50 = 30000 nM T56556 C8W9VD 25249649 IC50 > 10000 nM T56556 C78LKG 26213315 IC50 = 4100 nM T56556 CJPM47 31538107 IC50 = 1350 nM T56556 CI4AK1 39969954 IC50 = 14400 nM T56556 C0X8OT 44221093 IC50 = 10200 nM T56556 C9BNA1 44248179 EC50 = 63.2 nM T56556 C4DBF9 44257640 IC50 = 5900 nM T56556 C2NK1G 44428701 IC50 = 770 nM T56556 C4NCQ7 44428711 IC50 > 20000 nM T56556 CUIG60 44428712 IC50 = 450 nM T56556 CQ6A3K 44428713 IC50 = 560 nM T56556 CNBA28 44428714 IC50 = 1380 nM T56556 C43CIH 44451513 IC50 = 77624.71 nM T56556 CMHP85 44451563 IC50 = 263026.8 nM T56556 C29SBO 44451564 IC50 = 6606.93 nM T56556 C1G2CB 44451590 IC50 = 7585.78 nM T56556 C6NW0Q 44451617 IC50 = 14454.4 nM T56556 C1ENZ0 44451645 IC50 = 44668.36 nM T56556 CB0OL9 44451671 IC50 = 6025.6 nM T56556 CC9LK5 44451719 IC50 = 6025.6 nM T56556 CS4RX9 44451745 IC50 = 7244.36 nM T56556 C9Z4VY 44451773 IC50 = 12882.5 nM T56556 CTP09O 44451801 IC50 = 11481.54 nM T56556 CP69AF 44451832 IC50 = 22908.68 nM T56556 C45VCM 44451857 EC50 = 15000 nM T56556 C4T5UP 44451866 IC50 = 21877.62 nM T56556 CI1Y5L 44451888 IC50 = 64565.42 nM T56556 CP3B8R 44451889 IC50 = 36307.81 nM T56556 C3S5OK 44451912 IC50 = 5011.87 nM T56556 C6M3ZN 44451913 IC50 = 47863.01 nM T56556 C9AOQ4 44562411 IC50 = 15135.61 nM T56556 CLBO81 44565459 IC50 = 9080 nM T56556 C7NRZ8 44565460 IC50 = 6760 nM T56556 CN03BJ 44565480 IC50 = 2610 nM T56556 C38FXL 44565481 IC50 = 58400 nM T56556 CZUI80 44565482 IC50 = 74100 nM T56556 CZT54M 44565509 IC50 = 74100 nM T56556 C4Q2ER 44593438 IC50 = 24547.09 nM T56556 CE6F2U 45272659 IC50 = 22600 nM T56556 COPA25 46227750 IC50 = 10200 nM T56556 COA30H 46227751 IC50 = 630 nM T56556 CLWR13 46227752 IC50 = 500 nM T56556 C54HFY 46232422 IC50 > 100000 nM T56556 C5TJ4Y 46232423 IC50 = 25200 nM T56556 CY2RN7 46232494 IC50 > 100000 nM T56556 CW9J2R 46232495 IC50 > 100000 nM T56556 CO7V0S 46232496 IC50 > 100000 nM T56556 CZ89LA 46232497 IC50 = 15400 nM T56556 C4RUB7 46232498 IC50 = 6400 nM T56556 CR96LU 46232536 IC50 = 18800 nM T56556 C6UW4G 46232537 IC50 = 11100 nM T56556 C5ATF2 46232538 IC50 = 23200 nM T56556 CKXH76 46232539 IC50 > 100000 nM T56556 CXI72Q 46359934 IC50 = 1430 nM T56556 C0L6DC 46359963 IC50 = 60 nM T56556 CD64QE 49816175 IC50 = 1270 nM T56556 C72QDG 49844541 IC50 = 8920 nM T56556 CY4XL9 50806112 IC50 = 1890 nM T56556 C5PHF6 51041756 IC50 = 15500 nM T56556 C5M9DP 51041990 IC50 = 8400 nM T56556 CL29IG 53321447 IC50 = 6500 nM T56556 CPL41H 54341571 IC50 = 13600 nM T56556 C4Z7MF 54580539 IC50 > 100000 nM T56556 C96NWY 54580541 IC50 > 6200 nM T56556 CN30LW 54581539 IC50 > 5000 nM T56556 C6AIG3 54582535 IC50 = 183 nM T56556 CY24RJ 54582627 IC50 = 508 nM T56556 CN38OK 54583506 IC50 > 50000 nM T56556 CLTM38 54586400 IC50 > 50000 nM T56556 CK52PH 54586413 IC50 = 130 nM T56556 CIAU38 54587418 IC50 > 50000 nM T56556 CKZ01T 54587433 IC50 = 390 nM T56556 CB4DX1 54754510 IC50 = 450 nM T56556 CS7XP1 54754512 IC50 = 350 nM T56556 C4WO8B 56681840 IC50 = 270 nM T56556 C1H9ML 56764960 IC50 = 1390 nM T56556 C5EN2Q 56924700 IC50 = 170 nM T56556 CTX1N3 56924701 EC50 = 31 nM T56556 CP1VK5 56951135 IC50 = 16300 nM T56556 C2SF8B 56951136 IC50 = 470 nM T56556 C2KMN3 56951137 IC50 = 180 nM T56556 CAT80Q 56951138 IC50 = 200 nM T56556 CJ8C4Y 56951261 IC50 = 160 nM T56556 C0N9YK 57394942 IC50 = 7260 nM T56556 CTN9Q0 57396989 IC50 = 940 nM T56556 CR8MW5 57398461 IC50 = 1930 nM T56556 C9LPN4 57400130 IC50 = 3210 nM T56556 CW7B0M 57614266 IC50 = 2210 nM T56556 CQZS56 66636984 IC50 = 4100 nM T56556 C5RHD4 66637000 IC50 = 230 nM T56556 C5IT4O 70686509 IC50 = 28200 nM T56556 C9Y1TS 70686876 IC50 = 3270 nM T56556 C9B5TD 70690679 IC50 = 13300 nM T56556 CA1WO9 70696907 IC50 = 4300 nM T56556 CE1QO3 71296003 EC50 = 42 nM T56556 C2YIM8 71449571 IC50 = 5120 nM T56556 C7VGS2 71453183 IC50 = 1530 nM T56556 C1ZHB6 71453184 IC50 = 8220 nM T56556 C6ZOP0 71453185 IC50 = 970 nM T56556 CY5LI4 71454921 IC50 = 7950 nM T56556 C3OLA2 71454922 IC50 = 9350 nM T56556 C5T0NL 71454923 IC50 = 152 nM T56556 C0CIZ8 71458549 IC50 = 5910 nM T56556 CTWA64 71458550 IC50 = 5930 nM T56556 C0U5FJ 71458829 IC50 = 112 nM T56556 CA02ZE 71460396 IC50 = 3750 nM T56556 CZS0L5 71460397 IC50 = 2460 nM T56556 CPQ16X 71462088 IC50 = 6830 nM T56556 C4ZD2W 71492590 IC50 = 207 nM T56556 C0P6IG 71492759 IC50 = 176 nM T56556 C3T8ZF 71560811 EC50 = 18 nM T56556 CFN89Y 71560812 EC50 = 500 nM T56556 C42SMF 71560938 EC50 = 10000 nM T56556 C98LPJ 71560939 EC50 = 1000 nM T56556 CWCJ73 71624433 IC50 = 1100 nM T56556 CN3KI6 71624434 IC50 = 3214 nM T56556 C9RD7L 71624435 IC50 = 760 nM T56556 CGA8B3 71624544 IC50 = 544 nM T56556 C8YT2N 71624545 IC50 = 1461 nM T56556 CI7QT2 71624546 IC50 = 641 nM T56556 CA7P8Q 71624648 IC50 = 1540 nM T56556 C18BKV 71624649 IC50 = 1031 nM T56556 CMA90D 71624650 IC50 = 237 nM T56556 C3KVP8 71624651 IC50 = 591 nM T56556 CB40GR 71624766 IC50 = 943 nM T56556 CEF9J8 71624767 IC50 = 839 nM T56556 C0Z3PN 71682039 EC50 > 100000 nM T56556 CV5Z9M 71682040 EC50 > 100000 nM T56556 C1IZT7 71682041 EC50 > 100000 nM T56556 COV12T 71682195 EC50 > 100000 nM T56556 C3Y4FW 71682196 EC50 > 100000 nM T56556 CLF3I8 71682197 EC50 > 100000 nM T56556 CN6Q3L 71696716 EC50 = 12.3 nM T56556 CQCF98 71724480 EC50 = 29.5 nM T56556 C1PR7Z 71724504 EC50 = 7.2 nM T56556 CA7K8Z 71724506 EC50 = 57.5 nM T56556 CD9KH7 71724532 EC50 = 14.8 nM T56556 CWR2L5 71724556 EC50 = 0.9 nM T56556 C4ODQ2 71724557 EC50 = 160 nM T56556 C7T0UM 71724558 EC50 = 23.6 nM T56556 CUL9E2 71724582 EC50 = 38.7 nM T56556 CNW68B 71724606 EC50 = 371.7 nM T56556 CCZ9B3 71724628 EC50 = 18 nM T56556 C48CAR 72735227 IC50 = 400 nM T56556 CI6E4O 72735228 IC50 = 1550 nM T56556 CXWG13 72735229 EC50 = 3.5 nM T56556 CG7S2T 72735404 IC50 = 240 nM T56556 C2O8IJ 72735405 IC50 = 190 nM T56556 CVZK97 72735406 IC50 = 260 nM T56556 CFL45O 72735407 IC50 = 110 nM T56556 CKF0Q7 72735408 IC50 = 680 nM T56556 C5I7XA 72735580 IC50 = 610 nM T56556 CY20ED 72735581 IC50 = 470 nM T56556 C6D7QV 72735582 IC50 = 320 nM T56556 CR91NX 72735583 IC50 = 1520 nM T56556 CQ5NB6 72950792 IC50 = 426 nM T56556 CF57OZ 73346145 IC50 = 1060 nM T56556 CUX0H5 73346146 IC50 = 4270 nM T56556 C90GUQ 73347669 IC50 = 3070 nM T56556 C7KIJ0 73349189 IC50 = 2440 nM T56556 CC9F2B 73349190 IC50 = 11100 nM T56556 C7DAJ3 73352266 IC50 = 4970 nM T56556 CK3EX6 73355255 IC50 = 2710 nM T56556 CKH8D4 73355256 IC50 = 6120 nM T56556 C7NTB0 73356802 IC50 = 457 nM T56556 CIWH89 73356803 IC50 = 17900 nM T56556 C25AUR 73356804 IC50 = 4840 nM T56556 C8NC1P 76310339 EC50 = 220 nM T56556 CBDY35 76310340 EC50 = 570 nM T56556 CH9B2W 76317551 EC50 = 570 nM T56556 CVN95Y 76317552 EC50 = 530 nM T56556 C2U1VA 76321285 EC50 = 100 nM T56556 C3T5OH 76324898 EC50 = 1670 nM T56556 CCP3L1 76324899 IC50 > 2000 nM T56556 CD4V0F 76328460 IC50 = 250 nM T56556 CZ3P5R 76332141 EC50 = 80 nM T56556 C7ISD3 76335756 EC50 = 500 nM T56556 CPJ5M2 76335757 EC50 = 1270 nM T56556 CZ4SE6 76335758 EC50 = 500 nM T56556 C67ASV 76335759 EC50 = 1110 nM T56556 C5Z3GF 76335761 EC50 = 600 nM T56556 C73WDV 85922974 IC50 > 10000 nM T56556 CRB93S 89784681 EC50 = 69.3 nM T56556 CG71EX 89784708 EC50 = 28 nM T56556 C4ZOX6 89784717 EC50 = 190 nM T56556 C0ZQO6 89784722 EC50 = 32.8 nM T56556 C4U5CZ 89784733 EC50 = 54 nM T56556 CW17YB 89784735 EC50 = 59 nM T56556 C0VD4P 89784742 EC50 = 34.1 nM T56556 CZT7B9 89784751 EC50 = 47 nM T56556 CH70XJ 89784752 EC50 = 24.9 nM T56556 C6MRA2 89784753 EC50 = 24.5 nM T56556 C1JH4L 89784756 EC50 = 230 nM T56556 CN1RD8 89784760 EC50 = 195 nM T56556 C2YB6Q 89784818 EC50 = 54 nM T56556 CSK8X6 89784827 EC50 = 15.5 nM T56556 CENX80 89785043 EC50 = 32.5 nM T56556 CY46QV 89785047 EC50 = 17.5 nM T56556 CQL7T6 89785059 EC50 = 17 nM T56556 CENR59 89785064 EC50 = 235 nM T56556 CVZG56 89785117 EC50 = 86.1 nM T56556 CT43OU 89785127 EC50 = 32 nM T56556 C3FB6Q 89785132 EC50 = 30.5 nM T56556 C4S9WG 89785146 EC50 = 20 nM T56556 CCE95J 89785148 EC50 = 16.5 nM T56556 C9SBA1 89785178 EC50 = 90 nM T56556 CSI51G 89785190 EC50 = 19.7 nM T56556 CGB2P5 89785210 EC50 = 302.5 nM T56556 CTY1H5 89785238 EC50 = 48 nM T56556 CHGX10 89785254 EC50 = 195 nM T56556 CB1FR2 89794901 EC50 = 3.3 nM T56556 C43AXK 89795130 EC50 = 82.5 nM T56556 C70LJV 89795278 EC50 = 242.5 nM T56556 CFU4W2 89795305 EC50 = 152.5 nM T56556 CVB23M 89795326 EC50 = 3.6 nM T56556 CX1W9Z 89795330 EC50 = 0.9 nM T56556 C7XG4U 89795333 EC50 = 111 nM T56556 C7W1TP 89795335 EC50 = 36 nM T56556 CAX9S0 89795337 EC50 = 3.3 nM T56556 COB3Z9 89795340 EC50 = 1.7 nM T56556 C6BW0Q 89795341 EC50 = 15.8 nM T56556 COVK20 90142631 IC50 > 25000 nM T56556 CUHC90 90469229 EC50 = 3600 nM T56556 C05JQB 90469230 EC50 = 2500 nM T56556 C41EMT 90469289 EC50 = 1300 nM T56556 CA1VH0 90469291 EC50 = 2600 nM T56556 C4NX2Q 90469293 EC50 = 2600 nM T56556 C0NW8T 90469355 EC50 = 700 nM T56556 CJK73Q 90655473 EC50 = 700 nM T56556 CFX2C0 90655474 EC50 = 300 nM T56556 CYU3G9 90655475 EC50 = 400 nM T56556 CGWI98 90655476 EC50 = 15 nM T56556 C1D9TM 90655477 EC50 = 1400 nM T56556 C8A9RT 90655478 EC50 = 1100 nM T56556 CHKF72 90655479 EC50 = 2300 nM T56556 CFS75L 90655480 EC50 = 800 nM T56556 CA57QF 90655481 EC50 = 1300 nM T56556 C78PYH 90655482 EC50 = 500 nM T56556 CM1X5R 90655483 EC50 = 1100 nM T56556 CSD17I 90655484 EC50 = 1800 nM T56556 CF4Z8T 91669184 IC50 = 600 nM T56556 C3G6AI 91964346 IC50 = 953 nM T56556 CL15PA 91964352 IC50 = 300 nM T56556 C8BRG2 101876951 EC50 = 200 nM T56556 C24YLQ 101913604 IC50 = 490 nM T56556 CYM1I6 101913605 IC50 = 1600 nM T56556 CQ81YV 101913606 IC50 = 210 nM T56556 C86WSC 117777746 EC50 = 5.2 nM T56556 C9E0BT 117777811 EC50 = 4.1 nM T56556 C9YPJ7 117803128 EC50 = 25.5 nM T56556 C2UY8J 118017356 IC50 = 1700 nM T56556 CP14NL 118017358 IC50 = 1810 nM T56556 C7L8PT 118017419 IC50 = 1700 nM T56556 C7YH4G 118017423 IC50 = 610 nM T56556 C0OQ9P 118716252 EC50 = 4100 nM T56556 CK0H3V 118716255 EC50 = 400 nM T56556 C3VRT8 118716258 EC50 = 1500 nM T56556 CNS3X0 118716259 EC50 = 1300 nM T56556 CS9IV4 118716261 EC50 = 400 nM T56556 C5FD4B 118716262 EC50 = 800 nM T56556 C3BY1A 118716264 EC50 = 600 nM T56556 CLAZ45 118716265 EC50 = 3000 nM T56556 C62JPR 118716267 EC50 = 3400 nM T56556 C6JIC7 118717839 EC50 = 700 nM T56556 CLAF39 118719581 IC50 = 310 nM T56556 CHIB60 118719582 IC50 = 700 nM T56556 CFGK85 118719583 IC50 = 3000 nM T56556 CXO3V7 118719584 IC50 = 20000 nM T56556 CPI2F5 118719585 IC50 = 610 nM T56556 CCI1E7 118737162 IC50 = 184 nM T56556 C0D4GP 118737164 IC50 = 100 nM T56556 C5WYN2 118737166 IC50 = 261 nM T56556 CGT48U 118737167 IC50 = 78.9 nM T56556 CC8Q3G 118737168 IC50 = 118 nM T56556 CNZ06S 118737171 IC50 = 137 nM T56556 C3M9PE 118737173 IC50 = 451 nM T56556 C8O2WM 118737174 IC50 = 11200 nM T56556 C41ROW 118737175 IC50 = 106 nM T56556 C2UZG9 118737176 IC50 = 269 nM T56556 CUSI65 118737177 IC50 = 201 nM T56556 C85ZHJ 118737178 IC50 = 117 nM T56556 CR75MD 118737179 IC50 = 73 nM T56556 CEM28H 118737180 IC50 = 180 nM T56556 C3IH1T 118737181 IC50 = 64.2 nM T56556 C5SRA7 118737182 IC50 = 79.4 nM T56556 CU6EP1 122179376 IC50 = 357 nM T56556 CIL20J 122179390 IC50 = 45 nM T56556 C0OUW1 122179391 IC50 = 38 nM T56556 CRF71Q 122420973 IC50 = 1810 nM T56556 CCE46L 126587406 EC50 = 3.9 nM T56556 CN0LZ6 126739167 IC50 = 2330 nM T56556 CSR0Y7 127028060 IC50 > 100000 nM T56556 C8Z2XI 127028354 IC50 > 100000 nM T56556 C8Q9DG 127028355 IC50 > 100000 nM T56556 CRI72H 127028356 IC50 > 100000 nM T56556 C5A1NO 127028392 IC50 = 9640 nM T56556 CUC9I4 127040367 IC50 > 100000 nM T56556 C0I9VF 127040368 IC50 > 100000 nM T56556 CX9JE1 127040369 IC50 = 34900 nM T56556 CRM9W5 127040370 IC50 = 12000 nM T56556 CJY60W 127042304 IC50 > 100000 nM T56556 CO2P8K 127042305 IC50 = 99700 nM T56556 C56HDS 127042306 IC50 = 37600 nM T56556 CZ0E5J 127042554 IC50 = 230 nM T56556 C90ELS 127042555 IC50 = 230 nM T56556 C87PMI 127042802 IC50 = 87800 nM T56556 CRQ7U8 127042918 IC50 = 36900 nM T56556 C39PWZ 127042920 IC50 = 66600 nM T56556 C21DSU 127042921 IC50 > 100000 nM T56556 C6UZ7C 127042922 IC50 > 100000 nM T56556 CSBM31 127042943 IC50 = 12200 nM T56556 C12BJD 127042944 IC50 = 38200 nM T56556 C42ZKN 127044753 IC50 = 210 nM T56556 CA8P0B 127044754 IC50 = 310 nM T56556 CUF52K 127044901 IC50 = 840 nM T56556 CF3ML0 127044902 IC50 = 680 nM T56556 C7GXK0 127044903 IC50 = 1230 nM T56556 CP1K0B 127044904 IC50 = 390 nM T56556 CO3AX7 127044909 IC50 = 290 nM T56556 C63KNP 127044910 IC50 = 880 nM T56556 CP2U0C 127044913 IC50 = 360 nM T56556 C9SE5Y 127044914 IC50 = 3130 nM T56556 CB4JL3 127044915 IC50 = 1090 nM T56556 C9Z8XO 127045057 IC50 = 1710 nM T56556 C3FG1L 127045064 IC50 = 190 nM T56556 CM1B6D 127045208 IC50 = 1300 nM T56556 CZAL20 127045209 IC50 = 890 nM T56556 C4DH6E 127045210 IC50 = 320 nM T56556 CFX5J3 127045211 IC50 = 460 nM T56556 C5F2BE 127045212 IC50 = 970 nM T56556 CYT62M 127045213 IC50 = 680 nM T56556 C6R5MV 127045214 IC50 = 600 nM T56556 CZBJ54 127048170 IC50 = 8710 nM T56556 C6L0AF 127049502 IC50 = 8240 nM T56556 CK1SN3 127049508 IC50 = 14300 nM T56556 CB9EV4 127049509 IC50 = 6070 nM T56556 C1VP2D 127052887 IC50 = 7680 nM T56556 CG9TE5 127052888 IC50 = 9940 nM T56556 CA7N9R 127052889 IC50 = 4680 nM T56556 CX20OQ 129903920 EC50 = 10 nM T56556 CX48UI 129904103 IC50 = 1200 nM T56556 CK8S4T 132285218 IC50 = 26 nM T56556 C1WG6D 132510852 IC50 = 38 nM T56556 CH3VU5 132510853 IC50 = 29 nM T56556 C5CT0K 132547158 EC50 = 20 nM T56556 C1V7GY 134129908 IC50 = 127 nM T56556 C9VJC1 134129912 IC50 > 10000 nM T56556 CK1TS2 134129976 IC50 = 280 nM T56556 CQ5N3X 134129987 IC50 = 129 nM T56556 C3B1NJ 134130004 IC50 > 10000 nM T56556 CDG0S3 134130015 IC50 = 66.9 nM T56556 C13RTP 134130119 IC50 = 212 nM T56556 CG0NC4 134130126 IC50 = 117 nM T56556 C71PUG 134130154 IC50 = 308 nM T56556 CM40NH 134130306 IC50 > 10000 nM T56556 CCP16R 134130324 IC50 > 10000 nM T56556 C7EVF0 134130371 IC50 = 4390 nM T56556 CR6Z4W 134130497 IC50 = 150 nM T56556 C90RDH 134130514 IC50 = 223 nM T56556 CA7QF6 134130525 IC50 = 319 nM T56556 CZF1D2 134130601 IC50 = 168 nM T56556 CYLW12 134130603 IC50 > 10000 nM T56556 C63NSK 134130669 IC50 = 131 nM T56556 CK15FY 134130999 IC50 = 832 nM T56556 C6LRO0 134131064 IC50 = 208 nM T56556 C36TJZ 134131208 IC50 > 10000 nM T56556 CD69RC 134131216 IC50 = 300 nM T56556 CWP09Q 134131281 IC50 = 96.6 nM T56556 CYT40U 134131325 IC50 > 10000 nM T56556 C1JP2L 134131336 IC50 = 330 nM T56556 C6GIZ2 134131389 IC50 = 251 nM T56556 CB7A2U 134131478 IC50 = 311 nM T56556 CQ8PC9 134131521 IC50 = 679 nM T56556 C1Q0BR 134131558 IC50 = 793 nM T56556 C6QKS0 134131773 EC50 = 540 nM T56556 CDJ2L0 134133476 IC50 = 7100 nM T56556 CVRT47 134134470 IC50 = 4900 nM T56556 CA18ZH 134137512 EC50 = 4350 nM T56556 CJTO68 134140233 EC50 = 340 nM T56556 CQO05X 134141004 IC50 = 7800 nM T56556 C3PIE7 134141342 IC50 = 8900 nM T56556 CPJC31 134144364 EC50 = 380 nM T56556 C9FZI6 134147046 EC50 = 86 nM T56556 CMUK36 134147167 EC50 = 910 nM T56556 C8CIP6 134148609 EC50 = 360 nM T56556 C2Z5LD 134148627 EC50 = 360 nM T56556 CXV6P1 134149485 EC50 = 550 nM T56556 CUBF46 134149834 EC50 = 280 nM T56556 C9Q4YF 134151298 EC50 = 630 nM T56556 C48WKX 134151943 EC50 = 1050 nM T56556 CE14NO 134156590 IC50 = 7400 nM T56556 C4HTR0 134156671 EC50 = 260 nM T56556 CMN2A4 135418331 IC50 = 12800 nM T56556 C41IEM 135659059 IC50 > 20000 nM T56556 CO69BC 135885017 IC50 = 11900 nM T56556 C09BGP 135885019 IC50 = 5900 nM T56556 CV4F5D 137631464 IC50 = 507 nM T56556 COU58A 137631903 EC50 = 116 nM T56556 CL7J6T 137632165 IC50 = 128 nM T56556 CD5VI8 137632443 IC50 = 1267 nM T56556 CV09DQ 137632591 IC50 = 594 nM T56556 CXA82V 137632731 IC50 = 1100 nM T56556 C29XTR 137633043 IC50 = 621 nM T56556 CF73VM 137634351 EC50 = 85 nM T56556 CKCE38 137634438 EC50 = 72 nM T56556 C39YOJ 137634518 IC50 = 4260 nM T56556 CS26GV 137634543 IC50 = 541 nM T56556 CI2K0G 137634736 IC50 = 454 nM T56556 CB0ZJ4 137635897 EC50 = 16 nM T56556 CS3RK1 137636023 IC50 = 628 nM T56556 C54LGH 137636095 EC50 = 16 nM T56556 CI1S9R 137636359 IC50 = 146 nM T56556 C51AGO 137636525 EC50 = 8 nM T56556 CEUR16 137637400 IC50 = 605 nM T56556 CUWZ73 137637797 IC50 = 206 nM T56556 C15FLS 137638403 EC50 = 676 nM T56556 CJ57LP 137638487 EC50 = 141 nM T56556 CFL5V7 137638559 IC50 = 488 nM T56556 C1CAL5 137638992 IC50 = 882 nM T56556 CI3NO0 137639122 IC50 = 1070 nM T56556 CI5Z8K 137639498 EC50 = 47 nM T56556 CTNP09 137639885 EC50 = 4 nM T56556 C8DL5H 137639918 EC50 = 37.1 nM T56556 C5IP1S 137640378 EC50 = 210 nM T56556 C91SBQ 137640534 EC50 = 3 nM T56556 CV3QD9 137641058 EC50 = 13 nM T56556 CI0KU2 137643961 EC50 = 22 nM T56556 C36TRI 137644856 IC50 = 952 nM T56556 CS4Z5B 137644952 IC50 = 283 nM T56556 C9HCB1 137645106 EC50 = 11 nM T56556 CP42GX 137645755 IC50 = 1656 nM T56556 CN3Y8B 137646060 IC50 = 403 nM T56556 C5LFG0 137646752 EC50 = 7 nM T56556 CUP1D3 137646767 EC50 = 32 nM T56556 CTN5H3 137647282 IC50 = 2563 nM T56556 C1FM8R 137647675 EC50 = 4 nM T56556 CV2FL8 137647707 EC50 = 22 nM T56556 CVL5T7 137648146 EC50 = 79 nM T56556 CBL59T 137648334 EC50 = 8 nM T56556 CAU49L 137648335 EC50 = 4 nM T56556 C15MCA 137648533 IC50 = 838 nM T56556 CMR58G 137649090 IC50 = 164 nM T56556 C8UYC1 137649208 EC50 = 5 nM T56556 CX1NH9 137649265 EC50 = 14 nM T56556 CH07EY 137649297 IC50 = 355 nM T56556 C0W1LM 137649303 EC50 = 16 nM T56556 CYP3S6 137649349 IC50 = 325 nM T56556 CZF79C 137649780 IC50 = 1202 nM T56556 CLTE54 137650017 EC50 = 16 nM T56556 C03KMV 137650224 IC50 = 1515 nM T56556 CBAK32 137650656 IC50 = 1380 nM T56556 C5S9OL 137651096 IC50 = 512 nM T56556 C2ZVM8 137651212 IC50 = 1713 nM T56556 CC0H4S 137651220 EC50 = 82 nM T56556 C60QXZ 137651369 EC50 = 9 nM T56556 CM0SC5 137651605 EC50 = 140 nM T56556 C9PE5G 137652835 IC50 = 519 nM T56556 CDZ5I0 137652882 IC50 = 299 nM T56556 CS14NG 137652949 EC50 = 4 nM T56556 CXS2E7 137653095 EC50 = 4 nM T56556 C2B9JN 137653194 IC50 = 472 nM T56556 CN6QH5 137653329 EC50 = 85 nM T56556 C65IAD 137653455 IC50 = 985 nM T56556 C59ZRO 137653532 IC50 = 910 nM T56556 CB1Y8V 137655046 IC50 = 348 nM T56556 C6RP1Z 137655517 IC50 = 354 nM T56556 C89NMB 137655783 IC50 = 1530 nM T56556 C12YJV 137655818 IC50 = 5270 nM T56556 CTV4I1 137655973 IC50 = 122 nM T56556 C0N1TD 137656929 IC50 = 866 nM T56556 COY89M 137657641 EC50 = 145 nM T56556 C5C0KF 137658808 EC50 = 1540 nM T56556 CTO85K 137659047 IC50 = 6400 nM T56556 CB8CJ2 137659409 IC50 = 691 nM T56556 C9HU7R 137659989 IC50 = 325 nM T56556 C8MXN5 137661038 EC50 = 2 nM T56556 C31GEP 137661880 IC50 = 750 nM T56556 CPI3E4 137662036 IC50 = 1630 nM T56556 C7SH6Z 137662093 EC50 = 12 nM T56556 CP1M2F 137662213 IC50 = 2121 nM T56556 CC1QL5 139593871 IC50 = 2130 nM T56556 C5PKZ2 139593897 IC50 = 951 nM T56556 C9USZ1 145949183 EC50 = 4 nM T56556 C3H7QO 145949352 EC50 = 29 nM T56556 C43QGK 145949445 IC50 = 284 nM T56556 CFN6T2 145949660 EC50 = 11 nM T56556 C2X7WS 145950031 IC50 = 44.8 nM T56556 CHB1S3 145950435 IC50 = 57.7 nM T56556 CZRP27 145950520 IC50 = 51.5 nM T56556 CB7KD0 145950545 EC50 = 2 nM T56556 CUB64Y 145950625 EC50 = 690 nM T56556 CNG6V3 145950683 IC50 = 78.7 nM T56556 CK6YR0 145950764 EC50 = 19.5 nM T56556 C07XUY 145950844 IC50 = 61.4 nM T56556 C94HRD 145950874 EC50 = 577 nM T56556 CE4SY2 145950964 IC50 = 1150 nM T56556 CUY09I 145950988 IC50 = 127 nM T56556 CIZ82R 145951128 IC50 = 1040 nM T56556 CR31OX 145951139 IC50 = 336 nM T56556 C4TRJ3 145951213 IC50 = 799 nM T56556 C53MCJ 145951316 IC50 = 65.3 nM T56556 CSYV28 145951611 EC50 = 19 nM T56556 CUD94F 145952004 EC50 = 63 nM T56556 C8Y7ND 145952143 IC50 = 66.3 nM T56556 C5V1MZ 145952691 IC50 = 801 nM T56556 C9O3IC 145952963 IC50 = 1770 nM T56556 C1L4NV 145953000 EC50 = 0.6 nM T56556 CIF74V 145953301 IC50 = 726 nM T56556 C5Z0BT 145953360 IC50 = 33 nM T56556 COSR30 145953465 IC50 = 369 nM T56556 CW97IA 145953788 IC50 = 904 nM T56556 CC3GQ9 145954340 EC50 = 21.8 nM T56556 C21XAV 145954560 EC50 = 1230 nM T56556 C2KBR1 145954586 IC50 = 30.2 nM T56556 CQ7Y6U 145955013 EC50 = 48 nM T56556 C7LP2U 145955206 EC50 = 6 nM T56556 CJ3ET0 145955421 EC50 = 10 nM T56556 CBI96G 145955592 IC50 = 20 nM T56556 C06LAX 145955721 IC50 = 2120 nM T56556 C3CAG9 145955791 IC50 = 221 nM T56556 CM62WT 145956236 IC50 = 120 nM T56556 CHCB46 145956407 EC50 = 4 nM T56556 C6FS8J 145956778 IC50 = 119 nM T56556 CLD32M 145957548 IC50 = 48.2 nM T56556 C8ZAT2 145957575 IC50 = 44.8 nM T56556 CX32LO 145957840 IC50 = 106 nM T56556 C9F8TW 145957857 EC50 = 48.3 nM T56556 CXH7F4 145957934 IC50 = 820 nM T56556 CB5PZ6 145958054 EC50 = 71.2 nM T56556 CB9CF1 145958160 EC50 = 14 nM T56556 CL15OJ 145958265 EC50 = 10 nM T56556 C9QO8G 145958364 IC50 = 16200 nM T56556 CL76TP 145958566 IC50 = 1190 nM T56556 CDH0A1 145958606 IC50 = 642 nM T56556 CD46YZ 145958660 IC50 = 1640 nM T56556 C0T5ZE 145958944 IC50 = 1620 nM T56556 CBQ8K0 145959274 IC50 = 795 nM T56556 CPU4D2 145959408 IC50 = 33.1 nM T56556 C3ZLR8 145959442 IC50 = 84 nM T56556 C2XSC1 145959549 IC50 = 49.1 nM T56556 C4PQ5A 145959673 IC50 = 811 nM T56556 C3C6SA 145959746 EC50 = 34 nM T56556 CIA08G 145959888 IC50 = 101 nM T56556 CVX17O 145960171 EC50 = 5 nM T56556 CYL21E 145960198 IC50 = 570 nM T56556 C2T8PH 145960322 IC50 = 610 nM T56556 CR0J2I 145960997 IC50 = 57.2 nM T56556 CA7RL9 145962283 IC50 = 5310 nM T56556 CBU79J 145964049 IC50 = 501 nM T56556 C1A7DH 145964067 IC50 = 9930 nM T56556 C5YP9J 145964072 IC50 = 6910 nM T56556 C80ESB 145964513 IC50 = 1060 nM T56556 CM5W0B 145964551 IC50 = 733 nM T56556 CNM1G3 145964790 IC50 = 766 nM T56556 C2QI8W 145965708 IC50 = 90 nM T56556 CJRZ24 145966467 IC50 = 445 nM T56556 C4OZH5 145966511 IC50 = 880 nM T56556 CBL6O0 145966757 IC50 = 7670 nM T56556 C4ZA8I 145966835 IC50 = 1550 nM T56556 CVB80Y 145966874 IC50 = 14390 nM T56556 C58UJF 145968465 IC50 = 15800 nM T56556 CTP6I7 145971735 IC50 = 646 nM T56556 CYU1W6 145971955 EC50 = 11 nM T56556 CZ3N8M 145972213 IC50 = 210 nM T56556 CIT6S0 145972309 IC50 = 18500 nM T56556 C6DKL1 145972800 IC50 = 438 nM T56556 C9QW5V 145973127 IC50 = 59 nM T56556 C96ARL 145973335 IC50 = 3230 nM T56556 C65PUC 145973732 IC50 = 6730 nM T56556 CM1UP7 145973867 IC50 = 430 nM T56556 C14UYO 145974134 IC50 = 287 nM T56556 C8K3YC 145974263 IC50 = 130 nM T56556 C1CKI3 145974543 IC50 = 297 nM T56556 CH30BM 145974617 IC50 = 270 nM T56556 CGWT84 145974788 EC50 = 4 nM T56556 C2O0FG 145974893 IC50 = 351 nM T56556 CLZ4D7 145974899 IC50 = 8760 nM T56556 CQ53WA 145974921 IC50 = 1400 nM T56556 CZ4I8A 145975509 IC50 = 61.6 nM T56556 CAF5H4 145975609 IC50 = 9000 nM T56556 CRO97S 145975756 IC50 = 2830 nM T56556 CM05IS 145975969 IC50 = 176 nM T56556 CA3V5K 145976004 IC50 = 15300 nM T56556 CT4C0Y 145976071 IC50 = 23240 nM T56556 C3PU1W 145976134 IC50 = 77.4 nM T56556 CM0DC2 145976272 IC50 = 2720 nM T56556 CZ9EA3 145976337 IC50 = 4080 nM T56556 C7EP8H 145976472 IC50 = 6650 nM T56556 CV9W1U 145976531 IC50 = 39800 nM T56556 COA43R 145976548 IC50 = 190 nM T56556 C6SV1M 145976742 IC50 = 11400 nM T56556 C6W1PJ 145977012 IC50 = 228 nM T56556 CZP74I 145977357 IC50 = 129 nM T56556 CQ6PN4 145977383 IC50 = 8340 nM T56556 CB7WX4 145977891 IC50 = 102 nM T56556 CK89HF 145978336 IC50 = 2130 nM T56556 C3Q8JT 145978355 IC50 = 1130 nM T56556 C53TFX 145978471 IC50 = 259 nM T56556 C4S5RJ 145978614 IC50 = 287 nM T56556 C3FSQ9 145978662 IC50 = 267 nM T56556 CGY0D8 145978682 IC50 = 2360 nM T56556 CL4WJ5 145978764 IC50 = 565 nM T56556 CF8L7A 145979103 EC50 = 22.3 nM T56556 CM6Z4G 145979318 EC50 = 989 nM T56556 CDYJ89 145979389 IC50 = 5400 nM T56556 C3EX7W 145979504 EC50 = 51.7 nM T56556 C24OSG 145979776 IC50 = 8440 nM T56556 C4G7LT 145980033 EC50 = 38.3 nM T56556 CUSP05 145981621 IC50 = 10900 nM T56556 C26OWY 145981942 EC50 = 19.9 nM T56556 C10YDI 145982128 EC50 = 1170 nM T56556 CZ9N5Q 145982445 IC50 = 6950 nM T56556 C3ZG6V 145982714 IC50 = 6630 nM T56556 C13VFZ 145985646 EC50 = 6.4 nM T56556 CU1Z8M 145986566 EC50 = 1390 nM T56556 C37ULP 145986567 IC50 = 10000 nM T56556 C3KFN7 145987093 EC50 = 448 nM T56556 CFU24J 145987833 EC50 = 3.1 nM T56556 CGL02K 145988126 EC50 = 57 nM T56556 C4F5OW 145988257 IC50 = 20100 nM T56556 CCIF35 145989307 IC50 = 12000 nM T56556 CX3YR7 145990226 EC50 = 34.7 nM T56556 CN1V8K 145992500 EC50 = 7.4 nM T56556 CT02XU 145992768 EC50 = 14 nM T56556 CKZA78 145992770 EC50 = 107 nM T56556 C07OTB 145993028 EC50 = 25.2 nM T56556 C65JUT 145993130 EC50 = 10.9 nM T56556 C8WF7P 145993760 IC50 = 6330 nM T56556 C3UC5J 145994097 EC50 = 59.7 nM T56556 CKM79V 145994277 EC50 = 27.1 nM T56556 CF92IR 155510784 EC50 > 100000 nM T56556 C3MZ1E 155511724 EC50 = 2300 nM T56556 CE4C1X 155512695 IC50 = 1630 nM T56556 CC9X1U 155514114 IC50 = 13100 nM T56556 CVZ7D2 155514151 EC50 = 4600 nM T56556 C0AFT8 155514623 EC50 = 2.4 nM T56556 C17AZU 155515244 EC50 = 5100 nM T56556 CUHI07 155515592 IC50 = 994 nM T56556 CH6O3X 155515825 EC50 = 16000 nM T56556 CV9TF6 155516191 EC50 = 2.2 nM T56556 C75VID 155517095 EC50 = 46 nM T56556 C4IS7E 155518051 EC50 = 4500 nM T56556 CLQO05 155518383 IC50 = 202 nM T56556 CCL04Y 155518581 IC50 = 7400 nM T56556 CCK94U 155519382 IC50 = 2570 nM T56556 CA1BD2 155520579 EC50 = 3700 nM T56556 CE50TP 155521906 IC50 = 7270 nM T56556 C97CDW 155522930 IC50 = 20000 nM T56556 CS18PU 155523410 EC50 = 33500 nM T56556 CN6ST7 155523417 EC50 = 1.1 nM T56556 C1V9YM 155523822 EC50 = 3000 nM T56556 CBZ8K4 155524289 IC50 = 513 nM T56556 C4LK0P 155524329 IC50 = 47.3 nM T56556 C86ZPR 155525910 EC50 = 8100 nM T56556 C8C7VA 155525927 EC50 > 100000 nM T56556 C8TQ4G 155526547 EC50 = 13.5 nM T56556 C7WI3R 155526594 IC50 = 1070 nM T56556 CTW8I2 155526857 EC50 = 3800 nM T56556 C41JTR 155528166 EC50 = 5600 nM T56556 C9BGT5 155528240 EC50 = 55.4 nM T56556 C75OQS 155529248 IC50 = 1900 nM T56556 C56AHP 155530068 EC50 = 3.5 nM T56556 CE0F4W 155530435 IC50 = 3669 nM T56556 C2PW4J 155530538 IC50 = 2025 nM T56556 CQZD59 155530897 IC50 = 3948 nM T56556 C1HFX4 155531129 EC50 = 7200 nM T56556 CUL2G4 155531672 EC50 > 1000 nM T56556 C4IW9M 155533366 EC50 = 41000 nM T56556 C9QT4A 155533532 IC50 = 7.98 nM T56556 CRC20Y 155534149 EC50 = 6400 nM T56556 CP9C0M 155534240 EC50 = 1220 nM T56556 C52RYM 155534490 IC50 = 178 nM T56556 CHF7A6 155535686 EC50 = 84 nM T56556 COFC46 155536723 EC50 = 4700 nM T56556 CP3U4C 155536912 EC50 = 46000 nM T56556 CYG84N 155537154 EC50 = 9500 nM T56556 CB1FI9 155537197 EC50 = 793 nM T56556 C2J7TM 155537461 IC50 = 652 nM T56556 CGD47O 155537584 EC50 = 2.1 nM T56556 C8FX4B 155537647 IC50 = 5650 nM T56556 CVES34 155538494 EC50 = 2300 nM T56556 CS4WO9 155538718 IC50 = 10500 nM T56556 CFN41J 155538958 EC50 = 6200 nM T56556 C8WT1F 155539055 IC50 = 1460 nM T56556 CLU37N 155539307 EC50 = 8100 nM T56556 C9VW3C 155539729 IC50 = 31 nM T56556 C70PUH 155540561 IC50 = 335 nM T56556 CL9G5X 155541828 IC50 > 10000 nM T56556 CE0G9A 155542384 IC50 = 1100 nM T56556 C56DUX 155543049 IC50 > 10000 nM T56556 CP93FH 155543149 EC50 = 6800 nM T56556 CJ5Q2K 155543420 IC50 = 10080 nM T56556 C7JUC3 155543680 EC50 = 3800 nM T56556 CYE3M6 155544628 IC50 = 556 nM T56556 C0GVI7 155545772 EC50 = 1800 nM T56556 CQ3S7A 155545818 IC50 > 10000 nM T56556 CMIN20 155545978 IC50 = 846 nM T56556 CDO86V 155546844 IC50 = 1780 nM T56556 CEA2R7 155547184 IC50 = 2900 nM T56556 COM08I 155547388 IC50 = 1320 nM T56556 CDY82R 155549328 EC50 = 4600 nM T56556 C86HEA 155549333 IC50 = 811 nM T56556 C72IFK 155549366 IC50 = 10400 nM T56556 CDFC58 155549450 IC50 = 1230 nM T56556 C53PGC 155550195 EC50 = 446 nM T56556 CWK3L0 155550287 EC50 = 11000 nM T56556 CB8FC1 155550293 EC50 = 4300 nM T56556 C8F3HQ 155550402 IC50 = 2000 nM T56556 CGF1W0 155551433 IC50 = 1920 nM T56556 CP7A5R 155552128 EC50 = 3900 nM T56556 CIF4T8 155553306 EC50 = 2.8 nM T56556 CG9K4Y 155553476 EC50 > 100000 nM T56556 C5QE9O 155553583 IC50 = 1030 nM T56556 CEZ7B1 155554618 EC50 = 6.5 nM T56556 CX6CM0 155554919 EC50 = 64 nM T56556 C2Y9UG 155554959 EC50 = 2300 nM T56556 C7JI4C 155555932 EC50 = 60 nM T56556 C8M0BP 155556108 IC50 = 989 nM T56556 CDAP41 155557648 IC50 = 202 nM T56556 CG0H8N 155557744 EC50 = 3300 nM T56556 CM2J5L 155558116 EC50 = 6400 nM T56556 C27XQN 155558615 EC50 = 7.2 nM T56556 CUNV65 155558919 EC50 = 17.8 nM T56556 C21LPY 155559292 IC50 = 1260 nM T56556 CG6NC7 155560071 EC50 = 4200 nM T56556 C46KOL 155560381 IC50 = 698 nM T56556 CY6UB5 155561091 IC50 = 112 nM T56556 CS2B6P 155561257 EC50 = 97 nM T56556 C6VUX2 155561896 IC50 = 77.3 nM T56556 CX42YD 155562157 IC50 > 10000 nM T56556 CPOI59 155562875 IC50 = 883 nM T56556 CWM67C 155563340 EC50 = 2500 nM T56556 CS0NC2 155563858 IC50 = 805 nM T56556 CJ57SV 155563869 IC50 > 10000 nM T56556 CU1TG6 155564277 IC50 = 7820 nM T56556 CJ4GX0 155564603 IC50 = 1060 nM T56556 C7SMU4 155565022 IC50 = 1100 nM T56556 C6Z2XK 155566234 EC50 = 4700 nM T56556 CAN76P 155566986 EC50 > 100000 nM T56556 C8ZE6S 155567126 IC50 = 4490 nM T56556 CO1LU7 155567143 EC50 = 30.7 nM T56556 C9QA2H 155567258 IC50 = 4780 nM T56556 CHT79A 155568041 EC50 = 5900 nM T56556 CFCV37 155568122 IC50 = 14800 nM T56556 CTV5K3 155568177 EC50 = 24.5 nM T56556 C03SJY 155568508 EC50 = 2 nM T56556 CO08ZV 155568670 EC50 = 5400 nM T56556 CTXV81 155568869 EC50 = 2.4 nM T56556 COQJ76 155569267 IC50 = 1450 nM T56556 D00RIX 5280443 IC50 = 3100 nM T56556 D01UYI 5281607 IC50 = 1500 nM T56556 D02ZRO 735125 IC50 = 1080 nM T56556 D04GYT 15511439 IC50 = 3981.07 nM T56556 D07RSH 631105 IC50 = 5980 nM T56556 D09HIM 22004473 IC50 = 3890.45 nM T56556 D0A4TF 15511440 IC50 = 5011.87 nM T56556 D0E5IP 3795 EC50 = 189 nM T56556 D0G3TK 5280863 IC50 = 4700 nM T56556 D0I7GE 11790 IC50 = 1310 nM T56556 D0NJ4H 5281670 IC50 = 49000 nM T56556 D0S0RK 10680 IC50 = 17000 nM T56556 D0S8CE 15950351 IC50 = 676.08 nM T75907 C79IRE 71620755 IC50 = 360 nM T75907 C7PI9C 71620756 IC50 = 360 nM T75907 CGD70V 71620759 IC50 = 360 nM T75907 CX85HD 71621073 IC50 = 360 nM T75907 CZB46R 71621227 IC50 = 360 nM T75907 CNP1U5 86574151 IC50 = 360 nM T75907 C2LM9W 127026354 IC50 = 30 nM T75907 CRD02W 127026355 IC50 = 280 nM T75907 C6KE3B 127026667 IC50 = 80 nM T75907 CE2PX6 127026668 IC50 = 30 nM T75907 C7VP6A 127026669 IC50 = 10 nM T75907 C1IF8B 127028921 IC50 = 70 nM T75907 C5ZK6J 127029217 IC50 = 50 nM T75907 CZ3DS8 127029218 IC50 = 40 nM T75907 CMR68I 127029233 IC50 = 1 nM T75907 C7ZHE4 127029234 IC50 = 10 nM T75440 D01XOD 54897 Ki = 0.5 nM T75440 D04BNP 5391 IC50 = 62517269.28 nM T75440 D07JVL 3016 IC50 = 123594743.3 nM T75440 D09LDR 4616 IC50 = 55590425.73 nM T75440 D0CP4E 2802 IC50 = 555904257.3 nM T75440 D0E0OG 3958 IC50 = 285759054.3 nM T75440 D0T5WK 4506 IC50 = 100000000 nM T75440 D0W2NM 3380 IC50 = 263026799.2 nM T75440 D0Z5OV 17925 IC50 = 555904257.3 nM T75440 D0Z9VB 31640 IC50 = 10864256.24 nM T75440 D0G4YZ 11653141 Ki = 2.47 nM T75440 D0M2TS 71600087 IC50 = 800 nM T75440 D01LOJ 11595759 Ki = 6.68 nM T75440 D0FR9I 10430788 Ki = 0.188 nM T75440 D0ZK2Q 9841240 Ki = 2.5 nM T75440 D05UXF 6433109 Ki = 6.4 nM T75440 D08AWI 11430856 Ki > 2000 nM T75440 D0K5IQ 9844410 IC50 = 0.92 nM T75440 D0VN4K 1345 IC50 = 1.1 nM T75440 CCH08A 2997 IC50 = 106414301.8 nM T75440 C87SBM 4540 IC50 = 500034535 nM T75440 CWB1Y9 15024 IC50 = 285759054.3 nM T75440 C2B9SE 16795 IC50 = 76913044.03 nM T75440 CC9L3A 19011 IC50 = 2630267.99 nM T75440 CHL67Q 30401 IC50 = 40831938.63 nM T75440 C7H2PJ 65764 IC50 = 2328091.26 nM T75440 CSTD39 75849 IC50 = 25003453.62 nM T75440 CL25FN 76175 IC50 = 2857590.54 nM T75440 CV8O9T 78641 IC50 = 2588212.92 nM T75440 CB0PY6 92294 IC50 = 15381546.4 nM T75440 CJD8Z6 118749 IC50 = 345143739.3 nM T75440 CYOL58 128744 IC50 = 142889395.9 nM T75440 CH2JA9 148760 IC50 = 10423174.29 nM T75440 CIUV59 188298 IC50 = 13335214.32 nM T75440 C1RK6L 520217 IC50 = 666806769.2 nM T75440 CNA35U 528222 IC50 = 454988060.2 nM T75440 CQ8H2P 622885 IC50 = 1614358.56 nM T75440 C89UHQ 5458184 Ki = 0.242 nM T75440 C01SQJ 6603782 Ki = 0.41 nM T75440 CR5NV7 9975396 IC50 = 181970085.9 nM T75440 C48VJA 10264786 IC50 = 27797132.68 nM T75440 CM8L2J 10358803 IC50 = 277971326.8 nM T75440 C8MT4I 10453776 Ki = 3.9 nM T75440 C3QEM9 10469149 IC50 = 263026799.2 nM T75440 CYX7O2 10738832 Ki = 1.6 nM T75440 CR67IU 10833643 IC50 = 11.8 nM T75440 CFJG64 11059058 IC50 = 1040 nM T75440 CR97ZW 11488150 Ki = 2.68 nM T75440 CR6OL3 11780929 Ki = 30.1 nM T75440 CXLW54 11948707 Ki > 10000 nM T75440 CM1T4V 12790028 IC50 = 142889395.9 nM T75440 C50BWX 13292074 IC50 = 47643098.68 nM T75440 CLH94F 13485706 IC50 = 416869383.5 nM T75440 CKZI28 15294055 IC50 = 620 nM T75440 CZ2IS9 16660294 Ki > 10000 nM T75440 C3W8DT 16749353 IC50 > 5000 nM T75440 CCP1J0 20542073 IC50 = 33342641.28 nM T75440 CDJ23A 23275339 IC50 = 2172701.18 nM T75440 CSB68Q 23275675 IC50 = 195884467.4 nM T75440 CWYX46 23275762 IC50 = 35727283.82 nM T75440 C9S0VL 23275763 IC50 = 625172692.8 nM T75440 CHL6M4 23275854 IC50 = 55590425.73 nM T75440 CTG41H 24778289 IC50 > 2000 nM T75440 C54TYJ 24945827 Ki = 0.882 nM T75440 CL6RD3 25140330 Ki = 0.537 nM T75440 CV4ZB3 25140479 Ki = 0.15 nM T75440 CD5V1U 25140760 Ki = 0.86 nM T75440 CIKB38 25208880 Ki = 0.997 nM T75440 C0RWI9 44366034 IC50 = 23280912.58 nM T75440 CFG7O1 44366036 IC50 = 41686938.35 nM T75440 CF72JC 44366089 IC50 = 25003453.62 nM T75440 CG9YJ7 44366116 IC50 = 135207256.3 nM T75440 CQ19LG 44366138 IC50 = 71449632.61 nM T75440 C1X5TW 44366161 IC50 = 188799134.9 nM T75440 C4LPC1 44366162 IC50 = 20417379.45 nM T75440 C8LT0S 44366169 IC50 = 52601726.64 nM T75440 C24VAZ 44366175 IC50 = 3334264.13 nM T75440 C26GHA 44366179 IC50 = 58884365.54 nM T75440 CR2V5W 44366192 IC50 = 833681184.6 nM T75440 CNAU14 44366206 IC50 = 285759054.3 nM T75440 CL7MP2 44366219 IC50 = 333426412.8 nM T75440 C94OVZ 44366228 IC50 = 188799134.9 nM T75440 CSF51U 44366236 IC50 = 243781081.8 nM T75440 CIP40L 44366255 IC50 = 52601726.64 nM T75440 C5TOJ7 46853447 IC50 = 2000 nM T75440 C8ZCU1 50994211 Ki = 1.57 nM T75440 CMJ62D 53245590 Ki = 2540 nM T75440 C49IKC 56671767 Ki = 1.19 nM T75440 C9D8WH 68968012 IC50 = 1.6 nM T75440 C1U2OK 72793912 Ki = 8 nM T75440 C0ZT5N 90644973 Ki = 293 nM T75440 CWE5X6 90656115 IC50 = 350 nM T75440 CLM5N2 90656116 IC50 = 680 nM T75440 CEAH51 118731302 Ki = 0.87 nM T75440 C5X8MN 122186880 Ki = 2897 nM T75440 C7ODW3 122195524 Ki > 900 nM T75440 CEK04Y 122196423 Ki = 28.13 nM T75440 C7ZKE3 122196424 Ki = 224.46 nM T75440 CVLH25 122196425 Ki = 29.11 nM T75440 C2HUV5 122196426 Ki > 10000 nM T75440 C5L9BD 134143752 Ki = 2100 nM T75440 C71PIY 134144970 Ki = 2200 nM T75440 CGS61F 137553161 Ki = 2930 nM T75440 CD7X5J 145951649 Ki = 28.9 nM T75440 CI4F0U 145954243 Ki = 25.4 nM T75440 CUSI97 145954858 Ki = 54.3 nM T75440 CKA9Z4 145958209 Ki = 70 nM T75440 C9ZY4V 145960315 Ki = 31.5 nM T75440 CPN90L 145971987 Ki = 31.6 nM T75440 CCTO46 155512230 Ki > 10000 nM T75440 CV35ZN 155513505 Ki = 3980 nM T75440 CB65EC 155513663 Ki = 96.1 nM T75440 C23PQH 155514371 Ki = 243 nM T75440 CLD73A 155514689 Ki = 1531.3 nM T75440 CWH24L 155517967 Ki = 562.5 nM T75440 CB0JS3 155518392 Ki > 10000 nM T75440 CH4ZC6 155518977 Ki = 53 nM T75440 C8DNZ6 155519967 Ki = 4737.3 nM T75440 CKH8G2 155522433 Ki > 10000 nM T75440 C36DYH 155525138 IC50 = 2.13 nM T75440 CIW07A 155526405 Ki = 3.2 nM T75440 C2UL4X 155526804 Ki > 10000 nM T75440 C1O0IC 155527848 Ki > 10000 nM T75440 C78XNA 155528306 Ki = 385.3 nM T75440 C2XY8U 155531728 Ki = 184.2 nM T75440 CY0H3U 155533272 Ki = 2020 nM T75440 COT9U8 155535203 Ki = 2380 nM T75440 CTD7J5 155537862 Ki = 462.3 nM T75440 C4C9NY 155541492 Ki > 10000 nM T75440 C1LU5B 155541865 Ki = 200 nM T75440 CMT60C 155543832 Ki = 2890 nM T75440 CJS87Q 155545399 Ki = 3170 nM T75440 C1L0SN 155547768 Ki = 200.7 nM T75440 CJ61KL 155547788 Ki = 369 nM T75440 CRY61B 155548339 Ki = 1696 nM T75440 C6IL4E 155548476 Ki = 50 nM T75440 CGL97X 155555425 Ki > 10000 nM T75440 CDL16X 155555765 Ki = 693.8 nM T75440 CBS89O 155556618 Ki = 2020 nM T75440 CLQH75 155558424 Ki = 208.4 nM T75440 CIPF89 155559210 Ki = 214 nM T75440 CAQ4S5 155561301 Ki > 10000 nM T75440 CCOD50 155562467 Ki = 2220 nM T75440 COP4K5 155562523 Ki > 10000 nM T75440 CI12LD 155566336 Ki > 10000 nM T75440 CU9HA1 155566889 Ki > 10000 nM T75440 C13REG 44471685 Ki = 3166 nM T75440 C6VJE1 6603767 Ki = 4.5 nM T75440 C9TZG6 9842567 Ki = 1.4 nM T75440 D06DTT 193319 IC50 = 71449632.61 nM T75440 D0A0ED 132496 Ki = 3.25 nM T75440 D0FF6S 16038374 IC50 > 2000 nM T75440 D0O6JQ 24839733 Ki = 13.6 nM T94621 D03ZBT 11626560 IC50 > 10000 nM T94621 D01NEC 51042438 IC50 = 1 nM T94621 D01ZAQ 25227436 IC50 = 8 nM T94621 D02ZQS 16095342 IC50 = 1350 nM T94621 D09IYM 24905401 IC50 = 402 nM T94621 D0E3TC 44259 IC50 = 6.5 nM T94621 D0I4TH 24788740 IC50 = 18 nM T94621 D0MS3Z 16725726 Ki = 4 nM T94621 D0W3RW 24964624 IC50 = 12 nM T94621 D03BNU 59604787 IC50 > 10000 nM T94621 D0ZE5U 11161844 IC50 = 5 nM T94621 D0T3ME 156422 IC50 > 30000 nM T94621 COYW98 9222 IC50 > 100000 nM T94621 C3XD4Z 139106 IC50 = 135000 nM T94621 C5EH9L 139601 IC50 = 80000 nM T94621 CU73ST 599501 IC50 = 660000 nM T94621 CFC7G1 756695 IC50 = 41000 nM T94621 C1SVD2 2132479 IC50 = 1900 nM T94621 C9ZT2G 2753118 IC50 = 72000 nM T94621 CFY1D0 2974957 IC50 > 10000 nM T94621 CABJ52 3129049 IC50 = 59000 nM T94621 C98ITU 5327109 IC50 = 260 nM T94621 CWN6P7 5702541 IC50 = 590 nM T94621 CG17TN 6914611 IC50 = 6.8 nM T94621 C7E2QK 6914613 IC50 = 257 nM T94621 CIAL53 9819282 IC50 = 23000 nM T94621 CC7Y2O 9828163 IC50 = 220 nM T94621 C8QZD6 9829528 IC50 = 26 nM T94621 C16VXB 9863538 IC50 > 10000 nM T94621 CI0AW6 9871034 IC50 = 2057 nM T94621 C7H8EO 9871171 IC50 = 7356 nM T94621 C18HKQ 9885748 IC50 = 720 nM T94621 CUE4B5 9912061 IC50 > 50000 nM T94621 CU7FH2 9957031 IC50 > 50000 nM T94621 CJX43Z 10055074 IC50 = 359 nM T94621 CEV18B 10128689 IC50 > 50000 nM T94621 C7PK4U 10152003 IC50 = 15700 nM T94621 C4FUG5 10152760 IC50 = 4517 nM T94621 CMO32F 10152761 IC50 = 325 nM T94621 CMR17F 10174144 IC50 > 50000 nM T94621 CLP79V 10196532 IC50 = 388 nM T94621 CI8MW4 10216627 IC50 = 5 nM T94621 C0O8FI 10217663 IC50 = 1179 nM T94621 CY6MJ3 10218178 Ki = 325 nM T94621 CT97JL 10218280 IC50 = 577 nM T94621 C8V6RI 10240275 IC50 = 212 nM T94621 CD3W6Y 10289038 IC50 > 20000 nM T94621 C2LP9A 10289671 IC50 = 300 nM T94621 CT0M7Q 10311653 IC50 = 259 nM T94621 C4MOF8 10312133 IC50 = 144 nM T94621 CAK9U4 10415819 IC50 = 65 nM T94621 CNY45Z 11151075 IC50 = 10 nM T94621 CO48BE 11165629 IC50 = 14 nM T94621 CO2DA6 11165945 IC50 = 10 nM T94621 C53MZX 11168481 IC50 > 50000 nM T94621 C1GYU5 11175137 IC50 = 18000 nM T94621 C3IJ6D 11180030 IC50 > 50000 nM T94621 CPVK21 11180486 IC50 = 1228 nM T94621 CMA1U5 11196322 IC50 = 510 nM T94621 C7BN5E 11225451 IC50 > 50000 nM T94621 CC6V3Z 11225497 IC50 = 529 nM T94621 C1UZC6 11226082 IC50 = 37720 nM T94621 CKB72H 11237628 IC50 = 8141 nM T94621 CL0QN6 11246027 IC50 = 27 nM T94621 C2ON6C 11246455 IC50 = 118 nM T94621 CCF0G6 11249067 IC50 = 2062 nM T94621 C49NET 11256399 IC50 = 204 nM T94621 C3T6XF 11256709 IC50 = 8 nM T94621 C1TCF3 11260243 IC50 > 50000 nM T94621 COHW29 11272514 IC50 > 50000 nM T94621 C9FG0K 11293497 IC50 = 4 nM T94621 CBOP58 11293798 Ki = 1120 nM T94621 CHBC32 11296432 IC50 = 839 nM T94621 CO39LB 11312547 IC50 = 31000 nM T94621 C1KOA4 11325683 IC50 = 39 nM T94621 CPV82H 11341558 IC50 > 50000 nM T94621 C26BZX 11362471 Ki = 3970 nM T94621 C4G3RZ 11364261 IC50 > 50000 nM T94621 COF6V0 11370369 IC50 = 9 nM T94621 C5EP3S 11373564 IC50 = 11 nM T94621 C1LT9H 11374804 IC50 > 50000 nM T94621 CD2P0L 11383042 IC50 = 5 nM T94621 CWXB93 11397177 Ki > 10000 nM T94621 CPFW90 11399527 IC50 = 556 nM T94621 CRC7H2 11407608 IC50 = 29 nM T94621 C6KQ2U 11409661 IC50 > 50000 nM T94621 C4L5TF 11409804 IC50 = 7356 nM T94621 C4OT0X 11417334 IC50 = 10 nM T94621 CCP18F 11430140 IC50 = 6 nM T94621 C1FC5U 11431759 IC50 > 50000 nM T94621 CW53GT 11440050 IC50 = 57 nM T94621 C5H7KT 11453730 IC50 = 3 nM T94621 CI9L2T 11454186 IC50 > 50000 nM T94621 CQS3U5 11454871 IC50 > 50000 nM T94621 CE72WO 11489421 IC50 = 15390 nM T94621 C7XM4C 11504922 IC50 = 59 nM T94621 CPN02A 11513279 IC50 = 27 nM T94621 C38OKZ 11513374 IC50 = 177 nM T94621 C85JUO 11514232 IC50 = 1600 nM T94621 CJ7XT8 11526364 IC50 = 1909 nM T94621 CTM2Q3 11526695 IC50 = 85 nM T94621 CEX8Y5 11527102 IC50 = 44 nM T94621 C5NPU9 11534762 IC50 = 5127 nM T94621 CCJ7Z1 11535873 IC50 = 830 nM T94621 CTG83F 11539329 Ki > 8400 nM T94621 CG84SZ 11540975 IC50 = 1572 nM T94621 CWCN15 11541348 IC50 = 44 nM T94621 CY0JX9 11541985 IC50 = 21 nM T94621 CSCJ29 11542208 IC50 = 229 nM T94621 C2O3DZ 11543058 IC50 = 880 nM T94621 CA8R0K 11547290 IC50 = 928 nM T94621 CX96EC 11549174 IC50 = 22 nM T94621 C3Z8PI 11549180 IC50 = 31 nM T94621 CJEB45 11549190 IC50 = 2106 nM T94621 CJF21M 11549537 IC50 = 297 nM T94621 CN25UD 11556452 IC50 = 99 nM T94621 CACS26 11561968 Ki > 10000 nM T94621 C3WVM7 11564772 IC50 = 180 nM T94621 C4LI8C 11564882 IC50 = 770 nM T94621 C9LDN1 11577612 IC50 = 107.2 nM T94621 CPJZ24 11584546 IC50 = 696 nM T94621 C0SCK2 11585287 IC50 = 8923 nM T94621 CAP6N0 11588244 IC50 = 8 nM T94621 CMIL86 11590363 Ki > 8400 nM T94621 C6C0VR 11592032 IC50 = 1131 nM T94621 C61KCW 11596252 IC50 = 680 nM T94621 CK61VI 11606572 IC50 = 3706 nM T94621 C20IRX 11606613 IC50 = 1304 nM T94621 C7PA8T 11607451 IC50 = 27 nM T94621 CNA3X5 11608401 IC50 = 6900 nM T94621 C3FQP1 11614515 IC50 = 4 nM T94621 CBEG76 11621110 IC50 = 635 nM T94621 C7P8CI 11622815 IC50 = 9500 nM T94621 CP2R3O 11636277 IC50 = 45 nM T94621 C4YWT2 11636404 IC50 = 6 nM T94621 C9T6SC 11640926 Ki > 8400 nM T94621 C2OC8S 11642946 IC50 = 43 nM T94621 CDY01B 11643074 IC50 = 252 nM T94621 C9RLC8 11643116 IC50 = 77 nM T94621 CP0I2U 11643417 IC50 = 25 nM T94621 CPA5Y7 11650332 IC50 = 184 nM T94621 COR9B8 11650399 IC50 = 16 nM T94621 CBW0A4 11660816 IC50 = 250 nM T94621 C87JQN 11663666 IC50 = 281 nM T94621 C7XEV0 11664023 IC50 = 94.4 nM T94621 CESQ80 11670972 IC50 = 239 nM T94621 C43LDG 11671553 IC50 = 73 nM T94621 CTI6U1 11671757 IC50 = 47 nM T94621 CX1GS0 11672017 IC50 = 16 nM T94621 CON70D 11672049 IC50 = 68 nM T94621 C0V7SU 11675388 IC50 = 2.2 nM T94621 CC5B1E 11681688 IC50 = 16 nM T94621 C0Q7ZW 11688053 IC50 = 400 nM T94621 CU0E8O 11690457 Ki > 10000 nM T94621 C81CLV 11693440 IC50 = 138 nM T94621 C95XBF 11695362 IC50 = 430 nM T94621 CPK2W8 11696113 IC50 = 5 nM T94621 C0NRG1 11703456 IC50 = 8 nM T94621 CB0AP2 11705863 Ki > 10000 nM T94621 CG3RQ4 11708454 IC50 = 290 nM T94621 C3B2HN 11708521 IC50 = 3200 nM T94621 CCK3Q5 11712132 IC50 = 1242 nM T94621 CY8U0T 11713130 IC50 = 90 nM T94621 CM49IK 11715597 IC50 = 920 nM T94621 C0TN5D 11738219 IC50 = 200 nM T94621 CJKC74 11750389 IC50 = 17 nM T94621 C9A6KM 11857236 Ki = 2 nM T94621 CA9ST2 11959186 IC50 = 63 nM T94621 CC7M0D 11959190 IC50 = 50 nM T94621 C39VTW 11959283 IC50 = 63 nM T94621 CQ8U1P 11959284 IC50 = 16 nM T94621 C36HDX 11959286 IC50 = 40 nM T94621 CTE96C 11959310 IC50 = 25 nM T94621 CO0A4K 11959314 Ki = 5 nM T94621 C12CRJ 11959377 IC50 = 200 nM T94621 CUWL12 11959378 IC50 = 25 nM T94621 CVPT94 11959513 IC50 = 316 nM T94621 C5LZ9C 11959550 IC50 = 200 nM T94621 C3UVQ2 11959600 IC50 = 79 nM T94621 C1WDQ0 11959682 IC50 = 20 nM T94621 CMW89V 11959683 IC50 = 20 nM T94621 CA6K4Y 11959684 IC50 = 20 nM T94621 C7RNV1 15602982 IC50 = 280 nM T94621 C3P1ED 15602983 IC50 = 34000 nM T94621 C7N6CQ 15604547 IC50 = 21 nM T94621 CSA02I 15979148 IC50 = 14.6 nM T94621 CBE54Y 15979149 IC50 = 6.7 nM T94621 C9YE7I 15979150 IC50 = 2.8 nM T94621 C92FEN 15979151 IC50 = 10.4 nM T94621 C9QO8U 15979276 IC50 = 10 nM T94621 CFPW41 16007116 Ki > 8400 nM T94621 CZK8V6 16043304 IC50 = 23 nM T94621 C9TU1O 16046126 IC50 > 1000 nM T94621 CKV4G1 16079040 IC50 = 20 nM T94621 CBM80K 16091080 IC50 = 47.7 nM T94621 C7Z4LV 16095343 IC50 = 1950 nM T94621 CHR8G4 16122633 IC50 = 20 nM T94621 C51PSY 16122634 IC50 = 5200 nM T94621 C2RNZ0 16657945 IC50 = 9 nM T94621 C94ONJ 16658020 IC50 = 12000 nM T94621 CSR4V7 16658021 IC50 = 3000 nM T94621 C0O6SY 17751068 IC50 = 8.5 nM T94621 CSK49V 17751069 IC50 = 7 nM T94621 C9C5TV 17751819 IC50 = 6 nM T94621 CWK2H5 21103101 IC50 = 274 nM T94621 CA46OM 21103107 IC50 > 50000 nM T94621 CJXU82 21103111 IC50 = 1877 nM T94621 CF9YE6 21103119 IC50 = 332 nM T94621 C5AR9M 21103197 IC50 = 281 nM T94621 CN1O7X 23647016 IC50 > 50000 nM T94621 CJ3EO0 23647017 IC50 = 1755 nM T94621 CH14KD 23647018 IC50 = 45270 nM T94621 CQ5Z0J 23647019 IC50 = 5407 nM T94621 CT7XW8 23647020 IC50 > 50000 nM T94621 C2JTA3 23647573 IC50 = 5 nM T94621 C83PYS 23647592 IC50 = 9 nM T94621 CI90XG 23647594 IC50 = 21 nM T94621 CWE47K 23647595 IC50 = 45 nM T94621 CICB91 23647596 IC50 = 4 nM T94621 C7W0PE 23647597 IC50 = 4 nM T94621 CTI1F7 23647598 IC50 = 6 nM T94621 CSOG98 23647599 IC50 = 19 nM T94621 CJAI42 23647600 IC50 = 51 nM T94621 CUX75S 23647601 IC50 = 37 nM T94621 CUX5O6 23647602 IC50 = 5 nM T94621 CA4LE6 23647603 IC50 = 8 nM T94621 CGS7Q3 23647604 IC50 = 3 nM T94621 CH89JW 23647605 IC50 = 5 nM T94621 CLDV63 23647606 IC50 = 5 nM T94621 C2BHO1 23658108 IC50 = 25 nM T94621 CL8M1D 23658126 IC50 = 5 nM T94621 CC97WO 23658173 IC50 = 70 nM T94621 CSJ34W 24701731 IC50 = 270 nM T94621 C7YG1N 24759534 IC50 = 23000 nM T94621 C7R9TA 24762195 IC50 = 8 nM T94621 CQNP54 24764449 IC50 = 25000 nM T94621 CW3JR8 24783593 IC50 = 14 nM T94621 C05MQY 24783594 IC50 = 35 nM T94621 C93TIM 24786152 IC50 = 12 nM T94621 CSY9Z6 24788164 IC50 = 11 nM T94621 CFR62V 24788432 IC50 = 12 nM T94621 C2JNI3 24788623 IC50 = 17 nM T94621 CMR7F1 24788739 IC50 = 15 nM T94621 CY1ZS7 24803305 Ki = 3 nM T94621 C2ANO6 24804134 Ki = 8 nM T94621 CSH8A5 24804780 Ki = 6 nM T94621 CUTH13 24805273 IC50 = 125 nM T94621 C0AO5R 24828715 IC50 = 110000 nM T94621 C1H2AM 24828716 IC50 = 246 nM T94621 CU9E4W 24828717 IC50 = 12 nM T94621 C5U2ZM 24828854 IC50 = 3 nM T94621 CQ4G2E 24828855 IC50 = 7 nM T94621 C57SYK 24829098 IC50 = 25 nM T94621 C3YLM1 24829099 IC50 = 71 nM T94621 CM5AX9 24829102 IC50 = 25 nM T94621 CY97JK 24829220 IC50 = 7 nM T94621 CT7QD8 24829222 IC50 = 25 nM T94621 C5WS6R 24894100 IC50 = 48 nM T94621 CV5IE4 24963049 Ki = 1 nM T94621 C9YN2Q 24967131 IC50 > 10000 nM T94621 CLJ2N0 24971386 IC50 = 1299 nM T94621 CC7B8W 24971387 IC50 = 1709 nM T94621 CCWV70 24971388 IC50 = 1381 nM T94621 CSE34D 24971389 IC50 = 1160 nM T94621 C5NFP2 24971390 IC50 = 1514 nM T94621 C0B9HE 24971391 IC50 = 17470 nM T94621 CX1U6V 24971392 IC50 = 1792 nM T94621 C3JT8Q 24971393 IC50 = 494 nM T94621 C0PFZ7 24992842 IC50 = 35 nM T94621 CC61ER 24993160 IC50 = 46 nM T94621 CT81XK 24993161 IC50 = 44 nM T94621 CZK9Q1 24993162 IC50 = 5.5 nM T94621 CK0NZ8 24993163 IC50 = 27 nM T94621 CQ9BF6 24993164 IC50 = 15 nM T94621 C71EOU 24993165 IC50 = 90 nM T94621 C1Y3TF 24993166 IC50 = 20 nM T94621 CA9F3Y 25023714 IC50 = 1000 nM T94621 C8Z4PI 25023715 IC50 = 3980 nM T94621 CV96QX 25023716 IC50 = 2340 nM T94621 C5INV4 25023717 IC50 = 2510 nM T94621 CPOH02 25023718 IC50 = 10000 nM T94621 C6F7RD 25023719 IC50 = 2570 nM T94621 C1JEU6 25023729 IC50 = 9 nM T94621 C14NAT 25023731 IC50 = 20 nM T94621 C81XKW 25023732 IC50 = 4 nM T94621 CFH80B 25023733 IC50 = 13 nM T94621 CR8JP7 25023735 IC50 = 13 nM T94621 C4W7LY 25023736 IC50 = 6 nM T94621 CA6QU5 25023737 IC50 = 5 nM T94621 COV3Q4 25061501 IC50 = 9 nM T94621 C8NR9H 25170562 IC50 = 6 nM T94621 CS9LC3 25170563 IC50 = 22 nM T94621 CN8YZ4 25170991 IC50 = 29 nM T94621 CHN5O0 25190977 IC50 = 19 nM T94621 COWB90 25221040 IC50 = 130 nM T94621 CC25TV 25222706 IC50 = 13 nM T94621 C1IG7E 25243798 IC50 > 10000 nM T94621 CH65JV 25243799 IC50 > 10000 nM T94621 CBQO98 42602095 IC50 = 40 nM T94621 CJ61SE 42602096 IC50 = 23 nM T94621 CI42XG 42602097 IC50 = 30 nM T94621 CD2AH4 42602175 IC50 = 24 nM T94621 CSWA85 42602176 IC50 = 46 nM T94621 C1LUN4 42602178 IC50 = 14 nM T94621 C8O3EA 42602260 IC50 = 22 nM T94621 C93NKL 42602264 IC50 = 15 nM T94621 C59CDG 44389260 IC50 = 157 nM T94621 CEP4T0 44422924 IC50 = 10 nM T94621 C0PEK6 44426856 IC50 = 31 nM T94621 COP8A3 44449880 IC50 = 42 nM T94621 CMC82Z 44449900 IC50 = 1476 nM T94621 C3APO5 44449908 IC50 = 210 nM T94621 CA85HS 44449909 IC50 = 981 nM T94621 C4QJK8 44449942 IC50 = 1600 nM T94621 C0ICB5 44449973 IC50 = 280 nM T94621 CE15WY 44449975 IC50 = 900 nM T94621 CEWB75 44450002 IC50 = 260 nM T94621 CDEJ84 44450004 IC50 = 1075 nM T94621 C8OG1V 44517709 IC50 = 1500 nM T94621 C1EVH2 44560678 IC50 = 827 nM T94621 CI58CZ 44560679 IC50 = 224 nM T94621 CC4Z5M 44560681 IC50 = 165 nM T94621 CWOM65 44560715 IC50 = 40 nM T94621 C7YCO3 44560716 IC50 = 80 nM T94621 C5X7PO 44560717 IC50 = 130 nM T94621 COTH35 44560718 IC50 = 84 nM T94621 C6J0ZC 44560719 IC50 = 180 nM T94621 CL0A2D 44560720 IC50 = 140 nM T94621 CR8K0X 44560724 IC50 = 185 nM T94621 CE08JD 44560725 IC50 = 146 nM T94621 CSX84T 44560726 IC50 = 92 nM T94621 C1O0IG 44560727 IC50 = 43 nM T94621 CB7X4S 44560728 IC50 = 192 nM T94621 C94LIO 44560729 IC50 = 190 nM T94621 C3UQ8C 44560730 IC50 = 116 nM T94621 C8OD4F 44560731 IC50 = 225 nM T94621 CLB20U 44560732 IC50 = 230 nM T94621 CGY1X7 44561054 IC50 = 29 nM T94621 CZK43G 44561055 IC50 = 223 nM T94621 C4WLX8 44561056 IC50 = 421 nM T94621 CXC8I3 44561057 IC50 = 23 nM T94621 CS0QZ4 44561058 IC50 = 539 nM T94621 C1QG9P 44561059 IC50 = 3570 nM T94621 C9MTS4 44561060 IC50 = 59 nM T94621 CZ9L8F 44572052 IC50 = 24.1 nM T94621 CIV48S 44572053 IC50 = 483.3 nM T94621 CFVA91 44572054 IC50 = 55.1 nM T94621 CZE8M9 44572055 IC50 = 77.9 nM T94621 C0DJS1 44591843 Ki = 4 nM T94621 CX52YW 44591844 Ki = 4 nM T94621 C1LS6V 44591845 Ki = 16 nM T94621 CSZ5R9 44592438 IC50 = 500 nM T94621 C6X7FC 44592501 Ki = 40 nM T94621 CTS95L 44592502 Ki = 40 nM T94621 CSKZ16 44592503 IC50 = 8 nM T94621 COY57J 44592504 Ki = 0.63 nM T94621 C3CDV8 44592505 Ki = 2 nM T94621 CJK7L8 45141615 IC50 = 19 nM T94621 CUEX28 45141616 IC50 = 84 nM T94621 C7XZI3 45141617 IC50 > 1000 nM T94621 CZC94D 45141618 IC50 = 35 nM T94621 CY8DC7 45141619 IC50 = 16 nM T94621 C5N4FO 45141620 IC50 = 18 nM T94621 CSB9Q2 45141621 IC50 = 69 nM T94621 C9BXC0 45141812 IC50 = 7 nM T94621 CEU36T 45141813 IC50 = 36 nM T94621 CLED29 45141814 IC50 = 14 nM T94621 CC16ZH 45141815 IC50 = 11 nM T94621 CM57PW 45141816 IC50 = 29 nM T94621 CC3R8E 45141817 IC50 = 210 nM T94621 CQ7OZ9 45142021 IC50 = 4.9 nM T94621 C01CFQ 45142022 IC50 = 5.7 nM T94621 C7FS2V 45142023 IC50 = 11 nM T94621 CYBD69 45142024 IC50 = 8 nM T94621 CR37UP 45142025 IC50 = 4 nM T94621 CU2K8B 45142026 IC50 = 25 nM T94621 CE4D3F 45142255 IC50 = 31 nM T94621 CLCU70 45142256 IC50 = 12 nM T94621 CJQ28R 45142257 IC50 = 52 nM T94621 CJIA74 45142258 IC50 = 12 nM T94621 C1V2YL 45142259 IC50 = 58 nM T94621 CQ5SD4 46190876 IC50 = 39 nM T94621 CY3HW5 46224684 IC50 = 4200 nM T94621 CB5H9C 46225574 IC50 = 31 nM T94621 C8M1DT 46225589 IC50 = 6 nM T94621 C60XUQ 46226079 IC50 = 15 nM T94621 C5PCH8 46226080 IC50 = 15 nM T94621 C6UD1Y 46226095 IC50 = 250 nM T94621 C7IF4T 46226096 IC50 = 63 nM T94621 CUDZ46 46226135 IC50 = 6300 nM T94621 C0P4CT 46226136 IC50 = 12 nM T94621 CPH49S 46226137 IC50 = 7 nM T94621 CM5X8B 46226156 IC50 = 15 nM T94621 C64TVL 46226417 IC50 = 25 nM T94621 CLS29B 46872626 IC50 > 10000 nM T94621 C2O8RZ 46886323 IC50 > 1000 nM T94621 CM8RX4 46886549 Ki = 17 nM T94621 C70BLN 46886550 IC50 = 50 nM T94621 CCV96R 46886665 Ki = 39 nM T94621 CJ2E9Q 46929857 IC50 > 25000 nM T94621 CC1Y0M 52941299 IC50 = 4951 nM T94621 CDT94U 52941495 IC50 = 1485 nM T94621 C9UF6K 52941555 IC50 = 433 nM T94621 CYM80Q 52942489 IC50 = 37826 nM T94621 CS09YT 52942516 IC50 = 5027 nM T94621 CQ08WT 52942668 IC50 = 1288 nM T94621 CHW04J 52943916 IC50 = 630 nM T94621 CY8BV4 52944892 IC50 = 707 nM T94621 CEM95A 52946401 IC50 = 5586 nM T94621 CKE3C7 52946402 IC50 = 1067 nM T94621 C3Q4CU 52947490 IC50 = 8362 nM T94621 CR9E1Z 52947590 IC50 = 26500 nM T94621 CE81HA 52950003 IC50 = 279 nM T94621 C3TU8R 52950063 IC50 = 872 nM T94621 C7MC5G 52950205 IC50 = 4371 nM T94621 C8NA4L 53384644 IC50 > 30000 nM T94621 CO6B0E 54583043 IC50 > 10000 nM T94621 C3PGE2 54585958 IC50 > 10000 nM T94621 CV7HJ8 54585959 IC50 > 10000 nM T94621 CPC5D2 56603995 IC50 = 8 nM T94621 CFP56A 56604013 IC50 = 8 nM T94621 CM8JX1 56604907 IC50 = 25000 nM T94621 CN9QD7 56643097 IC50 > 10000 nM T94621 CT4E8R 56832546 IC50 = 3300 nM T94621 CS7U9L 56965952 IC50 = 18 nM T94621 CQ57PE 57345536 IC50 = 3021 nM T94621 CQP7E0 57750290 IC50 = 31 nM T94621 CNBO65 57750312 IC50 = 36 nM T94621 C2F9DS 57750315 IC50 = 159 nM T94621 CZ08KN 57750321 IC50 = 96 nM T94621 CUY8T6 57750329 IC50 = 709 nM T94621 CK4W1L 57750342 IC50 = 30 nM T94621 CM5X9L 57750343 IC50 = 836 nM T94621 CBY5E4 57750369 IC50 = 42 nM T94621 CSI9Y4 57750382 IC50 = 210 nM T94621 C6GH7X 57750391 IC50 = 190 nM T94621 CL7CW0 57750402 IC50 = 130 nM T94621 CA4G5W 57750407 IC50 = 13 nM T94621 CM7XL6 57750408 IC50 = 20 nM T94621 CY4Z8R 57750418 IC50 = 344 nM T94621 C87LKR 58191080 IC50 = 4 nM T94621 CZPF92 58191081 IC50 = 6 nM T94621 CZA32V 58344912 IC50 = 700 nM T94621 CPVF85 58344916 IC50 = 660 nM T94621 CD3LX9 58344922 IC50 = 15 nM T94621 CS8ZY7 58344924 IC50 = 25 nM T94621 C89NVR 58344941 IC50 = 47 nM T94621 CYK74H 58344983 IC50 = 32 nM T94621 CRJ47B 58345005 IC50 = 16000 nM T94621 CIOV02 58345019 IC50 = 800 nM T94621 CY62SG 58345029 IC50 = 30 nM T94621 CM5HE1 58345070 IC50 = 130 nM T94621 CO18NP 58345151 IC50 = 35 nM T94621 CV61YJ 58345169 IC50 = 51000 nM T94621 CW6SC9 58345215 IC50 = 20000 nM T94621 CFLZ87 58345232 IC50 = 24 nM T94621 CYBT41 58345302 IC50 = 80 nM T94621 C4PE7X 58345314 IC50 = 27 nM T94621 C8X3WB 58458198 IC50 = 4177 nM T94621 C20XPF 58458267 IC50 > 2000 nM T94621 CP85TJ 58458278 IC50 = 6 nM T94621 CT79LH 58458379 IC50 = 356 nM T94621 CXJ63M 59603829 IC50 > 100000 nM T94621 CQEU96 59603842 IC50 = 430 nM T94621 CPVD45 59670809 IC50 = 33 nM T94621 C32WHR 59670989 IC50 = 24 nM T94621 CDWQ04 59671004 IC50 = 31 nM T94621 C43HZT 59671085 IC50 = 249 nM T94621 C0BRA5 59671144 IC50 = 66 nM T94621 CEYW16 59671148 IC50 = 10 nM T94621 C50NWX 59671151 IC50 = 3 nM T94621 CZH4W5 59671179 IC50 = 18 nM T94621 C8FY0G 59671180 IC50 = 17 nM T94621 COH62U 60097413 IC50 > 5000 nM T94621 C1MR8Q 60097495 IC50 > 10000 nM T94621 CC3MB4 60155179 IC50 = 9300 nM T94621 C9QB8G 60155270 IC50 = 1900 nM T94621 CM6NF2 60155627 IC50 = 3500 nM T94621 C62SQG 60155628 IC50 = 24 nM T94621 COS39T 60155629 IC50 = 33 nM T94621 CG6XQ3 67161715 IC50 = 477 nM T94621 CNXU89 67162253 IC50 = 311 nM T94621 CV63UL 67240318 IC50 > 10000 nM T94621 CP8OI2 67304551 IC50 = 5300 nM T94621 CY76UR 67305743 IC50 = 4.5 nM T94621 C3UKG8 67312397 IC50 = 3.2 nM T94621 CM6TZ3 67312506 IC50 = 2.5 nM T94621 C5DGR9 69036886 IC50 = 10000 nM T94621 CS8UF1 70675988 IC50 = 6 nM T94621 C2W5BX 70675991 IC50 = 2005 nM T94621 CUJA60 70676312 IC50 = 6 nM T94621 CRBW21 70676316 IC50 = 30 nM T94621 CGX49K 70676464 IC50 = 5 nM T94621 C1IEJ2 70789254 IC50 = 66000 nM T94621 C8T7ZP 70789255 IC50 = 9500 nM T94621 CKT60L 71455860 Ki > 8000 nM T94621 C9DIK2 71512060 IC50 > 10000 nM T94621 CQV96E 71583048 IC50 = 8111 nM T94621 CSPR52 71583049 IC50 = 16498 nM T94621 CNT5F3 71583050 IC50 = 805 nM T94621 CH7I0W 71583051 IC50 = 8578 nM T94621 CXSI14 71718330 IC50 > 100000 nM T94621 C1TM3P 71720141 IC50 > 100000 nM T94621 CJ2T9E 76332983 IC50 > 10000 nM T94621 C1HW4B 89735655 IC50 = 2500 nM T94621 CQCX41 118737057 IC50 > 10000 nM T94621 C9J4ES 135503073 IC50 = 8 nM T94621 CK94UW 136036657 IC50 = 83 nM T94621 CO16JK 136099766 IC50 = 188 nM T94621 C3ZS9L 136099767 IC50 = 284 nM T94621 CLB4O7 136099768 IC50 = 98 nM T94621 CC73PA 138911338 IC50 = 1.2 nM T94621 CSU93V 155077019 IC50 = 0.54 nM T94621 C2MD1Q 155513187 IC50 > 10000 nM T94621 C86HPW 155518524 IC50 = 21000 nM T94621 CL5DR0 155525783 IC50 < 0.64 nM T94621 CHS21A 155553831 IC50 = 14 nM T94621 CG95WV 155563831 IC50 = 2.8 nM T94621 CEIW13 155566807 IC50 = 79 nM T94621 D00ERW 44444843 Ki = 4800 nM T94621 D00HVA 11624601 Ki > 8400 nM T94621 D05APZ 135398501 IC50 = 210 nM T94621 D09FFE 449241 IC50 = 590 nM T94621 D0I1FJ 11393719 IC50 = 741 nM T94621 D0L2WP 46225540 IC50 = 12 nM T94621 D0OX1T 10172943 IC50 = 30 nM T94621 D0Q3NG 11715520 Ki > 8400 nM T94621 D0R2WK 16038120 Ki > 10000 nM T94621 D0S7IE 11658882 Ki > 8400 nM T94621 D0V6GX 11311693 IC50 = 20 nM T59720 C9G0HL 10533268 Ki = 35 nM T59720 C0QN5G 10606215 Ki = 35 nM T59720 C4IZ1Y 10820377 Ki = 35 nM T59720 CA50FN 56662663 Ki = 35 nM T59720 CH3SW7 56679684 Ki = 35 nM T43031 D0E3TC 44259 IC50 = 18.4 nM T43031 C1SVD2 2132479 IC50 = 3500 nM T43031 C18HKQ 9885748 IC50 = 77000 nM T43031 CACS26 11561968 Ki > 2000 nM T43031 CU0E8O 11690457 Ki > 2000 nM T43031 CKV4G1 16079040 IC50 = 500 nM T43031 CL81VC 21100709 IC50 = 11500 nM T43031 CZ3XP5 46926535 IC50 = 2600 nM T43031 C75GBE 49837568 IC50 = 22500 nM T43031 CEQN27 52936621 Ki > 1000 nM T43031 CT4E8R 56832546 IC50 = 14000 nM T43031 C1MR8Q 60097495 IC50 > 1000 nM T43031 CV63UL 67240318 IC50 = 630 nM T43031 CXSI14 71718330 IC50 = 83000 nM T43031 C1TM3P 71720141 IC50 = 83000 nM T43031 CJ2T9E 76332983 IC50 > 10000 nM T43031 C07EKN 138454794 IC50 > 10000 nM T43031 C0BU2E 145954767 IC50 > 10000 nM T43031 C2MD1Q 155513187 IC50 > 10000 nM T43031 D0K0UJ 49837564 IC50 = 170 nM T55922 D05FFR 5351154 Ki > 1000 nM T55922 CD0Y2A 118705586 Ki = 1070000 nM T55922 CD64YM 118725236 Ki = 1207000 nM T55922 C4ZJU9 239269 IC50 > 180000 nM T55922 CL14FJ 240808 IC50 > 180000 nM T55922 C9BOU0 240809 IC50 > 180000 nM T55922 CD3MU4 388060 IC50 > 180000 nM T55922 CG8Y0J 463012 IC50 > 180000 nM T55922 C1EPW6 476291 IC50 = 1500 nM T55922 CWN21X 608203 IC50 > 180000 nM T55922 CHU71V 2766291 IC50 > 180000 nM T55922 C3KV6A 11742879 Ki = 21200 nM T55922 C7HG1T 15218331 Ki = 20600 nM T55922 C1M3XT 19754189 IC50 > 180000 nM T55922 C05HNS 25181313 IC50 = 400 nM T55922 CQ39IJ 25183746 IC50 = 31000 nM T55922 CV90QL 25231313 IC50 = 3000 nM T55922 CTN16A 25231650 IC50 = 4000 nM T55922 C7NB0S 25231818 IC50 = 170 nM T55922 CIF3B2 25231819 IC50 = 440000 nM T55922 CH84SG 25231821 IC50 = 500000 nM T55922 CDS82O 25232183 IC50 = 49 nM T55922 CP1DT0 25233591 IC50 = 88000 nM T55922 C5BL4R 25233958 IC50 = 157000 nM T55922 C2EMK0 29066960 IC50 > 180000 nM T55922 CHB02E 44564175 IC50 = 7 nM T55922 C1L3WI 44564176 IC50 = 86 nM T55922 CE0JM4 44564196 IC50 = 11 nM T55922 CMWC14 44564197 IC50 = 5 nM T55922 CAID84 44564238 IC50 = 15 nM T55922 CFB5I1 44564239 IC50 = 18 nM T55922 CB7U4V 44564271 IC50 = 7000 nM T55922 CS43LM 44564338 IC50 = 70000 nM T55922 C57HRM 44564339 IC50 = 420000 nM T55922 C9Q3ZV 45097405 IC50 > 180000 nM T55922 C8UP6J 56919646 IC50 > 180000 nM T55922 CNI72Y 56919796 IC50 > 180000 nM T55922 C6A4KE 56919816 IC50 > 180000 nM T55922 C8I4ZA 56919856 IC50 > 180000 nM T55922 COU16Q 56920121 IC50 > 180000 nM T55922 CKLS86 56920454 IC50 > 180000 nM T55922 C8B4NQ 56920865 IC50 > 180000 nM T55922 C4T8JN 56921130 IC50 > 180000 nM T55922 C5CHU3 56921153 IC50 > 180000 nM T55922 CZHJ85 56921749 IC50 > 180000 nM T55922 C4U2XL 56921808 IC50 > 180000 nM T55922 COC17L 56922155 IC50 > 180000 nM T55922 C84CMO 56922551 IC50 > 180000 nM T55922 CUB52I 56923076 IC50 > 180000 nM T55922 CFG3V8 61710896 IC50 > 180000 nM T55922 C0Q8VJ 71460033 Ki = 3800 nM T55922 CA5VM1 80647643 IC50 > 180000 nM T55922 CHF61P 80761654 IC50 > 180000 nM T55922 C5JT8K 80768222 IC50 > 180000 nM T55922 C1B3TQ 80768523 IC50 > 63000 nM T55922 CFB2V6 80768610 IC50 > 180000 nM T55922 CGM4L1 100765007 IC50 > 180000 nM T55922 C8AF7O 104032679 IC50 > 180000 nM T55922 CV6FI3 107371081 IC50 > 180000 nM T55922 CW9RE8 113977178 IC50 > 160000 nM T55922 CIZ98T 114563625 IC50 > 180000 nM T55922 CP68ZQ 118725161 Ki = 21200 nM T55922 CUX9J4 118725180 Ki = 19600 nM T55922 CI9ZG7 118725204 Ki = 7200 nM T55922 CTB96Z 118725211 IC50 = 9000 nM T55922 CG8LY5 118725234 Ki = 18000 nM T55922 CI7C4Q 118725235 Ki = 669000 nM T55922 CZ4AP8 118725238 Ki = 478000 nM T55922 CQI0V5 118725241 Ki = 415000 nM T55922 CX13CP 118725243 Ki = 960000 nM T55922 CL3QZ8 118725244 IC50 = 178600 nM T55922 CAQH86 118725250 IC50 = 204800 nM T55922 CMS1X0 137632229 IC50 > 180000 nM T55922 CA6JL1 137632834 IC50 > 180000 nM T55922 CS1V5F 137632899 IC50 > 180000 nM T55922 CVC92M 137634051 IC50 > 180000 nM T55922 C82GYX 137634161 IC50 > 180000 nM T55922 CX84ME 137634646 IC50 > 180000 nM T55922 CT85ZK 137635286 IC50 > 180000 nM T55922 CGWV42 137635709 IC50 > 180000 nM T55922 C0D3HO 137635782 IC50 > 180000 nM T55922 C9ANK4 137635823 IC50 > 180000 nM T55922 CIKN81 137637985 IC50 > 63000 nM T55922 C8LO3S 137638905 IC50 > 180000 nM T55922 C7IWK8 137639930 IC50 > 180000 nM T55922 C6K3NC 137640514 IC50 > 180000 nM T55922 CD9HO6 137641254 IC50 > 21000 nM T55922 CK4NM7 137642459 IC50 > 180000 nM T55922 CT9Z2B 137642510 IC50 > 180000 nM T55922 CP05EG 137642600 IC50 > 63000 nM T55922 CPL3I7 137642845 IC50 = 44000 nM T55922 CF3W1S 137644197 IC50 > 63000 nM T55922 CO2ZG3 137645098 IC50 > 180000 nM T55922 CZ39RI 137645795 IC50 > 180000 nM T55922 CR2G4T 137646814 IC50 > 63000 nM T55922 C5D8MS 137647022 IC50 > 180000 nM T55922 CYA0M8 137648601 IC50 > 180000 nM T55922 C8J6EA 137648725 IC50 > 180000 nM T55922 C5HQ3N 137648979 IC50 > 21000 nM T55922 C4XUM8 137649315 IC50 > 21000 nM T55922 CNK2S4 137650167 IC50 > 180000 nM T55922 CE8ID4 137650445 IC50 > 180000 nM T55922 C9K4XH 137651053 IC50 > 21000 nM T55922 C75RCW 137651145 IC50 > 7000 nM T55922 C4C9DG 137651239 IC50 > 180000 nM T55922 CD23LP 137651376 IC50 > 63000 nM T55922 C03QHT 137651433 IC50 > 180000 nM T55922 C0TO6G 137651822 IC50 > 180000 nM T55922 CQE98H 137652324 IC50 > 180000 nM T55922 CHM69W 137652349 IC50 > 180000 nM T55922 CE57MT 137652443 IC50 > 180000 nM T55922 C46JEQ 137652753 IC50 > 180000 nM T55922 CFCI38 137652950 IC50 > 180000 nM T55922 C4GMS8 137653057 IC50 > 180000 nM T55922 CPZ58N 137653090 IC50 > 21000 nM T55922 CGK5Y1 137653360 IC50 > 180000 nM T55922 CSQF12 137653636 IC50 > 180000 nM T55922 CP8TJ0 137654766 IC50 > 21000 nM T55922 C75NWC 137655212 IC50 > 180000 nM T55922 CR6N5Y 137656925 IC50 > 21000 nM T55922 C9PJD2 137657088 IC50 > 180000 nM T55922 C5Q0YO 137657983 IC50 > 180000 nM T55922 CJ4M7L 137658244 IC50 > 180000 nM T55922 C3RO8E 137659106 IC50 > 180000 nM T55922 C6BN1M 137659420 IC50 > 63000 nM T55922 CBXA79 137659429 IC50 > 63000 nM T55922 CYD2N8 137659438 IC50 > 180000 nM T55922 C71FOJ 137660126 IC50 > 180000 nM T55922 C89UTS 137660314 IC50 > 63000 nM T55922 CPZ9E8 137660942 IC50 > 180000 nM T55922 CD1Y9L 137660985 IC50 > 180000 nM T55922 C4QM7T 137662328 IC50 > 180000 nM T55922 D03OLX 25231309 IC50 = 9000 nM T55922 D0I7IA 25231315 IC50 = 5000 nM T55922 D0P5YR 446204 IC50 = 55 nM T55922 D0YM6B 25231308 IC50 = 600 nM T58130 CN8XM2 5311263 EC50 = 8.1 nM T58130 CLS96Y 6419701 EC50 = 83.18 nM T58130 COZF72 10322404 EC50 = 2.692 nM T58130 C7QRT8 11648176 EC50 = 3.8 nM T58130 CV86RF 44368508 EC50 = 4.898 nM T58130 C85ANH 46213949 IC50 > 8000 nM T58130 CET63X 46223906 EC50 = 3.3 nM T58130 C57TYK 71569053 EC50 = 3.8 nM T58130 CSN3I7 71569056 EC50 = 2.4 nM T58130 CPT5S2 71718248 EC50 = 4.467 nM T58130 CKC4U7 71719457 EC50 = 4.898 nM T58130 C5P1CQ 71720690 EC50 = 3.467 nM T58130 CG65XZ 122191108 Ki = 170 nM T58130 CWQ8Y3 122191544 IC50 = 266 nM T58130 D05TVG 23682233 Ki = 170 nM T58130 D0X0UR 5497152 EC50 = 570 nM T17345 D01KKQ 135400182 IC50 = 21000 nM T17345 D0AO5H 5578 Ki = 0.006 nM T17345 D0C0SK 4993 Ki = 8 nM T17345 D0H0KB 5070 IC50 = 312000 nM T17345 D0M4VM 5320 IC50 = 18000 nM T17345 D0SV8E 126941 Ki = 0.00034 nM T17345 D0Y4GO 135410875 Ki = 7 nM T17345 D0Y7TS 5583 IC50 < 1 nM T17345 D04LBC 213043 IC50 = 8 nM T17345 D09AYQ 54369 Ki = 0.025 nM T17345 D05HCO 177894 Ki = 0.0003 nM T17345 D05AHQ 68916 Ki = 58.88 nM T17345 D06YIB 135436405 IC50 > 100000 nM T17345 D0D2RN 169371 Ki = 0.0018 nM T17345 D0FC5T 21453 IC50 = 530 nM T17345 D0N3XT 57030 IC50 = 1.8 nM T17345 CND0P2 1881 Ki = 4.5 nM T17345 C7OTP8 3439 IC50 = 220 nM T17345 CU2C4N 3534 IC50 = 70000 nM T17345 C8Y3OG 3537 IC50 = 2000 nM T17345 CEJF30 19931 Ki = 1659.59 nM T17345 C1F2TO 25889 Ki = 110 nM T17345 CY85FK 38778 Ki = 77.62 nM T17345 CRV0E5 72468 IC50 = 1000 nM T17345 CZ8JM5 72509 IC50 = 2.7 nM T17345 C87TYO 72934 IC50 = 15 nM T17345 C7SXL6 87152 IC50 = 1040000 nM T17345 CJ19OK 101067 Ki = 9.6 nM T17345 C8OGL7 102185 IC50 = 9400 nM T17345 C1Q8JR 121750 Ki = 7.7 nM T17345 C4HSB8 125843 IC50 = 1.35 nM T17345 CZA4M3 158351 IC50 = 220 nM T17345 CRQ24H 160203 Ki = 22.39 nM T17345 CZM82G 269322 IC50 = 3.9 nM T17345 C82AVZ 275733 IC50 = 3.8 nM T17345 C5JO7S 316019 IC50 = 3000 nM T17345 C3BRV9 317332 IC50 = 2700 nM T17345 CV20SE 324351 IC50 = 4.1 nM T17345 CPI45H 324352 IC50 = 8.6 nM T17345 CWV02U 324357 IC50 = 5.8 nM T17345 CY8C9L 329597 IC50 = 25000 nM T17345 C9GDJ6 353015 Ki = 0.00089 nM T17345 C3QH5B 354441 Ki = 218.78 nM T17345 CE7IH3 354768 IC50 = 19 nM T17345 CHA7L8 360682 Ki = 0.00035 nM T17345 CT64FM 375312 IC50 = 5.8 nM T17345 CC3ZE0 381233 IC50 = 11.6 nM T17345 C7VFS0 381234 IC50 = 11.4 nM T17345 C3F5KM 382165 IC50 = 8.7 nM T17345 CT51LK 393599 Ki = 0.0004 nM T17345 C8WO4J 403898 Ki = 42000 nM T17345 CTO2D8 404585 Ki = 100 nM T17345 C2IZ4Q 405137 Ki = 1800 nM T17345 C0MKV6 405140 Ki = 600 nM T17345 CDC2L4 406510 Ki = 4000 nM T17345 C25WDV 406511 Ki = 4000 nM T17345 C58ZQB 406512 Ki = 3000 nM T17345 CU4O0N 407233 Ki = 93.33 nM T17345 CD27CT 407235 Ki = 70 nM T17345 C5E7QX 429008 IC50 = 740 nM T17345 C6P2YK 444617 IC50 = 8500 nM T17345 CS9OU4 447021 IC50 = 26 nM T17345 CTXS72 447022 IC50 = 2900 nM T17345 C65ECP 448780 Ki = 5200 nM T17345 CT4N6R 456183 Ki = 6 nM T17345 CYC5M0 456204 IC50 = 4.7 nM T17345 CU1IP4 456205 IC50 < 100 nM T17345 C5VDE1 456216 IC50 = 3900 nM T17345 C1GU8M 456245 IC50 = 820 nM T17345 CD83KY 456272 IC50 = 440 nM T17345 CA6RC1 456306 IC50 = 2700 nM T17345 CQ61JH 456893 IC50 = 5 nM T17345 CEQ98S 456897 IC50 = 18200 nM T17345 CI10YF 457336 IC50 = 150 nM T17345 CHUR38 457342 IC50 = 5.5 nM T17345 CB2ZR6 457343 IC50 = 300 nM T17345 CBD80Z 457349 IC50 = 2300 nM T17345 CX4L1I 457350 IC50 = 1000 nM T17345 C7SZQ6 457353 IC50 = 142 nM T17345 C23EKX 457354 IC50 = 5.1 nM T17345 CBDY12 457370 IC50 = 2600 nM T17345 C81HJP 457371 IC50 = 31000 nM T17345 C53LNC 457372 IC50 = 750 nM T17345 CSWJ43 457373 IC50 = 730 nM T17345 CI17EV 457374 IC50 > 10000 nM T17345 C38SDU 457375 IC50 > 10000 nM T17345 CQY5L9 457376 IC50 > 10000 nM T17345 CMI8V4 457377 IC50 > 10000 nM T17345 CM5JA3 459880 IC50 = 370 nM T17345 CFQ2A9 459881 IC50 = 1000 nM T17345 CW1Q3Y 459887 IC50 = 710 nM T17345 C9YRU0 460024 IC50 = 57 nM T17345 CT9FW6 461920 Ki = 10.2 nM T17345 C03TKX 462111 IC50 = 17 nM T17345 CM4T5X 462117 IC50 = 10 nM T17345 C97EVZ 462118 IC50 = 28000 nM T17345 CHI3D7 462119 IC50 = 28000 nM T17345 C08HAR 462121 IC50 = 26000 nM T17345 C4SOE5 462122 IC50 = 27000 nM T17345 CUO54Z 462123 IC50 = 11 nM T17345 CS04OY 462124 IC50 = 25000 nM T17345 C7DI1F 462125 IC50 = 140 nM T17345 C8WYK9 462127 IC50 = 1400 nM T17345 C6NS9C 462129 IC50 = 50 nM T17345 C4AI1C 462134 IC50 = 3.6 nM T17345 C0EH1R 462466 Ki = 42.66 nM T17345 C8YC0H 462467 Ki = 134.9 nM T17345 CAHX06 462469 Ki = 302 nM T17345 CINY32 462582 IC50 = 2400 nM T17345 C8F9IM 462583 IC50 = 3900 nM T17345 C8QJT5 462584 IC50 = 550 nM T17345 CC65NE 462585 IC50 > 10000 nM T17345 CO46NQ 462587 IC50 = 4300 nM T17345 C62CHU 462589 IC50 = 2100 nM T17345 CTO26P 462590 IC50 = 3100 nM T17345 CQ4DV2 462591 IC50 = 2000 nM T17345 CJ4H0N 462592 IC50 = 2600 nM T17345 C0W2ZP 462593 IC50 = 24000 nM T17345 CBM4S2 462594 IC50 = 33000 nM T17345 C5Z4WX 462595 IC50 = 320 nM T17345 CO05RB 462596 IC50 = 180 nM T17345 C7XI6R 462597 IC50 = 3500 nM T17345 CV80TA 462598 IC50 = 4100 nM T17345 CS1AR6 462599 IC50 = 4400 nM T17345 C74WHR 462600 IC50 = 1300 nM T17345 C3HUT1 462601 IC50 = 400 nM T17345 CEW0T1 462602 IC50 = 270 nM T17345 C52FZM 462603 IC50 = 92 nM T17345 C8PC9F 462604 IC50 = 4300 nM T17345 C7ZJP3 462605 IC50 = 9100 nM T17345 CXW5K6 462606 IC50 = 820 nM T17345 C59MPI 462607 IC50 = 30 nM T17345 CK60HY 463731 IC50 = 990 nM T17345 CO3N7T 463890 IC50 = 12 nM T17345 CVK3W9 463891 IC50 = 7.1 nM T17345 CV4Q2D 463908 IC50 = 1200 nM T17345 C0XBM2 464022 IC50 = 590 nM T17345 C9PX5G 464023 IC50 = 500 nM T17345 C87RIT 464024 IC50 = 850 nM T17345 CMN7V4 464028 IC50 = 6100 nM T17345 CLC49E 464033 IC50 = 440 nM T17345 C6Z1YM 464034 IC50 = 420 nM T17345 C4H1FO 464035 IC50 = 36 nM T17345 CC80XF 464040 IC50 = 10 nM T17345 CRF85I 464992 IC50 = 27 nM T17345 CX8Y6N 464994 IC50 = 670 nM T17345 CCD18G 466230 IC50 = 6.7 nM T17345 CIR4Z5 466231 IC50 = 2500 nM T17345 CZI41B 467890 Ki = 87 nM T17345 CQB5F2 467891 Ki = 29 nM T17345 C0HG3Q 467892 Ki = 10 nM T17345 C7EJH4 467893 Ki < 2 nM T17345 CL91XC 467894 Ki = 10 nM T17345 CI8A9R 467895 Ki = 6.4 nM T17345 CT9M6G 467896 Ki < 2 nM T17345 C68DYK 467897 Ki = 24 nM T17345 CS8GB6 467898 Ki = 0.1 nM T17345 C3VY2Z 467899 Ki = 0.4 nM T17345 C4WIB5 467900 Ki = 0.1 nM T17345 CI81OG 467901 Ki = 0.2 nM T17345 CL8X1M 467902 Ki = 0.2 nM T17345 CSMT16 467903 Ki = 30 nM T17345 C45HLJ 467904 Ki = 0.4 nM T17345 CRUW28 467905 Ki = 0.1 nM T17345 CF1M8Q 468708 IC50 = 450 nM T17345 CSO8F0 468709 IC50 > 26000 nM T17345 CRP1D3 468710 IC50 > 25000 nM T17345 CQM7K4 468711 IC50 > 15000 nM T17345 CT6B0K 468712 IC50 > 15000 nM T17345 C92GMA 470175 IC50 = 6.1 nM T17345 CS6A3D 470176 IC50 = 2.8 nM T17345 C41BHZ 470177 IC50 = 5.2 nM T17345 C1BU8E 470179 IC50 = 6.7 nM T17345 CA3U5C 470200 IC50 = 3.7 nM T17345 C1Y2GQ 470201 IC50 = 5.9 nM T17345 C4D2QK 470202 IC50 = 6.1 nM T17345 C0V5MT 470264 IC50 = 120 nM T17345 CLY84S 470265 IC50 = 8 nM T17345 CMT51S 470266 IC50 = 44 nM T17345 C76HNV 470281 IC50 = 69 nM T17345 CQA07O 470284 IC50 = 250 nM T17345 CWV91M 470285 IC50 = 19 nM T17345 C25WGL 470286 IC50 = 4.6 nM T17345 CX5KM2 470287 IC50 = 3.2 nM T17345 CPC2W8 470288 IC50 = 4.1 nM T17345 CGI39U 470317 IC50 = 4 nM T17345 CI81MK 470318 IC50 = 850 nM T17345 C3O4TZ 470332 IC50 = 5300 nM T17345 CMJ5I4 470333 IC50 = 1900 nM T17345 CLM7A5 472826 IC50 = 3400 nM T17345 C0IJ7Q 472845 IC50 = 3.8 nM T17345 CM6FH7 472846 IC50 = 6.2 nM T17345 CQGS78 472847 IC50 = 2 nM T17345 C8NJU3 472848 IC50 = 68 nM T17345 CNBY98 472849 IC50 = 14 nM T17345 CIHZ91 472850 IC50 = 33 nM T17345 C9H4YB 472852 IC50 = 277 nM T17345 C7VGW9 472853 IC50 = 20 nM T17345 CVFX53 472910 Ki = 24.4 nM T17345 CERP02 474750 IC50 = 15 nM T17345 C0SG1N 476032 IC50 = 2459 nM T17345 C1Z6AQ 476042 IC50 = 1526 nM T17345 CY37PZ 476043 IC50 = 942 nM T17345 C74WGU 477890 IC50 = 7300 nM T17345 C3JY5Z 479281 IC50 = 700 nM T17345 CM2GT8 479412 IC50 = 76000 nM T17345 CF3C8Q 479413 IC50 = 13000 nM T17345 C41TQB 479416 IC50 = 530 nM T17345 C59FRQ 479418 IC50 = 160000 nM T17345 CF2JD3 479421 IC50 = 6200 nM T17345 CRB65P 481401 IC50 > 19000 nM T17345 COV85S 482165 IC50 = 1300 nM T17345 C9KOB8 485848 IC50 = 0.0021 nM T17345 C3JX2W 490573 IC50 = 5000 nM T17345 C25VUD 490663 Ki = 96.3 nM T17345 CI74ZT 490664 Ki = 4.3 nM T17345 CEW3B0 490665 Ki = 33 nM T17345 C89KLU 490666 Ki = 310 nM T17345 C7LX8H 490667 Ki = 250 nM T17345 CR1SM3 490668 Ki = 49 nM T17345 CLTA76 504022 IC50 = 5000 nM T17345 CN5CJ7 688803 IC50 = 50000 nM T17345 CQ5E7D 789778 Ki = 9.8 nM T17345 C9JQC0 2437106 IC50 = 500 nM T17345 C7RW2A 2731323 Ki = 130 nM T17345 C67UFD 2737412 IC50 = 580 nM T17345 C5F6EO 3010592 IC50 = 6.8 nM T17345 CG6F5S 3132813 Ki = 6.4 nM T17345 C2IFO1 3145500 IC50 = 1900 nM T17345 CFRL82 5183677 IC50 = 830 nM T17345 CHGZ97 5288461 IC50 = 800 nM T17345 CQ1ZH4 5742617 IC50 = 1216 nM T17345 CQ75AN 5742620 IC50 = 624 nM T17345 CT79NS 5742621 IC50 = 1410 nM T17345 CM59DP 5742624 IC50 = 970 nM T17345 C2N0IR 6477203 Ki = 1600 nM T17345 CYP69H 6482470 IC50 = 10000 nM T17345 CXI43R 9805576 IC50 = 1530 nM T17345 CYZ79K 9846618 IC50 = 8.8 nM T17345 CVWX01 9881905 Ki = 15000 nM T17345 CC36EP 9889551 IC50 = 10000 nM T17345 CP75AV 9898639 IC50 = 18000 nM T17345 C5VZN4 9911146 IC50 = 420 nM T17345 C3GI6F 9931657 Ki = 0.005 nM T17345 CL0P6O 9932276 IC50 = 1000 nM T17345 CIDQ05 9952879 Ki = 0.12 nM T17345 CBQK30 9973530 Ki = 4.2 nM T17345 CG9ZU8 9976735 IC50 > 26000 nM T17345 C2C7WX 9980556 Ki = 0.54 nM T17345 C3FR4N 10004772 IC50 = 125 nM T17345 C7RD2X 10007840 Ki = 0.183 nM T17345 C9A1VX 10019413 Ki = 24 nM T17345 CID95L 10030947 Ki = 0.000014 nM T17345 CN4V0B 10053803 Ki = 0.00041 nM T17345 C04LWZ 10060600 Ki = 1.6 nM T17345 CQI0P1 10060703 IC50 = 20 nM T17345 C37ZPO 10065177 Ki = 977.24 nM T17345 C5THD4 10070986 IC50 = 16 nM T17345 C70FRM 10072852 IC50 = 66 nM T17345 CQ8U6T 10090457 Ki > 5000 nM T17345 CSJY78 10246793 Ki = 36 nM T17345 C8ME5O 10260430 IC50 = 2.5 ug.mL-1 T17345 CGT0H9 10326322 Ki = 0.00011 nM T17345 CKFP04 10403719 Ki = 140 nM T17345 C7KXJ2 10404647 IC50 = 560 nM T17345 C9PRM3 10405166 IC50 = 2.8 nM T17345 CTX6H7 10433577 IC50 = 210 nM T17345 CZD4B0 10456691 IC50 = 21000 nM T17345 CB15AR 10457642 IC50 = 1.3 nM T17345 CHM3X4 10478775 Ki = 3400 nM T17345 CPO4W7 10518330 Ki = 9.8 nM T17345 C12BJE 10522269 Ki = 52 nM T17345 CZ8YM9 10544281 Ki = 75 nM T17345 CM95NE 10565157 Ki = 7.1 nM T17345 CLK5H2 10590469 IC50 = 3185 nM T17345 CG83DM 10608757 Ki = 750 nM T17345 C9WCK2 10634047 Ki = 8.6 nM T17345 CI5SU7 10658874 Ki = 10.5 nM T17345 CBXD51 10682649 Ki = 8.8 nM T17345 CXZL07 10709354 Ki = 13 nM T17345 C41ICW 10719122 IC50 = 3100 nM T17345 C0B7YU 10805231 Ki = 131 nM T17345 CHK35G 10807265 Ki = 19 nM T17345 CMF9L1 10826074 Ki = 3.6 nM T17345 C7XFJ5 10828475 Ki = 11 nM T17345 C3R0FI 10860015 IC50 = 10 nM T17345 C0S6TG 10883066 IC50 = 22000 nM T17345 CYWT73 10884015 IC50 = 100000 nM T17345 C9HR0M 10902858 IC50 = 32000 nM T17345 C8B0FL 10961831 IC50 = 5400 nM T17345 C4ZML2 10981577 IC50 = 85 nM T17345 C9D4VK 10991113 IC50 = 44 nM T17345 C9LPA1 10993870 IC50 = 920 nM T17345 CCQ4P6 11003295 IC50 = 2 nM T17345 C2P3AT 11047021 IC50 = 1300 nM T17345 CZ90JL 11058970 IC50 = 450 nM T17345 C4RBD9 11078421 IC50 = 21 nM T17345 CP5YV0 11099765 IC50 = 27000 nM T17345 CY1A7Q 11102571 IC50 = 7 nM T17345 C9ZWB1 11154001 IC50 > 10000 nM T17345 CO2DY5 11247965 Ki = 0.034 nM T17345 C8Q6ZT 11248313 Ki = 2.1 nM T17345 CIG85H 11282247 IC50 = 300 nM T17345 CI2TD8 11340329 IC50 > 10000 nM T17345 C85DMO 11349789 IC50 = 28000 nM T17345 C4EL7T 11430583 IC50 > 10000 nM T17345 CH8IF2 11442040 IC50 > 10000 nM T17345 C41XHB 11452801 IC50 > 10000 nM T17345 CJS58R 11455251 IC50 > 10000 nM T17345 C03JKV 11478803 Ki = 0.0001 nM T17345 C3ROC9 11538533 IC50 < 10 nM T17345 C6K9EH 11573029 IC50 = 630 nM T17345 C1XJI4 11645134 IC50 = 10700 nM T17345 C71ZQD 11645349 IC50 = 34 nM T17345 CYL01H 11651834 IC50 = 9400 nM T17345 CRUQ79 11673839 IC50 = 98000 nM T17345 C8AEX7 11687971 Ki = 500 nM T17345 C19BQV 11688044 IC50 = 8400 nM T17345 CQ4H5E 11744008 IC50 = 9000 nM T17345 CE7DH6 11783065 IC50 = 30000 nM T17345 CTB69W 11822511 IC50 = 47 nM T17345 CR9GN2 11826533 IC50 = 22000 nM T17345 CWP0B9 11846624 IC50 = 1830 nM T17345 CCUF60 11846625 IC50 = 2300 nM T17345 CW5VO2 12214236 Ki = 56000 nM T17345 CU1CF0 12242319 IC50 = 377000 nM T17345 CML17O 12242320 IC50 = 242000 nM T17345 CZO4H8 12242322 IC50 = 57000 nM T17345 C9AQ3V 12242324 IC50 = 740000 nM T17345 C13ZHJ 12517699 IC50 = 28000 nM T17345 CRSM76 12517700 IC50 = 7000 nM T17345 CSN4H6 12517701 IC50 = 8000 nM T17345 CMT96B 12517702 IC50 = 11000 nM T17345 C32RLQ 12517703 IC50 = 903000 nM T17345 C3G8JV 12517705 IC50 = 168000 nM T17345 CYPT41 12655201 IC50 = 370 nM T17345 CI0Y1T 12655204 IC50 = 58 nM T17345 CUXC87 12803287 IC50 = 340000 nM T17345 C98JXK 13112734 IC50 = 120 nM T17345 CX3Q6D 13112736 IC50 = 49 nM T17345 C8EIC5 13112740 IC50 = 29 nM T17345 C1INA2 13112752 IC50 = 310 nM T17345 C5X3WZ 13112757 IC50 = 44 nM T17345 C84HXC 13170795 IC50 = 14000 nM T17345 CU4O5B 13739857 IC50 = 61 nM T17345 CZLB08 13877973 IC50 = 230 nM T17345 CU8A4L 13877981 IC50 = 1110 nM T17345 CZV23T 13953684 IC50 = 67 nM T17345 CIW97R 13953685 IC50 = 93 nM T17345 CQFS01 13953687 IC50 = 110 nM T17345 C49DCF 13953688 IC50 = 170 nM T17345 C47HUP 13953689 IC50 = 20 nM T17345 C25SRU 13989362 IC50 = 5.3 nM T17345 CHI71Y 13989363 IC50 = 5.4 nM T17345 CRN23J 14083105 IC50 = 72 nM T17345 CS1G8K 14503206 IC50 = 40 nM T17345 CD84TM 14503207 IC50 = 70 nM T17345 CZET95 14560097 IC50 = 3 nM T17345 CAM5O1 14570150 Ki = 0.8 nM T17345 C8XLI9 14570153 IC50 = 66 nM T17345 CM49FY 14570156 IC50 = 110 nM T17345 C46HSO 14570159 IC50 = 14 nM T17345 CEL4B9 14570163 IC50 = 46 nM T17345 C6N4JB 14570319 IC50 = 300 nM T17345 C20TUW 14570320 IC50 = 630 nM T17345 CFQ37R 14570325 IC50 = 1800 nM T17345 CK5JI7 14570338 IC50 = 540 nM T17345 C3B7AQ 14570339 IC50 = 140 nM T17345 C9W4IP 14776576 IC50 = 6.4 nM T17345 C9V3SY 14776579 IC50 = 88 nM T17345 CX4U2T 14776583 IC50 = 57 nM T17345 CU1M4X 14776589 IC50 = 5.3 nM T17345 CWDB20 14776590 IC50 = 5.9 nM T17345 C9EW5Z 14776615 IC50 = 6000 nM T17345 CA4HC9 14776619 IC50 > 20000 nM T17345 CW5C6T 14801655 IC50 = 32 nM T17345 CBKR63 14801660 IC50 = 35 nM T17345 C68YXF 14801666 IC50 = 30 nM T17345 C4UVQ0 14840934 IC50 = 27000 nM T17345 CL5H0X 14840943 IC50 = 35 nM T17345 CORH59 14840958 IC50 = 50 nM T17345 C7VK0C 15021215 IC50 = 1.34 nM T17345 C4D8IR 15523786 Ki = 14.1 nM T17345 CW1QA4 15523787 Ki = 0.107 nM T17345 C6QM7Z 15616236 IC50 = 19000 nM T17345 C8W1DB 15616238 IC50 > 50000 nM T17345 CQ1TU0 16038397 Ki = 9.6 nM T17345 CWKX69 16086910 Ki = 110000 nM T17345 C6V7GN 16086911 Ki = 35000 nM T17345 C3X9DE 16086912 Ki = 3900 nM T17345 C9KZ4H 16086913 Ki = 33000 nM T17345 CTK25X 16086914 Ki = 69000 nM T17345 C7MA5T 16086915 Ki = 13000 nM T17345 CD59VR 16086916 Ki = 35000 nM T17345 C6UX1P 16086917 Ki = 109000 nM T17345 CRWB95 16086918 Ki = 13000 nM T17345 C0RE7Z 16086919 Ki = 12000 nM T17345 C1BYA7 16110323 IC50 = 1460 nM T17345 C4XBM2 16110326 IC50 = 1380 nM T17345 CB36UF 16110328 IC50 = 5710 nM T17345 CS9FR8 16110329 IC50 = 1160 nM T17345 C31SJW 16110337 IC50 = 400 nM T17345 CJ73WY 16110338 IC50 = 1460 nM T17345 C3LHA7 16110339 IC50 = 14300 nM T17345 C8OYD1 16110341 IC50 = 1220 nM T17345 C81MTW 16110344 IC50 = 1380 nM T17345 CZJM43 16732891 IC50 = 2900 nM T17345 CGM38B 16732892 IC50 = 6000 nM T17345 CMC21Z 16732893 IC50 = 5800 nM T17345 C9IG0J 16733029 IC50 = 2700 nM T17345 CHL6F9 16733030 IC50 > 31000 nM T17345 C8X9EC 16733031 IC50 > 31000 nM T17345 CW5SB7 16733033 IC50 > 28000 nM T17345 CM80YI 16733034 IC50 = 5800 nM T17345 CM1I4D 16733035 IC50 > 32000 nM T17345 CP8VS3 16733036 IC50 = 1400 nM T17345 C83VHB 16733162 IC50 = 1400 nM T17345 CED2R5 16733163 IC50 = 2900 nM T17345 CDA8P5 16733164 IC50 = 18000 nM T17345 CXA71B 16733165 IC50 = 32000 nM T17345 CC09RL 19089924 IC50 = 430 nM T17345 CK1P0V 21496446 IC50 = 140 nM T17345 C7B8CR 21705470 IC50 = 83300 nM T17345 C27WPQ 23161237 IC50 = 1100 nM T17345 CE2XM5 23629645 Ki = 800 nM T17345 CT2G9I 23647976 IC50 = 2100 nM T17345 CUSF67 23648073 Ki = 94000 nM T17345 CI2F9K 23648074 Ki = 28000 nM T17345 C4SXQ7 23648075 Ki = 15000 nM T17345 CDUX91 23648076 Ki = 9500 nM T17345 CE4G3V 23729147 IC50 > 125000 nM T17345 C7TLP1 24202945 Ki = 2000 nM T17345 C4S9RX 24202946 Ki = 8000 nM T17345 C6H1RM 24202947 Ki = 8000 nM T17345 C7AXQ6 24203165 Ki = 6000 nM T17345 CUC7I6 24203167 Ki = 4000 nM T17345 CG7RU5 24203941 Ki = 3000 nM T17345 C9BO1H 24203942 Ki = 5000 nM T17345 COCG69 24203943 Ki = 3000 nM T17345 C6S0FC 24204135 Ki = 5000 nM T17345 C2M1JB 24204136 Ki = 11000 nM T17345 C5S8PW 24204221 Ki = 4000 nM T17345 C63PUM 24204222 Ki = 3000 nM T17345 C89JMH 24204223 Ki = 5000 nM T17345 CN13ZR 24204418 Ki = 5000 nM T17345 C1IN2K 24204433 Ki = 3000 nM T17345 C6Y0ZX 24204434 Ki = 7000 nM T17345 CP73JD 24204806 Ki = 5000 nM T17345 C6M5YP 24204807 Ki = 8000 nM T17345 CA3BT0 24204808 Ki = 4000 nM T17345 CEK8R6 24777136 IC50 = 39 nM T17345 C6O5CL 24778299 IC50 = 25 nM T17345 CL7KN4 24950538 IC50 = 2600 nM T17345 C2C4FZ 24950539 IC50 = 3000 nM T17345 C9LY5G 24950540 IC50 = 33000 nM T17345 CPEF92 24950541 IC50 > 30000 nM T17345 CD8QM2 24950542 IC50 = 28000 nM T17345 CX5Q0K 24950543 IC50 > 26000 nM T17345 CH9A4V 24950693 IC50 > 29000 nM T17345 CG6A8V 24950694 IC50 > 15000 nM T17345 C6F2CR 24950695 IC50 > 26000 nM T17345 CX1AR8 24950696 IC50 > 30000 nM T17345 C1PHA0 24950697 IC50 = 16000 nM T17345 CG2B8O 24950698 IC50 = 30000 nM T17345 CX97IY 24950699 IC50 > 28000 nM T17345 C32OJF 24950851 IC50 = 27000 nM T17345 CCY8U4 24950852 IC50 > 29000 nM T17345 C17DAP 24950853 IC50 > 29000 nM T17345 CPDN34 24950854 IC50 > 27000 nM T17345 C2BXV5 25002412 IC50 > 125000 nM T17345 CQ3AV2 25002763 IC50 > 125000 nM T17345 CNBS61 25007427 IC50 = 55200 nM T17345 C1ER2L 25007788 IC50 > 125000 nM T17345 CIB13V 25058133 IC50 = 1280 nM T17345 CZ9L1Y 25093361 IC50 = 1700 nM T17345 COHL97 25093362 IC50 = 1360 nM T17345 C7PUO6 25093363 IC50 = 1250 nM T17345 CZE0Q4 25093364 IC50 = 7200 nM T17345 CGRF64 25093365 IC50 = 1420 nM T17345 CU0M5T 25093366 IC50 = 2770 nM T17345 CMQR72 25093367 IC50 = 3370 nM T17345 COE57Z 25093368 IC50 = 4200 nM T17345 CJV6X5 25093369 IC50 = 1360 nM T17345 C49FRJ 25093370 IC50 = 1380 nM T17345 C6W1TN 25107577 IC50 = 3500 nM T17345 CHU9G1 25107640 IC50 = 1500 nM T17345 C5WV3Q 25107642 IC50 = 5600 nM T17345 C2FU7W 25107643 IC50 = 2500 nM T17345 C5EP2L 25107644 IC50 = 2800 nM T17345 C3YT9V 25107645 IC50 = 2900 nM T17345 CQV0S4 25107646 IC50 = 2600 nM T17345 CO01BE 25138222 IC50 = 3200 nM T17345 CCK4R2 25138223 IC50 = 1300 nM T17345 C7P2RD 25138224 IC50 = 1180 nM T17345 C4VFL0 25138225 IC50 = 57 nM T17345 CR2MW1 25138226 IC50 = 130 nM T17345 CQO1Y3 25138227 IC50 = 360 nM T17345 COB9G8 25181586 IC50 > 33000 nM T17345 CF8EX5 25187895 IC50 = 200 nM T17345 C5BH0D 25187896 IC50 = 290 nM T17345 C3F5HV 25187897 IC50 = 210 nM T17345 CJ51SH 25187898 IC50 = 180 nM T17345 C1J4CH 25195124 IC50 = 750 nM T17345 C4P5UX 25195125 IC50 = 1410 nM T17345 C8IJB9 25218207 IC50 > 31000 nM T17345 C2SY4Z 25243853 Ki = 10000 nM T17345 CS6HE5 42627761 IC50 = 110000 nM T17345 C3C2GH 44123767 IC50 = 2370 nM T17345 C93GYN 44123768 IC50 = 2150 nM T17345 COI2S4 44136999 Ki = 15430 nM T17345 CWH0S1 44137255 Ki = 590 nM T17345 CI0BF4 44201386 IC50 = 19 nM T17345 CZ6DE0 44221143 IC50 = 300 nM T17345 CL8B5Q 44221144 IC50 = 840 nM T17345 CSJ28V 44221145 IC50 = 280 nM T17345 COT01Q 44221146 IC50 = 620 nM T17345 CS14YU 44221147 IC50 = 300 nM T17345 CA64NZ 44221340 IC50 = 600 nM T17345 CK5OL1 44221343 IC50 = 2600 nM T17345 CW0IM7 44221344 IC50 = 260 nM T17345 C0QZ7V 44221345 IC50 = 290 nM T17345 C74PHB 44221346 IC50 = 2200 nM T17345 CW39YO 44221347 IC50 = 350 nM T17345 CBHT60 44221538 IC50 = 260 nM T17345 CN5QV6 44221539 IC50 = 540 nM T17345 C9O1JI 44239402 IC50 = 173 nM T17345 CL13YN 44239406 IC50 = 19.9 nM T17345 C2PA5U 44239552 IC50 = 1790 nM T17345 C4NWP5 44246325 Ki = 2500 nM T17345 C2EW0I 44246326 Ki = 770 nM T17345 CSD8T0 44246327 Ki = 650 nM T17345 CMKF08 44246328 Ki = 12000 nM T17345 CAO87V 44246329 Ki = 5300 nM T17345 CLU2V3 44246330 Ki = 4600 nM T17345 CZ8U9G 44264907 IC50 = 1 nM T17345 CCJ0E5 44272288 IC50 = 27 nM T17345 CZ83VS 44273520 Ki = 776.25 nM T17345 CB9ZO8 44281305 IC50 = 320 nM T17345 C2O1KM 44281312 IC50 = 650 nM T17345 CFB79E 44282924 Ki = 46.2 nM T17345 C8QZ2E 44282925 Ki = 55.7 nM T17345 C51OKF 44282953 Ki = 0.131 nM T17345 C41RVE 44283340 IC50 = 1.5 nM T17345 CTZ9E5 44291963 Ki = 0.00033 nM T17345 C0D1VX 44291964 Ki = 0.0006 nM T17345 CHSF50 44291965 Ki = 0.00035 nM T17345 CDW63J 44292014 Ki = 0.00062 nM T17345 CG4KS0 44292015 Ki = 0.00021 nM T17345 C2DQ9E 44300934 IC50 = 1000 nM T17345 CN9U6W 44300964 IC50 = 420 nM T17345 CEV8X6 44300967 IC50 = 220 nM T17345 C54FJZ 44301716 IC50 = 190 nM T17345 C9JG5P 44308541 IC50 = 4.6 nM T17345 C0LZ8X 44308557 IC50 = 5.7 nM T17345 C7Q4RC 44309078 IC50 = 10.2 nM T17345 C8KST2 44314297 IC50 = 12 nM T17345 CBK5E3 44338827 IC50 = 14 nM T17345 CE14LA 44342970 IC50 = 27 nM T17345 CV6U1R 44343198 IC50 = 600 nM T17345 C6GME8 44346127 IC50 = 200 nM T17345 CN0GE5 44366301 Ki = 0.00019 nM T17345 C05HEV 44366644 IC50 = 18 nM T17345 C8AQ0F 44372902 IC50 = 0.84 nM T17345 C5F0ZB 44378252 Ki = 0.29 nM T17345 CZ7Y4L 44378321 Ki = 9.87 nM T17345 C3W2YH 44378322 Ki = 0.69 nM T17345 CM4Z7A 44421498 Ki = 0.077 nM T17345 CZ4CF9 44424991 IC50 = 2800 nM T17345 C0G4XZ 44523554 IC50 = 382.1 nM T17345 CB3D5L 44529842 IC50 > 100000 nM T17345 CPDY84 44531062 IC50 = 7.6 nM T17345 CN76FA 44568860 IC50 = 20 nM T17345 CPT49L 44582168 IC50 = 560 nM T17345 C0O4GX 44582169 IC50 = 1408 nM T17345 CM67QY 44582180 IC50 = 9340 nM T17345 CPS34N 44654525 IC50 = 2900 nM T17345 CMH39V 45267084 IC50 > 22000 nM T17345 C2V1MK 45267934 IC50 = 110000 nM T17345 CA53OY 45267939 IC50 > 27000 nM T17345 CYGI67 45268817 IC50 > 16000 nM T17345 C9H3DZ 45269661 IC50 > 20000 nM T17345 CE6W3J 45269665 IC50 > 24000 nM T17345 CW82HJ 45270497 IC50 > 28000 nM T17345 CW37YT 45270501 IC50 > 19000 nM T17345 CUNA34 45270504 IC50 > 21000 nM T17345 CGU1K7 45271328 IC50 > 25000 nM T17345 C17OKU 45271331 IC50 > 19000 nM T17345 C9M2ET 45271332 IC50 > 22000 nM T17345 CVGQ38 45272213 IC50 = 813000 nM T17345 CTFO90 45273072 IC50 > 23000 nM T17345 C50PYG 45273073 IC50 > 42000 nM T17345 C70SNR 45481871 IC50 = 1200 nM T17345 CM65ZU 45481878 IC50 = 60 nM T17345 CIGZ82 45481879 IC50 = 2300 nM T17345 CM3BD5 45481892 IC50 = 290 nM T17345 CP82LD 45481893 IC50 = 1580 nM T17345 CD1G7Q 45481939 IC50 = 400 nM T17345 CM1BK5 45481950 IC50 = 88 nM T17345 C1YAE7 46231368 IC50 = 4000 nM T17345 C1PJ2K 46231369 IC50 > 200000 nM T17345 CV38CS 46231370 IC50 > 200000 nM T17345 C5WM1J 46231371 IC50 > 200000 nM T17345 C5D7UV 46231372 IC50 > 200000 nM T17345 C9OER4 46231373 IC50 > 200000 nM T17345 CW0UO4 46231409 IC50 > 200000 nM T17345 C7OG0U 46231410 IC50 > 200000 nM T17345 CU5T7G 46231411 IC50 > 200000 nM T17345 COML63 46231412 IC50 > 200000 nM T17345 CK21OD 46231413 IC50 > 200000 nM T17345 C7Y5MX 46231414 IC50 > 200000 nM T17345 CN3HM6 46844539 Ki = 49.8 nM T17345 C5NOF1 46844540 Ki = 11.8 nM T17345 C9OM6V 46844541 Ki = 13 nM T17345 C2K9SC 46844649 Ki = 188 nM T17345 C6N1YZ 46861681 IC50 = 900 nM T17345 CY3M7K 46861682 IC50 = 1000 nM T17345 CIL1Z3 46886064 IC50 = 2000 nM T17345 CDV7P4 46886065 IC50 = 500 nM T17345 CO6E2M 46886122 IC50 = 500 nM T17345 CVX23N 46886123 IC50 = 800 nM T17345 CE9TL8 46886124 IC50 = 1000 nM T17345 COQ64I 46886125 IC50 = 1000 nM T17345 CPF1G2 46886145 IC50 = 2000 nM T17345 CB4YL0 46886146 IC50 = 2000 nM T17345 CM8B7K 46886147 IC50 = 800 nM T17345 C42TQK 46886148 IC50 = 3000 nM T17345 C5USK9 46886149 IC50 = 700 nM T17345 CCGH29 46886469 IC50 = 4000 nM T17345 C3PZL9 46886489 IC50 = 1000 nM T17345 CF27TO 46886490 IC50 = 3000 nM T17345 C26DLM 46886513 IC50 = 6000 nM T17345 CN4JM7 46886546 IC50 = 3000 nM T17345 CLY37J 46898100 Ki = 34 nM T17345 CQ3E4W 46898103 Ki = 7.6 nM T17345 C9H4WN 46905455 Ki = 9 nM T17345 CF4UK7 46907163 Ki = 24.5 nM T17345 CL14GQ 50992060 Ki = 22.5 nM T17345 CE0VL8 50994805 IC50 = 300000 nM T17345 CJA45X 52914860 IC50 = 90 nM T17345 CV21AI 52914861 IC50 = 100 nM T17345 CT8R2P 52918390 Ki = 1026 nM T17345 C7BY6M 52942956 Ki = 830 nM T17345 CE02NU 52943039 IC50 = 42000 nM T17345 CX24TS 52943277 IC50 = 340 nM T17345 CA62KU 52944152 Ki = 1600 nM T17345 CE37DL 52944456 IC50 = 314 nM T17345 CQV34K 52945403 Ki = 1100 nM T17345 C97XZA 52946619 Ki = 11000 nM T17345 CD9S4I 52947801 Ki = 4300 nM T17345 CA6IL3 52947802 Ki = 1300 nM T17345 C0MQ9Y 53346505 Ki = 1138 nM T17345 C2EGS5 53346506 Ki = 12.2 nM T17345 CAK50X 53346507 Ki = 26.3 nM T17345 COSG28 53346508 Ki = 12 nM T17345 C5U3KJ 53346509 Ki = 11.1 nM T17345 CD60FA 53346510 Ki = 5.8 nM T17345 CX2NV9 53346511 Ki = 4.5 nM T17345 CK72UF 53387838 IC50 > 100000 nM T17345 CXOL35 56595784 Ki = 572 nM T17345 CT45OM 56595785 Ki = 854 nM T17345 C9OW8X 56658455 IC50 > 100000 nM T17345 C1VYN7 56658457 IC50 > 100000 nM T17345 CDWN05 56658459 IC50 > 100000 nM T17345 CEX01L 56659280 Ki = 323 nM T17345 C6UHW8 56659281 Ki = 11.1 nM T17345 C0OSM1 56662749 Ki = 95.6 nM T17345 CO14BL 56665108 IC50 = 155 nM T17345 C6ER2F 56665410 IC50 > 100000 nM T17345 C1KWA9 56665412 IC50 > 100000 nM T17345 C7IX2A 56665414 IC50 > 100000 nM T17345 CPO4V8 56665416 IC50 > 100000 nM T17345 CUPO65 56666113 IC50 > 20000 nM T17345 CDC24L 56666218 Ki = 44.1 nM T17345 C9C7KW 56666219 Ki = 85 nM T17345 CH91WP 56666648 IC50 = 14000 nM T17345 CMHP59 56668551 IC50 = 5330 nM T17345 CQP5U2 56668841 IC50 > 100000 nM T17345 C2F0BA 56668843 IC50 > 100000 nM T17345 CDGX83 56668845 IC50 > 100000 nM T17345 CML5O9 56669623 Ki = 743 nM T17345 C2FBW1 56669624 Ki = 702 nM T17345 CCS0D3 56669625 Ki = 253 nM T17345 CP91XV 56673137 Ki = 20.9 nM T17345 C3JKO4 56673138 Ki = 22.2 nM T17345 COK3Z5 56675436 IC50 = 134 nM T17345 CUQ67O 56675715 IC50 > 100000 nM T17345 C6RCQ7 56676341 IC50 > 20000 nM T17345 C8AQ1O 56676459 Ki = 138 nM T17345 C7T2IG 56676460 Ki = 27.5 nM T17345 COA13E 56676461 Ki = 245 nM T17345 COG17M 56678776 IC50 = 548 nM T17345 C6VS9Y 56679010 IC50 = 21800 nM T17345 CJZ9B0 56679012 IC50 > 100000 nM T17345 C2B0OZ 56679014 IC50 > 100000 nM T17345 C90TMJ 56679774 Ki = 129 nM T17345 C29UVR 56679775 Ki = 10.1 nM T17345 COF0V7 56680536 IC50 = 49.04 nM T17345 CKX0H5 56682332 IC50 > 100000 nM T17345 CLGR37 56682334 IC50 > 100000 nM T17345 CDH01Q 56683111 Ki = 41.1 nM T17345 CRLK58 57381314 IC50 = 289 nM T17345 CZBG69 57381532 IC50 = 599 nM T17345 CRB3F1 57404325 IC50 > 250000 nM T17345 CA6DB4 57404326 IC50 = 50000 nM T17345 CBOX49 59608000 Ki = 4330 nM T17345 CTW7K2 60142113 IC50 = 5960 nM T17345 C7NCS0 60142250 IC50 = 2110 nM T17345 CC1X7M 60142382 IC50 = 1610 nM T17345 C3SH4V 60194459 Ki = 33.6 nM T17345 C25XOP 60199138 Ki = 18.1 nM T17345 C0WYU6 60199139 Ki = 20.2 nM T17345 CSA7P4 66563689 Ki = 47.6 nM T17345 CLJ4S9 66924089 IC50 = 15000 nM T17345 C47NRM 67607115 Ki = 1164 nM T17345 C5C0VZ 67607544 Ki = 1086 nM T17345 C8YM7S 67607902 Ki = 663 nM T17345 CVQW83 67615348 Ki = 320 nM T17345 C23NBA 67889361 Ki = 943 nM T17345 C95DAH 67889364 Ki = 2.9 nM T17345 CG5J2I 70687448 IC50 > 250000 nM T17345 CJAF56 70689505 IC50 > 250000 nM T17345 CZ48NJ 70695829 IC50 = 340 nM T17345 C0OB8G 71307952 IC50 = 57 nM T17345 C7KSO5 71449539 IC50 = 420 nM T17345 CJ6SQ8 71451328 IC50 = 33 nM T17345 CQ5YE6 71451881 Ki = 4680 nM T17345 C2F5XK 71453144 IC50 = 800 nM T17345 CTP47E 71454881 IC50 = 1070 nM T17345 CB1WD6 71456658 IC50 = 32 nM T17345 CSU17Q 71460350 IC50 = 18 nM T17345 C0UXW2 71462049 IC50 = 33 nM T17345 C7FEJ4 71462050 IC50 > 100000 nM T17345 CFP1O3 71463580 IC50 = 150 nM T17345 CKA6Q2 71463581 Ki = 11 nM T17345 C9SU7T 71520360 Ki > 55000 nM T17345 C9M2JK 71520483 Ki > 332000 nM T17345 C5N4XG 71521660 Ki > 110000 nM T17345 CGP9N4 71525312 IC50 = 1300 nM T17345 C3GN0W 71560185 IC50 = 400 nM T17345 CRZK12 71560290 IC50 = 250 nM T17345 CF06NE 71560291 IC50 = 1500 nM T17345 C2SJ7K 71560296 IC50 = 60 nM T17345 CCP40I 71560419 IC50 = 45 nM T17345 CR38HE 71560424 IC50 = 140 nM T17345 C06WSC 71560425 IC50 = 260 nM T17345 CV3A1O 71680871 IC50 = 190 nM T17345 CL5G6W 71680872 IC50 = 3650 nM T17345 CN8E7Q 71680873 IC50 = 250 nM T17345 CLT08Y 71680874 IC50 = 1000 nM T17345 CBW3F2 71680875 IC50 = 3900 nM T17345 CX82PD 71680876 IC50 = 2100 nM T17345 CGR6J5 71680877 IC50 = 5900 nM T17345 C23EQL 71681031 IC50 = 2200 nM T17345 CI9Y4J 71681032 IC50 = 7200 nM T17345 CO4V1J 71681033 IC50 = 2100 nM T17345 CU5IC1 71681034 IC50 = 450 nM T17345 C3I5KR 71681035 IC50 = 3100 nM T17345 CYG8K1 71681036 IC50 = 12 nM T17345 CNT81J 71681037 IC50 = 14 nM T17345 CCS0L2 71681187 IC50 = 4.7 nM T17345 C1X8KC 71681188 IC50 = 4.6 nM T17345 C46UPB 71681189 IC50 = 32 nM T17345 C7A1WK 71681190 IC50 = 340 nM T17345 CTIX90 71681191 IC50 = 5.6 nM T17345 C38MXU 71681192 IC50 = 46 nM T17345 CMJ47I 72771095 Ki = 1101 nM T17345 CZ4D3T 73386686 IC50 = 180 nM T17345 C8HKV5 76308482 IC50 = 3000 nM T17345 CR1SA3 76310814 Ki = 4000 nM T17345 CBH3C5 76311133 Ki = 841 nM T17345 CE8K7X 76314747 Ki > 5000 nM T17345 CWYV16 76314759 Ki = 1607 nM T17345 C9L4RE 76314760 Ki = 2922 nM T17345 CWN21Q 76318014 Ki = 4000 nM T17345 CE9Q3J 76318015 Ki = 200 nM T17345 CFM0V3 76318330 Ki = 749 nM T17345 CY8T3V 76319350 IC50 = 1.3 nM T17345 C17BXW 76319351 IC50 = 8.9 nM T17345 C0WMC2 76319379 IC50 = 10 nM T17345 C1B0TE 76322025 Ki = 723 nM T17345 C7N0YG 76323015 IC50 = 7300 nM T17345 CN7LS9 76325171 IC50 = 100 nM T17345 CL62UB 76325172 IC50 = 500 nM T17345 C2TF7J 76325354 Ki = 6000 nM T17345 CZ5DA3 76325652 Ki > 3000 nM T17345 C3PJ8X 76325653 Ki > 3000 nM T17345 CUC0O5 76325779 IC50 > 1000000 nM T17345 CQYO16 76328899 Ki = 3000 nM T17345 C12PIT 76328900 Ki = 3000 nM T17345 C1W8SP 76329213 Ki = 610 nM T17345 CVS27U 76329214 Ki = 437 nM T17345 CU1N3X 76330211 IC50 = 94 nM T17345 C8CQ5G 76332587 Ki = 3000 nM T17345 CM7X0D 76332864 Ki = 1564 nM T17345 CIAJ89 76336478 Ki = 2299 nM T17345 CYZJ97 76336479 Ki > 5000 nM T17345 C60IHU 76336487 Ki = 170 nM T17345 CJEA39 77461251 IC50 = 1200 nM T17345 CI0BY7 86276188 IC50 = 688 nM T17345 CLN0B2 86276189 IC50 = 625 nM T17345 CMF27J 86577836 IC50 = 172 nM T17345 C9EMA6 86577876 IC50 = 127 nM T17345 CC0F4M 86577948 IC50 = 136 nM T17345 CMV52E 86578029 IC50 = 208 nM T17345 C6F0NA 86578120 IC50 = 477 nM T17345 CUMG18 86578123 IC50 = 170 nM T17345 C4L6CM 86578162 IC50 = 49 nM T17345 C7T4CU 86578197 IC50 = 147 nM T17345 C37MOB 86578230 IC50 = 148 nM T17345 CQ3I8M 86578301 IC50 = 174 nM T17345 CVD2Y7 90666046 IC50 = 2730 nM T17345 CQS9A6 90666047 IC50 = 3100 nM T17345 C1UY6B 90666049 IC50 = 8720 nM T17345 CIG5W1 121493974 Ki = 200.77 nM T17345 CY21HZ 122164615 IC50 = 92 nM T17345 C8QB7N 124080837 IC50 = 511 nM T17345 C9NQ7B 124080838 IC50 = 1372 nM T17345 CW2D6Y 124081250 Ki = 388.62 nM T17345 CS04TC 124081251 Ki = 234.23 nM T17345 CO5MJ2 124220265 IC50 = 45 nM T17345 CE5F7Z 124220266 IC50 = 16 nM T17345 C6WU1A 124220267 IC50 = 41 nM T17345 CRE75U 127031638 IC50 = 30000 nM T17345 CY2W5J 127032512 IC50 > 100000 nM T17345 CCQ0D9 127032513 IC50 = 56400 nM T17345 CJ2Q3G 127032813 IC50 = 2400 nM T17345 CAVH35 127033390 Ki = 5.83 nM T17345 C2J9OY 127033391 IC50 = 700 nM T17345 CWK31L 127033392 IC50 = 300 nM T17345 CO9HL0 127033684 IC50 = 8000 nM T17345 C3HRW8 127033994 IC50 > 100000 nM T17345 CBT27N 127034482 IC50 = 5000 nM T17345 CT2OP4 127034483 IC50 = 7000 nM T17345 C6V8HZ 127034484 IC50 = 20000 nM T17345 CK7AG3 127036397 IC50 = 42000 nM T17345 CU7ZS5 127041310 IC50 = 310 nM T17345 C6ZX0J 127041311 IC50 = 310 nM T17345 C2WOC5 127041312 IC50 = 110 nM T17345 C8FD5L 127041909 IC50 = 2 nM T17345 C5Q2OX 127041910 IC50 = 42400 nM T17345 CD8MQ0 127041911 IC50 = 720 nM T17345 C2ILO0 127041912 IC50 = 320 nM T17345 COL16A 127043134 Ki = 2494.9 nM T17345 CWQ6Y4 127043135 Ki = 346.15 nM T17345 CE2R6W 127043324 Ki = 158.77 nM T17345 CEM63B 127043325 Ki = 376.62 nM T17345 C6BF8K 127045460 Ki = 451.15 nM T17345 C14WFB 129906767 IC50 = 72490 nM T17345 CEWR32 130301107 IC50 = 935 nM T17345 CM7E0A 132574708 IC50 = 52000 nM T17345 C4W5JI 134132161 IC50 = 2500 nM T17345 C32OQG 134133398 IC50 > 10000 nM T17345 C4W7YT 134135190 IC50 = 920 nM T17345 CW84JC 134135508 IC50 = 33.56 nM T17345 CF2T9N 134136051 IC50 > 10000 nM T17345 CI45FO 134136319 IC50 = 36.01 nM T17345 C17NRB 134136557 IC50 > 10000 nM T17345 CW0P8B 134136864 IC50 = 32.49 nM T17345 CS27VL 134138165 IC50 = 7.46 nM T17345 CP5IW7 134138953 IC50 = 9200 nM T17345 CCWD64 134139368 IC50 = 1100 nM T17345 CVZI26 134141070 IC50 = 86.11 nM T17345 CTO84X 134141850 IC50 > 10000 nM T17345 C34GRK 134142208 IC50 = 11.07 nM T17345 C3WXJ9 134143008 IC50 = 2100 nM T17345 CWT7F2 134144326 IC50 = 760 nM T17345 CY1X2T 134144992 IC50 = 6.46 nM T17345 C20VFD 134145574 IC50 = 4.08 nM T17345 C86PJW 134146078 IC50 > 10000 nM T17345 C1KFQ9 134147493 IC50 > 10000 nM T17345 CTHA87 134147818 IC50 = 18.28 nM T17345 CQG73J 134147949 IC50 > 10000 nM T17345 CCZ38F 134148801 IC50 > 10000 nM T17345 C2H7AI 134149549 IC50 = 4200 nM T17345 CQ0B2P 134150774 IC50 = 8.23 nM T17345 CA0J6U 134151081 IC50 = 56.75 nM T17345 C3RTP9 134152596 IC50 > 10000 nM T17345 CL72SR 134153211 IC50 > 10000 nM T17345 C2B4RW 134154165 IC50 = 3.72 nM T17345 CK6CQ1 134154523 IC50 > 75000 nM T17345 C18MPZ 134154991 IC50 = 46.62 nM T17345 C5MA8G 134155232 IC50 > 10000 nM T17345 C31ZAM 134156833 IC50 = 2800 nM T17345 C1IX4T 134812633 IC50 = 308 nM T17345 C0LJE4 134816733 IC50 = 11990 nM T17345 C4SZU6 134816735 IC50 = 15320 nM T17345 C3MKJ4 134816970 IC50 = 3670 nM T17345 CCT84X 135399760 IC50 > 240000 nM T17345 CQ4F8Y 135402053 IC50 = 910 nM T17345 C6AY2U 135403832 IC50 > 20000 nM T17345 C0LTC1 135404992 IC50 = 2100 nM T17345 C9EA3J 135407589 IC50 > 100000 nM T17345 C3MHI2 135427303 IC50 = 640 nM T17345 CSNH87 135431649 IC50 = 2100 nM T17345 CJ51DM 135443603 IC50 = 83 nM T17345 CS0I8R 135469335 IC50 > 95000 nM T17345 CS4M7U 135471854 IC50 = 170 nM T17345 C7YPI6 135481470 IC50 = 330 nM T17345 C7BQ1O 135487985 IC50 = 420 nM T17345 C79OVQ 135488791 IC50 = 11 nM T17345 CPZ72B 135488819 IC50 = 460 nM T17345 C5WV3M 135488820 IC50 = 110 nM T17345 CD40CJ 135502983 IC50 > 26000 nM T17345 C98GZD 135511915 IC50 > 54000 nM T17345 CFH82R 135516724 IC50 > 32000 nM T17345 CLB45I 135543610 IC50 > 62000 nM T17345 CK4FS8 135543796 IC50 = 7000 nM T17345 CV7HQ6 135545795 IC50 = 10000 nM T17345 C8N5QD 135545810 IC50 > 21000 nM T17345 CCF8H5 135545819 IC50 > 80000 nM T17345 C9K8DE 135545856 IC50 = 11000 nM T17345 C9Z4ES 135567027 IC50 > 20000 nM T17345 CE5O9J 135570463 IC50 = 22600 nM T17345 C06IDH 135746097 IC50 > 30000 nM T17345 CGLI18 135749904 IC50 = 120 nM T17345 CQ49YZ 135749905 IC50 > 39000 nM T17345 CBUS79 135749906 IC50 > 37000 nM T17345 C2HZK8 135749907 IC50 > 37000 nM T17345 CD48XU 135749908 IC50 > 35000 nM T17345 C9NZA4 135749909 IC50 > 35000 nM T17345 C0ME1H 135749910 IC50 = 33000 nM T17345 CMVH39 135749911 IC50 > 35000 nM T17345 CR4DU1 135749912 IC50 > 35000 nM T17345 C1H6ZF 135749913 IC50 > 31000 nM T17345 CR5NK7 135749914 IC50 > 24000 nM T17345 C1LV7B 135749915 IC50 > 32000 nM T17345 CQF8P5 135800109 IC50 > 24000 nM T17345 C4IDQ3 135855753 IC50 = 66600 nM T17345 C39FIY 135855754 IC50 = 20300 nM T17345 C0N1LQ 135855759 IC50 = 66600 nM T17345 C6A4QR 135855760 IC50 = 100000 nM T17345 CRV4K7 135855761 IC50 = 10200 nM T17345 CAUV24 135855764 IC50 = 72600 nM T17345 CYAS86 135855765 IC50 = 37300 nM T17345 CTG51U 135887103 IC50 = 4700 nM T17345 CE6TP5 135887104 IC50 = 8500 nM T17345 CY5H4A 135887105 IC50 = 400 nM T17345 CHT2O4 135887106 IC50 = 220000 nM T17345 CWL71S 135887124 IC50 = 2000 nM T17345 CNKW46 135887125 IC50 = 12000 nM T17345 CH1W2S 135887126 IC50 = 210 nM T17345 C6U0PF 135887127 IC50 = 250 nM T17345 COA6S0 135887128 IC50 = 1950 nM T17345 CBO9A7 135887129 IC50 = 320 nM T17345 CFIG79 135887147 IC50 > 1000000 nM T17345 CDA05G 135887148 IC50 > 1000000 nM T17345 CZB8O6 135960753 IC50 = 22000 nM T17345 CZ6C4R 135964391 IC50 > 29000 nM T17345 CUOV62 135964392 IC50 > 34000 nM T17345 CG23QU 135964393 IC50 > 32000 nM T17345 CR5EG8 135964397 IC50 > 28000 nM T17345 C0T2QO 135964404 IC50 > 32000 nM T17345 CD8WY9 135964405 IC50 > 25000 nM T17345 CRXF18 135964411 IC50 > 31000 nM T17345 C87XGZ 135964413 IC50 > 32000 nM T17345 CF1N5G 136002190 IC50 = 750 nM T17345 C3LWJ1 136002235 IC50 = 460 nM T17345 CJ7ES6 136016316 IC50 = 290 nM T17345 C24FWM 136016317 IC50 = 370 nM T17345 C9SMI1 136016318 IC50 = 340 nM T17345 CMG1F8 136016319 IC50 = 300 nM T17345 C1GE3H 136016320 IC50 = 640 nM T17345 C56SPO 136046100 IC50 = 430 nM T17345 CT0NK9 136046104 IC50 > 40000 nM T17345 CA1R9P 136046152 IC50 = 950000 nM T17345 C6CMD5 136046154 IC50 = 1300 nM T17345 CDMI28 136056632 IC50 = 3800 nM T17345 CL8YP6 136056633 IC50 = 530 nM T17345 CZ0JY3 136056634 IC50 = 1500 nM T17345 CMQ87O 136056635 IC50 = 3800 nM T17345 C5X9UG 136078523 IC50 = 650 nM T17345 CTK4I6 136078526 IC50 = 260 nM T17345 CML42R 136092224 IC50 63300 nM T17345 C8O2GN 136109165 IC50 = 100 nM T17345 CALV20 136109177 IC50 = 100 nM T17345 CKI9N0 136136563 IC50 = 3000 nM T17345 CG3OA8 136136566 IC50 = 1400 nM T17345 C7QAB0 136171375 IC50 = 3200 nM T17345 C6XHI1 136171377 IC50 = 280 nM T17345 CVKL45 136171378 IC50 = 300 nM T17345 C23HGZ 136191424 Ki ~ 600 nM T17345 CVY71R 137300720 IC50 > 10000 nM T17345 CWE38X 137491959 IC50 = 12500 nM T17345 CM10NY 137631470 IC50 = 28000 nM T17345 CAZB89 137631503 IC50 = 2250 nM T17345 CWR72A 137632901 IC50 = 19000 nM T17345 CYF76S 137633375 IC50 = 5330 nM T17345 CFUY16 137633842 IC50 > 27000 nM T17345 CNT9K1 137634037 IC50 = 9.2 nM T17345 CZ5B9O 137634433 IC50 = 16900 nM T17345 CPB9Q3 137634556 IC50 = 1260 nM T17345 C0PNW5 137635062 IC50 = 450 nM T17345 CS23KQ 137635618 IC50 > 28000 nM T17345 CF5S9P 137636125 IC50 = 4 nM T17345 C7N6WS 137636390 IC50 > 150000 nM T17345 C53CKY 137636400 IC50 = 853 nM T17345 COE67T 137637328 IC50 > 50000 nM T17345 CL87FM 137638209 IC50 = 108 nM T17345 CA01DG 137638564 IC50 = 3.2 nM T17345 CP8X2O 137639098 IC50 = 290 nM T17345 CL95CK 137639545 IC50 = 6.1 nM T17345 CK6GP0 137640129 IC50 = 14800 nM T17345 C4QHY1 137640582 IC50 = 3610 nM T17345 C8MQ6U 137642178 IC50 = 2.6 nM T17345 C19WKB 137642364 IC50 = 6000 nM T17345 CU8YX6 137643005 IC50 > 27000 nM T17345 CW27XK 137644048 IC50 = 25000 nM T17345 C4N6GR 137644261 IC50 = 36 nM T17345 CT6CI1 137644294 IC50 = 710 nM T17345 C9YX2K 137644352 IC50 = 4000 nM T17345 CA7QW8 137645236 IC50 = 53.4 nM T17345 CSXF17 137645367 IC50 = 2840 nM T17345 CO0U6R 137646091 IC50 = 1400 nM T17345 C4NJB5 137646478 IC50 = 4.2 nM T17345 C83JEY 137646749 IC50 = 13.1 nM T17345 CRU6D2 137647615 IC50 = 5.3 nM T17345 CA7Y9F 137648264 IC50 = 4780 nM T17345 CZGU30 137648786 IC50 = 44 nM T17345 CQED79 137651284 IC50 = 2550 nM T17345 C5V4MO 137651590 IC50 = 14.1 nM T17345 CL1DZ0 137651595 IC50 = 5280 nM T17345 CQUY83 137652218 IC50 > 29000 nM T17345 CB3H5W 137652434 IC50 = 6.4 nM T17345 CSR07T 137654267 IC50 = 3190 nM T17345 CR71UO 137654559 IC50 = 950 nM T17345 C9JT1N 137655519 IC50 > 30000 nM T17345 C5XVK8 137656132 IC50 = 4130 nM T17345 C1M2YZ 137657601 IC50 = 2480 nM T17345 CQJD20 137657673 Ki = 13170 nM T17345 CX2T5K 137658038 IC50 = 35.6 nM T17345 CYV97X 137659199 IC50 = 4340 nM T17345 CO79SP 137659251 IC50 = 1670 nM T17345 CYML31 137659929 IC50 = 59.2 nM T17345 CETP42 137660220 IC50 = 3.4 nM T17345 C8W5GY 137660580 IC50 = 20100 nM T17345 C4UF6M 137660773 IC50 = 4.8 nM T17345 CD6VN2 137660870 IC50 = 9 nM T17345 C7V3LC 137661421 IC50 = 3.9 nM T17345 CFI5E0 137661591 IC50 = 18 nM T17345 CC8QH2 138460007 IC50 = 1090 nM T17345 C9NL0Q 138460276 IC50 = 1430 nM T17345 CL45VQ 145949793 Ki = 530 nM T17345 CX76CQ 145954183 Ki = 1400 nM T17345 C8QO7R 145955925 Ki = 640 nM T17345 CE0VX2 145967688 IC50 = 700 nM T17345 C49HWY 145967911 IC50 = 970 nM T17345 C4Q8MH 145968315 IC50 = 1101 nM T17345 CL72EN 145968368 IC50 = 1400 nM T17345 CK5H1X 145968380 IC50 = 579 nM T17345 C7ILN2 145968384 IC50 = 2730 nM T17345 CKC3W9 145968635 IC50 = 70510 nM T17345 C2V6SX 145968836 IC50 = 2318 nM T17345 CBP38L 145968849 IC50 = 590 nM T17345 C2LD6U 145968997 IC50 = 1917 nM T17345 CZ6LQ5 145969012 IC50 = 7930 nM T17345 C7N8WS 145969103 IC50 = 12290 nM T17345 CR9J7O 145970201 IC50 = 610 nM T17345 C04XEC 145970467 IC50 = 1130 nM T17345 C48KNM 145970614 IC50 = 811 nM T17345 CBXY67 145970730 IC50 = 2530 nM T17345 CT72GK 145970859 IC50 = 60 nM T17345 CIG4X8 145970868 IC50 = 11230 nM T17345 CHC2I0 145971065 IC50 = 2100 nM T17345 CEA95O 145971179 IC50 = 2046 nM T17345 CLY9F6 145988837 IC50 = 1104 nM T17345 CG36PF 145989276 IC50 > 100000 nM T17345 CUP4Z9 151456061 IC50 = 1360 nM T17345 CSL7O9 152598220 IC50 = 1790 nM T17345 C5OVQ3 152617142 IC50 = 347 nM T17345 CI79YB 155510882 IC50 = 1630 nM T17345 CB8J3L 155511255 IC50 = 37.94 nM T17345 C7GFM4 155512559 Ki = 18.41 nM T17345 CGK20J 155513582 IC50 = 819 nM T17345 C6D2CN 155514408 IC50 = 903 nM T17345 CS84IM 155515034 Ki = 555.55 nM T17345 CO9ZD7 155516975 IC50 = 29.29 nM T17345 CPX7N5 155517476 Ki = 23.42 nM T17345 CK8UH6 155518935 Ki = 13.41 nM T17345 C1ZA0M 155520729 IC50 = 1098 nM T17345 CHW46G 155523087 IC50 >= 1000 nM T17345 CUY38N 155523154 Ki = 18.24 nM T17345 CF4JM8 155523234 IC50 = 10 nM T17345 CEA02Z 155527030 Ki = 508.88 nM T17345 CT6S0G 155527248 IC50 = 237 nM T17345 CLO94T 155527394 Ki = 14.36 nM T17345 C3U4ED 155528338 IC50 = 300 nM T17345 C4N5QE 155528668 Ki = 19.55 nM T17345 C8PH3I 155529256 IC50 = 2626 nM T17345 C1GZ7W 155529285 Ki = 21.72 nM T17345 CR0O1S 155529844 IC50 > 30000 nM T17345 C87EWF 155530674 IC50 = 1100 nM T17345 CJ1P8L 155531623 IC50 = 1330 nM T17345 CT40PE 155532707 IC50 = 1800 nM T17345 C5H8LY 155532752 Ki = 32.89 nM T17345 C9OW3C 155533311 Ki = 74.16 nM T17345 C2P4MC 155534197 IC50 = 4125 nM T17345 C51XLA 155539843 Ki = 22.07 nM T17345 CFP3Y7 155540286 IC50 >= 1000 nM T17345 CG1S5K 155542983 IC50 = 65.88 nM T17345 C49SMW 155543062 IC50 = 2253 nM T17345 C0SNO1 155543141 IC50 = 3260 nM T17345 C5GZ1N 155543331 IC50 = 980000 nM T17345 CC20PV 155543847 IC50 = 1808 nM T17345 CP15AX 155544485 Ki = 48.67 nM T17345 C9MU3J 155546590 IC50 = 53.42 nM T17345 C9QN6E 155547319 IC50 = 100 nM T17345 CA4T8J 155548037 IC50 = 541 nM T17345 CNA65G 155549118 IC50 = 5980 nM T17345 CM5F3R 155550798 Ki = 8.72 nM T17345 CKBA16 155550915 IC50 = 973 nM T17345 C4SXE2 155551604 Ki = 32.43 nM T17345 CPV2I5 155552635 IC50 = 210 nM T17345 C2NIY4 155552687 Ki = 34.84 nM T17345 C3U7CK 155552787 IC50 = 1540 nM T17345 C0V2SW 155553051 IC50 = 125000 nM T17345 C1WXN8 155553663 IC50 = 2710 nM T17345 C4PLU8 155554619 Ki = 27.27 nM T17345 CVHM01 155555730 Ki = 12.5 nM T17345 C3KM4N 155556589 IC50 = 48.95 nM T17345 C4WH0C 155557612 Ki = 12.77 nM T17345 C8WB9O 155558582 IC50 >= 1000 nM T17345 CDB7F2 155560431 IC50 > 30000 nM T17345 CMYU10 155561126 Ki = 52.39 nM T17345 CE84AM 155561456 IC50 = 670 nM T17345 CXYW29 155562270 IC50 = 200 nM T17345 CU71YW 155562818 IC50 = 1571 nM T17345 CFM53Y 155563602 IC50 = 1576 nM T17345 CQ97VE 155565527 IC50 = 180000 nM T17345 C6COP9 155565754 IC50 = 1300 nM T17345 CV6WP8 155566484 IC50 = 9.28 nM T17345 C8BGX5 155567131 Ki = 29.05 nM T17345 CWON57 155567297 Ki = 45.97 nM T17345 C8M7LB 155567321 IC50 = 1338 nM T17345 CGMA98 155567948 Ki = 13.59 nM T17345 CUV9H3 155568251 IC50 = 2800 nM T17345 C9S2ON 155568330 IC50 = 468 nM T17345 C5ILH2 155568439 IC50 = 1373 nM T17345 D00IBG 643976 IC50 = 325000 nM T17345 D01HKU 44428667 IC50 = 120 nM T17345 D02ZCP 446244 IC50 = 620 nM T17345 D02ZPZ 6532431 Ki = 1.8 nM T17345 D03DRF 46886486 IC50 = 2000 nM T17345 D04PAW 16216218 IC50 = 250 nM T17345 D05WHM 6917908 IC50 = 4.4 nM T17345 D06DIH 158376 IC50 = 220 nM T17345 D06ERH 637760 IC50 > 100000 nM T17345 D06QEN 467889 Ki = 230 nM T17345 D06UPT 446752 IC50 = 4.3 nM T17345 D07LSP 135438608 IC50 = 1900 nM T17345 D07XLJ 462120 IC50 = 2400 nM T17345 D08GPU 490662 Ki = 2.9 nM T17345 D0B0UI 44428664 IC50 = 70 nM T17345 D0H8AW 291270 IC50 = 23000 nM T17345 D0J4KJ 446245 IC50 = 940 nM T17345 D0JY6J 93114 Ki = 10.4 nM T17345 D0LH5P 100516 IC50 = 4.1 nM T17345 D0ME8Z 24778025 IC50 = 0.39 nM T17345 D0O9YG 9049 Ki = 55.6 nM T17345 D0P9XE 46871716 Ki = 93 nM T17345 D0R4PS 135403648 Ki = 2370 nM T17345 D0S4ZT 46886512 IC50 = 5000 nM T17345 D0Y3TU 334409 Ki = 1 nM T17345 D0Z9QC 135517463 IC50 = 34 nM T17345 D0ZG7W 11441554 IC50 > 100000 nM T77393 C6F2WU 700755 Ki > 1000000 nM T77393 CZS6I0 720519 Ki > 1000000 nM T77393 CJL6Z8 765511 Ki = 323000 nM T77393 CQ2S4B 910123 Ki = 61000 nM T77393 C9AVC3 1006789 IC50 = 25000 nM T77393 C5XG0W 1006800 IC50 = 13620 nM T77393 C36IHN 1006808 IC50 = 24000 nM T77393 C3N7ZL 1006833 IC50 = 9630 nM T77393 CMD15J 1006856 IC50 = 22000 nM T77393 CA1X5I 1025961 IC50 = 22000 nM T77393 C3D1ZK 1266319 IC50 = 38000 nM T77393 CKR60Y 2810167 IC50 = 6000 nM T77393 CU0VC2 2943337 IC50 > 20000 nM T77393 CN9SE0 3308644 Ki = 843000 nM T77393 CAV9I1 3697667 Ki = 8440 nM T77393 C9FT3D 13430822 Ki = 589000 nM T77393 C9CR0M 15561337 Ki = 651000 nM T77393 C6C2JF 16483718 IC50 = 24000 nM T77393 C1XOL3 16487351 IC50 = 22000 nM T77393 CL3C9H 16645214 IC50 = 22000 nM T77393 C78LBG 16645215 IC50 = 30000 nM T77393 C4IAR3 16645216 IC50 = 12970 nM T77393 C6IM7Q 24757930 Ki = 27300 nM T77393 C6XPA0 39845054 IC50 = 48000 nM T77393 CC30IP 39845125 IC50 = 23000 nM T77393 CT4OS9 39845172 IC50 = 13000 nM T77393 CI9N1O 46864279 Ki = 120 nM T77393 CM51WO 46864280 Ki = 20 nM T77393 C81DFP 46866889 Ki = 200 nM T77393 C1U3KE 46867009 Ki = 3 nM T77393 CCKI47 46867010 Ki = 20 nM T77393 CT24XZ 46867121 Ki = 6300 nM T77393 C5WP7S 46867122 Ki = 7300 nM T77393 CM27BD 46867257 Ki < 1 nM T77393 CS6J9I 46889977 Ki = 160 nM T77393 C4DR8T 46889978 Ki = 30 nM T77393 CAJ5E1 46889979 Ki = 90 nM T77393 C8NY4I 46889980 Ki = 160 nM T77393 CK48PC 46889981 Ki = 80 nM T77393 CM5XP9 46889982 Ki = 27000 nM T77393 C0SFR4 46889983 Ki > 50000 nM T77393 C0L7GM 46889984 Ki = 3200 nM T77393 CPE06Y 46889985 Ki > 50000 nM T77393 CZ9VF6 46889986 Ki = 150 nM T77393 CXV0F2 46889987 Ki = 6500 nM T77393 COKG74 46889988 Ki = 1600 nM T77393 CP7E6H 46889989 Ki = 15100 nM T77393 CQTU62 46889993 Ki = 15000 nM T77393 CO7ZX4 46889994 Ki = 9000 nM T77393 C1WP0Q 46889995 Ki = 15600 nM T77393 C52WPZ 53356803 Ki < 1 nM T77393 C5JOC6 54766612 Ki < 1 nM T77393 CBT35C 54766613 Ki < 1 nM T77393 CH1KS7 70679466 IC50 = 338.2 nM T77393 C8IPK7 71586081 IC50 = 0.9 nM T77393 CY1J9L 85721372 IC50 > 20000 nM T77393 CN7F5K 127048565 IC50 = 660.9 nM T77393 C5J6QE 127048926 IC50 = 733.3 nM T77393 C9IK3M 127048927 IC50 = 127.4 nM T77393 CZ9T0Q 127048933 IC50 > 20000 nM T77393 C4DL6C 127048934 IC50 = 11400 nM T77393 CUN7F3 127048935 IC50 > 20000 nM T77393 CH1K3Y 127049251 IC50 = 206.1 nM T77393 CG84YX 127049252 IC50 = 207.2 nM T77393 CO0ZG4 127049253 IC50 = 130 nM T77393 C1IPG6 127049254 IC50 > 20000 nM T77393 CT10RI 127050095 IC50 > 20000 nM T77393 CL5V0S 127050385 IC50 = 1604 nM T77393 CXH7K0 127050386 IC50 = 198.5 nM T77393 C19BTR 127050387 IC50 = 465.7 nM T77393 C7T5WN 127052836 IC50 = 392.6 nM T77393 CC71PB 127052837 IC50 = 103.9 nM T77393 CBI1K8 127052955 IC50 > 20000 nM T77393 CO8X1P 127052956 IC50 > 20000 nM T77393 CR8JM3 127052957 IC50 > 20000 nM T77393 C75QVY 127052958 IC50 > 20000 nM T77393 CX8MA9 127052959 IC50 > 20000 nM T77393 CGY79B 127052960 IC50 > 20000 nM T77393 CQF37D 132580838 IC50 = 46.5 nM T77393 C0LHZ3 132580839 IC50 = 26.4 nM T77393 CN3MY7 134129874 IC50 > 20000 nM T77393 CVZS03 134129880 IC50 = 81.5 nM T77393 CO75BV 134129898 IC50 = 340.8 nM T77393 C15JEQ 134129903 IC50 = 13600 nM T77393 CSMF23 134129955 IC50 = 70.1 nM T77393 C8WNH1 134130001 IC50 > 20000 nM T77393 CZV10G 134130017 IC50 = 102.1 nM T77393 CMLA18 134130074 IC50 = 5800 nM T77393 C6OPH7 134130102 IC50 = 197.6 nM T77393 CZ9X1B 134130118 IC50 > 20000 nM T77393 CYO72F 134130195 IC50 = 47.9 nM T77393 C8M9NP 134130199 IC50 = 285.1 nM T77393 CN0HP5 134130274 IC50 = 104.6 nM T77393 C9DJC5 134130275 IC50 = 1363 nM T77393 C7A3FI 134130278 IC50 = 77.1 nM T77393 C1UR5D 134130359 IC50 > 20000 nM T77393 CL3Z2T 134130407 IC50 = 30.1 nM T77393 CO9BF6 134130408 IC50 = 1553 nM T77393 C9YS8H 134130465 IC50 = 92.5 nM T77393 CB08EV 134130500 IC50 = 62.5 nM T77393 CY24IA 134130560 IC50 = 113.4 nM T77393 C8XUN4 134130570 IC50 = 18.2 nM T77393 CRIW18 134130589 IC50 > 20000 nM T77393 CM5US2 134130592 IC50 = 8.5 nM T77393 CXH06K 134130734 IC50 = 285.3 nM T77393 CB61JP 134130757 IC50 = 7.6 nM T77393 C48BIF 134130903 IC50 > 20000 nM T77393 C5KRU7 134130925 IC50 = 75.8 nM T77393 CZ4J1P 134130945 IC50 = 95.6 nM T77393 CBP5O4 134130958 IC50 = 421.9 nM T77393 CYL7R9 134131003 IC50 = 88.7 nM T77393 CYFW16 134131026 IC50 = 50.2 nM T77393 CIN01V 134131045 IC50 = 15 nM T77393 CBF6E4 134131065 IC50 = 77.9 nM T77393 C4B7MN 134131117 IC50 = 3186 nM T77393 C59JMH 134131257 IC50 = 1093 nM T77393 CHJ39K 134131302 IC50 > 20000 nM T77393 C7GBH3 134131374 IC50 > 20000 nM T77393 C7SKU8 134131410 IC50 = 76 nM T77393 C3O4TN 134131411 IC50 > 20000 nM T77393 CF5S3O 134131548 IC50 = 70 nM T77393 C30GML 134131594 IC50 = 80.4 nM T77393 C56NTH 134135619 IC50 = 483.5 nM T77393 C17JRH 134135674 IC50 > 20 nM T77393 C7PN4W 134135702 IC50 = 263.5 nM T77393 C10RIC 134136312 IC50 = 1171 nM T77393 CCN03X 134137047 IC50 > 20 nM T77393 C3ZA5K 134137967 IC50 > 20 nM T77393 C71GIB 134140087 IC50 = 283.9 nM T77393 CB0NA6 134143014 IC50 = 162.4 nM T77393 C9IGQ2 134143930 IC50 > 20 nM T77393 C2RS6U 134144485 IC50 > 20 nM T77393 C3G6AQ 134145642 IC50 = 433.2 nM T77393 C9AJI4 134145666 IC50 > 20 nM T77393 C72APM 134148078 IC50 = 454 nM T77393 CO57LR 134148875 IC50 > 20 nM T77393 CG74JP 134149023 IC50 > 20 nM T77393 CCMR94 134149266 IC50 > 20 nM T77393 CRMX45 134149901 IC50 > 20 nM T77393 CG78KP 134153992 IC50 = 244.9 nM T77393 CF1KZ5 134155604 IC50 = 58.8 nM T77393 CI3CN5 134157644 IC50 = 811.6 nM T77393 CH1S6B 134364156 Ki = 3.53 nM T77393 C8LV1Q 134364178 Ki = 105 nM T77393 C4MIV7 134369551 Ki = 7540 nM T77393 CK6ZM1 134369552 Ki = 7210 nM T77393 C1OLR0 134369556 Ki = 665 nM T77393 CHNY14 134369557 Ki = 2600 nM T77393 C3LO6E 134369558 Ki = 17600 nM T77393 CLH26P 134369559 Ki = 219 nM T77393 C59CPA 134369560 Ki = 503 nM T77393 CJ3R0T 134369561 Ki = 3130 nM T77393 C12FZJ 134369563 Ki = 3910 nM T77393 C7QFN0 134369568 Ki = 690 nM T77393 CKUR59 134369576 Ki = 1380 nM T77393 C1Y3CD 134369579 Ki = 4130 nM T77393 C4F5BV 134369583 Ki = 1260 nM T77393 CK0JG5 134369594 Ki = 480 nM T77393 C0LKG2 134369619 Ki = 1460 nM T77393 CR6ZE1 134369620 Ki = 148 nM T77393 CYM14L 134369623 Ki = 118 nM T77393 C9Z7GJ 134369629 Ki = 42.5 nM T77393 CN8DO3 134369637 Ki = 27.6 nM T77393 CDVS67 134369647 Ki = 473 nM T77393 C3OE7I 134369648 Ki = 9.89 nM T77393 CLC39Q 134369650 Ki = 22.8 nM T77393 C71NAT 134369652 Ki = 28.9 nM T77393 CH8C7V 134369653 Ki = 76.1 nM T77393 C2C7AZ 134369665 Ki = 13.1 nM T77393 CT61JH 134369666 Ki = 185 nM T77393 CRW1A0 134369668 Ki = 184 nM T77393 CBW56J 134369669 Ki = 95 nM T77393 C6B9RO 134369670 Ki = 51.9 nM T77393 C4F1OP 134369672 Ki = 20.7 nM T77393 C15BUR 134369676 Ki = 2.82 nM T77393 CP46RA 134369681 Ki = 924 nM T77393 C63WBR 134369708 Ki = 16.4 nM T77393 C8B3LO 137349384 Ki = 85200 nM T77393 CSM61B 138319680 Ki = 0.044 nM T77393 CK27NV 138470399 Ki = 9.36 nM T77393 CMTD84 138470404 Ki = 65.1 nM T77393 CMG7V3 138470418 Ki = 2.51 nM T77393 CB24SI 138470423 Ki = 0.902 nM T77393 C8X5US 145981722 Ki = 109000 nM T77393 C9EAI7 145982119 Ki > 125000 nM T77393 CJ23AP 145988536 Ki = 1120 nM T77393 CF0BR7 145989019 Ki = 64000 nM T77393 C0IUB7 145989142 Ki = 117000 nM T77393 C49OYH 145990286 Ki > 125000 nM T77393 CK2C9E 145991249 Ki = 64300 nM T77393 C7YAG8 145992826 Ki = 118000 nM T77393 CX74VN 145992918 Ki = 29700 nM T77393 C2AHW4 145993387 Ki = 4.94 nM T49031 D00UVA 11556711 IC50 = 2.7 nM T49031 D01MML 49867936 IC50 = 8.44 nM T49031 D04AIT 5280445 IC50 = 1300 nM T49031 D0E7PQ 5311 IC50 > 25000 nM T49031 D0K8KX 5280343 IC50 = 2000 nM T49031 D0SH3I 387447 Ki = 0.55 nM T49031 D0T9TJ 3034010 IC50 > 100000 nM T49031 D05KED 53340666 IC50 > 25000 nM T49031 D07SDQ 969516 IC50 = 10000 nM T49031 D0DP0J 92135659 IC50 = 1670 nM T49031 D0F9BT 25067547 IC50 = 10 nM T49031 D0L4FS 5280961 IC50 = 9260 nM T49031 D0N0RN 11347535 IC50 = 22 nM T49031 D0U2BH 65064 IC50 = 86 nM T49031 D0VO0T 24800541 IC50 = 3 nM T49031 D0Y2SW 25183872 IC50 = 3 nM T49031 D0U7OU 3220 IC50 = 1220 nM T49031 CKGX24 7060 IC50 > 25000 nM T49031 C29BVT 11926 IC50 > 25000 nM T49031 CTK25Q 72277 IC50 = 1200000 nM T49031 CPSA65 80458 IC50 = 3000 nM T49031 CNIW58 107905 IC50 = 194 nM T49031 CDZ65K 199472 IC50 = 187 nM T49031 CA6ID2 241903 IC50 = 4580 nM T49031 C9A1KC 282849 IC50 > 25000 nM T49031 CF5T0S 282888 Ki = 2180 nM T49031 CPEL12 336327 IC50 > 100000 nM T49031 C46ZED 434315 Ki = 2120 nM T49031 C7HME8 439246 IC50 = 41600 nM T49031 C3YF4P 462382 IC50 = 1.2 nM T49031 C1MY6Z 490002 Ki = 2.3 nM T49031 CZ0AH3 638278 IC50 = 4880 nM T49031 C2DC6P 684753 Ki = 11500 nM T49031 CS4F8G 688857 IC50 = 5210 nM T49031 C2JU6P 833502 Ki = 10900 nM T49031 CS1P9Y 906456 IC50 = 172200 nM T49031 C2CR9F 1722365 Ki = 2010 nM T49031 C5FC0Z 2215326 IC50 = 3500 nM T49031 CL3KS0 5497183 IC50 = 61 nM T49031 CL9NX1 6610292 IC50 = 160 nM T49031 CK1U3G 6871286 IC50 > 10000 nM T49031 CL4VY9 9874885 Ki = 0.72 nM T49031 C3TDO0 9920246 IC50 = 1900 nM T49031 COK6X9 9960660 Ki < 1 nM T49031 CB2KX5 10032943 Ki = 0.5 nM T49031 CDPZ20 10099985 Ki = 5.7 nM T49031 C56PLQ 10258908 Ki = 0.72 nM T49031 CV25EX 10346881 IC50 = 51090 nM T49031 CO2HE7 10461001 Ki = 38 nM T49031 C5CBI2 10484581 Ki = 0.65 nM T49031 CDW5Y2 10542930 IC50 > 10000 nM T49031 CLU69K 10628969 IC50 = 420 nM T49031 CU8I1N 11243977 EC50 = 10 nM T49031 C1A2IM 11512726 IC50 = 2.9 nM T49031 C31TAR 11520347 Ki = 500 nM T49031 C6B5UF 11520360 IC50 = 52 nM T49031 C3GE9O 11532672 IC50 = 3360 nM T49031 CF2R5T 11534087 IC50 = 17 nM T49031 C61XQZ 11542118 IC50 = 1.5 nM T49031 CV56WA 11548000 IC50 = 6560 nM T49031 CWX6Y7 11549328 Ki = 32 nM T49031 C8MEH4 11549343 Ki = 140 nM T49031 C3BTN5 11556651 IC50 = 2.5 nM T49031 C2OPE1 11556685 IC50 = 2.4 nM T49031 CMH1V5 11563622 IC50 = 570 nM T49031 C8T5DM 11570453 IC50 = 170 nM T49031 C9KS5X 11578303 IC50 = 120 nM T49031 CB1L7I 11583999 IC50 = 260 nM T49031 CETS82 11585586 Ki = 45 nM T49031 CW7Z2P 11585713 IC50 = 2500 nM T49031 CH4RG7 11591941 IC50 > 10000 nM T49031 CFH34R 11598900 IC50 = 21000 nM T49031 CR9VG2 11599767 IC50 = 5.9 nM T49031 CKN7V8 11600122 Ki = 0.51 nM T49031 CO9PW8 11607192 IC50 = 78 nM T49031 CW0T9J 11613973 IC50 = 56000 nM T49031 C9OT1M 11621366 IC50 = 1.1 nM T49031 CX51NM 11636132 IC50 = 540 nM T49031 CB70KR 11636235 IC50 = 10 nM T49031 CLUA24 11636269 IC50 = 1400 nM T49031 CYR86V 11664755 IC50 = 49 nM T49031 CJFM60 11671614 IC50 = 4.3 nM T49031 CZ68VB 11672014 IC50 = 44 nM T49031 CZF9M1 11686028 Ki = 130 nM T49031 CE82UG 11692971 IC50 = 28000 nM T49031 CJE3N7 11693095 IC50 = 6.7 nM T49031 CJ1H4E 11700022 IC50 = 14 nM T49031 CX9D8R 11707332 IC50 = 2300 nM T49031 CF3Y2Q 11714595 IC50 = 49 nM T49031 CLBD57 15479395 IC50 = 220 nM T49031 C8D5OY 16084592 IC50 = 6670 nM T49031 C5RA8E 17480620 Ki = 7550 nM T49031 C7JCW4 21140132 Ki = 4700 nM T49031 C19EMT 23649126 IC50 = 700 nM T49031 CU0FE7 24752894 IC50 > 10000 nM T49031 C9E8MQ 24753965 IC50 = 7190 nM T49031 C7A4VT 24966905 IC50 > 10000 nM T49031 C5RCN7 24966906 Ki = 580 nM T49031 C1LJZ3 24966907 IC50 > 10000 nM T49031 C1MJ0W 25053219 IC50 = 1440 nM T49031 C64CJD 25111344 IC50 > 5000 nM T49031 CG52FR 42601513 Ki = 843 nM T49031 CB8H2Y 42612596 IC50 = 49 nM T49031 CN6D8U 44190246 IC50 = 4.37 nM T49031 CKH7Y0 44190247 IC50 = 1.6 nM T49031 CC8FG3 44191199 IC50 = 1.2 nM T49031 CKM83N 44307872 IC50 = 140 nM T49031 C21GXN 44410779 Ki > 450000 nM T49031 CXS71L 44411047 IC50 = 430 nM T49031 C90ZUI 44411546 IC50 = 2230 nM T49031 CMV46Q 44411707 IC50 = 4320 nM T49031 CP03SX 44411716 IC50 = 4150 nM T49031 CHFA42 44477958 IC50 = 15300 nM T49031 C69XJY 44477959 IC50 = 10000 nM T49031 C7NW5T 44555355 IC50 = 0.08 nM T49031 CN57MC 44583022 IC50 = 10 nM T49031 C9GUZ5 45140224 IC50 = 31 nM T49031 C5GAE4 45140225 IC50 = 3 nM T49031 C9RL7F 46233200 IC50 = 1 nM T49031 CNFQ84 46233201 IC50 = 2 nM T49031 CB57EF 46233202 IC50 = 100 nM T49031 CZ29GM 46233203 IC50 = 200 nM T49031 CQO52J 46233204 IC50 = 130 nM T49031 C4V9JP 46233205 IC50 = 300 nM T49031 C38TWK 46233206 IC50 = 524807460.3 nM T49031 CM81GQ 46864294 IC50 = 2.1 nM T49031 CX1YJ8 49799952 IC50 = 4.26 nM T49031 CHO3X2 49799953 IC50 = 7.63 nM T49031 C3XCL9 49859747 Ki = 2430 nM T49031 CIW0H6 50899478 IC50 = 0.55 nM T49031 C5QU2O 50899571 IC50 = 0.42 nM T49031 C8WD6E 50899573 IC50 = 0.39 nM T49031 CWDL81 52948098 IC50 = 16 nM T49031 C5EQD3 53362657 IC50 = 303.8 nM T49031 C7Q0RA 54455523 IC50 = 514 nM T49031 CV1P6X 56945245 IC50 = 92 nM T49031 CG2D5M 57149553 IC50 = 93 nM T49031 C3QG8L 59127842 IC50 = 1700 nM T49031 CLM1G5 60164712 IC50 > 30000 nM T49031 CGZ89B 65806958 IC50 = 24790 nM T49031 C82JTA 71305068 IC50 = 11600 nM T49031 CQD09I 71495550 Ki = 3744 nM T49031 CR38FB 71543331 Ki = 374.9 nM T49031 C2GAT5 71561597 IC50 = 1500 nM T49031 C62JWN 71561733 IC50 = 13000 nM T49031 CJ9AR2 71561735 IC50 = 5500 nM T49031 CXJP49 71561736 IC50 = 2800 nM T49031 CZ4I1N 71561866 IC50 = 10500 nM T49031 CHG65M 71561867 IC50 = 630 nM T49031 CA5T6O 71561868 IC50 = 2400 nM T49031 C2E9HV 71561869 IC50 = 480 nM T49031 C5FDT2 71561997 IC50 = 93 nM T49031 C2F0BJ 71561998 IC50 = 160 nM T49031 CSG26R 71561999 IC50 = 110 nM T49031 C45HOE 71562349 IC50 = 1200 nM T49031 CSDV65 71562351 IC50 = 1100 nM T49031 CKE98R 71625293 Ki = 101 nM T49031 CA95PY 71625294 Ki = 67 nM T49031 CVD0M7 71625412 Ki = 10.3 nM T49031 C6KP3Q 71625413 Ki = 10.8 nM T49031 CO9HD8 71625414 Ki = 11.4 nM T49031 CB7A3F 71625415 Ki = 10.6 nM T49031 CB24WG 71625416 Ki = 6 nM T49031 C6YL0H 71655218 IC50 = 38 nM T49031 CJ2B4Q 71655219 IC50 = 90 nM T49031 C58CEL 71655220 IC50 = 14 nM T49031 C4E2RB 71655221 IC50 = 5.7 nM T49031 C32PIH 71655289 IC50 = 35 nM T49031 C6BSW5 71655290 IC50 = 130 nM T49031 C19VOE 71655291 IC50 = 200 nM T49031 C6ZCI2 71655292 IC50 = 63 nM T49031 C7BIM2 71655353 IC50 = 29 nM T49031 CY78WU 71655354 IC50 = 230 nM T49031 C5H0IP 71655355 IC50 = 210 nM T49031 CW0Y5L 71655356 IC50 = 130 nM T49031 C8G6CQ 71655357 IC50 = 60 nM T49031 C2B4FJ 71655358 IC50 = 33 nM T49031 C1RYA4 71655419 IC50 = 300 nM T49031 C42YSR 71655420 IC50 = 57 nM T49031 CS3OP6 71655421 IC50 = 41 nM T49031 C7EW4B 71655422 IC50 = 47 nM T49031 C63MDL 71655423 IC50 = 30 nM T49031 CHCW60 71655482 IC50 = 28 nM T49031 C1Z7FJ 71655483 IC50 = 230 nM T49031 CZ0B7D 71655484 IC50 = 79 nM T49031 C75FOB 71655485 IC50 = 25 nM T49031 CQR98T 71655486 IC50 = 10 nM T49031 CM9U4L 71655547 IC50 = 77 nM T49031 CBMY45 71697266 Ki = 1620 nM T49031 CC1EV9 71697268 Ki = 260 nM T49031 CPW74Y 71697269 Ki = 800 nM T49031 CL0Q1G 71697270 Ki = 1450 nM T49031 CX1R7P 71697360 Ki = 300 nM T49031 C69BUX 71697361 Ki = 98 nM T49031 C2X5UT 71697363 Ki = 5900 nM T49031 C0UPY7 71697364 Ki = 440 nM T49031 C92HCM 71697365 Ki = 1340 nM T49031 CIPT74 71697366 Ki = 170 nM T49031 CJ52KP 71717087 Ki = 2.3 nM T49031 C7FLM2 72724741 IC50 = 50 nM T49031 CC65XM 72724804 IC50 = 28 nM T49031 C5IX8L 72724805 EC50 = 332 nM T49031 CK41SO 72724806 IC50 = 330 nM T49031 CR4A1Z 72724807 IC50 = 500 nM T49031 CJG3W2 73897219 IC50 = 63340 nM T49031 C0ER9W 74538726 IC50 = 5700 nM T49031 C1IN8Q 76310070 IC50 = 3380 nM T49031 CNYC80 76313773 IC50 = 1040 nM T49031 C0LU1D 76317291 IC50 = 900 nM T49031 C0U3XB 76317292 IC50 > 10000 nM T49031 CX6O8P 76317293 IC50 > 10000 nM T49031 CF8B7J 76320989 IC50 > 10000 nM T49031 CON57Y 76320990 IC50 > 10000 nM T49031 C3H2UI 76320991 Ki = 1100 nM T49031 CZO5L9 76320992 IC50 = 1660 nM T49031 C9P2HW 76320993 IC50 = 1650 nM T49031 CX5H3D 76320994 IC50 = 670 nM T49031 CP7R9O 76320995 IC50 = 1940 nM T49031 C1U5JY 76328224 IC50 = 1370 nM T49031 CN48JG 76328225 IC50 = 2190 nM T49031 CB89NY 76328226 IC50 = 800 nM T49031 CCF2T7 76328227 IC50 = 750 nM T49031 C4MAE1 76335476 IC50 = 580 nM T49031 CL30YE 76335477 IC50 = 2700 nM T49031 CG5E8R 76335478 IC50 > 10000 nM T49031 CV3S5J 76335479 IC50 = 1570 nM T49031 C4C2HT 76335480 IC50 = 1460 nM T49031 CQAL89 76335481 IC50 = 1660 nM T49031 CGY43C 78425867 IC50 = 2670 nM T49031 C0WA1V 86290925 Ki = 10260 nM T49031 C6FVI5 86302567 Ki = 560 nM T49031 C4T2MX 86302568 Ki = 330 nM T49031 CH1AU3 86302591 Ki = 1480 nM T49031 CNK78C 86302666 Ki = 0.14 nM T49031 CQLZ84 90381790 Ki = 39213 nM T49031 C0U9JN 90645047 Ki = 57 nM T49031 C9VK0E 90645048 Ki = 490 nM T49031 C8K2VQ 90645050 Ki = 85 nM T49031 CEN72L 90645051 Ki = 53 nM T49031 C4RAD1 90645052 Ki = 60 nM T49031 CJH69O 90645053 Ki = 4570 nM T49031 C54TGH 90645054 Ki = 80 nM T49031 C1EB8U 90645055 Ki = 2340 nM T49031 CFPT98 90655054 IC50 = 140 nM T49031 C5JZ8R 90655055 IC50 = 280 nM T49031 C3DWJ2 90655129 Ki = 8030 nM T49031 C5Z8EX 90655130 Ki = 10100 nM T49031 C6C2HX 90655131 Ki = 7670 nM T49031 C24PAH 90655132 Ki = 1450 nM T49031 CIXL21 90655133 Ki = 300 nM T49031 C2X7HV 90665951 IC50 > 1000 nM T49031 CRH4M3 90665952 IC50 > 1000 nM T49031 C5ZA4B 90665953 IC50 = 910 nM T49031 CPJ21F 90665954 IC50 = 50 nM T49031 C3KRH8 90665955 IC50 = 25 nM T49031 C1BA4E 90665956 IC50 = 12 nM T49031 CY80KV 90665957 IC50 = 8.4 nM T49031 CA48LV 90665958 IC50 = 5.4 nM T49031 CYB86O 90665959 IC50 = 22 nM T49031 CW8MS4 90665960 IC50 = 6.8 nM T49031 CQ67SO 90665961 IC50 = 4.8 nM T49031 CN94OJ 90665962 IC50 = 4.7 nM T49031 C2K9LZ 90665963 IC50 = 12 nM T49031 C81TAL 90665964 IC50 = 4 nM T49031 CP5S0X 90665965 IC50 = 3 nM T49031 C8IVK5 90665966 IC50 = 11 nM T49031 C7DL5F 90665967 IC50 = 3.7 nM T49031 C78ZBE 90665968 IC50 = 4 nM T49031 C2AG7C 90665969 IC50 = 3.9 nM T49031 C10CYW 90665970 IC50 = 1.1 nM T49031 CHBL08 90665971 IC50 = 940 nM T49031 CVZO36 90665972 IC50 = 22.6 nM T49031 C5EN3W 90665973 IC50 = 16 nM T49031 C62YEW 90665974 IC50 = 23 nM T49031 CF20ZD 90665975 IC50 = 160 nM T49031 CQE72G 90665976 IC50 = 7.3 nM T49031 CYF9H8 90665977 IC50 = 11.6 nM T49031 CJB32F 98103582 Ki = 17500 nM T49031 CG1IY3 98473743 Ki = 2350 nM T49031 C8NM0U 101553172 Ki = 2120 nM T49031 CG0N1O 101874275 IC50 = 16 nM T49031 CZX37E 102160215 IC50 = 14400 nM T49031 CVC0L7 102236951 IC50 = 93600 nM T49031 CXUQ14 102236952 IC50 = 31900 nM T49031 CHR18W 102579879 IC50 = 23600 nM T49031 C9C5OZ 117607839 IC50 = 782 nM T49031 C9BZ6E 117607841 IC50 = 185 nM T49031 CLHS74 117607901 IC50 = 926 nM T49031 CW9R0U 117607904 IC50 = 688 nM T49031 CKPU97 117607978 IC50 = 6630 nM T49031 C7QST8 117611788 IC50 = 6894 nM T49031 C2QDO6 117611839 IC50 = 54 nM T49031 CO1HJ9 117611880 IC50 = 18226 nM T49031 CZ6C1M 117611892 IC50 = 3620 nM T49031 C9YH1X 117611941 IC50 = 42468 nM T49031 C29AKS 118717990 IC50 = 0.38 nM T49031 CU4O3M 118718077 IC50 = 0.4 nM T49031 CS16DB 118718078 IC50 = 0.22 nM T49031 CK6E3L 118718085 IC50 = 0.34 nM T49031 CRZY67 118736272 IC50 = 290 nM T49031 CPY1S2 118736273 IC50 = 920 nM T49031 C2HWT3 118736382 IC50 = 17190 nM T49031 CY0VM1 118736383 IC50 = 12970 nM T49031 C6X0GY 118736384 IC50 = 13880 nM T49031 CS50HX 118736385 IC50 = 17310 nM T49031 C80ROJ 118736389 IC50 = 660 nM T49031 CIJ3E0 118736391 IC50 = 1630 nM T49031 CYO8P5 118736392 IC50 = 11730 nM T49031 C1DP4N 118899141 IC50 = 76000 nM T49031 CUH45I 118899149 IC50 = 78200 nM T49031 CA83ML 118899158 IC50 = 74870 nM T49031 C7YGZ8 122177663 IC50 = 360 nM T49031 CR80CE 122177664 IC50 = 930 nM T49031 CO0E6T 122189322 Ki = 3231 nM T49031 CG3U9I 122189323 Ki = 743.4 nM T49031 CM68CG 122189324 Ki = 7575 nM T49031 CWN52G 122189325 Ki = 906.2 nM T49031 CH08QC 122189326 Ki = 591.6 nM T49031 CSWG38 122189327 Ki = 951.9 nM T49031 C2ZJK1 122189328 Ki = 2113 nM T49031 CP7I6J 122189329 Ki = 963.1 nM T49031 CY7O0G 122189330 Ki = 1237 nM T49031 CO9E8A 122189331 Ki = 2347 nM T49031 CK7UV3 122189332 Ki = 1140 nM T49031 C8E7MQ 122189333 Ki = 1711 nM T49031 CI46QN 122189334 Ki = 949.8 nM T49031 CZ6LS4 122189335 Ki = 447 nM T49031 CZSI84 122189336 Ki = 385.2 nM T49031 C0OLW2 122204528 IC50 = 900 nM T49031 C90BKO 122520041 IC50 < 10 nM T49031 C3P0QD 122576697 IC50 = 220 nM T49031 C17FZG 127027248 IC50 = 26.24 nM T49031 C0DW3P 127027565 IC50 = 42.61 nM T49031 C6OVL9 127028490 IC50 = 49.5 nM T49031 CCF5E4 127028491 IC50 = 120.2 nM T49031 CV6JZ1 127028492 IC50 = 471 nM T49031 CO4D8I 127028814 IC50 = 24547089.16 nM T49031 C1Y9BP 127028815 IC50 = 3.34 nM T49031 CLB70K 127029400 IC50 = 8.32 nM T49031 C3FR6D 127029685 IC50 = 25.02 nM T49031 C6A1GD 127029686 IC50 = 4.6 nM T49031 CI6S1K 127030040 IC50 = 8.46 nM T49031 C4X7CO 127030041 IC50 = 2.34 nM T49031 C3LRH9 127030042 IC50 = 2.73 nM T49031 CAB69Z 127030043 IC50 = 16.4 nM T49031 CA50HP 127030044 IC50 = 114 nM T49031 C8DA4P 127030315 IC50 = 295120922.7 nM T49031 CQV32H 127030316 IC50 = 1.16 nM T49031 CI6P8J 127030317 IC50 = 1.15 nM T49031 CXQ69J 127030318 IC50 = 6.96 nM T49031 CQJ7F3 127030635 IC50 = 0.76 nM T49031 CZH53T 127030636 IC50 = 1.34 nM T49031 CO7WC6 127030637 IC50 = 2.46 nM T49031 CU0BJ3 127030638 IC50 = 862978547.8 nM T49031 C6Y2XQ 127031260 IC50 = 4.69 nM T49031 CJL9I1 127032443 IC50 = 1.02 nM T49031 CK3BX6 127032447 IC50 = 6.31 nM T49031 CI8RZ2 127032448 IC50 = 8.47 nM T49031 CV76UR 127032449 IC50 = 6.94 nM T49031 CVQ04L 127032450 IC50 = 4.82 nM T49031 CL36HN 127045979 IC50 = 26050 nM T49031 CI7H5T 127045980 IC50 = 23050 nM T49031 CIVH08 127045981 IC50 = 21540 nM T49031 C4ZG2O 127045982 IC50 = 16140 nM T49031 CWN9X5 127046160 IC50 = 14230 nM T49031 CUK8M7 127046161 IC50 = 13760 nM T49031 C4CAH2 127046162 IC50 = 13340 nM T49031 CDR54T 127047437 IC50 = 10250 nM T49031 CNL84P 127047438 IC50 = 17630 nM T49031 C3G7FU 127047439 IC50 = 9880 nM T49031 CED9T0 127047850 IC50 = 11860 nM T49031 C8QSW1 127048158 IC50 = 13800 nM T49031 CD51BP 127048159 IC50 > 25000 nM T49031 CP59LC 127048521 IC50 = 7800 nM T49031 CSLW65 127048522 IC50 > 25000 nM T49031 CADQ63 127048523 IC50 = 18700 nM T49031 C2A0UO 127048524 IC50 = 2300 nM T49031 CX65VA 127048525 IC50 = 21600 nM T49031 C5TS0O 127048526 IC50 > 25000 nM T49031 C3SY6Q 127049154 IC50 = 7600 nM T49031 CE5VT0 127049164 IC50 > 25000 nM T49031 CG9XP1 127049501 IC50 > 25000 nM T49031 CKYV35 127049817 IC50 > 25000 nM T49031 CVY2Q6 127049838 IC50 = 6300 nM T49031 CNX36Z 127049839 IC50 = 5600 nM T49031 COH67Z 127049840 IC50 = 9100 nM T49031 C1B4PE 127049841 IC50 = 5260 nM T49031 CJM29H 127049842 IC50 > 25000 nM T49031 CZIV95 127049843 IC50 = 15600 nM T49031 CDX7J4 127049844 IC50 = 5500 nM T49031 C3JE8G 127049845 IC50 = 6700 nM T49031 CEU1Y3 127050799 IC50 = 19200 nM T49031 CAS65J 127051646 IC50 = 8200 nM T49031 CLU6P9 127051647 IC50 > 25000 nM T49031 C9BFA0 127051648 IC50 > 25000 nM T49031 CMW2S6 127051649 IC50 > 25000 nM T49031 CE25WX 127051650 IC50 = 9900 nM T49031 C5REY7 127051651 IC50 > 25000 nM T49031 C4QXW2 127051652 IC50 > 25000 nM T49031 CL4N3G 127051653 IC50 = 8500 nM T49031 CFC43I 127052871 IC50 = 6100 nM T49031 C8AUE5 127053172 IC50 = 19900 nM T49031 C4YV1I 127053228 IC50 = 208929613.1 nM T49031 CPB1J8 127053229 IC50 = 3.21 nM T49031 CZR14W 127053267 IC50 = 4.18 nM T49031 CX53LM 127053268 IC50 = 1.12 nM T49031 CW3L9P 127053269 IC50 = 5.17 nM T49031 C6W2RO 127053272 IC50 = 524807460.3 nM T49031 C3AZ9G 127053273 IC50 = 5.24 nM T49031 CU8NW9 127053274 IC50 = 6.7 nM T49031 C4O6VG 127053280 IC50 = 162181009.7 nM T49031 C98AVC 127053285 IC50 = 1.26 nM T49031 CH2EP6 127053293 IC50 = 39 nM T49031 C3IVZ5 127053294 IC50 = 14.2 nM T49031 CDS47Y 127053295 IC50 = 17.2 nM T49031 CI2U8S 127053300 IC50 = 3.67 nM T49031 CQ6YW0 127053301 IC50 = 1.46 nM T49031 CT96PH 129047769 IC50 = 1140 nM T49031 CI24DQ 129047778 IC50 = 409 nM T49031 CI2J8F 129047830 IC50 = 110 nM T49031 C7BGS2 129047963 IC50 = 960 nM T49031 C4FRX1 132501288 IC50 = 26300 nM T49031 C34DQH 132501408 IC50 = 18500 nM T49031 CSP91A 132501468 IC50 = 5300 nM T49031 C1IFJ2 132501469 IC50 > 100000 nM T49031 CUT65O 132503175 IC50 = 370 nM T49031 CTQ8E6 132528967 IC50 = 2.4 nM T49031 CFB4V6 132528968 IC50 = 3 nM T49031 CM34ST 132528969 IC50 = 1.4 nM T49031 C5ZWQ8 132528970 IC50 = 4.3 nM T49031 C3WLQ2 134134387 IC50 = 15.7 nM T49031 CLM6F9 134134689 IC50 = 45.7 nM T49031 C5JS7V 134138393 IC50 = 669.9 nM T49031 CJ8ZN5 134139145 Ki = 420 nM T49031 C63QWU 134141164 IC50 = 16.9 nM T49031 C3EKC0 134142355 IC50 = 343.9 nM T49031 CEF0U1 134144291 IC50 = 601.4 nM T49031 CH9PI2 134146604 IC50 = 14.7 nM T49031 C8GH5D 134155148 IC50 = 152.9 nM T49031 C2Z5NM 134155499 Ki = 10980 nM T49031 C3K5UI 134155758 IC50 = 16.6 nM T49031 CH4XU1 134156052 IC50 = 23.7 nM T49031 C52IBY 134823859 IC50 = 394.2 nM T49031 C8VHK7 137632080 IC50 = 2710 nM T49031 CQO35X 137632519 IC50 = 2 nM T49031 CVSF43 137632662 IC50 = 25.7 nM T49031 C2NC9L 137633752 IC50 = 2180 nM T49031 CN78FJ 137633908 IC50 = 50 nM T49031 C08FKI 137634357 IC50 = 75 nM T49031 C3JI7B 137634520 IC50 = 5.5 nM T49031 CEJO70 137634807 IC50 = 510 nM T49031 CM3G2X 137635261 IC50 = 22160 nM T49031 CGPH59 137635270 IC50 > 1000 nM T49031 C40KOA 137635653 IC50 = 0.6 nM T49031 C64VSP 137636270 IC50 = 22290 nM T49031 C3H9XJ 137636488 IC50 = 41 nM T49031 CQP57Z 137636959 IC50 = 1 nM T49031 C3U2JC 137637883 IC50 > 50000 nM T49031 CW8D3F 137638026 IC50 = 197 nM T49031 C1HIY2 137638305 IC50 = 6.6 nM T49031 CNYU52 137639027 IC50 = 1.1 nM T49031 CZO8K2 137639142 IC50 = 5840 nM T49031 CNE56R 137639426 IC50 = 740 nM T49031 C0JQF2 137639470 IC50 = 39400 nM T49031 CG8V1S 137639601 IC50 = 3.8 nM T49031 CMK7O5 137639868 IC50 > 50000 nM T49031 CMSA73 137639962 IC50 = 260 nM T49031 C1KN9L 137640079 IC50 = 510 nM T49031 CVAK38 137640137 IC50 = 0.3 nM T49031 CB94IM 137640658 IC50 = 19600 nM T49031 CNVZ89 137640673 IC50 = 500 nM T49031 CIJ6E3 137640968 IC50 > 1000 nM T49031 C0B1FH 137641544 IC50 = 192.5 nM T49031 C6DF7U 137641807 IC50 > 1000 nM T49031 C0GWD7 137641958 IC50 = 10 nM T49031 CO1L4N 137642007 IC50 = 21.8 nM T49031 CH09CN 137642553 IC50 = 0.0002 nM T49031 C6DJF3 137642709 IC50 = 168 nM T49031 C3AEP5 137642951 IC50 = 99 nM T49031 CSXN16 137643018 IC50 = 44.25 nM T49031 CE0J4N 137643562 IC50 = 7 nM T49031 C0EY3T 137643629 IC50 = 2430 nM T49031 CB85DX 137643715 IC50 = 11.42 nM T49031 CJ6Z5F 137645427 IC50 > 1000 nM T49031 CL09KP 137645698 IC50 = 10 nM T49031 CEB8L5 137646135 IC50 > 50000 nM T49031 C5NF8R 137647268 IC50 = 90 nM T49031 CWOY74 137647871 IC50 = 1380 nM T49031 CC9R2E 137647922 IC50 = 2.6 nM T49031 C0KYZ2 137648206 IC50 = 237 nM T49031 CSF5N6 137648399 IC50 = 10.8 nM T49031 CNA75Z 137648431 IC50 = 8830 nM T49031 C7NYD8 137649498 IC50 > 1000 nM T49031 C19DEP 137649562 IC50 = 1360 nM T49031 C58EXC 137650165 IC50 = 200 nM T49031 CU9EK0 137650556 IC50 = 8.6 nM T49031 C7BUK5 137650655 IC50 = 12 nM T49031 CQ5AJ9 137650783 IC50 = 1.2 nM T49031 C7QW9D 137650914 IC50 = 57 nM T49031 C09QJA 137650983 IC50 = 1 nM T49031 C2NYK9 137651187 IC50 = 3 nM T49031 CCWZ51 137651207 IC50 = 20 nM T49031 CDQ41W 137651497 IC50 = 19.7 nM T49031 C04AZG 137651667 IC50 = 4 nM T49031 C57ZKC 137652515 IC50 = 182 nM T49031 C7R4DB 137653941 IC50 = 22 nM T49031 C8XLU1 137654027 IC50 = 29030 nM T49031 CGSU61 137654406 IC50 = 11.6 nM T49031 C2QMK8 137654413 IC50 = 40 nM T49031 CT08DG 137654519 IC50 = 1.5 nM T49031 CDAE50 137655349 IC50 = 23.17 nM T49031 CUC26W 137655738 IC50 = 20 nM T49031 CV8P6O 137656187 IC50 > 50000 nM T49031 CHV31Y 137656315 IC50 = 3570 nM T49031 CTA1F2 137656425 IC50 = 67 nM T49031 C90JMU 137656505 IC50 = 0.7 nM T49031 CSZ1A5 137657170 IC50 = 2.9 nM T49031 C1Y9RS 137657408 IC50 = 660 nM T49031 C5N2CB 137657727 IC50 > 1000 nM T49031 CNM6C4 137657944 IC50 > 1000 nM T49031 CJU5K7 137658335 IC50 = 110 nM T49031 CNFP69 137658811 IC50 = 2710 nM T49031 C3XE0H 137659182 IC50 = 0.9 nM T49031 CUFT31 137659572 IC50 = 17 nM T49031 CY6A3Q 137659779 IC50 = 18 nM T49031 C9CQ4N 137659903 IC50 = 25.93 nM T49031 CJQ6B7 137659959 IC50 = 3390 nM T49031 CY1S6E 137660489 IC50 = 24.58 nM T49031 C4BMO7 137660514 IC50 = 2 nM T49031 C8MH9V 137660779 IC50 = 18 nM T49031 CL1G7H 137661189 IC50 = 2.4 nM T49031 C01KBD 137661456 IC50 = 570 nM T49031 C1R9BC 137661627 IC50 = 13.3 nM T49031 CI96SM 137661745 IC50 = 1970 nM T49031 C1JH8K 138545006 IC50 > 100000 nM T49031 CLT78F 138545112 IC50 > 100000 nM T49031 C7DZ8K 138545235 IC50 > 100000 nM T49031 C5DJC6 138545265 IC50 = 10000 nM T49031 CIS28V 139209090 IC50 = 1412 nM T49031 CB46AI 139209092 IC50 > 100000 nM T49031 CMNL75 145960420 IC50 = 9.7 nM T49031 CL45BO 145960456 IC50 = 140000 nM T49031 C1W6TO 145960482 IC50 = 92 nM T49031 C0YF7Z 145960612 IC50 = 109 nM T49031 CU1EV5 145960693 IC50 = 126 nM T49031 C01WBE 145960929 IC50 = 335 nM T49031 C5G6LM 145961320 IC50 = 8900 nM T49031 C96AIF 145961391 IC50 > 100000 nM T49031 CI9QB0 145961558 IC50 = 210 nM T49031 CUIF27 145961566 IC50 = 10000 nM T49031 CQE07I 145961835 IC50 = 166 nM T49031 CI9JH6 145961877 IC50 = 6700 nM T49031 C3M4OD 145961898 IC50 = 18000 nM T49031 CBI7V1 145962019 IC50 = 27800 nM T49031 CN1I2C 145962168 IC50 = 69000 nM T49031 C8CSZ0 145962247 IC50 = 125000 nM T49031 CMD9X7 145962389 IC50 = 53 nM T49031 CVEF93 145962537 IC50 = 39000 nM T49031 C35NPT 145962676 IC50 = 192 nM T49031 C97URS 145962850 IC50 = 950 nM T49031 CVB9A4 145963178 IC50 = 36 nM T49031 CPA60M 145963188 IC50 = 65 nM T49031 CM95CN 145963260 IC50 = 155 nM T49031 CUL94O 145963403 IC50 = 275 nM T49031 COA19G 145963426 IC50 > 100000 nM T49031 C2LEB3 145963518 IC50 = 67000 nM T49031 CS6I8T 145964202 IC50 > 8000 nM T49031 CJ3Q5B 145964538 IC50 = 890 nM T49031 CKAS15 145964962 IC50 = 1100 nM T49031 CO83HL 145965095 IC50 > 8000 nM T49031 C15VCH 145966003 IC50 > 8000 nM T49031 C3L5IP 145966472 IC50 = 6300 nM T49031 C40QHP 145969617 IC50 > 8000 nM T49031 CV5NU9 145974241 IC50 = 2100 nM T49031 CQ42KP 145974420 IC50 > 8000 nM T49031 CRUD43 145974971 IC50 = 6100 nM T49031 CZ8H4Y 145975867 IC50 = 370 nM T49031 C38NRV 145976554 IC50 > 8000 nM T49031 CK2B4J 145978094 IC50 = 890 nM T49031 C9BWP4 145979302 IC50 = 2130 nM T49031 CN79HG 145979487 IC50 = 2800 nM T49031 CODE68 145979676 IC50 = 11.6 nM T49031 CEI3U1 145979850 IC50 = 4300 nM T49031 C24WEG 145980281 IC50 = 8.2 nM T49031 CIZU61 145980473 IC50 = 9.8 nM T49031 C35BOY 145980635 IC50 = 7.8 nM T49031 C69MQC 145980644 IC50 = 8.8 nM T49031 C07EJK 145980652 IC50 = 5.7 nM T49031 C5AYC4 145980811 IC50 = 64000 nM T49031 CG6UL0 145980995 IC50 = 1740 nM T49031 C2XPD3 145981337 IC50 = 2.7 nM T49031 C21VNK 145981642 IC50 = 22.8 nM T49031 CB67YT 145981691 IC50 = 1480 nM T49031 C41IRV 145981707 IC50 = 350 nM T49031 C5L8JM 145981943 IC50 = 12.9 nM T49031 CE94FB 145982013 IC50 = 7.7 nM T49031 C4UVP5 145982479 IC50 = 10.2 nM T49031 CLO3P1 145982669 IC50 = 74.86 nM T49031 C4B2NC 145982840 IC50 = 3.53 nM T49031 CL1F8N 145982922 IC50 = 28700 nM T49031 CGB54U 145983051 IC50 = 8.21 nM T49031 CQF0E2 145983505 IC50 = 4.16 nM T49031 CFE52X 145983530 IC50 = 27.75 nM T49031 C7SKN2 145983622 IC50 = 30.78 nM T49031 CG9LA8 145983719 IC50 = 5.89 nM T49031 C7WD8V 145983830 IC50 = 26.79 nM T49031 CSV4F0 145983965 IC50 = 20.44 nM T49031 C8WRQ7 145984091 IC50 = 21.17 nM T49031 C2UV4N 145984105 IC50 = 8.86 nM T49031 CPK4C5 145984357 IC50 = 4.82 nM T49031 C62OHN 145984529 IC50 = 5.26 nM T49031 CQ30LY 145984824 IC50 = 6.74 nM T49031 CF5R2L 145984944 IC50 = 3.22 nM T49031 CNZ16R 145985009 IC50 = 8.11 nM T49031 C16JLE 145985104 IC50 = 1.98 nM T49031 CVZ10A 145985697 IC50 = 42.79 nM T49031 C9G2VJ 145985757 IC50 = 387 nM T49031 C07VUG 145985780 IC50 = 2.31 nM T49031 C69VIS 145985988 IC50 = 593.7 nM T49031 CXBR78 145986043 IC50 = 12.89 nM T49031 C5X3GQ 145986425 IC50 = 6200 nM T49031 CRZE86 145986857 IC50 = 5100 nM T49031 CAJ5K8 145986961 IC50 = 3.6 nM T49031 CIB5Z9 145986993 IC50 = 5 nM T49031 CHWT73 145987085 IC50 = 6800 nM T49031 CM3H4F 145987197 IC50 = 2900 nM T49031 CNZ7R6 145987536 IC50 = 9200 nM T49031 CYBN31 145987734 IC50 = 835 nM T49031 C1EF3B 145988020 IC50 = 7.1 nM T49031 CM1U6F 145988104 IC50 = 15.9 nM T49031 CQIS01 145988427 IC50 = 6000 nM T49031 C4R3HC 145988596 IC50 = 7 nM T49031 CQ7W9S 145988601 IC50 = 13.2 nM T49031 CMW7U5 145989009 IC50 = 35.9 nM T49031 CN8K1E 145989337 IC50 = 3.1 nM T49031 CE16JH 145989568 IC50 = 113 nM T49031 CON2B3 145989641 IC50 = 7.7 nM T49031 CF3OZ9 145989730 IC50 = 18.7 nM T49031 CXG30R 145990249 IC50 = 11300 nM T49031 CWS03B 145991519 IC50 = 9.4 nM T49031 C8G1BT 145991875 IC50 = 10000 nM T49031 C8IL9E 145992200 IC50 = 5100 nM T49031 CBY18W 145992498 IC50 = 1400 nM T49031 CCU34H 145992780 IC50 = 360 nM T49031 C6GHQ9 145993211 IC50 = 22000 nM T49031 C2Q8BT 145993325 IC50 = 7.6 nM T49031 CVN3A5 145993374 IC50 = 6.6 nM T49031 CEVY70 145993649 IC50 = 880 nM T49031 CC24LD 145993770 IC50 = 19.7 nM T49031 CJO08K 145993925 IC50 = 125 nM T49031 C1UC2Z 147001460 IC50 = 77.1 nM T49031 CES1Y7 147009690 IC50 = 52.2 nM T49031 CYUM75 147335182 IC50 = 36.8 nM T49031 CSK1A5 147672609 IC50 = 4.6 nM T49031 CDX0I3 149045896 IC50 = 729 nM T49031 C1YFV0 155510465 IC50 < 10 nM T49031 CX74UV 155510547 IC50 < 10 nM T49031 C2AW9L 155510675 IC50 = 37 nM T49031 CLHB15 155510759 IC50 = 14 nM T49031 C4FH8S 155512766 IC50 = 48.3 nM T49031 C7J5BO 155512794 IC50 = 41.5 nM T49031 CZXI74 155513137 IC50 = 32 nM T49031 CL7I6A 155513548 IC50 = 30.8 nM T49031 C6IB7G 155513571 IC50 = 9 nM T49031 CY56QN 155514326 IC50 = 952 nM T49031 C5J0OF 155514653 IC50 = 253 nM T49031 C8E6ZX 155514792 IC50 = 1400 nM T49031 C0SDO2 155515259 IC50 = 230 nM T49031 CX76LO 155515463 IC50 = 34 nM T49031 CGW2M6 155516032 IC50 > 100000 nM T49031 C53ZEN 155516179 IC50 > 10000 nM T49031 CM3BV8 155516620 IC50 > 100000 nM T49031 CHU0Q9 155516696 IC50 = 111 nM T49031 C4VT1Y 155517101 IC50 = 430 nM T49031 C2BCH9 155517229 IC50 = 248 nM T49031 C6I7SU 155517529 IC50 = 154 nM T49031 CJ6ZU4 155517550 IC50 > 1000 nM T49031 CCB58J 155517652 IC50 = 481 nM T49031 CE95IQ 155518158 IC50 > 100000 nM T49031 CFQZ35 155518266 IC50 = 1410 nM T49031 CW8Z7I 155518578 IC50 = 8100 nM T49031 C5ATN1 155519023 IC50 = 232 nM T49031 C2OQU6 155519126 IC50 > 100000 nM T49031 CEF5D1 155519196 IC50 > 100000 nM T49031 C7FP0V 155519306 IC50 = 395 nM T49031 C5B4HU 155519323 IC50 = 14 nM T49031 CEJ56T 155519405 IC50 = 6700 nM T49031 CH9R4W 155520688 IC50 = 54 nM T49031 COL16B 155520712 IC50 = 8 nM T49031 C4WO3N 155521110 IC50 = 392 nM T49031 CNM0Q9 155521286 IC50 > 10000 nM T49031 CD4OH3 155521410 IC50 = 56 nM T49031 C0S4TP 155521499 IC50 = 30.6 nM T49031 CZKF54 155521690 IC50 = 1300 nM T49031 C8NOH2 155521815 IC50 = 6040 nM T49031 CJZT01 155522109 IC50 = 952 nM T49031 CTDK64 155522147 IC50 = 480 nM T49031 CN60CL 155522148 IC50 = 243 nM T49031 CB0WG8 155522381 IC50 = 2.1 nM T49031 C73DYM 155522560 IC50 = 5907 nM T49031 CQ3OD0 155522579 IC50 = 116 nM T49031 C8GNQ9 155522828 IC50 = 486 nM T49031 CM7ZA2 155523065 IC50 = 99 nM T49031 CW75YK 155523151 IC50 > 100000 nM T49031 CY3UP7 155523507 IC50 = 405 nM T49031 CL0IQ3 155523963 IC50 = 25.5 nM T49031 C94IEH 155524612 IC50 = 922 nM T49031 CZP1E6 155524975 IC50 = 30 nM T49031 CIP3E9 155526380 IC50 = 460 nM T49031 C5R3PX 155526504 Ki = 17 nM T49031 C78BVM 155526764 IC50 = 1130 nM T49031 CVJ70O 155526910 IC50 = 1561 nM T49031 CAC34Y 155527225 IC50 = 1800 nM T49031 COMG30 155527377 IC50 = 579 nM T49031 C6OC8R 155527614 IC50 = 836 nM T49031 CPHX68 155527880 IC50 = 1.5 nM T49031 CWZ17S 155528412 IC50 = 67 nM T49031 CROM71 155528428 IC50 = 436 nM T49031 C3PMD9 155529033 IC50 = 506 nM T49031 CW3G4Z 155529142 IC50 = 920 nM T49031 CCW71B 155529960 IC50 = 100 nM T49031 CYW5R1 155530452 IC50 > 100000 nM T49031 C2MW8Q 155530743 IC50 > 100000 nM T49031 CUP2B4 155531358 IC50 = 39 nM T49031 CIL2D0 155531506 IC50 = 51 nM T49031 CD84AS 155531896 IC50 = 40190 nM T49031 C9SH6Q 155532346 IC50 = 352 nM T49031 CLE8N1 155532865 IC50 = 660 nM T49031 CL9A0E 155532989 IC50 = 20.6 nM T49031 CK28QW 155533771 IC50 = 20 nM T49031 C2TR0X 155533978 IC50 = 50210 nM T49031 CEF08Q 155534115 IC50 > 100000 nM T49031 C9ODL6 155534328 IC50 = 968 nM T49031 CH9GO0 155534453 IC50 = 56.5 nM T49031 CG5E2L 155534840 IC50 = 16 nM T49031 C72EIY 155535051 IC50 = 89 nM T49031 C5G9LX 155535238 IC50 = 113 nM T49031 COZ5V6 155535430 IC50 = 46600 nM T49031 CT3A0N 155536062 IC50 = 14 nM T49031 C20BYW 155536148 Ki = 10.1 nM T49031 C9IL7E 155536781 IC50 = 38.8 nM T49031 C7O0SH 155537082 IC50 = 1111 nM T49031 CP7D4R 155537435 IC50 = 26.8 nM T49031 CCYI81 155537845 IC50 = 29370 nM T49031 C3EF7U 155538548 IC50 = 100 nM T49031 C2S5HL 155538665 IC50 = 52.1 nM T49031 C2NTI6 155538936 IC50 > 100000 nM T49031 CW5U4H 155539000 IC50 = 64.8 nM T49031 C6E1YP 155539344 IC50 > 100000 nM T49031 C69TOB 155539701 IC50 = 57 nM T49031 CLE9Y6 155539965 IC50 = 280 nM T49031 CT2V8E 155540850 IC50 = 4380 nM T49031 CTM03H 155540978 IC50 = 4726 nM T49031 C6RE8V 155540985 IC50 = 36.6 nM T49031 CQE43H 155541095 IC50 > 100000 nM T49031 C0T3CO 155541137 IC50 = 139.6 nM T49031 CNZ5B4 155541377 IC50 = 2000 nM T49031 C6OIY3 155541618 IC50 > 100000 nM T49031 C42XMS 155542291 IC50 = 3 nM T49031 C1K6NV 155542487 IC50 = 259 nM T49031 C41IBR 155542489 IC50 = 2200 nM T49031 CRU73P 155542979 Ki = 4.8 nM T49031 CHJY08 155543004 IC50 > 10000 nM T49031 CH92PY 155543085 IC50 = 1682 nM T49031 CH6X3Q 155543527 IC50 = 26 nM T49031 CTL46N 155543581 IC50 = 64 nM T49031 CB4K6P 155543584 IC50 = 274 nM T49031 C0EG5T 155543676 IC50 < 10 nM T49031 CR7WL1 155544072 IC50 = 35 nM T49031 C13HEG 155544089 IC50 > 10000 nM T49031 CH17XP 155544685 IC50 > 100000 nM T49031 C72ADE 155544797 IC50 = 162.2 nM T49031 CEC78A 155545362 IC50 > 1000 nM T49031 CB4J8F 155545830 IC50 = 162 nM T49031 C7YS2H 155546237 IC50 = 119 nM T49031 C3Q5GS 155546528 IC50 = 17 nM T49031 CV8T2E 155546596 IC50 = 269 nM T49031 C2R3FM 155546808 IC50 = 111.6 nM T49031 C0V4GT 155547050 IC50 = 2 nM T49031 CKY05M 155547055 IC50 = 37090 nM T49031 CBG9C3 155547430 IC50 = 98.2 nM T49031 CNS2J4 155548060 IC50 < 10 nM T49031 CQ0Z4K 155548281 IC50 = 35 nM T49031 C1LJ0G 155548285 IC50 = 257 nM T49031 CA8Z7D 155548324 IC50 = 9120 nM T49031 C8HVD1 155548349 IC50 > 100000 nM T49031 CZB82L 155548494 IC50 = 370 nM T49031 CC5H7R 155548878 IC50 > 100000 nM T49031 C8JC4L 155548940 IC50 = 50 nM T49031 CK4Q0J 155548955 IC50 = 3863 nM T49031 CX27NO 155549084 IC50 > 100000 nM T49031 CP7FQ0 155549178 IC50 > 1000 nM T49031 CIM5K2 155549227 IC50 = 39000 nM T49031 CH35KO 155550346 IC50 = 36 nM T49031 C12LPX 155551071 IC50 = 29 nM T49031 CRV20J 155551193 IC50 = 25 nM T49031 C6BZ4E 155551617 IC50 = 7 nM T49031 CCKN07 155551785 IC50 = 43.1 nM T49031 CX7P8L 155552184 IC50 = 853 nM T49031 CR7Q8D 155552542 IC50 = 2011 nM T49031 CH93MA 155553025 IC50 = 4.9 nM T49031 CBHM14 155553205 IC50 > 100000 nM T49031 C35NJC 155553210 IC50 = 45300 nM T49031 C2VBQ0 155553272 IC50 = 25 nM T49031 CK9FW3 155553273 IC50 = 60.7 nM T49031 CI15FC 155553565 IC50 = 8600 nM T49031 CVJ3E7 155553910 IC50 = 5000 nM T49031 C0DQC5 155554155 IC50 = 34.1 nM T49031 CDI56O 155554254 IC50 = 37.5 nM T49031 C1AIJ3 155554704 IC50 = 82070 nM T49031 C6YP0L 155554916 IC50 > 100000 nM T49031 C9GE3U 155554982 IC50 > 100000 nM T49031 C2IE7D 155555749 IC50 = 12430 nM T49031 CCI45A 155555926 IC50 = 361 nM T49031 C5SZB7 155556059 IC50 < 10 nM T49031 CJ0QX2 155556352 IC50 > 100000 nM T49031 CP58EH 155556856 IC50 = 26050 nM T49031 CW0K5V 155556875 IC50 < 10 nM T49031 CYJ92G 155557164 IC50 < 10 nM T49031 C6YSC7 155557266 IC50 < 10 nM T49031 C9M1NU 155557790 IC50 = 32 nM T49031 CXCF36 155558612 IC50 = 63 nM T49031 C0Z4ET 155558668 IC50 = 540 nM T49031 CK41QD 155558933 IC50 = 3.8 nM T49031 C5AQM2 155559051 IC50 < 10 nM T49031 CMH7V5 155559237 IC50 > 100000 nM T49031 CR3V7P 155559353 IC50 = 2.1 nM T49031 CT97AU 155559419 IC50 < 10 nM T49031 C7O2KR 155559420 IC50 = 638 nM T49031 CJ5UC9 155560661 IC50 = 33 nM T49031 C2GHS4 155561494 IC50 = 2.1 nM T49031 C98PWZ 155561783 IC50 = 1197 nM T49031 C5OM0U 155561976 IC50 = 12 nM T49031 CZJ52C 155562121 IC50 = 70450 nM T49031 CZXL78 155562443 IC50 = 530 nM T49031 CYB71Z 155563262 IC50 = 18 nM T49031 C2USA4 155563322 IC50 = 166 nM T49031 CZ3XY4 155563335 IC50 > 100000 nM T49031 C9CG3Y 155563835 IC50 = 189 nM T49031 C1UR9Y 155564187 IC50 = 118 nM T49031 CY83KQ 155564232 IC50 < 10 nM T49031 C3N8XZ 155564979 IC50 = 12030 nM T49031 C5YCE8 155565509 IC50 = 4 nM T49031 C0XSM3 155565602 IC50 = 44.9 nM T49031 CEAV80 155566012 IC50 = 5000 nM T49031 CV1L3T 155566407 IC50 > 10000 nM T49031 C7HP0L 155566550 IC50 = 770 nM T49031 CU53FD 155566562 IC50 = 49 nM T49031 CK87TX 155566958 IC50 = 21 nM T49031 C2T7GX 155567492 IC50 < 10 nM T49031 CT23WX 155567596 IC50 < 10 nM T49031 C5Z7YC 155567712 IC50 = 750 nM T49031 CG2KN0 155567727 IC50 > 100000 nM T49031 C7UPT8 155567911 IC50 = 127 nM T49031 CR1NB6 155568111 IC50 = 139 nM T49031 C63DVL 155568157 IC50 = 36.8 nM T49031 CIC1Q5 155568323 IC50 = 50.9 nM T49031 CV68GZ 155568757 IC50 = 1070 nM T49031 CUE8B1 155568787 IC50 = 205 nM T49031 C4ZV3Q 155568941 IC50 > 10000 nM T49031 C1I7QW 155568944 IC50 = 346 nM T49031 CL1QZ7 44583044 IC50 = 9 nM T49031 D00RIX 5280443 IC50 = 1800 nM T49031 D01NCW 11534772 IC50 = 460 nM T49031 D01UYI 5281607 IC50 = 4900 nM T49031 D05MDE 11505372 IC50 = 150000 nM T49031 D05VEV 11556056 IC50 = 120 nM T49031 D06NEB 11693148 IC50 = 35 nM T49031 D08AIJ 440735 IC50 = 14600 nM T49031 D09GZQ 11713852 IC50 = 1300 nM T49031 D09IMK 11621748 IC50 = 3.2 nM T49031 D0A5WN 11621347 IC50 = 2.1 nM T49031 D0B3US 11585523 IC50 = 3300 nM T49031 D0G3TK 5280863 IC50 = 10500 nM T49031 D0I0MU 11534625 IC50 = 69 nM T49031 D0K0KT 11621207 IC50 = 6.1 nM T49031 D0K4PY 114829 IC50 > 100000 nM T49031 D0M7BR 5280378 IC50 > 100000 nM T49031 D0Q4MO 23642227 IC50 = 150 nM T49031 D0QY3R 11513217 IC50 = 24 nM T49031 D0RB1V 6419835 IC50 = 124 nM T49031 D0RL4S 11714476 IC50 = 27 nM T49031 D0SY2M 5281708 IC50 > 100000 nM T49031 D0T3PW 5281672 IC50 = 10000 nM T49031 D0W3ON 416002 IC50 = 600 nM T49031 D0Y3TZ 370 IC50 = 7100000 nM T49031 D0Y6HD 90645049 Ki = 51 nM T00926 D0BP9C 193962 IC50 = 8500 nM T00926 D0K8KX 5280343 Ki = 2400 nM T00926 D0O3OS 104850 Ki = 1400 nM T00926 D0R0FE 2520 EC50 = 1925 nM T00926 D0R1RS 3715 IC50 = 12000 nM T00926 D0R3JB 4212 IC50 = 27.5 nM T00926 D0Z3DY 2333 Ki = 190 nM T00926 D02HTD 25167947 IC50 = 14900 nM T00926 D02QWY 24785538 IC50 = 36300 nM T00926 D0G7UX 5284373 EC50 = 1700 nM T00926 D0O2EF 56946615 IC50 > 100000 nM T00926 D0V7UQ 56946834 IC50 = 2500 nM T00926 D02VJY 3037617 IC50 = 5180 nM T00926 D07GTB 16760063 IC50 = 7570 nM T00926 C52MFS 1756 EC50 = 42000 nM T00926 C8C1JP 72343 IC50 = 38320 nM T00926 C5ZCH7 97332 IC50 = 26350 nM T00926 CL97OF 97548 IC50 = 9860 nM T00926 CA3NK8 193841 EC50 = 5100 nM T00926 CR67FB 243037 EC50 > 100000 nM T00926 CABJ72 276138 IC50 = 1760 nM T00926 CM70RQ 285815 IC50 = 16000 nM T00926 CN8ZL4 298546 EC50 = 45000 nM T00926 C7HME8 439246 Ki = 2400 nM T00926 COI2C9 560674 EC50 = 98000 nM T00926 CTF2J0 687260 EC50 > 100000 nM T00926 CH6MV7 715632 IC50 = 8770 nM T00926 C64RUF 877998 IC50 = 15900 nM T00926 CXR0P5 917533 IC50 = 8800 nM T00926 C7D1QN 921567 EC50 > 100000 nM T00926 CK8TP4 1019287 IC50 > 100000 nM T00926 CL27VW 1069464 IC50 = 3900 nM T00926 CXQ4P8 1183964 IC50 = 8130 nM T00926 CQT4J5 2094802 IC50 > 100000 nM T00926 C1A0FV 2298706 EC50 = 9800 nM T00926 CW6SA0 2787558 IC50 > 100000 nM T00926 C8PN0C 5280682 IC50 = 50000 nM T00926 CNI9X4 5281888 Ki = 600 nM T00926 CPHR19 5325373 EC50 > 100000 nM T00926 CJMT13 5325385 EC50 > 100000 nM T00926 C8VZ9T 5325386 EC50 > 100000 nM T00926 C81ZSW 5325387 EC50 = 85000 nM T00926 CTO51S 5352005 IC50 = 50000 nM T00926 CB2U6E 5467200 IC50 = 1100 nM T00926 C0EM5S 6509849 IC50 = 2800 nM T00926 C32UFI 9828452 IC50 = 61 nM T00926 C82UNW 9828532 IC50 = 1800 nM T00926 CI78PM 9848185 IC50 = 1050 nM T00926 C30DJS 9873998 IC50 = 800 nM T00926 CK5L6J 9904482 EC50 = 64000 nM T00926 CHI5S9 9975676 IC50 = 2900 nM T00926 CEG64W 9976758 EC50 = 2800 nM T00926 CDTB42 9979854 IC50 >= 250 nM T00926 CL5ZS9 9980860 IC50 = 650 nM T00926 C2B0CY 10004696 IC50 >= 250 nM T00926 CQI0Z7 10029563 IC50 = 76 nM T00926 C0HN4T 10031184 IC50 = 118 nM T00926 CG3RA9 10046544 IC50 = 1850 nM T00926 C5IQ2D 10047863 IC50 < 250 nM T00926 CK4A1L 10048669 IC50 = 1020 nM T00926 C2ZUK8 10051663 IC50 < 250 nM T00926 CC6U1G 10071405 IC50 >= 250 nM T00926 CSY05M 10072430 IC50 = 38 nM T00926 CO0QB1 10092403 IC50 = 7350 nM T00926 CWJ7R4 10094280 IC50 >= 250 nM T00926 CE6X4R 10221081 EC50 = 49100 nM T00926 C96LOC 10251349 IC50 > 50000 nM T00926 CQT7H4 10320818 IC50 = 65 nM T00926 C3I4DW 10322116 IC50 = 715 nM T00926 CY73KI 10322450 EC50 = 1800 nM T00926 CW6D4S 10333981 IC50 = 10800 nM T00926 CK9SQ7 10344755 IC50 = 533 nM T00926 CXG67L 10345205 IC50 = 500 nM T00926 C7Z4DU 10346312 IC50 >= 250 nM T00926 C7Z8IW 10379829 IC50 = 2870 nM T00926 CAO02N 10383921 IC50 = 789 nM T00926 CQU08N 10388318 IC50 >= 250 nM T00926 C36PIN 10407830 IC50 = 197 nM T00926 C1DYS4 10432300 IC50 = 920 nM T00926 CG40WP 10454772 IC50 = 910 nM T00926 CW4BK0 10455921 IC50 = 138 nM T00926 CE7IT1 10459316 IC50 >= 250 nM T00926 CCS90U 10472817 IC50 = 714 nM T00926 C78HZG 10495050 IC50 = 932 nM T00926 CE1U9A 10517005 EC50 > 100000 nM T00926 CCG5H3 10518339 IC50 = 14500 nM T00926 C8HWT1 10543161 IC50 = 2710 nM T00926 CD2EQ3 10585756 IC50 = 43100 nM T00926 CHE31J 10591449 IC50 > 100000 nM T00926 C58EFZ 10616146 IC50 = 4190 nM T00926 CH1V7U 10708375 IC50 = 20400 nM T00926 C7ANU6 10709061 IC50 = 8290 nM T00926 CH72SE 10709378 IC50 = 18300 nM T00926 CSK86O 10756523 IC50 = 2560 nM T00926 C01KTG 10758537 IC50 = 5970 nM T00926 CQF21J 10776189 IC50 = 26400 nM T00926 CI1RC8 10830017 IC50 = 4060 nM T00926 COHV95 10848828 IC50 = 4460 nM T00926 C53AIX 10850200 IC50 = 43400 nM T00926 C2BXZ1 11156535 IC50 >= 250 nM T00926 CKJ32I 11164648 IC50 = 6350 nM T00926 C5E8LY 11168500 IC50 = 20 nM T00926 C84PJK 11177283 IC50 = 94 nM T00926 C8HF7R 11177641 IC50 = 399 nM T00926 CYQ98P 11179994 IC50 = 138 nM T00926 CN3B9L 11186582 IC50 = 9000 nM T00926 CTBH70 11189272 IC50 = 2800 nM T00926 C8CWV4 11200621 IC50 = 632 nM T00926 C6XUE4 11201011 IC50 = 33 nM T00926 CLT87I 11212921 IC50 = 41 nM T00926 CFD6R7 11213871 IC50 = 48 nM T00926 CD8VO1 11214464 IC50 = 15 nM T00926 C63QRZ 11226516 IC50 = 17 nM T00926 C7PTZ8 11246811 IC50 >= 250 nM T00926 C79PBA 11247947 IC50 = 59 nM T00926 C86MWN 11249529 IC50 = 13.7 nM T00926 COJD26 11258566 IC50 = 2300 nM T00926 CEN76W 11261262 IC50 = 40.9 nM T00926 CI1M9O 11270541 IC50 = 28 nM T00926 CP13GR 11270563 IC50 = 59 nM T00926 C8NL3A 11281999 IC50 = 3440 nM T00926 C4I2ZV 11293873 IC50 = 2710 nM T00926 CY79US 11293906 IC50 = 110 nM T00926 CFX64S 11293909 IC50 = 166 nM T00926 CH7E1O 11293927 IC50 = 147 nM T00926 C1YH6T 11295806 IC50 = 97 nM T00926 CJYA49 11304370 IC50 = 24 nM T00926 CXKY42 11305058 IC50 = 45 nM T00926 CD9SN8 11316308 IC50 = 167 nM T00926 CE4HY2 11318194 IC50 = 88 nM T00926 CL8ZT6 11327691 IC50 = 3150 nM T00926 CY8G5H 11337594 IC50 >= 250 nM T00926 C78BGT 11339085 IC50 = 169 nM T00926 C65ZTX 11350733 IC50 = 820 nM T00926 C8P1QC 11351150 IC50 >= 250 nM T00926 CYZ51K 11359019 IC50 = 8370 nM T00926 C61ARN 11362459 IC50 = 1415 nM T00926 C31PLX 11376266 IC50 = 29 nM T00926 CZ9W0I 11385818 IC50 = 78 nM T00926 C8S3OV 11396606 IC50 = 87 nM T00926 C0G4AF 11408751 IC50 = 120 nM T00926 C13MRQ 11418752 IC50 = 955 nM T00926 CUO79V 11419244 IC50 = 63 nM T00926 C49LBJ 11432257 IC50 = 620 nM T00926 CTK09U 11443156 IC50 = 13 nM T00926 CLB97A 11443942 IC50 = 26.5 nM T00926 CM2J9W 11444700 IC50 < 250 nM T00926 CSK8F9 11453657 IC50 = 190 nM T00926 C19WQH 11454150 IC50 >= 250 nM T00926 CTQS76 11454703 IC50 = 10 nM T00926 C59DBU 11454819 IC50 < 250 nM T00926 CYCB17 11455462 IC50 = 107 nM T00926 C6W0MU 11477947 IC50 = 122 nM T00926 CH0T1B 11488138 IC50 = 27 nM T00926 CJXT34 11751643 IC50 = 67 nM T00926 CXWU95 11752839 IC50 < 250 nM T00926 C9X6DU 11774980 IC50 = 51 nM T00926 CLR59J 11775287 IC50 = 62 nM T00926 C2C3WI 11957988 IC50 > 20000 nM T00926 CG1CU7 12219475 EC50 > 100000 nM T00926 CS4D6C 12405466 EC50 = 15100 nM T00926 C4D7RX 12613559 EC50 = 26500 nM T00926 C6UJA5 13144102 EC50 > 100000 nM T00926 CT0DU8 13633111 IC50 = 20400 nM T00926 CO9ES2 13633119 IC50 = 1210 nM T00926 CJ9Z4M 15290116 EC50 = 72000 nM T00926 CLD92G 15999199 IC50 = 40600 nM T00926 C0A3IV 16092354 IC50 = 3730 nM T00926 CMVW98 16618023 EC50 = 728 nM T00926 CX06NR 17412108 IC50 = 39300 nM T00926 CB7T2K 20963109 IC50 = 7720 nM T00926 CFI13S 22310708 IC50 = 7820 nM T00926 CK4UG1 23323164 IC50 > 100000 nM T00926 C3ESV6 24178402 EC50 = 2800 nM T00926 C60EJI 25113688 EC50 = 9300 nM T00926 C6O2ZR 25225119 EC50 = 2700 nM T00926 C3J8PO 39176758 IC50 > 100000 nM T00926 CG7UZ6 44220872 IC50 = 12300 nM T00926 C8C9MJ 44220873 IC50 = 42600 nM T00926 CSLJ20 44220874 IC50 = 5380 nM T00926 CPIM70 44220875 IC50 = 21600 nM T00926 C01FMP 44220876 IC50 = 16200 nM T00926 C04ZKP 44220877 IC50 = 18300 nM T00926 CY9AW0 44221092 IC50 = 11600 nM T00926 C0X8OT 44221093 IC50 = 4510 nM T00926 C12MDG 44221095 IC50 = 14300 nM T00926 C3MNS1 44221096 IC50 = 27500 nM T00926 C2VWE1 44221097 IC50 = 1230 nM T00926 C9BNA1 44248179 EC50 = 73 nM T00926 CKA6N2 44276937 IC50 = 122 nM T00926 CTOA75 44368818 IC50 = 2020 nM T00926 CPLV23 44368900 IC50 > 10000 nM T00926 C26MFU 44368902 IC50 = 7600 nM T00926 CHO6P8 44368923 IC50 = 400 nM T00926 COWL28 44369026 IC50 = 1330 nM T00926 CDLX46 44369027 IC50 = 1560 nM T00926 C9VXD2 44369028 IC50 = 3840 nM T00926 CT0SK1 44369032 IC50 = 36000 nM T00926 CCD76W 44369044 IC50 = 37000 nM T00926 C1V6QO 44369052 IC50 = 900 nM T00926 CY08UQ 44369067 IC50 = 1000 nM T00926 C0FXA2 44369069 IC50 = 18570 nM T00926 C82JKC 44369082 IC50 = 1500 nM T00926 C0Z4TJ 44369087 IC50 = 15100 nM T00926 CZD46M 44369091 IC50 = 6350 nM T00926 CLIY42 44369110 IC50 = 1000 nM T00926 CTE65O 44369198 IC50 = 7200 nM T00926 C1J6DA 44369228 IC50 = 4500 nM T00926 CKPW47 44369229 IC50 = 3200 nM T00926 CA0PF4 44369232 IC50 > 100000 nM T00926 CU9H3K 44369247 IC50 = 39000 nM T00926 C05EUO 44369260 IC50 = 3330 nM T00926 CGU9Z8 44369264 IC50 = 2910 nM T00926 C5JLT0 44369265 IC50 = 2800 nM T00926 CE32OY 44369278 IC50 = 10000 nM T00926 C40XPZ 44404554 IC50 >= 250 nM T00926 CU97QG 44404555 IC50 < 250 nM T00926 CHX57V 44404558 IC50 < 250 nM T00926 C89BQU 44405535 EC50 = 420 nM T00926 CLV54W 44405572 EC50 = 250 nM T00926 C8A7CS 44405716 EC50 = 640 nM T00926 CM8O3W 44451264 EC50 > 100000 nM T00926 C45VCM 44451857 EC50 = 21000 nM T00926 CG61YX 44542293 EC50 > 100000 nM T00926 CI9VZ6 44542743 EC50 > 100000 nM T00926 C80EVI 44723582 EC50 > 100000 nM T00926 C43FNG 45266957 IC50 = 4180 nM T00926 C8C4ZS 45267881 IC50 = 22800 nM T00926 C8IYJ2 45268774 IC50 = 198000 nM T00926 CUE5Y2 45269621 IC50 = 29100 nM T00926 CJG13Y 45272176 IC50 = 24000 nM T00926 CAPW24 45272182 IC50 = 20700 nM T00926 COA30H 46227751 IC50 > 20000 nM T00926 CLWR13 46227752 IC50 > 20000 nM T00926 CX2EU1 46843551 EC50 = 13000 nM T00926 CON7Q5 46888534 EC50 = 46000 nM T00926 C53NLD 46888535 EC50 = 7610 nM T00926 CWO79T 46899560 EC50 = 12000 nM T00926 CUFI19 46899561 EC50 = 8700 nM T00926 C43WPR 46899562 EC50 = 8000 nM T00926 C2QX3P 46899563 EC50 = 63000 nM T00926 CBWT20 46899565 EC50 = 13600 nM T00926 CHR49C 46899724 EC50 > 100000 nM T00926 CZXN91 46899725 EC50 = 85800 nM T00926 C7ZS6E 46899726 EC50 = 29500 nM T00926 C1H9ML 56764960 IC50 = 22700 nM T00926 C2WYN9 56945196 IC50 > 100000 nM T00926 C7RW8P 56945197 IC50 = 11200 nM T00926 C7LDX6 56945198 IC50 > 100000 nM T00926 C2N8DS 56945199 IC50 > 100000 nM T00926 CN2WF6 56945201 IC50 > 100000 nM T00926 CB7W4E 56945202 IC50 > 100000 nM T00926 CT4BW6 56945299 IC50 > 100000 nM T00926 CTEJ21 56945300 IC50 = 45800 nM T00926 CU2HC7 56945301 IC50 = 40600 nM T00926 CUK5Q9 56945302 IC50 = 38800 nM T00926 C36HTV 56945303 IC50 = 46600 nM T00926 C7X2EU 56945304 IC50 = 44500 nM T00926 C4VNX9 56945305 IC50 = 16300 nM T00926 C1JCB9 56945418 IC50 = 44000 nM T00926 C6UD7F 56945419 IC50 = 32200 nM T00926 C98UJH 56945420 IC50 = 8000 nM T00926 C51PRX 56945421 IC50 = 22000 nM T00926 CES25H 56945422 IC50 = 9500 nM T00926 C2QB4L 56945423 IC50 = 7700 nM T00926 CA6UX7 56945524 IC50 = 74500 nM T00926 C4AVC1 56945525 IC50 = 40600 nM T00926 CC25LY 56945526 IC50 = 75800 nM T00926 C8KLW6 56945527 IC50 = 37900 nM T00926 C6ZSA3 56945528 IC50 = 30000 nM T00926 C2IAL8 56945529 IC50 = 28000 nM T00926 CP6G0O 56945530 IC50 > 100000 nM T00926 C27RQI 56946614 IC50 > 100000 nM T00926 CK1ZU5 56946616 IC50 = 23600 nM T00926 C73GCK 56946617 IC50 > 100000 nM T00926 CL8Z0F 56946723 IC50 = 23300 nM T00926 CIQ64Z 56946724 IC50 = 17200 nM T00926 CXMK07 56946726 IC50 > 100000 nM T00926 CRY4C6 56946727 IC50 = 80000 nM T00926 CV29FO 56946728 IC50 > 100000 nM T00926 CI69QT 56946831 IC50 > 100000 nM T00926 CDPU29 56946832 IC50 > 100000 nM T00926 C69ELZ 56946833 IC50 = 6100 nM T00926 CH7M4O 56946835 IC50 > 100000 nM T00926 CP1VK5 56951135 IC50 > 200000 nM T00926 C1XCE9 57393400 IC50 > 100000 nM T00926 CJXP74 71061793 EC50 > 100000 nM T00926 CA2N0L 71062020 EC50 = 31800 nM T00926 C0QGU2 71062093 EC50 = 33200 nM T00926 C5T0NL 71454923 IC50 = 11180 nM T00926 C4ZD2W 71492590 IC50 = 418 nM T00926 C0P6IG 71492759 IC50 = 434 nM T00926 CV9QS7 71524587 EC50 > 100000 nM T00926 C7JIG6 71524588 EC50 > 100000 nM T00926 C1EY6B 71524589 EC50 = 14700 nM T00926 C4LPZ3 71524590 EC50 = 3200 nM T00926 C60ZQJ 71524591 EC50 = 8800 nM T00926 CGV8F5 71525288 EC50 > 100000 nM T00926 CO9ZJ3 71560809 EC50 > 100000 nM T00926 C0E6OM 71560810 EC50 > 100000 nM T00926 C3T8ZF 71560811 EC50 > 100000 nM T00926 CFN89Y 71560812 EC50 > 100000 nM T00926 C42SMF 71560938 EC50 > 100000 nM T00926 C98LPJ 71560939 EC50 > 100000 nM T00926 CG8DU1 71618156 EC50 > 100000 nM T00926 C0Z3PN 71682039 EC50 > 100000 nM T00926 CV5Z9M 71682040 EC50 > 100000 nM T00926 C1IZT7 71682041 EC50 > 100000 nM T00926 COV12T 71682195 EC50 > 100000 nM T00926 C3Y4FW 71682196 EC50 > 100000 nM T00926 CLF3I8 71682197 EC50 > 100000 nM T00926 CN6Q3L 71696716 EC50 = 113 nM T00926 CQCF98 71724480 EC50 = 151 nM T00926 C1PR7Z 71724504 EC50 = 140 nM T00926 CA7K8Z 71724506 EC50 = 217 nM T00926 CD9KH7 71724532 EC50 = 250 nM T00926 CWR2L5 71724556 EC50 = 220 nM T00926 C4ODQ2 71724557 EC50 = 425 nM T00926 C7T0UM 71724558 EC50 > 1000 nM T00926 CUL9E2 71724582 EC50 = 238.3 nM T00926 CNW68B 71724606 EC50 = 616.7 nM T00926 CCZ9B3 71724628 EC50 = 230 nM T00926 C48CAR 72735227 IC50 = 14090 nM T00926 CQ5NB6 72950792 IC50 = 21800 nM T00926 CF57OZ 73346145 IC50 = 19000 nM T00926 CK3EX6 73355255 IC50 = 27500 nM T00926 C7NTB0 73356802 IC50 = 15100 nM T00926 CRB93S 89784681 EC50 = 301.7 nM T00926 CG71EX 89784708 EC50 = 175 nM T00926 C4ZOX6 89784717 EC50 = 670 nM T00926 C0ZQO6 89784722 EC50 = 171 nM T00926 C4U5CZ 89784733 EC50 = 208 nM T00926 CW17YB 89784735 EC50 = 272 nM T00926 C0VD4P 89784742 EC50 = 114 nM T00926 CZT7B9 89784751 EC50 = 135 nM T00926 CH70XJ 89784752 EC50 = 193 nM T00926 C6MRA2 89784753 EC50 = 87 nM T00926 C1JH4L 89784756 EC50 = 243.3 nM T00926 CN1RD8 89784760 EC50 = 333.3 nM T00926 C2YB6Q 89784818 EC50 = 137 nM T00926 CSK8X6 89784827 EC50 = 233.3 nM T00926 CENX80 89785043 EC50 = 103 nM T00926 CY46QV 89785047 EC50 = 172.3 nM T00926 CQL7T6 89785059 EC50 = 99 nM T00926 CENR59 89785064 EC50 = 263 nM T00926 CVZG56 89785117 EC50 = 78 nM T00926 CT43OU 89785127 EC50 = 133.8 nM T00926 C3FB6Q 89785132 EC50 = 219 nM T00926 C4S9WG 89785146 EC50 = 650 nM T00926 CCE95J 89785148 EC50 = 184 nM T00926 C9SBA1 89785178 EC50 = 246.7 nM T00926 CSI51G 89785190 EC50 = 225 nM T00926 CGB2P5 89785210 EC50 = 276.3 nM T00926 CTY1H5 89785238 EC50 = 155 nM T00926 CHGX10 89785254 EC50 = 292.7 nM T00926 CB1FR2 89794901 EC50 = 441.7 nM T00926 C43AXK 89795130 EC50 = 750 nM T00926 C70LJV 89795278 EC50 > 1000 nM T00926 CFU4W2 89795305 EC50 = 760 nM T00926 CVB23M 89795326 EC50 = 245 nM T00926 CX1W9Z 89795330 EC50 = 165 nM T00926 C7XG4U 89795333 EC50 = 950 nM T00926 C7W1TP 89795335 EC50 = 475 nM T00926 CAX9S0 89795337 EC50 = 457.5 nM T00926 COB3Z9 89795340 EC50 = 180 nM T00926 C6BW0Q 89795341 EC50 = 137.7 nM T00926 CUHC90 90469229 EC50 = 11900 nM T00926 C05JQB 90469230 EC50 = 7000 nM T00926 C41EMT 90469289 EC50 = 3900 nM T00926 CA1VH0 90469291 EC50 = 12400 nM T00926 C4NX2Q 90469293 EC50 = 6600 nM T00926 C0NW8T 90469355 EC50 = 5200 nM T00926 C8BRG2 101876951 EC50 = 1100 nM T00926 C0H9DF 101891699 EC50 = 23000 nM T00926 CXHQ89 102340685 IC50 = 4280 nM T00926 CJ7VI3 102340686 IC50 = 6260 nM T00926 CS1P5K 102340687 IC50 = 3380 nM T00926 C93SXK 102340688 IC50 > 100000 nM T00926 C86WSC 117777746 EC50 = 255 nM T00926 C9E0BT 117777811 EC50 = 135 nM T00926 C9YPJ7 117803128 EC50 = 579 nM T00926 C5GUV9 118708511 IC50 = 5800 nM T00926 CQLK93 118708512 IC50 > 100000 nM T00926 C5F8LY 118708513 IC50 = 13600 nM T00926 CL8H6M 118708514 IC50 > 100000 nM T00926 CCT4I2 118708515 IC50 > 100000 nM T00926 C7GI8W 118708516 IC50 > 100000 nM T00926 CE7Q3U 118708517 IC50 > 100000 nM T00926 C31MGA 118708518 IC50 > 100000 nM T00926 CKV6P1 118708519 IC50 > 100000 nM T00926 C1MJ4N 118708520 IC50 > 100000 nM T00926 C7WFJ3 118708521 IC50 = 2200 nM T00926 CVK89G 118708522 IC50 > 100000 nM T00926 C7G3ZV 118708523 IC50 = 94500 nM T00926 CG8S9M 118708524 IC50 = 15800 nM T00926 C9T4KE 118708525 IC50 = 11100 nM T00926 CG3LK4 118708526 IC50 = 8130 nM T00926 C42ETW 118708527 IC50 = 23600 nM T00926 C0OQ9P 118716252 EC50 = 41400 nM T00926 C3VRT8 118716258 EC50 = 5200 nM T00926 C4Z2DS 118719365 EC50 = 10000 nM T00926 CU6EP1 122179376 IC50 = 322 nM T00926 CIL20J 122179390 IC50 = 142 nM T00926 C0OUW1 122179391 IC50 = 141 nM T00926 CCE46L 126587406 EC50 > 1000 nM T00926 CZG92F 127028059 IC50 = 11300 nM T00926 CSR0Y7 127028060 IC50 > 100000 nM T00926 C8Z2XI 127028354 IC50 = 19800 nM T00926 C8Q9DG 127028355 IC50 = 20800 nM T00926 CRI72H 127028356 IC50 = 22700 nM T00926 C58QBI 127028357 IC50 > 100000 nM T00926 C6AIP3 127028358 IC50 > 100000 nM T00926 CG46ES 127028359 IC50 = 30100 nM T00926 CRP9U1 127028361 IC50 = 53300 nM T00926 CUC9I4 127040367 IC50 = 18500 nM T00926 C0I9VF 127040368 IC50 = 5500 nM T00926 CX9JE1 127040369 IC50 = 8300 nM T00926 CRM9W5 127040370 IC50 = 1800 nM T00926 CJY60W 127042304 IC50 = 58300 nM T00926 CO2P8K 127042305 IC50 = 26700 nM T00926 C56HDS 127042306 IC50 = 8300 nM T00926 CRI0X9 127042307 IC50 > 100000 nM T00926 CK4J8D 127042801 IC50 = 7300 nM T00926 C87PMI 127042802 IC50 = 13200 nM T00926 CRQ7U8 127042918 IC50 = 10900 nM T00926 CDL84X 127042919 IC50 > 100000 nM T00926 C39PWZ 127042920 IC50 = 38000 nM T00926 C21DSU 127042921 IC50 = 6800 nM T00926 C6UZ7C 127042922 IC50 > 100000 nM T00926 CSBM31 127042943 IC50 = 12100 nM T00926 C12BJD 127042944 IC50 = 18800 nM T00926 CZBJ54 127048170 IC50 = 1010 nM T00926 CO93BJ 127048171 IC50 = 8980 nM T00926 C6L0AF 127049502 IC50 = 636 nM T00926 CK1SN3 127049508 IC50 = 1070 nM T00926 CB9EV4 127049509 IC50 = 2500 nM T00926 C7PF5I 127050480 IC50 = 623 nM T00926 C59EXD 127050481 IC50 = 876 nM T00926 CUO40Y 127050796 IC50 = 910 nM T00926 C7MJ5X 127050797 IC50 = 586 nM T00926 CT6A2G 127050798 IC50 = 2360 nM T00926 C6V7JZ 127051981 IC50 = 418 nM T00926 C4P0LG 127051982 IC50 = 821 nM T00926 C5CX0B 127051983 IC50 = 200 nM T00926 CBQL62 127051984 IC50 = 340 nM T00926 C0FOG1 127051985 IC50 = 866 nM T00926 C1VP2D 127052887 IC50 = 9410 nM T00926 CG9TE5 127052888 IC50 = 643 nM T00926 CA7N9R 127052889 IC50 = 981 nM T00926 C6ZK3C 135449697 EC50 > 100000 nM T00926 CD2NR8 136110930 IC50 = 95000 nM T00926 C1EB8Q 136236384 EC50 > 100000 nM T00926 CI0KU2 137643961 IC50 = 15900 nM T00926 CHCB46 145956407 IC50 = 44200 nM T00926 C1F4LH 145971569 IC50 > 1000 nM T00926 CK61NI 145973976 IC50 > 1000 nM T00926 CF8L7A 145979103 EC50 = 298 nM T00926 C3EX7W 145979504 EC50 = 170 nM T00926 C4G7LT 145980033 EC50 = 95 nM T00926 C26OWY 145981942 EC50 = 156 nM T00926 C13VFZ 145985646 EC50 = 53 nM T00926 C4A1LN 145985882 EC50 = 38000 nM T00926 CI38SJ 145987174 EC50 = 28900 nM T00926 CFU24J 145987833 EC50 = 103 nM T00926 CGL02K 145988126 EC50 = 205 nM T00926 CX3YR7 145990226 EC50 = 200 nM T00926 CZRB08 145990960 EC50 = 62000 nM T00926 CN1V8K 145992500 EC50 = 208 nM T00926 CT02XU 145992768 EC50 = 121 nM T00926 CKZA78 145992770 IC50 = 12500 nM T00926 C07OTB 145993028 EC50 = 111 nM T00926 C65JUT 145993130 EC50 > 1000 nM T00926 C3UC5J 145994097 EC50 = 207.3 nM T00926 CKM79V 145994277 EC50 = 155.8 nM T00926 C5VRT4 155511477 IC50 > 100000 nM T00926 C1L0WJ 155511549 IC50 = 20000 nM T00926 CE4C1X 155512695 IC50 = 5800 nM T00926 C0AFT8 155514623 EC50 > 1000 nM T00926 CH6O3X 155515825 EC50 = 5080 nM T00926 CV9TF6 155516191 EC50 > 1000 nM T00926 C4IS7E 155518051 EC50 = 2200 nM T00926 CLQO05 155518383 IC50 = 9680 nM T00926 CA1BD2 155520579 EC50 = 12700 nM T00926 C8WFN9 155522227 IC50 > 100000 nM T00926 C8V3OE 155522345 IC50 > 100000 nM T00926 CQK86M 155522385 IC50 > 100000 nM T00926 CS18PU 155523410 EC50 = 5600 nM T00926 CN6ST7 155523417 EC50 > 1000 nM T00926 C86ZPR 155525910 EC50 = 4400 nM T00926 C8TQ4G 155526547 EC50 > 1000 nM T00926 C9BGT5 155528240 EC50 > 1000 nM T00926 C75OQS 155529248 IC50 = 2980 nM T00926 C3O4FR 155529325 IC50 > 100000 nM T00926 C56AHP 155530068 EC50 = 181.4 nM T00926 C9F3YI 155530680 IC50 = 44000 nM T00926 C6I0LU 155531567 IC50 = 18000 nM T00926 CUL2G4 155531672 EC50 > 1000 nM T00926 CJ5X8R 155532908 IC50 = 322 nM T00926 C4IW9M 155533366 EC50 = 5800 nM T00926 C9QT4A 155533532 IC50 = 85100 nM T00926 CHF7A6 155535686 EC50 > 1000 nM T00926 C28CPM 155536187 IC50 = 3600 nM T00926 CQC9E5 155536529 IC50 > 100000 nM T00926 CGM43D 155536878 IC50 = 40000 nM T00926 CYG84N 155537154 EC50 = 7300 nM T00926 C2J7TM 155537461 IC50 = 17300 nM T00926 CGD47O 155537584 EC50 > 1000 nM T00926 CNS83Y 155538210 IC50 = 33000 nM T00926 CVES34 155538494 EC50 = 1900 nM T00926 CLU37N 155539307 EC50 = 3000 nM T00926 CXN6C4 155539538 IC50 = 31000 nM T00926 CL6QG0 155542981 IC50 = 73000 nM T00926 C7JUC3 155543680 EC50 = 4500 nM T00926 C1HI5E 155550141 IC50 > 100000 nM T00926 CB8FC1 155550293 EC50 = 3500 nM T00926 C8B3LI 155551011 IC50 = 3700 nM T00926 CX43TI 155551742 IC50 = 41000 nM T00926 CIF4T8 155553306 EC50 > 1000 nM T00926 CEZ7B1 155554618 EC50 = 137 nM T00926 CX6CM0 155554919 EC50 = 530 nM T00926 CU9P0W 155555392 IC50 = 18000 nM T00926 C7JI4C 155555932 EC50 = 348.3 nM T00926 C27XQN 155558615 EC50 = 212 nM T00926 C8ATZ5 155558917 IC50 = 53000 nM T00926 CUNV65 155558919 EC50 > 1000 nM T00926 CFRS42 155559312 IC50 > 100000 nM T00926 CG6NC7 155560071 EC50 = 10100 nM T00926 CE6C4X 155562808 IC50 > 100000 nM T00926 CWM67C 155563340 EC50 = 2800 nM T00926 C6Z2XK 155566234 EC50 = 3700 nM T00926 CO1LU7 155567143 EC50 > 1000 nM T00926 C7KFG6 155567619 EC50 = 3900 nM T00926 CTV5K3 155568177 EC50 > 1000 nM T00926 C03SJY 155568508 EC50 = 139.3 nM T00926 CTXV81 155568869 EC50 > 1000 nM T00926 C0K1HQ 155569340 IC50 = 12900 nM T00926 D00RFY 5281612 IC50 = 3000 nM T00926 D00RIX 5280443 Ki = 2400 nM T00926 D01FGM 5280666 IC50 = 3000 nM T00926 D07NAY 5281692 Ki = 5000 nM T00926 D0G3TK 5280863 Ki = 2400 nM T00926 D0I7GE 11790 IC50 = 11300 nM T00926 D0T3PW 5281672 Ki = 2400 nM T17967 D03GFC 16741245 EC50 = 80 nM T17967 CHGI09 6597 IC50 = 9000000 nM T17967 CMC1D0 12892 Ki = 176 nM T17967 C6NQ9Y 1116656 IC50 = 3800 nM T17967 CHK89E 6102763 IC50 = 2000 nM T17967 C19DIZ 7178516 EC50 = 5200 nM T17967 CI5FC0 7178544 EC50 = 3800 nM T17967 CG7X9S 7178546 EC50 = 1100 nM T17967 CC28SV 16414363 IC50 = 10900 nM T17967 CHK6P1 16424570 IC50 = 5200 nM T17967 CKQY13 28361735 IC50 = 10500 nM T17967 C28NIL 29255080 IC50 = 1500 nM T17967 C80ODY 67932020 Ki = 1070 nM T17967 CXIN84 72376511 IC50 = 570 nM T17967 CELO13 72376512 EC50 = 456 nM T17967 C47XUW 86280454 IC50 = 65 nM T17967 CI7HO1 97281116 IC50 = 2500 nM T17967 CK6QG0 117972799 IC50 = 206 nM T17967 CUE2B5 118155888 IC50 = 1177 nM T17967 C2SA5C 118155890 IC50 = 416 nM T17967 C5CJ3D 118155894 IC50 = 154 nM T17967 C5Y8GW 118155895 IC50 = 432 nM T17967 C75WOG 118155906 IC50 = 195 nM T17967 C2OW7X 118155909 IC50 = 1196 nM T17967 C4QI2B 124201642 Ki = 2170 nM T17967 CRHZ85 124390110 IC50 = 7.8 nM T17967 C3FC0O 126200721 IC50 = 5900 nM T17967 C0VN5E 134561057 IC50 = 580 nM T17967 C46MPX 134561154 IC50 = 72 nM T17967 CKQ63N 134561155 IC50 = 58 nM T17967 C5X0YD 134561193 IC50 = 1514 nM T17967 CMQ04B 134561196 IC50 = 156 nM T17967 C30MTB 134561301 IC50 = 357 nM T17967 CHME32 134561302 IC50 = 67 nM T17967 C7WTU8 134561303 IC50 = 221 nM T17967 CR3V2E 134561305 IC50 = 65 nM T17967 CO3V2F 134561468 IC50 = 767 nM T17967 C8W3YG 136087021 IC50 = 1126 nM T17967 C0BUJ9 136249185 IC50 = 2600 nM T17967 CMO6K1 137636150 IC50 = 1657 nM T17967 CKU8P4 137638606 IC50 = 629 nM T17967 CAP1D8 137641886 IC50 = 1610 nM T17967 CS3KF0 137642154 Ki = 150 nM T17967 C7KIS8 137645507 IC50 = 1346 nM T17967 CSA49E 137646868 IC50 = 91 nM T17967 CI5TH3 137653481 Ki = 702 nM T17967 C7RB8J 137653507 Ki = 1330 nM T17967 C5XEM7 137655013 IC50 = 565 nM T17967 C0AZR8 137656816 IC50 = 68 nM T17967 C3SV7G 137659540 Ki = 1278 nM T17967 C9LP0W 137660248 IC50 = 4371 nM T17967 CHQ86U 149832647 IC50 = 140 nM T17967 CL6T4P 149986651 IC50 = 10 nM T17967 C24DWX 150179460 IC50 = 302 nM T17967 C7BM5V 150226583 IC50 = 126 nM T17967 CDO4W3 150362366 IC50 = 373 nM T17967 CJ17UR 150426809 IC50 = 18 nM T17967 CMS4L6 150703157 IC50 = 1620 nM T17967 C7J0AF 150821022 IC50 = 772 nM T17967 C1Z5DA 151004457 IC50 = 98 nM T17967 C02NBO 151026196 IC50 = 133 nM T17967 C0Q9PK 151406722 IC50 = 193 nM T17967 CY8OK4 151698036 IC50 = 110 nM T17967 C2RVC3 151777753 IC50 = 252 nM T17967 CKR2T1 151835909 IC50 = 113 nM T17967 CTI5R1 151961601 IC50 = 1455 nM T17967 CC3ME1 152131905 IC50 = 8 nM T17967 CAR6N3 152143591 IC50 = 132 nM T17967 C79SKI 152618834 IC50 = 184 nM T17967 C49BFR 155510663 IC50 = 2040 nM T17967 COH17B 155516961 IC50 > 10000 nM T17967 CRK41X 155523490 IC50 = 2660 nM T17967 C8K4NL 155527038 IC50 = 9910 nM T17967 CCG7K6 155528322 IC50 = 64 nM T17967 CNY40T 155534218 IC50 = 1960 nM T17967 CM20ZB 155534260 IC50 = 503 nM T17967 C8EH6M 155538895 IC50 = 95 nM T17967 C7BTJ9 155554053 IC50 = 8590 nM T17967 CA18GY 155563372 IC50 = 1660 nM T17967 C6Y5IM 155567964 IC50 = 7220 nM T89565 CV7IN2 104934 Ki = 210 nM T89565 C1KR5B 5327301 Ki = 98000 nM T89565 C37TKL 5327302 Ki = 12000 nM T89565 C64ZMN 5327304 Ki = 22000 nM T89565 C3IZ2W 5327307 Ki = 23000 nM T89565 C16DTL 5327308 Ki = 24000 nM T89565 C4O3QY 5327309 Ki = 63000 nM T89565 C3GUM7 5327310 Ki = 36000 nM T89565 CLAC59 9828058 Ki = 81 nM T89565 CDX7A4 10963183 Ki = 32000 nM T89565 CDT9G3 11467504 IC50 = 0.81 nM T89565 CJ57OA 14585243 Ki = 47 nM T89565 C8D5TB 44364680 Ki = 11000 nM T89565 C86ORE 44459987 IC50 = 13489.63 nM T89565 CDY2W5 49796910 IC50 = 0.2 nM T89565 CGY3W2 71471109 IC50 > 100000 nM T89565 CANH70 71716242 IC50 = 35200 nM T89565 C40WIR 71718085 IC50 = 750 nM T89565 CU75VK 71719897 IC50 = 19500 nM T89565 CBV6F1 71720507 IC50 = 560 nM T89565 CWM2E8 133081971 IC50 = 2980 nM T89565 CID3N6 134134572 Ki = 48 nM T89565 CV0R3B 134135432 Ki = 24 nM T89565 C3D7LQ 134136688 Ki = 59 nM T89565 CBY95D 134138690 Ki = 41 nM T89565 CG3EI1 134145896 Ki = 34 nM T89565 CI9X3K 134147411 Ki = 16 nM T89565 CP16IA 134148745 Ki = 111 nM T89565 CPE90G 134149983 Ki = 34 nM T89565 CBE39C 134151245 Ki = 135 nM T89565 CY0LD4 134152014 Ki = 59 nM T89565 C3K5HR 134153309 Ki = 28 nM T89565 CWQT79 134156687 Ki = 99 nM T89565 D0Y5IQ 44255320 IC50 = 5000 nM T50269 D00KHM 16362 EC50 = 1700 nM T50269 D01AZG 5073 EC50 = 320 nM T50269 D03YGR 156419 EC50 = 320 nM T50269 D09GDD 11167602 EC50 = 1800 nM T50269 D0A9YA 6918296 EC50 = 330 nM T50269 D0GQ7K 4046 EC50 = 2500 nM T50269 D0JC9N 60164 EC50 = 1300 nM T50269 D0K5WS 5280795 EC50 = 400 nM T50269 D0M8AB 750 EC50 = 94000 nM T50269 D0N6RF 65999 EC50 = 3200 nM T50269 D0P1FO 16078 EC50 = 1300 nM T50269 D0U5FS 3396 EC50 = 1200 nM T50269 D0Z5IU 1548887 EC50 = 380 nM T50269 D0Y2HR 2247 EC50 = 4200 nM T50269 C3O9AG 439709 EC50 = 12589.25 nM T50269 C8HZF2 783663 IC50 = 76 nM T50269 C9H1CE 5390854 EC50 = 590 nM T50269 C4SWU6 6324617 IC50 = 1700 nM T50269 C3W8ZK 17758335 IC50 > 100000 nM T50269 CH9J0Y 24846186 Ki = 67 nM T50269 COX8D7 44408895 IC50 > 100000 nM T50269 CR6CE1 44408940 IC50 > 100000 nM T50269 COY01R 44420834 IC50 = 3162.28 nM T50269 CE30WA 44420835 IC50 = 7400 nM T50269 C0DIM8 44420839 IC50 > 100000 nM T50269 CYE94N 44420840 IC50 > 100000 nM T50269 C59CNH 44420842 IC50 > 100000 nM T50269 C6N3DU 44420843 IC50 > 100000 nM T50269 C6Q1OE 44420847 IC50 > 100000 nM T50269 CKHC34 44420848 IC50 > 100000 nM T50269 C52YKX 44420851 IC50 > 100000 nM T50269 C23CLN 44420852 IC50 > 100000 nM T50269 C2NF6H 44420854 IC50 > 100000 nM T50269 CW2TL6 44420856 IC50 > 100000 nM T50269 C3XV2H 44420857 IC50 > 100000 nM T50269 CG30DJ 44420862 IC50 > 100000 nM T50269 C3AYZ8 44420865 IC50 > 100000 nM T50269 CVS4Z1 44420866 IC50 > 100000 nM T50269 CKG6M0 44420867 IC50 > 100000 nM T50269 CCB95G 44420868 IC50 > 100000 nM T50269 CYX7A3 44420870 IC50 > 100000 nM T50269 COH12C 44420871 IC50 > 100000 nM T50269 C9X7JH 44420872 IC50 > 100000 nM T50269 CR8HG1 44420875 IC50 > 100000 nM T50269 C19QZY 44420876 IC50 > 100000 nM T50269 CSZ5F4 44420878 IC50 = 2400 nM T50269 C6ZG0M 44420879 IC50 > 100000 nM T50269 C3IU8N 44420880 IC50 > 100000 nM T50269 CW80SJ 44420881 IC50 = 3981.07 nM T50269 CV8C2B 44420885 IC50 = 7943.28 nM T50269 CPBM16 44420891 IC50 = 3162.28 nM T50269 CYG93V 44427853 IC50 > 100000 nM T50269 C3C2OK 44427854 IC50 > 100000 nM T50269 C8Y9FW 44427856 IC50 > 100000 nM T50269 C19LSU 44427858 IC50 > 100000 nM T50269 C1FY4M 44427860 IC50 > 100000 nM T50269 CC2BE1 44427862 IC50 > 100000 nM T50269 CW95BM 44427864 IC50 > 100000 nM T50269 C3XJ4Z 44427866 IC50 > 100000 nM T50269 C84GXL 44427868 IC50 > 100000 nM T50269 C8CPX2 44427870 IC50 > 100000 nM T50269 CS17TJ 44427872 IC50 > 100000 nM T50269 CDL67C 44427876 IC50 > 100000 nM T50269 C9B6ER 44427877 IC50 > 100000 nM T50269 C15UHM 44427879 IC50 > 100000 nM T50269 CCAV10 44427881 IC50 > 100000 nM T50269 CXRV71 44427883 IC50 > 100000 nM T50269 CKX81C 44427885 IC50 > 100000 nM T50269 CG71DA 54467154 IC50 = 6900 nM T50269 C6DQT3 71450923 IC50 = 501.19 nM T50269 C2HUL4 90659973 IC50 > 100000 nM T50269 CO9ZU7 99118914 Ki = 40 nM T50269 CFW2V1 118195533 EC50 = 0.0012 nM T50269 CHM30C 118195560 EC50 = 0.06 nM T50269 C3HMN2 118195567 EC50 = 0.43 nM T50269 C8DSH5 118195581 EC50 = 0.00016 nM T50269 CKDM68 123133764 EC50 = 32 nM T50269 CPV2O3 132547348 EC50 = 327 nM T50269 CTN47D 135753560 IC50 = 8800 nM T50269 C8H3QG 135753564 IC50 > 200000 nM T50269 CLE71N 137631631 IC50 = 109 nM T50269 CL2X3J 137631882 IC50 = 690 nM T50269 C4L8SF 137635401 IC50 = 260 nM T50269 C1YE3F 137637510 IC50 = 720 nM T50269 CS41FM 137639832 IC50 = 4590 nM T50269 CKR79P 137644791 IC50 = 165.96 nM T50269 CVL25O 137645081 IC50 = 245.47 nM T50269 C3DZ4I 137650620 IC50 = 49 nM T50269 CDP0F7 137654599 IC50 = 220 nM T50269 C5QN0I 137655067 IC50 = 380.19 nM T50269 CU8FI4 137656578 IC50 = 75 nM T50269 CF1C3T 137657339 IC50 = 51.29 nM T50269 CRZY05 155519552 Ki = 741 nM T50269 CF27SE 155541454 Ki = 91 nM T50269 D04IEW 9909368 IC50 = 1900 nM T50269 D0H0BD 441071 Ki = 23 nM T50269 D0M4ZK 44420890 IC50 = 5011.87 nM T50269 D0X3TL 44420886 IC50 = 6200 nM T67710 D02CII 76943386 EC50 = 0.02 nM T67710 D03NHS 76283707 EC50 = 4100 nM T67710 CA6P1K 11963968 Ki = 0.912 nM T67710 CA4WI0 12001598 Ki = 707.95 nM T67710 CNF70V 16220269 IC50 = 68000 nM T67710 CH3KU5 23626097 Ki = 2818.38 nM T67710 CF1V4U 23626240 Ki = 3388.44 nM T67710 C5K7RJ 23626241 Ki = 562.34 nM T67710 C7O1ZX 23626243 Ki = 676.08 nM T67710 CS2FX3 23626399 Ki = 288.4 nM T67710 C0ZIC4 23626400 Ki = 154.88 nM T67710 CSI39A 23626402 Ki = 70.79 nM T67710 C0XE1Q 23626403 Ki = 3.802 nM T67710 CUTB14 23626557 Ki = 13.18 nM T67710 C5TJF3 23626558 Ki = 50.12 nM T67710 C0LNV5 23626559 Ki = 20.42 nM T67710 C27CIX 23626560 Ki = 6.761 nM T67710 CXU8E9 23626561 Ki = 3.548 nM T67710 C7JG9E 23626730 Ki = 1.445 nM T67710 C5N9AK 23626731 Ki = 1.82 nM T67710 CF8X4T 23626732 Ki = 6.761 nM T67710 C3B8PO 23626733 Ki = 616.6 nM T67710 CF4NW8 23626734 Ki = 8.71 nM T67710 CVO15W 23626891 Ki = 6.607 nM T67710 CB3D4J 23626894 Ki = 83.18 nM T67710 CU75YI 25118026 IC50 = 9400 nM T67710 CC9G1A 44270419 EC50 = 7.9 nM T67710 CS9AC3 44270511 EC50 = 4.4 nM T67710 C02OVQ 44270512 EC50 = 5.5 nM T67710 CC1OX8 44270513 EC50 = 9.1 nM T67710 CN3D6A 44428088 Ki < 100000 nM T67710 CPY82C 44428090 Ki = 933.25 nM T67710 CRS3H8 44428091 Ki = 380.19 nM T67710 C4FXJ3 44428092 Ki = 112.2 nM T67710 CN6WS7 44584917 EC50 = 32 nM T67710 CH14QN 44584920 EC50 = 13 nM T67710 CJR45V 44584921 EC50 = 0.06 nM T67710 CXSB17 44584922 EC50 = 0.15 nM T67710 CQS1U6 45485585 EC50 > 10000 nM T67710 C5XME6 49838154 EC50 > 1000000 nM T67710 C09VXY 49840922 EC50 = 1122 nM T67710 CPX2V6 49841000 EC50 = 0.2 nM T67710 CU3J0E 50908590 EC50 = 2.4 nM T67710 C24IPZ 56841901 EC50 = 0.07 nM T67710 C6Y8QI 66815925 EC50 > 1000000 nM T67710 CM8BP9 66817107 EC50 = 26000 nM T67710 C6IP4J 66817215 EC50 = 32000 nM T67710 CVCF27 66817553 EC50 = 33000 nM T67710 CAX82O 66817788 EC50 = 12000 nM T67710 C6CM8L 76283959 EC50 = 3600 nM T67710 C4WM1Z 137631923 EC50 = 19 nM T67710 C9XVZ4 137634846 EC50 = 0.51 nM T67710 CHV35B 137634885 EC50 = 0.26 nM T67710 CWA3V8 137635204 EC50 = 1.12 nM T67710 CIN0J6 137635394 EC50 = 0.08 nM T67710 CB64NJ 137636149 EC50 = 0.15 nM T67710 CP59IE 137636311 EC50 = 0.51 nM T67710 C7KQ9X 137637857 EC50 = 0.29 nM T67710 C6ZXO0 137637950 EC50 = 3 nM T67710 CLW1R3 137639371 EC50 = 14.57 nM T67710 CUZP78 137639372 EC50 = 0.13 nM T67710 C7O9IM 137639587 EC50 = 18.69 nM T67710 C05BRV 137640122 EC50 = 0.52 nM T67710 CT9B3U 137640833 EC50 = 0.34 nM T67710 C1O3FE 137641949 EC50 = 0.4 nM T67710 CSY1M3 137642287 EC50 = 0.14 nM T67710 C93LST 137642401 EC50 = 4.98 nM T67710 C3V6MW 137642849 EC50 = 0.12 nM T67710 C12BTY 137643019 EC50 = 0.34 nM T67710 CDR83Q 137643296 EC50 = 1.8 nM T67710 CQIU59 137645140 EC50 = 0.71 nM T67710 C71AOQ 137650056 EC50 = 11.51 nM T67710 C89VPB 137651582 EC50 = 0.18 nM T67710 C4A9EI 137652688 EC50 = 9.74 nM T67710 CL41NK 137654722 EC50 = 0.36 nM T67710 CV6G8Y 137657562 EC50 = 1.84 nM T67710 CRNM53 137657563 EC50 = 167 nM T67710 C79QHV 137657564 EC50 = 0.44 nM T67710 CN6V0J 137657565 EC50 = 0.83 nM T67710 CE0J2B 137657566 EC50 = 0.79 nM T67710 CQ8J3B 137657687 EC50 = 0.32 nM T67710 C5Q7KC 137657688 EC50 = 0.65 nM T67710 C38QDU 137657689 EC50 = 4.13 nM T67710 C5PM6C 137659455 EC50 = 0.48 nM T67710 CE5MN9 137659482 EC50 = 0.06 nM T67710 C3BK4S 137659489 EC50 = 2.59 nM T67710 C0ZJN1 137659716 EC50 = 0.17 nM T67710 C4TH5F 137660321 EC50 = 9.84 nM T67710 C8WFK3 137660410 EC50 = 0.27 nM T67710 CCT8K0 139035050 IC50 = 90 nM T67710 CDXQ89 145964425 EC50 = 67000 nM T67710 C60ZAH 145975286 EC50 = 50000 nM T67710 C9MJG6 145975813 EC50 > 1000000 nM T67710 CL3X2U 155513348 EC50 = 4600 nM T67710 C26GUZ 155518374 IC50 = 6800 nM T67710 CXZ5W0 155521869 IC50 > 100000 nM T67710 CB7Z3X 155522420 IC50 = 3500 nM T67710 CX2TS6 155522839 IC50 = 7600 nM T67710 CN5D9T 155526572 IC50 = 6100 nM T67710 C8LAP0 155529306 IC50 > 100000 nM T67710 CAE4T8 155533095 EC50 = 3600 nM T67710 CKW9P0 155536792 EC50 = 2.5 nM T67710 CTQ9U5 155536860 IC50 = 14000 nM T67710 C2I0PA 155540108 IC50 = 14000 nM T67710 CHM51V 155542161 EC50 = 5300 nM T67710 C2BHW9 155543526 IC50 = 38000 nM T67710 CGT23X 155546261 IC50 = 730 nM T67710 C59QIA 155547998 IC50 = 2300 nM T67710 C38KWY 155550447 IC50 = 4100 nM T67710 CGS61H 155551285 IC50 = 44000 nM T67710 CQ7ZP6 155553639 EC50 = 4600 nM T67710 C65GPR 155553648 EC50 > 100000 nM T67710 C6GAF5 155555773 IC50 = 4000 nM T67710 CFNP14 155557308 IC50 = 45000 nM T67710 CHDB02 155558265 IC50 = 23000 nM T67710 CGVN45 155559611 IC50 = 180 nM T67710 CTQ3H1 155560902 IC50 = 16000 nM T67710 C4DQ3V 155567876 EC50 > 100000 nM T68698 D0H1OL 135398635 Ki = 1472000 nM T68698 D0I7BL 65269 Ki = 110 nM T68698 D0I7TN 23190 IC50 = 4000 nM T68698 D0R2QS 72968 IC50 = 0.004 ug.mL-1 T68698 CY1P2C 72501 Ki = 4 nM T68698 CRG3J6 73651 Ki = 12 nM T68698 CI8KD2 97627 Ki = 410 nM T68698 C2CG8M 98567 Ki = 1930 nM T68698 CGF69C 99920 Ki = 3.3 nM T68698 C3BU7T 147104 Ki = 110 nM T68698 CHT80Q 275945 Ki = 22000 nM T68698 C8I2PG 358177 IC50 = 31 nM T68698 C3J5VD 402194 IC50 < 20000 nM T68698 CRU2Q9 443234 Ki = 39 nM T68698 CVQW71 451935 IC50 = 1000 nM T68698 C72EKO 469184 IC50 = 7600 nM T68698 CY0ZN2 472632 IC50 = 0.2 ug.mL-1 T68698 CA2U7Y 472655 IC50 > 10 ug.mL-1 T68698 C67BXW 481083 IC50 > 10 ug.mL-1 T68698 CJL5D2 489877 IC50 = 0.87 ug.mL-1 T68698 CLRY91 489878 IC50 = 3760 nM T68698 CLO12U 490351 Ki = 41 nM T68698 CJ2L8F 490432 IC50 = 123000 nM T68698 C5L8GI 490433 IC50 = 76000 nM T68698 CE9J3U 501516 Ki = 5020 nM T68698 C58AMW 501517 Ki = 27 nM T68698 CHNA61 501518 Ki = 586 nM T68698 C12AIT 501519 Ki = 22 nM T68698 C8T0YV 501520 Ki = 67600 nM T68698 CB4HR1 512554 IC50 > 10 ug.mL-1 T68698 CKIL63 512555 IC50 = 195 nM T68698 CTF70X 512656 IC50 > 10 ug.mL-1 T68698 CL24RG 512657 IC50 > 10 ug.mL-1 T68698 C1AU9I 512658 IC50 > 10 ug.mL-1 T68698 CL74IO 1362195 Ki = 1700 nM T68698 C13DGU 5358592 IC50 = 40 nM T68698 COLD86 6439007 Ki = 330 nM T68698 CX58IU 6450949 Ki = 125 nM T68698 CSB29R 6474190 IC50 = 90700 nM T68698 CW7NE1 6476927 IC50 = 8 nM T68698 CZR3N8 9816781 IC50 = 75020 nM T68698 CB01OK 9840103 Ki = 16000 nM T68698 CRAI41 9993207 Ki = 7900 nM T68698 C2SKW5 9997450 Ki = 134 nM T68698 CW21OU 10015023 IC50 = 7670 nM T68698 C3DI6E 10061387 Ki = 39 nM T68698 C4VB3K 10243225 Ki = 8800 nM T68698 CHG3J9 10400519 Ki = 273 nM T68698 C2FV5L 10422910 IC50 = 18 nM T68698 CNR64H 10655770 IC50 = 930 nM T68698 CR6A7V 11380460 IC50 = 12680 nM T68698 CJ8QH3 11537088 Ki = 17000 nM T68698 CV0F5A 11564784 Ki = 500 nM T68698 CTMK84 11615884 IC50 > 100000 nM T68698 CXEG94 11777524 Ki = 4500 nM T68698 C2RE5C 11779405 Ki = 110 nM T68698 CX35EZ 12097487 IC50 = 36460 nM T68698 C6IX0V 12769724 IC50 = 100000 nM T68698 C4SD3B 13712019 IC50 = 28000 nM T68698 CEC2K8 13939857 Ki = 35 nM T68698 CW0E2J 14134370 Ki = 160 nM T68698 CU06ED 14134371 IC50 = 1230 nM T68698 CB35KG 14134372 Ki = 200 nM T68698 C45LBI 14134395 IC50 = 950 nM T68698 CF9SO7 14134396 Ki = 200 nM T68698 CPJ92T 14134397 Ki = 170 nM T68698 C5YGX9 14134400 Ki = 90 nM T68698 CYGP51 14134401 Ki = 166 nM T68698 CCF8Z2 14134506 IC50 = 80 nM T68698 CFRL70 16075366 IC50 = 180 nM T68698 CZ03BO 21152084 Ki = 43400 nM T68698 CY07FB 25244925 Ki = 2600 nM T68698 C97ZIN 44189703 IC50 = 1.5 nM T68698 CL4K0U 44278585 Ki = 0.5 nM T68698 CYP2V1 44373339 IC50 > 100000 nM T68698 CS4NG1 44396071 IC50 > 100000 nM T68698 C7ZMI0 44396095 IC50 > 100000 nM T68698 C6BN5P 44396175 IC50 = 97270 nM T68698 CCW9P4 44432644 IC50 = 28940 nM T68698 CS2EY3 44450578 IC50 = 163000 nM T68698 C5JM9A 44450579 IC50 > 500000 nM T68698 CNI6X4 44451567 IC50 = 47200 nM T68698 CI3VJ8 44551468 IC50 = 400 nM T68698 CT8I2H 44561305 Ki = 12400 nM T68698 CVS3O8 44561306 Ki = 20300 nM T68698 C6BG4W 45110892 IC50 = 2.2 nM T68698 C7GN9D 45110893 IC50 = 36 nM T68698 CB5IQ2 45110895 IC50 = 98 nM T68698 CG5RZ9 45111029 IC50 = 4827 nM T68698 C5H3VJ 45111030 IC50 = 189 nM T68698 C36LBT 45111031 IC50 = 9.4 nM T68698 C50EYM 45111032 IC50 = 41 nM T68698 CJA7Q8 45111033 IC50 = 2.7 nM T68698 CL8NW5 45111034 IC50 = 1223 nM T68698 CYAQ84 45111036 IC50 = 28 nM T68698 C7RM9B 46174640 IC50 = 1.3 nM T68698 CZL10R 46874055 Ki = 94.6 nM T68698 CXH9E4 46874068 Ki = 4000 nM T68698 CY41AR 46874106 Ki = 67000 nM T68698 C3DB1E 46874218 Ki = 3100 nM T68698 CN59VL 46874243 Ki = 681 nM T68698 C0HY4G 46874757 Ki = 111 nM T68698 CS32QG 46874759 Ki = 101 nM T68698 C3F2PG 46874761 Ki = 10000 nM T68698 C0NLW6 46875043 Ki = 13700 nM T68698 C0DI9E 46875054 Ki = 45000 nM T68698 CD3C8F 46875063 Ki = 16000 nM T68698 CMGN58 46875065 Ki = 10000 nM T68698 CD28UB 46875621 Ki = 1100 nM T68698 CPHC63 46875632 Ki = 1700 nM T68698 CJ6EL3 46875710 Ki = 770 nM T68698 C19BFH 46875728 Ki = 48500 nM T68698 CE5O4A 46875732 Ki = 570 nM T68698 C8T2JI 46875733 Ki = 710 nM T68698 C7B8QH 46875922 Ki = 3600 nM T68698 CCE7X6 46875931 Ki = 3900 nM T68698 C2VZR9 46876033 Ki = 1300 nM T68698 CGJ03W 46876073 Ki = 96 nM T68698 CZ50WH 46876160 Ki = 3800 nM T68698 CY4L3V 46876365 Ki = 360 nM T68698 CTV70J 46876373 Ki = 570 nM T68698 CKB03R 46876407 Ki = 320 nM T68698 CH81PT 46877209 Ki = 75000 nM T68698 C5NFH6 46877212 Ki = 50000 nM T68698 C1O4WI 46877256 Ki = 750000 nM T68698 CWM2L0 46877257 Ki = 3200 nM T68698 C8IWQ3 46877302 Ki = 105000 nM T68698 CLG04P 46877303 Ki = 19000 nM T68698 C81YJV 46877310 Ki = 550 nM T68698 CJ23FN 46877328 Ki = 4000 nM T68698 CKE16H 46877337 Ki = 118500 nM T68698 CM4CG5 46877338 Ki = 96000 nM T68698 C0HQ5A 46877339 Ki = 17000 nM T68698 C6IRP9 46886640 IC50 > 250000 nM T68698 CW0Y4H 49797674 Ki = 19800 nM T68698 C8GU9B 51003093 IC50 = 60170 nM T68698 CM8WE3 51003094 IC50 > 1000000 nM T68698 C7M3KT 51003095 IC50 > 1000000 nM T68698 C46DIL 51003096 IC50 > 1000000 nM T68698 CZK6B3 53318848 IC50 > 1000000 nM T68698 CC6GR8 57522307 IC50 = 910 nM T68698 C0Z8LK 68364288 IC50 = 2300 nM T68698 CIX13E 73351185 Ki = 1900 nM T68698 C8H9WC 73352895 Ki = 800 nM T68698 CPHB93 90644119 IC50 > 10000 nM T68698 CWP2F5 90644120 IC50 = 2100 nM T68698 C28IXS 90644121 IC50 > 10000 nM T68698 C8INM3 90644122 IC50 = 672 nM T68698 C7ZQA6 90644123 IC50 = 878 nM T68698 C4Y6KI 90644124 IC50 = 1960 nM T68698 CD2X0B 90644125 IC50 = 976 nM T68698 CS3KR7 91824125 Ki = 1.5 nM T68698 C4F3MG 118710205 IC50 = 530 nM T68698 C1PIQ5 118710206 IC50 = 380 nM T68698 C6TMO4 118710207 IC50 = 340 nM T68698 C7IDP1 118710208 IC50 = 970 nM T68698 CG5M1W 118710209 IC50 = 8780 nM T68698 CN29AS 118710210 IC50 = 11360 nM T68698 C0RW1F 118710211 IC50 > 100000 nM T68698 C87EMG 118710212 IC50 = 17000 nM T68698 CMWO70 118710213 IC50 = 2700 nM T68698 C39PRU 118710214 IC50 = 52 nM T68698 CT9PF2 118710215 IC50 = 81 nM T68698 CV51BZ 118710216 IC50 = 530 nM T68698 C5YR2F 118710217 IC50 > 100000 nM T68698 CGT1A9 118710218 IC50 = 4600 nM T68698 CM64LA 118710219 IC50 = 230 nM T68698 CKP9S8 118710220 IC50 = 890 nM T68698 CBW08J 118710221 IC50 = 13 nM T68698 CLAB80 118710222 IC50 = 200 nM T68698 CD01LY 118710223 IC50 = 49 nM T68698 C7HJ8B 118710224 IC50 = 44 nM T68698 C5J7EQ 118710225 IC50 = 330 nM T68698 C01AOB 118710226 IC50 = 320 nM T68698 COMR26 118710227 IC50 = 130 nM T68698 C3AY7W 118710228 IC50 = 70 nM T68698 C91TJV 118710229 IC50 = 60 nM T68698 C1S0YD 118710230 IC50 = 49 nM T68698 C29JSZ 118710231 IC50 = 1200 nM T68698 CI8Z4P 118710232 IC50 = 1500 nM T68698 C34ARU 118710233 IC50 = 110 nM T68698 CR26QJ 118710234 IC50 = 600 nM T68698 CVL4C5 118710235 IC50 = 150 nM T68698 CEW89M 118718118 Ki = 224 nM T68698 CY4DU7 122178501 IC50 > 100000 nM T68698 CGY0N1 122178503 IC50 > 100000 nM T68698 CD98QW 122178504 IC50 > 100000 nM T68698 CX8FW7 122178506 IC50 > 100000 nM T68698 CA98UV 122183895 IC50 = 640 nM T68698 CQ0LA3 122183896 IC50 > 100000 nM T68698 CK6J3X 122183897 IC50 > 100000 nM T68698 CNOV-65 122183898 IC50 = 70 nM T68698 CQM0H1 122183899 IC50 = 60 nM T68698 C6JAU8 122183900 IC50 = 49 nM T68698 CMU94S 122183901 IC50 = 1200 nM T68698 CTU42V 122183902 IC50 = 1500 nM T68698 C0SZO2 122183903 IC50 = 110 nM T68698 CHM13L 122183904 IC50 = 600 nM T68698 C80TRM 122183905 IC50 = 150 nM T68698 CI8WG9 122183915 IC50 = 8.5 nM T68698 CP1FW4 135398641 Ki = 925000 nM T68698 CP4M0E 135976391 Ki 128000 nM T68698 C8WD3Z 135976393 Ki = 422000 nM T68698 CZD50N 137090971 IC50 > 100000 nM T68698 CJW84E 137090972 IC50 > 100000 nM T68698 C5ZM8O 137628302 IC50 > 10000 nM T68698 CW0C4P 155517779 IC50 > 3700 nM T68698 CNP67J 155524359 IC50 > 100000 nM T68698 CKN0W4 155530574 IC50 > 100000 nM T68698 CI2OR3 155531848 IC50 = 4390 nM T68698 CAE5R9 155536819 IC50 > 100000 nM T68698 CZXU90 155538219 IC50 > 100000 nM T68698 CTM53Z 155543643 IC50 > 100000 nM T68698 CKWS45 155544569 IC50 > 100000 nM T68698 CDU83I 155549525 IC50 = 760 nM T68698 CKP82O 155553203 IC50 = 1060 nM T68698 C09CGT 155568198 IC50 > 100000 nM T68698 C0I9OP 155568822 IC50 > 100000 nM T68698 D02XPR 73124 IC50 = 280 nM T68698 D02YYQ 23661679 IC50 = 7530 nM T68698 D0D2MS 11737492 IC50 = 15700 nM T68698 D0F5AJ 126704 Ki = 160 nM T68698 D0O2CM 498018 IC50 = 480 nM T68698 D0X3MK 73087 IC50 = 440 nM T04689 D0T8GD 89594 EC50 = 180000 nM T04689 D09ADT 119380 EC50 = 411000 nM T04689 CUI25G 115224 IC50 = 120000 nM T04689 CY1XN7 7446712 IC50 = 1000 nM T04689 C74CBS 9794141 EC50 = 34000 nM T04689 C0Z5RS 9859386 IC50 = 6000 nM T04689 CLWT60 9882021 EC50 > 100000 nM T04689 CDH4J3 10130527 IC50 = 11000 nM T04689 C6LB2N 10130752 IC50 = 8000 nM T04689 CIQ12L 11701287 Ki = 944 nM T04689 CY7F5O 15389735 EC50 > 1000000 nM T04689 CQ03LX 21290600 IC50 = 81000 nM T04689 CW2R4M 23624283 IC50 = 3981.07 nM T04689 CC1SF7 49863118 IC50 = 794.33 nM T04689 CJ34EQ 53483935 IC50 = 4200 nM T04689 CLH24J 56663402 IC50 > 10000 nM T04689 CU7OP3 56666825 IC50 > 10000 nM T04689 CY01LS 56666826 IC50 > 10000 nM T04689 CCP40B 56666827 IC50 > 10000 nM T04689 CVT85Q 56670262 IC50 = 7800 nM T04689 C7XK8I 56677105 IC50 = 5500 nM T04689 C02AZR 56677106 IC50 > 10000 nM T04689 CL45WN 57345320 IC50 > 30000 nM T04689 CV2J9A 57663655 IC50 = 6309.57 nM T04689 CU3D9N 73388373 EC50 = 19952.62 nM T04689 CI14LP 145949343 IC50 = 11300 nM T04689 CGW92C 145952721 IC50 > 30000 nM T04689 D0R4RN 1204 IC50 = 160 nM T33966 CSD1A3 125874 Ki = 200 nM T33966 CX7U8V 444797 Ki = 450 nM T33966 CF5A3T 9837547 IC50 > 50000 nM T33966 CHI95J 9926432 IC50 = 1400 nM T33966 CM1A0D 9943447 IC50 = 6400 nM T33966 CVK4L6 10418061 IC50 = 3900 nM T33966 C6FQ0R 10465893 IC50 = 1700 nM T33966 CT7IR8 12110710 IC50 > 100000 nM T33966 CFQW82 18955956 Ki = 207000 nM T33966 CYT07N 21575382 IC50 = 0.007 ug.mL-1 T33966 CG0M4T 21575383 IC50 = 3.4 ug.mL-1 T33966 C4UDA1 21606664 IC50 = 0.0052 ug.mL-1 T33966 CR1BW2 21606665 IC50 = 0.0076 ug.mL-1 T33966 C14ZMJ 24768537 Ki = 150 nM T33966 C7J1DP 24774575 Ki = 15000 nM T33966 CP2LY7 25033280 Ki = 17000 nM T33966 C4YKQ1 25033281 Ki = 22000 nM T33966 CA9D6R 25209871 IC50 = 0.12 ug.mL-1 T33966 C46SPD 44374719 Ki = 6500 nM T33966 C0NI9F 44374736 Ki = 5820 nM T33966 CFPX72 44374737 Ki = 4950 nM T33966 CPRQ07 44374750 Ki = 1200 nM T33966 C9RPC6 44374765 Ki = 1160 nM T33966 C1CPB2 44374994 Ki = 980 nM T33966 CXTF63 44374995 Ki = 560 nM T33966 CGD91Y 44374996 Ki = 5900 nM T33966 C4UBK7 44374998 Ki = 320 nM T33966 CG75AN 44377126 Ki = 1200 nM T33966 C6SV1C 44387258 IC50 = 1100 nM T33966 C06HJB 44446952 Ki = 11000 nM T33966 CNK7X5 44446953 Ki = 35000 nM T33966 CEB78N 44446954 Ki = 11000 nM T33966 CMO78A 44446956 Ki = 530 nM T33966 CV6H2M 44446957 Ki = 350 nM T33966 CF4KE1 44446959 Ki = 3600 nM T33966 CW9C0E 44446960 Ki = 7200 nM T33966 CQB5M0 44446963 Ki = 9900 nM T33966 C94POY 44446965 Ki = 5000 nM T33966 CBX2U9 44446967 Ki = 2300 nM T33966 CRZ6B3 44446968 Ki = 14000 nM T33966 CY9O4I 44446969 Ki = 8900 nM T33966 C4PQ7D 44446970 Ki = 1600 nM T33966 C96KIY 44446972 Ki = 5000 nM T33966 CK1EM5 44446974 Ki = 4600 nM T33966 C4V6RZ 44446975 Ki = 16000 nM T33966 CBL9E6 44446976 Ki = 1900 nM T33966 CVYX54 44446979 Ki = 3300 nM T33966 CAI9Z6 44446980 Ki = 4600 nM T33966 C86KVP 44446984 Ki = 11000 nM T33966 CYQN96 44452011 Ki = 2080 nM T33966 CFOM52 44452012 Ki = 790 nM T33966 CJ8G5P 44452013 Ki = 68000 nM T33966 CZI4H9 44452015 Ki = 62600 nM T33966 CC2IS3 44454957 Ki = 12000 nM T33966 C1ESI2 44454959 Ki = 12000 nM T33966 C8L0MV 44454960 Ki = 12000 nM T33966 CBG6T0 44454987 Ki = 15000 nM T33966 CN7UW3 44455013 Ki = 8900 nM T33966 CC5L7S 44455015 Ki > 50000 nM T33966 C6KDT1 44455016 Ki = 9300 nM T33966 CF4ML7 44455018 Ki = 14000 nM T33966 CZI6S1 44455047 Ki = 1700 nM T33966 C3UF6E 44455406 Ki = 5000 nM T33966 CJG71N 44455407 Ki = 32000 nM T33966 C0IR5W 44455428 Ki = 17000 nM T33966 C62KSV 44455429 Ki > 50000 nM T33966 CR9WL2 44455430 Ki = 11000 nM T33966 CXD0Q4 44558923 IC50 = 0.022 ug.mL-1 T33966 C48QBD 45101440 Ki = 160 nM T33966 CP43WZ 45484707 Ki = 430 nM T33966 C2Q9OC 45484717 Ki = 31000 nM T33966 C85MBH 112499885 Ki = 0.087 nM T33966 C2L8SI 112499886 Ki = 0.107 nM T33966 CS49EB 112499887 Ki = 0.04 nM T33966 CG9SC3 145949929 Ki = 289000 nM T33966 C8H1FK 145950532 Ki = 294000 nM T33966 CH02KU 145955234 Ki = 56000 nM T33966 CA6QF8 145956086 Ki = 413000 nM T33966 CZH6P7 145956217 Ki = 238000 nM T33966 CF01VH 145974566 Ki = 60400 nM T33966 CU65CB 155511784 Ki = 0.08 nM T33966 CFG96J 155514645 Ki = 5.9 nM T33966 CF64GH 155518335 Ki = 0.07 nM T33966 CY0H2S 155519530 Ki = 3.1 nM T33966 CA49SR 155523686 Ki = 1.7 nM T33966 C5X4TD 155524117 Ki = 0.1287 nM T33966 C4F1EB 155538870 Ki = 0.3 nM T33966 CD81NB 155547411 Ki = 1.2 nM T33966 D06LNX 3858 IC50 = 400 nM T33966 D0N4RO 44377139 Ki = 310 nM T06792 D00UVA 11556711 IC50 = 2420 nM T06792 D0SH3I 387447 IC50 = 3 nM T06792 D0DP0J 92135659 IC50 = 1840 nM T06792 D0VO0T 24800541 IC50 = 1 nM T06792 CLU69K 10628969 IC50 = 440 nM T06792 CU0FE7 24752894 IC50 = 104 nM T06792 CN62YJ 46850523 IC50 = 140 nM T06792 CEV5D1 49859748 IC50 = 10600 nM T06792 C3QG8L 59127842 IC50 = 36 nM T06792 C82JTA 71305068 IC50 = 21500 nM T06792 C45HOE 71562349 IC50 > 10000 nM T06792 CGY43C 78425867 IC50 = 1850 nM T06792 CC0OF1 101874274 IC50 = 300 nM T06792 CG0N1O 101874275 IC50 = 7100 nM T06792 CL50TR 101874276 IC50 = 7300 nM T06792 C0RY3V 101874277 IC50 = 6200 nM T06792 CVHC29 101874278 IC50 > 100000 nM T06792 C4VHU6 101874279 IC50 > 100000 nM T06792 C9C5OZ 117607839 IC50 = 3530 nM T06792 CLHS74 117607901 IC50 = 223 nM T06792 CW9R0U 117607904 IC50 = 0.623 nM T06792 C7QST8 117611788 IC50 = 51 nM T06792 CO1HJ9 117611880 IC50 = 140 nM T06792 C9YH1X 117611941 IC50 = 112 nM T06792 CO6E0B 118709670 IC50 = 170 nM T06792 C8WMH3 118709671 IC50 = 68 nM T06792 CZ8GE0 118709672 IC50 = 96 nM T06792 CZ70XF 118709673 IC50 = 67 nM T06792 C7C9PZ 118709674 IC50 = 220 nM T06792 CS05KF 118709675 IC50 = 22 nM T06792 C17ZTF 118709676 IC50 = 34 nM T06792 C0WZ3V 118709677 IC50 = 66 nM T06792 C14VLB 118709678 IC50 = 87 nM T06792 CO5CU1 118709679 IC50 = 42 nM T06792 C1RA9C 118709680 IC50 = 130 nM T06792 C9BWP4 145979302 IC50 = 5700 nM T06792 CN79HG 145979487 IC50 = 3500 nM T06792 CEI3U1 145979850 IC50 = 4800 nM T06792 CG6UL0 145980995 IC50 = 4000 nM T06792 CB67YT 145981691 IC50 = 16100 nM T06792 C41IRV 145981707 IC50 = 14000 nM T06792 CL1F8N 145982922 IC50 = 13000 nM T06792 C5X3GQ 145986425 IC50 = 12600 nM T06792 CRZE86 145986857 IC50 = 45000 nM T06792 CHWT73 145987085 IC50 = 8900 nM T06792 CM3H4F 145987197 IC50 = 4300 nM T06792 CNZ7R6 145987536 IC50 = 12500 nM T06792 C1EF3B 145988020 IC50 = 23800 nM T06792 CQIS01 145988427 IC50 = 7310 nM T06792 CE16JH 145989568 IC50 = 52000 nM T06792 CXG30R 145990249 IC50 = 21000 nM T06792 C8IL9E 145992200 IC50 = 10320 nM T06792 CBY18W 145992498 IC50 = 2770 nM T06792 C6GHQ9 145993211 IC50 = 59000 nM T06792 CEVY70 145993649 IC50 = 24600 nM T06792 CJO08K 145993925 IC50 = 8800 nM T06792 C8E6ZX 155514792 IC50 > 10000 nM T06792 CX76LO 155515463 IC50 > 10000 nM T06792 C53ZEN 155516179 IC50 > 100000 nM T06792 CM3BV8 155516620 IC50 > 100000 nM T06792 CE95IQ 155518158 IC50 > 100000 nM T06792 CNM0Q9 155521286 IC50 > 100000 nM T06792 CZKF54 155521690 IC50 > 10000 nM T06792 CB0WG8 155522381 IC50 = 743.5 nM T06792 C8GNQ9 155522828 IC50 > 25000 nM T06792 CW75YK 155523151 IC50 > 100000 nM T06792 CAC34Y 155527225 IC50 = 3100 nM T06792 CUP2B4 155531358 IC50 = 415 nM T06792 C2NTI6 155538936 IC50 > 100000 nM T06792 C6OIY3 155541618 IC50 > 100000 nM T06792 C12LPX 155551071 IC50 > 10000 nM T06792 CBHM14 155553205 IC50 > 100000 nM T06792 C35NJC 155553210 IC50 > 10000 nM T06792 CI15FC 155553565 IC50 > 10000 nM T06792 CVJ3E7 155553910 IC50 > 100000 nM T06792 C6YP0L 155554916 IC50 > 100000 nM T06792 C5Z7YC 155567712 IC50 > 10000 nM T06792 C4ZV3Q 155568941 IC50 > 10000 nM T06792 D0Q4MO 23642227 IC50 = 287 nM T01943 D04AIT 5280445 IC50 = 5000 nM T01943 D0K8KX 5280343 IC50 = 1500 nM T01943 D0L4FS 5280961 IC50 = 7000 nM T01943 D0U2BH 65064 IC50 = 400 nM T01943 CY0AL9 72279 IC50 = 30000 nM T01943 CNIW58 107905 IC50 = 400 nM T01943 CDZ65K 199472 IC50 = 600 nM T01943 CN7AQ6 15958429 IC50 = 14 ug.mL-1 T01943 CZR73C 16072317 IC50 = 12.5 ug.mL-1 T01943 C20YLR 22600366 IC50 = 0.58 ug.mL-1 T01943 C15VRN 44412009 IC50 = 40000 nM T01943 C6XHE9 49770727 IC50 = 12 ug.mL-1 T01943 CG4H0W 71768351 IC50 > 100000 nM T01943 CMAP17 71768352 IC50 = 16300 nM T01943 CW0T6G 72703050 IC50 > 100000 nM T01943 CPZO91 72703242 IC50 > 100000 nM T01943 CQ2IU6 72703243 IC50 = 90000 nM T01943 C0B3KS 72703244 IC50 = 13000 nM T01943 CE6HI7 72703245 IC50 = 28000 nM T01943 CJ12BK 72703246 IC50 = 10000 nM T01943 CESN04 73347724 IC50 > 100000 nM T01943 D01KKU 5281894 IC50 = 20000 nM T01943 D02TVS 985 IC50 > 100 ug.mL-1 T01943 D0MF5Y 5281614 IC50 = 2000 nM T01943 D0NJ4H 5281670 IC50 = 8000 nM T01943 D0RB1V 6419835 IC50 = 400 nM T01943 D0S9YX 5280373 IC50 = 8000 nM T01943 D0SY2M 5281708 IC50 = 30000 nM T01943 D0T3PW 5281672 IC50 = 2000 nM T19229 D01KKQ 135400182 IC50 = 99.5 nM T19229 D02LWU 148121 IC50 = 57 nM T19229 D0SV8E 126941 IC50 = 121 nM T19229 D0Y4GO 135410875 IC50 = 13.2 nM T19229 CPM3L5 67092576 IC50 > 1000 nM T19229 CTK64O 67092918 IC50 > 1000 nM T19229 C87FBU 135455948 IC50 = 80.2 nM T19229 CF8D5O 135465664 IC50 > 1000 nM T19229 C9Z4ES 135567027 IC50 = 5.21 nM T19229 C14LTO 135567028 IC50 = 43.4 nM T19229 CF39AI 135567029 IC50 = 3.34 nM T19229 C8N7ES 135567030 IC50 = 41.5 nM T19229 CGM2V5 135567031 Ki = 420 nM T19229 CFE2O7 135567034 IC50 = 40 nM T19229 C8KVP5 135567035 IC50 = 6.51 nM T19229 CSQX75 135567163 IC50 = 87.4 nM T19229 CQF8P5 135800109 IC50 = 9.71 nM T19229 C6XK3M 135862924 Ki = 100 nM T19229 CL8VN5 136015502 IC50 = 312 nM T19229 CR7UY3 136044173 IC50 > 1000 nM T19229 C0Q5FI 136044174 IC50 > 1000 nM T19229 CGX68Y 136044175 IC50 > 1000 nM T19229 C4C9FN 136044176 IC50 > 1000 nM T19229 CIPD35 136044177 IC50 > 1000 nM T19229 CZG8W6 136059167 IC50 = 30.4 nM T19229 CZC95Y 136059168 IC50 > 1000 nM T19229 CG2ID9 136059169 IC50 > 1000 nM T19229 C2WH0S 136059178 IC50 > 1000 nM T19229 CB3GL7 136059191 IC50 > 1000 nM T19229 CCHG08 136059192 IC50 > 1000 nM T19229 C4Q1HF 136180345 IC50 = 141 nM T19229 CDC83K 136180346 IC50 = 57.4 nM T19229 CF7NW6 136180347 IC50 > 1000 nM T19229 CPH52E 137150145 IC50 > 1000 nM T19229 C9XD1M 137150146 IC50 = 747 nM T19229 CHDB56 137150160 IC50 = 48.6 nM T19229 CUF8R1 155515541 IC50 = 207 nM T19229 CMKA64 155517044 IC50 = 81.7 nM T19229 CCL3Y9 155518053 IC50 = 20.4 nM T19229 C91SVN 155519837 IC50 = 57.5 nM T19229 CO7BN6 155524531 IC50 > 1000 nM T19229 CT70WU 155530762 IC50 = 5.01 nM T19229 CX42MF 155532591 IC50 = 267 nM T19229 CFU98A 155534971 IC50 = 88.5 nM T19229 C4K2RU 155538415 IC50 > 1000 nM T19229 C27BIX 155539477 IC50 > 1000 nM T19229 C6S7OC 155548982 IC50 = 3.82 nM T19229 CX3K8F 155549935 IC50 = 4.57 nM T19229 CJ0MK5 155554671 IC50 = 67 nM T19229 CYQ0I9 155555353 IC50 = 109 nM T90987 CJS23I 9868333 Ki = 7800 nM T90987 CY08WJ 10322755 Ki = 7800 nM T90987 C8C5AV 11294179 Ki > 1000 nM T90987 CZB81D 44395506 IC50 = 79 nM T90987 C52ESR 66559934 IC50 > 50000 nM T90987 C57ARI 66560021 IC50 > 50000 nM T90987 CU58DB 66560022 IC50 > 50000 nM T90987 C16RDM 66560389 IC50 > 50000 nM T90987 C8RZG9 66560479 IC50 > 50000 nM T90987 CKW2Q5 71453375 IC50 > 50000 nM T90987 D0H6CK 10160968 Ki = 776 nM T06569 D00STL 644241 Ki = 461 nM T06569 D01MUR 68844 Ki = 0.9 nM T06569 D02PJA 24841 Ki = 810000 nM T06569 D03QGM 5355 Ki = 0.8 nM T06569 D03RTS 2662 Ki = 94 nM T06569 D03UOT 785 Ki = 521000 nM T06569 D05OFX 219078 Ki = 412 nM T06569 D05UYW 5284549 Ki = 10 nM T06569 D07HBX 338 Ki = 11900 nM T06569 D07INV 3295 Ki = 43 nM T06569 D07VDZ 5284627 Ki = 45 nM T06569 D09NIA 2732 Ki = 1347 nM T06569 D09VAZ 5565 Ki = 43000 nM T06569 D0AZ3C 5291 Ki = 392 nM T06569 D0AZ8C 5213 Ki = 9700 nM T06569 D0C2II 4100 Ki = 10 nM T06569 D0C8FX 3005837 Ki = 2410 nM T06569 D0E1SW 1986 Ki = 11 nM T06569 D0H8FH 3702 Ki = 1606 nM T06569 D0J4GO 3038 Ki = 79 nM T06569 D0J7RK 36811 Ki = 9470 nM T06569 D0K0OZ 5702160 Ki = 98.2 nM T06569 D0K1QD 3998 Ki = 4800 nM T06569 D0K8KX 5280343 Ki = 6170 nM T06569 D0L4JT 5333 Ki = 941 nM T06569 D0L6DA 119607 Ki = 572 nM T06569 D0OT0O 44561 Ki = 1810000 nM T06569 D0PQ3G 3440 Ki = 245 nM T06569 D0SH3I 387447 Ki = 4380 nM T06569 D0U5QK 1983 Ki = 658000 nM T06569 D0Y2IZ 5560 Ki = 2459 nM T06569 D0Z3EI 6038 Ki = 33 nM T06569 D04IIU 216468 Ki = 47 nM T06569 D05NJI 5287541 Ki = 653 nM T06569 D06PII 5356 Ki = 134 nM T06569 D08BXT 1102 Ki = 1410 nM T06569 D0L6HN 996 Ki = 208000 nM T06569 D0U3EP 445154 Ki = 8070 nM T06569 D0V0UK 82267 Ki = 0.07 nM T06569 D03SLR 445858 Ki = 8450 nM T06569 D0NH9P 135 Ki = 5700 nM T06569 D0LD9S 1103 Ki = 990 nM T06569 CI0WH9 72 Ki = 4720 nM T06569 CUT2V4 260 Ki = 730000 nM T06569 COV5W3 402 Ki = 710000 nM T06569 CSZ43B 540 Ki = 690000 nM T06569 C97QXH 767 Ki = 690000 nM T06569 C39CTO 768 Ki = 70000 nM T06569 C1QDT0 781 Ki = 890000 nM T06569 CAD4R0 798 Ki = 3630 nM T06569 CW0R2L 944 Ki = 760000 nM T06569 CQV86E 1100 Ki = 14200000 nM T06569 C8W7BZ 1118 Ki = 9900000 nM T06569 CU12QE 1203 Ki = 4910 nM T06569 C5L7VX 2871 Ki = 2230 nM T06569 CJ2F6P 5056 Ki = 8630 nM T06569 CDJ4K6 5987 Ki = 0.09 nM T06569 CUP2F4 7043 Ki = 234700 nM T06569 C1CVT7 7121 Ki = 24420 nM T06569 C6NC4O 7414 Ki = 5100 nM T06569 CJKY76 7420 Ki = 3170 nM T06569 CIU0C8 7519 Ki = 234700 nM T06569 CUG8B9 11418 Ki = 402300 nM T06569 CCPT31 11419 Ki = 427100 nM T06569 CUA0L6 14917 Ki = 600000 nM T06569 C3NG2U 24529 Ki = 820000 nM T06569 CFM9L6 24530 Ki = 70000 nM T06569 C4OU6D 35703 Ki = 82300 nM T06569 C1N6SE 61127 Ki = 29138 nM T06569 CE5RZ1 76509 Ki = 780 nM T06569 CX47BZ 78479 Ki = 53000 nM T06569 CEC01M 97598 Ki = 12840 nM T06569 CN19UT 129695 Ki = 110 nM T06569 CUX39B 132037 Ki = 3410 nM T06569 CVB67D 134560 Ki = 73 nM T06569 CD2HC7 138614 Ki = 405600 nM T06569 C8AO0Z 165323 Ki = 114 nM T06569 C1QOB5 284045 Ki = 382473 nM T06569 CT3ZU4 388776 Ki = 1100 nM T06569 CH21KA 389641 Ki = 104000 nM T06569 C6CQO3 389642 Ki = 114000 nM T06569 CNPZ40 394897 Ki = 765 nM T06569 C4TD8M 2388085 Ki > 10000 nM T06569 C21FUI 2801263 Ki = 3790 nM T06569 CE2GR3 2900806 Ki = 109000 nM T06569 CI8JY0 5172475 Ki = 740 nM T06569 C9L8AX 6537802 Ki = 41 nM T06569 C65FRB 6852128 Ki = 136 nM T06569 CKCM96 7463376 Ki = 8580 nM T06569 CDCP43 7766335 Ki = 420 nM T06569 CY47OI 9998322 Ki = 24 nM T06569 CWM01R 10059806 Ki = 13692 nM T06569 CD58EL 10083644 Ki = 730 nM T06569 C58IYR 10366827 Ki = 590 nM T06569 C3HBY6 10375558 Ki = 4150 nM T06569 C73KXU 10586607 Ki = 6700 nM T06569 C9TSQ6 10632698 Ki = 43100 nM T06569 C8C6ER 11069133 Ki = 41 nM T06569 C39IDU 11183936 Ki = 12010 nM T06569 CHC42Y 11245700 Ki = 654 nM T06569 CA6T0Z 11322287 Ki = 11660 nM T06569 CXB86F 11579563 Ki = 12530 nM T06569 CDU79V 11637531 Ki = 10820 nM T06569 CX4W3J 11701693 Ki = 9870 nM T06569 CV7HN1 11795548 Ki = 65 nM T06569 CMPA32 12066940 Ki > 500000 nM T06569 CB15KR 12066941 Ki > 500000 nM T06569 CREV05 12140130 Ki = 12430 nM T06569 CHOG93 14611919 Ki = 2650 nM T06569 C8PER5 15938557 Ki > 500000 nM T06569 CC0Z4V 16119626 Ki = 510 nM T06569 C6SFI8 18268734 Ki > 10000 nM T06569 C61KUX 21726402 Ki = 9680 nM T06569 C54IUM 21778115 Ki = 17830 nM T06569 C27BJH 21778117 Ki = 17430 nM T06569 C9U4TE 22313850 Ki = 1230 nM T06569 CICR37 23426698 Ki = 38190 nM T06569 CPN2T5 25392418 Ki > 10000 nM T06569 C82MRL 44144383 Ki = 25 nM T06569 CI3O9B 44395149 Ki = 147 nM T06569 CZ4DF9 44399462 Ki = 76 nM T06569 CD5MJ6 44399571 Ki = 59 nM T06569 C2T7MB 44399654 Ki = 749 nM T06569 C8E0MV 44552472 Ki = 9210 nM T06569 CKG53H 44552473 Ki = 1920 nM T06569 C17XAJ 44552559 Ki = 4170 nM T06569 CF0KQ8 44581932 Ki = 73 nM T06569 C23MVW 45269009 IC50 = 35700 nM T06569 C0RG8K 45269749 Ki > 100000 nM T06569 CV5RQ3 45484187 Ki = 4300 nM T06569 CTG20B 45485271 Ki = 100 nM T06569 CK4U0V 45485283 Ki = 5600 nM T06569 CHE08Y 46225608 Ki = 10230 nM T06569 CIE2H3 46225609 Ki = 9640 nM T06569 CF42NR 46225631 Ki = 7610 nM T06569 C0ZG3L 46225639 Ki = 7960 nM T06569 CGW1I5 46225644 Ki = 7840 nM T06569 CEOQ06 46225645 Ki = 8310 nM T06569 CR0WO3 46225646 Ki = 8540 nM T06569 CC2BL5 46225656 Ki = 8980 nM T06569 CW52PZ 46225672 Ki = 4950 nM T06569 CXJ1C9 46225673 Ki = 4310 nM T06569 C93AIR 46899573 Ki = 156000 nM T06569 CJ0R2O 46911381 Ki = 921 nM T06569 CF89ML 53307609 Ki = 29670 nM T06569 C0NUM6 53386724 Ki = 980 nM T06569 C54FGU 53386866 Ki = 543 nM T06569 CRI54V 53386867 Ki = 1035 nM T06569 CUX7S4 53386868 Ki = 814 nM T06569 CIJ9V0 56684131 Ki = 8140 nM T06569 CH52DA 56921864 Ki = 8950 nM T06569 CUR32K 57334711 Ki = 480 nM T06569 C2CD1R 57334712 Ki = 470 nM T06569 C1K0DM 57334713 Ki = 470 nM T06569 CP7YR5 57345662 Ki = 8 nM T06569 C13FJU 57392368 Ki = 510 nM T06569 CY5G4Z 57395885 Ki = 960 nM T06569 C5RX6H 57396029 Ki = 5240 nM T06569 CP75OF 57397664 Ki = 158592 nM T06569 CUAG84 57397836 Ki = 765300 nM T06569 CW43HV 57397837 Ki = 5590 nM T06569 C1MCW8 57399336 Ki = 919182 nM T06569 C2CAM1 57399491 Ki = 4810 nM T06569 C2J7GW 66572313 Ki = 35450 nM T06569 C7J5RN 66573254 Ki = 45360 nM T06569 CQR91N 70692438 Ki = 28170 nM T06569 CWJ0Q8 70696540 Ki = 11143 nM T06569 CXJ16H 71450117 Ki = 8055 nM T06569 CB8JA3 71455488 Ki = 9340 nM T06569 C02UHX 71455489 Ki = 7116 nM T06569 CICJ97 71457274 Ki = 9280 nM T06569 CMHG14 71521493 Ki = 6200 nM T06569 CHN53G 71521494 Ki = 7700 nM T06569 CZJ5M6 71521495 Ki = 7900 nM T06569 CFBE53 71521496 Ki > 100000 nM T06569 CME27W 71521497 Ki = 8100 nM T06569 C24XWU 71521575 Ki = 8800 nM T06569 CJF68W 71521576 Ki > 100000 nM T06569 CX82JD 72696463 Ki = 130 nM T06569 COCV73 72696591 Ki = 1388 nM T06569 C5KHD7 72696592 Ki = 220 nM T06569 C4FBA6 72696593 Ki = 274 nM T06569 CO1JM5 72696594 Ki = 167 nM T06569 CUF61Q 72696595 Ki = 148 nM T06569 CO1JT3 73054728 Ki = 857 nM T06569 CDGZ03 101879106 Ki > 120 nM T06569 CY6ER7 101879108 Ki > 120 nM T06569 C0D1SQ 118724328 Ki > 120 nM T06569 C89YTC 118724329 Ki > 120 nM T06569 CBT87C 118724330 Ki > 120 nM T06569 C49AWZ 118724331 Ki > 120 nM T06569 CH1N0C 122193189 Ki = 560 nM T06569 C19HVL 122193190 Ki = 740 nM T06569 C5TQJ1 122193251 Ki = 540 nM T06569 C8XCL0 122193252 Ki = 470 nM T06569 CIX41M 138393379 Ki > 10000 nM T06569 CBOM51 138753317 Ki > 10000 nM T06569 COP4Q6 155516517 Ki = 9192 nM T06569 CAG9L4 155517430 Ki = 2440 nM T06569 CP49HE 155520274 Ki = 7428 nM T06569 CTJ3I7 155530506 Ki = 7218 nM T06569 CT5NG1 155534179 Ki > 10000 nM T06569 CVU5P6 155535355 Ki > 10000 nM T06569 C8RV6T 155541805 Ki > 10000 nM T06569 CU1NE7 155549031 Ki > 10000 nM T06569 CWB82E 155555878 Ki > 10000 nM T06569 CH5VU6 155568899 Ki > 10000 nM T06569 D00IUB 13019 Ki = 13700 nM T06569 D00RNZ 910172 Ki = 93100 nM T06569 D00XJA 711717 Ki = 65200 nM T06569 D00YEF 148885 Ki = 1414 nM T06569 D01BUB 94952 Ki = 90600 nM T06569 D01STY 9861037 Ki = 1024 nM T06569 D02DBP 5054 Ki = 550000 nM T06569 D02QGI 273 Ki = 740 nM T06569 D03NBX 637308 Ki = 770 nM T06569 D03ZMQ 323 Ki = 2000 nM T06569 D04CVC 4687472 Ki = 96 nM T06569 D04NSN 169682 Ki = 813 nM T06569 D05QUG 45485279 Ki > 500000 nM T06569 D05TLB 11117301 Ki = 795 nM T06569 D05WQF 637540 Ki > 1000000 nM T06569 D05XZM 10081162 Ki = 6680 nM T06569 D06DYP 234562 Ki = 44500 nM T06569 D06TPF 1057 Ki = 520 nM T06569 D07MTM 403 Ki = 23500 nM T06569 D07QJJ 289 Ki = 606000 nM T06569 D07TAJ 914298 Ki = 6600 nM T06569 D09JPC 16402 Ki = 720 nM T06569 D09PWX 8739 Ki = 887 nM T06569 D09QHC 7370 Ki = 2970 nM T06569 D09WSJ 19772348 Ki = 1334 nM T06569 D09WVV 8111 Ki = 11500 nM T06569 D0A0YX 5143 Ki = 935 nM T06569 D0A1CM 5281855 Ki = 7060 nM T06569 D0A6HS 6852129 Ki = 103 nM T06569 D0AU0M 637542 Ki = 6720 nM T06569 D0C7LR 313 Ki = 720000 nM T06569 D0D4OV 20043772 Ki = 1020 nM T06569 D0D6UR 12394434 Ki > 500000 nM T06569 D0E8CC 18794 Ki = 93 nM T06569 D0EJ9B 66827 Ki = 0.82 nM T06569 D0G0FJ 11206245 Ki = 1090 nM T06569 D0G3BI 25090 Ki = 54700 nM T06569 D0H3NS 10752 Ki = 76300 nM T06569 D0L5TZ 20195365 Ki = 9300 nM T06569 D0LU4S 156219 Ki = 13000 nM T06569 D0M3PO 69561 Ki = 955 nM T06569 D0M6RM 7365 Ki = 13.9 nM T06569 D0N1AW 45485270 Ki = 1300 nM T06569 D0NN3Q 78105 Ki = 1275 nM T06569 D0OI1H 72894 Ki = 772 nM T06569 D0OT5L 1631814 Ki = 7400 nM T06569 D0P6AM 3526523 Ki = 4680 nM T06569 D0Q7DJ 10742 Ki = 7550 nM T06569 D0R4WJ 16129778 Ki = 17800 nM T06569 D0R7QY 127676 Ki = 1860 nM T06569 D0RB0D 44268050 Ki > 500000 nM T06569 D0TY8X 31036 Ki = 86 nM T06569 D0U4BB 10748 Ki = 5500 nM T06569 D0V9EN 689043 Ki = 7330 nM T06569 D0VD7H 84724 Ki = 798 nM T06569 D0X5HL 15107 Ki = 640 nM T06569 D0X6IE 4422372 Ki = 55 nM T06569 D0Y3TZ 370 Ki = 6130 nM T06569 D0YU8J 1502014 Ki = 1097 nM T06569 D0Z1HY 67136 Ki = 608 nM T06569 D0ZC3W 6269 Ki = 1582 nM T03529 D07XOD 2733079 IC50 = 11000 nM T03529 CCI13U 11536910 IC50 = 20400 nM T03529 CN8LG9 13171484 IC50 = 37000 nM T03529 CXC3W5 20377108 IC50 = 28400 nM T03529 C3PDB6 20377110 IC50 = 122000 nM T03529 CI3Q2W 25125116 IC50 = 312000 nM T03529 C5NER0 25125122 IC50 = 7100 nM T03529 CGF7A0 25125458 IC50 = 12800 nM T03529 CS1RD3 25125461 IC50 = 7600 nM T03529 CJ4I7C 25125799 IC50 = 31600 nM T03529 CM6EV5 70681820 IC50 = 7500 nM T03529 CUYZ39 70681821 IC50 = 5600 nM T03529 C9BP5R 70681822 IC50 = 5200 nM T03529 CP6E4R 70681828 IC50 = 16400 nM T03529 CBHO57 70681829 IC50 = 11800 nM T03529 COQC31 70681830 IC50 = 17500 nM T03529 CUF80Q 70681831 IC50 = 15700 nM T03529 CXU67P 70681832 IC50 = 119000 nM T03529 C45NUH 70681833 IC50 = 70600 nM T03529 CV91MS 70681834 IC50 = 194000 nM T03529 CDN0C4 70683924 IC50 = 39800 nM T03529 CH2PL3 70683932 IC50 = 9900 nM T03529 C8E4JH 70683933 IC50 = 7700 nM T03529 CA27DC 70683934 IC50 = 98000 nM T03529 CUC9K6 70686055 IC50 = 17200 nM T03529 C48CLJ 70686056 IC50 = 12300 nM T03529 C59QXF 70688191 IC50 = 21300 nM T03529 C3S9IJ 70688192 IC50 = 11600 nM T03529 C1S3IH 70690203 IC50 = 11400 nM T03529 CJ5PK6 70690208 IC50 = 56000 nM T03529 CL0JW1 70692374 IC50 = 16200 nM T03529 CNW8O1 70692382 IC50 = 13200 nM T03529 CM2KW1 70692383 IC50 = 8400 nM T03529 C04XZL 70694433 IC50 = 6200 nM T03529 CD5O8R 70694437 IC50 = 9500 nM T03529 CTLH58 70696507 IC50 = 10900 nM T03529 C3TV8N 70696508 IC50 = 18700 nM T03529 D05AMQ 6539137 IC50 = 83500 nM T03529 D0M5DR 57330144 IC50 = 36100 nM T97822 D03RTS 2662 IC50 = 89 nM T97822 D0GY5Z 2244 IC50 = 15000 nM T97822 D0R1RS 3715 IC50 = 10 nM T97822 D0U2FN 71321 IC50 = 6500000 nM T97822 D05WPQ 6438354 IC50 = 3200 nM T97822 D09QRO 55390 IC50 = 10000 nM T97822 D0DP8P 47795 IC50 = 5800 nM T97822 D0JY4Y 443292 IC50 > 100000 nM T97822 D0N1SU 133021 IC50 = 160 nM T97822 D0O8ZE 5059 IC50 = 5300 nM T97822 D0S8YL 3969 IC50 = 44000 nM T97822 CH0L7P 71697 IC50 = 950000 nM T97822 CI5D9O 92656 IC50 = 100 nM T97822 CV7L0G 112230 IC50 = 100000000 nM T97822 CT2XZ0 116545 IC50 = 7079457.84 nM T97822 CAT4E3 129615 IC50 = 3388441.56 nM T97822 CCJ76H 512829 IC50 = 9000 nM T97822 CE2BC3 512830 IC50 = 14000 nM T97822 C16VBD 512831 IC50 = 12000 nM T97822 CT7E6Y 573683 IC50 > 800000 nM T97822 CZ0AH3 638278 IC50 = 130000 nM T97822 C6EVL8 854057 IC50 = 3467368.5 nM T97822 CQM64G 3037018 IC50 = 800 nM T97822 COH1C4 3052566 IC50 = 446683.59 nM T97822 C82IPJ 3052567 IC50 = 912010.84 nM T97822 C4VBK3 3253091 IC50 = 50000 nM T97822 CU86JL 4618600 IC50 = 40000 nM T97822 C4M1JC 5709318 IC50 = 44000 nM T97822 COQ7T3 5973690 IC50 = 63000 nM T97822 C3G7DT 6365297 IC50 = 4200 nM T97822 C40FZG 6366698 IC50 = 1300 nM T97822 C02AQY 6366699 IC50 ~ 1000 nM T97822 CWK1F9 6438990 IC50 = 110 nM T97822 C62UOZ 6439221 IC50 = 780 nM T97822 CHQ4Z3 6439222 IC50 = 1300 nM T97822 COC86Q 6439421 IC50 = 390 nM T97822 CLJ91K 6439912 IC50 = 260 nM T97822 C82TEX 7515046 IC50 < 10000 nM T97822 CUS6L8 9822795 IC50 = 30 nM T97822 C5C9ET 10042219 IC50 > 100000 nM T97822 C9T7YV 10063338 IC50 > 100000 nM T97822 CBL7R3 10220019 IC50 = 400 nM T97822 C2WE0I 10246235 IC50 = 9600 nM T97822 C20BTQ 10313997 IC50 = 5500 nM T97822 C8EQI3 10334136 IC50 > 100000 nM T97822 CC1UF0 10335738 IC50 > 100000 nM T97822 C25MYB 10425738 IC50 > 100000 nM T97822 CPR7J0 10469807 IC50 = 12589254.12 nM T97822 C6JI5F 10492615 IC50 > 300000 nM T97822 C0NRO9 10513373 IC50 = 570000 nM T97822 CK0OL2 10704667 IC50 = 27000 nM T97822 CUOI16 10729548 IC50 = 26000 nM T97822 C8IBM2 10801359 IC50 = 250000 nM T97822 CC8S6O 10801786 IC50 = 37000 nM T97822 CDZ94R 10826230 IC50 = 29000 nM T97822 CGLQ72 11723348 IC50 > 100000 nM T97822 CH9VC8 13245625 IC50 > 10000 nM T97822 CRA87I 13556944 IC50 = 14125375.45 nM T97822 C0P5AK 13914227 IC50 > 100000 nM T97822 C49OGE 13914253 IC50 > 100000 nM T97822 C4U3RD 14006855 IC50 = 5000 nM T97822 C6EZ0K 14312565 IC50 > 10000 nM T97822 C2X8PQ 14416570 IC50 = 34 nM T97822 C5PT1G 14416572 IC50 670 nM T97822 C1SG0F 14416576 IC50 = 10000 nM T97822 CRYI80 14416580 IC50 = 610 nM T97822 C27NOS 14416585 IC50 < 10000 nM T97822 C6BP2F 14416587 IC50 < 1000 nM T97822 CER87K 14762923 IC50 = 13803842.65 nM T97822 CGYF09 14762938 IC50 = 501187233.6 nM T97822 CX9AH8 14762939 IC50 = 501187233.6 nM T97822 CU3OT4 14762940 IC50 = 165958690.7 nM T97822 CXT3B5 14762942 IC50 = 100000000 nM T97822 CNZ45J 14762943 IC50 = 91201083.94 nM T97822 CL2A1E 14762944 IC50 = 91201083.94 nM T97822 C78IHC 14762948 IC50 = 50118723.36 nM T97822 CBL2O8 14762951 IC50 = 14791083.88 nM T97822 C8NKZ7 14762954 IC50 = 7079457.84 nM T97822 C4PS0F 14771889 IC50 < 10000 nM T97822 CV41BE 14771890 IC50 = 3100 nM T97822 CCX7K5 14771891 IC50 = 1400 nM T97822 CG57JP 14771892 IC50 = 1300 nM T97822 C91VJM 14771893 IC50 = 230 nM T97822 C0EMA5 14771894 IC50 < 1000 nM T97822 CZ4WJ2 14771895 IC50 = 730 nM T97822 CV5YH8 14771896 IC50 < 10000 nM T97822 C3HNQ2 14771897 IC50 < 10000 nM T97822 CH0TC9 14771898 IC50 < 10000 nM T97822 CX3N7Z 14771899 IC50 = 11000 nM T97822 CX7VA0 14771900 IC50 < 10000 nM T97822 CZC2D4 14771901 IC50 < 10000 nM T97822 CTY60Q 14771902 IC50 < 10000 nM T97822 C0D5OC 14771903 IC50 = 1500 nM T97822 CS3V5C 14771904 IC50 < 10000 nM T97822 CNH5M1 14771905 IC50 = 3200 nM T97822 CXN94C 14771906 IC50 = 510 nM T97822 CY2HF8 14771907 IC50 = 1400 nM T97822 CP5M9A 14771908 IC50 = 190 nM T97822 CI3XK7 14771909 IC50 < 10000 nM T97822 C8NTK2 14771910 IC50 = 750 nM T97822 C8H6XA 14771911 IC50 = 2500 nM T97822 CK53TR 14771912 IC50 < 1000 nM T97822 C10DIY 14771913 IC50 < 1000 nM T97822 C2F9TX 14771915 IC50 = 1100 nM T97822 C83VPQ 14771916 IC50 = 710 nM T97822 CA0C7U 14771917 IC50 = 1000 nM T97822 CK0AR5 14771918 IC50 < 1000 nM T97822 C8SRH6 14771919 IC50 > 10000 nM T97822 CCS9Y4 14771920 IC50 > 10000 nM T97822 C47LJK 14771921 IC50 > 10000 nM T97822 C9OWP0 14771922 IC50 = 1300 nM T97822 C1Z6FX 14771923 IC50 = 780 nM T97822 CHI8M3 14771924 IC50 < 10000 nM T97822 C4JX5S 14771927 IC50 = 590 nM T97822 CRGJ45 14771928 IC50 < 10000 nM T97822 C7L2ZJ 14771929 IC50 = 400 nM T97822 CXAG49 14771930 IC50 < 1000 nM T97822 C54ITL 14771931 IC50 = 110 nM T97822 CC4LM1 14771932 IC50 < 10000 nM T97822 CU6TO3 14771933 IC50 < 10000 nM T97822 C08CRZ 14771934 IC50 = 630 nM T97822 CA3D5U 14771935 IC50 = 1000 nM T97822 CZU2H5 14771936 IC50 = 300 nM T97822 C3B0LX 14771937 IC50 < 10000 nM T97822 CRT9E4 14771938 IC50 > 10000 nM T97822 C18DXV 14977360 IC50 = 71000 nM T97822 CD8YK4 15256755 IC50 = 140000 nM T97822 C53TQI 19044744 IC50 > 100000 nM T97822 CGPW68 19044748 IC50 > 100000 nM T97822 CLN6S5 19044753 IC50 > 100000 nM T97822 CR1W2E 19934882 IC50 > 100000 nM T97822 CF30ID 23275601 IC50 = 66069344.8 nM T97822 CUC36F 23680215 IC50 = 9772372.21 nM T97822 CN6F4H 23680216 IC50 = 4365158.32 nM T97822 C2JUV4 23680221 IC50 = 17782794.1 nM T97822 CHY73S 23680224 IC50 = 524807460.3 nM T97822 C7HV8Y 23680227 IC50 = 70794578.44 nM T97822 CZV8U1 23680228 IC50 = 4677351.41 nM T97822 C54NWH 23680229 IC50 = 741310241.3 nM T97822 CNU43B 23680230 IC50 = 891250938.1 nM T97822 C8A9UV 23689693 IC50 = 562341325.2 nM T97822 CJ1Z9S 44315480 IC50 = 794328234.7 nM T97822 C7UG4F 44315519 IC50 = 15135612.48 nM T97822 C8FEV0 44319113 IC50 = 25000 nM T97822 C1ZH6U 90664380 IC50 > 100000 nM T97822 C5T4EQ 131801158 IC50 = 23 nM T97822 C6JF0E 135616214 IC50 = 2500 nM T97822 CH4YE6 135987613 IC50 > 10000 nM T97822 CFNO28 145950339 IC50 = 34 nM T97822 CG37FR 145950583 IC50 = 27 nM T97822 CCN16Y 145952805 IC50 = 44 nM T97822 C2FVO7 145953074 IC50 = 38 nM T97822 C19TPY 145958203 IC50 = 50 nM T97822 C1BLR8 145959460 IC50 = 33 nM T97822 CUXQ13 145971245 IC50 = 41 nM T97822 C8U9TX 145971276 IC50 = 28 nM T97822 D00GBX 71751 IC50 = 5.7 nM T97822 D01TOR 667555 IC50 = 50000 nM T97822 D05EMX 14076674 IC50 = 10000000 nM T97822 D06VWH 11758240 IC50 = 2 nM T97822 D08GOT 13752584 IC50 = 4897788.19 nM T97822 D09AUL 10266864 IC50 = 51000 nM T97822 D0EW3L 5281222 IC50 = 120000 nM T97822 D0M6UM 129265 IC50 = 22000 nM T97822 D0P1LP 7090 IC50 = 12000 nM T97822 D0U0YE 14762941 IC50 = 165958690.7 nM T97822 D0U2YL 131820 IC50 = 36000 nM T97822 D0U8YQ 921562 IC50 = 14000 nM T23673 D00STL 644241 IC50 = 1100 nM T23673 D05ROI 44462760 IC50 = 150 nM T23673 D09GDD 11167602 IC50 = 1.5 nM T23673 D0E6XR 3062316 IC50 = 164 nM T23673 D0R0MW 5329102 IC50 > 10000 nM T23673 D0W5HK 216239 IC50 = 3 nM T23673 D0Y9EW 42611257 IC50 = 48 nM T23673 D03AND 11656518 IC50 = 19 nM T23673 D04AHQ 71721540 IC50 = 42 nM T23673 D0B9BU 6918454 IC50 = 12 nM T23673 D0E3TC 44259 IC50 = 130 nM T23673 D0F5JZ 24180719 Ki = 3.3 nM T23673 D0M6BD 16719221 IC50 = 56 nM T23673 D0N8RV 9868037 IC50 = 41 nM T23673 D0T4QA 90456533 IC50 = 0.2 nM T23673 D03BNU 59604787 IC50 > 3500 nM T23673 D02YAQ 6603857 IC50 = 49000 nM T23673 D0A9KI 9863367 IC50 > 50 nM T23673 D0F8DL 176155 IC50 = 330 nM T23673 D0T3ME 156422 IC50 = 1400 nM T23673 CB37VR 5034 IC50 = 77 nM T23673 C1YNB7 447721 IC50 > 1000 nM T23673 C73DGZ 656907 IC50 > 1000 nM T23673 CXJ40G 667570 IC50 = 1300 nM T23673 C3OKI4 1228884 IC50 = 1300 nM T23673 C1SVD2 2132479 IC50 = 6500 nM T23673 CVE5C7 2807754 IC50 = 6800 nM T23673 CK2QF5 4163701 IC50 = 17000 nM T23673 C2N9KR 5353919 IC50 = 9 nM T23673 C3G5DZ 9797863 IC50 = 6700 nM T23673 C1A0GW 9798540 IC50 = 1100 nM T23673 CR6T9K 9800910 IC50 = 11000 nM T23673 CNJE78 9811391 IC50 = 1500 nM T23673 CJ7TP1 9818992 IC50 = 4000 nM T23673 C5TVQ1 9819877 IC50 = 230 nM T23673 C1F0PU 9819906 IC50 = 3100 nM T23673 CY52NF 9819987 IC50 = 1200 nM T23673 C8Y9EF 9820630 IC50 = 2000 nM T23673 C1E2DV 9826083 IC50 > 10000 nM T23673 CSQ85J 9827373 IC50 = 700 nM T23673 CP1KY2 9827920 IC50 = 100 nM T23673 C36KUT 9842995 IC50 = 6000 nM T23673 C8UY4X 9844334 IC50 = 6600 nM T23673 C65RQN 9849174 IC50 = 6 nM T23673 C41QWA 9857146 IC50 = 5800 nM T23673 C1W4JG 9872939 IC50 = 400 nM T23673 C45ENX 9883939 IC50 = 3000 nM T23673 CVW95E 9884589 IC50 = 4900 nM T23673 C9KO2G 9884742 IC50 = 7600 nM T23673 CSZ72R 9884877 IC50 = 3700 nM T23673 C18HKQ 9885748 IC50 = 24000 nM T23673 CJ4QV2 9885993 IC50 = 470 nM T23673 CXTE43 9905562 IC50 = 3000 nM T23673 CG47NJ 9906915 IC50 = 6000 nM T23673 C5GE7T 9917045 IC50 = 880 nM T23673 C24UQF 9927821 IC50 = 11000 nM T23673 C5NE6S 9928371 IC50 = 8000 nM T23673 CJT0A3 9929998 IC50 = 7700 nM T23673 C3V6WA 9930407 IC50 = 500 nM T23673 CQ64LI 9935852 IC50 = 695 nM T23673 C61KBJ 9943464 IC50 = 7200 nM T23673 C5ZVD1 9949990 IC50 = 5000 nM T23673 C60EDC 9950128 IC50 = 1700 nM T23673 CW2N9R 9950282 IC50 = 590 nM T23673 CI4BL2 9950385 IC50 = 120 nM T23673 C30RGW 9950906 IC50 = 11000 nM T23673 C3MSR9 9950907 IC50 = 8100 nM T23673 C48ITV 9951822 IC50 = 1900 nM T23673 C2W3AV 9995236 IC50 > 100000 nM T23673 C26QHZ 10005638 IC50 > 10000 nM T23673 CBL7Y0 10127660 IC50 = 53 nM T23673 C0SB5R 10128380 IC50 = 88 nM T23673 CO2E8Y 10128955 IC50 = 73 nM T23673 C30ULG 10128960 IC50 = 410 nM T23673 CABY28 10129238 IC50 = 160 nM T23673 C4V8FQ 10151557 IC50 = 13 nM T23673 C9ZN8M 10151709 IC50 = 61 nM T23673 CS89XI 10152022 IC50 = 300 nM T23673 CLY75M 10173949 IC50 = 130 nM T23673 C6MYH8 10175138 IC50 = 160 nM T23673 C50CXW 10195382 IC50 = 50 nM T23673 C25XBS 10195523 IC50 = 330 nM T23673 C52OSM 10195599 IC50 = 26 nM T23673 C6T3MD 10196590 IC50 = 70 nM T23673 C5E7HJ 10217017 IC50 = 1 nM T23673 C1E6OC 10217682 IC50 = 2300 nM T23673 CE31PD 10218746 IC50 = 210 nM T23673 CLV62C 10238782 IC50 = 460 nM T23673 C2TO8Y 10239830 IC50 = 82 nM T23673 C5WCZ2 10269141 IC50 = 20000 nM T23673 CKF79I 10289214 IC50 = 110 nM T23673 CY6UR3 10289414 IC50 = 100 nM T23673 C26OJV 10289677 IC50 = 150 nM T23673 C3I0MT 10289813 IC50 = 230 nM T23673 CMF93A 10293379 IC50 = 12000 nM T23673 C59HOA 10310634 IC50 = 130 nM T23673 CIO14B 10311595 IC50 = 27 nM T23673 CSAJ01 10311596 IC50 = 170 nM T23673 CZKA14 10311642 IC50 = 44 nM T23673 CSR83F 10311959 IC50 = 63 nM T23673 C17NJQ 10312001 IC50 = 140 nM T23673 CRIA28 10312314 IC50 = 60 nM T23673 CIS0N3 10323382 IC50 = 3500 nM T23673 CA8B5T 10390073 IC50 = 2100 nM T23673 CD47LT 10522840 IC50 = 2600 nM T23673 CN2TU0 10526792 IC50 = 1000 nM T23673 C9Q5ON 10546780 IC50 = 1400 nM T23673 CXN40D 10565927 IC50 = 380 nM T23673 CGSD37 10567785 IC50 = 135 nM T23673 C8E3NI 10568528 IC50 = 90 nM T23673 CFP95Y 10591281 IC50 = 750 nM T23673 CW1L8E 10591928 IC50 = 110 nM T23673 C2JVA6 10595034 IC50 = 20 nM T23673 CJ2O7T 10601190 IC50 = 4500 nM T23673 C16KBG 10637813 IC50 = 5000 nM T23673 C0QC5K 10638921 IC50 = 23 nM T23673 C46ERK 10639924 IC50 = 210 nM T23673 CLSA43 10663963 IC50 = 2100 nM T23673 CTA89W 10664281 IC50 = 610 nM T23673 CK4EW1 10664282 IC50 = 56 nM T23673 CD94OB 10665884 IC50 = 320 nM T23673 CWM72U 10666557 IC50 = 1600 nM T23673 C2UFM7 10711296 IC50 = 950 nM T23673 C1FZ3L 10757716 IC50 = 3000 nM T23673 C29ITE 10829679 IC50 = 86 nM T23673 CKZ95C 10829684 IC50 = 80 nM T23673 C81JVA 10833164 IC50 = 2500 nM T23673 CP6K0I 11155829 IC50 = 210 nM T23673 CSK2W9 11166166 IC50 = 580 nM T23673 CXC91Z 11167118 IC50 = 76 nM T23673 CT1K6D 11167921 IC50 = 180 nM T23673 CZKL03 11190042 IC50 = 120 nM T23673 CGS76Q 11224163 IC50 = 200 nM T23673 C2W5RC 11235063 IC50 > 30000 nM T23673 C6QLP2 11235672 IC50 = 110 nM T23673 C8YQ6T 11235899 IC50 = 170 nM T23673 CH73GV 11258258 IC50 = 480 nM T23673 C2XQC6 11259227 IC50 = 280 nM T23673 CJ69GI 11283035 IC50 = 80 nM T23673 CC1K4L 11294093 IC50 = 490 nM T23673 CQ8CM9 11305234 IC50 = 140 nM T23673 C72GHB 11318236 IC50 = 230 nM T23673 CNFT61 11364677 IC50 = 340 nM T23673 CD57AN 11373388 IC50 = 190 nM T23673 CV24KW 11407374 IC50 = 360 nM T23673 C8W5UG 11407870 IC50 = 250 nM T23673 CFHN02 11407902 IC50 = 340 nM T23673 COT0F6 11418292 IC50 = 480 nM T23673 CP0WH6 11419121 IC50 = 240 nM T23673 C0APW4 11422034 IC50 = 1200 nM T23673 CM3ZU2 11429946 IC50 = 320 nM T23673 CIQ9K8 11430708 IC50 = 550 nM T23673 CD2R4S 11430860 IC50 = 160 nM T23673 C8DA5W 11454055 IC50 = 250 nM T23673 CX7ZP1 11454895 IC50 = 450 nM T23673 CEKC20 11477628 IC50 = 230 nM T23673 CVT10K 11487778 IC50 = 810 nM T23673 CB6ME8 11503895 IC50 = 9 nM T23673 CRP2U5 11526671 Ki > 50000 nM T23673 CO9KP5 11583459 IC50 > 10000 nM T23673 C4U7HM 11621097 IC50 = 116 nM T23673 CU0E8O 11690457 Ki > 10000 nM T23673 C8JW5Z 11696578 IC50 = 38150 nM T23673 CB0AP2 11705863 Ki > 10000 nM T23673 CGI1D9 11717001 Ki = 0.54 nM T23673 CZY05V 11719421 IC50 = 68 nM T23673 C63CKJ 11750387 IC50 = 370 nM T23673 CH3JL9 11750681 IC50 = 190 nM T23673 CO09LN 11750815 IC50 = 260 nM T23673 C8L9ZM 11751978 IC50 = 200 nM T23673 CT8P5W 11775428 IC50 = 660 nM T23673 CIY7C5 12972078 IC50 = 18 nM T23673 C89WYZ 16038368 IC50 > 10000 nM T23673 CZK8V6 16043304 IC50 > 10000 nM T23673 C9TU1O 16046126 IC50 > 1000 nM T23673 C2FR4D 16049771 IC50 = 4 nM T23673 CKV4G1 16079040 IC50 = 1600 nM T23673 C2IF3P 16678352 IC50 = 180 nM T23673 C3IO1C 16679060 IC50 = 1700 nM T23673 C0H8UN 16730109 IC50 > 30000 nM T23673 C8G9AL 16756850 IC50 > 10000 nM T23673 C8M6LZ 17755310 IC50 = 19 nM T23673 CE14ZT 17941505 IC50 = 800 nM T23673 CAF63H 18322354 IC50 = 13000 nM T23673 C14YFA 21024387 IC50 = 170 nM T23673 C4AK5J 21037180 IC50 = 4 nM T23673 C9YR7W 21037208 IC50 = 18 nM T23673 C8ID6R 21037243 IC50 = 41 nM T23673 C2V1EQ 21037245 IC50 = 2 nM T23673 C9MTS8 21037247 IC50 = 9 nM T23673 C1TBC5 21037266 IC50 = 4 nM T23673 CZ23BW 21037364 IC50 = 9 nM T23673 C1CA7H 22040368 IC50 = 53 nM T23673 CG67FQ 22040397 IC50 = 12 nM T23673 CJ4E1M 22040403 IC50 = 780 nM T23673 CSJ67N 22040407 IC50 = 1 nM T23673 C8VJ3A 22040410 IC50 = 210 nM T23673 CHFO54 22040436 IC50 = 1 nM T23673 C19FQT 22040598 IC50 = 1 nM T23673 CJ3UH0 22040625 IC50 = 4 nM T23673 C02DQZ 22040627 IC50 = 20 nM T23673 CCA1D7 22040647 IC50 = 19 nM T23673 C4RP8N 22040656 IC50 = 15 nM T23673 CFK41E 22040722 IC50 = 120 nM T23673 C9A4LW 22040760 IC50 = 14 nM T23673 CSKZ32 22040783 IC50 = 150 nM T23673 CLX26F 22040796 IC50 = 110 nM T23673 CI3V6C 22040802 IC50 = 48 nM T23673 C9WU0J 22040805 IC50 = 490 nM T23673 CDN61H 22040847 IC50 = 10 nM T23673 C3SX8H 22040857 IC50 = 950 nM T23673 CJCL02 22040865 IC50 = 4 nM T23673 C6NM3T 22040925 IC50 = 28 nM T23673 CC84UT 22040937 IC50 = 150 nM T23673 CZM5W1 22040941 IC50 = 6 nM T23673 C30PJQ 22040960 IC50 = 7 nM T23673 CNI32B 22040966 IC50 = 2 nM T23673 C6FMB5 22040978 IC50 = 45 nM T23673 C9A1HQ 22041020 IC50 = 200 nM T23673 CKT6M2 22041042 IC50 = 7300 nM T23673 CM50PH 22041067 IC50 = 27 nM T23673 CRJ4H3 22041111 IC50 = 3500 nM T23673 CO37NP 22041112 IC50 = 1100 nM T23673 C4UMZ2 22041119 IC50 = 56 nM T23673 CI5KM3 22041171 IC50 = 9 nM T23673 C51FDU 22041175 IC50 = 8 nM T23673 CR3G0K 22041260 IC50 = 3 nM T23673 C69BSO 22041261 IC50 = 15 nM T23673 CU85MA 22041278 IC50 = 2 nM T23673 CGX61W 22041319 IC50 = 4 nM T23673 C7HUS0 23585267 IC50 = 28 nM T23673 CHQ23N 23585318 IC50 = 16 nM T23673 COSI68 23585320 IC50 = 11 nM T23673 CV9U8E 24745781 IC50 > 10000 nM T23673 C6JCE7 24753323 IC50 = 26 nM T23673 C50GZI 24753409 IC50 = 13 nM T23673 CC4RZ6 24753410 IC50 = 530 nM T23673 CB3D1Y 24753411 IC50 = 180 nM T23673 C6JF2R 24753412 IC50 = 5 nM T23673 CWX89I 24753603 IC50 = 220 nM T23673 C4CY3V 24753607 IC50 = 300 nM T23673 CQJ2D3 24753784 IC50 = 8 nM T23673 CP1E4R 24753786 IC50 = 32 nM T23673 CA3I4T 24753787 IC50 = 8 nM T23673 CW36DL 24753877 IC50 = 120 nM T23673 COAY09 24753878 IC50 = 23 nM T23673 C9H7EZ 24753971 IC50 = 1500 nM T23673 C6CT7I 24753973 IC50 = 63 nM T23673 CS98MR 24754053 IC50 = 6 nM T23673 C9Q3DE 24754054 IC50 = 4 nM T23673 CRJ9G6 24754132 IC50 = 4 nM T23673 CBD59Z 24754133 IC50 = 45 nM T23673 CKV76A 24754134 IC50 = 37 nM T23673 CM8HY9 24754207 IC50 = 3600 nM T23673 C7YG1N 24759534 IC50 = 630 nM T23673 CCS1U0 24862785 IC50 = 6 nM T23673 C6R4ZU 24863189 IC50 = 1520 nM T23673 CUIS63 24878671 IC50 = 6960 nM T23673 CBUG02 24879141 IC50 > 100000 nM T23673 C2F6KO 24879328 IC50 = 20260 nM T23673 C43HWQ 24883287 IC50 = 10000 nM T23673 C8DA5Q 24883334 IC50 = 10000 nM T23673 C13QYB 24884503 IC50 = 25 nM T23673 C5E1YD 24891645 IC50 = 5840 nM T23673 CY8L7E 24896769 IC50 > 10000 nM T23673 CJZE02 24963588 IC50 = 27 nM T23673 C3DI7Y 24995523 IC50 = 100 nM T23673 CS3Q8B 24995659 IC50 > 2000 nM T23673 CUJZ08 25059320 IC50 = 3200 nM T23673 C2ICS7 25065806 IC50 = 21 nM T23673 CA61PS 25066845 IC50 = 14 nM T23673 CR46MG 25066846 IC50 = 1 nM T23673 CF5AO8 25093353 IC50 > 10000 nM T23673 CAB5K2 25114576 IC50 = 870 nM T23673 C9PL5S 25137959 IC50 = 2000 nM T23673 CVJ0S5 25137960 IC50 = 10 nM T23673 C6FGQ1 25206346 IC50 = 23 nM T23673 CC71QJ 27666048 IC50 > 100000 nM T23673 CIJ56L 44142782 IC50 > 10000 nM T23673 CCFQ29 44187005 IC50 = 8.52 nM T23673 CR7K2T 44223999 Ki = 0.3 nM T23673 CJ75IB 44250343 IC50 = 120 nM T23673 CS2CK9 44250550 IC50 = 105 nM T23673 CLY1A3 44251218 IC50 = 200 nM T23673 C4O0CH 44272164 IC50 = 18000 nM T23673 CX28HG 44272165 IC50 = 18000 nM T23673 CNIJ29 44309757 IC50 > 10000 nM T23673 CH1TA5 44309758 IC50 = 570 nM T23673 C4P9ZA 44312235 IC50 = 29 nM T23673 CX57BA 44312236 IC50 = 40 nM T23673 C2D7RK 44312254 IC50 = 32 nM T23673 C8MF2U 44312272 IC50 = 65 nM T23673 C4XCW8 44312367 IC50 = 25 nM T23673 CGRP10 44312380 IC50 = 16 nM T23673 C2IC8R 44326529 IC50 = 15000 nM T23673 CT74PB 44326530 IC50 = 12000 nM T23673 C1W6BM 44326737 IC50 = 25000 nM T23673 CO0UF5 44326798 IC50 = 19000 nM T23673 C0E4TU 44326810 IC50 = 16000 nM T23673 C0GRN1 44326814 IC50 = 15000 nM T23673 CV37KZ 44326926 IC50 = 22000 nM T23673 C4ZD0E 44326936 IC50 = 20000 nM T23673 C0KD4U 44346053 IC50 = 8700 nM T23673 CO0FN8 44378490 IC50 = 130 nM T23673 CR1MV0 44378504 IC50 = 68 nM T23673 C4D5ZM 44378534 IC50 = 120 nM T23673 CI3W6L 44378535 IC50 = 38 nM T23673 C39PLZ 44378637 IC50 = 500 nM T23673 C9E7ID 44378798 IC50 = 270 nM T23673 C7HGZ5 44378800 IC50 = 460 nM T23673 CBGZ52 44378801 IC50 = 140 nM T23673 CIV90F 44378900 IC50 = 130 nM T23673 CI6T9Z 44378901 IC50 = 5800 nM T23673 C6CW1H 44378902 IC50 = 370 nM T23673 CJH86A 44385063 IC50 > 50000 nM T23673 CG46BQ 44386338 IC50 > 10000 nM T23673 CJTF35 44418481 IC50 = 100 nM T23673 CKV61A 44418488 IC50 = 630 nM T23673 CJ49OD 44418525 IC50 = 1000 nM T23673 C8LB9S 44418539 IC50 = 250 nM T23673 CO8X1V 44418540 IC50 = 158 nM T23673 C1IX6V 44418547 IC50 = 251 nM T23673 C4Q5UL 44418563 IC50 = 40 nM T23673 C8NZ9D 44418572 IC50 = 10 nM T23673 CJ3DL4 44418573 IC50 = 7 nM T23673 C10MKH 44448311 IC50 = 49 nM T23673 C1QN4V 44448333 IC50 = 41 nM T23673 CLQF97 44448334 IC50 = 26 nM T23673 C73THQ 44448354 IC50 = 5 nM T23673 C0DPU3 44448725 IC50 = 2 nM T23673 CFQN07 44448726 IC50 = 17 nM T23673 CR85LO 44448746 IC50 = 20 nM T23673 C5Y2JR 44448747 IC50 = 1 nM T23673 CA76JX 44448748 IC50 = 0.5 nM T23673 C9I0DU 44453753 IC50 = 6300 nM T23673 C2T7UV 44454440 IC50 = 8600 nM T23673 C0TN9Z 44454441 IC50 = 6300 nM T23673 C3P2TG 44454464 IC50 = 3500 nM T23673 CDN4M7 44565710 IC50 = 44 nM T23673 CB39SW 44565730 IC50 = 160 nM T23673 C13WTF 44565731 IC50 = 230 nM T23673 CEU40V 44565732 IC50 = 440 nM T23673 C6HEU1 44565743 IC50 = 2700 nM T23673 C5VL3A 44565744 IC50 = 4400 nM T23673 CI5M9V 44565745 IC50 = 500 nM T23673 CCD0E2 44565749 IC50 = 700 nM T23673 C4P7KM 44565750 IC50 = 820 nM T23673 CBZ1H2 44565751 IC50 = 1000 nM T23673 C39TYG 44565752 IC50 = 1100 nM T23673 C8QDY6 44565771 IC50 = 7500 nM T23673 CQAB41 44565772 IC50 = 10000 nM T23673 CUK3E8 44565773 IC50 = 650 nM T23673 CK24HZ 44565794 IC50 = 9500 nM T23673 CG0PL1 44565795 IC50 = 1400 nM T23673 C53FHZ 44565817 IC50 = 1500 nM T23673 C9VXN3 44578709 IC50 = 80 nM T23673 C3Y5AW 44589519 IC50 = 41 nM T23673 C09EWJ 44590206 IC50 = 17 nM T23673 CUA97D 46209401 IC50 = 1.4 nM T23673 C2P9QO 46228508 IC50 = 198 nM T23673 C6E5PY 46228822 IC50 = 126 nM T23673 C3T8AM 46228951 IC50 = 3 nM T23673 C4MKC5 46870033 IC50 = 11 nM T23673 C7LK1C 46945257 IC50 = 765 nM T23673 CHSF07 49806372 IC50 > 1000 nM T23673 C5ME3S 49806721 IC50 > 50000 nM T23673 CS7J8G 50937465 IC50 = 79 nM T23673 C2Q0GE 50990922 IC50 = 3000 nM T23673 C61DVY 50990961 IC50 = 2.2 nM T23673 CV3UP9 50992247 IC50 = 2.5 nM T23673 COVJ29 50994971 IC50 = 169 nM T23673 C5X9OM 51354603 IC50 = 10 nM T23673 C4DSG2 51354885 IC50 = 6.2 nM T23673 CQ85FC 51354886 IC50 = 110 nM T23673 C7MOQ0 51354887 IC50 = 70 nM T23673 C5KVT1 51355181 IC50 = 4.5 nM T23673 CS5F4Z 51355182 IC50 = 780 nM T23673 C4NFL7 51355183 IC50 = 3.3 nM T23673 C4W6PY 51355459 IC50 = 4.6 nM T23673 C95FWU 51355461 IC50 = 45 nM T23673 C4J3RE 51355733 IC50 = 6 nM T23673 CEQN27 52936621 Ki > 2000 nM T23673 CM24LF 52938983 IC50 = 2.87 nM T23673 CFR21J 52939107 IC50 = 22.41 nM T23673 CJQ31I 53239946 IC50 = 11 nM T23673 C7B3DE 53239955 IC50 = 13 nM T23673 C8UZE6 53239978 IC50 = 46 nM T23673 C1SKV3 53249125 IC50 = 1 nM T23673 C4CO1V 53317057 IC50 = 240.3 nM T23673 CE73CS 53323686 IC50 = 8319 nM T23673 CFP84X 53324920 IC50 = 1100 nM T23673 CD4H3S 53354074 Ki > 1000 nM T23673 CM7P3W 53357328 IC50 > 50000 nM T23673 CVG90B 53389651 IC50 > 10000 nM T23673 C89YCL 54580728 IC50 = 3 nM T23673 CA9I0J 54580729 IC50 = 4 nM T23673 C4X6DP 54581730 IC50 = 3 nM T23673 C2KHN1 54581731 IC50 = 1 nM T23673 CQ3U7M 54582720 IC50 = 140 nM T23673 C6ZR1A 54583026 IC50 = 530 nM T23673 CP7U4T 54584640 IC50 = 1 nM T23673 CC7T2A 56674921 IC50 = 170 nM T23673 CT4E8R 56832546 IC50 = 8500 nM T23673 CP58NG 56954518 IC50 = 930 nM T23673 CAK91L 56955954 IC50 = 206 nM T23673 C8LZ5B 56966054 IC50 = 10.6 nM T23673 CCE7J3 56966055 IC50 = 75.9 nM T23673 CP10UK 56966056 IC50 = 87.8 nM T23673 CMS50K 56966057 IC50 = 13.1 nM T23673 CRPT61 56966123 IC50 = 69.2 nM T23673 C6X0EZ 56966125 IC50 = 94.9 nM T23673 CLI12D 56966126 IC50 = 120.3 nM T23673 C9L4IJ 56966199 IC50 = 147.9 nM T23673 CTP30L 56966200 IC50 = 77.7 nM T23673 COA5X2 56966201 IC50 = 35.9 nM T23673 CIBO79 56966202 IC50 = 22.1 nM T23673 C2KDZ7 56966273 IC50 = 16.5 nM T23673 CGJ6F0 56966274 IC50 = 64.8 nM T23673 C48QKV 56966276 IC50 = 46.7 nM T23673 C4G7QD 57343225 IC50 = 73 nM T23673 CU4FW8 57397383 IC50 = 1600 nM T23673 C0BGR6 57399335 IC50 = 3 nM T23673 CZSM95 57412684 IC50 > 10000 nM T23673 CVK0G4 58056356 IC50 > 50000 nM T23673 CKB3A4 58102283 IC50 > 10000 nM T23673 CX1G3L 58102286 IC50 = 100 nM T23673 C1R8NM 59139106 IC50 = 78 nM T23673 CB34LP 59139113 IC50 = 120 nM T23673 CWK9I8 59139139 IC50 = 2500 nM T23673 CWN47R 59139154 IC50 = 70 nM T23673 CT0JG1 59139161 IC50 = 16 nM T23673 CP5GY6 59139172 IC50 = 81 nM T23673 CL4X3Z 59139185 IC50 = 70 nM T23673 C1PE3R 59139202 IC50 = 2400 nM T23673 CE82OV 59139228 IC50 = 1100 nM T23673 C3T5OF 59139235 IC50 = 56 nM T23673 CWO17Q 59139262 IC50 = 5 nM T23673 C5IYT0 59139264 IC50 = 25 nM T23673 C91SBH 59139388 IC50 = 830 nM T23673 C62EVK 59139472 IC50 > 50000 nM T23673 CT3EW2 59292007 IC50 > 1000 nM T23673 CXJ63M 59603829 IC50 = 560 nM T23673 CQEU96 59603842 IC50 = 48 nM T23673 C1MR8Q 60097495 IC50 > 10000 nM T23673 C9W0PE 60150671 IC50 = 75 nM T23673 C9NAL6 60152613 IC50 = 0.6 nM T23673 CSZA16 60155724 IC50 = 1814 nM T23673 CW3G6N 60196633 IC50 = 340 nM T23673 CUV14K 60196634 IC50 = 4300 nM T23673 CU32ED 60196737 IC50 = 175 nM T23673 CKB59I 60196738 IC50 > 10000 nM T23673 C40LVZ 60196740 IC50 > 10000 nM T23673 CV63UL 67240318 IC50 > 10000 nM T23673 CW17YX 68281294 IC50 = 1000 nM T23673 C5DGR9 69036886 IC50 = 4012 nM T23673 C4BT3M 69037249 IC50 = 2.9 nM T23673 CVBR46 70696651 IC50 = 81.5 nM T23673 CRX81Q 71575642 IC50 = 72 nM T23673 CT93OP 71682347 IC50 > 10000 nM T23673 C3NV9Q 71682348 IC50 > 10000 nM T23673 CN7M9G 71682349 IC50 = 293 nM T23673 C8KU4O 71682499 IC50 > 10000 nM T23673 C0XEQ1 71682500 IC50 = 30 nM T23673 CXSI14 71718330 IC50 > 100000 nM T23673 C1TM3P 71720141 IC50 > 100000 nM T23673 CU83YL 71730951 IC50 = 2.8 nM T23673 C7F3ZM 71736390 IC50 = 1.6 nM T23673 C9EM5X 71736552 IC50 = 6.7 nM T23673 CKYO24 71736864 IC50 = 5.6 nM T23673 CSVW76 72546488 IC50 = 570 nM T23673 C7HBR1 72546491 IC50 = 40 nM T23673 CXYT34 72546730 IC50 = 56 nM T23673 C1DAW5 72546731 IC50 = 50 nM T23673 C6R8DI 72943374 IC50 = 80 nM T23673 C80SEC 73504974 IC50 = 652 nM T23673 C3KVB2 73505180 IC50 = 92 nM T23673 CP4ZX2 76317169 IC50 = 120 nM T23673 C4DT2Z 76335375 IC50 = 55 nM T23673 CA5O6K 78325057 IC50 = 0.1 nM T23673 CCD78B 86295666 IC50 = 0.2 nM T23673 C2OGP3 86296699 IC50 = 0.2 nM T23673 C80LAH 86298305 EC50 = 200 nM T23673 CI2CG1 89670173 IC50 = 7 nM T23673 C1HW4B 89735655 IC50 = 950 nM T23673 C7TJR3 89814000 IC50 = 1.2 nM T23673 C4WP7D 89827799 IC50 = 7.2 nM T23673 CJE4A5 90407961 IC50 = 0.6 nM T23673 C9KN1H 90408121 EC50 = 52 nM T23673 CF45CE 90408582 IC50 = 0.4 nM T23673 C6RZ7J 90408826 EC50 = 20 nM T23673 CXZ6M2 90408889 EC50 = 76 nM T23673 C7QD9P 90409579 EC50 = 80 nM T23673 CU0GW5 90442604 IC50 = 0.8 nM T23673 CA2E5S 90456597 EC50 = 8 nM T23673 CW6S8P 90655795 IC50 > 50000 nM T23673 CNYK35 90655796 IC50 = 27000 nM T23673 CE4LR9 90655797 IC50 = 21 nM T23673 CWD4O3 90655989 IC50 > 50000 nM T23673 C26BSU 90666124 IC50 = 3200 nM T23673 CVQ1O6 90666126 IC50 = 286 nM T23673 C5AN9J 90666128 IC50 = 4300 nM T23673 CP76NE 90666130 IC50 > 50000 nM T23673 C85GHD 90666131 IC50 = 16500 nM T23673 CRP9I5 90666132 IC50 = 9200 nM T23673 CX1NV3 117609603 EC50 = 3960 nM T23673 CQ40CN 117609669 EC50 = 5 nM T23673 C5XEY9 117610044 EC50 = 64 nM T23673 C8E9JO 117610115 EC50 = 27 nM T23673 CG7QL4 118705925 IC50 = 8.79 nM T23673 C4AHL2 118711367 IC50 > 10000 nM T23673 CQCX41 118737057 IC50 = 27 nM T23673 C9KWP7 118870913 IC50 = 0.4 nM T23673 CSR81B 118887129 EC50 = 21 nM T23673 CV3MY8 118938835 IC50 = 0.1 nM T23673 CU52FB 118938855 IC50 = 0.1 nM T23673 C9NDH0 118938856 IC50 = 2 nM T23673 CTLH73 118938861 IC50 = 0.03 nM T23673 CL4MP3 118938866 IC50 = 6 nM T23673 C0UT7G 122177477 IC50 = 3.1 nM T23673 CSF49R 122177478 IC50 = 5.2 nM T23673 C5B6QT 122189918 IC50 = 44.8 nM T23673 C4X7SD 122192466 IC50 > 10000 nM T23673 CNX0Q2 122193763 IC50 > 10000 nM T23673 CWV0C3 122193764 IC50 = 4020 nM T23673 CSG98Y 122193765 IC50 > 10000 nM T23673 CCLQ75 122193769 IC50 = 6220 nM T23673 CXDR48 122193770 IC50 > 10000 nM T23673 CPA8C5 122193773 IC50 = 5840 nM T23673 CWM37L 123897305 IC50 = 71 nM T23673 CF5WH1 127039888 IC50 = 38600 nM T23673 CAG9K7 127046489 IC50 = 15 nM T23673 C6DP7Y 127047275 IC50 = 111 nM T23673 C3DVM9 127047276 IC50 = 566 nM T23673 CM81AR 127047922 IC50 = 695 nM T23673 CA2C3D 129010136 EC50 = 200 nM T23673 C0FM1R 130196825 IC50 = 27920 nM T23673 CR5P1D 132067922 IC50 = 0.6 nM T23673 CU1H0W 132497402 IC50 = 43.4 nM T23673 CZ81AL 134142029 IC50 = 0.024 nM T23673 C7PS8C 135271570 IC50 = 76 nM T23673 C8B5GZ 135513879 IC50 = 390 nM T23673 CGL3F1 135957036 IC50 = 50 nM T23673 C4REH9 135957052 IC50 = 76 nM T23673 C58FQY 135957053 IC50 = 156 nM T23673 CG9PJ7 135993841 IC50 = 960.9 nM T23673 CUA72Z 136042194 IC50 = 667.8 nM T23673 CL2D1A 136086817 IC50 = 146 nM T23673 CKG0N2 136086821 IC50 = 370 nM T23673 CH70WS 136086832 IC50 = 839 nM T23673 CG1R7B 136087060 IC50 = 6500 nM T23673 CRB3M4 136609929 IC50 = 2500 nM T23673 C0A9VE 136609930 IC50 = 1300 nM T23673 CW5YL0 136609931 IC50 > 50000 nM T23673 C3FC1W 137631894 IC50 = 7500 nM T23673 C7NFX9 137632089 IC50 = 8.5 nM T23673 C0Y1AW 137632207 IC50 = 150 nM T23673 C10BTW 137632556 IC50 > 10000 nM T23673 C2J9GO 137633617 IC50 > 10000 nM T23673 C7MD0H 137635615 IC50 = 28 nM T23673 CML76T 137635976 IC50 = 6200 nM T23673 CS9AW4 137636754 IC50 = 272 nM T23673 C08MHJ 137636777 IC50 = 0.7 nM T23673 CV3A5G 137637973 IC50 = 34.5 nM T23673 C7R0MS 137638615 IC50 = 2300 nM T23673 CE96AL 137639657 IC50 = 17300 nM T23673 CEPU59 137640849 IC50 = 220 nM T23673 CGR5B1 137642299 IC50 = 51 nM T23673 CA13KP 137642491 IC50 = 18.7 nM T23673 C26HIT 137643417 IC50 = 2100 nM T23673 CAT49C 137645403 IC50 = 374 nM T23673 CUES49 137646218 IC50 = 1800 nM T23673 CS6J8X 137646633 IC50 > 10000 nM T23673 C9Z6NB 137646838 IC50 = 770 nM T23673 CL8W4P 137647062 IC50 = 21.4 nM T23673 CGQ02E 137648059 IC50 = 6.3 nM T23673 C2HFR6 137648529 IC50 = 690 nM T23673 CL9HT1 137648599 IC50 = 21.9 nM T23673 CYR2I7 137649411 IC50 = 3050 nM T23673 C17GBS 137649678 IC50 = 1840 nM T23673 CEO70C 137650358 IC50 > 10000 nM T23673 CE7KF3 137650390 IC50 = 13.3 nM T23673 C4NM0R 137650776 IC50 = 1280 nM T23673 C3LAD6 137652990 IC50 > 100000 nM T23673 CL3P8Q 137653011 IC50 = 89 nM T23673 C5B9AM 137653362 IC50 = 860 nM T23673 C8K0OY 137655533 IC50 = 670 nM T23673 C3F8ZD 137656536 EC50 = 700 nM T23673 CMPJ36 137656808 IC50 = 14.4 nM T23673 C83XOY 137657177 IC50 = 53 nM T23673 CF7U5Y 137657487 IC50 > 10000 nM T23673 C3SD7B 137658277 IC50 = 4900 nM T23673 CVY3F0 137658568 IC50 = 1510 nM T23673 CJK81S 137659431 IC50 = 99 nM T23673 CNWY53 137659664 IC50 = 370 nM T23673 CUS48N 137659983 IC50 = 327 nM T23673 CA4V9R 137661906 IC50 = 100 nM T23673 COB9P2 141456067 IC50 = 7900 nM T23673 C6CN8H 142739455 IC50 = 61 nM T23673 CT25FH 145950796 IC50 = 8.5 nM T23673 C2I5WD 145979310 IC50 = 13.3 nM T23673 C6T4MU 145982183 IC50 = 40 nM T23673 CI1VH9 145985185 IC50 > 200000 nM T23673 CI7M2B 145988861 IC50 = 17.5 nM T23673 CNLH48 145988888 IC50 = 17600 nM T23673 CRT48W 145993502 IC50 = 3150 nM T23673 C2NKF8 155076930 IC50 = 182 nM T23673 CY1ZH2 155510358 IC50 = 336 nM T23673 CZ5S2M 155512875 IC50 = 2.7 nM T23673 C2MD1Q 155513187 IC50 > 10000 nM T23673 C0MZ9A 155513534 IC50 = 5160 nM T23673 CI54TD 155514548 IC50 = 1420 nM T23673 C2BA1L 155514841 IC50 = 1310 nM T23673 CX6SR0 155516442 IC50 = 420 nM T23673 CS31UH 155519078 IC50 = 1520 nM T23673 CU6Z5O 155520650 IC50 = 130 nM T23673 CP4JL5 155521754 IC50 = 4490 nM T23673 CVQ35F 155522102 IC50 = 3540 nM T23673 CM3DB7 155523430 IC50 = 480 nM T23673 CLY07C 155530863 IC50 = 450 nM T23673 CVQ24P 155532080 IC50 = 990 nM T23673 CS69CA 155532132 IC50 = 0.5 nM T23673 CJP67I 155535248 IC50 = 5320 nM T23673 C8ZF4H 155544511 IC50 = 3660 nM T23673 C8T0MQ 155544690 IC50 = 840 nM T23673 CJL37G 155544854 IC50 = 16400 nM T23673 CHE5F1 155553390 IC50 = 6260 nM T23673 CYC23K 155560669 IC50 = 110 nM T23673 C81JZW 155563388 IC50 = 410 nM T23673 C62CIM 155565320 IC50 = 420 nM T23673 CH3NO1 155566774 IC50 = 31.7 nM T23673 C0V2MU 135398506 Ki = 1.72 nM T23673 D00NWF 5730 IC50 = 70 nM T23673 D02XHC 448912 IC50 > 100000 nM T23673 D03MUZ 17759555 IC50 > 100000 nM T23673 D05UPS 44418518 IC50 = 398 nM T23673 D06WJA 9950176 IC50 = 1.4 nM T23673 D08LYB 5166 IC50 > 50 nM T23673 D0C0ZC 11676786 IC50 = 380 nM T23673 D0IR6U 5494425 IC50 > 10000 nM T23673 D0J4YA 9943465 IC50 > 12000 nM T23673 D0QN6U 9806182 IC50 = 810 nM T23673 D0V0QJ 389898 IC50 = 34500 nM T23673 D0Z5TQ 5924208 IC50 = 10.6 nM T48598 D05ROI 44462760 IC50 = 5880 nM T48598 D0Y9EW 42611257 IC50 = 16600 nM T48598 D04AHQ 71721540 IC50 = 150 nM T48598 CE2VX1 1381961 IC50 = 155000 nM T48598 C4K3AC 9870962 EC50 = 1065 nM T48598 C3MSB4 9954645 EC50 > 10000 nM T48598 C4BT3M 69037249 IC50 = 91 nM T48598 C3D6WC 71515468 IC50 = 200 nM T48598 CU83YL 71730951 IC50 = 48 nM T48598 C7F3ZM 71736390 IC50 = 46 nM T48598 C9EM5X 71736552 IC50 = 270 nM T48598 CKYO24 71736864 IC50 = 120 nM T48598 C2A4YP 86279165 Ki = 200000 nM T48598 C7TJR3 89814000 IC50 = 16 nM T48598 C4WP7D 89827799 IC50 = 160 nM T48598 CHJ6B8 90665836 IC50 = 1200 nM T48598 CFI02E 90665837 IC50 = 10000 nM T48598 CI6DB8 90665838 IC50 = 1800 nM T48598 C61RVL 90665839 IC50 = 10000 nM T48598 CW2UX9 90665840 IC50 = 10000 nM T48598 CDN49I 90665841 IC50 = 700 nM T48598 C0KI6U 90665842 IC50 = 1100 nM T48598 C0W7UI 90665843 IC50 = 2000 nM T48598 CYU7W2 90665844 IC50 = 2300 nM T48598 CEJ3D4 118019010 IC50 = 496 nM T48598 C0UT7G 122177477 IC50 = 57 nM T48598 CSF49R 122177478 IC50 = 120 nM T48598 CYP1B7 132145599 IC50 > 16000 nM T48598 CG7J5E 132162814 IC50 = 7600 nM T48598 CDWB35 132162815 IC50 > 16000 nM T48598 C1DW2E 132162816 IC50 > 16000 nM T48598 CJ1MY3 132162817 IC50 > 16000 nM T48598 C74FYN 132162819 IC50 > 16000 nM T48598 C2SIJ4 132162853 IC50 = 1900 nM T48598 CB80ZS 132163177 IC50 = 1500 nM T48598 C6CL4S 132163178 IC50 = 540 nM T48598 C3GPQ1 132163222 IC50 = 70 nM T48598 CULE35 135148667 IC50 = 8 nM T48598 C6DYW3 135148885 IC50 = 220 nM T48598 CU8T3N 136346978 Ki = 9 nM T48598 CC20EZ 136346980 Ki = 280 nM T48598 CY2L6T 136346989 Ki = 5000 nM T48598 CUG30Y 136347012 Ki > 25000 nM T48598 CS8YP7 137003167 IC50 = 939 nM T48598 CGS71A 137278705 IC50 = 51 nM T48598 CJ9N2K 137278711 IC50 = 68 nM T48598 C1HX7O 137278713 IC50 = 63 nM T48598 CK4MJ2 137278717 IC50 = 25 nM T48598 CA7GT6 137283289 Ki = 382 nM T48598 CS4W8U 137288869 IC50 = 69 nM T48598 C34DAC 137288870 IC50 = 36 nM T48598 CB42LP 137289789 Ki = 374 nM T48598 C0GNH8 137290307 Ki = 50000 nM T48598 CN2U1R 137290313 Ki = 8000 nM T48598 CX30GO 137290327 Ki = 2200 nM T48598 CW7Y3V 137292511 Ki = 15200 nM T48598 CXM3Y9 137297869 IC50 = 3330 nM T48598 C2XJN7 137297879 IC50 = 903 nM T48598 CRZH30 137297882 IC50 = 101 nM T48598 CBG13S 137297890 IC50 = 1800 nM T48598 C7BL0Z 137297899 IC50 = 7150 nM T48598 C1TWR9 137297909 IC50 = 20100 nM T48598 C85PEX 137297911 IC50 = 28 nM T48598 CS9D7J 137297914 IC50 = 3520 nM T48598 CTU65M 137297915 IC50 = 51 nM T48598 CJY69R 137297923 IC50 = 9150 nM T48598 CTO29V 137303087 Ki > 10000 nM T48598 C9SZ6B 137303128 Ki = 920 nM T48598 CVH3G7 137304434 Ki = 36000 nM T48598 C2LV5C 137304502 Ki = 5000 nM T48598 CV9Q5S 137314428 Ki = 380 nM T48598 CG7F2B 137314429 Ki > 20000 nM T48598 C8KFZ5 137316419 Ki = 2700 nM T48598 CQ7Z4X 137316471 Ki = 1600 nM T48598 C2M5GX 137317563 Ki = 3500 nM T48598 CJ07SA 137636907 IC50 = 50 nM T48598 CFA74W 137637303 IC50 = 64 nM T48598 C17EOK 137637743 IC50 = 1190 nM T48598 C7JU3W 137639238 IC50 = 35.8 nM T48598 CS93CA 137639750 IC50 = 1.6 nM T48598 CUS40W 137643713 IC50 = 59 nM T48598 CN4FM5 137645102 IC50 = 6.1 nM T48598 CK7S3H 137646089 IC50 = 1630 nM T48598 CFT25U 137647500 IC50 = 2.7 nM T48598 CM2XF3 137648559 IC50 = 426 nM T48598 C0UKF3 137648822 IC50 = 764 nM T48598 CP4V6Y 137650846 IC50 = 15400 nM T48598 CRF93P 137650861 IC50 = 19 nM T48598 CXO6C3 137652506 IC50 = 20600 nM T48598 CBIZ98 137653897 IC50 = 243 nM T48598 CLWD10 137660005 IC50 = 83 nM T48598 C78JQW 137661919 IC50 = 11 nM T48598 CKWQ13 138678754 IC50 < 5 nM T48598 CWM42J 138678756 IC50 = 18 nM T48598 C8S1AT 138678759 IC50 = 16 nM T48598 CA18QI 138678764 IC50 = 70 nM T48598 C9J3EN 138678770 IC50 = 132 nM T48598 C6SPK8 138678774 IC50 = 387 nM T48598 C7EV3T 138678780 IC50 = 610 nM T48598 CE7Q0H 138678786 IC50 = 97 nM T48598 C92HTX 138678788 IC50 = 81 nM T48598 C27KFX 138678799 IC50 = 150 nM T48598 C30MEF 138678890 IC50 = 211 nM T48598 C2DOL1 138679046 IC50 = 52 nM T48598 CR5A6H 139388519 IC50 = 780 nM T48598 CYRW58 139388529 IC50 = 4860 nM T48598 C5GLR3 139388566 IC50 = 169 nM T48598 CG1MO4 139388571 IC50 = 116 nM T48598 CNVK52 139388599 IC50 = 129 nM T48598 CXB0Y3 139388605 IC50 = 214 nM T48598 C8CRF6 139600305 IC50 = 115 nM T48598 CEL25S 140956840 IC50 = 11 nM T48598 C0NV4K 140956861 IC50 = 66 nM T48598 C1SJI0 142468965 IC50 = 18 nM T48598 CB29ZR 142468976 IC50 = 12 nM T48598 C9PC5N 142468998 IC50 = 12 nM T48598 C6S0VF 142469011 IC50 = 21 nM T48598 C3PD0Y 142469055 IC50 = 32 nM T48598 C7X6QM 142469058 IC50 = 97 nM T48598 CUW9Y5 146234885 IC50 = 128 nM T48598 CN08TQ 146234893 IC50 = 25 nM T48598 CB30HO 146235053 IC50 = 80 nM T48598 C2B5VH 146235304 IC50 = 47 nM T48598 CKM1C3 146235420 IC50 = 90 nM T48598 C5QBX0 146235429 IC50 = 53 nM T48598 C91ANQ 146235452 IC50 = 142 nM T48598 CAVJ61 146235508 IC50 = 34 nM T48598 CFKC35 146235592 IC50 = 164 nM T48598 C3HCA7 146235786 IC50 = 65 nM T48598 C89YKH 146235843 IC50 = 38 nM T48598 C5KX3F 146235857 IC50 = 306 nM T48598 C42CDB 146235944 IC50 = 53 nM T48598 CQW98L 146236007 IC50 = 146 nM T48598 C76QJC 146236012 IC50 = 56 nM T48598 C06VPI 146254335 IC50 = 109 nM T48598 C0U1KX 146254417 IC50 = 442 nM T48598 CZ7P4M 146254588 IC50 = 25 nM T48598 C3S5WI 146461338 IC50 = 29 nM T48598 CBI9U1 146585881 IC50 = 109 nM T48598 C1EFX9 146585884 IC50 = 683 nM T48598 C3H9BP 146585895 IC50 = 139 nM T48598 C1VJ4L 146630440 IC50 = 17900 nM T48598 C6S1IB 146630461 IC50 = 2120 nM T48598 C9I2WV 146630653 IC50 > 250000 nM T48598 C4IA5T 146630666 IC50 = 299 nM T48598 C51IYS 146630676 IC50 = 638 nM T48598 CW34ZK 146630683 IC50 = 1370 nM T48598 CVL6A5 146630701 IC50 = 4260 nM T48598 C4QH7U 146630731 IC50 = 6630 nM T48598 C0WAB5 146630732 IC50 = 14200 nM T48598 CYH28N 146630894 IC50 = 369 nM T48598 C5IV8H 146630905 IC50 = 1290 nM T48598 CIX1C8 146630907 IC50 = 174 nM T48598 CNK71Q 146631214 IC50 = 1270 nM T48598 C8H9TW 155523678 IC50 = 73 nM T48598 CBR9O0 155524545 IC50 = 4342 nM T48598 CVQ3H7 155528727 IC50 = 7653 nM T48598 C7Y3FZ 155549278 IC50 = 627 nM T48598 CMA86J 155564813 IC50 = 2780 nM T58093 D0S7BQ 52918384 IC50 = 12 nM T58093 D0T2IQ 443600 IC50 = 20 nM T58093 C8A6FD 9849925 IC50 = 30 nM T58093 C04KRJ 16034963 IC50 = 2.5 nM T58093 CJ42NE 16034968 IC50 = 0.52 nM T58093 CEYX96 16035081 IC50 = 0.93 nM T58093 CH97SC 16035085 IC50 = 2.1 nM T58093 CTC5O9 16035087 IC50 = 1.4 nM T58093 C4OQ3K 16035189 IC50 = 1.4 nM T58093 CG83UV 16035293 IC50 = 3.8 nM T58093 CGN4W5 16035295 IC50 = 3.2 nM T58093 CSFC45 16035507 IC50 = 2.2 nM T58093 CNTW74 16035824 IC50 = 12 nM T58093 CCDG98 16035825 IC50 = 5.2 nM T58093 CZC1T5 16035827 IC50 = 8 nM T58093 C48ARB 16036037 IC50 = 4.5 nM T58093 C1SMZ2 16036156 IC50 = 2.2 nM T58093 CP3H6M 16036157 IC50 = 4.4 nM T58093 C9YZ6I 16036158 IC50 = 1.4 nM T58093 C2I1YX 16036160 IC50 = 1.5 nM T58093 C3ZIH1 16036281 IC50 = 2.4 nM T58093 C5SOI2 16036282 IC50 = 3.4 nM T58093 C7JG1B 16036394 IC50 = 10 nM T58093 C3NWE9 16036395 IC50 = 2 nM T58093 CW16UL 16036656 IC50 = 5 nM T58093 C2VOZ5 16036657 IC50 = 4 nM T58093 C3IU1P 16036659 IC50 = 2 nM T58093 C9SHM6 16036661 IC50 = 3.7 nM T58093 CMOB46 16046174 IC50 = 7500 nM T58093 C7WH3R 25123230 IC50 = 30 nM T58093 CV15JQ 25123888 IC50 = 30 nM T58093 CFD1Z5 57345646 IC50 = 35800 nM T58093 C4GTE0 57345647 IC50 = 100100 nM T58093 CO8R3H 57878092 IC50 = 5 nM T58093 C0HY5X 57878097 IC50 = 2.3 nM T58093 C3W6PE 57878101 IC50 = 10 nM T58093 C2GJ1F 57878102 IC50 = 1.7 nM T58093 CX9UE4 57878122 IC50 = 1.6 nM T58093 C2F9SP 57878124 IC50 = 1.4 nM T58093 CH48QS 57878125 IC50 = 1.2 nM T58093 C5UJ7H 57878129 IC50 = 0.9 nM T58093 CU2KR4 57878131 IC50 = 1.7 nM T58093 C0WIY3 57878141 IC50 = 0.86 nM T58093 C1R5WU 57878145 IC50 = 1 nM T58093 C3XHZ9 70681653 IC50 = 1.3 nM T58093 C0C5BI 70685926 IC50 = 3.3 nM T58093 CMH5K3 70692221 IC50 = 2.3 nM T58093 C5SH2R 70694300 IC50 = 5.9 nM T58093 C5W1AK 138454269 IC50 = 2 nM T58093 CZUO38 155511087 IC50 = 2 nM T58093 C9F6LQ 155511457 IC50 = 5 nM T58093 C5DKE6 155511474 IC50 = 16 nM T58093 C45DSK 155512893 IC50 = 6 nM T58093 C6BQA2 155514815 IC50 = 11 nM T58093 CD58RH 155518934 IC50 = 5 nM T58093 C3WQH0 155520436 IC50 = 2 nM T58093 C0P4AY 155523706 IC50 = 10 nM T58093 CX3FD5 155526303 IC50 = 1 nM T58093 CEU4S5 155526689 IC50 = 0.63 nM T58093 CV3SG0 155529612 IC50 = 1 nM T58093 CJL2C8 155535353 IC50 = 18 nM T58093 CF5T2J 155536889 IC50 = 158 nM T58093 C7D4BJ 155541590 IC50 = 2 nM T58093 CL5AO7 155553287 IC50 = 20 nM T58093 CQF91W 155554205 IC50 = 3 nM T58093 CB1SN4 155557831 IC50 = 2 nM T58093 C94TBM 155560644 IC50 = 2 nM T58093 C4AD6J 155563341 IC50 = 1 nM T20600 D0J3SU 9847835 EC50 > 5000 nM T20600 C3T8NF 5288850 IC50 > 5000 nM T20600 C1KR5B 5327301 Ki = 22000 nM T20600 C37TKL 5327302 Ki = 1000 nM T20600 C64ZMN 5327304 Ki = 1400 nM T20600 C3IZ2W 5327307 Ki = 2300 nM T20600 C16DTL 5327308 Ki = 540 nM T20600 C4O3QY 5327309 Ki = 9700 nM T20600 C3GUM7 5327310 Ki = 2400 nM T20600 C3LZX9 8027611 IC50 > 20000 nM T20600 CFN2P6 9800285 Ki = 7500 nM T20600 CLTO67 9821317 IC50 = 18 nM T20600 C4XO3K 9821545 IC50 > 5000 nM T20600 CJI5T3 9823027 IC50 = 37 nM T20600 C74QTI 9823074 IC50 = 940 nM T20600 C6S3KT 9840223 Ki > 25000 nM T20600 CD05OL 9867192 IC50 = 1500 nM T20600 C2DMG1 9914167 IC50 > 5000 nM T20600 C9CV0Y 10001828 IC50 = 940 nM T20600 CX67SZ 10826725 Ki = 1000 nM T20600 CDX7A4 10963183 Ki = 190 nM T20600 CM8O6L 11257152 IC50 = 50 nM T20600 C4F8DC 11444079 IC50 > 500000 nM T20600 CDT9G3 11467504 IC50 = 3.44 nM T20600 CV4CP9 11496333 IC50 > 5000 nM T20600 CGE2J0 11497112 IC50 > 5000 nM T20600 C6IS9K 11509289 IC50 > 5000 nM T20600 C6L2MY 11509300 IC50 > 5000 nM T20600 CC31QO 11509301 IC50 > 5000 nM T20600 CS8OX7 11510566 IC50 > 500000 nM T20600 C7FY9B 11512139 IC50 > 5000 nM T20600 C15VFG 11515586 IC50 > 500000 nM T20600 CW6PC0 11519268 IC50 > 5000 nM T20600 CZC5D9 11525874 IC50 > 5000 nM T20600 C5BNE1 11533326 IC50 > 5000 nM T20600 CDK3Z5 11533935 IC50 = 3700 nM T20600 C4IC7E 11541867 IC50 > 500000 nM T20600 C3USR9 11543714 IC50 = 283 nM T20600 C3P2GZ 11548424 IC50 > 500000 nM T20600 CVX4M6 11548909 EC50 > 5000 nM T20600 C17OJS 11572844 IC50 = 201 nM T20600 CF0V3P 11576540 IC50 > 5000 nM T20600 C1T9DY 11576622 IC50 > 5000 nM T20600 C03KPR 11576852 EC50 > 5000 nM T20600 CN67DR 11583840 IC50 > 5000 nM T20600 CPD0M8 11584106 IC50 > 5000 nM T20600 CL16IM 11591540 IC50 > 5000 nM T20600 CE2TX6 11591919 IC50 > 500000 nM T20600 CG4Z9A 11598106 IC50 > 10000 nM T20600 CV6MF1 11614728 IC50 > 500000 nM T20600 CFP19E 11619968 IC50 > 5000 nM T20600 CA0LH6 11624920 IC50 > 5000 nM T20600 CEY39D 11628992 IC50 > 500000 nM T20600 C6UAV3 11632008 IC50 = 216 nM T20600 C6Y5MG 11634372 IC50 > 5000 nM T20600 CKJE92 11634649 IC50 > 5000 nM T20600 C91JNO 11639020 IC50 = 124 nM T20600 C4MCW2 11646889 IC50 = 137 nM T20600 C2KFU3 11647018 IC50 > 5000 nM T20600 CH20JE 11652994 IC50 = 2850 nM T20600 CN32TX 11664423 IC50 > 500000 nM T20600 CUD05C 11670894 IC50 > 5000 nM T20600 CX97NT 11684618 IC50 > 5000 nM T20600 C05YRV 11699954 IC50 > 500000 nM T20600 CKEX64 11700402 IC50 > 500000 nM T20600 C89COT 11705942 IC50 > 5000 nM T20600 C86PAH 11712912 IC50 > 5000 nM T20600 CXH9M5 16749067 IC50 = 407 nM T20600 C2DJ5W 16749068 IC50 = 9550 nM T20600 COM07G 16749069 IC50 = 698 nM T20600 CPG8Q0 16749161 IC50 = 744 nM T20600 CG84TK 16749162 IC50 = 823 nM T20600 CT3HD1 16749163 IC50 = 650 nM T20600 CZM4X2 16749164 IC50 = 610 nM T20600 CUZ8N4 16749267 IC50 = 8900 nM T20600 CMEK96 16749268 IC50 = 5025 nM T20600 C01HBN 16749269 IC50 = 918 nM T20600 CWG3C8 16749270 IC50 = 840 nM T20600 C8R3GD 16749271 IC50 = 515 nM T20600 CTI80F 25178948 EC50 > 5000 nM T20600 C2GI4J 25178949 EC50 > 5000 nM T20600 CQ2GM9 25178950 EC50 > 5000 nM T20600 C4GFV6 25179140 EC50 > 5000 nM T20600 CYL36B 25179141 IC50 = 4425 nM T20600 CGC69Q 25179143 EC50 > 5000 nM T20600 C27YJF 25179144 IC50 = 9967 nM T20600 C2YTB7 25179145 EC50 > 5000 nM T20600 C6GTV3 25179324 EC50 > 5000 nM T20600 CIC46T 25179513 EC50 > 5000 nM T20600 CK96WB 25179514 EC50 > 5000 nM T20600 CGX78D 25217029 IC50 = 450 nM T20600 CW2L9Q 25217030 IC50 = 770 nM T20600 C8UTC4 25217031 IC50 = 509 nM T20600 CZ43KQ 25217032 IC50 = 927 nM T20600 C2P9NI 25217145 IC50 = 4930 nM T20600 C8C9XU 42618276 IC50 > 15000 nM T20600 CFO93N 42618277 IC50 = 12833 nM T20600 CS1KQ0 42618278 IC50 = 325 nM T20600 CVI16X 42618279 IC50 = 545 nM T20600 C3MRA0 42618280 IC50 = 568 nM T20600 C8UO9S 42618281 IC50 = 425 nM T20600 C68NPR 42618282 IC50 = 453 nM T20600 CL41SD 42618283 IC50 = 591.7 nM T20600 CJ7U2E 42618284 IC50 = 151 nM T20600 CZL8C7 42618285 IC50 = 188 nM T20600 CNIQ28 42618286 IC50 = 230 nM T20600 C91OMB 42618287 IC50 = 9833 nM T20600 C5AC1L 42618288 IC50 = 156 nM T20600 CFU5T2 42618289 IC50 = 197 nM T20600 CK9H3M 42618290 IC50 = 280 nM T20600 CV4H2J 42618291 IC50 = 241 nM T20600 C7VPU3 42618292 IC50 = 358 nM T20600 C6R2FM 42618293 IC50 = 468 nM T20600 CT7VO2 44157085 IC50 > 500000 nM T20600 CWMU91 44157086 IC50 > 500000 nM T20600 C6LZ5Y 44157087 IC50 > 500000 nM T20600 CYSJ79 44157089 IC50 > 500000 nM T20600 CMX7W1 44157090 IC50 > 500000 nM T20600 C7B3VE 44158086 IC50 > 500000 nM T20600 C20WEJ 44158089 IC50 > 500000 nM T20600 C68KOD 44158154 IC50 > 500000 nM T20600 C4C1RU 44158155 IC50 > 500000 nM T20600 CN1YR9 44158157 IC50 > 500000 nM T20600 C80XPD 44158237 IC50 > 500000 nM T20600 CN09UV 44158238 IC50 > 500000 nM T20600 CT9DF4 44158240 IC50 > 500000 nM T20600 CHDF62 44158242 IC50 > 500000 nM T20600 CS6X1C 44158325 IC50 > 500000 nM T20600 C17TEZ 44158326 IC50 > 500000 nM T20600 CZ0VT3 44158328 IC50 > 500000 nM T20600 CD8WB9 44304162 Ki = 57000 nM T20600 CAB39E 44331552 IC50 = 32400 nM T20600 CE0FW4 44331565 IC50 = 21400 nM T20600 C8SZN9 44331566 IC50 = 12000 nM T20600 CMFW61 44331567 IC50 = 22600 nM T20600 CHYL38 44331577 IC50 = 1620 nM T20600 C1I9QH 44331578 IC50 = 18900 nM T20600 C4VGZ1 44331579 IC50 = 10100 nM T20600 CRZ01H 44331580 IC50 = 20500 nM T20600 CFOR90 44331674 IC50 = 14500 nM T20600 CK7VI8 44331675 IC50 = 717 nM T20600 CH7GS4 44331676 IC50 > 50000 nM T20600 C4FOD3 44331693 IC50 > 50000 nM T20600 CJY5L2 44331739 IC50 = 28600 nM T20600 C8N2GQ 44331740 IC50 = 11800 nM T20600 CW9K4Q 44331815 IC50 = 3370 nM T20600 CT76DG 44331816 IC50 = 33400 nM T20600 CC70GF 44331830 IC50 = 2530 nM T20600 CNJ19L 44331876 IC50 = 11110 nM T20600 C46IPA 44331879 IC50 > 10000 nM T20600 CP0Y8M 44331898 IC50 = 10 nM T20600 CF3R6W 44331908 IC50 > 10000 nM T20600 CTM5W1 44331914 IC50 = 3.5 nM T20600 C0YZ9O 44331915 IC50 = 15 nM T20600 C4NK1S 44331942 IC50 = 10 nM T20600 CXKY19 44331943 IC50 = 18560 nM T20600 C3FC8D 44331944 IC50 > 10000 nM T20600 CH1ZF2 44331953 IC50 = 589 nM T20600 C0QJ8V 44331957 IC50 = 4600 nM T20600 C1HBX6 44331963 IC50 = 14030 nM T20600 C7UXK5 44331964 IC50 = 10000 nM T20600 C42PGN 44331965 IC50 = 308 nM T20600 C5J7KX 44331966 IC50 > 50000 nM T20600 CG83FS 44331967 IC50 = 12500 nM T20600 CGAJ95 44331977 IC50 = 3610 nM T20600 CCYX84 44331980 IC50 > 10000 nM T20600 C5UIO2 44331987 IC50 = 32500 nM T20600 C0PM5C 44332004 IC50 = 4180 nM T20600 C4ENB1 44332005 IC50 = 1010 nM T20600 CFK4Z1 44332024 IC50 = 1280 nM T20600 CTM3G2 44332026 IC50 = 2720 nM T20600 C48ZEW 44332028 IC50 > 50000 nM T20600 C30MKG 44332029 IC50 > 50000 nM T20600 C7OS9X 44332050 IC50 = 9750 nM T20600 C9Y6NP 44332051 IC50 = 5050 nM T20600 C0VGF8 44332058 IC50 = 5860 nM T20600 CQU84D 44332068 IC50 = 21200 nM T20600 CBL91D 44332078 IC50 = 51200 nM T20600 C4VCM3 44332093 IC50 = 5900 nM T20600 C92QVT 44332108 IC50 = 1430 nM T20600 CQLZ09 44332109 IC50 = 13800 nM T20600 C4CUL6 44332112 IC50 = 3030 nM T20600 CN2YM6 44332113 IC50 = 1900 nM T20600 C4CY8K 44332118 IC50 = 7000 nM T20600 CXZ2N1 44332120 IC50 = 42700 nM T20600 CD56PK 44332121 IC50 > 50000 nM T20600 C5A6OJ 44332128 IC50 = 14500 nM T20600 C6IZ2R 44332129 IC50 = 3160 nM T20600 C5DY0G 44332136 IC50 = 1430 nM T20600 CQ1K9H 44332311 IC50 = 37 nM T20600 C9LOS2 44332330 IC50 = 305 nM T20600 C2U6GB 44332331 IC50 = 10300 nM T20600 CH01QW 44332332 IC50 = 11800 nM T20600 C8D5TB 44364680 Ki = 120 nM T20600 CJ6QG4 44417479 IC50 > 500000 nM T20600 C7RX9I 44418960 Ki = 550000 nM T20600 CXR1V5 44434249 IC50 = 61 nM T20600 C8Z4WO 44459967 IC50 = 5128.61 nM T20600 C86ORE 44459987 IC50 = 3548.13 nM T20600 CDY2W5 49796910 IC50 = 1.7 nM T20600 C3M2BW 52918163 IC50 = 8700 nM T20600 CF24IM 52918177 IC50 = 6900 nM T20600 CR9I7F 52918178 IC50 = 13450 nM T20600 C2VPU1 52918179 IC50 = 7750 nM T20600 C8Z2TQ 54580470 IC50 > 10000 nM T20600 CMU0B4 54581481 IC50 > 10000 nM T20600 CCS8Y3 54581987 IC50 = 1165 nM T20600 CJEP38 54582484 IC50 = 7666 nM T20600 C61NWL 54582924 IC50 = 9125 nM T20600 CO0AG3 54583923 IC50 = 747 nM T20600 CI2DL4 54583924 IC50 = 3475 nM T20600 CV2WU1 54583925 IC50 = 4700 nM T20600 CXA51D 54584867 IC50 = 6950 nM T20600 C8YSL0 54585834 IC50 = 1012 nM T20600 C9B5OF 54586343 IC50 = 2987 nM T20600 C7A8ER 54587376 IC50 = 9200 nM T20600 CGY3W2 71471109 IC50 > 100000 nM T20600 CKZ2H0 71582971 IC50 > 500000 nM T20600 C4WJ5F 71582972 IC50 > 500000 nM T20600 CXA62J 71582973 IC50 = 1030 nM T20600 CNZS31 71582974 IC50 > 500000 nM T20600 CE4L9D 71582975 IC50 > 500000 nM T20600 CXMS80 71583078 IC50 > 500000 nM T20600 C30UIL 71583079 IC50 > 500000 nM T20600 CJBC14 71583080 IC50 = 2610 nM T20600 C57MOP 71583081 IC50 > 500000 nM T20600 CS0YK9 71583082 IC50 > 500000 nM T20600 C3UTO9 71583083 IC50 > 500000 nM T20600 CW1R5Q 71583084 IC50 > 500000 nM T20600 CR57LS 71583192 IC50 > 500000 nM T20600 C8B3NZ 71583193 IC50 > 500000 nM T20600 CB6DY7 71583194 IC50 > 500000 nM T20600 CANH70 71716242 IC50 > 100000 nM T20600 C40WIR 71718085 IC50 = 100000 nM T20600 CU75VK 71719897 IC50 = 600 nM T20600 CBV6F1 71720507 IC50 > 100000 nM T20600 C4U5TO 76311196 IC50 > 10000 nM T20600 CSI53E 76311200 IC50 > 10000 nM T20600 CNOL37 76311201 IC50 = 3878 nM T20600 C8IS5Q 76314800 IC50 = 5082 nM T20600 CK41QI 76314804 IC50 > 10000 nM T20600 CHS61N 76314805 IC50 > 10000 nM T20600 CDY7K0 76318413 IC50 = 3790 nM T20600 CB2N6G 76322078 IC50 > 10000 nM T20600 C8SPW6 76322082 IC50 > 10000 nM T20600 CC2EP6 76325698 IC50 > 10000 nM T20600 CFY79U 76332916 IC50 > 10000 nM T20600 CD35SI 76332917 IC50 > 10000 nM T20600 C3FQX0 76336535 IC50 > 10000 nM T20600 CV4PE6 76336536 IC50 > 10000 nM T20600 CKCI60 90663142 IC50 = 310 nM T20600 C3GPO7 118723314 IC50 = 500000 nM T20600 C8H0EL 118723315 IC50 = 28500 nM T20600 CTE1O2 118723316 IC50 = 500000 nM T20600 CE8O9P 118723317 IC50 = 500000 nM T20600 C48DEF 118723325 IC50 = 500000 nM T20600 C67QMY 118723326 IC50 = 500000 nM T20600 CCJ27M 118723327 IC50 = 500000 nM T20600 COG92V 118723328 IC50 = 500000 nM T20600 CSX85P 118723329 IC50 = 500000 nM T20600 CICB42 118723330 IC50 = 78900 nM T20600 C13BRQ 118723331 IC50 = 12900 nM T20600 CWM2E8 133081971 IC50 > 9999 nM T20600 D08ORM 15487887 IC50 = 8 nM T20600 D0N5MU 4117381 Ki > 50000 nM T20600 D0Q9XX 515950 Ki = 1700 nM T20600 D0V6DX 10640 IC50 = 474 nM T20600 D0Y5IQ 44255320 IC50 = 5000 nM T28330 D04JEE 4946 EC50 > 5011.87 nM T28330 D0H7FW 9870520 Ki = 28.84 nM T28330 D0LI1C 44469321 IC50 > 30000 nM T28330 D01ZXW 122077 IC50 = 0.5623 nM T28330 D0C8ZD 121964 IC50 = 1900 nM T28330 D0EG1F 9914672 Ki = 79.43 nM T28330 D0F6CT 51353551 EC50 = 0.0024 nM T28330 D0W8TS 9898185 IC50 = 3162.28 nM T28330 D0W9ZY 52949124 EC50 = 0.5248 nM T28330 D0XJ0S 108187 IC50 = 1047.13 nM T28330 C7YKF2 1098327 Ki < 10000 nM T28330 CR7Y4G 1109919 Ki > 10000 nM T28330 CA0XN1 3081599 EC50 = 28 nM T28330 CF74HA 6918156 IC50 = 0.5 nM T28330 C6E0TB 9832467 Ki < 10000 nM T28330 C07OFK 9892971 IC50 > 10000 nM T28330 C57IBS 9913081 Ki < 10000 nM T28330 CRT68S 9960432 Ki = 125.89 nM T28330 CKTR60 10008654 IC50 = 5.2 nM T28330 CV56TJ 10031013 IC50 = 75.86 nM T28330 CD7XO3 10032955 EC50 = 3.162 nM T28330 C7SQA8 10032956 IC50 = 229.09 nM T28330 CDT69G 10051431 IC50 = 440 nM T28330 CFO8L6 10071178 Ki = 31.62 nM T28330 CL8M2B 10320262 Ki = 25.12 nM T28330 C16YAW 10343558 Ki = 25.12 nM T28330 CM1D3V 10350069 IC50 = 724.44 nM T28330 C4DIK2 10366068 Ki = 25.12 nM T28330 CD6B7H 10373077 EC50 = 3.981 nM T28330 CTE7N2 10388627 Ki = 25.12 nM T28330 CA5B8O 10391834 IC50 = 1584.89 nM T28330 CYU58T 10415786 IC50 = 39.81 nM T28330 C5Z8IP 10433726 Ki = 25.12 nM T28330 CM97BA 10460632 Ki = 3006 nM T28330 CB1X4K 10483574 IC50 = 79.43 nM T28330 CVE86S 10507071 IC50 = 6850 nM T28330 C91ZVY 10507109 Ki = 50.12 nM T28330 C36HIS 10507561 IC50 = 15.85 nM T28330 CKY68B 10509945 EC50 = 9.12 nM T28330 C1AE8J 10531224 IC50 = 1318.26 nM T28330 C9SUK0 10531430 IC50 = 1584.89 nM T28330 C4S2YR 10555164 IC50 = 138.04 nM T28330 CJZ47Q 10555363 IC50 = 36.31 nM T28330 CRI50M 10555571 IC50 = 42.66 nM T28330 CIN1C4 10555804 IC50 = 13.8 nM T28330 CM7LP6 10556460 IC50 = 309.03 nM T28330 C6LR2W 10580108 IC50 = 389.05 nM T28330 C0IT5X 10603713 IC50 = 17.38 nM T28330 CBRX06 10603714 IC50 = 20.89 nM T28330 C0AV6Q 10626596 IC50 = 524.81 nM T28330 CG02LF 10627173 IC50 = 10.81 nM T28330 CWF78P 10649606 EC50 = 0.014 nM T28330 C1QT8S 10674604 IC50 = 891.25 nM T28330 CXZ4C9 10675328 IC50 = 14.45 nM T28330 C84WOB 10698051 IC50 = 87.1 nM T28330 C89BME 10698109 IC50 = 154.88 nM T28330 CX8P5U 10698905 IC50 = 29.51 nM T28330 C90UHA 10699165 IC50 = 660.69 nM T28330 CG1KP5 10700916 EC50 = 1.549 nM T28330 CN53KG 10721792 IC50 = 120.23 nM T28330 C3R0HF 10722103 IC50 = 112.2 nM T28330 CA9O7Y 10722372 IC50 = 2511.89 nM T28330 CHD26N 10746778 IC50 = 1995.26 nM T28330 C7MS8F 10769675 IC50 = 478.63 nM T28330 C7KR4C 10769902 IC50 = 13.18 nM T28330 CU8KV7 10770092 IC50 = 17.78 nM T28330 CU59WT 10793168 IC50 = 107.15 nM T28330 CLMG75 10793883 IC50 = 38.9 nM T28330 C4G5HX 10794311 IC50 > 10000 nM T28330 CV2LI6 10817241 IC50 = 128.82 nM T28330 C8VBP1 10817395 IC50 = 8.318 nM T28330 CNL17K 10817407 IC50 = 354.81 nM T28330 CPER12 10819755 EC50 = 0.02512 nM T28330 C25UOS 10841112 IC50 = 89.13 nM T28330 C3Y6WE 10841358 IC50 = 42.66 nM T28330 C0ODR4 11027990 IC50 = 35.2 nM T28330 CT7HI5 11154873 Ki > 10000 nM T28330 CGR9A8 11178846 Ki > 10000 nM T28330 C2O3XT 11202178 Ki > 10000 nM T28330 C3NCV9 11212985 Ki > 10000 nM T28330 C8WK7R 11248998 Ki < 10000 nM T28330 C72OIE 11259485 Ki < 10000 nM T28330 CVL2X8 11281656 Ki > 10000 nM T28330 C2ZUE8 11292979 Ki < 10000 nM T28330 CL38VT 11293780 Ki < 10000 nM T28330 CD4I0A 11305046 Ki > 10000 nM T28330 CKL0X6 11316421 Ki < 10000 nM T28330 CBNS24 11316813 Ki < 10000 nM T28330 C9VA4Z 11352971 Ki > 10000 nM T28330 CU75AT 11353036 Ki < 10000 nM T28330 C3QE5S 11362975 Ki > 10000 nM T28330 COG3H2 11363465 Ki > 10000 nM T28330 C9DF4G 11363566 Ki < 10000 nM T28330 CXH69E 11385416 Ki > 10000 nM T28330 C9IX1T 11396307 Ki > 10000 nM T28330 CRA51C 11420366 Ki < 10000 nM T28330 COSZ16 11430523 Ki < 10000 nM T28330 CT0RI9 11431264 Ki < 10000 nM T28330 CXIN31 11442229 Ki > 10000 nM T28330 C9U8VO 11453391 Ki < 10000 nM T28330 C6AYO0 11454197 Ki < 10000 nM T28330 CE96SJ 11464858 Ki > 10000 nM T28330 C58JUC 11465671 Ki < 10000 nM T28330 CF9U1W 11511721 Ki = 1174.9 nM T28330 CV02EM 11512151 Ki = 50.12 nM T28330 C9TE6V 11527738 Ki = 10000 nM T28330 CYF52S 11534407 Ki = 79.43 nM T28330 C21ELY 11534594 Ki = 31.62 nM T28330 CA8WL2 11541048 Ki = 63.1 nM T28330 C7QYJ1 11555166 Ki = 724.44 nM T28330 C16KZS 11556194 Ki = 501.19 nM T28330 C8B2SH 11584582 Ki = 79.43 nM T28330 CK4H5O 11584903 Ki = 8709.64 nM T28330 C24OIW 11592162 Ki < 10000 nM T28330 CN6AR3 11605814 Ki < 10000 nM T28330 CT29GZ 11613982 Ki < 10000 nM T28330 CO3F1P 11627917 Ki = 79.43 nM T28330 C4EHB7 11635377 Ki = 12.59 nM T28330 COM97A 11656338 Ki = 5888.44 nM T28330 C51UDK 11667741 IC50 = 8100 nM T28330 CW79UI 11693225 Ki = 199.53 nM T28330 C42YZA 11700410 Ki = 158.49 nM T28330 CV9M3K 11712880 Ki = 1513.56 nM T28330 CK4SG5 11754311 Ki = 25.12 nM T28330 C65DTB 11765552 IC50 = 60.26 nM T28330 CSX23A 11786290 Ki < 10000 nM T28330 C8L2NZ 11801335 IC50 = 100 nM T28330 CSH7X6 11801911 IC50 = 16.98 nM T28330 C30NLE 15002730 Ki = 25.12 nM T28330 C2LBG8 15002734 Ki = 25.12 nM T28330 C5I4LT 15667001 IC50 = 16 nM T28330 CDJF92 15667003 IC50 = 4.2 nM T28330 CXH92N 15667011 IC50 = 0.99 nM T28330 C6QDI1 16090646 Ki < 10000 nM T28330 C3UCY1 16090647 Ki < 10000 nM T28330 C3HO2S 16090649 Ki < 10000 nM T28330 C4FKT8 16090650 Ki < 10000 nM T28330 CB19JY 16090651 Ki < 10000 nM T28330 CW7KL5 16090652 Ki > 10000 nM T28330 C9Q5YA 16090653 Ki > 10000 nM T28330 CA4PD3 16090658 Ki > 10000 nM T28330 CY9MB5 16090684 Ki > 10000 nM T28330 CY91OD 16090685 Ki > 10000 nM T28330 C4P8KS 16090686 Ki < 10000 nM T28330 C17IOA 16090687 Ki > 10000 nM T28330 C4ETX5 16090688 Ki > 10000 nM T28330 C37DEW 16090689 Ki > 10000 nM T28330 C7Q8LP 16090690 Ki > 10000 nM T28330 COJ46W 16090691 Ki < 10000 nM T28330 CNSU17 16090692 Ki > 10000 nM T28330 C49PFE 16090693 Ki > 10000 nM T28330 CI0XC5 16090694 Ki > 10000 nM T28330 C6QDP7 16090695 Ki > 10000 nM T28330 C3AVH8 16090699 Ki = 3162.28 nM T28330 C9R2PB 16090700 Ki = 199.53 nM T28330 C9K8RC 16090701 Ki = 7943.28 nM T28330 CH1UB0 16090702 Ki = 1995.26 nM T28330 CD7S4Q 16090703 Ki > 10000 nM T28330 CRS7B1 16090773 Ki > 10000 nM T28330 C2KCS0 16090774 Ki > 10000 nM T28330 C8IGT2 16090780 Ki > 10000 nM T28330 CM72TB 16090781 Ki > 10000 nM T28330 C8CI1X 16090782 Ki < 10000 nM T28330 C9QGU2 16090783 Ki > 10000 nM T28330 CF2IW8 16090784 Ki < 10000 nM T28330 CKCX80 16090785 Ki > 10000 nM T28330 C3D8HU 16090786 Ki < 10000 nM T28330 C8WSC9 16090788 Ki > 10000 nM T28330 CYQP41 16090789 Ki = 2511.89 nM T28330 C6MV4D 16090790 Ki > 10000 nM T28330 CJ94QO 16090791 Ki > 10000 nM T28330 C2G8TD 16090792 Ki < 10000 nM T28330 CRF40D 16090793 Ki < 10000 nM T28330 CX68OS 16090794 Ki > 10000 nM T28330 C0V8WI 16090795 Ki < 10000 nM T28330 C06QBM 16090796 Ki < 10000 nM T28330 C5NER1 16090797 Ki < 10000 nM T28330 C3T9MH 16100406 Ki = 130 nM T28330 CH6F0V 16100408 Ki = 8300 nM T28330 CY5F4S 16162108 EC50 = 269.15 nM T28330 C7YG3M 16731537 Ki < 10000 nM T28330 C7U3FA 16731711 Ki = 371.54 nM T28330 C3G0VB 16731712 Ki < 10000 nM T28330 CD9KY3 16731870 Ki < 10000 nM T28330 C6RS1M 16731872 Ki < 10000 nM T28330 CQ45MJ 16731874 Ki > 10000 nM T28330 C8FH9C 16732017 Ki = 6456.54 nM T28330 C9I7PZ 16732018 Ki = 4073.8 nM T28330 C8JR5Q 16732019 Ki = 1737.8 nM T28330 C2OQ0S 16732020 Ki = 6456.54 nM T28330 C5VUZ7 16732021 Ki = 389.05 nM T28330 CXN1C3 16732022 Ki < 10000 nM T28330 C34EYO 16732162 Ki = 457.09 nM T28330 C6CF0K 16732163 Ki < 10000 nM T28330 C4GZY1 16732164 Ki = 549.54 nM T28330 C8DU5M 16732165 Ki = 2511.89 nM T28330 CB7X3W 16732442 Ki < 10000 nM T28330 CY57CK 16732443 Ki = 5754.4 nM T28330 CO95FT 16732444 Ki = 2137.96 nM T28330 CE9M8H 16732592 Ki = 8128.31 nM T28330 C3J2CB 16732593 Ki = 6918.31 nM T28330 CU2FT3 16732598 Ki < 10000 nM T28330 CFT09X 16732750 Ki < 10000 nM T28330 CM4P7G 16732753 Ki < 10000 nM T28330 C9K4UR 16732755 Ki = 7943.28 nM T28330 CB2JR3 16732909 Ki > 10000 nM T28330 CZ14YT 16732911 Ki = 645.65 nM T28330 C35MZK 16732916 Ki = 1905.46 nM T28330 CR0A7J 16733051 Ki = 2951.21 nM T28330 C3LUI7 16733057 Ki < 10000 nM T28330 C9FU1Q 16733182 Ki < 10000 nM T28330 C93FYR 16733185 Ki = 549.54 nM T28330 CF3I5J 16733307 Ki = 660.69 nM T28330 CUF2R0 16733462 Ki = 8511.38 nM T28330 C0RH7Y 16733466 Ki = 2511.89 nM T28330 C1XWA0 16733469 Ki = 2089.3 nM T28330 CK04YG 16733644 Ki = 1698.24 nM T28330 C1RC2P 16733790 Ki < 10000 nM T28330 C76HVW 16755781 EC50 = 0.094 nM T28330 CO7F1T 16755782 EC50 = 1.1 nM T28330 CILG48 21842317 IC50 = 111 nM T28330 CLTI86 21842327 IC50 = 1200 nM T28330 C3NT8C 21842331 IC50 = 480 nM T28330 C53MSQ 21842340 IC50 = 293 nM T28330 CK8GY0 21842400 IC50 = 720 nM T28330 CPQ3K5 22171012 Ki = 25.12 nM T28330 C6VR4P 22171037 Ki = 25.12 nM T28330 C4Y3DN 22171039 Ki = 25.12 nM T28330 CH4V5J 22171089 Ki = 25.12 nM T28330 CKA98D 22171092 Ki = 25.12 nM T28330 CFL43N 23652473 IC50 > 1000000 nM T28330 CZ2PW8 24769543 EC50 = 0.033 nM T28330 CA7XZ6 24769546 IC50 = 0.018 nM T28330 C2YDQ3 24769604 IC50 = 0.01 nM T28330 CO46AU 24769605 EC50 = 0.065 nM T28330 CSCY65 24784940 IC50 = 2.5 nM T28330 C7HSF9 24784941 IC50 = 2.3 nM T28330 C14APO 24784942 IC50 = 22 nM T28330 C6X5AL 24785176 IC50 = 43 nM T28330 C4S1BJ 24785177 IC50 = 6.9 nM T28330 CE32FM 24785178 IC50 = 1.9 nM T28330 C6Y0AR 24785179 EC50 = 7.4 nM T28330 C0O2KU 24785180 EC50 = 5.5 nM T28330 C6ZNQ8 24785430 IC50 = 30 nM T28330 CXH90U 24785431 IC50 = 1.9 nM T28330 CC9TD5 24785432 EC50 = 175 nM T28330 C8A3XU 24785703 EC50 = 1.9 nM T28330 CZ14DY 24785705 IC50 = 0.42 nM T28330 CC8IW7 24861060 IC50 = 0.04 nM T28330 CZ9AS2 24861113 EC50 = 0.048 nM T28330 C6TM1P 24861114 EC50 = 0.053 nM T28330 C39NSA 24861174 EC50 = 0.4 nM T28330 CM0Q9T 24861391 IC50 = 0.03 nM T28330 CA5WE4 24861392 EC50 = 0.14 nM T28330 CCN34R 24861394 EC50 = 0.077 nM T28330 C5C4QR 24990933 IC50 < 50 nM T28330 C8HMZ0 25032312 Ki < 10000 nM T28330 C3NGL2 25032468 Ki < 10000 nM T28330 CK96SR 25033064 Ki < 10000 nM T28330 CM2Z9H 25033065 Ki < 10000 nM T28330 C1O7NJ 25033066 Ki < 10000 nM T28330 CITF86 25033148 Ki < 10000 nM T28330 C67SOQ 25033149 Ki < 10000 nM T28330 CJ10TY 25033150 Ki < 10000 nM T28330 C19WBD 44215880 Ki = 3.9 nM T28330 C6J7EK 44303510 IC50 > 10000 nM T28330 CWKM16 44303511 IC50 = 36.7 nM T28330 CY5Q8R 44303654 IC50 = 2175 nM T28330 CNH0W1 44303663 IC50 > 10000 nM T28330 CD80VI 44303664 IC50 = 2700 nM T28330 C0L8GD 44303722 IC50 = 364 nM T28330 CA8Z0J 44304324 IC50 = 190 nM T28330 C1VM8Q 44306360 IC50 = 31.62 nM T28330 C3ZDK0 44306744 IC50 = 19.95 nM T28330 CB5Q6O 44306823 IC50 = 5.012 nM T28330 CG9HF2 44306868 IC50 = 100 nM T28330 CP92WE 44306887 IC50 = 63.1 nM T28330 CN0SR5 44306888 IC50 = 100 nM T28330 C3MR8J 44328894 Ki = 10 nM T28330 C10ORA 44328951 Ki = 50.12 nM T28330 CZFL34 44329156 Ki = 79.43 nM T28330 CT7I5W 44330874 IC50 = 5.3 nM T28330 C4G1WN 44336539 EC50 = 0.02 nM T28330 C4HYP6 44355590 Ki = 3330 nM T28330 CVO2G3 44355745 Ki = 1080 nM T28330 CMS4H1 44355747 Ki = 3900 nM T28330 C8VW0Y 44355787 Ki = 10000 nM T28330 CHAZ51 44365304 IC50 = 3162.28 nM T28330 CMV8Q7 44365359 IC50 = 251.19 nM T28330 C1RNC2 44365788 IC50 = 10 nM T28330 CTD71M 44367000 IC50 = 2500 nM T28330 CN8SF3 44379428 Ki = 3 nM T28330 C9TZV6 44398261 IC50 = 3.8 nM T28330 CD69PS 44408411 Ki = 1000 nM T28330 C7QV6M 44408483 Ki = 560 nM T28330 C96ELC 44408632 Ki = 840 nM T28330 CI26KP 44417427 Ki > 10000 nM T28330 C0CV9L 44417429 Ki < 10000 nM T28330 CNZ3I4 44417439 Ki < 10000 nM T28330 C5OI3W 44418923 Ki > 10000 nM T28330 C4UPR1 44418924 Ki = 10000 nM T28330 CWT4D8 44425005 Ki = 7079.46 nM T28330 C2PEJ5 44425006 Ki = 3981.07 nM T28330 C7R2IK 44444763 Ki = 25.12 nM T28330 C0C1JA 44444767 Ki = 25.12 nM T28330 C91GMK 44444777 Ki = 25.12 nM T28330 CL94GA 44451519 Ki = 446.68 nM T28330 CXJ5N0 44451522 Ki = 616.6 nM T28330 CN8B5I 44451523 Ki < 10000 nM T28330 CMF6V5 44451547 Ki = 2089.3 nM T28330 C2MP5A 44451581 Ki = 281.84 nM T28330 C9SC7M 44451622 Ki = 2344.23 nM T28330 CH1K6S 44451830 Ki < 10000 nM T28330 CWEV38 44451843 Ki = 3890.45 nM T28330 CIS9D2 44451877 Ki = 1548.82 nM T28330 CVN2E4 44451920 Ki = 2344.23 nM T28330 C4DL5C 44469677 IC50 = 1 nM T28330 C9HFJ2 44562296 EC50 = 0.097 nM T28330 C1UA9S 44562297 EC50 = 0.04 nM T28330 CWT26N 44562298 EC50 = 0.095 nM T28330 C42LFU 44562299 IC50 = 0.08 nM T28330 CK78HN 44562300 EC50 = 0.082 nM T28330 C3QH7F 44562301 IC50 = 0.016 nM T28330 CSJ76G 44562302 EC50 = 0.034 nM T28330 CZ1MF9 44562303 IC50 = 0.067 nM T28330 CQ72YB 44562304 EC50 = 0.074 nM T28330 C9CDJ6 44562305 IC50 = 0.24 nM T28330 CM8A3V 44562306 EC50 = 0.097 nM T28330 CS3C0V 44562307 EC50 = 0.1 nM T28330 CR5Y4S 44562308 EC50 = 0.21 nM T28330 C9APN5 44562309 EC50 = 0.16 nM T28330 CF1BD0 44562310 EC50 = 0.18 nM T28330 C2JL9N 44562311 EC50 = 0.77 nM T28330 CT57RP 44562312 EC50 = 0.097 nM T28330 C2Y5XD 44562313 EC50 = 0.46 nM T28330 CJ72VF 44562314 EC50 = 0.14 nM T28330 C3IB9C 44578251 EC50 = 74 nM T28330 C3HFG1 44578305 IC50 = 8 nM T28330 CQ1DN3 44578398 IC50 = 630 nM T28330 C5FA0D 44578399 EC50 = 9.1 nM T28330 CG5PO8 44578422 IC50 = 16 nM T28330 C97ZLF 44578423 IC50 = 1.9 nM T28330 C5X3RK 44578424 EC50 = 1.1 nM T28330 CCS0G8 44578455 IC50 = 8.6 nM T28330 C45QLM 44578456 EC50 = 106 nM T28330 CW0F5K 44578457 EC50 = 0.078 nM T28330 CV5X3L 44578529 EC50 = 962 nM T28330 C4U0QS 44578530 IC50 = 130 nM T28330 CB31ZF 44578531 EC50 = 1349 nM T28330 CB9X2L 44578562 EC50 = 471 nM T28330 C8ES9Z 44578611 IC50 = 35 nM T28330 C65UYX 44578647 IC50 = 1.9 nM T28330 C94RSO 44578686 EC50 = 0.25 nM T28330 CLW1R5 44578727 EC50 = 0.53 nM T28330 CDIW83 44578728 EC50 = 0.13 nM T28330 CCP04Y 44578729 EC50 = 0.12 nM T28330 CJE1O8 44578764 EC50 = 0.26 nM T28330 C2A4JT 44578767 IC50 = 0.45 nM T28330 CPV6Q1 44578772 EC50 = 308 nM T28330 C6FE1M 45102806 Ki = 158.49 nM T28330 CM6BH7 45255234 Ki = 251.19 nM T28330 CYTL70 45486933 Ki = 100 nM T28330 CQH80S 45486935 Ki = 251.19 nM T28330 C7YUL8 45486936 Ki = 158.49 nM T28330 C1KLB2 45486940 Ki = 1995.26 nM T28330 COT6U7 45486941 Ki = 398.11 nM T28330 CAQ7Z9 45486947 Ki = 199.53 nM T28330 C6FGL0 45486949 Ki = 3981.07 nM T28330 CSR39Z 45486955 Ki = 199.53 nM T28330 CDZ82O 45486958 Ki = 3162.28 nM T28330 CMI20Q 45486964 Ki = 398.11 nM T28330 CD02XL 45486967 Ki = 158.49 nM T28330 C1X3BW 45486968 Ki = 316.23 nM T28330 CC8W1B 45486969 Ki = 199.53 nM T28330 CV17ZB 45486970 Ki = 3981.07 nM T28330 CZ04GO 45486971 Ki > 10000 nM T28330 C2WJI9 45486974 Ki = 25.12 nM T28330 C5HP4B 45486976 Ki = 251.19 nM T28330 CXR7T6 45486985 Ki = 316.23 nM T28330 CIX0G1 45486994 Ki = 1000 nM T28330 C1PZ8J 45486995 Ki = 1995.26 nM T28330 C06PMK 45486997 Ki = 3981.07 nM T28330 CQ31XM 45487002 Ki = 125.89 nM T28330 C3YB8W 45487003 Ki = 79.43 nM T28330 C6SQZ7 45487006 Ki = 100 nM T28330 CGH4V3 46234820 IC50 = 80.1 nM T28330 C5KH7S 46234969 IC50 = 4.24 nM T28330 CQAS17 46234970 IC50 = 44.7 nM T28330 CD0WG8 46235271 EC50 = 0.1202 nM T28330 CHD2N7 46235272 EC50 = 2.7 nM T28330 C94EJG 46869398 EC50 = 0.063 nM T28330 C8Y2QS 49798104 Ki > 10000 nM T28330 C6LEM8 49798106 IC50 = 125.89 nM T28330 C8EG6Y 49798111 Ki = 1400 nM T28330 C24DUW 49798112 Ki = 9 nM T28330 C2US0X 52940616 EC50 = 522 nM T28330 C5T0BN 52942901 EC50 = 91.3 nM T28330 CCOU43 52943046 EC50 = 628 nM T28330 CS2DM8 52944224 EC50 = 160 nM T28330 CL5G9A 52945789 EC50 = 1810 nM T28330 CW60FV 52946666 EC50 = 645 nM T28330 C4QWB8 52946667 IC50 = 246 nM T28330 CP0NO1 52950956 IC50 > 700 nM T28330 C7PC2V 52950958 IC50 > 700 nM T28330 CMYU60 52951093 IC50 > 700 nM T28330 C8ZL7M 52951227 IC50 > 700 nM T28330 C2VK4G 52951333 IC50 > 700 nM T28330 CG80QW 52951789 IC50 > 700 nM T28330 CXZL73 52952034 IC50 > 700 nM T28330 C6UQ3N 53233689 EC50 = 0.065 nM T28330 C2DIE0 53465843 Ki = 973 nM T28330 CB90RU 53465844 Ki = 0.32 nM T28330 C9J3NZ 54580263 EC50 = 38 nM T28330 CN56CG 54580264 IC50 = 2925 nM T28330 C74EHP 54580265 EC50 = 286 nM T28330 CV4Z2K 54580266 IC50 = 2.4 nM T28330 C6WDJ8 54580267 EC50 = 61 nM T28330 CF0V5K 54580295 EC50 = 0.71 nM T28330 CE98TJ 54580296 EC50 = 17 nM T28330 CGP10T 54581259 IC50 > 10000 nM T28330 CK85VP 54581260 IC50 = 35 nM T28330 C0XN2Z 54581261 EC50 = 34 nM T28330 C4SC7B 54581301 EC50 = 41 nM T28330 C8YT9J 54581302 EC50 = 9.6 nM T28330 CXP3W9 54582287 EC50 = 6.1 nM T28330 C5NZ0G 54582288 EC50 = 37 nM T28330 C7MT8A 54582313 EC50 = 5020 nM T28330 C10GBP 54583260 EC50 = 1.8 nM T28330 CSD2T3 54583296 EC50 = 0.24 nM T28330 CF12HS 54583297 EC50 = 59 nM T28330 CK01LS 54583298 EC50 = 0.2 nM T28330 C40TZF 54584222 IC50 > 10000 nM T28330 COGN42 54584255 EC50 = 7.5 nM T28330 CW6E2U 54586147 IC50 = 35 nM T28330 CB7AL6 54586148 IC50 = 0.18 nM T28330 CF1M5T 54586149 IC50 = 174 nM T28330 C5ME1Z 54586174 IC50 = 16.9 nM T28330 CE5SJ2 54586175 IC50 = 9.9 nM T28330 C9XP0E 54587149 IC50 = 33 nM T28330 CZ9S1K 54587150 EC50 = 1.3 nM T28330 CT14KG 54587151 EC50 = 256 nM T28330 C4HMO9 56663037 IC50 > 700 nM T28330 CZL6U4 56663263 IC50 > 700 nM T28330 CRL92U 56666696 IC50 > 700 nM T28330 CV38BZ 56683899 IC50 > 700 nM T28330 CSX93Z 70681224 EC50 = 31.9 nM T28330 CP73WX 70683295 IC50 = 68.6 nM T28330 C9V7QF 70683305 IC50 = 87.6 nM T28330 C15FHQ 70685411 IC50 = 248 nM T28330 CCQ5U4 70689603 EC50 = 52.5 nM T28330 C7BJ3X 70689619 EC50 = 2116.8 nM T28330 CQXZ61 70691750 EC50 = 12.9 nM T28330 C07BDF 70693814 IC50 = 340 nM T28330 CCN89Z 70695922 EC50 = 400 nM T28330 C0IJ1E 70695933 IC50 = 373 nM T28330 CR6KF1 70695934 IC50 = 38.1 nM T28330 CWH6T3 72548703 IC50 = 0.12 nM T28330 CNC3S0 73345637 IC50 = 15000 nM T28330 C5KT3R 73346888 IC50 < 100000 nM T28330 CG2PW4 73348650 IC50 = 32 nM T28330 CYL21W 73348651 IC50 = 6450 nM T28330 CO8BC0 73350236 IC50 = 26660 nM T28330 CIFQ07 73350237 IC50 = 7460 nM T28330 C5G8NK 73350238 IC50 = 7200 nM T28330 CE17QO 73351737 IC50 = 26340 nM T28330 CEVU91 73353218 IC50 = 6940 nM T28330 CGSW23 73354720 IC50 = 24750 nM T28330 CA8MQ1 73354785 Ki = 15 nM T28330 C6C0SX 90663256 IC50 = 7400 nM T28330 CZ61LK 127034966 EC50 > 5011.87 nM T28330 CA0SN5 127034967 EC50 > 5011.87 nM T28330 C1GY2T 135156251 EC50 > 10000 nM T28330 C3ZNX5 135423404 Ki = 467.74 nM T28330 CR79SC 135529065 Ki = 117.49 nM T28330 C0OK8I 135610887 Ki = 588.84 nM T28330 CEX49M 136000594 EC50 = 88 nM T28330 C8IP3M 136036821 Ki = 72.44 nM T28330 C6EOV2 136036823 Ki = 316.23 nM T28330 CB89KA 155514270 EC50 = 0.2512 nM T28330 C9MB4S 155514432 EC50 = 0.2138 nM T28330 CDK7N6 155515427 EC50 = 0.3631 nM T28330 C07LPH 155516677 EC50 = 0.1288 nM T28330 CBJH23 155517239 IC50 = 0.1096 nM T28330 CB1SI3 155517761 EC50 = 0.5012 nM T28330 CBG5S4 155517868 EC50 = 912.01 nM T28330 CTV3M6 155521287 IC50 = 5940 nM T28330 CKC61A 155524181 EC50 = 0.06761 nM T28330 CH5AU4 155524770 EC50 = 0.1585 nM T28330 CAE58M 155526914 EC50 = 0.1622 nM T28330 C9HIR7 155530671 EC50 = 0.06026 nM T28330 C30VKS 155531277 EC50 = 11.75 nM T28330 CKL8Y2 155532425 EC50 = 0.1096 nM T28330 CN0VP5 155532759 IC50 = 0.1072 nM T28330 C12IEY 155533399 EC50 = 0.166 nM T28330 CVBR79 155533520 EC50 = 8.511 nM T28330 CHV1D9 155535107 EC50 = 0.1072 nM T28330 C09DZK 155535249 EC50 = 0.166 nM T28330 CNB7M5 155535579 EC50 = 0.1698 nM T28330 CKI3E1 155536333 EC50 = 0.1349 nM T28330 CO07KD 155537344 EC50 = 0.1072 nM T28330 C8QIH3 155539345 IC50 = 0.06026 nM T28330 C2FBL5 155540394 EC50 = 1.122 nM T28330 CWP54F 155540415 EC50 = 602.56 nM T28330 CMV82T 155540739 EC50 = 0.2455 nM T28330 CB18RV 155542488 EC50 = 0.1905 nM T28330 CGN96I 155542545 EC50 = 3.311 nM T28330 CY6E8B 155543163 EC50 = 0.2951 nM T28330 CS5N7E 155543846 EC50 = 0.9772 nM T28330 C39DSM 155543995 EC50 = 0.3715 nM T28330 C7K4ZA 155544674 EC50 = 0.1288 nM T28330 CLB1R7 155546692 EC50 = 0.3236 nM T28330 C7Z8OY 155547906 IC50 = 0.07943 nM T28330 C1PV3I 155548381 EC50 = 0.389 nM T28330 C1GEA7 155550911 EC50 = 1.622 nM T28330 CQ9S8X 155551968 EC50 = 0.2138 nM T28330 C1DG3Q 155552556 EC50 = 0.182 nM T28330 C4QSR2 155553269 IC50 = 40.74 nM T28330 C3K4NQ 155553502 EC50 = 11.75 nM T28330 C51ZHW 155555065 IC50 = 0.09772 nM T28330 C8V6RX 155555346 IC50 = 0.0871 nM T28330 CDF1E8 155557064 EC50 = 0.1148 nM T28330 CN68GS 155557285 EC50 = 229.09 nM T28330 CO1N8R 155558199 EC50 > 1000 nM T28330 C0GE9L 155559320 IC50 = 0.07586 nM T28330 C2DFE4 155560670 IC50 = 0.07943 nM T28330 CLI24D 155562281 IC50 = 0.04266 nM T28330 CFZ19O 155564367 EC50 = 117.49 nM T28330 CFYB81 155564421 EC50 = 0.1549 nM T28330 CQ8G9E 155566319 IC50 = 0.07413 nM T28330 CK98TD 155568312 EC50 = 0.5012 nM T28330 CP23WI 44572148 Ki = 173.78 nM T28330 D00OFV 3035433 IC50 = 1400 nM T28330 D01ADK 11693641 Ki > 10000 nM T28330 D01AQC 9811733 Ki = 3600 nM T28330 D02ZML 5311148 IC50 = 22.91 nM T28330 D03EPA 11051303 IC50 = 97.72 nM T28330 D05QBF 443375 Ki = 0.02344 nM T28330 D05RRZ 10348659 IC50 = 63.1 nM T28330 D05YZC 59751 Ki = 10.4 nM T28330 D06BRA 11520765 IC50 = 6456.54 nM T28330 D06CIH 11200806 IC50 = 4000 nM T28330 D06KWA 11442807 IC50 = 12700 nM T28330 D07ICW 11556976 Ki = 32 nM T28330 D07LQQ 11564210 Ki = 9.6 nM T28330 D09EMR 11136782 IC50 = 1949.84 nM T28330 D0E2OG 11614928 Ki = 910 nM T28330 D0F1VP 44409521 IC50 = 2800 nM T28330 D0F1XY 44408590 Ki > 10000 nM T28330 D0FF6S 16038374 IC50 > 2000 nM T28330 D0I8AF 9833444 EC50 = 0.04365 nM T28330 D0I9PH 16100409 Ki = 1900 nM T28330 D0J7GJ 44408484 Ki = 10000 nM T28330 D0N6DN 44408524 IC50 = 4073.8 nM T28330 D0O7PT 60182 IC50 = 195 nM T28330 D0QP2S 44408526 Ki = 1900 nM T28330 D0R4GI 11040230 Ki = 5100 nM T28330 D0S7SO 16100407 Ki > 10000 nM T28330 D0TR0U 10942040 IC50 = 1096.48 nM T28330 D0U6OA 10909103 Ki = 5700 nM T28330 D0V9DY 16100410 Ki = 7000 nM T28330 D0X7LC 11061906 Ki = 870 nM T28330 D0Z4SS 44572147 Ki = 3.715 nM T18143 D03VOJ 8768 IC50 = 239000 nM T18143 C54JUR 25043 IC50 = 141000 nM T18143 C70HVL 77888 IC50 = 137000 nM T18143 CPI2E4 80447 IC50 = 71600 nM T18143 C07AKH 786691 IC50 = 20000 nM T18143 CY4MC6 3505109 IC50 = 145000 nM T18143 CGN9J7 44267478 IC50 = 25000 nM T18143 CH4Q6A 145964401 IC50 = 6100 nM T18143 CHU61S 145964420 IC50 = 600 nM T18143 C6YCA8 145964710 IC50 = 700 nM T18143 CV6F7L 145966788 IC50 = 600 nM T18143 CBWX17 145967285 IC50 = 900 nM T18143 COR9X3 145972736 IC50 = 700 nM T18143 CQ0M2X 145972809 IC50 = 7500 nM T18143 CF95RZ 145972878 IC50 = 600 nM T18143 CXI0D1 145975081 IC50 = 700 nM T18143 CG84ZR 145975487 IC50 = 400 nM T18143 C91FOT 145976006 IC50 = 800 nM T18143 C3F4UH 145978039 IC50 = 500 nM T79062 D00TLN 2913 Ki = 50.12 nM T79062 D00XWD 135409453 Ki < 100 nM T79062 D01AZG 5073 Ki = 0.4 nM T79062 D01ZII 2726 Ki = 10.72 nM T79062 D02HED 4748 Ki = 23 nM T79062 D03ELL 2159 Ki = 25.12 nM T79062 D03WEX 9966051 Ki = 19 nM T79062 D04JEE 4946 EC50 > 5011.87 nM T79062 D05MBZ 129211 Ki = 84 nM T79062 D05XGO 11154555 Ki = 111 nM T79062 D05ZIK 4205 Ki = 265 nM T79062 D06XZR 27400 Ki = 25 nM T79062 D08VRO 3822 Ki = 1258.93 nM T79062 D09IOI 2170 Ki = 500 nM T79062 D09TPF 23897 Ki = 265 nM T79062 D0CQ0Z 33630 Ki = 280 nM T79062 D0D1AL 3559 Ki = 316.23 nM T79062 D0G8NN 119570 Ki = 1188 nM T79062 D0H3HM 60795 Ki = 10.3 nM T79062 D0H7KF 5002 Ki = 63.1 nM T79062 D0P0OU 11978813 Ki = 3.7 nM T79062 D0R1JV 60854 Ki = 5 nM T79062 D0R6RO 4184 Ki = 56 nM T79062 D0U1OE 5452 Ki = 70 nM T79062 D0UA0I 28693 Ki = 6.31 nM T79062 D0V4QS 135398745 Ki = 79.43 nM T79062 D0W5HK 216239 Ki = 7071 nM T79062 D0X6BV 6918314 Ki = 3900 nM T79062 D0Z1RV 135398737 Ki = 5.5 nM T79062 D0Z6UC 5358 Ki = 1000 nM T79062 D04GMY 11842633 Ki < 100 nM T79062 D08CJK 1150 Ki = 158.49 nM T79062 D09IRN 21071390 Ki = 8635 nM T79062 D0N1HW 5311200 Ki = 226.3 nM T79062 D0R9HI 11256720 Ki = 14230 nM T79062 D00OWF 5280953 Ki = 5500 nM T79062 D02JMI 9888211 Ki = 100 nM T79062 D03ZZH 9887537 Ki = 63.1 nM T79062 D06DZI 107780 Ki > 10000 nM T79062 D06ZVC 10150497 Ki = 679 nM T79062 D07BCO 5684 Ki = 10000 nM T79062 D08AWI 11430856 Ki = 700 nM T79062 D08PUW 64982 IC50 > 200000 nM T79062 D0B7SP 11292933 Ki = 158.49 nM T79062 D0K8NW 5074 Ki = 15.85 nM T79062 D0L9SN 4431 Ki = 0.6 nM T79062 D0M7LV 5761 Ki = 6.31 nM T79062 D0Q2JS 10436045 Ki = 63.1 nM T79062 D0U7VZ 11225102 Ki < 100 nM T79062 D0YP7L 6604889 Ki = 0.3388 nM T79062 CZUI83 2769 Ki = 1000 nM T79062 C5H9CN 9287 Ki = 102.33 nM T79062 CFGH18 27620 Ki = 364 nM T79062 C8Y6DE 37461 Ki = 63.1 nM T79062 C6WDL7 49756 Ki = 145 nM T79062 CIOE06 69729 Ki = 140 nM T79062 CN9GK1 104911 Ki > 10000 nM T79062 CBH8L0 156308 Ki = 5000 nM T79062 CGT8R0 160510 Ki = 280 nM T79062 CLK7P3 169713 IC50 = 143 nM T79062 C4J5ZF 185617 IC50 = 63400 nM T79062 C9XWA6 198914 Ki = 1100 nM T79062 CP2DY7 198967 Ki = 97000 nM T79062 CVI6X5 213046 Ki = 0.5 nM T79062 C2V5FA 398712 Ki = 30 nM T79062 CYV1R3 417052 Ki = 2960 nM T79062 CD8Z9H 424430 Ki = 26 nM T79062 C4O6RK 435595 Ki = 84 nM T79062 CFJ3R2 452533 Ki = 27 nM T79062 CGF6W2 642376 IC50 = 126600 nM T79062 CTN56Q 647533 Ki > 4000 nM T79062 CXQ6U0 735755 IC50 > 10000 nM T79062 C2VLP8 752521 Ki = 2083 nM T79062 C9FI5L 1296368 Ki = 25390 nM T79062 C6VZT7 1984087 Ki = 8000 nM T79062 CGS9R7 2133793 Ki = 4718 nM T79062 CG9N3A 2136365 Ki = 6371 nM T79062 CT8KN9 2232766 Ki = 2307 nM T79062 CA2OY6 2737389 Ki = 1.4 nM T79062 CE50LO 2756712 Ki = 25 nM T79062 C1C4LH 2843443 Ki = 12250 nM T79062 CRA6F5 2853434 Ki = 1473 nM T79062 C3QRD6 2867758 Ki = 6100 nM T79062 CL2G3H 2870750 Ki = 13020 nM T79062 CC74QS 2872937 Ki = 20090 nM T79062 CRF65H 2880253 Ki = 10100 nM T79062 CET7C8 2921525 Ki = 14100 nM T79062 C2DE6R 2927683 Ki = 3800 nM T79062 CF01YE 2928642 Ki = 8400 nM T79062 CY8R6Q 2948971 Ki = 18080 nM T79062 CLXQ01 2950739 Ki = 10400 nM T79062 CO0C7J 2962174 Ki = 84500 nM T79062 CAM8H3 3066250 IC50 = 9800 nM T79062 CT9L0D 3084440 Ki = 80 nM T79062 C6SA2G 3132842 Ki = 37200 nM T79062 CNX8I1 3245407 IC50 > 1000 nM T79062 CX8W7I 3377940 Ki = 1700 nM T79062 CS8KE2 3649661 Ki = 472 nM T79062 C6SHA4 4713248 Ki = 950 nM T79062 CRUB15 4723431 Ki = 1281 nM T79062 C7PX9E 4790508 Ki = 197 nM T79062 C9NKP1 5216959 Ki = 265 nM T79062 C4BKS2 5242341 Ki = 502 nM T79062 C4J3HP 5640104 Ki = 3490 nM T79062 CGM63Y 6540428 Ki = 12.59 nM T79062 C0QCK1 6918455 Ki = 3981.07 nM T79062 CW0ZE5 6918542 Ki = 600 nM T79062 CC5PQ0 6918601 Ki > 5800 nM T79062 C1WXY3 6918603 Ki < 7943.28 nM T79062 CD0Z4I 6918648 Ki = 3162.28 nM T79062 C8AL9V 6918689 Ki < 100000 nM T79062 CI0X2F 7059581 Ki = 1 nM T79062 C2F3BY 7125890 Ki = 9566 nM T79062 CUD06Z 9796627 Ki = 1600 nM T79062 CFC9Y5 9799318 Ki = 6.457 nM T79062 CG0UK3 9803482 Ki = 16.98 nM T79062 CE0DI5 9804612 Ki = 79.43 nM T79062 CNX4F0 9805456 Ki < 5011.87 nM T79062 CWOS30 9817810 Ki = 29 nM T79062 CFBH76 9820952 Ki = 31.62 nM T79062 CBN06W 9839050 Ki = 13 nM T79062 CE3W4V 9845006 Ki = 2.138 nM T79062 CM13ZV 9856041 Ki = 24000 nM T79062 C0ZR3E 9861687 IC50 > 1000 nM T79062 CNCK78 9862256 Ki = 460 nM T79062 C4H7DK 9864569 IC50 < 50 nM T79062 CB1F0C 9867475 Ki = 1300 nM T79062 C7AB8O 9870053 Ki < 5011.87 nM T79062 CQ4LC2 9872676 Ki = 1750 nM T79062 CCLN49 9878197 Ki = 49 nM T79062 C9NF3D 9881600 Ki = 0.6 nM T79062 C08DBF 9885982 Ki = 3 nM T79062 CL1W0B 9887186 Ki = 5.754 nM T79062 CJW1P5 9888494 Ki = 2.239 nM T79062 C6N8UE 9889681 Ki < 10000 nM T79062 CM52WU 9890119 Ki = 2511.89 nM T79062 CEG1K5 9891002 Ki = 1584.89 nM T79062 C7QMK5 9891617 Ki < 5011.87 nM T79062 CEL29O 9891618 Ki = 1995.26 nM T79062 C3J8GU 9892409 Ki < 7943.28 nM T79062 CAM25C 9894665 Ki = 10 nM T79062 CUN81Q 9905249 Ki > 10000 nM T79062 CYWQ50 9906447 Ki > 10000 nM T79062 C9B3EA 9911844 Ki = 7.24 nM T79062 C78MDV 9913554 Ki = 1000 nM T79062 CR9KM0 9921064 Ki = 290 nM T79062 C4UYZ7 9927441 Ki = 3700 nM T79062 CYVZ47 9934284 Ki = 39.81 nM T79062 CO2RS8 9934709 Ki = 0.6761 nM T79062 CWO45F 9935387 Ki = 630.96 nM T79062 CX6E8C 9945703 Ki = 6 nM T79062 CQ04ZS 9950396 Ki = 400 nM T79062 CK8NR2 9954121 Ki < 10000 nM T79062 CHOJ30 9956365 Ki = 3.548 nM T79062 CFR41N 9957068 Ki < 3981.07 nM T79062 CFN50J 9978683 Ki = 579 nM T79062 CS40QN 10015688 Ki = 0.7 nM T79062 CV7R9F 10020040 Ki = 335.9 nM T79062 CK18LT 10020895 Ki > 5000 nM T79062 C2EUY0 10035109 Ki > 10000 nM T79062 C57TZR 10042333 Ki = 1345 nM T79062 C0KWB6 10062885 Ki = 1.1 nM T79062 CR68SH 10064053 Ki = 9.78 nM T79062 C8Z6MA 10067306 IC50 = 1217 nM T79062 CKA5F4 10084076 Ki = 18 nM T79062 C93RNG 10090247 Ki = 7 nM T79062 CA5H7K 10106205 Ki = 16 nM T79062 C4Q3UL 10154897 Ki = 3 nM T79062 C7F1ED 10183148 IC50 = 135000 nM T79062 CW09SL 10202089 Ki = 6 nM T79062 C4Q2SH 10249573 Ki = 10 nM T79062 CMRA02 10257042 Ki < 794.33 nM T79062 CH31DX 10267394 Ki = 412.3 nM T79062 CTWJ70 10274894 Ki = 2.042 nM T79062 CU89JD 10314060 Ki = 102.8 nM T79062 C9IAV3 10346043 Ki = 1.023 nM T79062 CA7IM5 10379532 Ki = 1.096 nM T79062 CR3KU9 10380133 IC50 > 5000 nM T79062 CMZA83 10383646 Ki = 753 nM T79062 C4L5PQ 10404657 Ki = 8.511 nM T79062 C04WGF 10407367 IC50 = 511 nM T79062 C4TPN1 10413595 Ki = 0.3162 nM T79062 C2B0IU 10421236 IC50 > 10000 nM T79062 CR4LS0 10430623 Ki = 1563 nM T79062 CD7U5I 10433930 Ki = 1.995 nM T79062 CO7IV6 10450593 Ki = 0.1995 nM T79062 COV85C 10472143 Ki = 14 nM T79062 C5LBS7 10472158 IC50 = 1362 nM T79062 C26KCR 10475231 Ki = 2 nM T79062 CEF2O6 10478367 Ki = 1412 nM T79062 CL70NJ 10499156 Ki = 10 nM T79062 CN29IF 10500557 Ki = 2.138 nM T79062 CWH7R8 10521887 Ki = 26.33 nM T79062 C9B7LR 10552788 Ki = 19.95 nM T79062 CHE80N 10573876 Ki = 1.995 nM T79062 CAVR62 10596321 Ki = 10 nM T79062 CO23YX 10597140 Ki = 15.85 nM T79062 CZ6WS8 10619437 Ki = 125.89 nM T79062 CAPO49 10638372 Ki = 105 nM T79062 CK08CW 10643153 Ki = 10000 nM T79062 CN40TJ 10668422 Ki < 1000 nM T79062 CBE87R 10706626 Ki = 13.4 nM T79062 CU32PG 10714877 Ki = 10.35 nM T79062 C1PG3A 10715573 Ki = 31.62 nM T79062 CJ4HC8 10715998 Ki = 15.85 nM T79062 CZ3A0O 10737314 Ki = 100 nM T79062 CIVN21 10767321 Ki = 15.85 nM T79062 C2AFT6 10785644 Ki = 1584.89 nM T79062 C3SWV9 10785714 Ki = 5 nM T79062 C75SKC 10811746 Ki = 3.802 nM T79062 CG4X1R 10834268 Ki = 1.862 nM T79062 C8MHZ9 10835110 Ki = 3.981 nM T79062 C5Q4IJ 10862697 Ki = 2.344 nM T79062 CFY4V1 10862787 Ki = 12 nM T79062 CVT7J1 10873805 Ki = 7.32 nM T79062 CNEP25 10884517 Ki = 7.943 nM T79062 C67UIY 10884717 Ki = 6.457 nM T79062 CRI50E 10885636 IC50 = 1440 nM T79062 C9C2FI 10895284 Ki = 72.44 nM T79062 CD4YL2 10896196 Ki = 19.05 nM T79062 CX65PW 10907460 IC50 = 2040 nM T79062 CEGJ41 10917174 Ki = 6.026 nM T79062 CU09AV 10937901 IC50 = 762 nM T79062 C7PWT9 10938620 Ki = 109.65 nM T79062 CA42MT 10939416 Ki = 8.71 nM T79062 CNB39C 10947658 Ki = 12 nM T79062 CSLT97 10949380 IC50 = 663 nM T79062 C2MBP7 10949445 Ki = 8.128 nM T79062 C74SOA 10950559 Ki = 74 nM T79062 C47MYE 10960943 Ki = 97.72 nM T79062 CJD58C 10971401 Ki = 4.786 nM T79062 C51NOQ 10982183 Ki < 10000 nM T79062 CK6VF7 10991109 Ki = 63 nM T79062 C4O7MD 10994400 Ki = 101 nM T79062 CJC9K4 11005810 IC50 = 998 nM T79062 C3FIP5 11016205 Ki = 3.68 nM T79062 CS0Z2D 11024311 Ki < 10000 nM T79062 CRS62E 11025847 Ki = 3.548 nM T79062 C0HA7O 11047374 Ki = 1.995 nM T79062 C23JHR 11047568 IC50 = 1430 nM T79062 C80UIZ 11048252 Ki = 416.87 nM T79062 CONV96 11058267 Ki = 45.71 nM T79062 CD4BW6 11058564 Ki = 43.65 nM T79062 CZN25U 11059148 Ki = 23.99 nM T79062 CG41BK 11071079 IC50 = 726 nM T79062 C15USQ 11101733 Ki = 19.05 nM T79062 C7OFQ4 11102049 Ki = 29.51 nM T79062 CCJ1U3 11112531 Ki = 147 nM T79062 C7DE0U 11113605 IC50 = 1170 nM T79062 CVE8T3 11121216 Ki = 31 nM T79062 C5I0XL 11133795 Ki = 223.87 nM T79062 C0VZK2 11143387 Ki = 9.7 nM T79062 CS90QD 11145126 Ki = 7.079 nM T79062 CYJ79P 11153905 Ki = 2.55 nM T79062 C8ZN3B 11166042 Ki = 37 nM T79062 CEHV65 11173572 Ki = 13.4 nM T79062 C6CL1Y 11178830 Ki = 125.89 nM T79062 C0W4SM 11186523 Ki = 6.5 nM T79062 CXQ3K0 11186985 Ki = 2.91 nM T79062 C5J4NR 11199511 Ki = 8 nM T79062 C9N5QU 11200511 Ki = 74 nM T79062 C90WSG 11248705 Ki = 125.89 nM T79062 CM08DU 11259115 Ki = 200 nM T79062 C4S2VF 11277147 Ki = 17.6 nM T79062 CY6MX5 11282296 EC50 = 2460 nM T79062 CW40XM 11294248 Ki = 251 nM T79062 C9BLC7 11304596 Ki = 501.19 nM T79062 CJS9C0 11304851 IC50 = 25000 nM T79062 CI79LV 11307899 Ki = 6.31 nM T79062 C1VSE5 11327643 Ki = 1000 nM T79062 CGD42N 11361090 Ki > 5000 nM T79062 CXW6B5 11373831 Ki = 19 nM T79062 CBV52J 11384146 Ki = 24 nM T79062 C1BP0U 11385380 Ki > 1000 nM T79062 CF4OX6 11397149 Ki = 79.43 nM T79062 C30ZMW 11397459 Ki = 200 nM T79062 C7GXP9 11397799 Ki = 9 nM T79062 C85LYP 11430418 IC50 = 1000 nM T79062 CNF28A 11432177 EC50 = 6320 nM T79062 CJK2S4 11453751 Ki = 221 nM T79062 CMFC18 11453756 Ki = 200 nM T79062 C9K8UW 11515799 Ki = 7.65 nM T79062 CVAC51 11524003 Ki = 1.19 nM T79062 C7YRP3 11524413 Ki = 0.38 nM T79062 CFW50Y 11525867 Ki = 9.5 nM T79062 C2M0JG 11532105 Ki = 40 nM T79062 C5VHK0 11536843 Ki = 5.1 nM T79062 C0YZ7L 11536844 Ki = 3.3 nM T79062 C1V5CH 11559090 Ki > 10000 nM T79062 C14HEP 11560285 Ki = 296 nM T79062 C1HP5K 11566558 Ki = 4.31 nM T79062 CNH1K4 11568826 Ki = 520 nM T79062 C8NMI4 11575479 Ki = 600 nM T79062 C1I4DF 11582132 Ki = 25 nM T79062 C6D1MA 11584660 Ki > 1995.26 nM T79062 C1M2CP 11589069 Ki = 0.38 nM T79062 CU45DK 11595209 Ki > 10000 nM T79062 CE9W6J 11595790 Ki = 16.8 nM T79062 CGX8F6 11596869 Ki > 3980000 nM T79062 CX5ZM0 11603891 Ki = 5.38 nM T79062 C8EPV2 11610908 Ki = 64 nM T79062 CUA05E 11617668 Ki = 5.4 nM T79062 CD4HR8 11633354 Ki = 2.1 nM T79062 C2OU7Y 11638332 Ki > 10000 nM T79062 C9OLN0 11646336 Ki = 5 nM T79062 CJBV31 11652871 IC50 = 118100 nM T79062 CCX0S1 11653869 Ki = 0.49 nM T79062 CO1L8J 11661471 Ki = 1.02 nM T79062 C4L7TV 11662592 Ki = 4.48 nM T79062 CD91CP 11666595 Ki = 33 nM T79062 CXRC27 11667458 Ki = 10.9 nM T79062 C42RHW 11674602 Ki = 94 nM T79062 CL31JB 11683077 Ki = 11.1 nM T79062 CEQ6W7 11694810 Ki = 4.3 nM T79062 C2QCF5 11697434 Ki = 18 nM T79062 CHR8U4 11697659 Ki = 2.81 nM T79062 C3IML2 11709509 Ki = 0.3 nM T79062 C1N7MO 11725453 Ki = 1 nM T79062 CV82QX 11729084 Ki = 25.12 nM T79062 CLYJ75 11729823 Ki = 8.76 nM T79062 C7PVL8 11730467 IC50 = 2130 nM T79062 CG72CS 11732538 Ki = 20 nM T79062 CMO0I9 11739679 Ki = 1555 nM T79062 C57IKL 11740526 Ki = 9.772 nM T79062 CPG15O 11743399 IC50 > 1000 nM T79062 CYV02C 11747350 Ki = 510 nM T79062 C3F5DX 11761059 IC50 = 4420 nM T79062 C9LUA7 11773414 Ki = 800 nM T79062 C37LEP 11785183 EC50 = 1820 nM T79062 C7A2QD 11793826 Ki = 630.96 nM T79062 C3PY7W 11811833 Ki = 21.88 nM T79062 CQV92N 11825614 Ki = 10.47 nM T79062 CW4BC2 11826723 Ki = 12.3 nM T79062 CXLW54 11948707 Ki = 328 nM T79062 C8JQL7 11957735 IC50 = 1713 nM T79062 C1QY2P 12005903 Ki = 15770 nM T79062 C8EDN0 12088080 Ki = 3 nM T79062 C8RB6W 12088082 Ki = 9 nM T79062 CLC82F 12374770 Ki = 176 nM T79062 CCG14E 13091356 Ki = 420 nM T79062 CYN95Z 13091359 Ki = 97 nM T79062 C4V6AS 14135325 IC50 = 179000 nM T79062 CAO70J 14748689 IC50 = 949 nM T79062 C7VAI1 15011772 IC50 > 10000 nM T79062 C30CHU 15512229 Ki < 316.23 nM T79062 CKBD37 15542627 Ki = 17.38 nM T79062 C65SCN 15599151 Ki = 1240 nM T79062 CTPX97 15803947 Ki = 1.3 nM T79062 C1LWZ6 16006605 Ki = 2.4 nM T79062 CK36NS 16006607 Ki = 1 nM T79062 C3M8GJ 16026344 Ki = 5232 nM T79062 C1SR0O 16071847 Ki > 5000 nM T79062 CD3E8L 16093484 Ki = 8.7 nM T79062 CEW91O 16093485 Ki = 2.5 nM T79062 CZ1WJ4 16117151 Ki = 3970 nM T79062 CM32ZX 16117153 Ki > 5000 nM T79062 CXTB90 16117279 Ki = 3216 nM T79062 C1F2LS 16118795 Ki > 5000 nM T79062 C69VDS 16118923 Ki > 5000 nM T79062 CZ2IS9 16660294 Ki > 10000 nM T79062 CT9GP4 16763549 Ki = 13100 nM T79062 CR63LE 17055181 Ki = 3700 nM T79062 C0QX5J 17374371 Ki = 12590 nM T79062 CB2J3R 17747575 IC50 > 100 nM T79062 C42YEX 18133517 Ki = 3187 nM T79062 CI90UP 18133518 Ki = 2544 nM T79062 C7R1IG 18137015 Ki = 1029 nM T79062 C4I1FW 18137017 Ki = 1342 nM T79062 C07EOI 18137020 Ki = 1417 nM T79062 C9PV8A 18180076 IC50 = 1582 nM T79062 CI6TS8 18377342 Ki = 562.34 nM T79062 CHFJ09 18377388 Ki = 173.78 nM T79062 C5KB2J 18377409 Ki = 15.85 nM T79062 CI91VX 18377415 Ki = 812.83 nM T79062 CXR67I 18663036 Ki = 18.4 nM T79062 C6AOE8 19426635 IC50 = 18.62 nM T79062 CUI3R1 19605739 Ki = 1 nM T79062 C7T8JC 19958494 Ki = 318.2 nM T79062 C6LI5E 19958507 Ki = 411 nM T79062 CBY03N 20846175 Ki < 10000 nM T79062 CISE25 21091965 Ki = 80 nM T79062 C6H9WC 21092408 Ki = 88 nM T79062 C3T5HF 21509921 Ki = 100 nM T79062 CFN81Q 21527771 Ki = 656 nM T79062 CH59WN 21533446 Ki = 1044 nM T79062 C4B0TN 21557475 Ki = 1200 nM T79062 CT7XG9 21830793 Ki = 12.9 nM T79062 C9X8PI 22001618 Ki = 2.6 nM T79062 CBN84K 22065997 Ki = 212.9 nM T79062 C1QBE0 22273749 Ki = 11.22 nM T79062 C6UXL4 22330705 Ki = 21400 nM T79062 CZG9S2 22425072 Ki = 12710 nM T79062 CW0V5M 22449331 Ki = 4.467 nM T79062 CPD8Q7 22549784 Ki = 26650 nM T79062 CZ7J4B 22857296 Ki = 6.4 nM T79062 C0L5QK 23111951 Ki = 270 nM T79062 CY10BQ 23133427 Ki = 2.7 nM T79062 C5BUL7 23151712 Ki = 43 nM T79062 C3IF7P 23151734 Ki = 185 nM T79062 C0NI3J 23290944 Ki = 198 nM T79062 C57MVP 23369416 Ki = 3.4 nM T79062 C6HE8J 23369421 Ki = 26 nM T79062 CAE7K1 23369450 Ki = 1838 nM T79062 CWQ2X3 23369455 Ki = 48 nM T79062 C7EPU0 23369457 Ki = 1029 nM T79062 CRT2Z3 23661667 Ki = 54 nM T79062 CHGE36 23661734 Ki = 46 nM T79062 C5ZSR7 23661735 Ki = 1200 nM T79062 CQE1N7 23906630 Ki = 16020 nM T79062 CD7CV6 24771120 Ki = 6900 nM T79062 CCEH06 24781896 IC50 > 100 nM T79062 CD86PT 24781897 IC50 > 100 nM T79062 CP7TJ3 24781898 IC50 > 100 nM T79062 CF17PW 24781899 IC50 > 100 nM T79062 C1JSY8 24781900 IC50 > 100 nM T79062 CJI2O1 24782049 IC50 > 100 nM T79062 CK9T1F 24782050 IC50 > 100 nM T79062 C2O7MV 24782051 IC50 > 100 nM T79062 C0G3RV 24782052 IC50 > 100 nM T79062 CR8DV4 24782058 IC50 > 100 nM T79062 C58AMS 24829343 Ki = 0.79 nM T79062 CDC91N 24839550 Ki < 10000 nM T79062 CY21RE 24841480 Ki = 330 nM T79062 CT2YG6 24853955 Ki = 0.6 nM T79062 C2KD1T 24854037 Ki = 0.66 nM T79062 C1BPD9 24854039 Ki = 5.3 nM T79062 CGPC24 24854040 Ki = 8.27 nM T79062 CM01LB 24854041 Ki = 0.67 nM T79062 CI7G6M 24854043 Ki = 4.75 nM T79062 C4WUP5 24854044 Ki = 1.1 nM T79062 CY1XA8 24854103 Ki = 6.99 nM T79062 C42KBQ 24854105 Ki = 1.96 nM T79062 CUW23K 24854106 Ki = 44 nM T79062 CX7MK6 24854108 Ki = 33.38 nM T79062 CS90OD 24854109 Ki = 21 nM T79062 CFHM49 24854111 Ki = 1.45 nM T79062 C80ANM 24854181 Ki = 1.24 nM T79062 CSL8E3 24854183 Ki = 1.5 nM T79062 CFR74S 24854185 Ki = 1.8 nM T79062 CW2Z5A 24854186 Ki = 25.4 nM T79062 C9GYO8 24854187 Ki = 0.43 nM T79062 CB9M0N 24854266 Ki = 9.07 nM T79062 C0LQ1R 24854267 Ki = 3.4 nM T79062 CP23KC 24854269 Ki = 6.57 nM T79062 CI5LC8 24854270 Ki = 9.46 nM T79062 CCUS10 24854272 Ki = 5.97 nM T79062 CFX96I 24854273 Ki = 0.4 nM T79062 C6Y3AG 24854368 Ki = 2.07 nM T79062 CTS4E5 24854369 Ki = 2.55 nM T79062 COZ84H 24854370 Ki = 5.11 nM T79062 C3X9MD 24854371 Ki = 0.6 nM T79062 C7ZEF0 24856058 IC50 > 10000 nM T79062 C3HK0J 24865725 Ki = 19.95 nM T79062 C0O6FX 24865727 Ki = 15.85 nM T79062 C98ZIV 24882509 IC50 = 11.99 nM T79062 C6L7KS 24887518 Ki < 3162.28 nM T79062 CAOF91 24894071 IC50 > 10000 nM T79062 CMN75S 24901425 Ki = 1659.59 nM T79062 CF7IV1 24963856 Ki = 6.2 nM T79062 C8DJG7 24963860 Ki = 8.6 nM T79062 C35XOJ 24964217 Ki = 8.4 nM T79062 CP6K8J 25024727 IC50 > 10000 nM T79062 CI95EF 25192947 Ki = 0.47 nM T79062 CKAS93 25256850 Ki = 6 nM T79062 CW07GN 25256855 Ki = 7 nM T79062 CM2T9Y 25263297 Ki = 5100 nM T79062 CFJM71 25263302 Ki = 5800 nM T79062 CHJ35A 32354149 Ki = 885 nM T79062 CS5QG1 35391328 Ki = 773 nM T79062 C8G7EY 36418162 IC50 = 476 nM T79062 CDV36I 37219401 Ki = 855 nM T79062 CG56DF 42388639 IC50 = 20 nM T79062 C6VL8I 42388965 IC50 = 140 nM T79062 CS2G3E 42388975 IC50 = 289 nM T79062 CJ8FH4 42389129 IC50 = 681 nM T79062 CO51RQ 42389139 IC50 > 10000 nM T79062 CBV62E 42389293 IC50 = 3241 nM T79062 CNV94Z 42389303 IC50 = 9314 nM T79062 CSRX20 42389457 IC50 = 53 nM T79062 CH5QX6 42389467 IC50 = 47 nM T79062 CV9C4D 42428409 Ki = 78 nM T79062 C1SD3E 42618253 Ki = 1230 nM T79062 C0BWG1 42618254 Ki = 902 nM T79062 CAG71H 42618255 Ki = 864 nM T79062 CQ96KL 42618256 Ki = 566 nM T79062 CC1Z7P 42618257 Ki = 1867 nM T79062 CFB70T 42618258 Ki = 17960 nM T79062 CJV5N3 42618259 Ki = 2500 nM T79062 CHA26S 42618260 Ki = 296 nM T79062 CX1KC4 42618261 Ki = 168 nM T79062 C2VWK7 42618262 Ki = 267 nM T79062 CV0CD8 42618263 Ki = 243 nM T79062 CS5TJ8 42618264 Ki = 38 nM T79062 CKOJ59 42618265 Ki = 20 nM T79062 C4J9RQ 42618266 Ki = 78 nM T79062 C16TUL 42618267 Ki = 11 nM T79062 CH3NO7 42618269 Ki = 21 nM T79062 CMGJ03 42618270 Ki = 134 nM T79062 CR6OX0 42618271 Ki > 5000 nM T79062 C7SN5E 42618272 Ki = 31 nM T79062 C3VR7E 42618273 Ki = 335 nM T79062 CA0B9F 42625181 Ki = 68 nM T79062 C3L0TN 42625183 Ki = 69 nM T79062 CW0OU4 42625185 Ki > 1000 nM T79062 CHY12B 42625186 Ki > 1000 nM T79062 CP5X3K 42625188 Ki > 1000 nM T79062 C8QSX3 42625267 Ki = 193 nM T79062 CTM69J 42625269 Ki = 350 nM T79062 CPDG98 42625353 Ki = 63 nM T79062 CK3QD2 42625354 Ki > 1000 nM T79062 CJ64FG 42625356 Ki = 250 nM T79062 C27KEF 42625359 Ki = 160 nM T79062 CN81SE 42625440 Ki = 7 nM T79062 CF7DM0 42625445 Ki = 22 nM T79062 CJI51X 42625446 Ki = 69 nM T79062 CLH7Y0 42626289 Ki = 158 nM T79062 C75QPL 42626291 Ki = 203 nM T79062 C5VTZ6 42626293 Ki = 74 nM T79062 C70SWL 42626361 Ki = 63 nM T79062 CY7W2J 42631003 Ki = 0.153 nM T79062 CV2X5B 42635027 IC50 = 89 nM T79062 CBSD79 42635028 IC50 = 384 nM T79062 CR1S3J 42635029 IC50 = 339 nM T79062 CS9Q3H 42635204 IC50 = 12 nM T79062 C5XBV7 42635205 IC50 = 567 nM T79062 CQ2M5S 42635387 IC50 = 124 nM T79062 CR3KM7 42635388 IC50 = 107 nM T79062 C8TFQ9 42635389 IC50 = 580 nM T79062 CFO4Y1 42635570 IC50 = 223 nM T79062 CWU54L 42635571 IC50 = 373 nM T79062 CV27CE 42635572 IC50 = 377 nM T79062 CJ3NP5 42636941 IC50 > 1000 nM T79062 C0AI7N 43229249 Ki = 354.81 nM T79062 C2RSL9 43840296 Ki = 226 nM T79062 CJ41QV 44126269 Ki = 0.389 nM T79062 CVG6X1 44209472 Ki = 208 nM T79062 CD5AB7 44209480 Ki = 90 nM T79062 C2FDB1 44250364 IC50 > 10000 nM T79062 C8MC0Q 44251387 IC50 > 10000 nM T79062 C5YEA8 44251388 IC50 > 10000 nM T79062 C0BSF6 44251389 IC50 > 10000 nM T79062 CP8S2J 44266156 Ki = 4.467 nM T79062 CM0CW8 44266160 Ki = 6.918 nM T79062 C0P8IF 44266163 Ki = 0.4074 nM T79062 CU67NF 44266164 Ki = 9.333 nM T79062 C14ACY 44266178 Ki = 37.15 nM T79062 CN3ES2 44266182 Ki = 2.042 nM T79062 CKLS45 44266203 Ki = 14.13 nM T79062 CARU58 44266221 Ki = 0.5623 nM T79062 CA1WJ4 44266222 Ki = 2.754 nM T79062 CS2MU8 44266229 Ki = 20.42 nM T79062 CZ84XC 44266244 Ki = 9.12 nM T79062 CR16DY 44266245 Ki = 11.75 nM T79062 CVHM20 44266253 Ki = 27.54 nM T79062 CK7AF0 44266267 Ki = 25.12 nM T79062 C1FTY0 44266268 Ki = 1.66 nM T79062 CU61ZS 44266284 Ki = 11.22 nM T79062 C0C6RL 44266289 Ki = 10.23 nM T79062 C5NS9O 44266315 Ki = 2.512 nM T79062 CO5H2Q 44266317 Ki = 18.62 nM T79062 C6OW2N 44268087 Ki = 32 nM T79062 CNHE76 44276598 Ki = 2.138 nM T79062 CC2OD4 44278111 Ki > 10000 nM T79062 CRMA84 44278114 Ki = 713 nM T79062 CF0Y4M 44278115 Ki > 10000 nM T79062 CA93MC 44319240 Ki = 12.59 nM T79062 C34FTE 44319435 Ki = 8.318 nM T79062 CW16JD 44324737 Ki > 1000 nM T79062 CA84SN 44324765 Ki > 1000 nM T79062 COA3H4 44324800 Ki > 1000 nM T79062 CY04JW 44324972 Ki > 1000 nM T79062 C5VLY2 44326733 Ki = 9 nM T79062 CT7DN4 44327688 Ki = 2.399 nM T79062 CER86D 44327952 Ki = 83 nM T79062 CP9B2K 44340834 Ki = 1.82 nM T79062 CB23YQ 44340835 Ki = 0.7943 nM T79062 CC25ZK 44340836 Ki = 0.5012 nM T79062 CZBQ72 44340850 Ki = 0.8318 nM T79062 CTM65V 44340854 Ki = 0.7079 nM T79062 C6F9XL 44340882 Ki = 57.54 nM T79062 C2S1ZT 44340883 Ki = 6.457 nM T79062 CG6PD8 44340897 Ki = 22.91 nM T79062 CQ3WH6 44341114 Ki = 6.31 nM T79062 C9BDG2 44341126 Ki = 6.457 nM T79062 CK37NE 44341130 Ki = 25.7 nM T79062 CO0ZY5 44341131 Ki = 165.96 nM T79062 CD9ZS8 44342270 IC50 = 849 nM T79062 CPWJ26 44343212 Ki = 39.81 nM T79062 CMX45U 44348383 IC50 = 2.2 nM T79062 CUXH48 44352308 Ki = 1460 nM T79062 C3LKN1 44364048 Ki = 3.162 nM T79062 CND4W7 44368304 Ki = 19.95 nM T79062 C6CUM2 44368306 Ki = 31.62 nM T79062 CH3G4F 44368358 Ki = 31.62 nM T79062 C2S8AQ 44368373 Ki = 100000 nM T79062 C1EO8C 44368383 Ki = 1584.89 nM T79062 CAEZ93 44368384 Ki = 630.96 nM T79062 CK9OQ3 44368683 Ki = 125.89 nM T79062 CB0E1J 44368705 Ki = 10 nM T79062 CS21UK 44368731 Ki = 1.995 nM T79062 CRF67K 44368732 Ki = 3.981 nM T79062 C61PEQ 44368754 Ki = 15.85 nM T79062 CT2BR5 44372581 Ki = 5.012 nM T79062 C08EKS 44374206 Ki = 1200 nM T79062 CVL3U2 44374207 Ki = 7.2 nM T79062 CV8CP3 44374225 Ki = 22 nM T79062 C7FE5A 44374226 Ki = 6800 nM T79062 CX9S1K 44374227 Ki = 3200 nM T79062 C04WKH 44374233 Ki = 4.1 nM T79062 CB2S7T 44374234 Ki = 100 nM T79062 CV62ZP 44374298 Ki = 170 nM T79062 CJ4A2U 44374299 Ki = 12 nM T79062 C4VXQ1 44388858 Ki = 4.3 nM T79062 CTPG47 44388956 Ki > 2000 nM T79062 C1UMV6 44393001 Ki = 60 nM T79062 C64IKJ 44393004 Ki = 4 nM T79062 CT8Y5A 44393007 Ki = 4 nM T79062 C1F5IX 44393021 Ki = 13 nM T79062 C9VH1B 44393022 Ki = 16 nM T79062 CG9S1O 44393045 Ki = 2 nM T79062 CGRD59 44393052 Ki = 23 nM T79062 CBJ84O 44393053 Ki = 54 nM T79062 CPS9T7 44393056 Ki > 1000 nM T79062 C4HVE3 44393057 Ki > 1000 nM T79062 CKV3Z0 44393069 Ki = 3 nM T79062 C7HIJ9 44393072 Ki = 10 nM T79062 C20PMS 44393073 Ki = 0.4 nM T79062 C1E0QH 44393074 Ki = 36 nM T79062 C3H6ML 44393075 Ki = 8 nM T79062 C53UVJ 44393088 Ki = 2 nM T79062 C89NKB 44393089 Ki > 1000 nM T79062 C2QX0I 44393090 Ki > 1000 nM T79062 C0F9MP 44393091 Ki = 0.3 nM T79062 CCS5Q4 44393092 Ki = 0.4 nM T79062 C1KBZ7 44393093 Ki > 1000 nM T79062 CO6EY0 44393113 Ki = 2 nM T79062 C9GEU3 44393114 Ki = 33 nM T79062 CX4C9P 44393133 Ki = 6 nM T79062 CE03ZW 44393134 Ki = 1 nM T79062 C69CFB 44393154 Ki > 41000 nM T79062 CP9K0J 44393161 Ki = 2 nM T79062 CY60BQ 44393162 Ki > 1000 nM T79062 CG5UE1 44393169 Ki = 0.3 nM T79062 CG18AU 44393170 Ki = 5 nM T79062 CZ18RL 44393171 Ki = 5 nM T79062 CHV6D3 44393180 Ki = 0.6 nM T79062 CZB65R 44393192 Ki = 0.4 nM T79062 CK85EB 44393193 Ki = 0.4 nM T79062 CVC86L 44393228 Ki = 3 nM T79062 C7AR1C 44393229 Ki = 4 nM T79062 C4B0OI 44397588 Ki = 1000 nM T79062 C5FP0R 44397589 Ki = 1258.93 nM T79062 CE3G8U 44397670 Ki = 3981.07 nM T79062 CX7O9S 44401041 Ki = 80 nM T79062 C5XC2B 44401042 Ki = 92 nM T79062 CD56EA 44401105 Ki = 35 nM T79062 CW3PC2 44401106 Ki = 34 nM T79062 C9WH7P 44401164 Ki = 6.2 nM T79062 C9CWX1 44401194 Ki = 57 nM T79062 CXT84G 44401243 Ki = 251 nM T79062 C1B4QL 44403095 Ki > 10000 nM T79062 C1YL7Z 44403098 Ki > 10000 nM T79062 CFV98A 44403101 Ki > 10000 nM T79062 C6OY9S 44403102 Ki > 10000 nM T79062 CH4SX6 44403105 Ki > 10000 nM T79062 C4LKC1 44404394 Ki = 342 nM T79062 C3EJ4G 44404396 Ki > 10000 nM T79062 CG87PW 44409290 Ki > 1000 nM T79062 CXO64D 44437860 Ki = 107 nM T79062 CWO35N 44437861 Ki > 5000 nM T79062 CKZF16 44439165 Ki = 39.81 nM T79062 CA4HZ3 44439167 Ki = 79.43 nM T79062 CRC2Y5 44439387 Ki = 800 nM T79062 C3ZT7I 44439388 Ki = 3500 nM T79062 CKU9N8 44439389 Ki = 7800 nM T79062 C20VDP 44439390 Ki = 45 nM T79062 C6RKA9 44439391 Ki = 36 nM T79062 CI9D7G 44439392 Ki = 20 nM T79062 CDE27X 44439393 Ki = 35 nM T79062 CIQW67 44439394 Ki = 170 nM T79062 CV93LJ 44439395 Ki = 46 nM T79062 CPX5Q2 44439396 Ki = 200 nM T79062 C2R0SX 44439397 Ki = 2200 nM T79062 C4CMV7 44439398 Ki = 400 nM T79062 C8YQ4P 44439399 Ki = 500 nM T79062 C6YA9O 44439400 Ki = 5300 nM T79062 C89ZPX 44439401 Ki = 25000 nM T79062 CE60JL 44439402 Ki = 2700 nM T79062 C65GSE 44439403 Ki = 1000 nM T79062 CKUG90 44439404 Ki = 100 nM T79062 CTYP87 44439405 Ki = 300 nM T79062 C3UBA6 44439406 Ki > 300000 nM T79062 C7HV8X 44439407 Ki = 36000 nM T79062 CD4T3S 44439408 Ki = 200 nM T79062 C07XPE 44439409 Ki = 100 nM T79062 CMU43Q 44439410 Ki = 3600 nM T79062 C2S6HQ 44448054 Ki = 55 nM T79062 C3Z7FI 44451927 IC50 = 119.95 nM T79062 CSD7R5 44451929 IC50 = 2197.86 nM T79062 C3MCY7 44451930 IC50 = 1300 nM T79062 C3R7BH 44451931 IC50 = 369.83 nM T79062 CRFN53 44451952 IC50 = 260.02 nM T79062 CZE3T1 44451953 IC50 = 199.99 nM T79062 CJTX92 44451954 IC50 = 190 nM T79062 CINR86 44451957 IC50 = 2500 nM T79062 CK4GN8 44451959 IC50 = 500 nM T79062 CL29TJ 44451979 IC50 = 620 nM T79062 C57SBC 44451980 IC50 = 16 nM T79062 CEST18 44451982 IC50 = 54.95 nM T79062 CV7EY2 44451984 IC50 = 500 nM T79062 C7L9DK 44451985 IC50 = 939.72 nM T79062 C15JOU 44451986 IC50 = 510 nM T79062 CM34IO 44452005 IC50 = 190 nM T79062 C39KGW 44452006 IC50 = 269.77 nM T79062 CRN4F8 44452007 IC50 = 49 nM T79062 CY43VF 44452008 IC50 = 42 nM T79062 CW80FP 44452010 IC50 = 680 nM T79062 C3L6IQ 44452037 IC50 = 28.97 nM T79062 CR4N5K 44452038 IC50 = 1199.5 nM T79062 CN6PT7 44452039 IC50 = 130.02 nM T79062 CB0CK5 44452040 IC50 = 769.13 nM T79062 C74KEA 44452041 IC50 = 769.13 nM T79062 CL2EH4 44452042 IC50 = 8994.98 nM T79062 CO1W6H 44452078 IC50 = 97 nM T79062 CT2VN0 44452080 IC50 = 199.99 nM T79062 CA91RH 44452081 IC50 = 419.76 nM T79062 C6U4YS 44452082 IC50 = 928.97 nM T79062 C7DAM2 44452084 IC50 > 10000 nM T79062 CP1E6V 44452114 IC50 = 1000 nM T79062 COR7N6 44452115 IC50 = 16 nM T79062 C65HFP 44452117 IC50 = 470 nM T79062 C8F7IQ 44452118 IC50 = 349.95 nM T79062 CN4YL1 44452139 IC50 = 230 nM T79062 CMP20V 44452141 IC50 = 680 nM T79062 CG1C6X 44452142 IC50 = 92 nM T79062 C7A9JI 44452143 IC50 = 26 nM T79062 C78UTQ 44452144 IC50 = 1999.86 nM T79062 CQR12V 44452145 IC50 > 10000 nM T79062 CF3H6V 44452166 IC50 = 19 nM T79062 C6SC1Q 44452167 IC50 = 91 nM T79062 C56JMP 44452169 IC50 > 10000 nM T79062 CQ5U1I 44452170 IC50 = 20.99 nM T79062 CX8OK7 44452171 IC50 = 45 nM T79062 CS72NU 44452193 IC50 = 54.95 nM T79062 C5ZF1H 44452195 IC50 = 97.95 nM T79062 CTAP34 44452196 IC50 = 199.99 nM T79062 CUG1W4 44452197 IC50 = 420 nM T79062 C5DNK1 44452199 IC50 = 710 nM T79062 CA3Y7E 44452217 IC50 = 48 nM T79062 CFUM27 44452219 IC50 = 1100 nM T79062 CAI2D5 44452221 IC50 = 690 nM T79062 CVAU93 44452222 IC50 = 460.26 nM T79062 CD0CQ5 44452223 IC50 = 1400 nM T79062 C6TN5J 44452224 IC50 = 79.98 nM T79062 CD8AJ3 44452243 IC50 = 79 nM T79062 C69RGK 44452244 IC50 > 10000 nM T79062 C1HEZ2 44452245 IC50 = 110 nM T79062 CJD35V 44452246 IC50 = 84.92 nM T79062 C23DZP 44452247 IC50 = 159.96 nM T79062 CLPR24 44452249 IC50 = 449.78 nM T79062 CJY18I 44452251 IC50 = 1099.01 nM T79062 C0G6ZC 44452273 IC50 = 28.97 nM T79062 CD5IY1 44452274 IC50 = 210 nM T79062 CX4DR9 44452275 IC50 = 590 nM T79062 CDLB90 44452276 IC50 = 1500 nM T79062 C6CT8L 44452277 IC50 = 109.9 nM T79062 CF5G0O 44452278 IC50 = 130 nM T79062 CKU52M 44452279 IC50 = 639.73 nM T79062 CP4M7B 44452298 IC50 = 590.2 nM T79062 CMBT16 44452301 IC50 = 939.72 nM T79062 CFH72P 44452302 IC50 = 2398.83 nM T79062 CRE1X3 44452305 IC50 = 95 nM T79062 C4B8JL 44452324 IC50 = 74 nM T79062 C0B3LC 44452327 IC50 = 75 nM T79062 C6SF7C 44452328 IC50 = 449.78 nM T79062 C6V1WM 44452329 IC50 = 400 nM T79062 CQX6I3 44452331 IC50 = 650 nM T79062 C8HI7Q 44452332 IC50 = 730 nM T79062 CCHJ25 44452357 IC50 = 349.95 nM T79062 C5U3VQ 44452359 IC50 = 920 nM T79062 C2QBM9 44452362 IC50 = 7294.58 nM T79062 CZL97F 44455426 Ki = 116 nM T79062 CYS7T4 44455943 Ki = 73 nM T79062 C6BFI0 44456033 Ki = 6 nM T79062 CG91RD 44456395 Ki = 12.4 nM T79062 C12XGE 44456400 Ki = 1148.15 nM T79062 C13YGE 44460471 Ki = 31 nM T79062 CHA10N 44460639 Ki = 166 nM T79062 C7KP0I 44460641 Ki = 125 nM T79062 C7HNZ8 44460642 Ki = 140 nM T79062 CVF5C3 44460669 Ki = 109 nM T79062 CQ2ID1 44460701 Ki = 139 nM T79062 C9DUW7 44460708 Ki = 10 nM T79062 C4YB7R 44460724 Ki = 109 nM T79062 CN6K9F 44460725 Ki = 23 nM T79062 CF6A9J 44460738 Ki = 34 nM T79062 C46ZGA 44460739 Ki = 158 nM T79062 CV0PU6 44460744 Ki = 182 nM T79062 C8P1MO 44460759 Ki = 288 nM T79062 CCL32X 44460808 Ki = 88 nM T79062 C9UW7I 44460917 Ki = 70 nM T79062 C3PK8D 44460918 Ki = 145 nM T79062 CSI97R 44460980 Ki = 70 nM T79062 CCX4G5 44461045 Ki = 17 nM T79062 C0RE6D 44461048 Ki = 9 nM T79062 CR6J9L 44461052 Ki = 163 nM T79062 C05GVU 44461064 Ki = 1573 nM T79062 C7G4MW 44461065 Ki = 10 nM T79062 CKE9C5 44461066 Ki = 16 nM T79062 C62CSN 44461069 Ki = 37 nM T79062 CK5SR9 44461070 Ki = 14 nM T79062 C4DL5C 44469677 IC50 > 10000 nM T79062 CEX18U 44517732 Ki = 195 nM T79062 C3I9NZ 44517733 Ki = 339 nM T79062 C3D4HR 44537940 Ki > 5000 nM T79062 CJ7U3K 44554227 Ki > 5000 nM T79062 CM0I1P 44554393 Ki > 5000 nM T79062 CNHA47 44554395 Ki > 5000 nM T79062 C0NGQ3 44575261 IC50 > 150000 nM T79062 CEGL62 44576914 IC50 > 10000 nM T79062 CW8OI7 44576978 IC50 = 103 nM T79062 C1S9PB 44576979 IC50 > 10000 nM T79062 C0TN9C 44576980 IC50 > 10000 nM T79062 C3R0YE 44577013 IC50 > 10000 nM T79062 CRCH48 44582675 Ki = 59 nM T79062 CEJ4R8 44582676 Ki = 210 nM T79062 CZGP86 44582677 Ki = 5170 nM T79062 C5QB4K 44582678 Ki = 498 nM T79062 C01RCI 44582705 Ki = 731 nM T79062 CXL25V 44582706 Ki > 10000 nM T79062 C8MR1X 44582707 Ki = 6241 nM T79062 C4IT1N 44582708 Ki = 2862 nM T79062 CB0S4Z 44592109 IC50 > 1000 nM T79062 C6KTM4 45028192 Ki = 9549.93 nM T79062 C0DLU3 45109862 IC50 = 456 nM T79062 CGB2Z0 45113400 Ki = 42 nM T79062 CV1F6P 45268647 Ki = 276 nM T79062 CGZ08S 45269494 Ki = 198 nM T79062 CR2QP3 45272864 Ki = 177 nM T79062 CX15SL 45272891 Ki = 140 nM T79062 CTD71C 45273807 Ki = 161 nM T79062 C13MCR 45273816 Ki = 150 nM T79062 CZ71RN 45278805 IC50 = 333 nM T79062 CZN6M7 45278882 IC50 = 408 nM T79062 C6NT3Q 45278883 IC50 = 493 nM T79062 CS5BA4 45278886 IC50 = 524 nM T79062 C0CHF4 45482789 IC50 > 10000 nM T79062 CH90CZ 45488126 Ki > 500 nM T79062 CG9U2R 45488130 Ki > 500 nM T79062 C7N4GP 45488138 Ki > 500 nM T79062 CH29KP 45488139 Ki > 500 nM T79062 CDAJ27 45488143 Ki > 500 nM T79062 CZYC01 45488151 Ki > 500 nM T79062 C8PH0Y 45488152 Ki > 500 nM T79062 CC2OU0 45488156 Ki > 500 nM T79062 CL4G8T 45488165 Ki > 500 nM T79062 C5NDO6 45488166 Ki > 500 nM T79062 C0GMN4 45488171 Ki > 500 nM T79062 C3ZAL4 45488172 Ki > 500 nM T79062 C3PYL9 45488174 Ki > 500 nM T79062 CFT7C5 45488175 Ki > 500 nM T79062 CX1A2N 45488179 Ki > 500 nM T79062 CA8I7U 45488180 Ki > 500 nM T79062 C01QBM 45488181 Ki > 500 nM T79062 COX47A 45488183 Ki > 500 nM T79062 C8ETO2 45488184 Ki > 500 nM T79062 C5FQ4S 46224879 Ki = 0.2089 nM T79062 CXUL12 46232559 IC50 = 195 nM T79062 CU2RG8 46232560 IC50 = 456 nM T79062 C9RQ8U 46232586 IC50 = 110 nM T79062 C2B3ZP 46232587 IC50 = 87 nM T79062 C3I8TO 46232588 IC50 = 567 nM T79062 COW9V6 46232589 IC50 = 172 nM T79062 CGV2J5 46232620 IC50 = 678 nM T79062 CWHG97 46232621 IC50 = 980 nM T79062 CUQW08 46232622 IC50 = 1236 nM T79062 C5REP7 46232623 IC50 = 500 nM T79062 C2QOW0 46232652 IC50 = 888 nM T79062 C9I7XS 46232653 IC50 = 1508 nM T79062 C5D0BH 46232654 IC50 = 419 nM T79062 C5PAL9 46232689 IC50 = 24 nM T79062 CT5C0M 46232690 IC50 = 160 nM T79062 CF53BL 46232691 IC50 = 442 nM T79062 CE1ID7 46232729 IC50 = 2296 nM T79062 CN0CO9 46232730 IC50 = 152 nM T79062 C0VXA5 46232731 IC50 = 334 nM T79062 C1C4OF 46232732 IC50 = 147 nM T79062 CMR8O9 46232770 IC50 = 500 nM T79062 CTY9H7 46232771 IC50 = 121 nM T79062 C5TBE8 46232772 IC50 = 316 nM T79062 COH03R 46232773 IC50 = 124 nM T79062 CZ2W7X 46232817 IC50 = 93 nM T79062 C0N4YP 46232818 IC50 = 117 nM T79062 CTJ89I 46232819 IC50 = 188 nM T79062 CS98DM 46232820 IC50 = 342 nM T79062 C8P3HD 46232858 IC50 = 49.6 nM T79062 CP04TS 46232859 IC50 = 749 nM T79062 C8W0IJ 46232860 IC50 = 12.3 nM T79062 CF5M2T 46232861 IC50 = 6.3 nM T79062 C21CHG 46232975 IC50 = 35.3 nM T79062 CO41KX 46232976 IC50 = 657 nM T79062 CIK94R 46232977 IC50 = 316 nM T79062 CB67ST 46232978 IC50 = 363 nM T79062 CRU0F7 46233014 IC50 = 526 nM T79062 C7W5TE 46233349 Ki = 2240 nM T79062 C10LFM 46233350 Ki = 128 nM T79062 C5NT9Y 46233351 Ki = 1614 nM T79062 C4T3HL 46233352 Ki = 26 nM T79062 C75PCA 46233382 Ki = 669 nM T79062 CV2FO0 46233383 Ki = 1429 nM T79062 C0QBP6 46233384 Ki > 10000 nM T79062 CL54OR 46233385 Ki > 10000 nM T79062 C3RH1V 46233448 Ki > 10000 nM T79062 C8USF7 46233449 Ki = 1485 nM T79062 C69MQR 46233450 Ki = 0.3 nM T79062 CNGP15 46233483 Ki > 10000 nM T79062 C42SVX 46700866 IC50 > 10000 nM T79062 CD0K6E 46700867 IC50 = 5600 nM T79062 C5TC2S 46830335 IC50 > 10000 nM T79062 C1K7FL 46830336 IC50 > 10000 nM T79062 C1N4KX 46842383 IC50 > 10000 nM T79062 CC62SX 46866711 IC50 = 2874 nM T79062 C03LTM 46869265 Ki = 220000 nM T79062 CB8GE1 46884818 IC50 > 10000 nM T79062 C4MQ0A 46884856 IC50 > 10000 nM T79062 CCNT25 46884898 IC50 > 10000 nM T79062 C3MSG2 46885027 IC50 > 10000 nM T79062 CB7XI0 46885213 IC50 > 10000 nM T79062 CY28OS 47556338 Ki = 888 nM T79062 C2LZJ0 49783209 Ki = 5702 nM T79062 C57SMG 49783415 Ki > 10000 nM T79062 C0TG6I 49783419 Ki > 10000 nM T79062 CR40BA 49836386 IC50 > 1000 nM T79062 C4R2YS 49850567 Ki = 199.53 nM T79062 C07JTU 49850570 Ki = 39.81 nM T79062 CK68QR 49850672 Ki = 25.12 nM T79062 CN5XR1 49850772 Ki = 125.89 nM T79062 CR4EZ0 49850870 Ki = 100 nM T79062 C5K4EC 49850872 Ki = 63.1 nM T79062 C8AW0R 49850874 Ki = 79.43 nM T79062 C6OQV2 49862237 Ki = 15 nM T79062 C9KIU1 49864289 IC50 = 3038 nM T79062 CHO9C0 49864292 IC50 = 2044 nM T79062 C90MTG 49864602 IC50 = 1006 nM T79062 C5BCS4 49864722 IC50 = 4425 nM T79062 CKZO79 49864723 IC50 = 3865 nM T79062 C74LZS 49864724 IC50 = 2059 nM T79062 C2RY0J 50878551 Ki = 16.98 nM T79062 C1W6TV 50898777 Ki > 10000 nM T79062 CXMZ73 50898778 Ki > 10000 nM T79062 CX48AD 51002362 Ki = 1956 nM T79062 C8TA1J 51003550 IC50 > 10000 nM T79062 CQ1UJ7 51003551 IC50 = 2007 nM T79062 CGMI37 51003586 IC50 > 10000 nM T79062 CE4KP1 51050257 Ki > 10000 nM T79062 CT3HG0 52952098 Ki > 100000 nM T79062 CDM75V 52952099 Ki = 14125.38 nM T79062 CR0ES9 52952100 Ki > 100000 nM T79062 CI9BF4 52952200 Ki = 91201.08 nM T79062 C31KMJ 52952201 Ki > 100000 nM T79062 CG4AW2 52952202 Ki = 15135.61 nM T79062 C3KZA4 52952203 Ki > 100000 nM T79062 C0MC9X 52952204 Ki > 100000 nM T79062 CT7A6Q 52952304 Ki > 100000 nM T79062 CR96JZ 52952305 Ki > 100000 nM T79062 CN70EP 52952306 Ki > 100000 nM T79062 CUI85Q 52952307 Ki = 9120.11 nM T79062 CJ94KO 52952308 Ki = 7244.36 nM T79062 C39XRU 52952309 Ki = 4786.3 nM T79062 C53DTC 52952419 Ki = 53703.18 nM T79062 COZ2U3 52952420 Ki = 12589.25 nM T79062 CG0L5I 52952421 Ki = 8709.64 nM T79062 CHC1S3 52952422 Ki = 263.03 nM T79062 CP37CU 52952423 Ki > 100000 nM T79062 C6LRO4 52952424 Ki = 27542.29 nM T79062 CMJ62D 53245590 Ki = 930 nM T79062 CGY45S 53248361 Ki = 161 nM T79062 CE9L8G 53248365 Ki = 50 nM T79062 C61DNP 53320009 IC50 = 143 nM T79062 C9ZDR5 53320010 IC50 = 620 nM T79062 CQLK01 53322638 IC50 > 10000 nM T79062 C32YWL 53324045 Ki = 326 nM T79062 CY28UP 53324535 Ki = 14 nM T79062 CRQF15 53325242 Ki = 969 nM T79062 C70WHV 53361627 Ki = 404 nM T79062 CU4B6N 53370045 Ki = 125 nM T79062 CKQ6A3 53376040 Ki = 739 nM T79062 C65CWD 53377240 Ki > 10000 nM T79062 CSGU70 53377324 Ki = 418 nM T79062 CG24AT 53381002 Ki = 1985 nM T79062 CMOZ61 53475319 Ki = 770 nM T79062 C0J8XZ 54598062 Ki = 26 nM T79062 C8SJ1Z 54758201 Ki = 107 nM T79062 C6G2AC 54758202 Ki = 72 nM T79062 CU6HI4 54758203 Ki = 96 nM T79062 C5KGQ3 54758204 Ki = 11 nM T79062 CS6PX1 54758293 Ki = 5.1 nM T79062 C6X3OI 54758294 Ki = 139 nM T79062 CS9L0P 54758295 Ki = 4 nM T79062 CUD7N0 54758296 Ki = 52 nM T79062 C1H2GP 54758297 Ki = 16 nM T79062 CG3UJ4 54758298 Ki = 6.7 nM T79062 C89NYL 54758391 Ki = 40 nM T79062 CTH56O 54758392 Ki = 13 nM T79062 CAZ5T6 54764323 Ki = 13 nM T79062 COZ82F 55479093 Ki = 155 nM T79062 CW89BT 56595402 Ki > 1000 nM T79062 C4C3XQ 56595529 Ki > 1000 nM T79062 C6W1RA 56649648 Ki = 132 nM T79062 C2SW7J 56649649 Ki = 77 nM T79062 CQTR49 56649650 Ki = 97 nM T79062 CH37LU 56663451 IC50 > 10000 nM T79062 CJKO58 56852956 Ki = 338.84 nM T79062 C1ZG7A 56933434 Ki = 0.6 nM T79062 CO0N2W 56943599 Ki = 6.7 nM T79062 C3DF5Z 56943600 Ki = 3.2 nM T79062 C19BDH 56943695 Ki = 10 nM T79062 CS7K3T 56943891 Ki = 6.9 nM T79062 CZ4L3S 56944082 Ki = 0.1 nM T79062 C5NI3K 56944086 Ki = 67 nM T79062 C37BYO 56944186 Ki = 5.1 nM T79062 C9UOZ6 56944189 Ki = 5.9 nM T79062 CH7V9J 56944190 Ki = 5.1 nM T79062 CE49MC 56944191 Ki = 4.4 nM T79062 CX2RP5 56944287 Ki = 15 nM T79062 CB0P9N 56944383 Ki = 1.6 nM T79062 CEQ7I3 56944384 Ki = 1.3 nM T79062 CHWI01 56944473 Ki = 13 nM T79062 C6Y4ZQ 56944564 Ki = 1.8 nM T79062 C3B0MZ 56944565 Ki = 1.6 nM T79062 CI4KW0 56944664 Ki = 1.1 nM T79062 C39YHD 56944665 Ki = 0.8 nM T79062 C1W3GL 56944666 Ki = 1.4 nM T79062 C7J4UT 56944667 Ki = 1.5 nM T79062 CZT80U 56944668 Ki = 0.8 nM T79062 CTW2F5 56944763 Ki = 0.4 nM T79062 C50WEX 56944764 Ki = 1.1 nM T79062 CX0ZW2 56944859 Ki = 1.3 nM T79062 C1ST9U 56944860 Ki = 140 nM T79062 CQKL90 56944861 Ki = 110 nM T79062 CS5J6Y 56944862 Ki = 90 nM T79062 CFLB40 56944863 Ki = 65 nM T79062 C53OTR 56944864 Ki = 70 nM T79062 C5T3RI 56944951 Ki = 18 nM T79062 CR6H7U 56944952 Ki = 10 nM T79062 C1Y2RP 56944953 Ki = 6 nM T79062 C1BH7I 56944954 Ki = 2 nM T79062 CTK9I8 56944955 Ki = 29 nM T79062 CCF1A5 56944956 Ki = 2 nM T79062 C2YVT8 56945042 Ki = 51 nM T79062 CNI2G3 56945043 Ki = 17 nM T79062 CF9V3Q 56945045 Ki = 33 nM T79062 CE4S5M 56945046 Ki = 38 nM T79062 C1TC7Q 56963799 Ki > 10000 nM T79062 C3ZG6J 57325520 Ki = 56 nM T79062 CDK7B0 57325521 Ki = 47 nM T79062 CR9MZ4 57384073 Ki = 16 nM T79062 CO7BG0 57390335 Ki = 335 nM T79062 CP05DB 57390336 Ki = 235 nM T79062 C1TH4R 57390337 Ki = 41 nM T79062 CATM39 57390694 Ki = 2060 nM T79062 C6S0IE 57390695 Ki = 2810 nM T79062 C83GWU 57391158 Ki = 604 nM T79062 CPE8N4 57391622 Ki = 68 nM T79062 CHG51U 57391624 Ki = 36 nM T79062 CIHJ73 57392107 Ki = 55 nM T79062 CY02VL 57392108 Ki = 38 nM T79062 C93QRW 57393876 Ki = 267 nM T79062 CUF40C 57393877 Ki = 334 nM T79062 CR7FB5 57393878 Ki = 1255 nM T79062 C7VFQ3 57394663 Ki = 50 nM T79062 CEW0O4 57395084 Ki = 88 nM T79062 CL96RC 57395086 Ki = 25 nM T79062 CSI7X2 57395597 Ki = 360 nM T79062 CJ15YT 57395598 Ki = 228 nM T79062 CK53EW 57395599 Ki = 37 nM T79062 C51GCK 57396417 Ki = 207 nM T79062 CZ2SJ8 57396419 Ki = 40 nM T79062 CZ8KA2 57396855 Ki = 381 nM T79062 CN7QE4 57396857 Ki = 334 nM T79062 C2Q6CJ 57397410 Ki = 132 nM T79062 CFQA13 57397411 Ki = 995 nM T79062 C7W5XA 57398619 Ki = 113 nM T79062 CFT56H 57399088 Ki = 3010 nM T79062 CGX5Q1 57399089 Ki = 79 nM T79062 CTF76G 57399090 Ki = 156 nM T79062 C0XFB2 57399091 Ki = 90 nM T79062 CI6ET3 57399092 Ki = 29 nM T79062 CMX4K5 57399093 Ki = 33 nM T79062 CJ41PW 57399432 Ki = 413 nM T79062 CAN0W7 57399866 Ki = 145 nM T79062 C9BG7C 57399868 Ki = 126 nM T79062 C5HGO2 57400281 Ki = 69 nM T79062 CT7Q3E 57400828 Ki = 506829 nM T79062 CFBP89 57400829 Ki = 1420 nM T79062 C3D1UP 57400830 Ki = 187 nM T79062 C5GPJ0 57401515 Ki = 210 nM T79062 CG8MF3 57401516 Ki = 353 nM T79062 CZX05B 57401706 Ki = 291 nM T79062 CN9J5I 57402588 Ki = 224 nM T79062 C92HON 57402951 Ki = 356 nM T79062 CX0B5M 57403525 Ki = 1042 nM T79062 C3A1YW 57403839 Ki = 310 nM T79062 CA10YX 57403841 Ki = 335 nM T79062 CYSV60 60165411 Ki = 337 nM T79062 CB9GC6 60165412 Ki = 62.6 nM T79062 CI5PM3 60165413 Ki = 107 nM T79062 C2Q5VD 60165416 Ki = 329 nM T79062 C9JL3F 60165418 Ki = 228.9 nM T79062 C31PEN 60165535 Ki = 35.6 nM T79062 CP60YF 60165537 Ki = 211 nM T79062 C85OTH 60165541 Ki = 425.8 nM T79062 CJO91V 60165543 Ki = 2467 nM T79062 CJDC53 60165545 Ki = 242 nM T79062 C3K5JN 60165681 Ki = 2917 nM T79062 C5RUP6 60167166 Ki = 790 nM T79062 CRH49P 60167309 Ki = 983 nM T79062 COHK72 60167451 Ki = 125.89 nM T79062 C30SVG 60167452 Ki = 512.86 nM T79062 CB4HT7 60195992 Ki = 109 nM T79062 C4Q6LO 60195993 Ki = 1.9 nM T79062 C04CRJ 60195994 Ki = 93 nM T79062 C4BG3H 60195995 Ki > 5000 nM T79062 C87FDE 60195996 Ki = 7 nM T79062 C6VWY1 60196073 Ki = 13 nM T79062 CM92UX 60196074 Ki = 23 nM T79062 C18AVJ 60196075 Ki = 80 nM T79062 CZN64D 60196076 Ki = 96 nM T79062 CIN29U 60196077 Ki = 7.1 nM T79062 C3LTC1 60196078 Ki = 8.2 nM T79062 C7WLN1 60196079 Ki = 6.9 nM T79062 C5N3SG 60196080 Ki = 1.4 nM T79062 C6AUO2 66800823 Ki = 25 nM T79062 C34ACQ 66800909 Ki = 2 nM T79062 CGT9E6 66800910 Ki = 6.3 nM T79062 C0QY7D 66800916 Ki = 4.6 nM T79062 CM58FG 66800926 Ki = 200 nM T79062 CQ43WD 66800934 Ki = 19 nM T79062 CK0I5J 66800939 Ki = 1.5 nM T79062 C0X2SF 66800942 Ki = 3.8 nM T79062 CN30YT 66800947 Ki = 9 nM T79062 CZ3MR6 66800959 Ki = 180 nM T79062 C92CMO 66800965 Ki = 91 nM T79062 CFPK92 66800991 Ki = 6.3 nM T79062 C13GMO 66801000 Ki = 13 nM T79062 CZ1TF9 66801018 Ki = 2.6 nM T79062 CBO9U3 66801028 Ki = 8.8 nM T79062 C3K8DC 66801052 Ki = 80 nM T79062 CA4DM3 66801062 Ki = 4.1 nM T79062 C2OUX9 66801107 Ki = 1.7 nM T79062 C4J5RZ 66801115 Ki = 54 nM T79062 C1H8BS 66801116 Ki = 41 nM T79062 C4JGC6 66801120 Ki = 18 nM T79062 CX2GN1 66801139 Ki = 0.9 nM T79062 C1NG8S 66801140 Ki = 5.3 nM T79062 CR7OW6 66801158 Ki = 0.8 nM T79062 CJU53X 66801160 Ki = 9.5 nM T79062 CH3BJ8 66801167 Ki = 0.5 nM T79062 C0AV5M 66801173 Ki = 9.9 nM T79062 C0V9EF 66801186 Ki = 3.2 nM T79062 CTHY41 66801210 Ki = 0.7 nM T79062 CSD67P 66801225 Ki = 4.3 nM T79062 C8J3YU 66801226 Ki = 9.9 nM T79062 CX45OZ 66801229 Ki = 1.5 nM T79062 C1S0EV 66801230 Ki = 3.2 nM T79062 C7S1KY 66801234 Ki = 0.9 nM T79062 CB53AV 66801246 Ki = 14 nM T79062 C3F1TZ 66801251 Ki = 34 nM T79062 CF8O9U 66801259 Ki = 57 nM T79062 C2Q9FS 66801263 Ki = 0.7 nM T79062 C7Y9VP 66801267 Ki = 2500 nM T79062 CED17M 66801271 Ki = 0.9 nM T79062 C41VYW 66801295 Ki = 14 nM T79062 C2FYL1 66801333 Ki = 180 nM T79062 CS75LK 66801335 Ki = 29 nM T79062 CR2N0J 66801344 Ki = 15 nM T79062 CDH7S9 66801346 Ki = 1.2 nM T79062 CGC4U6 66801354 Ki = 120 nM T79062 CY4FM5 66801379 Ki = 3.4 nM T79062 C3RX4C 66801425 Ki = 120 nM T79062 C7JD0I 66801429 Ki = 24 nM T79062 CN8OU1 66801430 Ki = 150 nM T79062 C93EGP 66801455 Ki = 4.1 nM T79062 COR1H8 66801528 Ki = 80 nM T79062 C1F3YV 66801537 Ki = 69 nM T79062 CIRW86 66801551 Ki = 0.2 nM T79062 C75WXP 66801561 Ki = 240 nM T79062 C8H5PD 66801565 Ki = 1.3 nM T79062 CT5SP8 66801605 Ki = 9 nM T79062 C8MH0I 66801613 Ki = 20 nM T79062 CC8JV6 66801624 Ki = 520 nM T79062 C3EI2F 66801625 Ki = 150 nM T79062 C49XBJ 66801673 Ki = 34 nM T79062 C0XG6B 66801701 Ki = 380 nM T79062 C42EBQ 66801837 Ki = 610 nM T79062 CW3AI2 66803474 Ki = 0.6 nM T79062 CPKH06 66803497 Ki = 12 nM T79062 CNJE57 66803500 Ki = 61 nM T79062 CN6FZ1 66803595 Ki = 1 nM T79062 C1LEH8 67268994 Ki = 30 nM T79062 CLA7F3 68281136 Ki = 23 nM T79062 C84MZH 68281137 Ki = 270 nM T79062 CR5KY1 71061607 Ki = 18 nM T79062 C72XPZ 71061659 Ki = 23.8 nM T79062 CKE2Y4 71061750 Ki = 26.1 nM T79062 CD1ET2 71061756 Ki = 23.5 nM T79062 C5KM2W 71061887 Ki = 11.2 nM T79062 C0D5SC 71062035 Ki = 15.2 nM T79062 CNQ65S 71062123 Ki = 12.7 nM T79062 CC43QK 71151588 Ki = 180 nM T79062 C3PUX5 71449549 Ki = 27 nM T79062 CN82LY 71449550 Ki = 311 nM T79062 C40DOC 71449627 Ki = 276 nM T79062 C8U6NR 71449628 Ki = 709 nM T79062 C7Y6LC 71449629 Ki = 7 nM T79062 C91SZN 71449641 Ki = 13 nM T79062 C2GCN7 71449642 Ki = 121 nM T79062 CQN93U 71449643 Ki = 7 nM T79062 CEJ3B4 71449644 Ki = 16 nM T79062 C5SAJ1 71449645 Ki = 28 nM T79062 C3XNC2 71450247 Ki = 1914 nM T79062 C9VZ8J 71450550 Ki = 3505 nM T79062 C2IXB6 71451344 Ki = 409 nM T79062 C7DCR4 71451345 Ki = 1672 nM T79062 CC6QP7 71451441 Ki = 161 nM T79062 CHT21G 71451454 Ki = 2222 nM T79062 C2QZL4 71451455 Ki = 78 nM T79062 CXI5Q2 71451456 Ki = 2375 nM T79062 CKJZ57 71451457 Ki = 29 nM T79062 C0F1HU 71451458 Ki = 15 nM T79062 CTZ24N 71451459 Ki = 6 nM T79062 C70JUP 71451460 Ki = 4 nM T79062 C4NDR3 71452382 Ki = 6259 nM T79062 C6ZWV2 71452383 Ki = 6873 nM T79062 CGO4M1 71453156 Ki = 815 nM T79062 C6EFP9 71453157 Ki = 391 nM T79062 CUK2P5 71453252 Ki = 12 nM T79062 CKI58Z 71453278 Ki = 21 nM T79062 C1QM8D 71453279 Ki = 58 nM T79062 C6O4KT 71453280 Ki = 9 nM T79062 CL49VI 71453281 Ki = 4 nM T79062 CGXT64 71453282 Ki = 12 nM T79062 CQ3XC8 71454898 Ki = 865 nM T79062 CWY38Z 71454899 Ki = 1188 nM T79062 CGO13Q 71454997 Ki = 20 nM T79062 C0K1JV 71454998 Ki = 46 nM T79062 C3JF1D 71454999 Ki = 0.3 nM T79062 C2QZ1N 71455000 Ki = 7 nM T79062 C6FE5D 71455001 Ki = 293 nM T79062 C4L0JN 71455002 Ki = 2 nM T79062 C8YH0J 71455083 Ki = 60 nM T79062 CAQF34 71455625 Ki = 1945 nM T79062 C6G2HC 71455894 Ki = 3647 nM T79062 C5O6LT 71456677 Ki = 1500 nM T79062 CLX0G4 71456770 Ki = 85 nM T79062 CE19SD 71456779 Ki = 97 nM T79062 CWR40I 71456780 Ki = 2195 nM T79062 CZUX67 71456781 Ki = 10 nM T79062 CZ17FC 71456782 Ki = 9 nM T79062 CKF09U 71456783 Ki = 16 nM T79062 CJKV72 71456784 Ki = 10 nM T79062 C7MNB5 71457264 Ki = 6371 nM T79062 CMJ1O9 71457409 Ki = 1018 nM T79062 CVI7S2 71457690 Ki = 2447 nM T79062 CG83QI 71458516 Ki = 334 nM T79062 CE6OC0 71458622 Ki = 1144 nM T79062 CZ8L0D 71458623 Ki = 17 nM T79062 CW79AY 71458624 Ki = 59 nM T79062 C2XV5L 71458625 Ki = 5 nM T79062 CUAC42 71458626 Ki = 5 nM T79062 C37EBC 71458647 Ki = 60 nM T79062 CM6OP1 71458648 Ki = 1362 nM T79062 CRGE05 71458649 Ki = 1438 nM T79062 CJN4S1 71458650 Ki = 14 nM T79062 CNT5J9 71458651 Ki = 10 nM T79062 C3NAM7 71458652 Ki = 11 nM T79062 CS83IF 71459269 Ki = 150 nM T79062 CK5T4P 71459604 Ki = 3601 nM T79062 CG0WO9 71459954 Ki = 329 nM T79062 CMW0T6 71460453 Ki = 93 nM T79062 C9W7CF 71460454 Ki = 3372 nM T79062 C09VSE 71460455 Ki = 1104 nM T79062 CBU8J7 71460456 Ki = 2224 nM T79062 CT17XB 71460468 Ki = 178 nM T79062 C63YLA 71461049 Ki = 3473 nM T79062 CJD96I 71461050 Ki = 384 nM T79062 CZ6G8V 71462064 Ki = 2674 nM T79062 CI0K3L 71462065 Ki = 415 nM T79062 CD0G8Q 71462066 Ki = 407 nM T79062 CK5JC7 71462067 Ki = 329 nM T79062 C42IZX 71462068 Ki = 873 nM T79062 CB30LT 71462154 Ki = 204 nM T79062 C7Y1XU 71462155 Ki = 427 nM T79062 CLS2A6 71462156 Ki = 1108 nM T79062 C7AX1Q 71462178 Ki = 41 nM T79062 C1CS0Z 71462179 Ki = 27 nM T79062 C4P3JU 71462776 Ki = 153 nM T79062 C3GUQ2 71462777 Ki > 10000 nM T79062 CT2ME3 71574204 Ki = 21 nM T79062 C3SXR5 71574206 Ki = 46 nM T79062 C2YRI9 71574208 Ki = 31 nM T79062 C62RWV 71574210 Ki = 12 nM T79062 CKC53S 71574212 Ki = 30 nM T79062 CNV42M 71574298 Ki = 41 nM T79062 C9PGQ1 71574300 Ki = 124 nM T79062 C2LXH5 71574302 Ki = 31 nM T79062 C2YPB8 71574304 Ki = 27 nM T79062 CK7GM0 71574306 Ki = 56 nM T79062 C7EQ2F 71602523 Ki = 537 nM T79062 C29INM 71602524 Ki > 10000 nM T79062 CK2C5Q 71602525 Ki > 10000 nM T79062 C1T0VP 71602526 Ki > 10000 nM T79062 C4BFZ0 71602581 Ki > 10000 nM T79062 C82MIC 71602582 Ki > 10000 nM T79062 C69MFB 71602583 Ki = 432 nM T79062 CG21CD 71602584 Ki > 10000 nM T79062 CQZ2O3 71602585 Ki > 10000 nM T79062 C9UE3T 71602586 Ki = 1850 nM T79062 C6B4VK 71602587 Ki = 1737.8 nM T79062 C9XWR8 71602639 Ki = 1200 nM T79062 CH91JF 71602640 Ki = 2754.23 nM T79062 C2KRC8 71602641 Ki > 10000 nM T79062 C1I9AS 71602642 Ki > 10000 nM T79062 CW3Z9S 71602643 Ki > 10000 nM T79062 C6MH1U 71602644 Ki > 10000 nM T79062 CKR10Z 71602687 Ki = 658 nM T79062 C3ZQ5D 71602688 Ki = 295.12 nM T79062 CJ89YE 71602689 Ki = 218.78 nM T79062 C6L3DJ 71602690 Ki = 199.53 nM T79062 C2ABS7 71602691 Ki = 309.03 nM T79062 CI86QM 71602692 Ki = 42.66 nM T79062 CC45VZ 71602739 Ki = 77 nM T79062 CXP3V8 71602740 Ki = 45.71 nM T79062 CVL36N 71678345 Ki = 1659.59 nM T79062 C0PF3I 71678857 Ki = 15 nM T79062 C0W2YA 71727193 Ki = 195 nM T79062 C79TLS 71727194 Ki = 16950 nM T79062 CFB10W 71727195 Ki = 13500 nM T79062 C6CIB5 71727196 Ki = 1145 nM T79062 C7Z3JS 71727308 Ki = 426 nM T79062 C3ATN5 72197484 IC50 = 1564 nM T79062 C20HSN 72197485 IC50 = 1059 nM T79062 CN8A5R 72197486 IC50 = 1003 nM T79062 CL3BF7 72197668 IC50 = 497 nM T79062 CUVJ59 72197845 Ki = 196 nM T79062 CIKU20 72198011 Ki = 345 nM T79062 COH95V 72198014 Ki = 589 nM T79062 C0WY2V 72198191 Ki = 1165 nM T79062 C7AOY4 72198754 IC50 = 62 nM T79062 C4M7KP 72198756 IC50 > 100 nM T79062 CWHF29 72547876 Ki = 43.7 nM T79062 CF47JC 72547878 Ki = 32.4 nM T79062 C12CIH 72548115 Ki = 26.1 nM T79062 C1UX8Q 72548117 Ki = 47.6 nM T79062 C4K1WO 72548349 Ki = 66.1 nM T79062 CWH6T3 72548703 IC50 = 0.39 nM T79062 C4T0SK 72549767 Ki = 186.5 nM T79062 CE4U6J 72549768 Ki = 64.5 nM T79062 C1QZ4F 72549986 Ki = 37.9 nM T79062 C17XNV 72549988 Ki = 43.7 nM T79062 CD7V6P 72550196 Ki = 36.5 nM T79062 C1SZ3K 72550200 Ki = 34.7 nM T79062 C62EFS 72550423 Ki = 34.7 nM T79062 CK0F1L 72550641 Ki = 46.6 nM T79062 C8Z0NM 72550642 Ki = 8.69 nM T79062 CL6W2Q 72550645 Ki = 15.9 nM T79062 CUH4Z3 72550864 Ki = 405.3 nM T79062 C9J4QU 72550865 Ki = 25.9 nM T79062 C8A3DU 72551082 Ki = 31.4 nM T79062 C78LYM 72698087 Ki > 10000 nM T79062 C63HPK 72698088 Ki > 10000 nM T79062 C7W4RH 72734860 Ki = 12.4 nM T79062 C8UCZ5 72734861 Ki > 100 nM T79062 CZ6SQ7 72734863 Ki = 42 nM T79062 C8JT6B 72734864 Ki = 144 nM T79062 CW4IB9 72734866 Ki > 1000 nM T79062 CY0AE3 72735038 Ki = 239 nM T79062 CAZ84Y 72735039 Ki > 1000 nM T79062 C0MT4E 72735040 Ki > 1000 nM T79062 C0CK8H 72735041 Ki > 100 nM T79062 CC6Q5R 72771081 Ki < 100 nM T79062 CC65OA 73213195 Ki = 199.53 nM T79062 CW83DK 73213196 Ki = 194.98 nM T79062 CCV91B 73346042 Ki = 17.2 nM T79062 CXM8O2 73347306 IC50 = 3100 nM T79062 C9X8GY 73347307 IC50 > 1000 nM T79062 C4ZM8R 73347582 Ki = 9.7 nM T79062 C6BS5L 73349361 Ki = 4423 nM T79062 CL38VQ 73351112 Ki > 1000 nM T79062 CC8I7X 73351903 IC50 = 1800 nM T79062 CG4M8P 73351905 IC50 = 3700 nM T79062 CAR7Z5 73354882 IC50 = 480 nM T79062 CET52A 73356443 IC50 = 690 nM T79062 CUB97Z 74538690 Ki = 35 nM T79062 C2E7QW 75201901 Ki = 7800 nM T79062 C8IDL3 75306277 Ki = 79.43 nM T79062 CX17RZ 76280896 Ki = 71 nM T79062 C45OSP 76284193 Ki = 53 nM T79062 C0CRJ1 76284452 Ki = 34.5 nM T79062 CS17IJ 76284453 Ki = 12.8 nM T79062 CH82JU 76284455 Ki = 45.2 nM T79062 CRO7Q9 76284721 Ki = 15.9 nM T79062 C4BIC2 76284724 Ki = 3.82 nM T79062 C0EKY7 76284725 Ki = 66.7 nM T79062 C3GXV8 76310809 Ki = 1200 nM T79062 C19EPD 76310810 Ki = 48 nM T79062 CK2X7A 76310812 Ki = 92 nM T79062 CXJG08 76314094 Ki > 1000 nM T79062 CN7GD5 76314435 Ki = 317 nM T79062 CLO9M1 76314437 Ki = 1920 nM T79062 CD8A5H 76318011 Ki = 6.9 nM T79062 C1Y9SX 76318012 Ki = 20 nM T79062 CEHK31 76321734 Ki = 4.5 nM T79062 C5F1XU 76321735 Ki = 4.5 nM T79062 CC8TR0 76321736 Ki = 70 nM T79062 C94VNF 76324975 Ki = 64.2 nM T79062 C18OSZ 76325346 Ki = 17 nM T79062 C62CZO 76325348 Ki = 27 nM T79062 COGC62 76325350 Ki = 18 nM T79062 C1Q5NC 76325352 Ki = 8.7 nM T79062 CZ6P1E 76328545 Ki > 1000 nM T79062 C0OI2M 76328889 Ki = 283 nM T79062 C51CME 76328891 Ki = 41 nM T79062 CBFE85 76328893 Ki = 62 nM T79062 C5WG9E 76328895 Ki = 60 nM T79062 C6OV4J 76328897 Ki = 65 nM T79062 CL83OY 76332574 Ki = 649 nM T79062 CN3QO1 76332576 Ki = 15 nM T79062 CDBS57 76332578 Ki = 34 nM T79062 C97OVP 76332580 Ki = 4440 nM T79062 C1LT6C 76332582 Ki = 3907 nM T79062 CP0D6T 76332584 Ki = 94 nM T79062 CW3AK0 76335863 Ki = 33.4 nM T79062 CYT34W 76336176 Ki = 33 nM T79062 C9XFL1 76336178 Ki = 18 nM T79062 C0GD2B 76336180 Ki = 20 nM T79062 CV90GC 76336182 Ki = 189 nM T79062 C51CXD 76336183 Ki = 54 nM T79062 CMG58X 76336185 Ki = 10.8 nM T79062 C28RIZ 76518514 Ki = 472 nM T79062 C9S0XK 86288947 Ki = 3 nM T79062 CEPC94 86288948 Ki = 3 nM T79062 CHE2U4 90178632 Ki = 16 nM T79062 CFDW68 90644074 Ki = 10 nM T79062 C0T8RE 90644075 Ki = 380 nM T79062 C2KE9G 90644076 Ki = 94 nM T79062 C1SOF5 90644077 Ki = 150 nM T79062 CIE9Z2 90644078 Ki = 900 nM T79062 C37CYS 90654670 Ki = 101 nM T79062 C0IQ5R 90654671 Ki = 51 nM T79062 CVG2C1 90654672 Ki = 78 nM T79062 CU0ON1 90654673 Ki = 111 nM T79062 CJR3Y9 90654674 Ki = 148 nM T79062 CO1H4U 90654675 Ki = 551 nM T79062 CAY64Z 90654676 Ki = 302 nM T79062 CH0R8B 90654677 Ki = 579 nM T79062 CRFB56 90654678 Ki = 476 nM T79062 CPR21O 90654679 Ki = 393 nM T79062 C6YLV3 90654680 Ki = 725 nM T79062 CGUY51 90654681 Ki = 223 nM T79062 CK8X4O 90654682 Ki = 295 nM T79062 CH8UQ9 90654683 Ki = 107 nM T79062 CTQ23Z 90654684 Ki = 95 nM T79062 C9Q2JW 90654685 Ki = 1196 nM T79062 C98TJR 90654686 Ki = 18 nM T79062 CG3OI7 90654687 Ki = 22 nM T79062 CKTV83 90654688 Ki = 28 nM T79062 CVK85U 90654689 Ki = 163 nM T79062 CLG75D 90654690 Ki = 153 nM T79062 C7T9HW 90654691 Ki = 495 nM T79062 C92BZL 90654692 Ki = 567 nM T79062 C6CD9R 90654693 Ki = 634 nM T79062 C6H9NV 90654694 Ki = 1199 nM T79062 CR74SD 90654695 Ki = 4151 nM T79062 C7VM4O 90654696 Ki = 1865 nM T79062 CGFU53 90654697 Ki = 1312 nM T79062 C7BEZ8 90654698 Ki = 3134 nM T79062 CZ3IM2 90654699 Ki = 478 nM T79062 C8TMK5 90654700 Ki = 1188 nM T79062 C7GK3C 90654701 Ki = 113 nM T79062 CN8BO1 90654702 Ki = 179 nM T79062 CHIW63 90654703 Ki = 108 nM T79062 C1SAW2 90654704 Ki = 50 nM T79062 CJG31T 90654831 Ki = 95 nM T79062 CMU45O 90654832 Ki = 77 nM T79062 C3C4BW 90654834 Ki = 157 nM T79062 C8QWR3 90654835 Ki = 34 nM T79062 C6ZR9L 90654837 Ki = 70 nM T79062 C0AC7R 90654839 Ki = 72 nM T79062 CKLG40 90654841 Ki = 122 nM T79062 C5JS8D 90654843 Ki = 135 nM T79062 C4VHZ6 90654845 Ki = 45 nM T79062 CG78PS 90654847 Ki = 172 nM T79062 CL39WP 90654849 Ki = 123 nM T79062 C0TVQ9 90654851 Ki = 46 nM T79062 C4I1CU 90654853 Ki = 31 nM T79062 CZ28YC 90654855 Ki = 78 nM T79062 CRO83N 90654857 Ki = 456 nM T79062 C72RKV 90656669 Ki = 20.8 nM T79062 CJ8H1R 90656670 Ki = 92.5 nM T79062 CSF25H 90656671 Ki = 90.1 nM T79062 CGD60Y 90656672 Ki = 12.1 nM T79062 C4H1SB 90656673 Ki = 81.4 nM T79062 CID83U 90656674 Ki = 161.4 nM T79062 C0VDH3 90656675 Ki = 252.1 nM T79062 CC1L7T 90656676 Ki = 57 nM T79062 CCQU80 90656678 Ki = 84.8 nM T79062 CNSW31 90656679 Ki = 161.2 nM T79062 CITS52 90656680 Ki = 179.2 nM T79062 C3GA5B 90656681 Ki = 111.7 nM T79062 C9SX5R 90656682 Ki = 10.1 nM T79062 CGEF35 90656683 Ki = 2.9 nM T79062 C76OIR 90656684 Ki = 434.2 nM T79062 CH9F4Q 90656685 Ki = 20 nM T79062 C8NB7D 90656686 Ki = 161.1 nM T79062 C13YLN 90656687 Ki = 39.6 nM T79062 CU82QN 90656688 Ki = 63.3 nM T79062 CNB76X 90656689 Ki = 77.9 nM T79062 CPQ46T 90656690 Ki = 108.8 nM T79062 C6QO1P 90656691 Ki = 13.2 nM T79062 C6TF2G 90656692 Ki = 8.1 nM T79062 CGP76X 90656694 Ki = 30 nM T79062 C3O2KS 90656695 Ki = 16.7 nM T79062 CYLZ26 90656696 Ki = 12 nM T79062 C9RH6O 90656697 Ki = 226 nM T79062 C5MP1J 90656699 Ki = 39.4 nM T79062 C5L9IQ 90656701 Ki = 95.6 nM T79062 C6NG4Q 90656703 Ki = 191 nM T79062 C63JKH 90656705 Ki = 137.5 nM T79062 C7NV3E 90656707 Ki = 242.1 nM T79062 CK6UO3 90656708 Ki = 310 nM T79062 C6N5CS 90656709 Ki = 40 nM T79062 CX49HI 90656710 Ki = 3.1 nM T79062 CRX47O 90656711 Ki = 11.6 nM T79062 CTHD25 90656712 Ki = 6.6 nM T79062 CID86Z 90656713 Ki = 12.8 nM T79062 C5Q8PH 90656714 Ki = 63.1 nM T79062 CS9E1R 90656715 Ki = 332 nM T79062 CCOV98 90664359 Ki = 10490 nM T79062 CA8B0H 90664441 Ki = 328 nM T79062 CP48OR 90664581 Ki = 612 nM T79062 C4MUI2 90664601 IC50 = 11 nM T79062 CXD5Q9 90664621 Ki = 17420 nM T79062 CP2MK1 90664692 Ki = 5800 nM T79062 CO9H3P 90664694 Ki = 153 nM T79062 CE6D5M 90664808 Ki = 296 nM T79062 CT7Z1V 90664944 Ki = 184 nM T79062 CHT7D5 90664962 IC50 = 6.8 nM T79062 CQCE48 90665063 Ki = 276 nM T79062 C4EQ5K 90665189 Ki = 484 nM T79062 C0J5YH 91864602 Ki = 3.548 nM T79062 CDWS84 91937906 Ki = 157 nM T79062 CEN10X 92042876 Ki = 5.2 nM T79062 CW6XB3 92042877 Ki = 15 nM T79062 CUQ6V0 92042918 Ki < 1000 nM T79062 CS62HU 101747513 Ki = 5.6 nM T79062 C4DG3V 102364516 Ki = 0.7 nM T79062 C4WDR8 109018769 Ki = 4.34 nM T79062 CD76TH 109026949 Ki = 52 nM T79062 C3DMI5 109026956 Ki = 29.5 nM T79062 C2G0WH 109026957 Ki = 23.5 nM T79062 CYB18Z 109027017 Ki = 26.2 nM T79062 C0M3CD 118051679 Ki = 42 nM T79062 CEMZ15 118464420 Ki = 401 nM T79062 CV2L6O 118464425 Ki = 516 nM T79062 CFNG86 118464427 Ki = 427 nM T79062 CMSN80 118626035 Ki = 19 nM T79062 CT3AI0 118626042 Ki = 75 nM T79062 CKNJ72 118626045 Ki = 23 nM T79062 CGB42Y 118626088 Ki = 66 nM T79062 C0XJT5 118626089 Ki = 19 nM T79062 CIE4C7 118626101 Ki = 4 nM T79062 C1NYS5 118626120 Ki = 142 nM T79062 CPG04R 118626121 Ki = 3 nM T79062 C3S5LJ 118626129 Ki = 1 nM T79062 CY3F0N 118626140 Ki = 97 nM T79062 CE07IQ 118626142 Ki = 4 nM T79062 C72OZY 118626161 Ki = 1 nM T79062 CY3E7S 118626169 Ki = 52 nM T79062 CHRB75 118626208 Ki = 349 nM T79062 CSN13R 118706278 Ki = 41 nM T79062 CIG56H 118706280 Ki > 1000 nM T79062 CF5ZR8 118706282 Ki = 14 nM T79062 CD1XJ5 118706284 Ki = 29 nM T79062 CL4Y6K 118706285 Ki = 4.1 nM T79062 C32KAS 118706287 Ki = 160 nM T79062 C1K5NC 118706290 Ki = 87 nM T79062 CGA0O1 118706292 Ki = 41 nM T79062 CA0V9U 118706294 Ki = 50 nM T79062 C0NSU5 118706296 Ki = 180 nM T79062 CFOE72 118706299 Ki = 57 nM T79062 C1DI6Y 118706301 Ki = 4.1 nM T79062 CH3Z8R 118706732 Ki = 4 nM T79062 CN4I3G 118706734 Ki = 2.3 nM T79062 C2Q4OP 118709739 Ki = 28 nM T79062 CZ68PL 118709740 Ki = 24 nM T79062 CSB25E 118709750 Ki = 917 nM T79062 CD4S9R 118709751 Ki = 882 nM T79062 CBP52O 118709752 Ki = 36 nM T79062 CO72SF 118709753 Ki = 29 nM T79062 CJQR81 118709754 Ki = 41 nM T79062 CPW1D5 118709755 Ki = 62 nM T79062 C1TMO7 118709756 Ki = 2.7 nM T79062 CZ9H5G 118711997 Ki = 22 nM T79062 CH9W0A 118713587 Ki = 36.48 nM T79062 CK43CN 118713588 Ki = 7.77 nM T79062 CL0TS7 118713589 Ki = 0.99 nM T79062 C4RD6F 118713590 Ki = 41.93 nM T79062 CIG13W 118713591 Ki = 46.83 nM T79062 CX5L1H 118713592 Ki = 1.72 nM T79062 CDWY84 118713593 Ki = 2.84 nM T79062 CO5S1I 118713594 Ki = 57.39 nM T79062 CI91US 118713595 Ki = 20 nM T79062 CW92LT 118713679 Ki = 5.9 nM T79062 C8P9YT 118713680 Ki = 5.16 nM T79062 CZ1K5R 118713681 Ki = 14.1 nM T79062 CH7ZE8 118713682 Ki = 2.96 nM T79062 CKX78H 118713683 Ki = 11.68 nM T79062 C5LSA7 118713684 Ki = 2.9 nM T79062 CPAI54 118713685 Ki = 45.57 nM T79062 C6U2LR 118713686 Ki = 7.58 nM T79062 CYA6E4 118713687 Ki = 7.73 nM T79062 CZ9UL2 118713688 Ki = 8.49 nM T79062 CI5XK3 118717210 Ki = 1.2 nM T79062 CYJQ09 118717212 Ki > 100 nM T79062 C1TSR8 118717214 Ki = 1.4 nM T79062 C7YX3Q 118717215 Ki = 0.6 nM T79062 CEZ4M6 118717216 Ki = 0.76 nM T79062 C1E4GL 118717218 Ki = 4.9 nM T79062 CSJ6N3 118717219 Ki = 1.8 nM T79062 C5LFW4 118717221 Ki = 1.7 nM T79062 CZ65GI 118717222 Ki = 1.3 nM T79062 C1F9ZM 118724639 Ki = 346 nM T79062 CGA86P 118728506 Ki = 168 nM T79062 C9PGE7 118728507 Ki = 357 nM T79062 CR4GE1 118728510 Ki = 30.1 nM T79062 C14LZH 118728511 Ki = 147 nM T79062 C14RAC 118728513 Ki = 68.4 nM T79062 CQK04P 118728514 Ki = 1464 nM T79062 CK9CG4 118728521 Ki = 307 nM T79062 C1N9JU 118728522 Ki = 1082 nM T79062 C1UZ8G 118728523 Ki = 35.8 nM T79062 CPCE84 118728524 Ki = 12.9 nM T79062 CBN06J 118728525 Ki = 6.88 nM T79062 CF3QE0 118728526 Ki = 143 nM T79062 CJG4Q1 118728527 Ki = 1650 nM T79062 C4NFW1 118728528 Ki = 88.5 nM T79062 CO8LF9 118728529 Ki = 213 nM T79062 CCN7R8 118728530 Ki = 2.99 nM T79062 C5O2NU 118729733 Ki = 17890 nM T79062 CB3Y2W 118731347 Ki = 116 nM T79062 CWZF06 118731348 Ki = 18 nM T79062 CA3O1H 118731349 Ki = 30 nM T79062 CU8P4W 118731350 Ki = 43 nM T79062 C8GKX6 118731351 Ki = 6 nM T79062 C2J4VC 118731352 Ki = 10 nM T79062 CF7NH5 118731353 Ki = 11 nM T79062 CQ8F6C 118731354 Ki = 77 nM T79062 CR9J0O 118731355 Ki = 135 nM T79062 CU12XM 118731356 Ki = 5 nM T79062 C4CEV7 118731357 Ki = 16 nM T79062 CU6T2D 118731358 Ki = 15 nM T79062 C95WKJ 118731359 Ki = 30 nM T79062 C20QAO 118731360 Ki = 40 nM T79062 CT6J8V 118731361 Ki = 22 nM T79062 C7QVJ4 118731362 Ki = 10 nM T79062 CA2X3O 118731363 Ki = 9 nM T79062 C4DV8I 118731364 Ki = 9 nM T79062 CHVY82 118731365 Ki = 12 nM T79062 CM5FG1 118731366 Ki = 9 nM T79062 C75OXS 118736395 Ki = 473 nM T79062 C74FCM 118736396 Ki = 61 nM T79062 C3F8PA 118736397 Ki > 1000 nM T79062 CHI8V7 121209051 Ki = 322 nM T79062 C7W3EY 122178698 Ki = 69 nM T79062 CF8P1H 122178699 Ki = 15 nM T79062 C48MFR 122178700 Ki = 24 nM T79062 CZ72QS 122178701 Ki = 58 nM T79062 C4VY8A 122178702 Ki = 52 nM T79062 C2KF4Z 122178703 Ki = 28 nM T79062 CX6MJ2 122178704 Ki = 34 nM T79062 CA53KF 122178705 Ki = 24 nM T79062 C8XD3F 122178706 Ki = 38 nM T79062 CTRC59 122178707 Ki = 22 nM T79062 C5QV8D 122178708 Ki = 50 nM T79062 C84UED 122178709 Ki = 20 nM T79062 CV96JK 122178710 Ki = 23 nM T79062 CM89KS 122178711 Ki = 54 nM T79062 C7ODW3 122195524 Ki > 900 nM T79062 CBHT01 122377930 Ki = 9 nM T79062 CG63UZ 122483217 Ki = 281.84 nM T79062 C3RX0B 122483224 Ki = 2336 nM T79062 C57RDF 122483225 Ki = 1071.52 nM T79062 C7PL6Q 122483228 Ki = 588.84 nM T79062 CW32JF 122483234 Ki = 251.19 nM T79062 C7K4ZC 122483237 Ki = 1307 nM T79062 C4JFD9 122483243 Ki = 549.54 nM T79062 CZ27HR 122483245 Ki = 151.36 nM T79062 C89LZM 122483248 Ki = 794.33 nM T79062 CM8HO9 122483250 Ki = 616 nM T79062 CB9U5S 122483253 Ki = 1398 nM T79062 CL4J6V 122483257 Ki = 831.76 nM T79062 C86NGA 122483259 Ki = 309.03 nM T79062 C24ZNM 122483261 Ki = 512.86 nM T79062 C2SWA8 122483263 Ki = 1047.13 nM T79062 C1G4YN 122483273 Ki = 676.08 nM T79062 CLW53P 122483274 Ki = 86 nM T79062 C8IZ9U 122483279 Ki = 949 nM T79062 CO63ET 122483280 Ki = 30 nM T79062 CJ84WM 122483287 Ki = 125.89 nM T79062 C5IV3P 122483288 Ki = 1281 nM T79062 C0Y7NI 122483295 Ki = 1905.46 nM T79062 CKSQ23 122483303 Ki = 2137.96 nM T79062 C4QM2E 124247485 Ki = 104 nM T79062 CLWM12 126720394 Ki = 8748 nM T79062 C8Q1JB 126720403 Ki = 11920 nM T79062 C1U3SZ 126720425 Ki = 7139 nM T79062 C5G8FD 126720440 Ki = 12340 nM T79062 CD50YM 127024949 Ki = 20 nM T79062 C4GF2D 127024950 Ki = 40 nM T79062 CJ76IB 127024951 Ki = 4 nM T79062 CKB42V 127025036 Ki = 157 nM T79062 CIHZ54 127025242 Ki = 2 nM T79062 CCY7P3 127025243 Ki = 1 nM T79062 CNJ4Z1 127025244 Ki = 9 nM T79062 CTBN56 127026052 Ki = 398.11 nM T79062 C26NMB 127026071 Ki = 74 nM T79062 C1YD7M 127026119 Ki = 344 nM T79062 CUO7Y8 127026120 Ki = 27 nM T79062 CDU21O 127026131 Ki = 4 nM T79062 C9HDP8 127026132 Ki = 70 nM T79062 CTYP30 127026133 Ki = 14 nM T79062 C19BOM 127026141 Ki = 50 nM T79062 CZFB49 127026142 Ki = 285 nM T79062 C2FT3B 127026143 Ki = 197 nM T79062 CP4J5H 127026144 Ki = 264 nM T79062 C6BIU4 127026145 Ki = 201 nM T79062 C1FA2U 127026146 Ki = 198 nM T79062 CE43NR 127026147 Ki = 39 nM T79062 CDAP16 127026434 Ki = 1918 nM T79062 C2XO3L 127026443 Ki = 54 nM T79062 C80QHX 127026444 Ki = 17 nM T79062 CBF64M 127026450 Ki = 12 nM T79062 CO1FB4 127026451 Ki = 14 nM T79062 CC13RA 127026452 Ki = 20 nM T79062 CBE56W 127026514 Ki = 74 nM T79062 C0SZI4 127026515 Ki = 38 nM T79062 CX6EI2 127026750 Ki = 19 nM T79062 CEG15O 127026751 Ki = 16 nM T79062 C1J4QY 127026752 Ki = 14 nM T79062 C0WB2U 127026753 Ki = 7 nM T79062 C62UMZ 127027143 Ki = 602.56 nM T79062 C4L0KU 127027144 Ki = 363.08 nM T79062 C0UOJ6 127027386 Ki = 72 nM T79062 C9IH1A 127027387 Ki = 26 nM T79062 C0TC7E 127027388 Ki = 53 nM T79062 CZ4W6I 127027389 Ki = 168 nM T79062 C4YR7A 127027390 Ki = 162 nM T79062 C3FA0I 127027391 Ki = 319 nM T79062 CC71UE 127027715 Ki = 292 nM T79062 CY2TW9 127028152 Ki = 223 nM T79062 CAZJ04 127028153 Ki = 89 nM T79062 CR48GO 127028154 Ki = 234 nM T79062 C8MC1I 127028408 Ki = 1023.29 nM T79062 CD8H7W 127028471 Ki = 47 nM T79062 C4EAY5 127028472 Ki = 10 nM T79062 CUS8R9 127028473 Ki = 14 nM T79062 CA10BY 127028634 Ki = 163 nM T79062 CZ26YR 127028797 Ki = 17 nM T79062 CI2R1N 127028798 Ki = 56 nM T79062 CS8GJ5 127028799 Ki = 837 nM T79062 CU0WQ3 127029375 Ki = 908 nM T79062 CS1GX5 127029649 Ki = 1190 nM T79062 C9N3BE 127029650 Ki = 141 nM T79062 CQFS48 127029651 Ki = 177 nM T79062 C7F3YE 127029652 Ki = 79 nM T79062 CZ61LK 127034966 EC50 > 5011.87 nM T79062 CA0SN5 127034967 EC50 > 5011.87 nM T79062 CQ0ZT9 127035062 Ki = 700 nM T79062 CU49VE 127036186 Ki = 154.88 nM T79062 CG06BD 127036932 Ki = 74.13 nM T79062 CVW71O 127036953 Ki = 48.98 nM T79062 C7N5DF 127037679 Ki = 8 nM T79062 CD13VY 127037680 Ki = 24 nM T79062 CTE43C 127037681 Ki = 19 nM T79062 C0LGK6 127037682 Ki = 21 nM T79062 C2XBE8 127037921 Ki = 49 nM T79062 CX0CN4 127037922 Ki = 18 nM T79062 CDAE15 127038033 Ki = 7 nM T79062 CFA6Q8 127038034 Ki = 44 nM T79062 CERL85 127038035 Ki = 49 nM T79062 C8TC9G 127038281 Ki = 10 nM T79062 CPK2Z7 127038282 Ki = 84 nM T79062 CYJ2D5 127039593 Ki = 56 nM T79062 CQED51 127039753 Ki = 7 nM T79062 CL4E2K 127039754 Ki = 36 nM T79062 CES26L 127039755 Ki = 6 nM T79062 CQ36LP 127039756 Ki = 7 nM T79062 C7KA2C 127040443 Ki = 200 nM T79062 CKBZ01 127040444 Ki = 42 nM T79062 CFAB12 127040760 Ki = 8 nM T79062 CWQ47G 127040761 Ki = 28 nM T79062 C8D4AV 127040908 Ki = 13 nM T79062 CE12AY 127041106 Ki = 19 nM T79062 C71LGS 127041107 Ki = 9 nM T79062 C6RI9V 127041108 Ki = 8 nM T79062 C15BGV 127041244 Ki = 9 nM T79062 CU0J4S 127041258 Ki = 18 nM T79062 C20MZH 127041259 Ki = 10 nM T79062 CP16CZ 127041260 Ki = 70 nM T79062 CZT53S 127041261 Ki = 68 nM T79062 C0FJP2 127041563 Ki = 58 nM T79062 CUC3F9 127041564 Ki = 58 nM T79062 COG9D2 127041874 Ki = 100 nM T79062 CS4WH1 127042184 Ki = 5 nM T79062 C13AIN 127042185 Ki = 7 nM T79062 CR59TP 127042539 Ki = 56 nM T79062 C54IZC 127042540 Ki = 28 nM T79062 C8G1HF 127042841 Ki = 53 nM T79062 CC7BU0 127049059 Ki = 1511 nM T79062 C42FHY 127049060 Ki > 10000 nM T79062 CF2QY9 127049061 Ki = 286 nM T79062 CX53AC 127050632 Ki = 1584.89 nM T79062 CTL0S1 127051516 Ki = 626 nM T79062 CTL8J1 127051843 Ki = 755 nM T79062 CF6V9Q 127051844 Ki = 12 nM T79062 C8TNB1 127051845 Ki = 16.98 nM T79062 C5ONG1 127051864 Ki = 1000 nM T79062 CVQW26 127051865 Ki = 79.43 nM T79062 CRF85X 127052458 Ki = 10 nM T79062 CCY71I 127052465 Ki = 330 nM T79062 C2E9VX 127052467 Ki = 51.29 nM T79062 CPO4C3 127052468 Ki = 86 nM T79062 CSQ2N8 127052486 Ki = 313 nM T79062 C4YJ8H 127052487 Ki = 111 nM T79062 CT9RS4 127052488 Ki = 778 nM T79062 CLU7C1 127052757 Ki = 26.92 nM T79062 C95KYT 127052758 Ki = 100 nM T79062 CYNR02 127052759 Ki = 48.98 nM T79062 C14YJU 127052778 Ki = 501.19 nM T79062 C1JAS7 127052779 Ki = 189 nM T79062 C7MQK8 127053042 Ki = 22.5 nM T79062 C50GOC 130442480 Ki = 8100 nM T79062 CM04RF 130442572 Ki = 4100 nM T79062 C4LJ2Y 132503215 Ki = 55 nM T79062 CM8B1L 132525569 Ki = 7.1 nM T79062 CU5L0K 132525570 Ki = 1.6 nM T79062 CA10SQ 132547275 Ki = 44.8 nM T79062 C6E1GN 132547276 Ki = 23.5 nM T79062 C6VTW3 132547277 Ki = 35.1 nM T79062 CI70OP 132547278 Ki = 45.1 nM T79062 C3Q1LA 132547279 Ki = 8.42 nM T79062 CAVB41 132584404 Ki > 10000 nM T79062 CS0MB3 132938109 Ki = 33 nM T79062 C8O2EP 134130246 Ki = 37 nM T79062 C8M9FH 134130379 Ki = 613 nM T79062 CA4GX3 134130447 Ki = 143 nM T79062 C7ZDA2 134130462 Ki = 53.7 nM T79062 CWL50Q 134130594 Ki = 1310 nM T79062 C8TG2O 134130846 Ki = 327 nM T79062 CHP3J4 134131015 Ki = 1377 nM T79062 CQ4IF8 134131147 Ki = 94.7 nM T79062 C6N5FS 134131151 Ki = 1328 nM T79062 CH4XB2 134131159 Ki = 990 nM T79062 CR32SP 134131265 Ki = 181 nM T79062 C0JKL5 134131283 Ki = 276 nM T79062 C0RQC6 134131976 Ki = 27 nM T79062 CQX4U3 134133064 Ki = 6.31 nM T79062 CTS3J4 134133483 Ki = 18.5 nM T79062 C0J2ML 134133604 Ki = 0.4677 nM T79062 CP0E5M 134133632 Ki = 497 nM T79062 CM0TS6 134133967 Ki = 44.67 nM T79062 CNV91Q 134134210 Ki = 23 nM T79062 C0ZLJ3 134134279 Ki = 648 nM T79062 CC1DO8 134134456 Ki = 25.5 nM T79062 CMS79H 134135372 Ki = 1038 nM T79062 C2Q3JY 134135516 Ki = 76 nM T79062 CJG3U0 134136134 Ki = 9.5 nM T79062 CGX03A 134136246 Ki = 131.83 nM T79062 C4VR6O 134137104 Ki = 18 nM T79062 C08ZBY 134137332 Ki = 32 nM T79062 CXF52V 134137560 Ki = 15.5 nM T79062 CN4LI8 134137732 Ki = 11.5 nM T79062 CWO5R6 134138168 Ki = 18 nM T79062 CRC2V0 134139826 Ki = 54 nM T79062 CG30KH 134140472 Ki = 126 nM T79062 CHK39T 134141166 Ki = 8 nM T79062 CLW86T 134141354 Ki = 257 nM T79062 C2NOX7 134141985 Ki = 34 nM T79062 CK54QW 134142259 Ki = 259 nM T79062 C6PSI9 134142907 Ki = 87 nM T79062 CR5L4K 134144303 Ki = 138 nM T79062 CYF16Z 134144798 Ki = 3063 nM T79062 C80TGJ 134144864 Ki = 25 nM T79062 CGW1D0 134145143 Ki = 1476 nM T79062 CK5RU9 134145903 Ki = 10 nM T79062 C2E0ID 134146185 Ki = 44 nM T79062 CC9P2T 134146194 Ki = 43.65 nM T79062 CV0QZ5 134147124 Ki = 52 nM T79062 C41XSD 134147935 Ki = 108 nM T79062 CFD13P 134147951 Ki = 1019 nM T79062 C8NBO0 134148917 Ki = 772 nM T79062 CBU81N 134149168 Ki > 10000 nM T79062 C0J8HT 134150597 Ki = 691 nM T79062 CE6LN3 134151118 Ki = 21 nM T79062 CLU34D 134151427 Ki = 265 nM T79062 C2JN8Y 134151729 Ki = 36.5 nM T79062 C76BZW 134151980 Ki = 16 nM T79062 CIV4H5 134152583 Ki = 254 nM T79062 CB6M5Y 134153538 Ki = 144 nM T79062 CX4W7F 134153716 Ki = 12 nM T79062 C79TEI 134154068 Ki = 25 nM T79062 C5B4GR 134154108 Ki = 1123 nM T79062 CMJ1U3 134154387 Ki = 65 nM T79062 C4M0FW 134154531 Ki = 79 nM T79062 C4VGJ5 134154679 Ki = 67 nM T79062 C6QAY2 134155116 Ki = 1.585 nM T79062 C79QLN 134155460 Ki = 91 nM T79062 CIUZ94 134155476 Ki = 10.5 nM T79062 C90QNV 134155645 Ki = 14 nM T79062 C97EWM 134155651 Ki = 389 nM T79062 CVR87Q 134156222 Ki = 125.89 nM T79062 CAB4K6 134156305 Ki = 19 nM T79062 C50XNE 134156520 Ki = 4.5 nM T79062 CUHE07 134157171 Ki = 6.5 nM T79062 CV8JU6 134157289 Ki = 73 nM T79062 CL6DN0 134157769 Ki = 14.5 nM T79062 C5IM7X 135367399 Ki = 363.08 nM T79062 C41JQV 135367400 Ki = 501.19 nM T79062 C2RN9U 135367403 Ki = 1407 nM T79062 C74JIA 135367404 Ki = 881 nM T79062 C6N8GM 135367405 Ki = 46.77 nM T79062 C6LU0C 135367816 Ki = 70 nM T79062 CTX68N 135367817 Ki = 883 nM T79062 CD2TH9 135367820 Ki = 52.48 nM T79062 CM7SA8 135367821 Ki = 369 nM T79062 CP21LA 135367855 Ki = 425 nM T79062 C5AMD9 135367857 Ki = 16 nM T79062 C6SKM3 135367858 Ki = 707.95 nM T79062 C5URG0 135367869 Ki = 1230.27 nM T79062 CBA7P6 135367917 Ki = 1436 nM T79062 C9DVI7 135367936 Ki = 386 nM T79062 CR0U6A 135367959 Ki = 316.23 nM T79062 CVE08Y 135458392 Ki = 15.3 nM T79062 CP7HN4 135458393 Ki = 33.3 nM T79062 CS8XJ6 135458394 Ki = 13.2 nM T79062 C9B7XA 135458410 Ki = 23.3 nM T79062 CFV9A3 135458427 Ki = 4.2 nM T79062 CKX4N8 135458428 Ki = 38.9 nM T79062 C9ZCL5 135458672 Ki = 4194 nM T79062 CTE23K 135464118 Ki = 512 nM T79062 CD6L8Q 135895192 Ki = 13.6 nM T79062 CA1M8B 135966709 Ki = 2.4 nM T79062 CUKO20 136020617 Ki > 10000 nM T79062 COF0U5 136020618 Ki > 10 nM T79062 CF89JI 136030596 Ki > 10000 nM T79062 CE8GB9 136030693 Ki > 10000 nM T79062 C65VFI 136030744 Ki > 10000 nM T79062 COIX80 136054961 Ki > 10000 nM T79062 C19GLK 136116062 Ki = 366.3 nM T79062 CQ2GP6 136118614 Ki = 1223 nM T79062 C8RH6M 136118617 Ki = 4114 nM T79062 CG5TX8 136118653 Ki = 3350 nM T79062 C40LYH 136118659 Ki = 5367 nM T79062 CY5GU4 136118730 Ki = 799 nM T79062 CB12QP 136152964 Ki = 24.8 nM T79062 CFX06E 136152966 Ki = 17.6 nM T79062 C37YXA 136152971 Ki = 7.7 nM T79062 CY0C1X 136152972 Ki = 1704 nM T79062 CX53NC 136180316 Ki = 145 nM T79062 CZ7WT9 136180317 Ki = 21.2 nM T79062 CQP2Y6 136180318 Ki = 1135 nM T79062 CQT9H5 136180319 Ki = 228 nM T79062 CLPU18 136180320 Ki = 11.9 nM T79062 C0LO6Q 136180321 Ki = 101 nM T79062 CAE39V 136188797 Ki > 10000 nM T79062 CWP0V5 136216703 Ki = 1600 nM T79062 CLAP52 136259032 Ki > 10000 nM T79062 CHM36P 137631892 Ki = 52 nM T79062 CU01TV 137633827 Ki > 10000 nM T79062 CC51JN 137635185 Ki > 10000 nM T79062 C94VXJ 137635884 Ki = 95 nM T79062 CFM92C 137636384 Ki = 3692 nM T79062 CDX39B 137637994 Ki = 142 nM T79062 C3LYX9 137641832 Ki > 10000 nM T79062 C5WS6Q 137642134 Ki = 14 nM T79062 CWUM83 137644521 Ki > 10000 nM T79062 CDA80E 137644790 Ki = 36 nM T79062 CZ8CU6 137645501 Ki = 56 nM T79062 CCP38D 137645926 Ki = 37 nM T79062 CVX74E 137646045 Ki = 438 nM T79062 CPI68E 137646281 Ki = 128 nM T79062 CMXI62 137649997 Ki = 209 nM T79062 C52IRM 137650705 Ki = 37 nM T79062 CKG08R 137650961 Ki = 165 nM T79062 CU4S1W 137651887 Ki = 5 nM T79062 CVK26R 137652044 Ki = 174 nM T79062 CHFK13 137652210 Ki > 10000 nM T79062 C51CGJ 137652310 Ki = 29 nM T79062 C2E3FV 137653850 Ki = 18 nM T79062 CX82HS 137654666 Ki = 32 nM T79062 C0SKV1 137654850 Ki > 10000 nM T79062 C4VG0U 137655411 Ki = 39 nM T79062 CO3L7F 137656918 Ki > 10000 nM T79062 CX4D7Y 137660741 Ki = 52 nM T79062 C0R6XM 138691314 Ki = 6 nM T79062 CU3Y7W 138691316 Ki = 20 nM T79062 CH2W4P 138691317 Ki = 531 nM T79062 CHSC40 138691321 Ki = 36 nM T79062 C18UZA 138691329 Ki = 42 nM T79062 C1XWV0 138691338 Ki = 30 nM T79062 C6LE1A 138691362 Ki = 44 nM T79062 CN9R4A 138691364 Ki = 5 nM T79062 C8H2KR 138691366 Ki = 302 nM T79062 C2Z9CD 139488518 Ki = 386 nM T79062 CJK95T 139488527 Ki = 22 nM T79062 CZ6H9M 139488539 Ki = 16 nM T79062 CAF2H8 139488606 Ki = 4 nM T79062 C54CIL 139488740 Ki = 18 nM T79062 CN3G0A 140936451 Ki > 10000 nM T79062 C4EU2S 141745651 Ki = 0.99 nM T79062 CCO6R0 141745657 Ki = 2.2 nM T79062 CO5DR9 145949220 Ki = 23 nM T79062 CWAF96 145949371 Ki = 10 nM T79062 CHG2W6 145950605 Ki = 9 nM T79062 COU57L 145950881 Ki = 7 nM T79062 CD4M6B 145951915 Ki = 85 nM T79062 C78AUI 145952711 Ki = 8 nM T79062 CA2J5S 145954503 Ki = 71200 nM T79062 C0JO8B 145954831 Ki = 10 nM T79062 CHI1V8 145956064 Ki = 566 nM T79062 CSER68 145956892 Ki = 20 nM T79062 CLVI07 145957637 Ki = 213 nM T79062 C91IDE 145958490 Ki = 1205 nM T79062 C8VS7K 145959257 Ki = 94 nM T79062 CSIZ31 145959706 Ki = 12 nM T79062 C67GQI 145961372 Ki = 2797 nM T79062 C4Y1PK 145963314 Ki = 6 nM T79062 C7KC3T 145963830 Ki > 10000 nM T79062 C5VWM7 145963860 Ki = 74 nM T79062 CCK5G1 145963863 Ki = 902 nM T79062 C4Y2AL 145964000 Ki = 3142 nM T79062 CV7YW9 145964086 Ki = 170 nM T79062 CHDN35 145964150 Ki > 10000 nM T79062 CR2B9G 145964154 Ki = 290 nM T79062 C1KH2E 145964159 Ki = 3600 nM T79062 C7YKQ4 145964390 Ki = 93 nM T79062 C95NZO 145964427 Ki = 89 nM T79062 C2P5NK 145964621 Ki = 67 nM T79062 CK0T1M 145964694 Ki = 213 nM T79062 C6T4RY 145964846 Ki = 90 nM T79062 CE9K3L 145964944 Ki = 12 nM T79062 C12OVL 145965034 Ki > 10000 nM T79062 CBS74V 145965054 Ki = 4 nM T79062 C9D8IB 145965203 Ki = 15 nM T79062 C1MIR9 145965401 Ki = 258 nM T79062 CLP94W 145965668 Ki = 245 nM T79062 C8TF9G 145965840 Ki = 121 nM T79062 C5W4LM 145965940 Ki > 10000 nM T79062 C53EFW 145966154 Ki = 547 nM T79062 CB05QA 145966199 Ki = 59 nM T79062 C1T4DN 145966418 Ki = 55 nM T79062 CV03XA 145967457 Ki = 1580 nM T79062 C81VUO 145967771 Ki > 10 nM T79062 CJS56K 145967795 Ki > 10000 nM T79062 CQ8EM6 145969402 Ki = 29 nM T79062 CA82FL 145970078 Ki = 2 nM T79062 CF74MR 145971390 Ki = 1671 nM T79062 C1T7GL 145971527 Ki = 12500 nM T79062 C8A2XG 145971561 Ki = 38 nM T79062 CN64ZR 145971588 Ki = 1154 nM T79062 CQJ5O8 145971635 Ki > 10000 nM T79062 C56RAO 145972025 Ki = 284 nM T79062 C79TNE 145972796 Ki > 10000 nM T79062 CJHI43 145972875 Ki = 52 nM T79062 CS7WG8 145973438 Ki = 1154 nM T79062 C8KYV6 145973487 Ki = 313 nM T79062 CEOY46 145973577 Ki = 388 nM T79062 CL74IP 145973853 Ki = 6 nM T79062 CR0CX6 145974087 Ki = 50 nM T79062 C6XIN0 145974114 Ki > 10000 nM T79062 C8KZ5T 145974165 Ki = 0.75 nM T79062 C05IVJ 145974184 Ki = 172 nM T79062 CW6EX3 145974189 Ki = 32 nM T79062 CD8ZL6 145974750 Ki > 10 nM T79062 C3WG0J 145975106 Ki = 52 nM T79062 C6PH4F 145975226 Ki > 10000 nM T79062 CN8U3P 145975289 Ki = 86 nM T79062 CSVR94 145975713 Ki = 408 nM T79062 COY2P3 145975720 Ki = 21 nM T79062 CL7EX5 145975776 Ki = 1050 nM T79062 C1BI8E 145975778 Ki = 534 nM T79062 C7R2MD 145975905 Ki = 100 nM T79062 C71CYU 145975946 Ki > 10000 nM T79062 C0V4AL 145975992 Ki = 275 nM T79062 C2TN8W 145976085 IC50 > 10000 nM T79062 C8XFM7 145976120 Ki = 3027 nM T79062 CF5B0W 145976158 Ki = 41 nM T79062 C8BJI2 145976292 Ki = 58 nM T79062 CZ5XK2 145976408 Ki = 67 nM T79062 C14OJW 145976618 Ki = 34 nM T79062 C0LRB2 145976686 Ki = 110 nM T79062 C34XME 145976696 Ki = 70 nM T79062 CTCM92 145976698 Ki = 415 nM T79062 CIZ69S 145976722 Ki = 228 nM T79062 CT7WO5 145976787 Ki = 213 nM T79062 CI8AN3 145976890 Ki = 32 nM T79062 C81CSM 145976946 Ki = 931 nM T79062 CXDR94 145977222 Ki = 3160 nM T79062 C8NW7Y 145977256 Ki = 43 nM T79062 CHS96B 145977297 Ki = 3.2 nM T79062 C6BFY7 145977338 Ki = 7400 nM T79062 C4L8EZ 145977467 Ki = 64 nM T79062 CC1DZ5 145977555 Ki = 204 nM T79062 C0Y6QO 145977799 Ki = 3300 nM T79062 C3BI1R 145978113 Ki > 10000 nM T79062 CP8C6M 145978146 Ki = 104 nM T79062 C6HQI0 145978420 Ki = 203 nM T79062 C8VL3Y 145978472 Ki = 529 nM T79062 C82NXP 145978482 Ki = 602 nM T79062 CQU8R0 145978665 Ki > 10000 nM T79062 C6AV9G 145978819 Ki > 10000 nM T79062 C20XQJ 145979626 Ki = 3609 nM T79062 C87MSW 145980271 Ki = 812 nM T79062 CW2CO4 145980458 Ki = 11 nM T79062 C8I7QL 145980875 Ki = 1120 nM T79062 CPK34X 145981875 Ki = 1.1 nM T79062 COY79P 145982165 Ki = 5 nM T79062 CEK60A 145982506 Ki = 165 nM T79062 CI59TX 145983018 Ki = 1119 nM T79062 CYC58R 145983059 Ki = 45 nM T79062 C4F5OT 145983128 Ki = 14 nM T79062 C5ZG9M 145983139 Ki = 7 nM T79062 CV2GU9 145983144 Ki = 65 nM T79062 C4PKM2 145983390 Ki = 19 nM T79062 C9LR8C 145983405 Ki = 0.55 nM T79062 CIAF74 145983468 Ki = 57 nM T79062 CE7MF4 145983751 Ki = 69 nM T79062 CDQ4U7 145983760 Ki = 19 nM T79062 CYW9B2 145983794 Ki = 32 nM T79062 C8I1WG 145983961 Ki = 3 nM T79062 CP5H4D 145984065 Ki = 8 nM T79062 CJ35DM 145984299 Ki = 9 nM T79062 CU7E4M 145984511 Ki = 51 nM T79062 C6JUY0 145984737 Ki = 12 nM T79062 CID02G 145984807 Ki = 672 nM T79062 CM5X3V 145985050 Ki = 0.4 nM T79062 CG10LK 145985224 Ki = 17 nM T79062 CFJ9B3 145985233 Ki = 12 nM T79062 C5AOI6 145985289 Ki = 24 nM T79062 CW30NA 145985505 Ki = 10 nM T79062 C7ZRP1 145985527 Ki = 12 nM T79062 C2XY8Q 145985533 Ki = 7 nM T79062 C7NI4X 145985585 Ki = 6 nM T79062 C9LJ5T 145985692 Ki = 1 nM T79062 C7QIX0 145985718 Ki = 52 nM T79062 C6V5QS 145985823 Ki = 12 nM T79062 C07GKD 145985958 Ki = 1340 nM T79062 CCM18E 145986031 Ki = 22 nM T79062 CR0XQ3 145986138 Ki = 31 nM T79062 CT37DW 145986720 Ki = 824 nM T79062 CNJH37 145986752 Ki = 949 nM T79062 C3VN5O 145987559 Ki = 165 nM T79062 CI0PA9 145987771 Ki = 3.3 nM T79062 CIS9P2 145988193 Ki = 12 nM T79062 CUGO10 145988693 Ki = 1574 nM T79062 C9D2OG 145988738 Ki = 3 nM T79062 C4C0YP 145988913 Ki = 172 nM T79062 CDY48U 145989143 Ki = 0.26 nM T79062 C3GPR9 145990093 Ki = 2085 nM T79062 C2Q5UK 145990353 Ki = 3 nM T79062 CT7AB8 145990459 Ki = 2172 nM T79062 C4GV8Q 145990586 Ki = 120 nM T79062 CVBR36 145991084 Ki = 0.79 nM T79062 C9TK6G 145991864 Ki = 2.6 nM T79062 CB8CM6 145992305 Ki = 209 nM T79062 CCP2U1 145992489 Ki = 10000 nM T79062 CLPU06 145992567 Ki = 224 nM T79062 CBI94R 145992877 Ki = 1.1 nM T79062 CI19KS 145993474 Ki = 2.3 nM T79062 C0TL8E 145993714 Ki = 19 nM T79062 CC2G1V 146025727 Ki = 3800 nM T79062 C5ZOJ3 146680920 Ki = 7832 nM T79062 CG97ER 146709966 Ki = 1000 nM T79062 CF5B2L 147653864 Ki = 398.11 nM T79062 C9T0PS 153061504 Ki = 691.83 nM T79062 CAF36V 153287539 Ki = 1000 nM T79062 C1FA0K 153287541 Ki = 19.95 nM T79062 CEQ69Z 153287542 Ki = 23.44 nM T79062 C6P3SR 153287553 Ki = 6.3 nM T79062 C3G5CJ 153287557 Ki = 199.53 nM T79062 CW31CT 153287566 Ki = 2.692 nM T79062 CYP86E 153287567 Ki = 199.53 nM T79062 CS73ZC 153287568 Ki = 1258.93 nM T79062 CV9G7Z 153287572 Ki > 10000 nM T79062 CO85KL 153287574 Ki = 1000 nM T79062 CZ1K4D 155510674 Ki = 21 nM T79062 CLX3D8 155510732 IC50 = 650 nM T79062 CC3KP7 155510927 Ki = 1148 nM T79062 CM4RB0 155511262 Ki = 3147 nM T79062 C9KX6O 155511928 Ki = 280 nM T79062 CZ7HP4 155512406 Ki = 40.1 nM T79062 C4OL0A 155512409 Ki = 3.43 nM T79062 CXF90M 155512487 Ki = 895 nM T79062 CO68LC 155512944 Ki = 49 nM T79062 C90FST 155513438 Ki = 51 nM T79062 C95QOT 155514378 Ki = 2352 nM T79062 C3SQI7 155514459 Ki > 10000 nM T79062 CI4DT8 155514575 Ki = 2455 nM T79062 CJUI87 155514774 Ki = 45 nM T79062 CQ84DA 155514889 Ki = 298 nM T79062 C3NB0D 155515324 Ki = 98430 nM T79062 C0Q8PR 155515407 Ki = 1833 nM T79062 CWO56B 155515415 Ki > 10000 nM T79062 CU0PY6 155515687 Ki = 9.42 nM T79062 C2TN5D 155515890 Ki = 184 nM T79062 C7KT0D 155515919 Ki = 1096 nM T79062 C13LOV 155515942 Ki = 6660 nM T79062 C7OF4C 155516118 Ki = 13750 nM T79062 CJ1Z0D 155516162 Ki > 10000 nM T79062 CG5M1O 155516282 Ki = 3743 nM T79062 CG53LH 155516399 Ki = 0.85 nM T79062 CU8TC0 155517162 Ki = 25 nM T79062 CW0B5K 155518159 Ki > 10000 nM T79062 CYB12O 155518974 Ki = 116500 nM T79062 CHVF41 155519045 Ki = 401 nM T79062 CCEZ93 155519102 Ki = 38730 nM T79062 CQD2J7 155519393 Ki = 9855 nM T79062 C2SXT1 155519515 Ki = 167 nM T79062 C0KLD8 155519559 Ki = 6248 nM T79062 C07BTO 155519598 Ki = 291 nM T79062 CUSA24 155519891 Ki = 1258.93 nM T79062 C5FL7R 155520499 Ki = 822 nM T79062 C8OC3W 155520552 Ki = 140 nM T79062 CTV2F6 155521010 Ki = 380 nM T79062 CQ76MP 155521503 Ki = 3715 nM T79062 C1OS6D 155522116 Ki > 10000 nM T79062 C98RDQ 155522218 Ki = 1115 nM T79062 C2TV4Y 155522487 Ki > 10000 nM T79062 CP6H1D 155522562 Ki = 432 nM T79062 CUQ61M 155522867 Ki = 7.54 nM T79062 CUG8L3 155522920 Ki > 10000 nM T79062 CD9QU6 155523519 Ki = 20 nM T79062 C5KYB4 155524228 Ki = 458 nM T79062 C6APG2 155524374 Ki = 36.6 nM T79062 CK4B0R 155524491 Ki = 1361 nM T79062 CUO93F 155524808 Ki = 305 nM T79062 CQB0M8 155524884 Ki > 10000 nM T79062 C65UZD 155524956 Ki = 286 nM T79062 C6MZJ9 155525703 Ki = 74 nM T79062 C81OCJ 155526014 Ki = 80.3 nM T79062 CZ81JA 155526026 Ki = 120 nM T79062 C1U2XO 155526651 Ki = 119 nM T79062 CXH79K 155526720 Ki = 11 nM T79062 CW68KC 155528355 Ki > 10000 nM T79062 C7C1EF 155528967 Ki = 1444 nM T79062 C5J7AU 155529153 Ki = 4247 nM T79062 C9KS5C 155529450 Ki = 58 nM T79062 CKZ25Y 155529679 Ki = 195 nM T79062 C3X4IA 155530328 Ki = 233 nM T79062 C9PC3D 155530350 Ki = 5996 nM T79062 CVLC03 155530779 Ki = 871 nM T79062 C98YQF 155531012 Ki = 258 nM T79062 C4W6VC 155531065 Ki = 1622 nM T79062 C5HWP4 155531362 Ki > 10000 nM T79062 CKDE38 155531753 Ki = 1 nM T79062 CCT8V9 155531846 Ki = 9531 nM T79062 C05KFL 155532137 Ki = 56.2 nM T79062 CMPU81 155532470 Ki > 10000 nM T79062 CX35QS 155532545 Ki > 10000 nM T79062 CX6DV4 155533028 Ki = 696 nM T79062 C23GDV 155533534 Ki = 1712 nM T79062 C3OEH2 155533648 Ki = 710 nM T79062 C15RYP 155533660 Ki > 10000 nM T79062 CY01GZ 155533850 Ki = 1384 nM T79062 CP3J8B 155534152 Ki = 3467 nM T79062 C3L0CP 155534184 Ki = 2431 nM T79062 CG85SB 155534301 Ki = 475 nM T79062 CG8Y7W 155534312 Ki = 366 nM T79062 C3VGT0 155534362 Ki = 1922 nM T79062 CW7SV9 155534575 Ki = 35 nM T79062 C75FSY 155534794 Ki = 2512 nM T79062 CTO4S9 155534839 Ki = 2 nM T79062 C6KF4E 155535154 Ki = 546 nM T79062 C8G7AW 155535428 Ki > 10000 nM T79062 C8O4IQ 155535827 Ki = 35 nM T79062 C14JEX 155535878 Ki = 776 nM T79062 CB79ZW 155536080 Ki > 10000 nM T79062 C5I1JA 155536087 Ki = 322 nM T79062 C72FLG 155536152 Ki = 3804 nM T79062 CW2SC8 155536533 Ki = 106 nM T79062 CTB93R 155536809 Ki = 462 nM T79062 C7FVE8 155537034 Ki = 6 nM T79062 C36FRH 155537074 Ki = 2095 nM T79062 CD75GP 155537227 Ki > 10000 nM T79062 CVS04L 155537788 Ki = 23 nM T79062 CB8IC7 155538144 Ki = 273 nM T79062 C5F2GI 155538236 Ki = 1092 nM T79062 COYG20 155538350 Ki = 933 nM T79062 C9TIU2 155538367 Ki = 53 nM T79062 CYC1P3 155538451 Ki = 73 nM T79062 CM08NT 155538716 Ki > 10000 nM T79062 CQ69UA 155538814 Ki = 5818 nM T79062 C0Q5NT 155538877 Ki = 133 nM T79062 CAT98F 155539483 Ki = 1158 nM T79062 C6S8BA 155539600 Ki = 4570 nM T79062 C9S2IA 155539605 Ki = 2765 nM T79062 C42GUK 155540147 Ki > 10000 nM T79062 C1X0IO 155540198 Ki = 197 nM T79062 C9J3BQ 155540635 Ki = 65.1 nM T79062 C1KA8C 155540755 Ki = 43.8 nM T79062 CR2K1T 155540795 Ki > 10000 nM T79062 CNU92V 155540807 Ki = 25 nM T79062 CUY87S 155540823 Ki = 119 nM T79062 COS2E7 155541072 Ki = 6417 nM T79062 CP7UG2 155541866 Ki = 3298 nM T79062 COZ46W 155541871 Ki = 53 nM T79062 CB62ZS 155542237 Ki = 2455 nM T79062 CXCW81 155542321 Ki = 11950 nM T79062 C9FS3Y 155542461 Ki > 10000 nM T79062 C9RV7W 155542678 Ki = 1.99 nM T79062 CT6HY4 155543250 Ki = 29 nM T79062 C68MSK 155543653 Ki = 8361 nM T79062 CZ7O0A 155544139 Ki = 5840 nM T79062 CD84VK 155544810 Ki = 336 nM T79062 C2XZD8 155545087 Ki = 404 nM T79062 CCX6T2 155545402 Ki = 3.3 nM T79062 CO9X1Z 155545526 Ki > 10000 nM T79062 CI0YL8 155545625 Ki = 70 nM T79062 C74GFO 155546189 Ki = 203 nM T79062 CH3W9N 155546350 Ki = 1445 nM T79062 C4UT5Z 155546595 Ki = 125 nM T79062 C98AIL 155546781 Ki = 3.54 nM T79062 CD02EN 155547436 Ki = 371 nM T79062 COJ27N 155547693 Ki = 10660 nM T79062 CAT9X4 155548275 Ki = 8511 nM T79062 C5LYE8 155548677 Ki = 5316 nM T79062 C0KZB5 155549018 Ki = 50.2 nM T79062 C87JGN 155549153 Ki > 10000 nM T79062 CGP8O5 155549315 Ki = 291 nM T79062 C52FRY 155549978 Ki = 192 nM T79062 C8HPN7 155551113 Ki = 420 nM T79062 C61IVC 155551353 Ki = 8 nM T79062 CHS71N 155551685 Ki = 119 nM T79062 CM26AV 155551704 Ki > 1000 nM T79062 C6E9LK 155552054 Ki = 366 nM T79062 CQ48CS 155552188 Ki = 0.9 nM T79062 CA1WS9 155552212 Ki = 5095 nM T79062 C38YJB 155552311 Ki = 2761 nM T79062 C87PTM 155552707 Ki = 11 nM T79062 CDQ7C2 155552798 Ki = 48960 nM T79062 CPV35U 155552826 Ki = 161 nM T79062 CDV6B9 155554036 Ki = 9247 nM T79062 CKF75H 155554324 Ki = 124 nM T79062 C6ZSU3 155554462 Ki = 2871 nM T79062 C8JKT1 155555378 Ki = 19.3 nM T79062 C2E5TR 155555506 Ki = 525 nM T79062 CUNK28 155555525 Ki > 10000 nM T79062 CO52HW 155556527 Ki = 5888 nM T79062 C1N5VF 155556756 Ki > 10000 nM T79062 CJCL47 155556806 Ki = 75.8 nM T79062 CJBX01 155557042 Ki = 199.53 nM T79062 C5QYS0 155557134 Ki = 34 nM T79062 CD2L3K 155557443 Ki = 21 nM T79062 CER48T 155557500 Ki > 10000 nM T79062 C2L0PC 155557720 Ki = 16 nM T79062 CF6H3V 155558408 Ki = 15180 nM T79062 C4I2OY 155558563 Ki = 27.8 nM T79062 C9TB5D 155559092 Ki = 2366 nM T79062 CP4JO7 155559794 Ki > 10000 nM T79062 COG70U 155560942 Ki = 7079 nM T79062 C2HF6P 155561581 Ki = 2329 nM T79062 COL7N8 155561901 Ki = 46 nM T79062 CL45NV 155561914 Ki = 17780 nM T79062 CJ57BI 155561978 Ki = 22 nM T79062 C0SDZ8 155561990 IC50 = 12 nM T79062 CW7M1D 155561995 Ki = 1112 nM T79062 C93KWN 155562202 Ki = 266 nM T79062 CO3C6L 155562423 Ki > 10000 nM T79062 C5AI0S 155562519 Ki = 641 nM T79062 C5BQ8U 155562652 Ki = 958 nM T79062 CF6B4W 155562834 Ki = 344 nM T79062 CZ6IA2 155562918 Ki = 514 nM T79062 CRCW25 155562997 Ki = 50 nM T79062 CBH14K 155563164 Ki > 10000 nM T79062 CG1L8E 155563286 Ki > 10000 nM T79062 C38WXS 155563374 Ki = 7322 nM T79062 C0INS4 155563826 Ki > 10000 nM T79062 CK0IW3 155563911 Ki = 6 nM T79062 C5TS7Q 155564824 Ki = 710 nM T79062 CQK8E3 155565209 Ki = 54.7 nM T79062 CE2YG1 155565215 Ki = 12.2 nM T79062 C2MIU5 155565813 Ki = 2730 nM T79062 C7P5VG 155566191 Ki = 206 nM T79062 C7O6YP 155566439 Ki = 16050 nM T79062 CG35LB 155566508 Ki = 24.2 nM T79062 CU46EB 155566665 Ki > 10000 nM T79062 C67LAG 155566854 Ki = 9120 nM T79062 CW1TN7 155566925 Ki = 14 nM T79062 C41UWT 155567307 Ki = 84 nM T79062 CA8OE0 155567476 Ki = 9.08 nM T79062 CC06FO 155567938 Ki = 1.86 nM T79062 CA68TK 155568224 Ki = 614 nM T79062 C4EX7C 155568246 Ki = 320 nM T79062 C4POS3 155568373 Ki = 32.7 nM T79062 C67MIN 155568606 Ki = 0.8 nM T79062 CXP3E4 155568794 Ki = 1501 nM T79062 CB5IP9 155569021 Ki = 166 nM T79062 C0CZK6 155569337 Ki > 10000 nM T79062 CP9V7M 155569396 Ki = 138 nM T79062 C3ZNX6 155569414 Ki = 552 nM T79062 CZ8RV4 155569568 Ki = 2170 nM T79062 C3N9VU 10251906 Ki > 500 nM T79062 CP9TR0 10324985 Ki = 9.1 nM T79062 D00CRA 1574 Ki = 1258 nM T79062 D00GSD 25107716 Ki = 0.58 nM T79062 D00MXS 5281703 IC50 > 350000 nM T79062 D00OBS 44559159 Ki > 10000 nM T79062 D00VRV 10171 Ki = 10 nM T79062 D00YEV 5281605 IC50 > 350000 nM T79062 D01KAX 135453290 EC50 = 5600 nM T79062 D01KVG 9843179 Ki = 1.995 nM T79062 D01WWC 16573 Ki = 20 nM T79062 D02HZG 888311 Ki = 2663 nM T79062 D02RAY 16754 Ki = 43 nM T79062 D02UWB 1809 Ki = 0.3981 nM T79062 D02YSX 197033 Ki = 7.943 nM T79062 D03DET 10287730 Ki = 501.19 nM T79062 D03NBX 637308 IC50 = 47600 nM T79062 D03TDN 1342 Ki = 83 nM T79062 D03TSY 24825775 Ki = 2.5 nM T79062 D03ZHB 44455973 Ki = 97.4 nM T79062 D04AQE 1833 Ki = 2 nM T79062 D04TPO 16006492 Ki = 15.85 nM T79062 D05EQG 5265 Ki = 19.95 nM T79062 D05GDP 599482 Ki = 1400 nM T79062 D05LKO 44414722 Ki = 840 nM T79062 D05XGR 6918647 Ki = 2511.89 nM T79062 D05ZUX 44207909 Ki >= 1000 nM T79062 D06VDN 443391 IC50 > 1000 nM T79062 D07JRV 46233381 Ki = 553 nM T79062 D07JTZ 9843889 Ki = 89 nM T79062 D07LRJ 5312149 Ki = 260 nM T79062 D08BCF 5011 Ki = 3033 nM T79062 D08CKM 9863250 Ki = 3 nM T79062 D08DOG 25130235 Ki = 5900 nM T79062 D08OFG 11177588 Ki > 10000 nM T79062 D08UOX 5281148 IC50 = 117500 nM T79062 D08VGJ 9904281 Ki = 294 nM T79062 D09BNS 439280 Ki = 2.12 nM T79062 D09RPR 16737207 Ki > 10000 nM T79062 D09RXU 45488131 Ki > 500 nM T79062 D09WIL 10028436 Ki = 1.995 nM T79062 D0B9TN 46233353 Ki = 4110 nM T79062 D0BG5H 11957684 Ki = 1.259 nM T79062 D0C5GF 6918515 Ki = 155 nM T79062 D0C5XQ 1832 Ki = 30 nM T79062 D0CA9H 25107518 Ki = 16.6 nM T79062 D0CK9K 6918513 Ki = 300 nM T79062 D0F0IA 11301655 Ki > 2000 nM T79062 D0F6CD 5202 Ki = 0.11 nM T79062 D0FF6S 16038374 IC50 > 10000 nM T79062 D0FU5E 10220053 Ki > 1000 nM T79062 D0G7QT 10131112 IC50 = 3000 nM T79062 D0G8CV 9954003 Ki = 7.943 nM T79062 D0H3KU 172267 Ki = 466 nM T79062 D0H7PC 6918553 Ki > 10000 nM T79062 D0H9QG 5312148 Ki = 31.6 nM T79062 D0HE4S 68788 Ki = 18 nM T79062 D0I0ML 35985234 Ki = 7.5 nM T79062 D0J6JT 1355 Ki = 304 nM T79062 D0K0HU 16747715 Ki = 7.6 nM T79062 D0K5NZ 68848 Ki = 7.943 nM T79062 D0KS0I 24894910 EC50 > 10000 nM T79062 D0L5MW 181743 Ki = 67 nM T79062 D0LT5D 11267988 Ki = 3.38 nM T79062 D0LV7U 10667433 Ki = 32 nM T79062 D0O3GF 1220 Ki = 388 nM T79062 D0OG0R 10337743 IC50 = 4764 nM T79062 D0R3GW 10296414 Ki = 199.53 nM T79062 D0T2RY 9948320 Ki >= 1000 nM T79062 D0X4PH 11224758 Ki = 0.22 nM T79062 D0X6MT 4106 EC50 = 0.6 nM T79062 D0X7SD 888197 Ki = 156 nM T79062 D0X9YS 23642275 Ki = 0.6 nM T79062 D0XX2U 16006606 Ki = 8.2 nM T79062 D0Y0SA 135399666 EC50 > 10000 nM T79062 D0Y9TL 13702393 Ki = 793 nM T68251 D00HNB 25419 IC50 = 145000 nM T68251 D00MDP 466151 Ki = 0.05 nM T68251 D01UBX 451415 IC50 = 9900 nM T68251 D01XWG 30323 IC50 = 1900 nM T68251 D04AIT 5280445 IC50 = 3610 nM T68251 D07VLY 31703 IC50 = 1100 nM T68251 D0K8KX 5280343 IC50 = 6680 nM T68251 D0Q8CS 60937 IC50 = 7200 nM T68251 D0R9BG 1990 IC50 = 15000000 nM T68251 D0RA5Q 72172 IC50 = 3400 nM T68251 D0S0LZ 54671203 IC50 = 24000 nM T68251 D0V4GY 9552079 IC50 = 7630 nM T68251 D0VM2L 68740 IC50 = 7000 nM T68251 D04LTF 9868980 IC50 = 0.46 ug.mL-1 T68251 D05VZE 119031 IC50 = 0.43 nM T68251 D0F2JS 15547703 IC50 = 190 nM T68251 D0MW3H 9824350 Ki = 154 nM T68251 D0N4IV 10718956 IC50 = 1.7 nM T68251 D0U2BH 65064 IC50 = 9600 nM T68251 D09EFW 46861776 IC50 = 3.42 nM T68251 D0G1LL 74221072 IC50 = 35000 nM T68251 D0LO1Z 5281858 IC50 = 6300 nM T68251 D0N6ZA 74221131 IC50 > 100000 nM T68251 D0UM5R 74221070 IC50 = 4700 nM T68251 D00UCC 9827497 IC50 = 0.78 nM T68251 D01DVX 9847838 IC50 = 482 nM T68251 D03BOZ 3342298 Ki = 0.22 nM T68251 D05VNG 9908389 IC50 = 1.8 nM T68251 D08CEE 10478364 Ki = 200 nM T68251 D0E5GY 9904965 IC50 = 7.4 nM T68251 D0P8YC 5362422 IC50 = 0.73 nM T68251 D0Q1CD 6918336 Ki = 11 nM T68251 D0T2IQ 443600 IC50 = 3000 nM T68251 D0T9HG 132519 IC50 = 0.104 nM T68251 D0Y1XT 128564 Ki < 1 nM T68251 CNA81R 1836 Ki = 80 nM T68251 CQS47H 2299 IC50 = 0.5 nM T68251 CZ45IU 4219 IC50 = 3.6 nM T68251 C24IRS 4222 Ki = 2000 nM T68251 CW1H7U 4323 IC50 = 5.998 nM T68251 CS8X0P 16124 IC50 = 49000 nM T68251 CL2W6Q 38422 IC50 = 7100 nM T68251 CA3M5F 68443 IC50 = 389000 nM T68251 CYEU83 69033 Ki = 70000 nM T68251 C0PY5N 77754 Ki > 100 nM T68251 C5Z1QA 96028 IC50 > 200000 nM T68251 CP4O2C 121255 Ki = 65000 nM T68251 CCY6L8 169853 IC50 = 31400 nM T68251 C7ROG5 177347 IC50 = 91.3 nM T68251 CP7Q8T 240910 Ki = 15000 nM T68251 CX3DK6 283995 Ki = 9000 nM T68251 CBN39D 285263 IC50 = 86.74 nM T68251 COFX01 352863 Ki = 70000 nM T68251 CNM0P3 391527 IC50 = 7 nM T68251 C4U7SY 401129 IC50 = 18700 nM T68251 CV60YH 445010 IC50 = 5 nM T68251 CK9M3P 445018 IC50 = 1 nM T68251 C4D7TS 448002 IC50 = 9.1 nM T68251 CR51PG 448593 Ki = 210 nM T68251 CC54LQ 450256 IC50 > 100000 nM T68251 CG1I8P 467296 IC50 = 88000 nM T68251 CTPW02 467297 IC50 = 34000 nM T68251 C9I8WB 478379 Ki = 0.2 nM T68251 C45JSH 639942 IC50 = 5.28 nM T68251 CP91NX 677915 IC50 = 1649.92 nM T68251 CS4O7K 685005 IC50 > 500000 nM T68251 CDE9V2 689424 IC50 = 1945.82 nM T68251 C5O0TJ 690158 IC50 = 8.95 nM T68251 C7TPR6 690965 IC50 = 5.37 nM T68251 CP1Q6R 703233 IC50 = 61000 nM T68251 C9FL2X 721434 IC50 = 1785.67 nM T68251 CTO15S 727131 IC50 = 9.17 nM T68251 CTV50K 727184 IC50 = 1859.32 nM T68251 C2CL6X 732134 IC50 = 6.32 nM T68251 CPKI76 765318 IC50 = 9.99 nM T68251 CXME85 766168 IC50 = 9.72 nM T68251 CWQG91 770865 IC50 > 1000 nM T68251 CQB03J 780790 IC50 = 6.41 nM T68251 C7EHR1 787183 IC50 = 5.46 nM T68251 C5MF2E 795596 IC50 = 1853.73 nM T68251 C1K0NF 795855 IC50 = 9.13 nM T68251 CW56XG 875024 IC50 = 9.66 nM T68251 C17IXT 910211 IC50 = 9.02 nM T68251 C9IFC6 1348435 IC50 = 2700 nM T68251 C8A5CX 1800786 IC50 = 500 nM T68251 CN9C8D 2140735 IC50 = 350000 nM T68251 C36DGS 2211098 IC50 = 53 nM T68251 CN6E3U 2366268 IC50 = 3600 nM T68251 C1ND5S 2734394 IC50 = 121000 nM T68251 CN62WX 2800809 IC50 > 10000 nM T68251 CEHZ37 3042462 IC50 = 383000 nM T68251 CY3TD6 3348132 Ki = 20 nM T68251 CME24U 3649035 IC50 = 26000 nM T68251 C3EI6T 4085085 IC50 = 67000 nM T68251 CBN96T 4358655 IC50 = 50118.72 nM T68251 CC5O4E 4369384 IC50 = 2000 nM T68251 CP8D7Y 4478236 IC50 = 20 nM T68251 CQ4Y5M 4626827 IC50 = 4.6 nM T68251 CZBY34 5220706 Ki = 72000 nM T68251 C20HRJ 5273475 IC50 = 6.24 nM T68251 CZS0G5 5276565 IC50 > 100000 nM T68251 C3JN0F 5277465 IC50 > 100000 nM T68251 CRJK67 5277481 IC50 = 37400 nM T68251 CYF7S5 5277490 IC50 = 15500 nM T68251 CQ4VL5 5287415 IC50 = 0.8 nM T68251 CW5SE3 5288615 IC50 = 4.7 nM T68251 CJ3QI1 5288814 IC50 = 2905 nM T68251 C5IDT0 5289314 Ki = 115 nM T68251 CVLS16 5319161 IC50 = 3880 nM T68251 CZC3I7 5326979 IC50 = 58000 nM T68251 CL89FO 5496920 Ki = 33 nM T68251 CDI23X 5941957 IC50 > 100000 nM T68251 C1K8FQ 6439677 IC50 = 800 nM T68251 CJG2B7 6476333 IC50 = 8960 nM T68251 CL5DH0 6479915 IC50 = 3580 nM T68251 CQEF36 6539670 IC50 = 1 nM T68251 C1LQD2 6540261 IC50 = 1100 nM T68251 CP7BG0 6852146 IC50 = 5 nM T68251 CN5L2B 6852147 IC50 = 1.5 nM T68251 CP2XK7 6882342 IC50 = 120000 nM T68251 CPFV65 6916013 Ki = 81.28 nM T68251 C7AZE5 6930803 IC50 = 100 nM T68251 C7Y1BX 9543420 IC50 = 13.3 nM T68251 CIJ25V 9794947 IC50 = 20000 nM T68251 CLK61C 9797144 Ki = 73 nM T68251 C7NP9Z 9798247 IC50 = 28 nM T68251 CET56A 9801414 Ki = 10 nM T68251 C76RCQ 9801569 IC50 = 341 nM T68251 C68HMJ 9801786 IC50 = 380 nM T68251 CJY12B 9802219 Ki > 3000 nM T68251 CIXD67 9802768 IC50 = 0.33 nM T68251 CUSD58 9803469 IC50 = 19 nM T68251 C4A0XM 9804305 IC50 = 457 nM T68251 CQ46XD 9804842 IC50 = 8700 nM T68251 CP65QD 9805079 Ki = 482 nM T68251 C1HP7E 9805710 IC50 = 25 nM T68251 CASW18 9806452 Ki = 17 nM T68251 C76CKA 9807105 Ki = 805 nM T68251 CTK6J8 9808181 IC50 = 34200 nM T68251 C9RQM7 9808674 IC50 = 0.3 nM T68251 CTO36D 9817594 IC50 = 30000 nM T68251 C5OE1B 9821883 Ki = 11 nM T68251 CJC20A 9822095 IC50 = 17 nM T68251 C6KJ9W 9822461 IC50 = 8.7 nM T68251 C6IX7G 9822926 IC50 < 0.1 nM T68251 C1MPW9 9823182 IC50 = 19 nM T68251 CTF8V4 9823391 Ki > 3000 nM T68251 CVN5Z3 9823395 IC50 = 12 nM T68251 C1PW5U 9824010 IC50 = 998 nM T68251 CDJB86 9825720 IC50 = 0.1 nM T68251 CXL65P 9825920 Ki > 3300 nM T68251 CL0G8K 9825927 IC50 = 602.56 nM T68251 C65ZHY 9826199 IC50 = 0.61 nM T68251 C1I6KQ 9826286 Ki = 500 nM T68251 C1A7NJ 9827355 Ki = 0.71 nM T68251 C3SZ8Y 9827469 Ki = 1244 nM T68251 C7I2FO 9828039 Ki = 324 nM T68251 C1GR4N 9828276 IC50 > 25000 nM T68251 CC1NG5 9829581 IC50 = 20 nM T68251 C7SRM4 9837496 IC50 = 3000 nM T68251 C9PW7L 9841168 Ki = 28.5 nM T68251 C5XL7R 9841323 IC50 = 0.6 nM T68251 CA7DJ9 9842114 IC50 = 3.199 nM T68251 C32JRZ 9843079 IC50 = 140 nM T68251 C6YT5W 9843479 IC50 = 40 nM T68251 CWY1J9 9846501 Ki > 3000 nM T68251 CE9AL3 9847113 IC50 < 0.1 nM T68251 CA1IP0 9847191 Ki > 3000 nM T68251 C8IMT2 9847787 IC50 = 1.1 nM T68251 C7VXJ5 9848025 IC50 = 3.9 nM T68251 C4IEK0 9850035 IC50 = 0.2 nM T68251 CD1KW6 9851858 Ki = 0.01 nM T68251 C5DGI9 9851911 IC50 = 6.6 nM T68251 C2FYO3 9852206 Ki = 0.01 nM T68251 C5TUJ7 9862317 IC50 = 39 nM T68251 C8GE7U 9862764 IC50 = 59 nM T68251 CS5JT6 9864502 IC50 = 59 nM T68251 CQ0J1G 9865191 IC50 = 17 nM T68251 CI8Z0R 9866250 IC50 = 1.6 nM T68251 CQ9SG1 9866486 IC50 = 1208 nM T68251 CR10NL 9866770 Ki > 3000 nM T68251 C0YN1X 9867935 IC50 = 20 nM T68251 CK3F1T 9868079 IC50 = 1.3 nM T68251 CX57RB 9868249 Ki > 3000 nM T68251 CJS23I 9868333 Ki > 3333 nM T68251 CJ8DP1 9868672 IC50 > 6000 nM T68251 C24JSB 9868858 IC50 = 2 nM T68251 CLQ29X 9869597 IC50 = 262 nM T68251 CG17NZ 9869811 IC50 = 4 nM T68251 CMEA71 9869947 IC50 = 0.5 nM T68251 C38BVX 9870100 IC50 = 19 nM T68251 CZO2I0 9870133 IC50 = 3 nM T68251 CA48SX 9870269 IC50 = 743 nM T68251 CD1XQ2 9871305 IC50 = 1.9 nM T68251 CSM16R 9871355 IC50 = 158 nM T68251 CHU9I8 9871883 IC50 < 1 nM T68251 C5NM6P 9872886 Ki = 91 nM T68251 C0TCJ2 9880675 Ki = 667 nM T68251 CW8IC4 9882151 IC50 > 100000 nM T68251 C0ZT7A 9883002 Ki = 13.9 nM T68251 C75DAZ 9885136 IC50 = 0.65 nM T68251 CG35XZ 9885916 IC50 = 148 nM T68251 CZBK85 9886177 IC50 = 21 nM T68251 C2M4EC 9887473 Ki > 3333 nM T68251 C4PB5Z 9887544 IC50 = 2.6 nM T68251 C3ZG6O 9887870 IC50 = 4 nM T68251 C8AJB7 9888429 Ki > 3000 nM T68251 CVP45O 9888530 IC50 = 175 nM T68251 CDW1O4 9888922 IC50 = 196 nM T68251 CD1U5P 9889190 IC50 = 12 nM T68251 C27HMG 9889517 IC50 = 1.6 nM T68251 C26SZX 9890226 IC50 = 0.4 nM T68251 CWN19T 9890526 IC50 = 3.3 nM T68251 CD79UJ 9890632 IC50 = 92000 nM T68251 CU65HY 9891358 IC50 = 0.06 nM T68251 C3QSE6 9891814 IC50 = 18 nM T68251 CF1X0W 9892321 IC50 = 534 nM T68251 CH69LT 9892815 IC50 < 0.1 nM T68251 CZU7Y4 9892876 IC50 = 73 nM T68251 CK1F3O 9892889 Ki > 305 nM T68251 C1NCU4 9894184 IC50 = 300 nM T68251 CX5G0F 9894469 IC50 = 1300 nM T68251 CZK6O9 9895099 IC50 = 300 nM T68251 CSIB97 9896504 IC50 > 30000 nM T68251 C5DW9S 9902427 IC50 > 30000 nM T68251 C97GSC 9903557 Ki = 1915 nM T68251 CD78ZQ 9907286 IC50 = 0.7 nM T68251 CN6WJ1 9909994 IC50 = 230 nM T68251 CJ3K1I 9910075 IC50 = 1480 nM T68251 CPO8V1 9910282 IC50 = 430 nM T68251 CM2F7R 9910302 IC50 = 1.1 nM T68251 C6NUE9 9910550 IC50 = 0.5 nM T68251 CP4LS8 9910727 IC50 = 87 nM T68251 CT50EC 9912183 Ki = 194 nM T68251 C62VZI 9912382 IC50 = 0.7 nM T68251 C3AZP0 9913479 IC50 = 0.3999 nM T68251 CR98KH 9913488 IC50 = 853 nM T68251 CSZV76 9913881 IC50 = 41 nM T68251 C7ZY1L 9914029 IC50 = 62 nM T68251 CA3FW0 9918908 IC50 = 0.004 nM T68251 CG1A6B 9924640 IC50 > 100000 nM T68251 C4YGT6 9928325 IC50 = 7.5 nM T68251 CK5OV9 9930210 IC50 = 33 nM T68251 C03GVA 9932290 Ki = 210 nM T68251 C1I2FW 9932632 Ki > 3000 nM T68251 CCHZ97 9932731 IC50 = 58000 nM T68251 CDXR37 9933197 IC50 = 0.1 nM T68251 CX17KQ 9933408 IC50 = 29 nM T68251 CF26MY 9934052 Ki > 3000 nM T68251 CA5V8M 9934053 Ki = 433 nM T68251 C57WSD 9934240 IC50 = 7 nM T68251 C65ION 9935032 IC50 = 0.1 nM T68251 CGFD83 9936194 IC50 = 188 nM T68251 C1HRU9 9936228 IC50 = 4.1 nM T68251 C68MQN 9936625 Ki = 435 nM T68251 C9OUC8 9936681 IC50 = 196 nM T68251 CG38KL 9936728 Ki = 1.1 nM T68251 CE59TP 9936926 IC50 = 547 nM T68251 CX7VQ9 9937188 IC50 = 10.96 nM T68251 CLM2R8 9941370 Ki = 3.5 nM T68251 C0IBF2 9941371 Ki = 0.03 nM T68251 CA30JY 9946988 IC50 = 70 nM T68251 CWZC93 9947332 IC50 > 100000 nM T68251 CSN61C 9948296 Ki = 1497 nM T68251 C16HTN 9948666 Ki = 27 nM T68251 CF1DO9 9950475 Ki > 567 nM T68251 CQY54S 9952396 IC50 = 2.1 nM T68251 C8C3DL 9953278 IC50 = 539.51 nM T68251 C16GIN 9953861 Ki > 1267 nM T68251 CR6EX3 9953909 Ki = 446 nM T68251 C8RXN6 9954304 IC50 = 297 nM T68251 C9X0YR 9954867 Ki = 6300 nM T68251 CK9HX0 9955125 IC50 = 0.4 nM T68251 C05HGV 9955795 IC50 = 1.1 nM T68251 C8M2RB 9956613 IC50 > 10000 nM T68251 C3Q2UJ 9956686 IC50 = 0.4 nM T68251 CS73TB 9956692 Ki = 2800 nM T68251 CI5TW9 9956699 IC50 = 529 nM T68251 CN76XI 9957653 IC50 = 1 nM T68251 CVG0O2 9959014 IC50 = 0.9 nM T68251 CN8TK0 9959428 IC50 = 661 nM T68251 CV40RB 9960075 Ki = 391 nM T68251 C9DRB7 9966028 IC50 = 110 nM T68251 C8K5VD 9969928 IC50 > 30000 nM T68251 CFQ15E 9976696 IC50 = 22 nM T68251 C0HL2X 9976697 IC50 = 2.7 nM T68251 C09LSY 9979489 Ki > 3333 nM T68251 CUA65C 9982414 IC50 = 12 nM T68251 CJGR30 9983604 IC50 = 0.5 nM T68251 CILK24 9983687 Ki = 1 nM T68251 CO0TX7 9993891 Ki > 600000 nM T68251 C3KX1B 9998685 Ki = 1 nM T68251 CB2J3S 9999667 IC50 = 10 nM T68251 C8W5UK 9999879 IC50 = 120 nM T68251 C6TO0A 10001582 Ki = 1.5 nM T68251 C59WEK 10001843 IC50 < 0.1 nM T68251 C5HN3L 10001964 IC50 = 222 nM T68251 CP5N4E 10005114 Ki = 43 nM T68251 C6U3CK 10006134 IC50 = 0.5 nM T68251 CA8C6U 10008733 Ki = 0.01 nM T68251 CR7T3J 10009978 Ki = 700 nM T68251 C71YGT 10025307 Ki = 4.7 nM T68251 C6O0MN 10026682 Ki = 5300 nM T68251 C6DGR7 10027203 Ki = 1.5 nM T68251 C4VJX9 10027747 IC50 = 32000 nM T68251 CM52RO 10030422 IC50 = 10 nM T68251 CJR59P 10031295 Ki > 3333 nM T68251 CX2W9O 10037048 IC50 = 200 nM T68251 C7J9ZF 10039403 IC50 = 32 nM T68251 C1X0SA 10041385 Ki = 8 nM T68251 CO39PK 10042482 Ki = 39.81 nM T68251 CW2MK1 10043732 Ki = 46 nM T68251 C7CT4E 10045150 IC50 = 0.34 nM T68251 CHF92V 10047100 Ki = 0.23 nM T68251 CCF5Z4 10047585 IC50 = 0.3 nM T68251 CAN59F 10047708 IC50 = 2.2 nM T68251 CV59KC 10049292 Ki = 340 nM T68251 CLZ87W 10051236 Ki = 1598 nM T68251 CSHD67 10054852 IC50 = 0.4 nM T68251 C42YWK 10055393 IC50 = 229.09 nM T68251 CSW7B3 10067146 Ki = 2.8 nM T68251 C69DPZ 10068042 IC50 = 15800 nM T68251 CD3RL7 10070821 Ki > 10000 nM T68251 CB28NP 10073353 IC50 = 30 nM T68251 CJK0R1 10074190 IC50 = 1 nM T68251 CU7DJ1 10081163 Ki = 77000 nM T68251 C8AEK4 10093420 IC50 = 0.38 nM T68251 C5W4ZA 10094362 IC50 = 300 nM T68251 CA6X2Z 10095338 IC50 = 0.6 nM T68251 CMY3X2 10098158 IC50 = 6.1 nM T68251 C2XV5J 10098250 IC50 = 0.4 nM T68251 C3V2HW 10099112 IC50 = 2 nM T68251 CXV2Y3 10109170 Ki = 433 nM T68251 CY6HZ7 10111132 IC50 = 74900 nM T68251 C0G7IY 10114318 Ki = 1870 nM T68251 C4P1LB 10116618 IC50 = 0.44 nM T68251 CU0D4S 10117481 Ki > 3333 nM T68251 CP5L0W 10117663 Ki > 3300 nM T68251 C7OPQ8 10118047 IC50 = 35 nM T68251 C7A8MI 10120093 IC50 < 0.1 nM T68251 CT4V0P 10120622 IC50 = 0.39 nM T68251 CY2N3D 10127629 Ki > 3330 nM T68251 C1N4MJ 10127670 Ki > 3330 nM T68251 CIL09Z 10127889 Ki > 3330 nM T68251 CYU19P 10127901 Ki > 3330 nM T68251 C07KFI 10128313 Ki > 3330 nM T68251 CB3I6K 10128659 Ki > 3330 nM T68251 C6ZK3A 10128916 Ki > 3330 nM T68251 CH0UW2 10129190 Ki > 3330 nM T68251 CZM7F4 10132758 IC50 = 80000 nM T68251 CDR73P 10135184 Ki > 2128 nM T68251 C7KR3Y 10136680 Ki = 440 nM T68251 CNU93J 10136924 Ki = 450 nM T68251 C1CDF2 10136925 Ki = 340 nM T68251 CJ9EX4 10138303 Ki = 550 nM T68251 CFXC89 10139040 Ki > 3333 nM T68251 CGC6S5 10139402 Ki > 3333 nM T68251 CP8QV4 10140363 Ki = 1920 nM T68251 CU6Y9T 10140438 Ki > 3333 nM T68251 CE75BY 10140776 Ki = 1400 nM T68251 CIH36M 10141214 IC50 = 18 nM T68251 C6MSI0 10141443 IC50 = 33000 nM T68251 CLXF15 10141613 Ki > 3300 nM T68251 C7VF1K 10141614 Ki > 3300 nM T68251 CWB5O4 10142326 Ki > 3300 nM T68251 CL7P6G 10143019 IC50 = 0.098 nM T68251 CPXB21 10143028 Ki > 3333 nM T68251 C23WZR 10143587 Ki > 3300 nM T68251 CZW98O 10156375 Ki = 3.8 nM T68251 CYO8D2 10159633 Ki > 3333 nM T68251 CQ4SJ5 10160197 Ki > 3333 nM T68251 CQ41YI 10161391 Ki > 3333 nM T68251 C7SXD4 10162245 Ki > 3300 nM T68251 CO6PS3 10162900 Ki = 150 nM T68251 CR5H6E 10163627 Ki > 2128 nM T68251 CI9VJ5 10163857 Ki > 3333 nM T68251 CR17PV 10164205 Ki > 3333 nM T68251 CZO5V4 10164317 IC50 < 0.4 nM T68251 CCM0Y8 10165180 Ki = 2167 nM T68251 C5ZO9J 10166232 IC50 = 0.53 nM T68251 C6IW4O 10173876 Ki > 3330 nM T68251 CGB27E 10174981 Ki > 3330 nM T68251 CL47AR 10175070 Ki > 3330 nM T68251 C4ULO6 10175077 Ki > 3330 nM T68251 C4QY3V 10175210 Ki = 3100 nM T68251 C84ZQD 10175219 Ki > 3330 nM T68251 CIT0H4 10175323 Ki > 3330 nM T68251 C95IGP 10175331 Ki = 2170 nM T68251 C4PDJ5 10175366 Ki = 110 nM T68251 CT7U0M 10175426 Ki > 3330 nM T68251 CD4AO0 10180362 IC50 = 2300 nM T68251 CEWF13 10180993 IC50 = 81800 nM T68251 CCX3T6 10183064 Ki > 15000 nM T68251 CDM94B 10183693 Ki > 3300 nM T68251 CHB2D3 10184071 Ki > 3333 nM T68251 C3E9NF 10184537 Ki > 3300 nM T68251 CTDP62 10184579 Ki > 3300 nM T68251 CXQ8N0 10185100 Ki > 3333 nM T68251 CK0P3F 10186536 Ki > 2128 nM T68251 CV7YI1 10186544 Ki > 3300 nM T68251 C51RPY 10195069 Ki > 3330 nM T68251 CCHX74 10195307 Ki = 200 nM T68251 C94KHT 10195527 Ki = 930 nM T68251 CDG35O 10196192 Ki = 370 nM T68251 CY36NO 10196425 Ki > 3330 nM T68251 C1JG5W 10196775 Ki > 3330 nM T68251 CVRZ27 10198038 IC50 = 80 nM T68251 C5CUM9 10202769 Ki > 3333 nM T68251 CX8BS3 10203685 Ki > 3333 nM T68251 CE1LI3 10204303 Ki = 90 nM T68251 C32RAQ 10204620 Ki > 3300 nM T68251 CQFP69 10206106 Ki = 270 nM T68251 CS1CA5 10207780 Ki = 1333 nM T68251 C4K1MJ 10208262 Ki > 2128 nM T68251 CYE02Q 10209301 IC50 = 2.6 nM T68251 CD76KE 10209382 Ki > 3333 nM T68251 CG8FA4 10218128 Ki > 3330 nM T68251 C7Y2US 10218353 Ki > 3330 nM T68251 C1C7AH 10223757 Ki > 3333 nM T68251 CYG10Z 10223774 Ki > 3333 nM T68251 CV5X8A 10224181 IC50 > 30000 nM T68251 CGKU70 10224396 Ki = 240 nM T68251 C7K1OR 10224602 IC50 = 1800 nM T68251 CLH71C 10225319 Ki > 3333 nM T68251 C2X1KF 10226116 Ki = 2566 nM T68251 C9CSG3 10226996 IC50 = 650 nM T68251 CUE63Q 10227853 Ki > 3300 nM T68251 C19DFP 10227854 Ki > 3300 nM T68251 CM7B5T 10228228 Ki > 3333 nM T68251 C7T0WH 10229644 IC50 = 1.1 nM T68251 CD2HP3 10230012 Ki = 1333 nM T68251 CCRM18 10231253 IC50 = 1.2 nM T68251 CCTY95 10237492 Ki > 3330 nM T68251 CQH2U3 10238391 IC50 = 200 nM T68251 CO8M7Q 10239526 Ki > 3330 nM T68251 CCQ9V5 10239716 Ki > 3330 nM T68251 CEO4X5 10239762 Ki > 3330 nM T68251 CU7TQ3 10239803 Ki > 3330 nM T68251 CLAX20 10250594 IC50 = 4.2 nM T68251 C0J3TC 10250722 Ki = 60 nM T68251 CL67DT 10252311 Ki < 2.8 nM T68251 CQJ0R3 10252900 Ki = 0.66 nM T68251 CK9DF5 10253223 IC50 = 12000 nM T68251 CQF3V9 10253673 IC50 = 9 nM T68251 CD8QY2 10253933 IC50 > 10000 nM T68251 CB6SE4 10256227 IC50 = 91 nM T68251 C7HZ1M 10270281 IC50 = 21700 nM T68251 C3XD1E 10271240 IC50 > 100000 nM T68251 C2MES9 10271604 Ki > 100000 nM T68251 CWJ02G 10273315 IC50 > 30000 nM T68251 C0K2ES 10273642 Ki > 3333 nM T68251 CJZP24 10273657 Ki > 3333 nM T68251 CK18DB 10273985 Ki > 2128 nM T68251 CGP97S 10274748 Ki = 140 nM T68251 C13NKU 10275545 Ki > 3333 nM T68251 C1NGV9 10276473 Ki > 3333 nM T68251 CES6A5 10276821 Ki = 1566 nM T68251 C1W7SN 10277073 Ki > 3333 nM T68251 CO18TA 10277120 Ki > 3333 nM T68251 CY6K1G 10277706 Ki > 3300 nM T68251 C2XU3O 10278147 IC50 = 0.67 nM T68251 C3IG0K 10280852 IC50 = 0.2 nM T68251 C80WUO 10282084 IC50 = 0.33 nM T68251 C7TWG0 10289551 Ki > 3330 nM T68251 CJ63ER 10289607 Ki > 3330 nM T68251 CR48SA 10289842 Ki > 3330 nM T68251 CO60CU 10290029 Ki = 2700 nM T68251 CJTV12 10293283 IC50 > 30000 nM T68251 CS69YG 10293394 IC50 = 3500 nM T68251 C89YGA 10295733 Ki > 2128 nM T68251 CDU36Y 10296475 Ki = 520 nM T68251 CTL3Y8 10296608 Ki > 3333 nM T68251 C48IRP 10296785 Ki = 500 nM T68251 CQ1Z0G 10298111 IC50 = 35 nM T68251 CN14MI 10298369 Ki > 3333 nM T68251 CU5E9Z 10299198 Ki = 1357 nM T68251 C25EKM 10299665 Ki > 3300 nM T68251 CQ5BE8 10299709 IC50 = 0.35 nM T68251 C1BR6A 10300063 Ki > 3333 nM T68251 C80VEU 10300077 Ki > 3333 nM T68251 C8U3KW 10301524 IC50 = 0.57 nM T68251 CFAU84 10301584 Ki > 3333 nM T68251 CP5AU1 10302088 Ki > 3333 nM T68251 C63BRA 10303333 IC50 = 34 nM T68251 CE1KM9 10311498 Ki > 3330 nM T68251 CJ15OB 10311501 Ki > 3330 nM T68251 C5F0EV 10311947 Ki > 3330 nM T68251 C4R9ZK 10311997 Ki = 83 nM T68251 CE6MB0 10312141 Ki = 116 nM T68251 C7G6QW 10312268 Ki > 3330 nM T68251 CQ5IT9 10312372 Ki > 3330 nM T68251 CP1GW0 10318094 Ki = 0.57 nM T68251 CIDW49 10319098 Ki > 3333 nM T68251 CF4KT9 10320002 Ki > 3333 nM T68251 CG23FV 10320328 IC50 = 4 nM T68251 CJWH74 10321975 Ki > 3333 nM T68251 CVKT01 10322744 IC50 = 50 nM T68251 CY08WJ 10322755 Ki > 3000 nM T68251 CQH5D4 10324032 IC50 = 0.1 nM T68251 CPI8R0 10324532 Ki = 3 nM T68251 CSFZ76 10325592 Ki = 1376 nM T68251 C1C4VZ 10326004 Ki = 0.9 nM T68251 C7UZA4 10340758 IC50 = 3.2 nM T68251 CCK1A4 10342176 IC50 = 8 nM T68251 CFO74N 10343375 Ki = 430 nM T68251 CJIW74 10343996 IC50 = 0.31 nM T68251 C94ANQ 10347529 IC50 = 0.6 nM T68251 C9FU5G 10362663 IC50 = 1 nM T68251 CWIM61 10364088 IC50 = 756 nM T68251 CL4B2U 10364155 IC50 = 567 nM T68251 CBA5I4 10365560 Ki = 1.1 nM T68251 CH89GT 10365752 IC50 = 3.4 nM T68251 CI0T8K 10366352 Ki > 3333 nM T68251 C6WZ4F 10367355 IC50 = 16 nM T68251 CT81YN 10370089 IC50 = 30 nM T68251 CBTO07 10370226 Ki > 3333 nM T68251 C0IUQ7 10387351 Ki > 3333 nM T68251 CZNT94 10389113 IC50 = 4 nM T68251 CY2G0R 10391428 Ki > 3333 nM T68251 C16BSA 10394828 IC50 = 50 nM T68251 CFKA79 10395015 Ki > 2000 nM T68251 C9HM1A 10402302 IC50 = 76000 nM T68251 CLP05D 10407603 IC50 = 5.2 nM T68251 C98HMP 10413940 Ki = 249 nM T68251 C7K0HG 10414437 Ki = 31 nM T68251 CH1S2G 10414974 Ki = 2.5 nM T68251 C4J7IP 10416507 Ki = 86 nM T68251 C0V9FN 10433382 IC50 = 0.1995 nM T68251 CS32HR 10435935 IC50 = 5.1 nM T68251 C7XE1L 10437629 IC50 = 5000 nM T68251 C5WV1N 10439082 Ki = 1867 nM T68251 C54UDR 10453826 IC50 = 891.25 nM T68251 CQUR30 10454592 Ki = 0.21 nM T68251 C6T8VC 10456675 Ki = 0.6918 nM T68251 C8M9FE 10462640 Ki = 30000 nM T68251 CA7DM9 10474389 IC50 = 0.7 nM T68251 CNQZ36 10483139 Ki = 410 nM T68251 COT6G1 10492779 Ki > 200000 nM T68251 C9KHT4 10495552 Ki = 30 nM T68251 CA7HT2 10498521 Ki = 15 nM T68251 C6KD0A 10498747 IC50 = 1.4 nM T68251 CL8O6I 10500340 Ki = 69 nM T68251 CGK80V 10500816 Ki = 35 nM T68251 CVID65 10500886 Ki = 17.78 nM T68251 CP37WK 10501527 Ki = 17 nM T68251 CK6YN5 10501862 Ki = 6 nM T68251 CZ2UY0 10502046 IC50 = 1 nM T68251 C36OMW 10502172 IC50 = 1 nM T68251 C9QE1B 10502327 Ki = 8 nM T68251 CHOX65 10502351 IC50 = 6.7 nM T68251 C5V8HJ 10502382 IC50 < 0.4 nM T68251 CJZ5T8 10502487 IC50 = 2770 nM T68251 CZ1R5Q 10502869 Ki = 8100 nM T68251 CBNM82 10503128 IC50 < 0.4 nM T68251 CO9S5H 10503708 Ki = 12 nM T68251 C5Y4IA 10504081 IC50 = 104 nM T68251 CD80YF 10504445 IC50 = 0.38 nM T68251 C2C7TE 10504472 IC50 = 2 nM T68251 CT2NM3 10505241 Ki = 19 nM T68251 CK2AB5 10505370 Ki = 2400 nM T68251 CH6S8Y 10505729 IC50 > 10000 nM T68251 C65KOE 10506125 IC50 = 33 nM T68251 C6D7JF 10506147 IC50 = 7 nM T68251 C7S0DB 10506158 IC50 = 16 nM T68251 CNH3L8 10506415 IC50 = 280 nM T68251 CS8V1G 10507004 Ki = 30 nM T68251 CV2T7C 10507137 Ki = 1800 nM T68251 C03MRW 10507152 Ki = 1.2 nM T68251 CDSO53 10507214 IC50 = 8.3 nM T68251 CFJ96A 10507282 Ki = 84 nM T68251 CC6H8T 10507755 Ki = 0.8 nM T68251 C9C5EL 10521197 IC50 = 8.4 nM T68251 CBT12Q 10522080 IC50 = 0.8 nM T68251 CXD8I5 10523292 Ki = 75 nM T68251 CZ36JW 10523383 IC50 = 530 nM T68251 C90HBF 10523728 Ki = 13 nM T68251 CQEH42 10524134 IC50 = 0.7 nM T68251 CYU87N 10524260 IC50 = 0.5 nM T68251 CX6EB7 10524337 Ki = 1800 nM T68251 CQTF46 10524338 Ki = 300 nM T68251 CYB53K 10525912 Ki = 33 nM T68251 CJK6G1 10526509 IC50 < 0.4 nM T68251 CSLO13 10526877 IC50 = 1000 nM T68251 CEK90M 10527263 IC50 = 50 nM T68251 CA83ON 10527749 IC50 = 18 nM T68251 CYGU41 10529315 IC50 = 1475 nM T68251 CBV6X5 10529587 IC50 = 4.4 nM T68251 CGK37L 10529602 Ki = 1.5 nM T68251 CIOJ69 10529720 Ki = 3000 nM T68251 C6PGE1 10530040 Ki = 380 nM T68251 C30UCT 10530499 Ki = 13 nM T68251 CQ82VY 10530944 Ki = 24 nM T68251 CEV6I5 10531005 Ki = 50 nM T68251 CJ2TZ3 10531167 Ki = 19 nM T68251 CS0AD8 10532048 Ki 17 nM T68251 C0WHA9 10546565 Ki = 9 nM T68251 C06NQR 10547080 IC50 = 66 nM T68251 C40ZXE 10547784 Ki = 7 nM T68251 CS10ZB 10549106 Ki = 19 nM T68251 C4PK0U 10549114 IC50 = 2.4 nM T68251 C4TA1K 10549256 IC50 < 0.4 nM T68251 C5JS8L 10549329 Ki = 10 nM T68251 CG27UI 10549756 Ki = 39 nM T68251 C82HQE 10550145 Ki = 6 nM T68251 C7WQ5Z 10550399 IC50 = 1 nM T68251 C1FA6T 10551440 IC50 = 50 nM T68251 CC2FM6 10551489 IC50 = 2391 nM T68251 C5UD0A 10551910 IC50 = 19 nM T68251 C4K3UD 10552661 Ki = 11 nM T68251 CU8QP7 10552732 Ki = 10 nM T68251 COYU34 10553872 Ki = 1900 nM T68251 C0S6GT 10554037 Ki = 16 nM T68251 CSQC42 10554611 Ki = 80 nM T68251 C7P5AW 10554727 Ki = 34 nM T68251 CI8XG0 10554869 IC50 = 8 nM T68251 CYJ41F 10554927 Ki = 3600 nM T68251 CZ41HP 10554978 Ki = 16 nM T68251 CD3R8V 10562830 IC50 = 8.32 nM T68251 CT7O9M 10569678 IC50 = 2 nM T68251 C8RWE4 10569743 IC50 = 36 nM T68251 C0M4VN 10570699 IC50 < 100 nM T68251 CE14GM 10570702 IC50 = 3 nM T68251 CUQ29Z 10571396 Ki = 170 nM T68251 CBXZ79 10572150 IC50 = 6 nM T68251 CPF0R5 10572544 Ki = 20 nM T68251 C21VZS 10573362 IC50 = 1.6 nM T68251 C42IAF 10573603 Ki = 15 nM T68251 CG39CF 10574279 Ki = 13 nM T68251 C8LYR6 10574340 IC50 < 1000 nM T68251 C42BTA 10576058 IC50 < 40 nM T68251 CH7Z2V 10576110 IC50 = 81 nM T68251 CK3JV9 10576740 IC50 = 3.3 nM T68251 CJ7KH8 10578213 Ki = 49 nM T68251 C1KH7E 10578728 IC50 = 9 nM T68251 CK05ZH 10579086 Ki = 0.7 nM T68251 C3R2SO 10580533 Ki = 20 nM T68251 C8J6HS 10591505 Ki = 83.18 nM T68251 CIUO27 10593253 IC50 = 2 nM T68251 CB20LM 10594000 Ki = 18 nM T68251 CUTS47 10594564 IC50 = 33 nM T68251 CN4Y6H 10594565 IC50 = 7 nM T68251 CD65OG 10594830 IC50 = 10.96 nM T68251 CJQY74 10595685 IC50 = 50 nM T68251 CI71CK 10595804 Ki = 10 nM T68251 CYNC76 10596158 IC50 = 12 nM T68251 CD65NF 10597516 Ki = 25 nM T68251 CP2H8O 10597673 Ki = 9 nM T68251 CL7EX4 10598952 IC50 > 1000 nM T68251 CUZ73T 10599048 IC50 = 50 nM T68251 CQCW86 10599579 IC50 < 0.4 nM T68251 CW18QK 10599594 IC50 = 1.2 nM T68251 CR1JI4 10600645 IC50 = 7 nM T68251 CN3E8J 10600844 Ki = 1.3 nM T68251 CJ86TP 10601066 IC50 > 1000 nM T68251 C5WUG1 10601082 Ki = 810 nM T68251 CEJ1U0 10603377 Ki = 18 nM T68251 C5G9MI 10610114 Ki = 120 nM T68251 C84URB 10610500 Ki > 100000 nM T68251 CPW6A4 10617505 IC50 > 1000 nM T68251 CL02BO 10618584 IC50 = 12 nM T68251 C06CAN 10619639 Ki = 12 nM T68251 CV14UH 10619971 Ki = 15 nM T68251 CR69NK 10621302 IC50 = 20 nM T68251 CSQ96T 10621933 Ki = 0.44 nM T68251 CVZ32G 10622447 Ki = 20 nM T68251 CL62YC 10622822 IC50 = 24 nM T68251 CL67UQ 10623250 IC50 = 8 nM T68251 C4FYL1 10623748 IC50 = 34 nM T68251 C6R4EG 10624005 Ki = 2 nM T68251 CR8X1Q 10624346 IC50 = 0.65 nM T68251 CKF6D7 10625329 Ki = 7.3 nM T68251 CGB29T 10625771 IC50 = 0.6 nM T68251 C6H9CT 10626366 Ki = 6900 nM T68251 C70MFZ 10626445 Ki = 18 nM T68251 C5VGB1 10626732 Ki = 21 nM T68251 C3NKC0 10626927 Ki = 17 nM T68251 CA63VQ 10640307 Ki = 36 nM T68251 C7KGM3 10642071 IC50 = 0.3 nM T68251 CI2QB9 10642965 IC50 < 0.4 nM T68251 CM1OZ6 10643325 IC50 = 5.9 nM T68251 C41RKE 10643401 Ki = 10 nM T68251 CUAI71 10643973 Ki = 2 nM T68251 CPYV83 10647658 Ki = 71000 nM T68251 CVX7Q2 10648390 Ki = 11 nM T68251 C4TXZ1 10648776 Ki = 100 nM T68251 C6S1KA 10649216 IC50 > 10000 nM T68251 C07FPQ 10649518 Ki = 55 nM T68251 COT6B8 10650624 Ki = 15 nM T68251 C69SPO 10650906 Ki = 0.6 nM T68251 CT23XW 10650907 Ki = 1.8 nM T68251 C13GKL 10658560 IC50 = 315000 nM T68251 C97KZU 10665624 IC50 = 39 nM T68251 CW1E7L 10667540 IC50 = 310 nM T68251 CF0E6H 10668745 IC50 = 13 nM T68251 CSCL07 10668823 Ki = 6.3 nM T68251 C4HJS1 10669027 Ki = 50 nM T68251 CFYC35 10669215 Ki = 3 nM T68251 C6TC0Z 10669216 Ki = 2.5 nM T68251 C78GYJ 10670529 IC50 = 1.3 nM T68251 C5FWS1 10670820 IC50 = 10 nM T68251 C4QVL0 10670896 Ki = 3 nM T68251 CB1F4G 10671203 IC50 = 110 nM T68251 C3DXN5 10671411 Ki = 0.92 nM T68251 CWB19K 10671441 Ki = 1.4 nM T68251 CXDM24 10671863 Ki = 0.54 nM T68251 C17LYV 10672346 IC50 = 26 nM T68251 CMU74I 10672857 IC50 = 6 nM T68251 CU6Y4O 10674458 Ki = 1600 nM T68251 CXTP56 10688727 IC50 < 1 nM T68251 CU5M1J 10691797 Ki = 42 nM T68251 CSA80H 10692194 IC50 < 1 nM T68251 CS5CL7 10692307 IC50 < 0.4 nM T68251 CR5KF8 10692994 IC50 = 535 nM T68251 CDI12G 10693559 IC50 = 6.8 nM T68251 C8JX1G 10693698 Ki = 3 nM T68251 CVML68 10693881 IC50 = 0.7 nM T68251 CM1T7K 10694510 Ki = 2.6 nM T68251 C7SM1E 10694604 Ki = 3.5 nM T68251 C3E1DX 10695165 IC50 = 4.4 nM T68251 C7ZQM4 10695491 Ki = 0.6 nM T68251 CZGC63 10695865 IC50 = 24 nM T68251 CVQF97 10695971 IC50 = 0.3 nM T68251 CW6CF7 10696226 IC50 = 2 nM T68251 C1YFC3 10696977 IC50 = 9 nM T68251 C4BME8 10697140 IC50 = 23 nM T68251 CBN9K8 10697378 Ki = 22 nM T68251 C1O5CQ 10697393 Ki = 210 nM T68251 CM4AI6 10698165 Ki = 100 nM T68251 C4THQ9 10698311 Ki = 280 nM T68251 C6Y1OU 10698367 Ki = 150 nM T68251 CG5JM9 10698412 Ki = 2.8 nM T68251 C56VSE 10698786 Ki = 1.5 nM T68251 C5E8QF 10707457 Ki = 87 nM T68251 C2GL3A 10714610 Ki = 44 nM T68251 C4IWF2 10714988 IC50 = 6 nM T68251 CO9KV7 10715115 IC50 < 1 nM T68251 C78CKH 10715629 IC50 > 20000 nM T68251 CE1D6G 10716217 IC50 = 3.5 nM T68251 C0ZX6T 10717308 IC50 = 9 nM T68251 C3TGW8 10717400 Ki = 61.66 nM T68251 CZ1M3L 10718058 Ki = 19 nM T68251 CQZ7M8 10718133 Ki = 13 nM T68251 CB96HF 10718916 IC50 > 1000 nM T68251 CN8AK6 10718996 Ki = 0.52 nM T68251 C2IS9D 10719476 Ki = 0.73 nM T68251 CVW81M 10719595 IC50 = 28 nM T68251 CI96XV 10720740 Ki = 14 nM T68251 CIV3P5 10720775 Ki = 760 nM T68251 C65IGZ 10720864 Ki = 21 nM T68251 CTGL64 10721152 Ki = 580 nM T68251 CF46SQ 10721337 Ki = 19 nM T68251 C4J1WN 10721454 IC50 = 0.2 nM T68251 CC1FB8 10721904 Ki = 2.5 nM T68251 CB2QD0 10723468 Ki = 0.9 nM T68251 CO7VP4 10737552 Ki = 18 nM T68251 C51DZG 10737732 IC50 = 11 nM T68251 C1LS5U 10738104 IC50 = 1 nM T68251 CL74TG 10738165 IC50 = 0.4 nM T68251 CB8G2D 10739728 Ki = 15 nM T68251 C4FWC9 10740485 Ki = 66 nM T68251 CKJD45 10741133 IC50 = 450 nM T68251 C0WKL7 10741470 Ki = 10 nM T68251 CPDX27 10741484 IC50 > 1000 nM T68251 C0QT2F 10741956 Ki = 7 nM T68251 CLI7B3 10742101 IC50 > 1000 nM T68251 CKX5R3 10742142 IC50 = 33 nM T68251 C39DPG 10742191 IC50 = 4.8 nM T68251 CHW23E 10742387 IC50 = 20 nM T68251 CY2BZ0 10742536 Ki = 41 nM T68251 C1LF0S 10744337 Ki = 48 nM T68251 CEV8X0 10744751 Ki = 25 nM T68251 CSM9H7 10745124 Ki = 800 nM T68251 C5BZ0J 10745489 Ki = 25 nM T68251 C9ILP3 10745718 IC50 = 31 nM T68251 C4IF2L 10745725 Ki = 25 nM T68251 CK30AE 10745748 Ki = 1.6 nM T68251 CWF50D 10745851 Ki = 21 nM T68251 CE09PI 10757715 IC50 = 6 nM T68251 CA3F1N 10758013 Ki = 43.65 nM T68251 CTKR07 10758266 Ki > 200000 nM T68251 CY9W4M 10760229 IC50 > 1000 nM T68251 CLEG16 10761206 Ki = 30 nM T68251 CDX13Z 10761730 Ki = 13 nM T68251 CA4U7D 10762262 Ki = 18 nM T68251 CP2G0N 10763745 Ki = 0.89 nM T68251 C68THN 10763851 IC50 = 0.3 nM T68251 CM54WS 10764477 Ki = 2400 nM T68251 CAG53Y 10764489 IC50 = 11.4 nM T68251 C7X6EC 10764497 Ki = 1500 nM T68251 CY8LV5 10765345 IC50 = 4.7 nM T68251 C3P2TS 10766036 IC50 = 17 nM T68251 CA6C0Z 10766622 Ki = 0.7943 nM T68251 CN6P1J 10766950 IC50 = 2.2 nM T68251 C0R1ZA 10767025 Ki = 0.64 nM T68251 CWR5Z3 10767105 IC50 = 29 nM T68251 CR4I1E 10767157 IC50 = 6 nM T68251 C7Q2EM 10767236 IC50 = 3 nM T68251 CNT4D0 10767387 Ki = 19 nM T68251 C18QVD 10768090 Ki = 61 nM T68251 C01YKA 10768236 IC50 = 13 nM T68251 CQ7J4I 10769007 IC50 = 12 nM T68251 C6VKJ9 10769394 Ki = 16 nM T68251 CQ6U2Y 10780743 Ki = 19 nM T68251 CIN4A9 10783989 Ki = 20 nM T68251 C15PVT 10785952 Ki = 20 nM T68251 CLAP90 10785969 IC50 = 23 nM T68251 C8AF9L 10787938 Ki = 0.88 nM T68251 C0DFB9 10788617 IC50 = 1 nM T68251 CNAE08 10788733 IC50 = 5 nM T68251 CXQD12 10789326 IC50 = 100 nM T68251 CM74LH 10789594 IC50 = 13 nM T68251 C8EOY6 10790150 Ki = 47 nM T68251 CHWG02 10790787 IC50 = 33 nM T68251 C0NP2Z 10790811 IC50 > 1000 nM T68251 C31EHR 10791372 IC50 = 84 nM T68251 C3P7LZ 10792025 Ki = 1.9 nM T68251 C8D1EN 10792133 IC50 = 3.9 nM T68251 C9VML0 10807861 Ki = 226000 nM T68251 CN8I3Z 10808172 IC50 = 9 nM T68251 CP72JG 10810483 IC50 = 4.8 nM T68251 CT1AI4 10810573 IC50 = 2 nM T68251 CU9F7V 10810684 Ki = 15 nM T68251 CS0O7M 10811110 Ki = 17 nM T68251 C49HCM 10812120 IC50 < 40 nM T68251 CEM1J0 10812918 IC50 < 40 nM T68251 CZB7L2 10812929 IC50 = 1.3 nM T68251 C4TF0K 10813874 IC50 < 0.4 nM T68251 CIUN51 10814028 IC50 = 46 nM T68251 CS7BY4 10816934 IC50 = 4 nM T68251 C3AI5Z 10831752 IC50 = 49 nM T68251 CMX2J7 10832371 IC50 > 1000 nM T68251 CF50HD 10832925 IC50 = 4 nM T68251 COE82D 10833334 Ki = 38.9 nM T68251 C5OG4U 10833497 IC50 = 61 nM T68251 C2A0IX 10833840 IC50 = 46.3 nM T68251 CH90ZB 10834348 IC50 = 14 nM T68251 C9M1JI 10834357 Ki = 10.96 nM T68251 CND0X1 10834889 IC50 = 130 nM T68251 CT3MN0 10837022 Ki = 4.6 nM T68251 CGR16B 10837261 IC50 = 1000 nM T68251 CR0E9Q 10837740 Ki = 3.89 nM T68251 C9H4CP 10838922 Ki = 0.52 nM T68251 CB32OK 10838949 IC50 > 1000 nM T68251 CR50UM 10839419 Ki = 5 nM T68251 CHWQ34 10839761 Ki = 1300 nM T68251 CA76MU 10840059 IC50 = 1160 nM T68251 CPD3L7 10840455 Ki = 32 nM T68251 CR2UX3 10840602 Ki = 94 nM T68251 CL1KG7 10840630 Ki = 24 nM T68251 CI0HR4 10840639 Ki = 39 nM T68251 C6ZSP8 10862104 Ki < 2.8 nM T68251 CQ1L7C 10863755 Ki = 690 nM T68251 C0AQL8 10873958 Ki < 2.8 nM T68251 CBQ70P 10874312 IC50 = 6.3 nM T68251 CLG40T 10874819 IC50 = 260 nM T68251 CXY47P 10875332 IC50 = 383 nM T68251 CJ0LE4 10876254 Ki = 50 nM T68251 CIB8Y1 10884337 Ki = 8 nM T68251 C3AY8O 10885569 IC50 = 20 nM T68251 CAU0I3 10885834 IC50 = 0.9 nM T68251 CDZ04P 10887027 Ki = 11 nM T68251 C7AMS4 10895808 Ki = 49 nM T68251 CPJ0I8 10896934 IC50 = 76 nM T68251 CU7YE0 10896986 IC50 = 0.7 nM T68251 C3FQT7 10903871 Ki = 82 nM T68251 CAF1N8 10906013 IC50 = 2500 nM T68251 CX93MR 10907320 IC50 = 9 nM T68251 CM9G8A 10907701 IC50 = 0.42 nM T68251 C13CJH 10907740 IC50 = 62 nM T68251 C69ZTR 10913644 Ki = 312 nM T68251 C2QR0W 10914151 Ki = 701 nM T68251 C7XE3L 10917417 Ki < 2.8 nM T68251 CGI2T1 10928606 IC50 = 176 nM T68251 CXHA75 10928874 IC50 = 1 nM T68251 CXY4L6 10929354 IC50 = 829 nM T68251 CDSQ41 10929404 IC50 = 106 nM T68251 C1QVT6 10939850 IC50 = 0.93 nM T68251 CWO29J 10940364 IC50 = 13 nM T68251 C89IYC 10948209 Ki < 2.8 nM T68251 CC46WL 10950008 Ki > 3000 nM T68251 C9YOU4 10951375 IC50 = 16 nM T68251 CJI1G0 10951750 IC50 = 1 nM T68251 CNBR78 10952384 IC50 = 8.82 nM T68251 C0A2IR 10958121 Ki = 14 nM T68251 C5HS4F 10961382 Ki = 491 nM T68251 CMY8S6 10961569 IC50 = 1.3 nM T68251 CPA1Q2 10961828 IC50 = 2.8 nM T68251 C30FBA 10970628 Ki = 19 nM T68251 CU2Q8S 10971085 IC50 = 320 nM T68251 CQ68IE 10972732 IC50 = 0.34 nM T68251 CJHO94 10972891 IC50 = 1.7 nM T68251 CTP6I0 10973485 IC50 = 3.6 nM T68251 C9DM0P 10980832 Ki = 11 nM T68251 CL7K8S 10983560 Ki < 3 nM T68251 C3UH2B 10983665 Ki = 647 nM T68251 CR9J5B 10983887 IC50 = 1.7 nM T68251 C68LPK 10983913 IC50 = 1.4 nM T68251 CS7D0Z 10984030 IC50 = 0.72 nM T68251 CV4J2F 10984597 IC50 = 0.3 nM T68251 C0G8TE 10993343 Ki = 11 nM T68251 CW8Z6R 10993677 Ki = 2518 nM T68251 CCX0L6 10994350 IC50 = 3.2 nM T68251 CW0Y6I 10994897 IC50 = 2.4 nM T68251 C3QX0T 11005761 IC50 = 0.45 nM T68251 CJM41O 11006091 IC50 = 1.3 nM T68251 C4PNK3 11006191 IC50 = 1810 nM T68251 C95NXQ 11006894 Ki = 0.64 nM T68251 C7WEZ4 11009332 Ki = 21000 nM T68251 C9WPH7 11016072 Ki = 880 nM T68251 CBE68H 11016073 Ki = 850 nM T68251 CG2DK0 11016448 IC50 < 0.4 nM T68251 C3IYK8 11016511 IC50 = 0.32 nM T68251 CF30UR 11016519 IC50 = 3.78 nM T68251 CODQ51 11016616 IC50 < 0.4 nM T68251 C6IHF5 11026991 IC50 > 8 nM T68251 C3LF1Y 11027584 Ki = 3001 nM T68251 CF5KU1 11027718 IC50 = 1.5 nM T68251 CA49QF 11027968 IC50 = 0.91 nM T68251 CLXZ15 11037377 Ki = 4.3 nM T68251 CT2S0G 11038175 IC50 = 7.4 nM T68251 C3W9IT 11046880 Ki = 408 nM T68251 C5R7JX 11049650 Ki = 1595 nM T68251 CW42KO 11049937 IC50 = 1.9 nM T68251 CQ08SN 11049982 IC50 = 1.8 nM T68251 C23KPN 11050468 IC50 = 2.3 nM T68251 C9RU4I 11059620 IC50 = 2.8 nM T68251 CH8O1E 11060081 Ki = 154 nM T68251 CM6X1E 11061555 Ki > 2000 nM T68251 C1N5PT 11070986 IC50 = 3.2 nM T68251 C18EIZ 11071831 IC50 = 0.6 nM T68251 C43JOG 11080156 Ki = 38 nM T68251 CT3VX4 11080936 Ki = 361 nM T68251 CG0A4C 11081333 IC50 = 25 nM T68251 C05MUK 11081992 IC50 = 1.6 nM T68251 CUNM68 11083152 Ki = 231 nM T68251 CS29GX 11091928 IC50 = 2.8 nM T68251 CE8V9B 11092295 IC50 = 4.22 nM T68251 CR8ZA7 11092551 IC50 = 14 nM T68251 CT2CH7 11092701 IC50 = 9.5 nM T68251 C6R7XB 11092861 Ki = 960 nM T68251 CX69YN 11093502 IC50 = 1.2 nM T68251 CR4V2D 11101785 Ki = 410 nM T68251 C8CK3E 11102531 IC50 = 24 nM T68251 C6G2DI 11111616 Ki = 23 nM T68251 CUK03P 11112062 Ki = 5812 nM T68251 CWV45Z 11112302 Ki < 2.8 nM T68251 CY1SR9 11113744 IC50 = 58.1 nM T68251 CNGP50 11122963 IC50 = 0.35 nM T68251 C8YVE5 11123989 IC50 = 5 nM T68251 CNBG53 11124956 IC50 = 1.6 nM T68251 CX2B6C 11125147 Ki = 450 nM T68251 C9GJ7C 11133809 Ki = 94 nM T68251 C2YBQ7 11134935 IC50 = 7.2 nM T68251 C8DMW5 11135133 IC50 = 83 nM T68251 CD3N8B 11135304 IC50 = 16 nM T68251 CF52TX 11143173 Ki = 1507 nM T68251 CH61QF 11144824 IC50 = 2.4 nM T68251 C8HM2R 11145437 Ki = 75 nM T68251 CHF19X 11146467 Ki = 32 nM T68251 C5WS3E 11147931 IC50 = 1000 nM T68251 CM0QK6 11156328 IC50 = 10 nM T68251 C9H1CW 11156691 IC50 = 16 nM T68251 CD1Q0L 11157488 IC50 = 1590 nM T68251 CZ8KI2 11157757 IC50 = 1500 nM T68251 CM04FR 11168103 IC50 = 10 nM T68251 CVR01T 11168326 IC50 = 7.21 nM T68251 CMKT17 11168614 IC50 = 886 nM T68251 C63CLD 11169065 IC50 = 1200 nM T68251 CD3WL8 11179683 IC50 = 8.4 nM T68251 C2LZ7F 11191803 IC50 = 85 nM T68251 CPA84O 11192618 IC50 = 1630 nM T68251 CCQ6N8 11194666 IC50 = 150 nM T68251 C43ONW 11202395 Ki > 3333 nM T68251 CO76XI 11205873 IC50 = 5000 nM T68251 C9R7OM 11207122 IC50 = 50000 nM T68251 CO87YZ 11215538 IC50 = 5000 nM T68251 CIZW31 11226189 IC50 = 323 nM T68251 C3LEA2 11226622 IC50 = 7 nM T68251 CEL1F0 11248884 IC50 = 19 nM T68251 CUOH67 11252195 IC50 = 500 nM T68251 CJZ3P6 11257884 Ki = 0.4 nM T68251 CO7T3M 11261246 IC50 = 0.41 nM T68251 CWG8Y6 11271094 IC50 = 236 nM T68251 C2OJ8Q 11272747 IC50 = 15000 nM T68251 CJX60I 11284255 IC50 = 5110 nM T68251 C6LJM4 11284404 IC50 = 522 nM T68251 CP17ID 11284983 IC50 = 1700 nM T68251 CF9O2R 11286824 IC50 = 3000 nM T68251 C1IW7N 11292680 IC50 = 0.09 nM T68251 C8C5AV 11294179 Ki > 3333 nM T68251 C7H9JG 11295013 IC50 = 26 nM T68251 C0ZI3J 11298263 IC50 > 200000 nM T68251 C78QSH 11307739 IC50 = 16 nM T68251 CRP08M 11310883 IC50 = 1000 nM T68251 CJ09XO 11317090 IC50 = 5 nM T68251 CK91YW 11317404 IC50 = 68 nM T68251 CLH50U 11318841 IC50 = 1760 nM T68251 C1SN8I 11319030 IC50 = 63 nM T68251 CN2P4G 11328571 IC50 = 321 nM T68251 C9FW7I 11330706 IC50 = 3650 nM T68251 C0XR3B 11330861 IC50 = 3010 nM T68251 CQH57S 11342435 IC50 = 135 nM T68251 CZ8B0D 11349945 Ki < 3.3 nM T68251 CYAK73 11353754 IC50 = 81 nM T68251 CA5P8H 11355488 IC50 = 76000 nM T68251 C7QNX8 11363138 IC50 = 1662 nM T68251 CHG6W0 11365417 IC50 = 62 nM T68251 CM8Y1J 11367571 IC50 = 3000 nM T68251 CTQK48 11373358 Ki > 3333 nM T68251 CLE30X 11374591 IC50 = 2.14 nM T68251 C5KU3Z 11376005 IC50 = 595 nM T68251 CEM0A7 11387990 IC50 = 6200 nM T68251 COZN84 11388372 IC50 = 15 nM T68251 CUJ4V0 11391937 IC50 = 8.2 nM T68251 C9ABX8 11397130 Ki > 3333 nM T68251 CF78WB 11398934 IC50 = 1410 nM T68251 C13NCF 11400989 IC50 = 300 nM T68251 CZM5E8 11410471 IC50 = 30 nM T68251 CU04HF 11419551 IC50 = 47 nM T68251 C4K9DO 11421151 IC50 = 3.2 nM T68251 C30PFC 11421763 IC50 = 2060 nM T68251 CK95HW 11429232 Ki = 0.4 nM T68251 C01FLQ 11441438 Ki = 3.2 nM T68251 CFE6A0 11443957 IC50 = 37 nM T68251 CZY3W9 11444262 IC50 = 12 nM T68251 CI0V6L 11447356 IC50 = 4000 nM T68251 COS67B 11456566 IC50 = 1370 nM T68251 CCMT46 11457732 IC50 = 20 nM T68251 C96DRO 11466734 IC50 = 581 nM T68251 C7QF0G 11467517 IC50 = 2150 nM T68251 CQ1D6E 11470070 IC50 = 200 nM T68251 C1KP2Q 11473879 Ki > 3333 nM T68251 CZBF91 11476645 IC50 = 156 nM T68251 C5Z4UP 11504653 IC50 > 2000 nM T68251 CWS35C 11510523 IC50 = 1270 nM T68251 C5G8PM 11511807 IC50 > 2000 nM T68251 C5VUM2 11517085 Ki = 300 nM T68251 C43OXZ 11519233 IC50 = 9 nM T68251 C5MO0U 11526826 IC50 = 5.3 nM T68251 CI8R5J 11529867 IC50 = 23100 nM T68251 C9Y6LH 11533683 IC50 = 3270 nM T68251 CE01PG 11543178 IC50 = 15370 nM T68251 C2OA3K 11547967 IC50 = 546 nM T68251 C1NZB9 11548265 IC50 = 0.3 nM T68251 CIWP38 11555036 IC50 = 18 nM T68251 C47VIT 11562805 IC50 = 4000 nM T68251 C61BQP 11562817 IC50 = 1563 nM T68251 CO9BC3 11562986 IC50 = 1272 nM T68251 CW5A4S 11569716 IC50 = 6.3 nM T68251 CHV2G1 11575995 Ki > 10000000 nM T68251 C3H2DG 11577137 IC50 = 135 nM T68251 CM6GO2 11577517 IC50 > 2000 nM T68251 CXT05D 11581283 IC50 = 1120 nM T68251 CX2PQ5 11588332 IC50 = 5740 nM T68251 C0Q5FU 11592023 IC50 > 2000 nM T68251 CSQ5M8 11598899 IC50 = 264 nM T68251 CTQ87G 11599024 IC50 = 1440 nM T68251 COT65V 11599397 IC50 > 2000 nM T68251 CUL5H2 11605631 IC50 = 4 nM T68251 CQ7G5D 11613116 IC50 = 1999 nM T68251 C0VCJ8 11613810 IC50 = 3.6 nM T68251 CXKU59 11620780 IC50 > 5000 nM T68251 CCBS59 11634234 IC50 = 280 nM T68251 CZO71U 11639846 IC50 = 550 nM T68251 CNY92D 11640694 Ki > 30000 nM T68251 CFV49P 11641262 IC50 < 1.5 nM T68251 CH3V8F 11663480 IC50 > 2000 nM T68251 CR2UN0 11669859 IC50 = 7.4 nM T68251 CK9F4P 11673778 IC50 = 9000 nM T68251 C90GCV 11675055 IC50 = 2110 nM T68251 C0WV8R 11678029 IC50 > 2000 nM T68251 CFC74O 11678245 IC50 = 574 nM T68251 C28WNK 11682752 Ki = 16 nM T68251 CY0T4D 11685065 IC50 > 2000 nM T68251 CRF7V9 11691964 IC50 = 1.3 nM T68251 CKGR97 11692294 IC50 = 1999 nM T68251 C6ORK5 11692747 IC50 = 655 nM T68251 C3U6ZR 11697504 Ki = 33000 nM T68251 C4BGI2 11698938 IC50 = 6958 nM T68251 C6PM1J 11713686 IC50 = 1380 nM T68251 C1MJ3P 11713694 IC50 = 126 nM T68251 C2BJ3X 11716217 Ki = 4599 nM T68251 C4FU2H 11717997 IC50 = 3430 nM T68251 C4ECU2 11720597 IC50 = 315 nM T68251 CCD93H 11730086 Ki = 80 nM T68251 C68KBY 11732585 Ki = 85 nM T68251 C7CED0 11733417 IC50 = 549 nM T68251 CI0KL2 11733573 IC50 = 13 nM T68251 C64LQC 11733862 Ki > 3000 nM T68251 CIU03K 11734219 Ki = 332 nM T68251 CJOE40 11748355 Ki = 4.8 nM T68251 C4HD9K 11751106 IC50 = 271 nM T68251 CG8U3H 11753351 IC50 = 3810 nM T68251 CO8QT0 11753905 Ki = 1100 nM T68251 C3P0TZ 11754739 Ki = 238 nM T68251 CJ4G5D 11754907 IC50 = 16.2 nM T68251 CD6S0B 11757331 IC50 > 100000 nM T68251 C5E7KU 11757592 Ki = 0.6 nM T68251 CUC9R5 11758082 IC50 = 0.7 nM T68251 CF2J8V 11758099 IC50 = 1000 nM T68251 CQ3Y4E 11761293 IC50 = 110 nM T68251 C6K8HR 11761578 Ki = 136 nM T68251 C04DFH 11783486 Ki = 4.8 nM T68251 CQP12F 11787159 IC50 = 86 nM T68251 C7BV5P 11792968 Ki = 40.74 nM T68251 CV16JZ 11793588 IC50 > 1000 nM T68251 CCSD72 11795621 IC50 = 7.8 nM T68251 CY8N1U 11795715 Ki = 5 nM T68251 CY7H2T 11795824 Ki = 12 nM T68251 C3DE6J 11796352 IC50 = 5.4 nM T68251 CK24XT 11796481 Ki = 8 nM T68251 C46KHU 11796490 IC50 = 5.2 nM T68251 C47OIA 11797154 IC50 = 0.8 nM T68251 CJ4VL3 11797382 IC50 = 10 nM T68251 C7VLP9 11798303 IC50 < 200 nM T68251 CHQR96 11798386 IC50 < 0.4 nM T68251 CZ3C9P 11798873 IC50 = 1.5 nM T68251 CXFP23 11798966 IC50 = 3.311 nM T68251 C19RCP 11799753 Ki = 3.7 nM T68251 CHS4I2 11800528 Ki = 38 nM T68251 CZ5LP1 11800650 IC50 = 10 nM T68251 CQ9HE2 11811551 IC50 = 53 nM T68251 CK03NI 11811717 Ki = 35 nM T68251 CLW3F1 11812791 IC50 = 24.2 nM T68251 C20PYA 11813392 IC50 = 12 nM T68251 CH3SV6 11813493 IC50 = 76 nM T68251 C8DY3Z 11817193 IC50 = 1000 nM T68251 CEN02U 11822212 Ki = 75 nM T68251 CDU9S2 11824087 Ki = 52 nM T68251 C3VO5H 11824148 Ki = 0.3 nM T68251 CKEM29 11827006 IC50 = 46 nM T68251 CV2MX4 11832221 Ki = 108 nM T68251 C48QEH 11833533 Ki < 2.8 nM T68251 CI2OP1 11942810 IC50 = 2700 nM T68251 C4XR5G 11963536 IC50 = 664 nM T68251 C02BWA 11967143 Ki > 2000 nM T68251 CB80OT 12000718 IC50 > 20000 nM T68251 C43PJZ 12000720 IC50 > 20000 nM T68251 CN72PQ 12037467 IC50 = 82.17 nM T68251 CKI97Z 12344252 IC50 > 200000 nM T68251 C0K8ZX 12404978 IC50 > 500000 nM T68251 C0JID3 12447203 Ki > 100000 nM T68251 CKSL53 12507616 IC50 > 200000 nM T68251 CTHQ39 12635073 Ki = 14000 nM T68251 CIQX87 12635074 Ki = 72000 nM T68251 C0XKJ1 12671872 IC50 = 1000 nM T68251 COF8W3 13008156 IC50 > 200000 nM T68251 CC9DK6 13384604 IC50 = 300 nM T68251 CSR94V 13559594 IC50 = 3.28 nM T68251 C71ASU 13644537 IC50 = 8.22 nM T68251 CQTX49 13738810 IC50 > 100000 nM T68251 CVH7N1 13746652 IC50 = 9800 nM T68251 C1AJO7 13968141 IC50 > 300000 nM T68251 CP8L5J 14104451 IC50 = 2000 nM T68251 CLS53V 14151811 IC50 = 9500 nM T68251 CQ3D9C 14151815 IC50 = 18000 nM T68251 C8TH1O 14177156 IC50 > 500000 nM T68251 CM9PD5 14237653 IC50 = 12400 nM T68251 CA2H8V 14303060 IC50 = 170 nM T68251 C7KDL3 14616290 IC50 = 98020 nM T68251 CY4XO2 14616291 IC50 > 500000 nM T68251 C1Q5JU 14616298 IC50 = 67010 nM T68251 C9TF7I 14616299 IC50 = 246260 nM T68251 CHU6J5 14616300 IC50 = 81010 nM T68251 C86DNV 14616301 IC50 = 64300 nM T68251 C47DQP 14732854 IC50 = 19000 nM T68251 C1IZ7D 15296597 Ki = 15 nM T68251 CGH19T 15296844 IC50 > 300000 nM T68251 CSU04W 15406874 IC50 = 5.8 nM T68251 C63MFQ 15435266 IC50 = 3 nM T68251 CH80JI 15435267 Ki = 25 nM T68251 CZ0NL1 15484680 IC50 = 6 nM T68251 CT68FI 15487434 Ki = 120 nM T68251 CJR3Z8 15487435 Ki = 110 nM T68251 C46XNB 15487436 Ki = 560 nM T68251 CP2C4Z 15524387 Ki = 31600 nM T68251 CAF7R5 15524388 Ki = 52 nM T68251 C17HGN 15524389 Ki = 6600 nM T68251 CFH8Y6 15524390 Ki = 35000 nM T68251 C3N1KV 15629940 IC50 > 100000 nM T68251 CVUY27 15631189 IC50 = 8490 nM T68251 C5TLB4 15765753 IC50 = 3.97 nM T68251 C5FA3L 15871222 IC50 = 0.7 nM T68251 CB3A4Z 15941413 Ki = 78 nM T68251 CA40FE 15941550 Ki = 6 nM T68251 CM3D1L 15941553 Ki = 110 nM T68251 CQ0ZL7 15941677 Ki = 23 nM T68251 C6F9WV 15941679 Ki = 70 nM T68251 C7C1HI 15941680 Ki = 34 nM T68251 CU2C1R 15987326 IC50 = 1040 nM T68251 CL7KX3 16040152 IC50 = 3 ug.mL-1 T68251 CTZ3R1 16040153 IC50 = 12.4 ug.mL-1 T68251 C4VW5F 16058482 IC50 = 35 nM T68251 C4WX2I 16108938 IC50 > 1000 nM T68251 CD51GI 16108939 IC50 = 5 nM T68251 C5YVB0 16108940 IC50 = 446 nM T68251 CB4DU9 16108941 IC50 > 5000 nM T68251 CBW71J 16108942 IC50 > 5000 nM T68251 CG6R9L 16108943 IC50 = 960 nM T68251 CN62KM 16108944 IC50 = 150 nM T68251 C7YS5Q 16108947 IC50 = 200 nM T68251 CLD2Y4 16108948 IC50 > 5000 nM T68251 CJR95O 16108949 IC50 > 1000 nM T68251 CRQ26L 16108950 IC50 = 350 nM T68251 CH80AG 16108951 IC50 = 13 nM T68251 CWB0G9 16108952 IC50 = 64 nM T68251 CS46XU 16126723 IC50 = 1.2 nM T68251 CC6OH2 16129741 IC50 = 43200 nM T68251 CH7D2Q 16420684 IC50 = 21200 nM T68251 C91EXN 16655061 IC50 = 555 nM T68251 CQS0F5 16719301 IC50 = 180 nM T68251 C0OUC6 16726064 IC50 = 23000 nM T68251 C75XDI 16730519 IC50 > 2000 nM T68251 C2W1VA 16739287 Ki = 5000 nM T68251 C6F9LM 16748789 IC50 > 30000 nM T68251 CXB10H 16748901 IC50 > 100000 nM T68251 C7YJZ5 17748252 IC50 = 2200 nM T68251 C3S2TQ 17754305 IC50 = 431 nM T68251 CQG89Z 17853548 IC50 = 64190 nM T68251 C2ZAX1 18002715 Ki > 3300 nM T68251 C12UGK 18002722 Ki > 3300 nM T68251 C0IYW8 18002726 Ki > 3300 nM T68251 C8N1DM 18002729 Ki > 3300 nM T68251 CCG96A 18002736 Ki > 3300 nM T68251 C5MLG1 18002745 Ki > 3300 nM T68251 CXT4H2 18002752 Ki > 3300 nM T68251 C26WHK 18002758 Ki > 3300 nM T68251 CV90XS 18002764 Ki > 3300 nM T68251 C8KPM7 18002765 Ki > 3300 nM T68251 CMJ0K3 18002771 Ki > 3300 nM T68251 C2CO9Z 18002775 Ki > 3300 nM T68251 CK8FS7 18173159 IC50 = 6 nM T68251 CX10BM 18173179 IC50 = 24 nM T68251 CQO70Y 18173222 IC50 = 82 nM T68251 C6F8WH 18319167 IC50 = 6 nM T68251 C57FQG 18319202 IC50 = 1790 nM T68251 CJ8G9A 18319234 IC50 = 334.97 nM T68251 CE4J1B 18319263 IC50 = 1300 nM T68251 CXG1K2 18363133 IC50 > 10000 nM T68251 C37BNA 18363136 IC50 > 10000 nM T68251 C0KOW7 18363142 IC50 > 10000 nM T68251 CP04KS 18363146 IC50 > 10000 nM T68251 CLZD96 18363152 IC50 > 10000 nM T68251 CW3KB9 18363153 IC50 > 10000 nM T68251 CK30ZO 18363159 IC50 > 10000 nM T68251 CZU27R 18363164 IC50 > 10000 nM T68251 CC0UV8 18363169 IC50 > 10000 nM T68251 CR3CQ4 18363187 IC50 > 10000 nM T68251 CH5IU9 18363209 IC50 > 10000 nM T68251 CJGZ27 18363210 IC50 > 10000 nM T68251 CWI2A9 18363212 IC50 > 10000 nM T68251 C31LQZ 18363213 IC50 > 10000 nM T68251 CE60WD 18363216 IC50 > 10000 nM T68251 C3L6DU 18363223 IC50 > 10000 nM T68251 CI53DY 18379040 Ki > 3333 nM T68251 CB1U5T 18379077 Ki > 3333 nM T68251 CSX97G 18379115 Ki > 3333 nM T68251 CJHL25 18379123 Ki > 3333 nM T68251 CR0B8G 18379149 Ki > 3333 nM T68251 CS4V5K 18379187 Ki > 3333 nM T68251 CCTY94 18379210 Ki > 3333 nM T68251 CA6K5S 18379235 Ki > 3333 nM T68251 CCSK49 18379254 Ki > 3333 nM T68251 CP4T7S 18379435 Ki > 3333 nM T68251 C9Y5GX 18379443 Ki > 3333 nM T68251 CXL6T9 18379569 IC50 = 173 nM T68251 CKY98M 18379668 IC50 = 9 nM T68251 CSY0N8 18394511 IC50 > 300000 nM T68251 C9J8IN 18445902 IC50 = 800 nM T68251 C5B9WG 18533077 IC50 = 800 nM T68251 C50AEZ 18616892 IC50 = 23.5 nM T68251 CYA3H7 18790040 IC50 > 10000 nM T68251 CBN28Y 18790155 Ki = 270 nM T68251 C03CET 18914685 Ki = 2000 nM T68251 CIEH93 19382975 IC50 = 6400 nM T68251 C60WKH 20196702 IC50 = 5.09 nM T68251 CK8MP3 20620240 Ki = 230 nM T68251 CPC4G6 20620273 Ki = 410 nM T68251 C26UJT 20620561 IC50 = 16 nM T68251 C2E3CY 20620614 IC50 = 48 nM T68251 CVEX54 20620688 IC50 = 6.6 nM T68251 CV1SD8 20620714 IC50 = 11 nM T68251 C3GAC4 20620715 IC50 = 270 nM T68251 C7QV8K 20620757 IC50 = 1100 nM T68251 CVO73Y 20620827 IC50 = 450 nM T68251 CQ14NY 20620831 IC50 = 940 nM T68251 C5RQ8A 20620860 IC50 = 10 nM T68251 CPK09X 20651316 IC50 = 1.4 nM T68251 CG1BD4 20689551 IC50 = 180 nM T68251 C48TWB 20728102 IC50 > 2000 nM T68251 C18RXS 20735191 IC50 < 0.1 nM T68251 C4I1OM 20735209 IC50 = 400 nM T68251 CF1CK9 20735364 IC50 = 0.5 nM T68251 CW3D7O 20760308 Ki = 1002 nM T68251 C09JTR 21130554 IC50 = 0.2 nM T68251 C6VP1T 21130556 IC50 = 0.2 nM T68251 C15UGO 21130558 IC50 = 5 nM T68251 C9H3IG 21130559 IC50 = 1.3 nM T68251 C8Q2OD 21130561 IC50 = 1.3 nM T68251 C25FAD 21130562 IC50 = 0.2 nM T68251 CW2Q5A 21130590 IC50 = 79.98 nM T68251 C9HMC0 21130591 IC50 = 184 nM T68251 CT87YK 21699971 IC50 = 5200 nM T68251 CH4G5T 21699977 IC50 = 400 nM T68251 CQ1GI3 21699983 IC50 = 650000 nM T68251 CJZ58F 21699985 IC50 = 37000 nM T68251 CA3WG1 21699989 IC50 = 4 nM T68251 CE72FU 21700004 IC50 = 950000 nM T68251 CRG8J9 21700008 IC50 = 20 nM T68251 C5JC6W 21700038 IC50 = 160000 nM T68251 CY18IE 21700054 IC50 = 89 nM T68251 CW1YS9 21700072 IC50 = 20 nM T68251 C3QAP8 21700080 IC50 = 45000 nM T68251 CG0RI5 21700124 IC50 = 5900 nM T68251 CR81NU 21700137 IC50 = 1300 nM T68251 CJ4C3K 21700144 IC50 = 85 nM T68251 C94FZS 21700146 IC50 = 26 nM T68251 CXME27 21700151 IC50 = 3400 nM T68251 CFK4Y7 21700160 IC50 = 6900 nM T68251 CIJ93L 21700163 IC50 = 25000 nM T68251 CN80JR 21700178 IC50 = 4 nM T68251 CB1QH3 21700191 IC50 = 480000 nM T68251 CUVE24 21700204 IC50 = 260000 nM T68251 CM42ZR 21700258 IC50 = 4 nM T68251 CMW12T 21700264 IC50 = 1 nM T68251 CKAJ52 21867770 IC50 = 0.7 nM T68251 C45UGA 21996090 IC50 = 16 nM T68251 CIC4S9 22004232 IC50 = 3.4 nM T68251 C36WFA 22096205 IC50 > 100000 nM T68251 CO91AD 22341241 Ki > 3333 nM T68251 CE5DH1 22484408 IC50 = 1.8 nM T68251 CZT05X 22484417 Ki = 550 nM T68251 CZT64B 22484431 Ki = 410 nM T68251 C1O7RC 22485248 IC50 = 400 nM T68251 CAM10T 22485252 IC50 = 0.8 nM T68251 CBJS34 22485260 IC50 < 0.1 nM T68251 C9MU7N 22485263 IC50 = 4.4 nM T68251 CEGJ03 22485276 IC50 = 3.3 nM T68251 C7VB8G 22485289 IC50 = 0.5 nM T68251 CNB02I 22485291 IC50 < 0.1 nM T68251 CAY3N6 22485292 IC50 = 1 nM T68251 C94OCJ 22485302 IC50 = 0.1 nM T68251 C3YL5X 22485311 IC50 = 0.1 nM T68251 C80RSQ 22485314 IC50 = 0.1 nM T68251 CWA03L 22485327 IC50 = 0.2 nM T68251 C6JRW5 22485340 IC50 = 0.1 nM T68251 C5JZF1 22485344 IC50 = 0.35 nM T68251 CI7MY5 22485346 IC50 = 0.1 nM T68251 CI1YL7 22485347 IC50 = 0.25 nM T68251 C25OBD 22485356 IC50 = 0.3 nM T68251 C7I0EW 22485367 IC50 = 0.2 nM T68251 CL64TJ 22485368 IC50 = 0.2 nM T68251 CT4GF9 22485381 IC50 = 6350 nM T68251 C27NDB 22485386 IC50 = 1.7 nM T68251 CTJ9I3 22485392 IC50 = 0.3 nM T68251 C3MG9P 22485396 IC50 = 0.4 nM T68251 CZY10U 22485408 IC50 = 0.3 nM T68251 C89AGT 22485413 IC50 = 0.2 nM T68251 C03NLM 22485417 IC50 = 0.1 nM T68251 C8GHU9 22485432 IC50 = 0.2 nM T68251 C9BT5F 22626996 IC50 = 77 nM T68251 C2Q4XK 22707806 IC50 = 0.1 nM T68251 CD4Z6P 22707833 IC50 = 3500 nM T68251 CMYK90 22707860 IC50 < 0.1 nM T68251 CVF9M4 22922043 IC50 = 23320 nM T68251 CX2JO7 22950015 IC50 = 335 nM T68251 COCN69 22956916 Ki = 1111 nM T68251 C85PXN 22956934 Ki = 771 nM T68251 CIYA45 22985930 IC50 < 0.1 nM T68251 CF75MS 23017979 IC50 = 60000 nM T68251 CQJ3S4 23018008 IC50 = 30000 nM T68251 CM5H2P 23061661 IC50 > 10000 nM T68251 C97LAR 23061665 IC50 > 10000 nM T68251 C2DG6O 23288322 Ki = 2000 nM T68251 C5XW9M 23310222 IC50 = 9 ug.mL-1 T68251 C9IW3E 23433373 IC50 = 1000 nM T68251 CX32YK 23513795 IC50 = 19 nM T68251 C6IZ1S 23513821 IC50 = 113 nM T68251 CPNM93 23513825 IC50 = 62 nM T68251 CML90Q 23513831 IC50 = 54 nM T68251 C87RTM 23513845 IC50 = 249 nM T68251 C4R2AJ 23625454 IC50 = 513 nM T68251 CD3U8A 23627203 Ki = 1300 nM T68251 C8UIC6 23644662 Ki > 100000 nM T68251 CCLA40 23644663 Ki > 100000 nM T68251 CSZ6J4 23645528 Ki = 3.2 nM T68251 C6UH9Q 23645529 Ki = 0.8913 nM T68251 CD0JP3 23645530 Ki = 0.7943 nM T68251 CM37EC 23645531 Ki = 2.399 nM T68251 C9PD5F 23645532 Ki = 2.884 nM T68251 C1OE7R 23645533 Ki = 0.7943 nM T68251 CCSN04 23645534 Ki = 1.4 nM T68251 CU08WI 23645535 Ki = 0.6918 nM T68251 CY41UC 23645536 Ki = 15 nM T68251 CX15EH 23645537 Ki = 3.7 nM T68251 CD3Q6G 23645538 Ki = 12 nM T68251 CE6NQ2 23645539 Ki = 19000 nM T68251 C4VK3U 23645540 Ki = 14000 nM T68251 C8VM1C 23645541 Ki = 73000 nM T68251 C0MUT6 23645542 Ki = 21000 nM T68251 CNI07H 23645543 Ki = 23000 nM T68251 CHK2X1 23645544 Ki = 38000 nM T68251 CW1V2Z 23645545 Ki = 14000 nM T68251 C6SP7T 23645546 Ki = 11000 nM T68251 CD9QO2 23645547 Ki = 900 nM T68251 C25YLZ 23645548 Ki = 90 nM T68251 CL1KC0 23652834 IC50 = 8.37 nM T68251 CL24JR 23655078 IC50 = 940 nM T68251 COIZ43 23655713 IC50 = 4350 nM T68251 CURM98 23655714 IC50 > 100000 nM T68251 CO90JC 23655717 IC50 = 5590 nM T68251 C3M2NQ 23655718 IC50 = 207 nM T68251 C56NMQ 23655910 IC50 = 9110 nM T68251 C9QZX5 23655911 IC50 = 6120 nM T68251 CA8W3K 23656106 IC50 = 239 nM T68251 CU4R7T 23656291 IC50 = 4 nM T68251 CVZ2M1 23656293 IC50 = 22 nM T68251 CL5C1I 23656295 IC50 = 30 nM T68251 CZP12E 23656450 IC50 = 2 nM T68251 CA2PY5 23657418 IC50 = 335 nM T68251 CN9TY1 23657419 IC50 = 992 nM T68251 C9FHZ1 23657421 IC50 = 19 nM T68251 CY9LF1 23657422 IC50 = 8 nM T68251 C28SPW 23657691 IC50 = 41000 nM T68251 CVJ1T7 23657695 IC50 = 20000 nM T68251 CAL05Q 23657697 IC50 = 35000 nM T68251 C6AW7U 23692637 IC50 = 2000 nM T68251 C7KF1N 23729138 IC50 = 6.8 nM T68251 C35QME 24742028 IC50 = 3 nM T68251 CY6KA0 24755074 IC50 = 5000 nM T68251 CG3J2L 24768528 IC50 = 120 nM T68251 CQCJ17 24768595 IC50 = 0.53 nM T68251 C5M3YW 24799779 Ki = 1000000 nM T68251 CWLT01 24806172 IC50 = 61 nM T68251 CN59KZ 24806173 IC50 = 1233 nM T68251 CH4X8K 24806175 IC50 = 13 nM T68251 C9RW0A 24806176 IC50 = 5.2 nM T68251 C18FRG 24807817 IC50 > 100000 nM T68251 CW3X0F 24852010 IC50 = 5.6 nM T68251 C2U0NS 24852011 IC50 = 8.3 nM T68251 C6YPS8 24852048 IC50 = 5 nM T68251 CUK6F1 24852487 IC50 = 95.9 nM T68251 C0MPV5 24852489 IC50 = 59.4 nM T68251 CK0CI6 24860421 IC50 = 334 nM T68251 CZI59C 24860423 IC50 = 97 nM T68251 CE29HI 24860424 IC50 = 1530 nM T68251 CT10JE 24860425 IC50 = 216 nM T68251 CRC98J 24860426 IC50 = 46 nM T68251 C8MKR0 24860427 IC50 = 1312 nM T68251 C3S6DX 24860428 IC50 = 56 nM T68251 C2LNE4 24860429 IC50 = 4181 nM T68251 CF4D0X 24860430 IC50 > 1666 nM T68251 CNR3U7 24866945 IC50 > 100000 nM T68251 CRZ7Y6 24868315 IC50 = 1.8 nM T68251 CFL04M 24881245 IC50 > 300000 nM T68251 CLIC14 24881246 IC50 = 60000 nM T68251 C3U8ZQ 24882385 IC50 = 230 nM T68251 C02WIB 24882535 IC50 = 20 nM T68251 C4FI5C 24901479 IC50 = 40 nM T68251 C6F0ZP 24901485 IC50 = 4.6 nM T68251 C4SP3O 24936157 IC50 = 0.67 nM T68251 CBUA83 24936183 IC50 = 12.6 nM T68251 CQ2K9H 24936215 IC50 = 488 nM T68251 C0EA5F 24936382 IC50 = 0.04 nM T68251 C78OAU 24944977 IC50 = 114 nM T68251 CO6CJ5 24945161 IC50 = 3600 nM T68251 C1C0NX 24945244 IC50 = 5300 nM T68251 CLTQ28 24945246 IC50 = 250 nM T68251 C7ZA6S 24945247 IC50 = 380 nM T68251 CH3O0V 24951588 IC50 = 83 nM T68251 C8I4PT 24951589 IC50 = 17 nM T68251 C2Q1BK 24951590 IC50 = 11 nM T68251 COMJ45 24951950 IC50 = 333 nM T68251 C3JGU2 24951952 IC50 = 24 nM T68251 CC7U2T 24951953 IC50 = 12 nM T68251 CV86KA 24952316 IC50 = 27 nM T68251 CYJ2E9 24952318 IC50 = 2535 nM T68251 CYKM71 24952674 IC50 = 139 nM T68251 C7MC8J 24952678 IC50 = 9.2 nM T68251 C0ZB8O 24953024 IC50 = 5.7 nM T68251 C5Z8XR 24953380 IC50 = 47 nM T68251 C2LN5E 24953381 IC50 = 119 nM T68251 CT2N3H 24953730 IC50 = 9.9 nM T68251 C1KH2Q 24953731 IC50 = 8.6 nM T68251 C0Q5BT 24954067 IC50 = 5.5 nM T68251 C6FI8O 24954068 IC50 = 5.6 nM T68251 CN29BR 24954070 IC50 = 5.5 nM T68251 CL1YO0 24954431 IC50 = 2.5 nM T68251 C3H9EO 24954432 IC50 = 7.6 nM T68251 CB60LR 24954795 IC50 = 24 nM T68251 C7P5YH 24954798 IC50 = 2.8 nM T68251 C5BG6I 24955154 IC50 = 32 nM T68251 CCE45B 24955155 IC50 = 56 nM T68251 CH53AG 24955156 IC50 = 47 nM T68251 CZC1P7 24955511 IC50 = 35 nM T68251 CL2G8J 24955513 IC50 = 281 nM T68251 CXG36M 24955514 IC50 = 4.8 nM T68251 CXO9Y4 24955857 IC50 = 36 nM T68251 CKY2F6 24955858 IC50 = 9.3 nM T68251 C4LJ8N 24955859 IC50 = 70 nM T68251 CX4MY3 24955861 IC50 = 67 nM T68251 CR29SO 24956227 IC50 = 509 nM T68251 CSM26P 24956228 IC50 = 102 nM T68251 C13JHO 24956229 IC50 = 4 nM T68251 C01QMC 24956580 IC50 = 1057 nM T68251 C8M5PJ 24956581 IC50 = 142 nM T68251 CC90AR 24956582 IC50 = 2382 nM T68251 CQH6I4 24956585 IC50 = 178 nM T68251 CHJ50Q 24956943 IC50 = 202 nM T68251 CN2AS5 24956945 IC50 = 670 nM T68251 C2HN8M 24956948 IC50 = 9.5 nM T68251 C2VEZ0 24957161 IC50 = 1318 nM T68251 CNCA57 25004194 Ki = 1.6 nM T68251 CIO26D 25022463 IC50 = 3 nM T68251 CWO3E0 25022465 IC50 = 170000 nM T68251 CAQ9Z1 25022681 Ki > 3333 nM T68251 CU6M9K 25060725 IC50 = 5400 nM T68251 CF7X2P 25060975 IC50 = 19000 nM T68251 CVR52U 25066764 IC50 = 60 nM T68251 CD2KA4 25102047 IC50 = 1.5 nM T68251 CRW96X 25102048 IC50 = 1 nM T68251 CQ3O9P 25102050 IC50 = 0.33 nM T68251 CSHA26 25102051 IC50 = 1.4 nM T68251 C7ADO2 25102197 IC50 = 0.37 nM T68251 CUR58H 25116339 IC50 = 297300 nM T68251 CA5DJ4 25138228 Ki = 2267000 nM T68251 CX6D9J 25138245 Ki > 3000 nM T68251 C7A6JQ 25138250 Ki = 5700 nM T68251 C6N7EQ 25138258 Ki > 3333 nM T68251 C7AD1J 25138259 Ki = 2933 nM T68251 CJ9TQ2 25138260 Ki > 3333 nM T68251 CUT8I7 25138261 Ki = 3300 nM T68251 CBD9X6 25138262 Ki > 3333 nM T68251 C8LX1S 25138263 Ki = 1367 nM T68251 C3OV1L 25138264 Ki > 3333 nM T68251 C92WVM 25138265 Ki > 3333 nM T68251 CMCS41 25138266 Ki > 3333 nM T68251 C1FJV5 25138267 Ki > 3333 nM T68251 C9N6WT 25138268 Ki > 3333 nM T68251 CF4QI1 25138269 Ki > 3333 nM T68251 C6P5UL 25138270 Ki > 3333 nM T68251 CQE0L7 25138271 Ki > 3333 nM T68251 C59XWU 25138272 Ki > 3333 nM T68251 C1TNQ3 25141117 Ki = 8.5 nM T68251 CYZ2J7 25141282 IC50 = 2 nM T68251 CR35QP 25144971 IC50 > 2500 nM T68251 C0Y5BC 25145683 IC50 > 2500 nM T68251 CGW49I 25146686 IC50 > 200000 nM T68251 CP0YF8 25146956 IC50 = 2900 nM T68251 C12AVL 25146957 IC50 = 3400 nM T68251 C10MBE 25146958 IC50 = 1500 nM T68251 CIUY75 25146959 IC50 = 2100 nM T68251 C5MG9N 25146960 IC50 = 6100 nM T68251 C83IOD 25147056 IC50 = 2200 nM T68251 C1IA0W 25147057 IC50 = 100 nM T68251 CB3W1I 25147058 IC50 = 800 nM T68251 CC35MZ 25147059 IC50 = 2200 nM T68251 CO5H9V 25147060 IC50 = 1600 nM T68251 CM20ZC 25147061 IC50 = 5 nM T68251 C2KZ0T 25147062 IC50 = 12 nM T68251 C5RMI2 25147153 IC50 = 100 nM T68251 C43YCQ 25147154 IC50 = 16 nM T68251 CPQW89 25147155 IC50 = 109 nM T68251 CQ3I6B 25147156 IC50 = 1100 nM T68251 CA34UT 25147158 IC50 = 4200 nM T68251 C3R0DB 25147159 IC50 = 5200 nM T68251 CV4ZE9 25147248 IC50 = 2100 nM T68251 C73HYI 25147249 IC50 = 3000 nM T68251 CV14TY 25147250 IC50 = 1 nM T68251 CUW8X2 25147251 IC50 = 4 nM T68251 C0Z7NX 25147252 IC50 = 11 nM T68251 CU1KO6 25147352 IC50 = 1000 nM T68251 CB1DY9 25147768 IC50 = 182900 nM T68251 CB7V8Y 25147773 IC50 = 0.35 nM T68251 C3KF1V 25178145 IC50 = 1.57 nM T68251 C8PMK7 25178356 IC50 > 100000 nM T68251 CG5Y2R 25178357 IC50 = 24.7 nM T68251 C4PZY6 25180866 IC50 = 145 nM T68251 CEP9Q2 25180867 IC50 = 0.5 nM T68251 C9HZG2 25181078 IC50 = 5120 nM T68251 CMYP34 25181079 IC50 = 2230 nM T68251 C7U1YC 25181080 IC50 = 25.3 nM T68251 C85HLG 25181081 IC50 = 16.2 nM T68251 CHR2P1 25183768 Ki > 25000 nM T68251 CZ8CR1 25190501 Ki > 3333 nM T68251 CO8CD1 25190502 Ki > 3333 nM T68251 C0R6MU 25212135 IC50 > 100000 nM T68251 C76PIF 26183540 IC50 = 33260 nM T68251 C9GCO4 28602444 IC50 = 48000 nM T68251 CW17CN 40516924 IC50 > 500000 nM T68251 C89YBJ 40582645 IC50 > 500000 nM T68251 C6AR8O 42623563 IC50 = 22000 nM T68251 CX0VP7 42623564 IC50 = 28000 nM T68251 C0H3RD 42627769 IC50 = 270 nM T68251 CB0QL3 42630085 IC50 = 37800 nM T68251 C7OX3C 42630086 IC50 = 47600 nM T68251 CAR56O 42645280 IC50 = 170200 nM T68251 CA6PS7 42645281 IC50 = 23500 nM T68251 C7R4JW 42645285 IC50 = 11200 nM T68251 CS29ZL 42645288 IC50 = 99700 nM T68251 C9JE0F 42645511 IC50 = 112100 nM T68251 CMK8T4 42645513 IC50 = 99700 nM T68251 CUF1L4 42645514 IC50 = 201900 nM T68251 C9WL3F 42645516 IC50 = 219400 nM T68251 C8OK0L 42645753 IC50 = 100700 nM T68251 C6K7LG 42645755 IC50 = 328500 nM T68251 CWS5M7 42645986 IC50 = 221000 nM T68251 CQBN65 42645987 IC50 = 632400 nM T68251 C6PI2X 42645989 IC50 = 211300 nM T68251 C8KM4E 43366432 IC50 = 8000 nM T68251 CPO1Z3 44123600 IC50 = 0.2 nM T68251 CWS64Q 44143474 IC50 > 15000 nM T68251 C7HV5Q 44143475 IC50 = 1590 nM T68251 C06IJY 44143476 IC50 = 1401 nM T68251 CVM82U 44143477 IC50 = 1241 nM T68251 C5XEB8 44143478 IC50 = 516 nM T68251 C0ZW7S 44143480 IC50 = 1093 nM T68251 C7K0YS 44143481 IC50 = 2674 nM T68251 CWU1K0 44143482 IC50 = 3614 nM T68251 CA29EQ 44143483 IC50 = 96 nM T68251 CA5P3E 44143484 IC50 = 15099 nM T68251 C7ER1N 44143485 IC50 = 855 nM T68251 C8YNO3 44143486 IC50 = 145 nM T68251 CLJG93 44143487 IC50 = 1743 nM T68251 CJB54F 44143488 IC50 = 2140 nM T68251 CH1IR0 44144307 IC50 = 14110 nM T68251 CT96JB 44199512 IC50 = 142900 nM T68251 C85BFQ 44199516 IC50 = 331100 nM T68251 CT80ED 44219901 Ki = 25 nM T68251 C94JVY 44219902 IC50 = 74 nM T68251 C7J6GH 44219903 IC50 = 26 nM T68251 C9J7WL 44219904 IC50 = 360 nM T68251 CRQ71E 44219905 IC50 = 310 nM T68251 C4Z0ID 44219906 IC50 = 56 nM T68251 CRNA25 44220092 IC50 = 17 nM T68251 C9T5ZF 44220093 IC50 = 9.6 nM T68251 CV38TE 44222825 IC50 = 5.5 nM T68251 CJI73R 44222826 IC50 = 1.5 nM T68251 CGQ30N 44222827 Ki = 3.8 nM T68251 CCI64J 44224245 IC50 = 66 nM T68251 CLRT69 44247751 IC50 = 3.5 nM T68251 CAR34Y 44263877 IC50 = 8.8 nM T68251 CEV08N 44263913 IC50 = 1.6 nM T68251 C5ZI0X 44263926 IC50 = 0.68 nM T68251 CO3C1E 44263994 IC50 = 2.7 nM T68251 C9XJ7U 44264020 IC50 = 3.4 nM T68251 C6L0MJ 44264021 IC50 = 2.4 nM T68251 CJ1WE7 44264036 IC50 = 0.7 nM T68251 C50QFR 44264375 IC50 = 5.3 nM T68251 CDL25C 44265349 Ki < 2.8 nM T68251 C3W4QO 44265401 Ki = 48 nM T68251 C2Q3JV 44265407 Ki = 2033 nM T68251 CN59QT 44265437 Ki = 500 nM T68251 CZA61K 44265475 Ki = 4.5 nM T68251 CD4A7F 44265476 Ki = 1133 nM T68251 CT6FK0 44265480 Ki < 2.8 nM T68251 C67HUL 44265485 Ki < 1 nM T68251 CH0O3I 44265492 Ki = 39 nM T68251 C4C7DY 44265493 Ki = 21 nM T68251 C0DFG7 44265501 Ki = 27 nM T68251 CXSD62 44265506 Ki = 310 nM T68251 CCM8K0 44265512 Ki = 2.8 nM T68251 CB3E6O 44265527 Ki < 2.8 nM T68251 COU3Y8 44266817 IC50 = 31 nM T68251 CUA5E0 44266818 IC50 = 8 nM T68251 CG23BI 44266830 IC50 = 8 nM T68251 C3YK0O 44268937 IC50 = 1000 nM T68251 C5DG8Z 44268941 IC50 = 200 nM T68251 C3SGT4 44268967 IC50 = 400 nM T68251 C1Z0GQ 44269012 IC50 = 1000 nM T68251 C18VGL 44269017 IC50 = 10000 nM T68251 CRF2Z5 44271421 IC50 = 8.05 nM T68251 CG7X5F 44272675 IC50 = 42.5 nM T68251 C2MWR0 44275913 Ki = 6.1 nM T68251 CKV1E7 44275972 Ki = 20 nM T68251 C6YT3K 44280285 Ki = 300 nM T68251 CC2O3U 44280323 Ki = 14 nM T68251 CIE09F 44280336 Ki = 0.3 nM T68251 CA1V6Y 44280345 Ki = 2 nM T68251 CI9L2E 44280411 Ki = 472 nM T68251 C8KZ2F 44281541 IC50 = 50 nM T68251 CRK8H6 44281557 IC50 = 66 nM T68251 CTJ7Q2 44281563 IC50 = 2.5 nM T68251 COU71D 44281564 IC50 = 64 nM T68251 CJ2PG9 44281705 IC50 = 23 nM T68251 C1M3JR 44281777 IC50 = 6.2 nM T68251 CL18QW 44281786 IC50 = 52 nM T68251 C3ES4Z 44281796 IC50 = 1.3 nM T68251 C60HIN 44281797 IC50 = 2.3 nM T68251 C8U5GR 44281941 IC50 = 110 nM T68251 CN23FC 44282968 IC50 = 1700 nM T68251 C2TV5I 44282969 IC50 = 50 nM T68251 CG3LF0 44282970 IC50 = 200 nM T68251 CC5XL3 44286083 IC50 = 48 nM T68251 CXT37W 44286406 IC50 = 35000 nM T68251 CB1R9G 44286414 IC50 > 10000 nM T68251 C7CU3J 44286466 IC50 = 19000 nM T68251 CZ2AL1 44286483 IC50 > 100000 nM T68251 C8I2EF 44286485 IC50 > 10000 nM T68251 C48FEB 44286518 IC50 = 130 nM T68251 CKM8V6 44286563 IC50 = 61 nM T68251 CJ1HT6 44288855 IC50 > 10000 nM T68251 CT38HI 44289140 IC50 > 10000 nM T68251 CAH30U 44289181 IC50 > 10000 nM T68251 CH1TS5 44289182 IC50 > 10000 nM T68251 CMZ2O6 44289200 IC50 > 10000 nM T68251 CBLC60 44289352 Ki = 31 nM T68251 CZO75J 44289369 Ki = 0.8 nM T68251 CRT7O2 44289382 Ki = 8 nM T68251 C7WUJ2 44289459 IC50 > 10000 nM T68251 CJ73FW 44289479 IC50 > 10000 nM T68251 CWMI67 44289482 IC50 > 10000 nM T68251 C1L4ZU 44289489 IC50 > 10000 nM T68251 C19EJM 44289515 IC50 > 10000 nM T68251 C6TI3X 44289520 Ki > 10000 nM T68251 CA52ED 44289521 Ki > 10000 nM T68251 C30KSP 44289579 Ki = 38 nM T68251 CHC08W 44289601 Ki = 36 nM T68251 CZ4EI7 44289602 Ki = 8 nM T68251 CEML82 44289603 Ki = 88 nM T68251 CM26JT 44289604 Ki = 27 nM T68251 CLY4K5 44289640 Ki = 4 nM T68251 C7GY8M 44289643 Ki > 10000 nM T68251 CV9B2F 44289867 Ki > 10000 nM T68251 CJ7VW3 44291166 IC50 = 0.7 nM T68251 C75IEN 44291420 IC50 = 30 nM T68251 CF21CS 44291532 IC50 = 0.7 nM T68251 CU75TB 44291559 IC50 = 53 nM T68251 C06JAO 44291626 IC50 = 49 nM T68251 C5XS0I 44294322 Ki = 1533 nM T68251 CC4V8S 44295180 IC50 = 50 nM T68251 CRW07Z 44295181 IC50 = 20 nM T68251 CL5QG6 44295202 IC50 = 540 nM T68251 CF0T8W 44295423 IC50 = 180 nM T68251 CVS7I1 44295425 IC50 = 550 nM T68251 CAFB18 44296974 Ki = 75 nM T68251 C5RSX9 44300181 IC50 = 19000 nM T68251 CKN3P7 44302022 IC50 = 100 nM T68251 C2Y0PK 44302023 IC50 = 9 nM T68251 C5S3UO 44302024 IC50 = 8 nM T68251 C8ERW6 44302042 IC50 = 10 nM T68251 C6JXH0 44302043 IC50 = 90 nM T68251 CI56DL 44302044 IC50 = 50 nM T68251 CWB83G 44302076 IC50 = 3 nM T68251 CY1J9U 44302096 IC50 = 5 nM T68251 CW94ZQ 44302164 IC50 = 47 nM T68251 C2FSR6 44302165 IC50 < 0.15 nM T68251 CQ54PZ 44302166 IC50 = 0.5 nM T68251 C9U3XT 44302167 IC50 = 0.6 nM T68251 C5X1WY 44302183 IC50 = 7 nM T68251 CQS19O 44302187 IC50 = 39810.72 nM T68251 C7G3BN 44302200 IC50 = 7 nM T68251 CMB4Q8 44302221 IC50 = 200 nM T68251 C70QWV 44302327 IC50 = 900 nM T68251 CZP20C 44302339 IC50 = 14 nM T68251 CO73BW 44302357 IC50 = 9 nM T68251 C6R0VK 44302358 IC50 = 500 nM T68251 CXUZ19 44302359 IC50 = 1 nM T68251 CNL4E2 44302361 IC50 = 19.95 nM T68251 C6YB0Q 44302364 IC50 = 10000 nM T68251 CCW65Y 44302378 IC50 = 1.995 nM T68251 CDK9W1 44302383 IC50 = 30.2 nM T68251 CYG80V 44302385 IC50 = 15 nM T68251 C7ZBR4 44302396 IC50 = 0.6 nM T68251 C8S5WT 44302397 IC50 = 1 nM T68251 CPC25G 44302409 IC50 = 13 nM T68251 C4QL0I 44302411 IC50 = 1 nM T68251 C4NDA2 44302416 IC50 = 12 nM T68251 C24ZWF 44302429 IC50 = 17 nM T68251 C4I6WO 44302430 IC50 = 0.8 nM T68251 CYL71W 44302432 IC50 = 3 nM T68251 C2X3QG 44302433 IC50 = 1000 nM T68251 C1J2AN 44302479 IC50 = 794.33 nM T68251 CE3BX0 44302505 IC50 = 200 nM T68251 C5H6OV 44302627 IC50 = 8 nM T68251 C6QR7C 44302634 IC50 = 15 nM T68251 CG8KJ0 44302661 IC50 = 5 nM T68251 CUZS20 44302663 IC50 = 600 nM T68251 CX1M3Q 44302666 IC50 = 6 nM T68251 C36CQP 44302952 IC50 = 12 nM T68251 CALD50 44304020 Ki > 3000 nM T68251 CTU4S6 44304048 Ki > 3000 nM T68251 CSVK45 44304230 Ki > 3000 nM T68251 CLH14M 44305978 IC50 = 5.9 nM T68251 CZ49UN 44305988 IC50 = 2.3 nM T68251 C6I8JA 44306058 IC50 = 1.9 nM T68251 CB5EY3 44306200 IC50 = 6.5 nM T68251 C0YOH1 44306202 IC50 = 3.8 nM T68251 CMA39E 44306203 IC50 = 2.1 nM T68251 CL58OS 44306208 IC50 = 14000 nM T68251 CAY2S4 44306209 IC50 = 1400 nM T68251 C27NJX 44306277 IC50 = 0.3 nM T68251 C6O1AN 44306279 IC50 = 0.8 nM T68251 C5AM6P 44308844 IC50 = 1587.17 nM T68251 CZUY51 44310789 Ki = 8.1 nM T68251 CH92OI 44310813 Ki = 3 nM T68251 CI4Y5N 44310825 Ki = 13 nM T68251 C5W8QH 44310847 Ki = 6.9 nM T68251 CLQV12 44310863 Ki = 0.44 nM T68251 CN9P5A 44310921 Ki = 0.42 nM T68251 CXB76U 44310932 Ki = 0.7 nM T68251 CMW5G3 44310933 Ki = 8.1 nM T68251 CBY0T1 44310973 Ki = 25 nM T68251 C5D9FS 44311011 Ki = 0.59 nM T68251 C2GC9W 44311172 Ki = 18 nM T68251 C0K1IL 44311187 Ki = 1.3 nM T68251 CL3CS0 44311254 Ki = 43 nM T68251 CV63JP 44311265 Ki = 1.9 nM T68251 CS56ER 44311267 Ki = 46 nM T68251 C5MBT7 44311268 Ki = 7.5 nM T68251 CM64HK 44311313 Ki = 1.9 nM T68251 CLQ48B 44311332 Ki = 6.7 nM T68251 C5AO7Z 44311335 Ki = 0.7 nM T68251 C78TEU 44311349 Ki = 0.96 nM T68251 CJEM64 44311491 Ki = 1.1 nM T68251 C2W5NQ 44311510 Ki = 0.47 nM T68251 C2MIT8 44311525 Ki = 1 nM T68251 CP7L6Q 44311566 Ki = 4 nM T68251 C0B4HZ 44312333 Ki = 12.88 nM T68251 CK9XB7 44314087 IC50 = 20 nM T68251 C8MRB1 44314322 IC50 = 0.36 nM T68251 CB6UL7 44314349 IC50 = 1.5 nM T68251 C3R0DL 44314366 IC50 = 1.9 nM T68251 C5ZTU6 44314442 Ki = 3.82 nM T68251 C2JUX9 44314443 Ki = 1.17 nM T68251 C92MGV 44314566 IC50 = 0.86 nM T68251 CLT6E0 44314618 IC50 = 3.7 nM T68251 CC95EZ 44314744 Ki = 0.33 nM T68251 CY63DG 44314754 Ki = 0.01 nM T68251 C8ZD7F 44314755 Ki = 10 nM T68251 COF0B1 44314762 Ki = 0.08 nM T68251 C59CBZ 44314763 Ki = 0.06 nM T68251 C9L1NY 44314788 Ki = 0.01 nM T68251 CM04TG 44314789 Ki = 0.03 nM T68251 C7LCN0 44314824 Ki = 10.3 nM T68251 CNM6W8 44314841 Ki = 0.01 nM T68251 C9K8JZ 44314900 Ki = 0.254 nM T68251 CXRE70 44314901 Ki = 0.06 nM T68251 CK3H1Y 44314929 Ki = 2.24 nM T68251 CS5A6Z 44314930 Ki = 0.06 nM T68251 CNB72W 44314931 Ki = 0.05 nM T68251 CBXI30 44314932 Ki = 0.02 nM T68251 CCF80X 44314958 Ki = 812 nM T68251 C3N8RQ 44314969 Ki = 1.83 nM T68251 C9SRT4 44314970 Ki = 1.03 nM T68251 C61DST 44314974 Ki = 0.03 nM T68251 CE2J4M 44314975 Ki = 0.01 nM T68251 CQE0D3 44314976 Ki = 0.59 nM T68251 CI2V1Y 44314995 Ki = 123 nM T68251 C48NVD 44314999 Ki = 0.01 nM T68251 CB7F0J 44315000 Ki = 0.3 nM T68251 CSY78M 44315028 Ki = 1300 nM T68251 CDZ5O3 44315029 Ki = 550 nM T68251 C6HW5G 44315084 Ki = 0.01 nM T68251 CV6KW1 44315085 Ki = 0.02 nM T68251 CH48TD 44315155 IC50 = 110 nM T68251 CAUQ47 44315167 Ki = 6 nM T68251 COA01P 44315179 Ki = 3000 nM T68251 CQ1R9E 44315204 Ki = 3.06 nM T68251 CL32FZ 44315221 Ki = 620 nM T68251 CDN4Y5 44315222 Ki = 860 nM T68251 C62FXJ 44315244 IC50 = 2.6 nM T68251 CP9M6W 44315277 Ki = 0.1 nM T68251 C3SZO4 44315279 Ki = 18.9 nM T68251 CSG05N 44315321 Ki = 0.02 nM T68251 COD08C 44315324 Ki = 46.5 nM T68251 C50IQE 44315333 IC50 = 6.6 nM T68251 C37JMW 44315348 Ki = 6.4 nM T68251 C89IQW 44318090 IC50 = 1 nM T68251 CJU31O 44321285 Ki = 17 nM T68251 C41VFA 44321286 Ki = 8 nM T68251 C5S2ZU 44321484 Ki = 85 nM T68251 CLQ23M 44321485 Ki = 202 nM T68251 CHF76Q 44321540 Ki = 9 nM T68251 CVOL49 44321593 Ki = 30 nM T68251 CB97GK 44321601 Ki = 26 nM T68251 CT0O7Y 44321602 Ki = 260 nM T68251 CU62BP 44321746 Ki = 11 nM T68251 CQU2K9 44321782 Ki = 100 nM T68251 CV8T3N 44321783 Ki = 19 nM T68251 CIBO50 44321801 Ki = 6 nM T68251 C4E8GU 44321802 Ki = 30 nM T68251 CYDN18 44321803 Ki = 40 nM T68251 C7Z4DQ 44321887 Ki = 24 nM T68251 CFJ20T 44321932 Ki = 10 nM T68251 C2E3RF 44321966 Ki = 75 nM T68251 CW9S1N 44321967 Ki = 330 nM T68251 C1FI3O 44321975 Ki = 14 nM T68251 CLB8J6 44321976 Ki = 80 nM T68251 CR0KN1 44322209 Ki = 250 nM T68251 C5LE1P 44322210 Ki = 31 nM T68251 CQ7AW8 44322211 Ki = 250 nM T68251 CJY2O7 44322214 Ki = 275 nM T68251 CR9GI0 44322215 Ki = 145 nM T68251 CYR6E5 44323170 Ki = 2000 nM T68251 C29OCD 44325165 Ki = 90 nM T68251 C20UGO 44325517 Ki = 157 nM T68251 C1SRC9 44325555 Ki = 6.9 nM T68251 CHMC02 44325564 Ki = 210 nM T68251 C8P6UA 44325625 Ki = 0.02 nM T68251 CBY75J 44325686 Ki = 1900 nM T68251 C6A1JX 44325696 Ki = 0.05 nM T68251 CJU3R8 44325730 Ki = 0.01 nM T68251 CBV73K 44325744 Ki = 0.03 nM T68251 C06ZAH 44325745 Ki = 0.01 nM T68251 C70UFH 44325749 Ki = 0.02 nM T68251 C8EWP2 44325750 Ki = 0.02 nM T68251 C2QL0B 44325810 Ki = 0.03 nM T68251 CS4EV5 44325831 IC50 = 3000 nM T68251 CU9B2Q 44325832 IC50 = 220 nM T68251 CP1NU9 44325834 Ki = 0.59 nM T68251 C7VRX2 44325907 Ki = 0.01 nM T68251 C80RKL 44326171 IC50 > 100000 nM T68251 C64XEI 44326172 IC50 = 670 nM T68251 C08MOK 44326187 IC50 > 100000 nM T68251 C3UB9D 44326260 IC50 = 17000 nM T68251 C1D8RA 44326261 IC50 = 2000 nM T68251 CK6P3C 44326668 IC50 = 370 nM T68251 C63XAO 44327476 IC50 = 90000 nM T68251 C7S4GH 44327780 IC50 = 200000 nM T68251 CXO1S8 44327801 IC50 = 100000 nM T68251 CW1QN6 44327818 IC50 > 500000 nM T68251 CTH2Y7 44327914 IC50 = 120000 nM T68251 CWYJ75 44327915 IC50 = 150000 nM T68251 C27ZST 44327916 IC50 = 60000 nM T68251 COAF26 44327936 IC50 > 500000 nM T68251 C9O8LM 44327939 IC50 = 160000 nM T68251 CB5L2U 44327940 IC50 = 72000 nM T68251 CI29FZ 44327960 IC50 = 155000 nM T68251 CV2U6R 44327961 IC50 = 54000 nM T68251 C8HUF1 44328149 IC50 > 500000 nM T68251 C85QTP 44328155 IC50 = 1000 nM T68251 CLK87J 44328168 IC50 = 150000 nM T68251 CMHZ13 44328169 IC50 > 500000 nM T68251 CZQ6N7 44328189 IC50 > 100000 nM T68251 C1IG0A 44328244 IC50 = 230000 nM T68251 CEI1V4 44328245 IC50 = 40000 nM T68251 CPI3A5 44328246 IC50 = 100000 nM T68251 CPU60Z 44328254 IC50 = 150000 nM T68251 CW3RX8 44328256 IC50 = 370000 nM T68251 CN81EA 44328258 IC50 = 43000 nM T68251 CR8XQ3 44328259 IC50 = 114000 nM T68251 CCD48V 44328263 IC50 = 2000 nM T68251 C31OKH 44328271 IC50 > 500000 nM T68251 CUA04P 44328279 IC50 = 125000 nM T68251 CHB05O 44328283 IC50 = 52000 nM T68251 CLC39W 44328295 IC50 = 110000 nM T68251 C36FCK 44328296 IC50 = 51000 nM T68251 CI46AP 44328297 IC50 > 500000 nM T68251 CR9YN5 44328312 IC50 > 500000 nM T68251 C8W9KN 44328316 IC50 = 50000 nM T68251 CPT80U 44328317 IC50 = 60000 nM T68251 CBD0Z2 44329014 IC50 = 5.97 nM T68251 CMLA39 44329018 IC50 = 1.3 nM T68251 C84MVU 44329019 IC50 = 5.73 nM T68251 C90CHA 44329405 IC50 = 7079.46 nM T68251 C2PB4Z 44329622 IC50 = 500 nM T68251 CI3Z4K 44329623 IC50 = 80 nM T68251 C6OL8M 44329636 IC50 = 10000 nM T68251 CB0G1H 44329644 IC50 = 1995.26 nM T68251 CA65RO 44329672 IC50 = 1995.26 nM T68251 CK9HO7 44329673 IC50 = 2000 nM T68251 C07GRS 44329693 IC50 = 60 nM T68251 CBH16R 44329694 IC50 = 600 nM T68251 CG3E7A 44329712 IC50 = 19.95 nM T68251 C9SN6I 44329713 IC50 = 3000 nM T68251 CZ2FW6 44329725 IC50 = 1995.26 nM T68251 CDKI48 44329741 IC50 = 500 nM T68251 CK3M2H 44329742 IC50 = 3000 nM T68251 C39RDS 44329886 IC50 = 50 nM T68251 C3YAF6 44329898 IC50 = 7000 nM T68251 C63RHP 44329909 IC50 = 95.5 nM T68251 CVQA75 44329910 IC50 = 398.11 nM T68251 C84SLI 44329926 IC50 = 100 nM T68251 CJS6B1 44329927 IC50 = 398.11 nM T68251 C2K6OU 44329943 IC50 = 95.5 nM T68251 C5BYR4 44329998 IC50 = 3400 nM T68251 C0SMC9 44330092 IC50 = 21 nM T68251 C35SIO 44330094 IC50 = 12.88 nM T68251 C3NM2G 44330095 IC50 = 0.7943 nM T68251 C6SCU5 44330119 IC50 = 0.26 nM T68251 C69KPL 44330130 IC50 = 109.65 nM T68251 C9P6ZF 44330131 IC50 = 10 nM T68251 C9R1ZE 44330132 IC50 = 55000 nM T68251 CKS01F 44330133 IC50 = 2187.76 nM T68251 CLU8I7 44330135 IC50 = 7000 nM T68251 C1IE0S 44330147 IC50 > 100000 nM T68251 CPG7N2 44330149 IC50 = 15000 nM T68251 CYP6S4 44330152 IC50 = 6000 nM T68251 CMGA28 44330163 IC50 = 41000 nM T68251 CXI49L 44330197 IC50 = 4000 nM T68251 CDQM84 44330198 IC50 = 0.048 nM T68251 CH6EN4 44330225 IC50 = 3388.44 nM T68251 C3GA9Q 44330226 IC50 = 0.23 nM T68251 CG2Q8W 44332306 IC50 = 36 nM T68251 C5NG0R 44334948 IC50 = 30 nM T68251 CFP3X8 44334949 IC50 = 53 nM T68251 CV5RF0 44334963 IC50 = 441 nM T68251 C4AOZ7 44334981 IC50 = 143 nM T68251 CXW59C 44334982 IC50 = 4.6 nM T68251 CCH1W8 44334983 IC50 = 2.5 nM T68251 CQ0UI1 44335017 IC50 = 32 nM T68251 CX58SB 44335240 IC50 = 1.64 nM T68251 CA96JG 44335285 IC50 = 15.4 nM T68251 CI5X0G 44339523 IC50 = 7.2 nM T68251 CB9K8T 44339536 IC50 = 9.5 nM T68251 C2R3XN 44339554 IC50 = 6.5 nM T68251 C2CRY1 44339556 IC50 = 8.6 nM T68251 CTBU53 44339564 IC50 = 23 nM T68251 C58OSK 44339567 IC50 = 7.2 nM T68251 CX2KJ3 44339574 IC50 = 110 nM T68251 CEK3G0 44339588 IC50 = 8.5 nM T68251 C7ZR6H 44339589 IC50 = 1100 nM T68251 C0WP9C 44339590 IC50 = 2.7 nM T68251 C5C2LI 44339654 IC50 = 1 nM T68251 CLD2P9 44339900 Ki = 4400 nM T68251 C2D6VN 44339918 Ki = 2.1 nM T68251 CRQJ09 44339936 Ki = 1300 nM T68251 C4JLG8 44340091 Ki = 6.1 nM T68251 CXW34P 44340094 Ki = 19 nM T68251 CGV94P 44340160 Ki = 7.3 nM T68251 C3IS1O 44340161 Ki = 130 nM T68251 CPK5W0 44340172 Ki = 26 nM T68251 CJ4Z9W 44340207 Ki = 570 nM T68251 CZ31VY 44340208 Ki = 12 nM T68251 C4B9QZ 44340327 Ki = 20 nM T68251 C2XY8H 44340328 Ki = 2.1 nM T68251 CAT48Z 44340657 Ki = 20 nM T68251 C3CYZ8 44340673 Ki = 1100 nM T68251 CRI8Q4 44340696 Ki = 1100 nM T68251 CF1QZ3 44340718 Ki = 70 nM T68251 C09ILT 44340727 Ki = 120 nM T68251 C6AS8J 44340740 Ki = 570 nM T68251 CL0U9T 44340810 Ki = 60 nM T68251 CV6W7Z 44340812 Ki = 770 nM T68251 C3WZM0 44340828 Ki = 2300 nM T68251 CW53EF 44340868 Ki = 350 nM T68251 C6ZDV3 44340869 Ki = 120 nM T68251 CR1ID4 44340923 Ki = 110 nM T68251 CL9I4M 44341538 Ki = 1533 nM T68251 CE3MT4 44341611 Ki = 4650 nM T68251 CJTZ45 44341652 Ki = 200000 nM T68251 C2XP4N 44342352 Ki = 3000 nM T68251 C2SZB1 44342614 IC50 = 6 nM T68251 CTQ6P4 44344631 IC50 = 34200 nM T68251 CBH9I5 44344658 IC50 = 750 nM T68251 CCF94Z 44349787 IC50 = 572 nM T68251 C1L2GF 44350073 IC50 = 20 nM T68251 CQ5RN6 44350101 IC50 = 130 nM T68251 CE2X3Q 44350116 IC50 > 100 nM T68251 CO9R4W 44356376 Ki > 3333 nM T68251 C3MZA1 44356386 Ki > 3333 nM T68251 CH1E2S 44356406 Ki > 3333 nM T68251 C84LUM 44356631 Ki > 3333 nM T68251 CG6T9A 44356632 Ki > 3333 nM T68251 C3WFH7 44356634 Ki > 3333 nM T68251 CB8KY4 44356635 Ki > 3333 nM T68251 COIA82 44356636 Ki > 3333 nM T68251 C4BU6T 44356644 Ki > 3333 nM T68251 CH9YT4 44356659 Ki > 3333 nM T68251 C68LMR 44356675 Ki > 3333 nM T68251 C69YIP 44356686 Ki > 3333 nM T68251 CT05XN 44356687 Ki 1079 nM T68251 CML03W 44356689 Ki > 3333 nM T68251 CQ4NP5 44356690 Ki > 3333 nM T68251 CE8U2Y 44356714 Ki > 3333 nM T68251 CCY5U3 44356804 Ki = 200 nM T68251 C27LMU 44356852 Ki > 3333 nM T68251 CTU64D 44356889 Ki > 3333 nM T68251 C4TM1I 44356890 Ki > 3333 nM T68251 C1WA4B 44356906 Ki > 3333 nM T68251 C50ELY 44356907 Ki 675 nM T68251 CVU8L2 44356924 Ki > 3333 nM T68251 CD1GW2 44356953 Ki > 1011 nM T68251 CR41QN 44356969 Ki > 2454 nM T68251 C3BT0N 44356971 Ki = 642 nM T68251 C81OIZ 44356983 Ki > 3333 nM T68251 CHNC03 44356993 Ki > 3333 nM T68251 C9Z3RT 44356998 Ki > 3333 nM T68251 CR4A7G 44356999 Ki = 476 nM T68251 C2VS6P 44357000 Ki = 1537 nM T68251 CES1G8 44357007 Ki > 3333 nM T68251 C6NQ7K 44357012 Ki = 656 nM T68251 C2HIN3 44357023 Ki > 3333 nM T68251 CI4JO7 44357024 Ki 585 nM T68251 CW4VQ3 44357029 Ki > 3333 nM T68251 C2AIT6 44357209 Ki > 3333 nM T68251 CJK2P7 44357220 Ki > 3333 nM T68251 CIX6G5 44357225 Ki > 3333 nM T68251 CT4C6P 44360260 IC50 = 4.2 nM T68251 CY5I3O 44360286 IC50 = 35 nM T68251 C40OCB 44360287 IC50 = 1.8 nM T68251 C3IW9L 44360784 IC50 = 1.4 nM T68251 CGQ92A 44364037 IC50 = 33 nM T68251 C36YLM 44364111 IC50 = 150 nM T68251 CN4T7Q 44364119 IC50 = 76 nM T68251 CH4TE7 44364121 IC50 = 24 nM T68251 CPE91Y 44364122 IC50 = 18 nM T68251 CG2X0C 44364224 IC50 = 430 nM T68251 C1F8XN 44364249 IC50 = 26 nM T68251 CWM47H 44364250 IC50 = 27 nM T68251 C0W5TL 44364251 IC50 = 1099 nM T68251 C3TPO7 44364266 IC50 = 853 nM T68251 CJ2B8F 44364280 IC50 = 724 nM T68251 C90CYD 44367175 IC50 = 4 nM T68251 C2DV0R 44367276 IC50 = 0.5 nM T68251 C5BAW2 44367284 IC50 < 0.4 nM T68251 C2YG5E 44367285 IC50 = 11 nM T68251 CUDF82 44367309 IC50 = 1 nM T68251 CA0CJ1 44368580 IC50 = 25.7 nM T68251 CW0Y3K 44368632 IC50 = 30 nM T68251 CU8FD2 44368650 IC50 = 109.65 nM T68251 CLE71V 44368654 IC50 = 15.14 nM T68251 CQ27XL 44368655 IC50 = 3.388 nM T68251 CH9G3O 44368849 IC50 = 1 nM T68251 CV6ZG4 44368850 IC50 = 1.288 nM T68251 CB2U9G 44368858 IC50 = 270 nM T68251 CN78UB 44368864 IC50 = 5.754 nM T68251 CV8ZA4 44368865 IC50 = 1.585 nM T68251 CW8O3S 44368924 IC50 = 50.12 nM T68251 C6CD9A 44368928 IC50 = 280 nM T68251 C5HF6P 44368940 IC50 = 330 nM T68251 CE30XV 44368941 IC50 = 50 nM T68251 CG2P9T 44368942 IC50 = 83.18 nM T68251 C7HT1U 44368944 IC50 = 3467.37 nM T68251 C1CW5A 44368946 IC50 = 6165.95 nM T68251 CV86QS 44368963 IC50 = 331.13 nM T68251 C4C7UJ 44368968 IC50 = 38 nM T68251 C3EW6B 44368969 IC50 = 416.87 nM T68251 C4I6ME 44368970 IC50 = 61 nM T68251 C8IZC4 44369030 IC50 = 2430 nM T68251 CDW8V9 44369031 IC50 = 6.4 nM T68251 C82BOI 44369038 IC50 = 776.25 nM T68251 C65FBJ 44369041 IC50 = 53.7 nM T68251 CI0S2R 44369094 IC50 = 310 nM T68251 CFI10T 44369095 IC50 = 34 nM T68251 CQGM80 44369096 IC50 = 210 nM T68251 CIR84S 44369104 IC50 = 920 nM T68251 C6SBW5 44369107 IC50 = 100 nM T68251 CAF5P0 44369163 IC50 = 52000 nM T68251 CHC71X 44369164 IC50 = 1700 nM T68251 CY5L0D 44369186 IC50 = 1 nM T68251 C1JZK6 44369209 IC50 = 86 nM T68251 C9BAO2 44369213 IC50 = 6800 nM T68251 CCJ63B 44369214 IC50 = 11 nM T68251 C4E7DM 44369266 IC50 = 41 nM T68251 CI0ZD9 44371783 IC50 = 20 nM T68251 C4VR5M 44371799 IC50 = 251 nM T68251 C4FHG7 44371800 IC50 = 38 nM T68251 CQ5UR4 44372530 IC50 = 240 nM T68251 CCZ6J3 44379232 Ki = 470 nM T68251 CW20ML 44379249 Ki = 110 nM T68251 CXM06G 44379250 Ki = 5.7 nM T68251 CK0B1D 44379273 Ki = 220 nM T68251 COD6P1 44379499 Ki = 2.6 nM T68251 C84YPO 44379547 Ki > 1000 nM T68251 C3EV2A 44384940 IC50 = 530 nM T68251 C0XE8K 44384941 IC50 = 13000 nM T68251 C3IJO9 44384994 IC50 > 50000 nM T68251 CZ6PU7 44389401 Ki = 1.8 nM T68251 CO4W0Y 44389552 Ki = 0.4 nM T68251 CWQ19I 44389560 IC50 = 10.3 nM T68251 C5R4EW 44389591 IC50 = 935 nM T68251 CC7QW9 44391352 IC50 = 21 nM T68251 C89FTQ 44393434 Ki > 3300 nM T68251 CCO3S9 44393444 Ki > 3300 nM T68251 CNO4P6 44393516 Ki > 3300 nM T68251 C5OIK4 44393520 Ki > 3300 nM T68251 C80NZE 44394179 Ki > 3300 nM T68251 CXD05N 44394645 Ki > 100000 nM T68251 CGQ98X 44394681 Ki = 153000 nM T68251 C8MY4S 44394703 Ki = 88000 nM T68251 CCEI41 44394814 Ki > 2000000 nM T68251 CCZ09V 44394886 Ki > 100000 nM T68251 CZB81D 44395506 IC50 = 5 nM T68251 CAU5R4 44397021 IC50 = 23.3 nM T68251 CQR73V 44397047 IC50 = 27.8 nM T68251 CSO92L 44397377 IC50 = 1.9 nM T68251 CMWU78 44397457 IC50 = 19 nM T68251 CU1E2Z 44397536 IC50 = 14 nM T68251 CQ1Y4E 44397568 IC50 = 4 nM T68251 C12MNT 44397632 IC50 = 2 nM T68251 CZ45GV 44397680 IC50 = 12.1 nM T68251 C7Y1VK 44397699 IC50 = 3.9 nM T68251 CHL9S2 44399294 Ki = 2530 nM T68251 CD49UI 44399312 Ki = 600 nM T68251 C3LS8N 44399509 Ki = 3330 nM T68251 CIA8T3 44399555 Ki > 3330 nM T68251 C8PR7S 44400182 IC50 = 9 nM T68251 CQ9F0K 44400232 IC50 = 9 nM T68251 C91POV 44402021 IC50 = 197 nM T68251 CYCJ78 44402280 IC50 = 9.8 nM T68251 CWG3M4 44402281 IC50 > 10000 nM T68251 C9KGL0 44404474 IC50 = 0.91 nM T68251 C92KDG 44404475 IC50 = 7.1 nM T68251 C07CGB 44404477 IC50 = 1050 nM T68251 C7VH3G 44404484 IC50 = 259 nM T68251 CC29XL 44404490 IC50 = 1770 nM T68251 CCN16G 44404500 IC50 = 164 nM T68251 C69GZU 44404501 IC50 = 688 nM T68251 CY6WL5 44404502 IC50 = 1490 nM T68251 CWGQ46 44404503 IC50 = 1610 nM T68251 CLXM58 44404504 IC50 = 2500 nM T68251 C1F9HO 44404506 IC50 = 4340 nM T68251 CLU41O 44404507 IC50 = 7000 nM T68251 C30DKN 44404553 IC50 = 0.04 nM T68251 C0G4MR 44405997 IC50 > 380000 nM T68251 CZ0XC1 44405998 IC50 = 685000 nM T68251 CIC60V 44406452 IC50 = 28 nM T68251 CHM26J 44406652 Ki = 8100 nM T68251 C1K3QM 44406655 IC50 = 20 nM T68251 C6YG5S 44406678 IC50 = 2.6 nM T68251 CB5ZS0 44411587 IC50 = 52 nM T68251 C4Z0BX 44411591 IC50 = 3060 nM T68251 CHV64P 44411592 IC50 = 0.84 nM T68251 CL6IG9 44411599 IC50 = 6.8 nM T68251 C6IKL1 44411602 IC50 = 0.7 nM T68251 CM2UL0 44411603 IC50 = 1.5 nM T68251 CBT4E7 44411614 IC50 = 4 nM T68251 CH8B4W 44411639 IC50 = 1.1 nM T68251 CS74LI 44411640 IC50 = 54 nM T68251 C43HTC 44411693 IC50 = 3 nM T68251 C8HSN2 44411697 IC50 = 1.2 nM T68251 CKQ8P6 44411698 IC50 = 0.74 nM T68251 CVQ82B 44411701 IC50 = 33 nM T68251 C87VNZ 44411702 IC50 = 1.3 nM T68251 C83MTG 44411776 IC50 = 0.98 nM T68251 CT1A8Q 44411815 IC50 = 295 nM T68251 CQLV08 44411816 IC50 = 556 nM T68251 CP16XL 44411819 IC50 = 1.8 nM T68251 C9COT4 44411820 IC50 = 6.5 nM T68251 C3Q8PM 44411822 IC50 = 4.4 nM T68251 CEB0S4 44411823 IC50 = 0.7 nM T68251 CRB85W 44411826 IC50 = 2.3 nM T68251 CV1NO8 44411829 IC50 = 1.7 nM T68251 CPH6V5 44411830 IC50 = 0.62 nM T68251 CRKL06 44411835 IC50 = 145 nM T68251 C0FDM1 44411836 IC50 = 8.6 nM T68251 CUV27I 44411839 IC50 = 19 nM T68251 CD5KV9 44411846 IC50 = 12 nM T68251 C7CU1F 44411852 IC50 = 1.3 nM T68251 CA9OS4 44411865 IC50 = 1.9 nM T68251 CVM7Y3 44413975 IC50 = 49 nM T68251 C4X0GA 44413977 IC50 = 15 nM T68251 CH01EO 44413978 IC50 = 24 nM T68251 CQ8HK9 44413979 IC50 = 553 nM T68251 CBT0P2 44413982 IC50 = 46 nM T68251 CIJ39D 44413983 IC50 = 16 nM T68251 C9BA0V 44413987 IC50 = 111 nM T68251 CE3WP0 44413991 IC50 = 518 nM T68251 CDUI73 44413992 IC50 = 3.1 nM T68251 CH2X6W 44413997 IC50 = 44 nM T68251 CHN85S 44414002 IC50 = 345 nM T68251 C2OJ4B 44414029 IC50 = 302 nM T68251 CT5PC9 44422672 IC50 = 2.3 nM T68251 CS9D5U 44422720 IC50 = 0.39 nM T68251 CNWM05 44422723 IC50 = 1.8 nM T68251 C58LAY 44422724 IC50 = 20 nM T68251 CDQU41 44422736 IC50 = 53 nM T68251 CVUB56 44422737 IC50 = 30 nM T68251 CB8G2W 44422743 IC50 = 24 nM T68251 CFX42T 44422744 IC50 = 980 nM T68251 C9EL7F 44422749 IC50 = 790 nM T68251 CY49HT 44423674 IC50 = 9600 nM T68251 CHI5G1 44423675 IC50 = 1060 nM T68251 CFC3M6 44423676 IC50 = 1500 nM T68251 CO24JF 44423677 IC50 = 5000 nM T68251 C7F9DB 44423678 IC50 = 30000 nM T68251 CJ6GW5 44423679 IC50 = 1980 nM T68251 CUKM29 44423680 IC50 = 2100 nM T68251 C3R0FS 44423681 IC50 = 660 nM T68251 C14DBJ 44423682 IC50 = 730 nM T68251 CU5QV9 44425142 IC50 > 100000 nM T68251 CW8RY1 44425150 IC50 = 5900 nM T68251 C45WZX 44426073 IC50 = 10 ug.mL-1 T68251 CK5H7O 44429877 IC50 = 5000 nM T68251 CQL1X9 44429878 IC50 = 73 nM T68251 C1CYV2 44429879 IC50 = 82 nM T68251 C7AXP9 44429880 IC50 = 58 nM T68251 CXOS97 44429881 IC50 = 11 nM T68251 C2MQ0I 44429882 IC50 = 37 nM T68251 CQ5PT8 44429883 IC50 = 37 nM T68251 CQRO36 44429884 IC50 = 161 nM T68251 CM27YB 44429885 IC50 = 54 nM T68251 C9JH0T 44429886 IC50 = 4 nM T68251 CD2B3T 44429887 IC50 = 62.6 nM T68251 C6V1CO 44429888 IC50 = 2058 nM T68251 CBC6W4 44429889 IC50 = 40 nM T68251 C7A0LF 44429890 IC50 = 176 nM T68251 CS0M3L 44429891 IC50 = 99.5 nM T68251 CX93QY 44429892 IC50 = 19 nM T68251 C7SWV1 44429893 IC50 = 33 nM T68251 C8QKS0 44429894 IC50 = 22 nM T68251 CBS47K 44429896 IC50 = 32 nM T68251 CI7TG1 44429897 IC50 = 61.3 nM T68251 CLJ48T 44429898 IC50 = 51 nM T68251 C3F9CK 44429899 IC50 = 51 nM T68251 C8PVF7 44429900 IC50 = 31 nM T68251 C6U0TK 44429901 IC50 = 20 nM T68251 CBK9M5 44429902 IC50 = 58 nM T68251 C72YFT 44429903 IC50 = 172 nM T68251 CMO9Q3 44429905 IC50 = 183 nM T68251 C8BHL5 44431844 IC50 > 2000 nM T68251 CR1DN9 44431845 IC50 > 2000 nM T68251 CHFB16 44431846 IC50 > 2000 nM T68251 C0C3ZT 44431847 IC50 > 2000 nM T68251 CS49GV 44431848 IC50 > 2000 nM T68251 C4AVK5 44431849 IC50 > 2000 nM T68251 C5DH4Q 44431850 IC50 > 2000 nM T68251 CLHE45 44431851 IC50 > 2000 nM T68251 CYG29L 44431852 IC50 > 2000 nM T68251 C4OF5L 44431853 IC50 > 2000 nM T68251 CWU7G8 44434565 IC50 = 123 nM T68251 CF9HU5 44434566 IC50 = 280 nM T68251 CV3M6F 44434578 IC50 = 120 nM T68251 CJN1K9 44439853 Ki = 20 nM T68251 C71IPQ 44439982 IC50 = 4000 nM T68251 C2WJP3 44439983 IC50 = 4400 nM T68251 CU9Z1H 44439984 IC50 = 1000 nM T68251 C0G4AS 44439985 IC50 = 3800 nM T68251 CV8D9L 44439986 IC50 = 4300 nM T68251 CKP8T1 44439987 IC50 = 2200 nM T68251 CUT86C 44439988 IC50 = 1200 nM T68251 CKC81R 44439990 IC50 = 1200 nM T68251 CPNM45 44439991 IC50 = 600 nM T68251 CROG92 44439992 IC50 = 300 nM T68251 C30RNZ 44439993 IC50 = 1200 nM T68251 C19MPB 44439994 IC50 = 13000 nM T68251 C2N1UC 44439995 IC50 = 1400 nM T68251 C4T0AW 44439996 IC50 = 1800 nM T68251 CJT4H2 44439997 IC50 = 1300 nM T68251 CYM08I 44439998 IC50 = 1700 nM T68251 C83KQO 44439999 IC50 = 15600 nM T68251 C4Y9JD 44440000 IC50 = 500 nM T68251 C5PWG9 44440001 IC50 = 10600 nM T68251 C70MGQ 44440455 Ki > 3333 nM T68251 CDY53F 44440460 Ki > 3333 nM T68251 CTB9P6 44440461 Ki = 307 nM T68251 C63RLK 44440462 Ki > 3333 nM T68251 C23JBO 44440463 Ki > 3333 nM T68251 CT9P3Y 44440464 Ki > 3333 nM T68251 CX32AM 44440465 Ki > 3333 nM T68251 C6FOC7 44440466 Ki > 3333 nM T68251 CMPX37 44440467 Ki > 3333 nM T68251 CV4F6Z 44440468 Ki > 3333 nM T68251 C6K8VB 44440469 Ki > 3333 nM T68251 C4Y0UM 44440470 Ki > 3333 nM T68251 CHU49A 44440471 Ki > 3333 nM T68251 C8OI4L 44440472 Ki > 3333 nM T68251 CV58YW 44441018 Ki > 3333 nM T68251 CV85PN 44441019 Ki > 3333 nM T68251 C5O2WK 44441020 Ki > 3333 nM T68251 CU67WS 44441021 Ki > 3333 nM T68251 CXZ53B 44441022 Ki > 3333 nM T68251 C8S7UT 44441023 Ki > 3333 nM T68251 CT4PZ9 44441024 Ki > 3333 nM T68251 CU9GE6 44441025 Ki > 3333 nM T68251 CB2IT4 44441026 Ki > 3333 nM T68251 CN4X2F 44441027 Ki > 3333 nM T68251 CPF45Y 44441028 Ki > 3333 nM T68251 CAM23N 44441029 Ki > 3333 nM T68251 C23BPG 44441030 Ki > 3333 nM T68251 C5YMT6 44441031 Ki > 3333 nM T68251 C9A6GJ 44441032 Ki > 3333 nM T68251 CYSU19 44441033 Ki > 3333 nM T68251 CB9P0C 44442303 IC50 = 870 nM T68251 C7HO0Y 44442304 IC50 = 1630 nM T68251 CAR3S2 44442305 IC50 = 960 nM T68251 CZK0A9 44442306 IC50 = 2230 nM T68251 C71MCV 44442307 IC50 = 840 nM T68251 CN70HO 44442308 IC50 = 520 nM T68251 CVE5P0 44442309 IC50 = 1110 nM T68251 C3PT7N 44442310 IC50 = 840 nM T68251 CGS18B 44442311 IC50 = 1620 nM T68251 CIZL27 44442312 IC50 = 760 nM T68251 CCFV76 44442313 IC50 = 700 nM T68251 C4HYM6 44442314 IC50 = 260 nM T68251 CZ2PE6 44442315 IC50 = 1030 nM T68251 C3I7RG 44442317 IC50 = 2570 nM T68251 CGR6E7 44442318 IC50 = 1230 nM T68251 C97ZHM 44442319 IC50 = 1450 nM T68251 C3DIB8 44442320 IC50 = 1000 nM T68251 C0HX1L 44445199 IC50 = 67000 nM T68251 CPQT35 44445200 IC50 = 66000 nM T68251 C2X6IP 44445201 IC50 = 72000 nM T68251 CSRB79 44445202 IC50 = 70000 nM T68251 C2O6KZ 44445203 IC50 = 101000 nM T68251 CASF34 44445204 IC50 = 65000 nM T68251 CQZ6M0 44445205 IC50 = 69000 nM T68251 CH7Z5M 44445206 IC50 = 73000 nM T68251 C71CPO 44445207 IC50 > 150 nM T68251 CO9QA4 44445209 IC50 = 70000 nM T68251 CH3UQ5 44445210 IC50 = 110000 nM T68251 C6B4LG 44445211 IC50 > 150 nM T68251 C1WA5N 44445212 IC50 = 90000 nM T68251 CM2CD0 44445213 IC50 = 71000 nM T68251 C6ZX2P 44445214 IC50 = 70000 nM T68251 C9KE8P 44445215 IC50 = 71000 nM T68251 C68QEF 44445216 IC50 = 66000 nM T68251 CCK7W2 44445217 IC50 = 70000 nM T68251 C58BQA 44445218 IC50 = 69000 nM T68251 C4CGN2 44445219 IC50 = 39000 nM T68251 C1IVR6 44445220 IC50 = 86000 nM T68251 CG2U7H 44445221 IC50 = 64000 nM T68251 CVW48J 44445222 IC50 = 69000 nM T68251 CL3HZ8 44445223 IC50 = 69000 nM T68251 CPY73U 44445224 IC50 = 57000 nM T68251 C9MA2F 44445225 IC50 = 68000 nM T68251 C9SJM3 44445226 IC50 = 107000 nM T68251 CH91WG 44445228 IC50 = 90000 nM T68251 CO59HI 44445229 IC50 = 109000 nM T68251 C62WPE 44445230 IC50 = 125000 nM T68251 COIR35 44445231 IC50 = 107000 nM T68251 CBH0M7 44445233 IC50 = 33000 nM T68251 CIS7M5 44445234 IC50 > 150 nM T68251 CKN60A 44445235 IC50 = 73000 nM T68251 CP4XL8 44445237 IC50 = 65000 nM T68251 CJA79R 44445239 IC50 = 111000 nM T68251 CA72BI 44445240 IC50 = 103000 nM T68251 CZJB48 44445241 IC50 > 150000 nM T68251 C85EVH 44445242 IC50 > 150000 nM T68251 C9DI7F 44445243 IC50 = 73000 nM T68251 CVLH67 44445244 IC50 = 85000 nM T68251 CIP3X8 44445245 IC50 = 119000 nM T68251 CL1MK6 44445246 IC50 = 100000 nM T68251 C0CX7T 44445247 IC50 = 7000 nM T68251 CEZ2P7 44445248 IC50 = 98000 nM T68251 CL0K9Q 44445249 IC50 = 110000 nM T68251 C9T2SH 44445250 IC50 = 125000 nM T68251 C5EFP9 44445251 IC50 = 90000 nM T68251 CLJ71G 44445252 IC50 = 91000 nM T68251 C8TF3E 44445253 IC50 = 63000 nM T68251 C4CAY7 44445254 IC50 = 124000 nM T68251 CH1LE5 44445255 IC50 = 108000 nM T68251 CLP96W 44445256 IC50 = 66000 nM T68251 CK8S4Z 44445257 IC50 = 79000 nM T68251 C03EJW 44445258 IC50 = 90000 nM T68251 CO9SM5 44445261 IC50 = 96000 nM T68251 C3FX8B 44445262 IC50 = 108000 nM T68251 CZS8N5 44445263 IC50 = 98000 nM T68251 CMW2U6 44445264 IC50 = 100000 nM T68251 CB47AH 44445265 IC50 = 110000 nM T68251 CA43LS 44445266 IC50 = 42000 nM T68251 C23MDF 44445267 IC50 = 46000 nM T68251 C9K3DI 44445268 IC50 = 93000 nM T68251 C2ZAK4 44445269 IC50 = 77000 nM T68251 CIVC64 44445270 IC50 = 85000 nM T68251 C8W1HX 44445271 IC50 > 150000 nM T68251 CTFR27 44445272 IC50 > 150000 nM T68251 C20DNO 44445273 IC50 > 150000 nM T68251 CWLC15 44445274 IC50 > 150000 nM T68251 CZD5M3 44445275 IC50 > 150000 nM T68251 CJET46 44445276 IC50 > 150000 nM T68251 CI58AM 44445277 IC50 = 149000 nM T68251 CDN37V 44445278 IC50 > 150000 nM T68251 CE36AB 44445279 IC50 > 150000 nM T68251 CV9KX5 44445280 IC50 > 150000 nM T68251 C4S2WX 44445281 IC50 > 150000 nM T68251 C0HXS4 44445391 IC50 = 620 nM T68251 CT1CP7 44445392 IC50 = 4380 nM T68251 CRNK10 44445393 IC50 = 3080 nM T68251 CF0LR3 44445394 IC50 = 776 nM T68251 C9WQ8E 44445790 IC50 = 3.388 nM T68251 CEGL68 44445796 IC50 = 3981.07 nM T68251 CH2Y7W 44445813 Ki = 2.1 nM T68251 C4J2QM 44445814 Ki = 6.1 nM T68251 CP5H1Q 44446267 IC50 = 6 nM T68251 C30TQK 44446273 IC50 = 1470 nM T68251 CB76CO 44446275 IC50 = 860 nM T68251 C20HIJ 44446753 IC50 = 13 nM T68251 C9CS8E 44446754 IC50 = 21 nM T68251 C4Z7IQ 44446755 IC50 = 50 nM T68251 C4K5QT 44446756 IC50 = 1100 nM T68251 CZEH45 44446757 IC50 = 24 nM T68251 C47SRV 44446758 IC50 = 433 nM T68251 C8CVO1 44446759 IC50 = 2500 nM T68251 C8HM5N 44446763 IC50 = 159 nM T68251 CU5Z4V 44446765 IC50 = 14 nM T68251 C9USL8 44446766 IC50 = 4999 nM T68251 CYO65B 44446797 IC50 = 63 nM T68251 CPI3T0 44446799 IC50 < 5 nM T68251 CGH0A2 44446805 IC50 = 32 nM T68251 CH72RW 44446806 IC50 > 5000 nM T68251 CTKX08 44446807 IC50 = 391 nM T68251 CJ1MP7 44446808 IC50 = 1387 nM T68251 CJN1L7 44446821 IC50 = 39 nM T68251 C4LF6Y 44446822 Ki = 302 nM T68251 C9FG5A 44446823 IC50 = 35 nM T68251 C1P0BV 44446824 IC50 = 37 nM T68251 C5AW3N 44446825 IC50 = 50 nM T68251 C17YSI 44446827 IC50 = 53 nM T68251 C3O8AX 44446835 IC50 = 472 nM T68251 CE2OM1 44446839 IC50 = 106 nM T68251 C49VJF 44446842 IC50 = 86 nM T68251 CF4DL2 44446843 IC50 = 960 nM T68251 C8OS4K 44446845 IC50 > 5000 nM T68251 CIP23G 44447330 IC50 = 10 nM T68251 CPS5M4 44447343 IC50 = 64 nM T68251 CB3F0E 44447344 IC50 = 53 nM T68251 C6WSC7 44447346 IC50 = 52 nM T68251 C6MOB0 44447348 IC50 = 549 nM T68251 CM7JV0 44447353 IC50 = 13 nM T68251 CY2XR5 44447363 IC50 = 1400 nM T68251 CU2BC6 44447364 IC50 > 10000 nM T68251 CXS34M 44447371 IC50 = 262 nM T68251 CD8RX4 44447437 IC50 > 2000 nM T68251 CLNK98 44447442 IC50 > 2000 nM T68251 CA5J9Q 44454525 IC50 > 10000 nM T68251 C6L1OH 44454554 IC50 = 283 nM T68251 CHTY64 44454555 IC50 = 297 nM T68251 CLNM62 44454612 IC50 = 247 nM T68251 CZ2QY4 44454641 IC50 = 344 nM T68251 C7DIB0 44454661 IC50 = 401 nM T68251 CTR91D 44454664 IC50 = 582 nM T68251 CR3PO9 44454741 IC50 = 1262 nM T68251 C1ZSK0 44454742 IC50 = 286 nM T68251 CM8AG1 44454790 IC50 = 2917 nM T68251 CCH42M 44454856 IC50 = 893 nM T68251 CQG09B 44454861 IC50 = 61 nM T68251 CQ5YK3 44454864 IC50 = 73 nM T68251 CLG57Z 44454888 IC50 = 2317 nM T68251 CMEJ96 44454891 IC50 = 147 nM T68251 CV07DO 44455123 IC50 = 4591 nM T68251 C9MHD2 44455124 IC50 = 108.4 nM T68251 C2L1VK 44455161 IC50 = 5.7 nM T68251 C4CZ7N 44455196 IC50 = 4.9 nM T68251 CZ15QG 44455197 IC50 = 104.5 nM T68251 CJ6L1K 44455200 IC50 = 1.7 nM T68251 CLK5O7 44455240 IC50 = 6.1 nM T68251 CSKN69 44455242 IC50 = 5 nM T68251 C3U9VM 44455265 IC50 = 22.4 nM T68251 CG65TZ 44455266 IC50 = 6.5 nM T68251 C14QTI 44455267 IC50 = 41 nM T68251 CSX4F2 44455294 IC50 = 6.1 nM T68251 CJ29BT 44455298 IC50 = 66.4 nM T68251 CCK15P 44455331 IC50 = 66.2 nM T68251 CW8IB7 44455332 IC50 = 662 nM T68251 C9ZXF4 44455360 IC50 = 242 nM T68251 CFB78A 44455363 IC50 > 1000 nM T68251 CW46RV 44455498 Ki = 1500 nM T68251 CXNP45 44455499 Ki = 2733 nM T68251 C6CED5 44455528 Ki > 3333 nM T68251 CUQH30 44455553 Ki = 1700 nM T68251 C83KYJ 44455582 Ki > 3333 nM T68251 CK5N1S 44455612 Ki > 3333 nM T68251 CU2E7V 44455613 Ki > 3333 nM T68251 CH1DI4 44455614 Ki > 3333 nM T68251 CFQ79A 44455647 Ki > 3333 nM T68251 C3J1SV 44455676 IC50 = 36.8 nM T68251 CS6HL1 44455704 IC50 > 1000 nM T68251 CR4EX3 44455706 IC50 > 1000 nM T68251 CC01WS 44455737 IC50 = 377 nM T68251 C0R9SH 44455760 IC50 = 167.5 nM T68251 C6FV2Z 44455783 Ki > 3333 nM T68251 C7W6XV 44455786 IC50 = 72 nM T68251 CO58GJ 44455787 IC50 = 184 nM T68251 CPYV60 44455807 Ki = 2633 nM T68251 CLAT19 44455811 IC50 > 1000 nM T68251 C3TS1X 44455813 IC50 = 10.6 nM T68251 C92AFN 44455816 IC50 = 84.5 nM T68251 CGA0T4 44455829 Ki > 3333 nM T68251 CIR06N 44455835 IC50 = 16.7 nM T68251 C38VBL 44455836 IC50 = 17.2 nM T68251 CKB6E7 44455837 IC50 = 468 nM T68251 CV2B4N 44455858 Ki > 3333 nM T68251 CL6UY9 44455865 IC50 > 1000 nM T68251 CVR58Q 44455879 Ki > 3333 nM T68251 CWZ8K6 44455880 Ki > 3333 nM T68251 CEN93Y 44460382 Ki > 10000 nM T68251 CL30OP 44460588 Ki = 220 nM T68251 C0A1KH 44460605 Ki = 77 nM T68251 CDN1V6 44460606 Ki = 110 nM T68251 CJ6PN3 44460646 Ki = 11 nM T68251 CU8A1O 44460672 Ki = 6100 nM T68251 CIQ87B 44460676 Ki = 4840 nM T68251 C5B8NZ 44460690 Ki = 12 nM T68251 CK4WU2 44460737 Ki = 130 nM T68251 CG0Z7I 44478924 IC50 = 1300 nM T68251 CFO27Y 44478926 IC50 = 230 nM T68251 CBZJ29 44478927 IC50 = 9.7 nM T68251 CRJ24K 44479197 IC50 = 7 nM T68251 CGOH82 44479198 IC50 = 710 nM T68251 CLV56M 44479199 IC50 = 47 nM T68251 CY92OQ 44479458 IC50 = 9900 nM T68251 CH1QG9 44479459 IC50 = 100 nM T68251 CB1NT7 44479460 IC50 = 38 nM T68251 C0JQ9L 44479699 IC50 = 73 nM T68251 C0DN1Q 44479700 IC50 = 58000 nM T68251 CTG24W 44479702 IC50 = 2400 nM T68251 CGZ49M 44479703 IC50 = 190 nM T68251 CAK94X 44563337 IC50 = 193 nM T68251 CSH4K3 44563364 IC50 = 10000 nM T68251 CAF95R 44563365 IC50 = 10000 nM T68251 CO4FQ1 44563366 IC50 = 10000 nM T68251 C6WA3X 44563401 IC50 = 10000 nM T68251 CX5L7N 44563402 IC50 = 24 nM T68251 CJ8V4U 44563403 IC50 = 18 nM T68251 CN2BM4 44563404 IC50 = 100 nM T68251 C3KCV6 44563405 IC50 = 740 nM T68251 CI0R5M 44563465 IC50 = 310 nM T68251 C5IQ9Z 44563466 IC50 = 320 nM T68251 C6ZEW9 44563467 IC50 = 1400 nM T68251 CZ2EL1 44563468 IC50 = 300 nM T68251 CDV6R7 44563469 IC50 = 92 nM T68251 CJ2BU5 44563487 IC50 = 37 nM T68251 CP54WT 44563489 IC50 = 1813 nM T68251 C1UXP6 44563490 IC50 = 310 nM T68251 CZ0W1A 44563491 IC50 = 1273 nM T68251 C37UAM 44563492 IC50 = 65 nM T68251 C4BD0N 44563493 IC50 = 247 nM T68251 CNP6M7 44563494 IC50 = 45 nM T68251 C0J6LB 44563970 IC50 = 2600 nM T68251 CR6NO2 44564180 IC50 = 6 nM T68251 C3US0I 44569010 IC50 = 3200 nM T68251 C3TAN1 44569011 IC50 = 2200 nM T68251 CF0L2W 44569012 IC50 = 50 nM T68251 CGI35S 44569013 IC50 = 200 nM T68251 C8PO5Q 44569024 IC50 = 40 nM T68251 C52JXP 44569036 IC50 = 3500 nM T68251 CU1NI6 44569037 IC50 = 2700 nM T68251 CS9CH4 44569038 IC50 = 40 nM T68251 C63ZQK 44569039 IC50 = 10 nM T68251 C2WE7H 44569040 IC50 = 1300 nM T68251 CO8FB4 44569058 IC50 = 90 nM T68251 C3K4ED 44569059 IC50 = 5200 nM T68251 CPWR76 44569060 IC50 = 1500 nM T68251 CU39FK 44569061 IC50 = 200 nM T68251 CR6H0X 44569062 IC50 = 700 nM T68251 CTWR37 44569063 IC50 = 8900 nM T68251 C6M9SH 44569081 IC50 = 500 nM T68251 C5RN7U 44569082 IC50 = 4 nM T68251 CQ9OA7 44569083 IC50 = 20 nM T68251 C70UVG 44571513 IC50 = 50500 nM T68251 CCV74H 44576563 IC50 = 400 nM T68251 C59TCG 44576564 IC50 = 2000 nM T68251 CMI9S4 44576565 IC50 = 9500 nM T68251 CD8ZI4 44576587 IC50 = 100 nM T68251 CQ87CS 44576614 IC50 = 200 nM T68251 CJY2W3 44576615 IC50 = 300 nM T68251 CL92CH 44576616 IC50 = 200 nM T68251 CIU84E 44576617 IC50 = 1100 nM T68251 C9ODS1 44576618 IC50 = 1500 nM T68251 C35DWL 44576631 IC50 = 6 nM T68251 C6ZL1U 44576632 IC50 = 8 nM T68251 CK09LV 44576633 IC50 = 8 nM T68251 CFL76T 44576634 IC50 = 11 nM T68251 CC58GQ 44576635 IC50 = 12 nM T68251 CPT42K 44580109 IC50 > 5000 nM T68251 CQ7W5I 44580110 Ki > 3000 nM T68251 CWD32S 44580184 IC50 = 664 nM T68251 CQ4ZR1 44580422 IC50 = 750 nM T68251 C0XJ5C 44580496 Ki > 3333 nM T68251 CK68GT 44580539 Ki = 1.37 nM T68251 CXIY57 44580801 Ki > 10000000 nM T68251 C0OA8Y 44580802 Ki > 10000000 nM T68251 CNC4D7 44581071 Ki = 7000000 nM T68251 CDF48U 44581111 Ki > 10000000 nM T68251 C06BRD 44582547 IC50 = 107200 nM T68251 C51VNE 44582548 IC50 = 287300 nM T68251 CLK3R4 44582549 IC50 = 76800 nM T68251 CZTW24 44582550 IC50 = 52800 nM T68251 CP0AJ7 44582568 IC50 = 59900 nM T68251 CCZ07T 44582586 IC50 = 76100 nM T68251 CN58BM 44582588 IC50 = 71200 nM T68251 C3UJ2Q 44582621 IC50 = 659600 nM T68251 C35BEJ 44582622 IC50 = 501500 nM T68251 C3UE5R 44582644 IC50 = 116300 nM T68251 CX1GV0 44582645 IC50 = 71400 nM T68251 C3IU2S 44582646 IC50 = 64300 nM T68251 C63ODU 44582647 IC50 = 120800 nM T68251 C7EAZ1 44582685 IC50 = 235800 nM T68251 CZW4O6 44582686 IC50 = 159100 nM T68251 C3AX6W 44582687 IC50 = 211400 nM T68251 CC0LO7 44582688 IC50 = 283600 nM T68251 CX63IA 44582689 IC50 = 256100 nM T68251 CL73BH 44582717 IC50 = 79600 nM T68251 CY2PM8 44582718 IC50 = 83200 nM T68251 C9EPQ6 44582719 IC50 = 76800 nM T68251 CF1G7I 44582720 IC50 = 101500 nM T68251 C15RUQ 44582746 IC50 = 76500 nM T68251 C3CJD0 44582747 IC50 = 397600 nM T68251 C16RAH 44582748 IC50 = 368100 nM T68251 CQ9XG5 44582769 IC50 = 470600 nM T68251 C7UTR1 44582771 IC50 = 470700 nM T68251 CE2D6Z 44582793 IC50 = 340800 nM T68251 CUR8M1 44582868 IC50 = 55300 nM T68251 CNK9C7 44582869 IC50 = 628000 nM T68251 CX49HN 44582873 IC50 = 369400 nM T68251 C56WPA 44582874 IC50 = 169400 nM T68251 C8TGB1 44582875 IC50 = 114900 nM T68251 CYV0N5 44582876 IC50 = 26100 nM T68251 CR4SF2 44582887 IC50 = 52300 nM T68251 C50OTD 44582888 IC50 = 54400 nM T68251 CDX63O 44582890 IC50 = 33600 nM T68251 C6X0FM 44582904 IC50 = 71200 nM T68251 CY3N7I 44582905 IC50 = 86300 nM T68251 CY4A6F 44582906 IC50 = 108700 nM T68251 CD0J5R 44582907 IC50 = 122400 nM T68251 C2Z4HB 44583600 IC50 = 1277 nM T68251 CD4Q8C 44583601 IC50 = 8 nM T68251 CD2AQ7 44583620 IC50 = 92 nM T68251 CLZ6X5 44583621 IC50 = 81 nM T68251 C5HA4P 44583622 IC50 = 180 nM T68251 C7PR8I 44583623 IC50 = 106 nM T68251 CDRC42 44583654 IC50 = 100 nM T68251 C5HEX6 44583655 IC50 = 1090 nM T68251 CM79HD 44583656 IC50 > 5000 nM T68251 C20FCM 44583672 IC50 > 5000 nM T68251 CLAU98 44586492 IC50 = 8760 nM T68251 CY8X7P 44586493 IC50 = 2930 nM T68251 CDS86C 44586529 IC50 = 3140 nM T68251 COD20L 44586530 IC50 = 12700 nM T68251 C1W2SV 44586531 IC50 = 17800 nM T68251 C5S0OJ 44586532 IC50 = 50500 nM T68251 CB2P7I 44586533 IC50 = 7480 nM T68251 CKRT49 44586578 IC50 = 19200 nM T68251 C8XY1Z 44586579 IC50 = 13100 nM T68251 CE9BZ5 44586580 IC50 = 25500 nM T68251 CXDF71 44586581 IC50 = 14300 nM T68251 COFY06 44586582 IC50 = 8080 nM T68251 CI2PT3 44586626 IC50 = 8000 nM T68251 C4GQ6Y 44586627 IC50 = 12600 nM T68251 CTO94B 44586628 IC50 = 3540 nM T68251 C9Y0CR 44586662 IC50 = 11700 nM T68251 CBV5P8 44586663 IC50 = 32000 nM T68251 C2U0CY 44586664 IC50 = 9940 nM T68251 C1IBA2 44588219 IC50 = 151400 nM T68251 C6XE5V 44588251 IC50 = 771900 nM T68251 C1UW6M 44588252 IC50 = 802300 nM T68251 CXF40R 44588253 IC50 = 78800 nM T68251 CQF2I5 44588254 IC50 = 546800 nM T68251 CBA1Y8 44588279 IC50 > 1000000 nM T68251 C8RI4Q 44591819 IC50 = 30000 nM T68251 C6BXS2 44591880 IC50 = 37700 nM T68251 CM9IN6 44592481 IC50 = 14400 nM T68251 CZNQ90 44593458 IC50 = 9 nM T68251 CR3Q4N 44593532 IC50 = 7100 nM T68251 CH8QS0 44596287 IC50 = 128 nM T68251 CTW7F2 44601281 IC50 = 1.6 nM T68251 CW5A2D 44608129 IC50 = 86 nM T68251 CT7KX5 44608938 IC50 = 96 nM T68251 CJRP30 44608939 IC50 = 458 nM T68251 COI5K3 44608942 IC50 = 706 nM T68251 CS4C5T 44609098 IC50 = 200 nM T68251 CMLV87 44609099 IC50 = 706 nM T68251 C3T9SV 44609100 IC50 = 54 nM T68251 C19LWR 44634267 IC50 = 0.13 nM T68251 CM0I4J 45101511 IC50 = 1475 nM T68251 CZP79X 45268488 IC50 = 379 nM T68251 CK50JB 45268522 IC50 = 8990 nM T68251 C2B0GI 45268787 Ki = 1 nM T68251 CVG5I2 45269378 IC50 = 4000 nM T68251 CQC5Y4 45269386 IC50 = 2840 nM T68251 CACH13 45269631 IC50 = 12 nM T68251 CTOH60 45270200 IC50 = 4410 nM T68251 C2H5IY 45271017 IC50 = 3590 nM T68251 C0YT8W 45271893 IC50 = 1150 nM T68251 CVNO86 45271894 IC50 = 1410 nM T68251 C7OQB3 45271912 IC50 = 2470 nM T68251 C3SWC7 45272759 IC50 = 7500 nM T68251 CH4NL1 45376336 IC50 = 1937.23 nM T68251 C36HRP 45377138 IC50 > 22000 nM T68251 C6B7ZY 45377564 IC50 > 500000 nM T68251 C5HAR6 45377565 IC50 > 20000 nM T68251 CKR0Q8 45377703 IC50 > 24000 nM T68251 C3SQL2 45378250 IC50 = 190 nM T68251 CQE49A 45378251 IC50 = 1.5 nM T68251 CO4AC6 45378252 IC50 = 17 nM T68251 C42FPG 45378253 IC50 = 4.2 nM T68251 CI82BN 45378254 IC50 = 21 nM T68251 C6MY2W 45380188 IC50 = 190 nM T68251 C9P0DG 45380189 IC50 = 29 nM T68251 CRY0E8 45380190 IC50 = 0.7 nM T68251 C0MPH3 45380191 IC50 = 390 nM T68251 CMPE63 45482676 IC50 = 1500 nM T68251 CZS39O 45487302 IC50 = 210 nM T68251 C4ZWY7 45487310 IC50 = 432 nM T68251 C9SV0H 45487311 IC50 = 581 nM T68251 C6GCM7 45487332 IC50 < 5 nM T68251 CCF05Q 45487333 IC50 = 102 nM T68251 C23NRD 45487334 IC50 > 2000 nM T68251 CY09ZU 45487335 IC50 = 344 nM T68251 CQHJ85 45487342 IC50 = 11 nM T68251 C3ZLN1 45487343 IC50 = 12 nM T68251 CI6DW2 45487357 IC50 < 5 nM T68251 COX40Y 45487358 IC50 = 102 nM T68251 CF1T7M 45487359 IC50 = 843 nM T68251 CRXI29 45487373 IC50 > 2000 nM T68251 CYL32E 45487376 IC50 = 235 nM T68251 CO5P9I 45487386 IC50 = 506 nM T68251 CS9Y8G 45487387 IC50 > 2000 nM T68251 CAN4J2 45487388 IC50 = 1662 nM T68251 CWLC18 45487393 IC50 = 471 nM T68251 CO9NJ2 45487398 IC50 = 365 nM T68251 CDN5Q6 45487399 IC50 = 502 nM T68251 CI4KJ5 45487400 IC50 = 613 nM T68251 C49HOI 45487401 IC50 = 730 nM T68251 CBK43U 45487402 IC50 < 5 nM T68251 C56WVI 46184724 Ki > 50000 nM T68251 CMB53L 46212112 IC50 = 159390 nM T68251 CX58KQ 46212114 IC50 = 58220 nM T68251 C9PXD0 46212116 IC50 = 17170 nM T68251 C6KHO2 46212117 IC50 = 36040 nM T68251 C9XGD0 46212861 IC50 = 187410 nM T68251 CLWA85 46228171 IC50 > 1000000 nM T68251 CFQ67J 46228182 IC50 > 1000000 nM T68251 CCV7T2 46228183 IC50 > 1000000 nM T68251 CU2WI8 46228191 IC50 > 1000000 nM T68251 CT6JZ9 46228192 IC50 = 594300 nM T68251 C6H7AB 46228205 IC50 = 999000 nM T68251 CJ9SD0 46228215 IC50 = 447200 nM T68251 C7WS9P 46228222 IC50 > 1000000 nM T68251 C71RSJ 46228223 IC50 > 1000000 nM T68251 CKCE97 46228233 IC50 > 1000000 nM T68251 CWUG47 46228234 IC50 = 324400 nM T68251 CM3YZ1 46228235 IC50 > 1000000 nM T68251 CYUM78 46228241 IC50 > 1000000 nM T68251 C6HCD2 46228242 IC50 > 1000000 nM T68251 C0GX8M 46228245 IC50 > 1000000 nM T68251 C9FM5N 46228246 IC50 = 176500 nM T68251 C4KA1Y 46228247 IC50 > 1000000 nM T68251 C7HIE4 46228248 IC50 = 131000 nM T68251 CQVZ58 46228249 IC50 > 1000000 nM T68251 C5WV8N 46228250 IC50 > 1000000 nM T68251 CR0BP8 46228264 IC50 > 1000000 nM T68251 CGW3Q4 46228265 IC50 > 1000000 nM T68251 CVN7J0 46228266 IC50 = 166600 nM T68251 C51LDC 46228283 IC50 > 1000000 nM T68251 C2JVF4 46228308 IC50 = 196600 nM T68251 C7Z6XB 46228317 IC50 > 1000000 nM T68251 C0S8FV 46231953 IC50 = 400 nM T68251 CN3OS2 46232362 IC50 = 6460800 nM T68251 CF9D2G 46232363 IC50 = 124320 nM T68251 C5GT8X 46232364 IC50 = 624480 nM T68251 C9A8BO 46232365 IC50 = 2000000 nM T68251 CP49KE 46232415 IC50 = 24180 nM T68251 CFZX82 46232416 IC50 = 26170 nM T68251 C3L7VK 46232417 IC50 = 1362800 nM T68251 C4XOU1 46232418 IC50 = 56600 nM T68251 C1S8BQ 46232490 IC50 = 106000 nM T68251 CAV06U 46232491 IC50 = 105300 nM T68251 CVF9D5 46232492 IC50 = 9426500 nM T68251 C18JTQ 46232493 IC50 = 1750000 nM T68251 CFA58J 46232533 IC50 = 2757800 nM T68251 C9C7IE 46232534 IC50 = 11520000 nM T68251 CFU05P 46232535 IC50 = 1920500 nM T68251 CSU81E 46233057 IC50 = 58140 nM T68251 C8SM5H 46233058 IC50 = 30050 nM T68251 C8W7RP 46233059 IC50 = 10490 nM T68251 C3IA9P 46233060 IC50 = 37290 nM T68251 CZ6C8P 46703060 IC50 = 5.97 nM T68251 C0DHL4 46703061 IC50 = 1721.82 nM T68251 CYA45K 46703062 IC50 = 3.55 nM T68251 CY72WL 46703063 IC50 = 5.27 nM T68251 C1YHS2 46703064 IC50 = 1679.56 nM T68251 C8HX7K 46840956 IC50 = 45820 nM T68251 CH0Z1E 46844314 Ki = 1208 nM T68251 C8MR0H 46847340 IC50 = 4000 nM T68251 C20BTY 46856241 Ki = 43600 nM T68251 C0ECU2 46861775 IC50 = 8.95 nM T68251 C0Y9NZ 46861793 IC50 = 8.31 nM T68251 C2S4YC 46866644 IC50 = 15000 nM T68251 C7QR8Y 46866645 IC50 = 10000 nM T68251 CUH07J 46866646 IC50 = 7000 nM T68251 C8GK4C 46866647 IC50 = 4000 nM T68251 C5L8GF 46871738 IC50 = 12.1 nM T68251 CR1KF7 46871739 IC50 = 3.7 nM T68251 C8Q6YR 46871740 IC50 = 5.3 nM T68251 C58YSM 46871741 IC50 = 6000 nM T68251 C3X5EN 46873064 IC50 = 53670 nM T68251 CR96AK 46890762 IC50 > 10000 nM T68251 C5G9FX 46890763 IC50 = 1400 nM T68251 COP78K 46890764 IC50 = 4500 nM T68251 C60QSB 46890765 IC50 = 1600 nM T68251 CQ5P9V 46890766 IC50 = 700 nM T68251 CB90YN 46890767 IC50 = 5600 nM T68251 CUA7L6 46890821 IC50 = 3600 nM T68251 C9BNQ7 46890822 IC50 = 1600 nM T68251 CTF20Y 46890823 IC50 = 1750 nM T68251 CR3QW7 46891107 IC50 = 21.1 nM T68251 C5MK3A 46891108 IC50 = 88 nM T68251 CQ5E1H 46891109 IC50 = 40 nM T68251 C0NW9D 46891110 IC50 = 370 nM T68251 C91LGI 46891170 IC50 = 48.5 nM T68251 CGI5B4 46891171 IC50 = 330 nM T68251 CZPM12 46891172 IC50 = 18.4 nM T68251 C2V6MW 46891173 IC50 = 35 nM T68251 CZWT45 46891207 IC50 = 1400 nM T68251 CFE58Q 46891208 IC50 = 5.4 nM T68251 C8S7QX 46891209 IC50 = 32.6 nM T68251 C5Y0MN 46891255 IC50 = 3700 nM T68251 CJ16SE 46891256 IC50 = 2 nM T68251 C7Y9TE 46891257 IC50 = 82 nM T68251 C7DT6W 46891258 IC50 = 700 nM T68251 CLF7Y4 46891311 IC50 = 900 nM T68251 C2IN7Y 46891312 IC50 = 3100 nM T68251 CNXU57 46891313 IC50 = 70 nM T68251 CJB5D0 46891314 IC50 = 5400 nM T68251 CVK0E5 46891356 IC50 = 500 nM T68251 C89RPO 46891357 IC50 = 505 nM T68251 CVB6K4 46891358 IC50 = 1750 nM T68251 C67WEK 46891359 IC50 = 800 nM T68251 CPQ37V 46891414 IC50 > 10000 nM T68251 C5LTI6 46891459 IC50 = 2900 nM T68251 C92FBL 46891460 IC50 = 2100 nM T68251 C1A0OE 46891522 IC50 = 2100 nM T68251 C2I6FV 46891523 IC50 = 2400 nM T68251 CAZ9Q5 46891524 IC50 = 7300 nM T68251 CG02KB 46891525 IC50 = 1700 nM T68251 C7ZG8J 46891526 IC50 > 10000 nM T68251 CRQ13J 46891580 IC50 = 2500 nM T68251 CERM39 46891581 IC50 = 5500 nM T68251 CN8WF9 46891582 IC50 = 7000 nM T68251 C86RLM 46891583 IC50 = 900 nM T68251 CM7S5T 46891584 IC50 = 6000 nM T68251 CRY18A 46891617 IC50 = 900 nM T68251 C0F7SU 46905989 IC50 = 112000 nM T68251 C49PYF 46907509 IC50 = 8.92 nM T68251 C2U1GW 46907510 IC50 = 9.11 nM T68251 C7MUS8 46907512 IC50 = 1820.53 nM T68251 C71YRF 46907513 IC50 = 1873.02 nM T68251 CVH58U 46907580 IC50 = 8.3 nM T68251 C0S9WB 46919610 Ki = 1900 nM T68251 CXDL74 46927871 IC50 = 8270 nM T68251 CE3H7I 46938726 IC50 < 0.1 nM T68251 C9T0HR 46938727 IC50 < 0.1 nM T68251 C0YR7M 46938728 IC50 < 0.1 nM T68251 C2TE8J 47162079 IC50 = 60000 nM T68251 CC42DK 49863560 IC50 = 129000 nM T68251 C4UWB6 49863561 IC50 = 18500 nM T68251 CMR3B0 49863562 IC50 = 121000 nM T68251 CBE6H5 49863563 IC50 = 127000 nM T68251 CR0I9V 49863564 IC50 = 12000 nM T68251 CD17YP 49863589 IC50 = 272000 nM T68251 CXW4C6 49863590 IC50 = 107000 nM T68251 C1B6ZU 49863591 IC50 = 155000 nM T68251 C0S2OT 49863592 IC50 > 1000000 nM T68251 CT3W2H 49863593 IC50 > 1000000 nM T68251 CG96WY 49863619 IC50 = 22700 nM T68251 CG40UX 49863620 IC50 = 315650 nM T68251 C0IX5P 49863621 IC50 > 1000000 nM T68251 CSC7K2 49863622 IC50 = 141000 nM T68251 C1FLD5 49863915 IC50 = 122000 nM T68251 CL90XE 49863932 IC50 > 1000000 nM T68251 CXZ8Y3 49863933 IC50 = 60400 nM T68251 CKXZ37 49863934 IC50 = 62700 nM T68251 CFD6O0 49863953 IC50 = 71600 nM T68251 C1L6TV 49863954 IC50 = 131000 nM T68251 CEL71O 49863955 IC50 = 46900 nM T68251 CJB0T7 49863956 IC50 = 454000 nM T68251 C7S9QA 50913428 IC50 > 500000 nM T68251 CO4XE9 50913573 IC50 > 500000 nM T68251 C2T1AZ 50925490 IC50 = 3000 nM T68251 CJG7H2 50941564 IC50 = 8800 nM T68251 C5B6SP 50941565 IC50 = 7200 nM T68251 CV4BM3 50941566 IC50 = 10800 nM T68251 C29WVD 50941567 IC50 = 8400 nM T68251 CKN8Z0 50941568 IC50 = 5600 nM T68251 CQ64FL 50941569 IC50 = 3900 nM T68251 CC4V0N 50941747 IC50 = 4300 nM T68251 C7AU4S 50943150 IC50 > 100000 nM T68251 CXF4V3 50990921 IC50 > 6300 nM T68251 CAS94N 51346773 Ki = 390 nM T68251 CP65WT 51346774 Ki = 90 nM T68251 C5OIA2 51346775 Ki = 280 nM T68251 CU2SX3 51355576 Ki > 10000 nM T68251 CQM4E7 52936345 IC50 = 19 ug.mL-1 T68251 CLA96C 53232689 Ki = 400 nM T68251 C3BGW0 53233015 Ki = 20500 nM T68251 CZ06OY 53233469 IC50 = 360 nM T68251 CMQZ70 53242178 IC50 > 23000 nM T68251 CC9HK5 53245646 IC50 = 6309.57 nM T68251 CRI92N 53311230 IC50 > 10000 nM T68251 C74CKF 53318123 Ki = 61 nM T68251 C47DIU 53318911 IC50 = 120 nM T68251 CC6DR2 53318912 IC50 = 4200 nM T68251 C7V1NC 53320225 IC50 = 350 nM T68251 CVH2B7 53320226 IC50 = 2800 nM T68251 CO8QK2 53320227 IC50 = 180 nM T68251 CNS3F2 53321542 IC50 = 1900 nM T68251 C4UE6R 53322469 IC50 = 30000 nM T68251 C1N2BX 53322876 IC50 = 1700 nM T68251 CSYW40 53322877 IC50 = 35000 nM T68251 CGUC59 53322878 IC50 = 2400 nM T68251 C3QHA6 53322879 IC50 = 2200 nM T68251 CI3WL5 53323418 Ki = 240 nM T68251 C0H7FQ 53324260 IC50 = 26000 nM T68251 CU7YG9 53325497 IC50 = 170 nM T68251 C4G1HK 53325498 IC50 > 9100 nM T68251 CO5L1I 53325499 IC50 = 12000 nM T68251 CZA03W 53326760 IC50 = 530 nM T68251 CM53CG 53326761 IC50 = 2500 nM T68251 CWR6T4 53326860 IC50 = 500 nM T68251 CPY02U 53327890 IC50 = 2.3 nM T68251 CPGE80 53327891 IC50 = 6 nM T68251 CLJ4G2 53328858 IC50 = 1.5 nM T68251 C4G3QL 53328859 IC50 = 2.5 nM T68251 CX1TW0 53328860 IC50 = 1.3 nM T68251 C0ZX5G 53329215 IC50 = 4 nM T68251 CSU52A 53329216 IC50 = 17 nM T68251 CHF62Q 53361485 IC50 = 140 nM T68251 CJ3F4R 53361486 IC50 = 37 nM T68251 C6Y2EV 53374826 IC50 > 100000 nM T68251 CNY03Z 53378637 Ki = 440 nM T68251 CX3DU4 53378973 Ki = 390 nM T68251 CTD1H9 53378974 Ki = 240 nM T68251 CQ04KO 53389286 IC50 = 384 nM T68251 C1IFJ8 53957122 IC50 = 210000 nM T68251 CTJ48R 54185618 IC50 = 17800 nM T68251 C24SIM 54334252 IC50 = 39 nM T68251 CSUW40 54352406 IC50 = 10 nM T68251 C7RC3A 54371779 IC50 = 10 nM T68251 C3M8GZ 54580051 IC50 = 61000 nM T68251 CL0WM9 54580052 IC50 > 10000 nM T68251 CK26XF 54580053 IC50 > 10000 nM T68251 C3LF0P 54580544 Ki = 9200 nM T68251 CA8U9V 54580837 IC50 = 4000 nM T68251 CVO09J 54581546 Ki = 110 nM T68251 CWB2Q6 54581896 IC50 = 170 nM T68251 CVK72M 54582073 IC50 = 1300 nM T68251 CBK18O 54582074 IC50 > 10000 nM T68251 CP2F1B 54582075 IC50 > 10000 nM T68251 CZNU23 54582076 IC50 > 10000 nM T68251 C0U5HZ 54582077 IC50 > 10000 nM T68251 C8SG9Y 54582079 IC50 > 10000 nM T68251 CZI6S3 54582080 IC50 = 3500 nM T68251 CD09BZ 54582543 IC50 = 1300 nM T68251 CH6Q2Z 54583016 IC50 > 10000 nM T68251 C3V9LQ 54583017 IC50 = 150 nM T68251 CT80KQ 54583018 IC50 = 620 nM T68251 CPT4L5 54583019 IC50 > 10000 nM T68251 CK52YD 54583511 Ki = 530 nM T68251 CF0SK8 54583712 IC50 = 2.5 nM T68251 CBEV27 54584024 IC50 = 3300 nM T68251 CM87DP 54584025 IC50 = 1100 nM T68251 C28GKQ 54585927 IC50 > 10000 nM T68251 CAZ76E 54586892 IC50 > 10000 nM T68251 CM0OQ3 54586893 IC50 > 10000 nM T68251 CK1NS7 54586894 IC50 > 10000 nM T68251 CMC4Y1 54586895 IC50 > 10000 nM T68251 C2MKX5 54586896 IC50 = 3800 nM T68251 CU91QP 54586897 IC50 > 10000 nM T68251 CI08RQ 54586898 IC50 = 1400 nM T68251 C6PRI4 54586899 IC50 = 7600 nM T68251 CG37UX 54587429 Ki = 430 nM T68251 CL9SC3 54587769 Ki > 40000 nM T68251 C13FSJ 54669762 Ki = 24 nM T68251 CHS01Z 54669766 Ki = 520 nM T68251 C8YLA4 54669829 IC50 = 7.5 nM T68251 C1KA8X 54669830 IC50 = 2.55 nM T68251 CZA6Q9 54669831 IC50 = 24 nM T68251 CF23NJ 54669841 IC50 = 23 nM T68251 C71KLJ 54679182 IC50 = 1260 nM T68251 CC67RV 54681831 IC50 = 610 nM T68251 C83NUI 54687474 IC50 = 9300 nM T68251 CZ6V0U 54724681 IC50 > 50000 nM T68251 CJ6HT4 54726662 IC50 = 19000 nM T68251 C9P5ES 54752445 IC50 = 0.39 nM T68251 C0HKC9 54752446 IC50 = 0.57 nM T68251 C6D9IE 54753443 IC50 = 1729.19 nM T68251 CLP2C1 54753981 IC50 = 393140 nM T68251 CQD2Z6 54757100 IC50 = 63.6 nM T68251 C7E9SG 54757202 Ki = 78000 nM T68251 CMJ90D 54757404 Ki = 62 nM T68251 CD1A3F 54757406 Ki = 69 nM T68251 C4EFI5 54757409 Ki = 420 nM T68251 C5D1TI 56649332 IC50 = 1.8 nM T68251 CGTV56 56658262 IC50 = 151600 nM T68251 C9Z4TW 56658263 IC50 = 110100 nM T68251 CAV9S4 56658410 IC50 = 42200 nM T68251 CLKA98 56659256 IC50 = 73 nM T68251 CAFN81 56659257 IC50 = 269 nM T68251 C5ATG7 56659258 IC50 = 95 nM T68251 CR0HX7 56659259 IC50 = 25 nM T68251 CI8RY0 56659946 IC50 = 249240 nM T68251 C0NK1P 56659952 IC50 = 307270 nM T68251 CL6GF3 56659954 IC50 = 166110 nM T68251 CP5K7G 56661758 IC50 = 100100 nM T68251 C1EW4P 56661759 IC50 = 105600 nM T68251 C5FR4E 56661895 IC50 = 119500 nM T68251 CG7E1O 56662736 IC50 = 13 nM T68251 CZF86Q 56662737 IC50 = 264 nM T68251 CT2G8L 56662738 IC50 = 24 nM T68251 C3LQY5 56662739 IC50 = 31 nM T68251 CQY15M 56663413 IC50 = 463380 nM T68251 CWM2L3 56663417 IC50 = 836490 nM T68251 C48JHP 56663421 IC50 = 267730 nM T68251 CIG9J2 56663694 IC50 = 1021 nM T68251 C8YPU6 56665194 IC50 = 84300 nM T68251 CV46HL 56665195 IC50 = 173100 nM T68251 C3L5SO 56665196 IC50 = 108900 nM T68251 CH4M6V 56665197 IC50 = 40600 nM T68251 C20IZG 56665371 IC50 > 1000000 nM T68251 C8ZD7Q 56666204 IC50 = 45 nM T68251 CKB12J 56666205 IC50 = 54 nM T68251 CR21IL 56666206 IC50 = 100 nM T68251 CT65HD 56666207 IC50 = 311 nM T68251 C2IVE9 56666208 IC50 = 706 nM T68251 CPM8U1 56666842 IC50 = 540030 nM T68251 CC8HS0 56669604 IC50 = 9.8 nM T68251 CLO80F 56669605 IC50 = 60 nM T68251 CPS48C 56669606 IC50 = 329 nM T68251 CGMF96 56669607 IC50 = 47 nM T68251 CG0N1D 56670269 IC50 = 251910 nM T68251 CD1UX2 56670273 IC50 = 276440 nM T68251 C6O4TD 56672133 IC50 > 1000000 nM T68251 CRZF93 56672134 IC50 = 157400 nM T68251 C5C3OA 56672135 IC50 = 149200 nM T68251 CSU81T 56672275 IC50 = 133800 nM T68251 CBX8M4 56673120 IC50 = 15 nM T68251 C6Z7VA 56673121 IC50 = 86 nM T68251 C2YJZ8 56673122 IC50 = 2.9 nM T68251 C3BD9S 56673123 IC50 = 264 nM T68251 CG10FP 56673124 IC50 = 681 nM T68251 CMNQ68 56673125 IC50 = 20 nM T68251 CY80GQ 56673788 IC50 = 656770 nM T68251 C8C3QL 56675664 IC50 = 111300 nM T68251 CWI28X 56676443 IC50 = 16 nM T68251 CSPX53 56676444 IC50 = 22 nM T68251 CJU1M7 56676445 IC50 = 16 nM T68251 CGD90C 56676446 IC50 = 268 nM T68251 CCA39I 56676447 IC50 = 83 nM T68251 CL67JD 56677116 IC50 = 516830 nM T68251 CWH5R6 56677118 IC50 = 939570 nM T68251 CX80RM 56677120 IC50 = 157420 nM T68251 CKLQ67 56678865 IC50 = 67400 nM T68251 C3ZAX6 56678866 IC50 = 44100 nM T68251 C2M1TR 56678867 IC50 = 119300 nM T68251 CNE08Y 56678974 IC50 = 40400 nM T68251 C7G9AH 56678975 IC50 = 94000 nM T68251 C02GOU 56679764 IC50 = 9.4 nM T68251 CFDR70 56679765 IC50 = 13 nM T68251 CLPF34 56679766 IC50 = 29 nM T68251 C0XP1D 56679767 IC50 = 50 nM T68251 CTE68Z 56679768 IC50 = 30 nM T68251 CES0V3 56679769 IC50 = 411 nM T68251 C0L2JS 56682178 IC50 = 61300 nM T68251 C8UB9G 56682179 IC50 = 83900 nM T68251 C4XL3Y 56682293 IC50 = 86600 nM T68251 CK70XW 56682294 IC50 = 107100 nM T68251 C67VUX 56682295 IC50 = 52700 nM T68251 CIB34L 56683087 IC50 = 10 nM T68251 CM79IH 56683088 IC50 = 1.1 nM T68251 CSL1X7 56683089 IC50 = 104 nM T68251 CSR32E 56683090 IC50 = 86 nM T68251 CWJ65H 56683091 IC50 = 308 nM T68251 CEO93F 56683092 IC50 = 106 nM T68251 CO8FP7 56683093 IC50 = 80 nM T68251 C6KT1Z 56683094 IC50 = 25 nM T68251 CJCI10 56683095 IC50 = 54 nM T68251 C5F7WT 56683096 IC50 = 142 nM T68251 C62FZC 56835063 IC50 = 501 nM T68251 CKJ9S1 56835167 IC50 = 30 nM T68251 C21CLZ 56835168 IC50 = 240 nM T68251 C0L2TS 56835169 IC50 = 1200 nM T68251 CKEV19 56850269 IC50 > 500000 nM T68251 C13DBR 56850270 IC50 > 500000 nM T68251 C05CTJ 56850271 IC50 = 30000 nM T68251 CX8QD5 56850272 IC50 = 310000 nM T68251 C1I9RE 56850407 IC50 > 500000 nM T68251 CVJ90W 56850408 IC50 = 24000 nM T68251 CPI5G0 56850409 IC50 = 83000 nM T68251 C8TH2F 56945850 IC50 = 203 nM T68251 CD72TG 56945851 IC50 = 5 nM T68251 C8J4SC 56945854 IC50 = 64 nM T68251 C1AIZ6 56945963 IC50 = 29 nM T68251 CXQC91 56945964 IC50 = 58 nM T68251 CM4H9D 56945965 IC50 = 44 nM T68251 CUT4S2 56946063 IC50 = 202 nM T68251 C2CQR8 56946064 IC50 = 22 nM T68251 C2H8PG 56946065 IC50 = 13 nM T68251 CW2P6A 56946167 IC50 = 12 nM T68251 CT8S3G 56946168 IC50 = 52 nM T68251 C6LR7O 56964014 IC50 = 328 nM T68251 CE12KU 56964015 IC50 = 158 nM T68251 CL42CX 56964110 IC50 = 219 nM T68251 C0KPD8 57384084 IC50 = 9 nM T68251 CV67JB 57384091 IC50 = 53 nM T68251 C5WFN6 57391082 IC50 = 1 nM T68251 C9BN4F 57391101 IC50 = 7 nM T68251 CI0X9S 57391136 IC50 = 10 nM T68251 CD9J1C 57391201 IC50 > 10000 nM T68251 CN2H9K 57391204 IC50 = 5011.87 nM T68251 CR8MW2 57391205 IC50 = 5011.87 nM T68251 CA25DM 57391224 IC50 = 200 nM T68251 C6P9XK 57391225 IC50 = 144 nM T68251 COT76D 57391411 IC50 > 500000 nM T68251 CJZ0U8 57391412 IC50 > 500000 nM T68251 CAQB32 57391413 IC50 = 4000 nM T68251 CCB9H2 57391414 IC50 = 9 nM T68251 CC57MO 57392866 IC50 = 3.7 nM T68251 C4IWN7 57392867 IC50 = 85 nM T68251 C1ZG3T 57392880 IC50 = 2 nM T68251 CH1I4N 57392901 IC50 = 102 nM T68251 C7CV1B 57392902 IC50 = 6913 nM T68251 C25FAK 57392903 IC50 = 16 nM T68251 C4CK0Q 57392968 IC50 = 7943.28 nM T68251 CNQ9B2 57392969 IC50 = 19952.62 nM T68251 CTYP14 57392972 IC50 = 7943.28 nM T68251 C5VB0U 57392973 IC50 = 6309.57 nM T68251 CMQL31 57392974 IC50 > 10000 nM T68251 C39OHF 57392975 IC50 = 7943.28 nM T68251 CX89EL 57392993 IC50 = 607 nM T68251 C0F3ZD 57393177 IC50 > 500000 nM T68251 CUJD65 57393178 IC50 = 400000 nM T68251 CMB13S 57393179 IC50 = 9000 nM T68251 CJ30LT 57393180 IC50 = 340000 nM T68251 CT2E8Z 57393181 IC50 = 31000 nM T68251 C2O9QP 57394596 IC50 = 2 nM T68251 CN9X5F 57394606 IC50 = 2 nM T68251 CP5BX6 57394607 IC50 = 3.9 nM T68251 CA09RY 57394649 IC50 = 197 nM T68251 CDCW73 57394678 IC50 > 500000 nM T68251 CH6BA3 57394709 IC50 > 10000 nM T68251 CNOH63 57394711 IC50 = 7300 nM T68251 C1CYK9 57394729 IC50 = 25 nM T68251 C9JC3H 57394730 IC50 = 200 nM T68251 C80FML 57394731 IC50 = 111 nM T68251 CYFJ06 57394732 IC50 = 3286 nM T68251 CE5X3D 57394850 IC50 = 10 nM T68251 C82ATC 57394900 IC50 = 3000 nM T68251 C2X8UO 57394901 IC50 > 500000 nM T68251 CN8A6U 57394902 IC50 = 330000 nM T68251 CG43ME 57394903 IC50 = 13 nM T68251 C18PVK 57396348 IC50 > 1000 nM T68251 CM8K2T 57396360 IC50 > 1000 nM T68251 COXA03 57396390 IC50 = 308 nM T68251 CO17CH 57396398 IC50 = 306 nM T68251 CDES09 57396473 IC50 = 1995.26 nM T68251 CONH52 57396474 IC50 = 7943.28 nM T68251 CV51ME 57396475 IC50 = 6309.57 nM T68251 CJB27Z 57396489 IC50 = 81 nM T68251 C34RZI 57396490 IC50 = 178 nM T68251 CD5G3V 57396665 IC50 > 500000 nM T68251 CEB81P 57396666 IC50 > 500000 nM T68251 CMNU14 57396667 IC50 > 500000 nM T68251 CN0LI1 57396668 IC50 = 710 nM T68251 C2MI0H 57398136 IC50 = 1599 nM T68251 C98EXD 57398159 IC50 = 3 nM T68251 C1BIM8 57398160 IC50 = 11 nM T68251 C0KPT7 57398161 IC50 = 2.4 nM T68251 CD6Q9F 57398187 IC50 = 163 nM T68251 CSX81J 57398194 IC50 = 1610 nM T68251 CBH82N 57398195 IC50 = 45 nM T68251 C0YHM7 57398273 IC50 = 83 nM T68251 C5R1PU 57398274 IC50 = 3670 nM T68251 C0ZL1D 57399843 IC50 = 2050 nM T68251 CI6WB3 57399844 IC50 = 30083 nM T68251 C5SVE2 57399911 IC50 > 10000 nM T68251 CZ4GX2 57399912 IC50 = 7943.28 nM T68251 C4J5LE 57399913 IC50 = 7943.28 nM T68251 CH1J9Q 57399914 IC50 > 10000 nM T68251 CD50CO 57399918 IC50 = 3981.07 nM T68251 C82HGR 57399936 IC50 = 4370 nM T68251 CAX15U 57399937 IC50 = 9200 nM T68251 C1CN3U 57401566 IC50 = 2319 nM T68251 C3EKY4 57401585 IC50 = 4 nM T68251 CBZ36R 57401604 IC50 = 3 nM T68251 CM9D3A 57401688 IC50 > 10000 nM T68251 CF02UP 57401689 IC50 = 3981.07 nM T68251 CVO56U 57401690 IC50 = 7943.28 nM T68251 CN27EP 57401691 IC50 = 6309.57 nM T68251 CJLZ14 57401692 IC50 > 10000 nM T68251 C2AI8P 57401693 IC50 > 10000 nM T68251 CLNT30 57401717 IC50 = 798 nM T68251 CKL68A 57401718 IC50 = 307 nM T68251 C5IYO8 57401900 IC50 > 500000 nM T68251 CI1ML6 57401901 IC50 > 500000 nM T68251 C2IE0C 57401902 IC50 = 6800 nM T68251 C39ELP 57403329 IC50 = 15 nM T68251 CWP09F 57403330 IC50 > 1000 nM T68251 CIB91W 57403331 IC50 = 0.55 nM T68251 C63WPS 57403332 IC50 = 0.49 nM T68251 CXF62Z 57403333 IC50 = 16 nM T68251 CT26AL 57403355 IC50 = 931 nM T68251 C6OQH8 57403420 IC50 = 1258.93 nM T68251 C2Z6EC 57403421 IC50 = 5011.87 nM T68251 CA5Z2V 57403422 IC50 = 6309.57 nM T68251 CK68EY 57403424 IC50 = 7943.28 nM T68251 CQN8L6 57403445 IC50 = 232 nM T68251 C2L1SE 57403446 IC50 = 180 nM T68251 C0G2VY 57403564 IC50 = 0.8 nM T68251 CK4CJ0 57403617 IC50 = 290000 nM T68251 C5D0WE 57403618 IC50 > 500000 nM T68251 C7K2AP 57403619 IC50 > 500000 nM T68251 CE9B2P 57403620 IC50 = 1700 nM T68251 C1DRY0 57403621 IC50 = 200 nM T68251 C2MH8O 57523473 IC50 = 0.35 nM T68251 C57CEM 57523505 IC50 = 4 nM T68251 CS8W4L 57523538 IC50 = 5 nM T68251 CIT7B9 57523539 IC50 = 2 nM T68251 C56QXU 57523540 IC50 = 4 nM T68251 CX8IU3 57523541 IC50 = 30 nM T68251 CE8CL9 57523575 IC50 = 107 nM T68251 CWUP89 57523576 IC50 = 0.13 nM T68251 CT2QS3 57523577 IC50 = 0.07 nM T68251 CK6M0Y 57523578 IC50 = 0.1 nM T68251 C0HVU7 57523611 IC50 = 3 nM T68251 C5Q0ND 57523641 IC50 = 1.2 nM T68251 CWH7V8 57561293 IC50 = 533 nM T68251 C1PHI6 57708731 IC50 = 510 nM T68251 CF2Z7W 57708783 IC50 = 62 nM T68251 C9KV2W 57708792 IC50 = 660 nM T68251 CE36GP 57708799 IC50 = 670 nM T68251 C23QGY 57708843 IC50 > 1000 nM T68251 C2J5CW 57708880 IC50 = 230 nM T68251 C1K6AP 57708886 IC50 = 14 nM T68251 CY1N3J 57792153 IC50 = 1167 nM T68251 C6BKQ0 57874709 IC50 = 46000 nM T68251 CCKD80 58307579 Ki = 2.3 nM T68251 CX73PT 59033102 IC50 > 25000 nM T68251 CAT67H 59910477 IC50 = 79 nM T68251 CTZJ24 59910497 IC50 = 885 nM T68251 C1T2QI 60144811 IC50 = 545000 nM T68251 CZ18UT 67684770 IC50 = 10700 nM T68251 CLOE02 70682288 Ki = 600 nM T68251 CH2Q3V 70682301 IC50 = 53 nM T68251 C4NG7I 70682302 IC50 = 24 nM T68251 C6YOW4 70682303 IC50 = 10 nM T68251 CH76IU 70684364 Ki = 450 nM T68251 CZ63AG 70684365 Ki = 300 nM T68251 C6YH8C 70684382 IC50 = 3.8 nM T68251 CQ50YR 70684390 IC50 = 66 nM T68251 CTR64D 70686538 IC50 = 149 nM T68251 C0Q6JA 70686539 IC50 = 179 nM T68251 C8B6WD 70688393 IC50 = 11650 nM T68251 CGR3J2 70688394 IC50 = 23280 nM T68251 CTUN76 70688632 Ki = 61 nM T68251 C3LCG0 70688633 Ki = 180 nM T68251 CV9Y7S 70688643 IC50 = 7.3 nM T68251 CB4ZL3 70690154 IC50 > 500000 nM T68251 CJY19I 70690714 IC50 = 15 nM T68251 CFM0Q5 70690777 IC50 = 0.2 nM T68251 CWVI71 70691250 IC50 = 144 nM T68251 CJ3OY4 70692312 IC50 > 500000 nM T68251 C1A0VU 70692840 Ki = 110 nM T68251 CY4E9Z 70692916 IC50 > 100000 nM T68251 C0HFX4 70694371 IC50 > 500000 nM T68251 C0HE2P 70694634 IC50 = 15470 nM T68251 CLE79H 70696450 IC50 > 500000 nM T68251 CENQ98 70697478 IC50 = 450 nM T68251 C1XNI9 70941086 IC50 > 100000 nM T68251 C7BHO9 70941091 IC50 = 34700 nM T68251 C37VPQ 70941121 IC50 = 10300 nM T68251 CF7PC5 70941155 IC50 > 100000 nM T68251 CL7JF9 71304794 IC50 = 63 nM T68251 CSY30R 71304795 IC50 = 10 nM T68251 CNPG78 71304796 IC50 = 170 nM T68251 CA92XR 71449332 IC50 = 85500 nM T68251 COM1B0 71449369 IC50 = 143 nM T68251 CA6IB0 71450469 IC50 > 1000000 nM T68251 CK2AT8 71451145 IC50 = 12500 nM T68251 C5NYF7 71451146 IC50 = 1400 nM T68251 CW06TJ 71451147 IC50 = 67 nM T68251 CA7M9F 71451166 IC50 = 39000 nM T68251 CD4CP2 71451167 IC50 = 60000 nM T68251 C6M9VL 71451168 IC50 = 8100 nM T68251 C7HUF5 71451169 IC50 = 120 nM T68251 CMW3O0 71451330 Ki > 200000 nM T68251 CT5J7F 71452300 IC50 > 1000000 nM T68251 C23NVO 71452301 IC50 > 1000000 nM T68251 C7UIS9 71452970 IC50 = 67500 nM T68251 CC1B0Z 71452971 IC50 = 83700 nM T68251 CNMP23 71452972 IC50 = 27600 nM T68251 CIP9J5 71452973 IC50 = 8100 nM T68251 CUZ9S0 71452974 IC50 = 120 nM T68251 C71TWC 71452975 IC50 = 3900 nM T68251 CE98YL 71452999 IC50 = 184 nM T68251 C8VC6N 71453000 IC50 = 30 nM T68251 C4VKI1 71453001 IC50 = 87 nM T68251 C4E6PS 71453593 IC50 = 20000 nM T68251 C5K8WS 71454094 IC50 = 573000 nM T68251 CP2D3C 71454095 IC50 > 1000000 nM T68251 CGE27K 71454723 IC50 = 3000 nM T68251 C3VQW4 71455829 IC50 > 1000000 nM T68251 C4EJX2 71456472 IC50 = 37 nM T68251 C9QS6E 71456659 Ki = 20 nM T68251 C1JI6W 71458326 IC50 = 74600 nM T68251 C8ZR2I 71458327 IC50 = 1700 nM T68251 CV2J5Y 71458328 IC50 = 460 nM T68251 C29YHS 71458330 IC50 = 900 nM T68251 CXC1U7 71458350 IC50 = 121 nM T68251 C4IZ5V 71458351 IC50 = 181 nM T68251 CKR4D0 71459517 IC50 > 1000000 nM T68251 CKV4Q6 71460169 IC50 = 4500 nM T68251 CYF62U 71460170 IC50 = 750 nM T68251 C3LFX2 71460171 IC50 = 270 nM T68251 CDRO30 71460172 IC50 = 25 nM T68251 C6WN3A 71460173 IC50 = 13 nM T68251 CZO86D 71460193 IC50 = 278 nM T68251 C6UQW4 71461261 IC50 > 1000000 nM T68251 CKW27N 71461578 IC50 = 19.6 nM T68251 CX7W4A 71461879 IC50 = 2400 nM T68251 CKXO81 71461880 IC50 = 6300 nM T68251 CI4M8V 71461881 IC50 = 7600 nM T68251 CHD70Q 71461882 IC50 = 29 nM T68251 C7MLC8 71461883 IC50 = 17 nM T68251 CWL97M 71461905 IC50 = 301 nM T68251 CUT3H5 71461906 IC50 = 148 nM T68251 C06AXC 71461907 IC50 = 58 nM T68251 CSW59Y 71461908 IC50 = 1340 nM T68251 C9QE5X 71462985 IC50 > 1000000 nM T68251 CATP87 71465323 IC50 = 32.8 nM T68251 C0H3BX 71465324 IC50 = 6.4 nM T68251 CTM24Y 71465370 IC50 = 7.2 nM T68251 C6ZV0X 71465371 IC50 = 9.3 nM T68251 C7NYO8 71465420 IC50 = 6.3 nM T68251 C0E3FD 71465421 IC50 = 3.9 nM T68251 CW1K8M 71465466 IC50 > 100000 nM T68251 C28OYX 71465467 IC50 = 35700 nM T68251 C12BUO 71465468 IC50 > 100000 nM T68251 CP37ZB 71465510 IC50 = 2100 nM T68251 CR2T8F 71503450 IC50 = 2.8 nM T68251 C56YRV 71516803 IC50 < 1 nM T68251 C52QIK 71516804 IC50 = 5.1 nM T68251 C79ZRK 71516805 IC50 = 1.6 nM T68251 C3L7SD 71533484 IC50 = 227 nM T68251 CZH5S9 71533485 IC50 = 52 nM T68251 C4YRC7 71533486 IC50 = 21 nM T68251 CGM72Q 71540498 IC50 = 57 nM T68251 CXA1I5 71540599 IC50 = 54 nM T68251 C7CV9E 71540600 IC50 = 149 nM T68251 CA4BP6 71540601 IC50 = 82 nM T68251 CMZ3T2 71540715 IC50 = 67 nM T68251 CXY83G 71540716 IC50 = 56 nM T68251 C1ZH2G 71540717 IC50 = 69 nM T68251 CT4UD5 71540831 IC50 = 145 nM T68251 CP7SX8 71540832 IC50 = 71 nM T68251 C9IW7R 71540833 IC50 = 54 nM T68251 C6MA8T 71540949 IC50 = 598 nM T68251 C52FXB 71547352 IC50 = 1.7 nM T68251 C9RE0A 71559535 IC50 = 8.44 nM T68251 C47TMN 71559652 IC50 = 8.46 nM T68251 CN2XB4 71559653 IC50 = 5.57 nM T68251 CZHQ79 71559654 IC50 = 1524.69 nM T68251 CO59LK 71559762 IC50 = 4.18 nM T68251 CGL35Z 71559763 IC50 = 5.62 nM T68251 C7U5LE 71559764 IC50 = 1674.81 nM T68251 CD6L1J 71559765 IC50 = 4.32 nM T68251 CXKO04 71559766 IC50 = 5.73 nM T68251 CA14SK 71559767 IC50 = 1724.94 nM T68251 COZ56A 71559768 IC50 = 9.09 nM T68251 CZ9X1J 71559769 IC50 = 1867.71 nM T68251 C5NHI1 71559770 IC50 = 8.59 nM T68251 CF9JE8 71559897 IC50 = 9.11 nM T68251 CGT96R 71559898 IC50 = 5.47 nM T68251 C01PTX 71559899 IC50 = 1674.23 nM T68251 C96OCB 71559900 IC50 = 5.53 nM T68251 CJB0D9 71559901 IC50 = 1764.37 nM T68251 C6Y1IE 71559902 IC50 = 4.09 nM T68251 C24ZYC 71559903 IC50 = 5.62 nM T68251 CC3MY7 71559904 IC50 = 1754.54 nM T68251 C7WMU5 71560026 IC50 = 9.01 nM T68251 C60VEX 71560027 IC50 = 1578.64 nM T68251 CN1VF7 71560028 IC50 = 8.39 nM T68251 CSY3D5 71560029 IC50 = 9.04 nM T68251 CH5J4A 71602247 IC50 = 16 nM T68251 CH53IU 71602248 IC50 = 230 nM T68251 C97EWQ 71602249 IC50 = 61 nM T68251 CNX9B1 71652215 IC50 = 1.4 nM T68251 C7RZN9 71652216 IC50 = 3.8 nM T68251 C0NTU7 71652382 IC50 = 0.43 nM T68251 CA5XS1 71652383 IC50 = 46 nM T68251 CYS46I 71652677 IC50 = 3200 nM T68251 CX67VE 71654516 IC50 = 3000 nM T68251 C6KEH0 71680708 Ki = 27 nM T68251 C7DMX5 71680709 Ki = 3.9 nM T68251 CFPM82 71680710 Ki = 35 nM T68251 C9ZOM7 71680866 Ki = 3.1 nM T68251 CQ68LT 71680868 Ki = 7000 nM T68251 CFH2V0 71681183 Ki = 49 nM T68251 CV3X1T 71682766 Ki = 810 nM T68251 C5EAO8 71682767 Ki = 430 nM T68251 C80EYX 71682913 Ki = 7200 nM T68251 CIBD03 71682914 Ki = 240 nM T68251 C41BYG 71682915 Ki = 4.6 nM T68251 C93XEI 71682916 Ki = 67 nM T68251 CQ29PJ 71682917 Ki = 50000 nM T68251 CFWN65 71683062 Ki = 5700 nM T68251 CM4E5A 71716445 IC50 = 4.19 nM T68251 C45PSZ 71717046 IC50 = 9.26 nM T68251 C9Z4PI 71718276 IC50 = 8.41 nM T68251 C2XW5I 71718291 IC50 = 9.41 nM T68251 C3L4XU 71718301 IC50 = 3.3 nM T68251 C18RDB 71719502 IC50 = 4.43 nM T68251 C6FVE5 71734008 IC50 < 1 nM T68251 CN95PL 71734104 IC50 < 1 nM T68251 CV37BJ 71734105 IC50 = 4.8 nM T68251 C7H8VM 71734106 IC50 < 1 nM T68251 CHBV73 71734107 IC50 < 1 nM T68251 C6C1JF 71734108 IC50 = 14 nM T68251 CR28AW 71734195 IC50 = 7 nM T68251 C2YJR3 71734196 IC50 = 141 nM T68251 CJC6N5 71734197 IC50 = 5.2 nM T68251 CEF50T 71734198 IC50 = 3.6 nM T68251 CLWC38 72193198 IC50 < 1 nM T68251 CX4G0R 72204928 IC50 = 28200 nM T68251 CG9C6U 72204929 IC50 = 6000 nM T68251 C5A6XZ 72204930 IC50 = 20000 nM T68251 C0XZK4 72204931 IC50 = 15000 nM T68251 CM8Y7X 72204932 IC50 = 36000 nM T68251 C6RY4X 72204933 IC50 = 6600 nM T68251 C4N5AB 72204934 IC50 = 20800 nM T68251 C3H2FZ 72205111 IC50 = 42000 nM T68251 CQ0VX7 72205112 IC50 = 25000 nM T68251 CQ7TI1 72205113 IC50 = 2800 nM T68251 CPAW52 72205114 IC50 = 2100 nM T68251 C2LD3J 72205115 IC50 = 2800 nM T68251 CE4J8F 72711063 Ki = 290 nM T68251 CW2RF1 72711064 Ki = 490 nM T68251 CC5T1Q 72711065 Ki = 680 nM T68251 C7YFC8 72711513 IC50 = 1045 nM T68251 CTM4P2 72713638 IC50 = 1.2 nM T68251 C0N2JX 72713639 IC50 = 3 nM T68251 CF4K8Y 72713862 IC50 = 7.5 nM T68251 C3R6JO 72713863 IC50 = 48 nM T68251 CW9D3V 72713864 IC50 = 15 nM T68251 CQ6FH3 72713865 IC50 = 7.8 nM T68251 C4FYB0 72713866 IC50 = 20 nM T68251 CH6SI1 72713867 IC50 = 41 nM T68251 CS21QM 72713868 IC50 = 670 nM T68251 CB56AP 72714081 IC50 = 18 nM T68251 C1CK0E 72714082 IC50 = 1750 nM T68251 CP5Q8W 72714083 IC50 = 1870 nM T68251 CA03NU 72714084 IC50 = 125000 nM T68251 CRUH64 72714085 IC50 = 3800 nM T68251 COQZ24 72714091 Ki = 160 nM T68251 CC0ZX4 72714092 Ki = 230 nM T68251 CW8I1S 72714093 Ki = 310 nM T68251 C3Q9LV 72714094 Ki = 480 nM T68251 CZFY06 72714322 IC50 = 4100 nM T68251 CDY70J 72714323 IC50 = 1440 nM T68251 CD56BA 72714324 IC50 = 240 nM T68251 CE51LQ 72714333 Ki = 550 nM T68251 CK6D5F 72714334 Ki = 760 nM T68251 C1R2UZ 72714335 Ki = 690 nM T68251 CH4VF7 72714336 Ki = 440 nM T68251 C4VSK6 72714337 Ki = 560 nM T68251 CG4KW2 72714338 Ki = 420 nM T68251 C9FL7V 72714339 Ki = 50 nM T68251 CT5U1W 72734852 IC50 = 428990 nM T68251 C4OEI9 72734853 IC50 = 20620 nM T68251 C4AT5M 72734854 IC50 = 6559 nM T68251 CA7I9Q 72734855 IC50 = 10800 nM T68251 CJ5N2K 72734856 IC50 = 679 nM T68251 CCQ27I 72734857 IC50 = 1802 nM T68251 CCP65R 72735032 IC50 = 5438 nM T68251 C5XL1A 72735033 IC50 = 386 nM T68251 CYT1H0 72735034 IC50 = 530 nM T68251 CW6IE4 72735035 IC50 = 325 nM T68251 C58RHN 72735036 IC50 = 678.1 nM T68251 CFB5U1 72735037 IC50 = 325 nM T68251 CXY79G 72737387 IC50 = 2776 nM T68251 C6M1OD 72737388 IC50 = 834.9 nM T68251 CY4M3X 72737389 IC50 = 28190 nM T68251 CQM2E0 72737390 IC50 = 9480 nM T68251 CFQX60 72737391 IC50 = 878 nM T68251 C4BAJ5 72737560 IC50 = 77930 nM T68251 CRP56E 72737561 IC50 = 3093 nM T68251 C3J8GN 72737562 IC50 = 7480 nM T68251 CS2JM8 72737563 IC50 = 678 nM T68251 CZ0G7Y 72737564 IC50 = 786 nM T68251 COHR84 72737565 IC50 = 877 nM T68251 CLV1F5 72737566 IC50 = 516 nM T68251 CDX2F9 72984326 IC50 = 9.25 nM T68251 C6SR0A 73106454 IC50 = 61.94 nM T68251 CUKG79 73292708 IC50 = 0.9 nM T68251 C5D3CJ 73292709 IC50 = 4 nM T68251 CL69NM 73292710 IC50 = 4 nM T68251 CQ4RO1 73292711 IC50 = 0.7 nM T68251 C7CT2E 73292869 IC50 = 4 nM T68251 CA0LS6 73292870 IC50 = 0.9 nM T68251 CJU3V6 73292871 IC50 = 5 nM T68251 C3PGF2 73292872 IC50 = 3 nM T68251 C0O8VM 73292873 IC50 = 2 nM T68251 CBR9I5 73293034 IC50 = 3 nM T68251 C9FD2C 73293035 IC50 = 3 nM T68251 C7LP5J 73293036 IC50 = 2 nM T68251 C9PQG1 73293037 IC50 = 5 nM T68251 C4PF1H 73293038 IC50 = 0.4 nM T68251 CE39WF 73293196 IC50 = 4 nM T68251 CU96XE 73293197 IC50 = 9 nM T68251 CGC51Z 73293198 IC50 = 2 nM T68251 CC83FW 73293199 IC50 = 2 nM T68251 CS6T8M 73293200 IC50 = 0.5 nM T68251 C38IDL 73345835 Ki = 1.7 nM T68251 CR1LT3 73346934 IC50 = 200630 nM T68251 C25SOB 73349251 IC50 = 0.8 nM T68251 CW01EA 73349535 IC50 > 10000 nM T68251 C8ROG3 73350414 Ki = 14 nM T68251 CF7AB2 73350415 Ki = 17 nM T68251 C2PFM4 73351930 Ki = 200 nM T68251 COC60V 73352986 IC50 = 671560 nM T68251 CI09CY 73354906 Ki = 8.5 nM T68251 CA5T7P 73603957 IC50 = 3000 nM T68251 C8VN1R 74221194 IC50 = 1800 nM T68251 C7M4FT 74430862 IC50 = 35670 nM T68251 CD28XO 74966628 IC50 = 109.9 nM T68251 CG1AU5 74991907 IC50 = 2.6 nM T68251 C65RFS 74991938 IC50 = 6.6 nM T68251 CX89MG 75002237 IC50 = 34197.94 nM T68251 CD7P3T 75002250 IC50 = 750 nM T68251 CU73SM 75018048 IC50 = 26 nM T68251 C1BTU7 75018058 IC50 = 29.99 nM T68251 CX9VB7 75018063 IC50 = 15 nM T68251 CLHO50 75018065 IC50 = 3.396 nM T68251 CQL0E1 75018100 IC50 = 1 nM T68251 CC9UA2 75018101 IC50 = 1.3 nM T68251 CYB42V 75018103 IC50 = 269.77 nM T68251 C1FTQ8 75018104 IC50 = 5.8 nM T68251 C5M2FT 75018105 IC50 = 1.6 nM T68251 CF5ZC7 75018120 IC50 = 50 nM T68251 CFW35X 75018121 IC50 = 280 nM T68251 C4GK3X 75018123 IC50 = 5105.05 nM T68251 C6FPO0 75018124 IC50 = 84 nM T68251 CMS1L6 75018126 IC50 = 3500 nM T68251 CW78YB 75018133 IC50 = 38.02 nM T68251 CZP6X1 75018134 IC50 = 414 nM T68251 CS1D6P 75018135 IC50 = 0.4 nM T68251 CHAP32 75018146 IC50 = 2430 nM T68251 CEF3L5 75018147 IC50 = 6.397 nM T68251 CPMC39 75018148 IC50 = 779.83 nM T68251 CBNW85 75018149 IC50 = 53.95 nM T68251 C57SNU 75018158 IC50 = 309.74 nM T68251 CCL95X 75018159 IC50 = 33.96 nM T68251 CXC24A 75018160 IC50 = 210 nM T68251 C9F8BU 75018162 IC50 = 920 nM T68251 C4OP3D 75018163 IC50 = 100 nM T68251 C7YPR3 75018171 IC50 = 51999.6 nM T68251 CT8Y6H 75018172 IC50 = 1698.24 nM T68251 C5Z1CN 75018180 IC50 = 1 nM T68251 CW7OX3 75018184 IC50 = 6800 nM T68251 C68QBF 75018185 IC50 = 10.99 nM T68251 CSBO46 75018194 IC50 = 41 nM T68251 CUB7V9 76329513 IC50 = 0.26 nM T68251 C5LB0U 78426619 IC50 > 100000 nM T68251 CET6N8 78426757 IC50 > 100000 nM T68251 CKD41G 81689861 IC50 = 1000 nM T68251 CBL02O 85040463 IC50 = 27.99 nM T68251 CHAG58 85052312 IC50 = 6.6 nM T68251 CJ67RP 85055259 IC50 = 59 nM T68251 CVHM18 85082338 IC50 = 11.99 nM T68251 CRC43U 85102289 IC50 = 0.4 nM T68251 C3Z0PJ 85141621 IC50 = 0.2 nM T68251 C28SQI 85198610 IC50 = 11 nM T68251 CUE7G4 86287514 IC50 = 24000 nM T68251 CGQ8F3 86287515 IC50 = 1800 nM T68251 CJ37XE 86287516 IC50 = 3200 nM T68251 COV8I9 86291010 IC50 = 1088 nM T68251 C76RBA 86298624 IC50 = 230 nM T68251 C93FKI 86298625 IC50 = 110 nM T68251 CVLU48 86298626 IC50 = 192 nM T68251 CAB2F5 87349434 Ki = 13000 nM T68251 CY74HT 89136066 IC50 = 2 nM T68251 C1MDQ8 89136114 IC50 = 1400 nM T68251 CO2FL5 90137145 IC50 = 310 nM T68251 CIJ96H 90644155 IC50 = 4800 nM T68251 CX7EW1 90644156 IC50 = 30000 nM T68251 CK5GZ4 90644157 IC50 = 52000 nM T68251 C7O1YN 90644158 IC50 = 19000 nM T68251 CEN6C1 90644159 IC50 = 4900 nM T68251 C8X9UZ 90644160 IC50 = 16000 nM T68251 C3H6SG 90656558 IC50 = 980 nM T68251 CFE10C 90656560 IC50 = 1030 nM T68251 CD4L8R 90656562 IC50 = 4190 nM T68251 CEST81 90656564 IC50 = 2710 nM T68251 C7J0CO 90656566 IC50 = 520 nM T68251 CE9Y4D 90656568 IC50 = 1940 nM T68251 CZVG63 90656570 IC50 = 720 nM T68251 CT0QG6 90656572 IC50 = 760 nM T68251 CFPR48 90656574 IC50 = 3360 nM T68251 CDF06N 90656576 IC50 = 1810 nM T68251 CQ3R1A 90656578 IC50 = 270 nM T68251 CWV0Z9 90656580 IC50 = 1280 nM T68251 CGX01J 90656582 IC50 = 430 nM T68251 C6M1VH 90656584 IC50 = 26180 nM T68251 C1GUD2 90656586 IC50 = 38320 nM T68251 C5KWT1 90656588 IC50 = 7430 nM T68251 CS7PZ6 90656590 IC50 = 5760 nM T68251 CGF9P3 90656592 IC50 = 1520 nM T68251 CM46JO 90656594 IC50 = 5210 nM T68251 CXL84V 90656596 IC50 = 2070 nM T68251 C7EIO6 90656598 IC50 = 2320 nM T68251 CRH7F2 90656600 IC50 = 4360 nM T68251 CKW64G 90656602 IC50 = 2950 nM T68251 C4CU3D 90656604 IC50 = 2050 nM T68251 CVPH63 90663059 Ki = 18000 nM T68251 C6AK3O 90663060 Ki = 15000 nM T68251 CUZD67 90663061 Ki = 8000 nM T68251 CTQ17J 90663062 Ki = 33000 nM T68251 CQGJ90 90663063 Ki = 6000 nM T68251 C0ZH1K 90663064 Ki = 17000 nM T68251 CD53CF 90663065 Ki = 5000 nM T68251 C1A4QT 90663067 Ki = 8000 nM T68251 CLW7Q8 90663069 Ki = 24000 nM T68251 C6JY4Q 90663070 Ki = 36000 nM T68251 C7YU1I 90663071 Ki = 10000 nM T68251 C07RTW 90663072 Ki = 11000 nM T68251 CZ68QM 90663073 Ki = 18000 nM T68251 CVTJ63 90663074 Ki = 7000 nM T68251 C9J8HB 90663075 Ki = 4000 nM T68251 C06GRV 90663076 Ki = 2000 nM T68251 CF2L9A 90663077 Ki = 40000 nM T68251 CGL0N7 90663078 Ki = 12000 nM T68251 COP05M 90663079 Ki = 13000 nM T68251 C1E5CB 90663080 Ki = 35000 nM T68251 C6IXP4 90663081 Ki = 41000 nM T68251 C0S7NT 90663082 Ki = 12000 nM T68251 C8MOY6 90663083 Ki = 20000 nM T68251 C4NP9W 90663084 Ki = 16000 nM T68251 CD3C8E 90663085 Ki = 16000 nM T68251 C63NOF 90663086 Ki = 15000 nM T68251 CU3LC2 90663087 Ki = 17000 nM T68251 CQ9C5I 90667651 IC50 = 0.53 nM T68251 CGXO89 90667652 IC50 = 0.61 nM T68251 CRT54C 101910871 IC50 = 11000 nM T68251 C1J3CK 117094707 IC50 = 5400 nM T68251 CDO15M 118721026 IC50 = 12.5 nM T68251 CHO72Q 118721027 IC50 = 1449 nM T68251 C5ZS4E 118722686 IC50 = 2100 nM T68251 CIZB24 118722687 IC50 = 6100 nM T68251 C5C0ZX 118722688 IC50 = 7100 nM T68251 C4V3FD 118723755 IC50 = 3 nM T68251 CH6OW5 122179777 IC50 = 85350 nM T68251 CLCW15 122181996 IC50 > 100000 nM T68251 CZO32N 122181998 IC50 > 100000 nM T68251 C40DWG 122181999 IC50 > 100000 nM T68251 CJFS09 122190237 IC50 = 590 nM T68251 CRN56G 122191012 IC50 = 235.2 nM T68251 CGC3E2 122191014 IC50 = 144.6 nM T68251 CS61WU 122191016 IC50 = 256.2 nM T68251 CV3SP6 122191017 IC50 = 299.2 nM T68251 C8ZOT4 122191645 IC50 = 7920 nM T68251 CU6LT0 122191646 IC50 = 2884.03 nM T68251 CER90U 122191647 IC50 = 8511.38 nM T68251 C8X2BN 122191648 IC50 = 3235.94 nM T68251 CQ3US9 122191649 IC50 = 4830 nM T68251 C86DWE 122191650 IC50 = 11220.18 nM T68251 CQ14HT 122191651 IC50 = 9430 nM T68251 C8B1HC 122191652 IC50 = 6760.83 nM T68251 CN6WP3 122191653 IC50 = 208.93 nM T68251 CJ5R2S 122192039 IC50 = 4168.69 nM T68251 CK45AP 122192040 IC50 = 794.33 nM T68251 C2W4VX 122192041 IC50 = 2700 nM T68251 C3R5YP 122192042 IC50 = 12589.25 nM T68251 C8EB9C 122192043 IC50 = 11440 nM T68251 CF2K9Z 122192044 IC50 = 14791.08 nM T68251 C68DRB 122192045 IC50 = 2089.3 nM T68251 C2L7ZO 122192046 IC50 = 2150 nM T68251 C1BH0V 122192047 IC50 = 23820 nM T68251 C9MX4H 122192048 IC50 = 17782.79 nM T68251 CE4MD1 122192049 IC50 = 15488.17 nM T68251 CU13GZ 122192050 IC50 = 2818.38 nM T68251 CN1OP2 122192051 IC50 = 9900 nM T68251 C2WV6G 122192052 IC50 = 14791.08 nM T68251 CD2I6H 122192053 IC50 = 16840 nM T68251 CQ7RZ6 122192054 IC50 = 3630.78 nM T68251 COIP89 122195564 IC50 = 360 nM T68251 C8Z1BF 124196387 IC50 = 17000 nM T68251 CF9C4N 127025165 IC50 = 6.5 nM T68251 CH59PY 127025166 IC50 = 791 nM T68251 CT03QA 127026888 IC50 = 370 nM T68251 CO1DJ9 127027301 IC50 = 11.66 nM T68251 CM7B5S 127029507 IC50 = 628 nM T68251 C6HA8I 127029508 IC50 > 100000 nM T68251 CPM3N2 127029509 IC50 = 56.3 nM T68251 C3B9EY 127029510 IC50 > 100000 nM T68251 C9NLI6 127030239 IC50 = 112260 nM T68251 CW3C0H 127030240 IC50 = 38650 nM T68251 CHC1V8 127031459 IC50 = 34790 nM T68251 C5GJB1 127031460 IC50 = 9390 nM T68251 C3R8PS 127031461 IC50 = 13220 nM T68251 C07FRX 127031462 IC50 = 90810 nM T68251 C9QC5M 127031784 IC50 = 1050 nM T68251 CX25ZP 127031785 IC50 = 210410 nM T68251 CIP36Q 127032630 IC50 = 1890 nM T68251 CA5I7G 127032946 IC50 = 410 nM T68251 CEO26U 127032998 IC50 = 28520 nM T68251 CL16WE 127033305 IC50 = 5520 nM T68251 C9RZO5 127033306 IC50 = 640 nM T68251 C20GLU 127033307 IC50 = 240 nM T68251 C2XUV8 127033875 IC50 = 74910 nM T68251 COM48Q 127033876 IC50 = 28760 nM T68251 C30DFR 127033877 IC50 = 223370 nM T68251 CA8HJ9 127033878 IC50 = 36790 nM T68251 CQ3HV1 127034380 IC50 = 566890 nM T68251 CV1YR6 127036461 IC50 = 2000 nM T68251 CDIC57 127037442 IC50 = 3 nM T68251 CV3NQ6 127037443 IC50 = 2400 nM T68251 CWI7K3 127037444 IC50 > 10000 nM T68251 C9QLI2 127037445 IC50 = 9000 nM T68251 CCA0R8 127037446 IC50 = 1100 nM T68251 C89QOM 127043503 IC50 = 51 nM T68251 CK3I0F 127043504 IC50 = 263 nM T68251 C9E5YJ 127043505 IC50 = 31 nM T68251 CW1Q3D 127043506 IC50 = 76 nM T68251 CFDC75 127043682 IC50 = 193 nM T68251 C1C7WB 127044036 IC50 = 123 nM T68251 C16UNQ 127044037 IC50 = 472 nM T68251 CN58BX 127044038 IC50 = 672 nM T68251 C5DMP0 127044039 IC50 = 419 nM T68251 CPF6U7 127044139 IC50 = 177 nM T68251 C5FPE1 127044169 IC50 > 500 nM T68251 C7YE9B 127044170 IC50 > 500 nM T68251 CT9B0Q 127044462 IC50 = 44.65 nM T68251 CL3X1A 127044649 IC50 = 98 nM T68251 C7X1YO 127044650 IC50 = 186 nM T68251 C8RZ7T 127044651 IC50 = 41 nM T68251 C3I4PT 127044652 IC50 = 103 nM T68251 CBR1V9 127044680 IC50 = 85.9 nM T68251 CDX86T 127044818 IC50 = 30 nM T68251 C56OJV 127044819 IC50 = 24 nM T68251 CF7A5N 127044986 IC50 = 843 nM T68251 CGLJ92 127045131 IC50 = 203 nM T68251 C4HY6K 127045132 IC50 = 208 nM T68251 CWO1X0 127045258 IC50 = 806 nM T68251 C43ORS 127045609 IC50 = 291 nM T68251 C21LIW 127053364 IC50 = 0.19 nM T68251 CR5VQ8 127053365 IC50 = 2.2 nM T68251 C19QXS 127053368 IC50 > 10000 nM T68251 CJ0G9N 127053369 IC50 > 10000 nM T68251 C2Q6UH 127053370 IC50 > 10000 nM T68251 CWM7U2 127053371 IC50 = 21.8 nM T68251 C1VRM8 127053372 IC50 > 10000 nM T68251 CT76DR 127053375 IC50 = 2.05 nM T68251 CYA92R 130282633 IC50 = 890 nM T68251 CO3QE2 130282636 IC50 = 1000 nM T68251 C4MB7N 132285189 Ki = 85 nM T68251 CTN42D 132941363 IC50 = 11000 nM T68251 C83FAY 134130294 Ki = 15.9 nM T68251 CT3G2U 134133460 IC50 = 0.16 nM T68251 C8VLY0 134144890 IC50 = 110 nM T68251 C93ZLI 134145328 IC50 = 107 nM T68251 CN9D7G 134155756 IC50 = 2600 nM T68251 CU24IK 134694685 IC50 = 190 nM T68251 CHV2U1 135438561 IC50 = 5300 nM T68251 C4FVJ1 135487604 IC50 = 79600 nM T68251 C6GR3K 135567051 IC50 = 83 nM T68251 C1MOD4 135567320 IC50 = 730 nM T68251 CYH23I 136054468 IC50 = 32 nM T68251 CZ8DW1 136054472 IC50 = 86 nM T68251 C9H0DL 136054473 IC50 = 120 nM T68251 CX7MI0 136054475 IC50 = 65 nM T68251 CA5JR6 136054481 IC50 = 14 nM T68251 CO2VU9 136054484 IC50 < 10 nM T68251 CV47JN 136054485 IC50 = 10 nM T68251 CZ48WO 136054487 IC50 = 23 nM T68251 CR9CY5 136054490 IC50 < 10 nM T68251 C8FGT0 136054495 IC50 = 110 nM T68251 CGH39U 136054498 IC50 < 10 nM T68251 C2TO7Y 136054508 IC50 = 160 nM T68251 CG70BZ 136054516 IC50 = 3 nM T68251 CSM57W 136054520 IC50 = 0.57 nM T68251 CXNG40 136118011 Ki = 2472 nM T68251 C1IOH9 136118012 Ki > 3333 nM T68251 CTY79S 136118013 Ki > 3333 nM T68251 CTE87J 136118014 Ki > 3333 nM T68251 CJG54U 136219136 IC50 > 30000 nM T68251 C3CAV5 136219141 IC50 > 30000 nM T68251 CPB07Z 136241630 IC50 = 800 nM T68251 CIEW62 136380958 IC50 = 8.3 nM T68251 CSEY19 137175240 IC50 = 7170 nM T68251 C9HS7J 137287436 IC50 = 1.9 nM T68251 C4UMY5 137636781 IC50 > 5000 nM T68251 CR8H9Z 137644167 IC50 > 5000 nM T68251 CB8M6U 137646865 IC50 > 5000 nM T68251 CK4LE6 137647628 IC50 = 2700 nM T68251 C9CIY6 137651719 IC50 = 2 nM T68251 CS80YI 137652598 IC50 = 280 nM T68251 CZB75K 137657128 IC50 > 10000 nM T68251 CC3I9B 137660260 IC50 > 5000 nM T68251 C4H0EM 137661370 IC50 = 3100 nM T68251 CZ8H6N 137661550 IC50 = 5800 nM T68251 C37HMX 137701229 Ki = 37 nM T68251 C5FWA2 145949488 IC50 = 584 nM T68251 CZS1N7 145949693 IC50 = 936 nM T68251 C6IPV3 145949783 IC50 = 4800 nM T68251 C72LGN 145950074 IC50 = 2850 nM T68251 CU53BP 145950331 IC50 > 5000 nM T68251 CY8C4A 145950332 IC50 = 189 nM T68251 CAJ25P 145951291 IC50 > 5000 nM T68251 C3EF7N 145952515 IC50 = 114 nM T68251 CW1GS2 145952760 IC50 > 5000 nM T68251 CFN1R7 145952843 IC50 = 187 nM T68251 CV80WQ 145954107 IC50 > 5000 nM T68251 C16VNH 145954604 IC50 = 500 nM T68251 CQF50V 145954863 IC50 = 128 nM T68251 C2HAG8 145955226 IC50 = 8520 nM T68251 CH0ZO5 145955778 IC50 = 362 nM T68251 CVZ5U7 145955868 IC50 = 232 nM T68251 C8TPR1 145956198 IC50 > 5000 nM T68251 COR96H 145956298 IC50 = 2120 nM T68251 CR8U7Y 145956318 IC50 > 5000 nM T68251 C7R3FE 145956426 IC50 = 1650 nM T68251 CUS0Y9 145957234 IC50 > 5000 nM T68251 C6MHN7 145957508 IC50 > 5000 nM T68251 CQ15DP 145957734 IC50 = 4070 nM T68251 C5K7PV 145958060 IC50 > 5000 nM T68251 CBE02W 145958354 IC50 > 5000 nM T68251 CQL4O0 145959327 IC50 > 5000 nM T68251 CG03OE 145959777 IC50 = 210 nM T68251 CIQ9J2 145960035 IC50 = 5340 nM T68251 CRY63E 145963538 IC50 > 5000 nM T68251 CX7PL8 145963779 IC50 = 75.25 nM T68251 CPRZ56 145963828 IC50 = 72.02 nM T68251 C5JTM2 145963892 IC50 = 38.68 nM T68251 CFLU54 145964255 IC50 = 57.24 nM T68251 C3MDU9 145965508 IC50 = 81210 nM T68251 C8ZI7P 145965593 IC50 = 53.14 nM T68251 C6ASH4 145965758 IC50 = 58.02 nM T68251 CABQ48 145965824 IC50 = 54.74 nM T68251 C8M7FR 145966330 IC50 = 660 nM T68251 CCO03H 145966492 IC50 = 32.71 nM T68251 CZG2P7 145966498 IC50 = 33.47 nM T68251 C4P0GM 145966951 IC50 = 53.82 nM T68251 C5ICD0 145967022 IC50 = 1350 nM T68251 CI80WY 145967366 IC50 = 19.57 nM T68251 CFE1A5 145971595 Ki = 127 nM T68251 CWY5X0 145971805 IC50 = 414 nM T68251 C1FPG2 145972660 IC50 = 219 nM T68251 CYFI60 145973042 IC50 = 2500 nM T68251 CZHR42 145973116 IC50 = 203400 nM T68251 CQF05Z 145973471 IC50 = 50.55 nM T68251 CJF73O 145973630 IC50 = 172 nM T68251 CC1BF5 145973750 IC50 = 58.08 nM T68251 COA47B 145973991 IC50 = 54.68 nM T68251 C1VO8L 145974965 IC50 = 73.82 nM T68251 CQ0DP4 145975098 IC50 = 55.13 nM T68251 CV9D1F 145975682 IC50 > 100000 nM T68251 CI9VB4 145975902 IC50 > 10000 nM T68251 CX7M9L 145976456 IC50 > 5000 nM T68251 C5C6VJ 145976464 IC50 = 54180 nM T68251 C1KPL5 145976497 IC50 = 670 nM T68251 C7RG1J 145976981 IC50 = 62.87 nM T68251 C18OCA 145976989 IC50 = 230000 nM T68251 C5HW7O 145977208 IC50 = 36.83 nM T68251 CPD1B0 145977213 IC50 > 5000 nM T68251 C79VAX 145977588 IC50 = 49.69 nM T68251 CG9KD3 145977825 IC50 > 1000 nM T68251 C60INE 145977843 IC50 = 83.04 nM T68251 CN6JB8 145978296 IC50 > 1000 nM T68251 C5Z7XW 145983264 IC50 = 182 nM T68251 C0EMZ9 145984335 IC50 = 345 nM T68251 CBNO84 145985441 IC50 = 414 nM T68251 CDW7K5 145986213 IC50 = 102 nM T68251 CM7YB8 145998092 IC50 = 1300 nM T68251 C2C8QR 153033791 IC50 = 58430 nM T68251 C2CZ9B 155511425 IC50 = 5700 nM T68251 CZ25LW 155512044 IC50 = 11000 nM T68251 CV10AF 155512426 IC50 = 151 nM T68251 C1V4CS 155512637 IC50 > 10000 nM T68251 CMQ8W6 155512861 IC50 = 7500 nM T68251 CFHU79 155514943 IC50 = 55 nM T68251 C13OQY 155515143 IC50 = 8800 nM T68251 CND4L8 155515645 IC50 = 9549.93 nM T68251 CC15YH 155515706 IC50 > 10000 nM T68251 C98HMU 155515777 IC50 = 1.2 nM T68251 C0OSL9 155516668 IC50 = 21379.62 nM T68251 C6N3DB 155517141 IC50 = 0.28 nM T68251 C3I5AL 155519394 IC50 = 6500 nM T68251 CS6ZT7 155519964 IC50 = 21 nM T68251 CG2RF3 155520398 IC50 = 2100 nM T68251 CL16UE 155520835 IC50 > 10000 nM T68251 C5C1SL 155521791 IC50 > 10000 nM T68251 C59YHT 155522902 IC50 = 503 nM T68251 C4AH9W 155525335 IC50 > 10000 nM T68251 CM9AP3 155526116 IC50 > 10000 nM T68251 C6RBG9 155527660 IC50 = 2800 nM T68251 C83IXL 155528558 IC50 = 0.16 nM T68251 CT4PA7 155528661 IC50 > 10000 nM T68251 CWB4X1 155529076 IC50 > 10000 nM T68251 CSG54J 155529234 IC50 > 10000 nM T68251 C2G0BE 155529579 IC50 > 10000 nM T68251 CC5FA9 155529859 IC50 > 10000 nM T68251 CQUA53 155531128 IC50 = 3000 nM T68251 C7TP3R 155531151 IC50 > 10000 nM T68251 CZSY48 155533962 IC50 = 3600 nM T68251 C5WTE3 155534754 IC50 = 6700 nM T68251 CG47PB 155534833 IC50 = 3000 nM T68251 C4VCN3 155535749 IC50 = 12860 nM T68251 C2WCU5 155536887 IC50 = 10715.19 nM T68251 C4DSL8 155536899 IC50 > 10000 nM T68251 C12LFZ 155540134 IC50 = 620 nM T68251 CNH2K4 155540729 IC50 = 3300 nM T68251 CO90SD 155541304 IC50 = 11748.98 nM T68251 CRY3D4 155541376 IC50 = 13 nM T68251 CV0ZI3 155542003 IC50 = 12302.69 nM T68251 CJN8X5 155542058 Ki = 0.5 nM T68251 CO8ZY9 155542845 IC50 = 0.048 nM T68251 CH9E0W 155543836 IC50 = 34673.69 nM T68251 C1VL8X 155544079 IC50 > 10000 nM T68251 CYK18P 155544623 IC50 > 10000 nM T68251 CBSJ86 155544856 IC50 = 11220.18 nM T68251 CWEG57 155545190 IC50 = 3 nM T68251 CP6W3Q 155545205 IC50 > 10000 nM T68251 CLWS20 155545852 IC50 = 47863.01 nM T68251 COH0W2 155546374 IC50 = 492 nM T68251 CLT8Z2 155546617 IC50 = 2.38 nM T68251 C3FRY8 155547834 IC50 = 0.096 nM T68251 C1FP0M 155548067 IC50 = 32 nM T68251 C9AOK6 155550135 IC50 = 3000 nM T68251 C9ZUH8 155553520 IC50 = 6200 nM T68251 CPQ84I 155553728 IC50 > 10000 nM T68251 CM7C1P 155555245 IC50 = 16240 nM T68251 CS62RN 155556052 IC50 = 13803.84 nM T68251 C94NQE 155556307 IC50 > 10000 nM T68251 C9FC1W 155557598 IC50 = 3200 nM T68251 CJHM29 155557941 IC50 = 8310 nM T68251 CD3M6P 155558654 IC50 = 16870 nM T68251 CPDF57 155558916 IC50 = 57543.99 nM T68251 CG2DI6 155560100 IC50 = 8800 nM T68251 CQJ07L 155561559 IC50 = 8800 nM T68251 C3BA9L 155561798 IC50 = 5 nM T68251 CH40UO 155562232 IC50 = 4.1 nM T68251 C6SAE0 155562336 IC50 = 8.9 nM T68251 CD18KU 155563750 IC50 = 7600 nM T68251 CM0LN1 155563771 IC50 = 810 nM T68251 CQ4WE0 155563852 IC50 = 28183.83 nM T68251 C29SMF 155565303 IC50 > 10000 nM T68251 C51ZMC 155565586 IC50 = 700 nM T68251 CZ0WK1 155566979 IC50 = 3800 nM T68251 CP9YX2 155567218 IC50 = 2400 nM T68251 C8D5VK 155567855 IC50 = 3500 nM T68251 CHL0F3 155567858 IC50 > 10000 nM T68251 C5U9LI 155569346 IC50 = 570 nM T68251 CLT4Y6 10138589 Ki = 300 nM T68251 C5U3AO 57394286 IC50 = 23 nM T68251 C0YL9R 9975488 IC50 = 1900 nM T68251 D00RNA 44446270 IC50 = 200 nM T68251 D00TRF 44423683 IC50 = 94000 nM T68251 D01UNE 44580457 Ki = 30 nM T68251 D02ECA 448942 IC50 > 100000 nM T68251 D02EFQ 10549609 IC50 = 5 nM T68251 D02UYR 9907830 Ki = 0.3 nM T68251 D03AMR 9849669 Ki = 7 nM T68251 D04GOO 10111838 IC50 > 100000 nM T68251 D04PAW 16216218 IC50 = 60000 nM T68251 D04VPH 45376872 IC50 = 18000 nM T68251 D04WWO 9889867 Ki > 3333 nM T68251 D05BMD 44423684 IC50 = 137000 nM T68251 D05JPV 44406790 IC50 = 3070 nM T68251 D05THD 44478925 IC50 = 1300 nM T68251 D06EHW 11625778 IC50 = 35 nM T68251 D06HSC 136117931 IC50 = 65000 nM T68251 D06NDR 44423687 IC50 = 81800 nM T68251 D06ZRX 5281717 IC50 = 27600 nM T68251 D07DRT 46175162 Ki = 3.8 nM T68251 D07GEL 10344307 Ki = 1.1 nM T68251 D07MJD 44479701 IC50 = 510 nM T68251 D07VXX 16721024 IC50 = 151000 nM T68251 D08ICI 44446277 IC50 = 590 nM T68251 D08NSS 5288596 IC50 < 0.1 nM T68251 D09GIL 66160 IC50 = 50000 nM T68251 D09USO 5277466 IC50 > 100000 nM T68251 D09ZOA 25049753 IC50 = 2 nM T68251 D0A0FY 44479457 IC50 = 35000 nM T68251 D0A4TC 446504 IC50 = 3 nM T68251 D0A5MV 11581319 IC50 = 1660 nM T68251 D0B3UN 44580458 Ki = 192 nM T68251 D0D7GL 10789 IC50 = 146000 nM T68251 D0E5MB 44411812 IC50 = 792 nM T68251 D0F2HJ 45257111 IC50 = 196500 nM T68251 D0F7BE 4369084 Ki = 3000 nM T68251 D0FO2B 1923 IC50 = 130000 nM T68251 D0G0OP 44423685 IC50 = 68000 nM T68251 D0G3YZ 11391583 IC50 = 4520 nM T68251 D0H2PA 9886977 Ki = 0.5 nM T68251 D0H6CK 10160968 Ki > 3333 nM T68251 D0J0WJ 45257110 IC50 = 232500 nM T68251 D0K4TI 49292 IC50 = 1300 nM T68251 D0L4EO 11609208 IC50 = 440 nM T68251 D0L6ND 10089677 IC50 = 1.7 ug.mL-1 T68251 D0N8YA 159596 IC50 = 15000 nM T68251 D0NP8A 10370504 IC50 = 1790 nM T68251 D0NV9C 22004198 IC50 = 40 nM T68251 D0P2TS 9818682 IC50 > 60000 nM T68251 D0Q4TA 10044321 IC50 = 12 nM T68251 D0Q9LC 44385624 IC50 = 868 nM T68251 D0R2BO 194777 IC50 = 0.7 nM T68251 D0S9OL 10155934 IC50 = 1200 nM T68251 D0T1FR 44457233 IC50 = 4000 nM T68251 D0UI1P 46228278 IC50 = 178600 nM T68251 D0V9EN 689043 IC50 = 24.26 nM T68251 D0VI2A 44447430 IC50 = 537 nM T68251 D0W2UK 6914621 Ki = 2050 nM T68251 D0W3ME 4369080 Ki = 3000 nM T68251 D0XK7G 10445302 IC50 = 32 nM T68251 D0Y1XM 44423686 IC50 = 33700 nM T68251 D0Y5IQ 44255320 IC50 = 5000 nM T68251 D0Y7NV 2220392 IC50 = 898 nM T68251 D0Z4LO 9832179 IC50 = 23 nM T68251 D0Z4NU 46228282 IC50 = 285900 nM T72319 CV39DH 1072048 Ki = 33100 nM T72319 C64ZSL 43430547 IC50 > 30000 nM T72319 CQ4P5B 44755448 IC50 > 30000 nM T72319 C3NE8O 46931242 IC50 > 30000 nM T72319 C6O8RT 55872720 IC50 > 30000 nM T72319 C2P7SD 56577044 IC50 > 10000 nM T72319 CXY3E4 57720618 IC50 > 30000 nM T72319 CY9Z8F 60735522 IC50 > 30000 nM T72319 CB0SA4 61041645 IC50 > 30000 nM T72319 CT9M2C 61041646 IC50 > 30000 nM T72319 C3I5DM 61041804 IC50 > 30000 nM T72319 C84MGB 61242835 IC50 > 30000 nM T72319 C0Y6KO 62947261 IC50 > 30000 nM T72319 C8XEI4 63259457 IC50 > 30000 nM T72319 C0WX5O 70679311 IC50 > 30000 nM T72319 CEW3R6 71598546 IC50 > 30000 nM T72319 CUD65X 73333125 IC50 > 10000 nM T72319 CHQ18I 73333126 IC50 > 10000 nM T72319 C9UDN1 73333127 IC50 > 10000 nM T72319 C9K1NV 73333128 IC50 > 10000 nM T72319 C4UE6G 73333129 IC50 > 10000 nM T72319 CV2SJ4 73333225 IC50 > 10000 nM T72319 CF8HO3 73333226 IC50 > 10000 nM T72319 CVH9F0 73333227 IC50 > 10000 nM T72319 C4PYG2 73333229 IC50 > 10000 nM T72319 CBJC52 73333322 IC50 > 10000 nM T72319 CVEN67 73334066 IC50 > 10000 nM T72319 CYL3M7 73334067 IC50 > 10000 nM T72319 C6T7YX 73334068 IC50 > 10000 nM T72319 C70XCT 73334069 IC50 > 10000 nM T72319 C8QWP1 73334070 IC50 > 10000 nM T72319 CR98DL 73334157 IC50 > 10000 nM T72319 CJD9C1 73334158 IC50 > 10000 nM T72319 CLRM71 73334159 IC50 > 10000 nM T72319 C43NER 73334160 IC50 > 10000 nM T72319 CD2HX4 73334161 IC50 > 10000 nM T72319 CC89FN 73334162 IC50 > 10000 nM T72319 COV3R1 73334262 IC50 > 10000 nM T72319 CZD0N1 73334263 IC50 > 10000 nM T72319 CU3KG0 73334264 IC50 > 10000 nM T72319 CMLV27 73334265 IC50 > 10000 nM T72319 CD0VK7 73334266 IC50 > 10000 nM T72319 C1SGJ3 73334267 IC50 > 10000 nM T72319 C3PYF5 73334361 IC50 > 10000 nM T72319 C8H9JF 73334363 IC50 > 10000 nM T72319 C8XE1J 73334364 IC50 > 10000 nM T72319 CN40ZI 73334365 IC50 > 10000 nM T72319 CF9GA5 73334366 IC50 > 10000 nM T72319 C69WLM 73334479 IC50 > 10000 nM T72319 CG32QB 73334480 IC50 > 10000 nM T72319 CVE0S2 73334481 IC50 > 10000 nM T72319 C2S8XN 73334482 IC50 > 10000 nM T72319 CXJP87 73334483 IC50 > 10000 nM T72319 C57KSE 73334484 IC50 > 10000 nM T72319 CAQ18T 73334592 IC50 > 10000 nM T72319 CA67YG 73334593 IC50 > 10000 nM T72319 CNS84D 73334594 IC50 > 10000 nM T72319 C93HWE 73334595 IC50 > 10000 nM T72319 C87UBE 73334596 IC50 > 10000 nM T72319 CKSY83 73334696 IC50 > 10000 nM T72319 C36QHM 73334697 IC50 > 10000 nM T72319 CF63HU 73334698 IC50 > 10000 nM T72319 CQBX27 73334699 IC50 > 10000 nM T72319 C0OW1V 73334700 IC50 > 10000 nM T72319 C2VFJ9 73349256 IC50 > 30000 nM T72319 CG80NF 73349257 IC50 > 10000 nM T72319 COY1J2 73349259 IC50 > 10000 nM T72319 CNO9Z5 73350843 IC50 > 10000 nM T72319 C8U0ZX 73352326 IC50 > 10000 nM T72319 CRZ62F 73355036 IC50 = 8100 nM T72319 CD26ZM 73386663 IC50 = 73000 nM T72319 C2OXQ5 76314887 IC50 > 30000 nM T72319 C3X7EW 76314888 IC50 > 30000 nM T72319 C1YKN5 76314889 IC50 > 30000 nM T72319 C4E1BN 76318504 IC50 > 30000 nM T72319 CF76CT 76318505 IC50 > 30000 nM T72319 CLVA91 76318506 IC50 > 30000 nM T72319 C9LNK4 76318507 IC50 > 30000 nM T72319 CL87KC 76318508 IC50 > 30000 nM T72319 CET23F 76318509 IC50 > 30000 nM T72319 C01JLF 76322168 IC50 > 30000 nM T72319 C2SEM0 76322169 IC50 > 30000 nM T72319 CRH48X 76322170 IC50 > 30000 nM T72319 C5CZV2 76325789 IC50 > 30000 nM T72319 CS6GL0 76333019 IC50 > 30000 nM T72319 C7IUX5 76333020 IC50 > 30000 nM T72319 CZC8W2 76336632 IC50 > 30000 nM T72319 CYQ0B9 76336633 IC50 > 30000 nM T72319 CK2N0L 76336634 IC50 > 30000 nM T72319 CS4W5I 76336635 IC50 > 30000 nM T72319 CM6H9O 76336636 IC50 > 30000 nM T72319 CL8E1A 83748040 IC50 > 30000 nM T72319 CK5MX8 90655573 IC50 = 11000 nM T72319 C0S3XK 90655574 IC50 = 6800 nM T72319 CC50PO 90655575 IC50 = 5700 nM T72319 CA07UL 90655576 IC50 = 67000 nM T72319 CSUT18 90655577 IC50 = 23000 nM T72319 CD43OR 90655578 IC50 = 62000 nM T72319 C2A3RQ 90655579 IC50 = 35000 nM T72319 CEOP54 90655580 IC50 = 10100 nM T72319 CAM67V 90655581 IC50 = 10300 nM T72319 CLR17Q 90655582 IC50 = 13000 nM T72319 C28HZW 90655583 IC50 = 11000 nM T72319 CA1Y5I 90655584 IC50 = 21000 nM T72319 CQY83C 90655585 IC50 = 11200 nM T72319 CQTF13 90655586 IC50 = 6000 nM T72319 C83EFC 90655587 IC50 = 8800 nM T72319 C25ZNR 90655588 IC50 = 39000 nM T72319 C0GIC4 90655589 IC50 = 120000 nM T72319 CR6VS0 90655590 IC50 = 53000 nM T72319 C6KU2N 90655591 IC50 > 500000 nM T72319 C65HLO 90655592 IC50 = 9000 nM T72319 C4ACU9 90655593 IC50 = 79000 nM T72319 C74MKT 90655594 IC50 = 560000 nM T72319 CM21PY 90655595 IC50 > 250000 nM T72319 C78GYV 90655596 IC50 > 500000 nM T72319 C86DBC 90655597 IC50 > 250000 nM T72319 C9QU1T 90655598 IC50 > 250000 nM T72319 CWXY79 90655599 IC50 = 35000 nM T72319 C8M3HN 90655600 IC50 = 102000 nM T72319 C1MDL6 90655601 IC50 = 26000 nM T72319 C1MDK2 90655602 IC50 = 23000 nM T72319 CCD42S 90655603 IC50 = 22000 nM T72319 C7C9MF 90655604 IC50 = 105000 nM T72319 C27CIT 90655605 IC50 = 8600 nM T72319 C9PUC5 90655606 IC50 = 7800 nM T72319 CK2F6S 90655607 IC50 = 26000 nM T72319 C5T9WY 90655608 IC50 = 57000 nM T72319 C2EUX8 90655609 IC50 = 91000 nM T72319 C2A3CS 90655610 IC50 = 23000 nM T72319 C45VLK 90655611 IC50 = 89000 nM T72319 CN54XB 90655612 IC50 = 26000 nM T72319 C14LVC 90655613 IC50 = 67000 nM T72319 C64DAW 90655614 IC50 = 58000 nM T72319 C5H9VJ 90655615 IC50 = 100000 nM T72319 C9Z6BP 90655616 IC50 = 58000 nM T72319 C31VJO 90655617 IC50 > 250000 nM T72319 CAFW32 90655618 IC50 > 250000 nM T72319 CNZ4D8 90655619 IC50 = 34000 nM T72319 CY1PL8 90655620 IC50 = 53000 nM T72319 C5F6MO 90655621 IC50 > 2000000 nM T72319 C54UJD 90655622 IC50 > 2000000 nM T72319 C3OB0Z 90655623 IC50 = 4600 nM T72319 CW2ND5 90655624 IC50 = 6200 nM T72319 C87RLM 90655625 IC50 = 6300 nM T72319 C05HED 90655626 IC50 = 6700 nM T72319 C2BM7J 90655627 IC50 > 250000 nM T72319 CM51GQ 90655628 IC50 = 8800 nM T72319 CSL98F 90655629 IC50 = 57000 nM T72319 CLT0P1 90655635 IC50 = 27000 nM T72319 CW25YP 90666882 IC50 > 30000 nM T72319 CQI7D0 90666883 IC50 > 30000 nM T72319 C72IZG 90666884 IC50 > 30000 nM T72319 CCDK35 90666885 IC50 > 30000 nM T72319 C2DCW6 90666886 IC50 > 30000 nM T72319 CXN36J 90666887 IC50 > 30000 nM T72319 CG2S0B 90666888 IC50 > 30000 nM T72319 C19VSG 90666889 IC50 > 30000 nM T72319 CBG12J 90666890 IC50 > 30000 nM T72319 C90LPT 90666891 IC50 > 30000 nM T72319 C0IOH4 90666892 IC50 > 30000 nM T72319 C1CU2X 101043861 IC50 = 37 nM T72319 C0YL6Q 102602632 IC50 = 16000 nM T72319 C4Z1BN 102602634 IC50 = 130 nM T72319 C30MVB 127034580 IC50 = 1700 nM T72319 CR72CK 127044991 Ki = 25000 nM T72319 CVT1R7 127044992 Ki = 10000 nM T72319 CFJ30Y 127044993 Ki = 16900 nM T72319 CWA1V6 127044994 Ki = 10000 nM T72319 CMY6T7 127045145 Ki = 4800 nM T72319 CW6BT0 127045602 Ki = 39300 nM T72319 C6NBV2 134130627 IC50 = 35 nM T72319 COEW21 134131637 IC50 > 60000 nM T72319 C9XOG1 134131644 IC50 > 60000 nM T72319 CUW67R 134133875 IC50 = 240 nM T72319 CA1LH4 134133965 IC50 > 60000 nM T72319 C7PCM8 134134706 IC50 > 60000 nM T72319 C3PR2V 134134858 IC50 = 3100 nM T72319 CZB51D 134137731 IC50 = 51000 nM T72319 CKI23U 134139941 IC50 > 60000 nM T72319 C1OEI2 134140369 IC50 > 60000 nM T72319 C62JBE 134141602 IC50 = 220 nM T72319 CB20QF 134142297 IC50 > 60000 nM T72319 C29JUC 134142686 IC50 = 56 nM T72319 CS69VL 134143576 IC50 = 25000 nM T72319 C3XG2N 134144118 IC50 = 81 nM T72319 CZ83CB 134144237 IC50 = 51000 nM T72319 C48DSU 134145156 IC50 > 60000 nM T72319 C5C0HU 134145218 IC50 = 32000 nM T72319 CX1QB4 134145347 IC50 = 53000 nM T72319 C5IMF8 134145736 IC50 > 60000 nM T72319 CQX43Z 134145760 IC50 = 570 nM T72319 CX71GT 134146508 IC50 = 47 nM T72319 CE0C7P 134146658 IC50 = 740 nM T72319 CJY6D2 134146764 IC50 > 60000 nM T72319 C7NBT1 134148174 IC50 = 1700 nM T72319 C02JMB 134148668 IC50 = 61 nM T72319 CTL0D2 134149263 IC50 = 1200 nM T72319 C3BD1U 134149299 IC50 = 250 nM T72319 CS73OF 134149994 IC50 = 41000 nM T72319 C1MLU3 134151077 IC50 > 60000 nM T72319 C21YGK 134151685 IC50 > 60000 nM T72319 CES73F 134152016 IC50 = 1100 nM T72319 CIZV46 134152824 IC50 > 60000 nM T72319 C38AYE 134153154 IC50 = 230 nM T72319 CD5VJ0 134153698 IC50 = 18000 nM T72319 C4C7VM 134154055 IC50 = 75 nM T72319 CPAK59 134154083 IC50 = 4400 nM T72319 C9SAU3 134154301 IC50 = 32 nM T72319 CVK52O 134155339 IC50 = 35 nM T72319 CUH81S 134156240 IC50 = 26000 nM T72319 CB3YE8 134156251 IC50 = 63 nM T72319 CQ35RF 134157076 IC50 > 60000 nM T72319 CU0Z1S 134157587 IC50 = 28000 nM T72319 CFHK68 134157612 IC50 = 2600 nM T72319 D0W9RR 57339144 IC50 > 10000 nM T97353 D01TJY 53340771 IC50 > 10 nM T97353 CS24BW 11973730 IC50 = 15 nM T97353 CG3FV0 16727128 IC50 = 214 nM T97353 CAVY89 23636144 IC50 = 102 nM T97353 C1VUH4 23636254 IC50 = 17 nM T97353 C6LR7V 23636255 IC50 = 50 nM T97353 C5MSF6 23636502 IC50 = 29 nM T97353 C8B7QE 72949858 IC50 > 5000 nM T97353 C5ALQ2 76285468 IC50 = 4 nM T97353 CQ8BX7 76310576 IC50 = 163 nM T97353 C0JKX6 76310577 IC50 = 588 nM T97353 CUAH40 76310578 IC50 = 978 nM T97353 C4EK9U 76310579 IC50 > 4000 nM T97353 COZ54T 76310580 IC50 > 1000 nM T97353 CHI2U7 76310581 IC50 > 1000 nM T97353 COI21T 76310597 IC50 = 34 nM T97353 CL3EO0 76310599 IC50 = 470 nM T97353 CA9X2E 76310600 IC50 > 4000 nM T97353 CT1AJ4 76314216 IC50 = 114 nM T97353 C90ZKU 76314217 IC50 = 233 nM T97353 CA42YR 76314218 IC50 = 731 nM T97353 CXQ41E 76314219 IC50 > 10000 nM T97353 CUHZ51 76314232 IC50 = 667 nM T97353 COQ48X 76314233 IC50 = 1297 nM T97353 C1M7ZG 76317786 IC50 = 178 nM T97353 CIQ0T7 76317787 IC50 = 745 nM T97353 C1I6HO 76317788 IC50 = 1050 nM T97353 CSA72F 76317789 IC50 > 1000 nM T97353 CC3U8I 76317804 IC50 > 1000 nM T97353 C5UPA9 76317805 IC50 = 366 nM T97353 CBR9F0 76317806 IC50 = 36 nM T97353 CV23LI 76317807 IC50 > 5000 nM T97353 C0O4QY 76321498 IC50 = 101 nM T97353 CG7H4W 76321513 IC50 = 792 nM T97353 C1BQF4 76321514 IC50 = 38 nM T97353 C2ZH7K 76321515 IC50 = 497 nM T97353 CS9W7I 76321516 IC50 = 909 nM T97353 C7HC0P 76321517 IC50 > 4000 nM T97353 C8QH1P 76321518 IC50 = 731 nM T97353 CI9T5J 76325099 IC50 = 142 nM T97353 C2C6EW 76325100 IC50 > 4000 nM T97353 CSVC17 76325118 IC50 > 4000 nM T97353 CMH79B 76325119 IC50 = 12 nM T97353 C1HJO0 76325120 IC50 = 869 nM T97353 CCN7M6 76328682 IC50 = 1900 nM T97353 CP7AC0 76328683 IC50 > 5000 nM T97353 CX3Y7N 76328684 IC50 = 270 nM T97353 CZM19H 76332361 IC50 = 134 nM T97353 C18OJH 76332362 IC50 = 176 nM T97353 CA1LM2 76335971 IC50 = 106 nM T97353 C4I5DV 76335989 IC50 > 1000 nM T97353 CVI67F 90665342 EC50 = 2000 nM T19567 C3MA9U 342139 Ki = 3200 nM T19567 CDUE24 778225 IC50 < 200 nM T19567 CL16MS 822778 IC50 = 1000 nM T19567 CDX3Q5 5289024 Ki = 10 nM T19567 C7W8IX 5486943 Ki = 46 nM T19567 C3X1UJ 11507040 Ki = 600 nM T19567 C8N6MC 24808481 Ki = 420 nM T19567 C75WCL 52949691 Ki = 700 nM T19567 C54CBK 54585170 Ki = 5900 nM T19567 CTL94E 57520838 Ki = 9.4 nM T19567 CJQ9O0 57520839 Ki = 11 nM T19567 C8S9PM 57520840 Ki > 3000 nM T19567 C9G2HN 57520841 Ki = 50 nM T19567 C3N4MF 57520842 Ki = 29 nM T19567 CU4NZ2 57520938 Ki = 41 nM T19567 CD0M8V 57520940 Ki = 14 nM T19567 CCS1L3 57520941 Ki = 0.53 nM T19567 CEL56T 57520942 Ki = 20 nM T19567 CM6RX9 57520943 Ki = 9 nM T19567 C9Q4XE 57520944 Ki = 180 nM T19567 C1Z0LC 57520945 Ki = 1200 nM T19567 CE09OR 57520946 Ki = 200 nM T19567 C3Z6AE 57521037 Ki = 14 nM T19567 C6XB7H 57521039 Ki = 2.4 nM T19567 CXN9G4 57521040 Ki = 74 nM T19567 C9RU7B 57521041 Ki = 760 nM T19567 CC6UT9 57521043 Ki = 26 nM T19567 C78HYG 57521133 Ki = 0.36 nM T19567 C42KWH 57521134 Ki = 5.3 nM T19567 C9DFB0 57521135 Ki > 3000 nM T19567 C6SZ1P 57521138 Ki = 50 nM T19567 CR23AT 57521139 Ki = 58 nM T19567 CCQM76 59153288 Ki = 5.5 nM T19567 C4K2LU 59153299 Ki = 5.6 nM T19567 CK76DI 60202405 Ki = 2.8 nM T19567 C2LBW7 66551925 Ki = 190 nM T19567 C9CZS3 67205978 Ki = 70 nM T19567 C10MDK 69082696 Ki = 13 nM T19567 C39VMJ 69082892 Ki = 3.3 nM T19567 CYH83A 69083992 Ki = 1800 nM T19567 CT1PN0 69084444 Ki = 1700 nM T19567 CPV2D7 69085518 Ki = 960 nM T19567 CBZ82I 69085541 Ki = 72 nM T19567 CY2W3Z 69085646 Ki > 3000 nM T19567 C6BE5X 71271461 Ki = 270 nM T19567 C74PAB 86223063 Ki = 2200 nM T19567 CL0ZX5 86223064 Ki > 100000 nM T19567 CPT0J9 86275056 IC50 < 200 nM T19567 CIOU35 86275306 IC50 = 1000 nM T19567 CT4E5W 102436701 Ki = 4.1 nM T19567 C53VJW 135301646 IC50 = 3.715 nM T19567 C26OPR 135301656 IC50 = 147.91 nM T19567 CZVS32 135301671 IC50 = 3.89 nM T19567 CZJV94 135301685 IC50 = 18.2 nM T19567 CS4UK6 135301687 IC50 = 181.97 nM T19567 C9LA1K 135301762 IC50 = 20.42 nM T19567 CVW5G9 135301817 IC50 = 77.62 nM T19567 CG93EF 135301914 IC50 = 6.026 nM T19567 CGL0U2 135301919 IC50 = 13.18 nM T19567 C94GAU 135301927 IC50 = 2630.27 nM T19567 CY4MV6 135566354 Ki = 0.41 nM T19567 C4OVP2 136416802 Ki = 44 nM T19567 C7ZCT8 136416815 Ki = 69 nM T19567 C1OA7D 136416820 Ki = 0.55 nM T19567 C50OXS 136416829 Ki = 23 nM T19567 CX54DV 136416830 Ki = 28 nM T19567 CH94UL 136416849 Ki = 7.9 nM T19567 C9L0UB 136416923 Ki = 3 nM T19567 C0QWG9 142408858 IC50 = 10.23 nM T19567 CLZ91U 145971636 Ki > 200000 nM T19567 C4YPL9 145972068 Ki = 3460 nM T19567 CZVU97 155511644 Ki = 800 nM T19567 CMI8N3 155513321 Ki = 1600 nM T19567 C2CI4A 155514380 Ki = 600 nM T19567 CJ45PR 155520478 Ki = 2000 nM T19567 C95LZD 155522194 Ki = 700 nM T19567 CA35VB 155524076 Ki = 2100 nM T19567 C2QA1Z 155525301 Ki = 3200 nM T19567 C1E0UF 155535661 Ki = 3800 nM T19567 C2DI7E 155536657 IC50 = 3700 nM T19567 C3K1BZ 155537205 Ki = 15900 nM T19567 C9F2JN 155538608 Ki = 35 nM T19567 C5T9KE 155542416 Ki > 3000 nM T19567 C08TBV 155543421 IC50 = 223.87 nM T19567 C9S4MT 155549437 Ki = 1200 nM T19567 CAM36F 155550472 Ki = 3500 nM T19567 C3XE9Y 155554199 Ki = 900 nM T19567 C3WT2Q 155556441 Ki > 3000 nM T19567 C3PHB1 155557026 Ki = 2200 nM T19567 C3FA0E 155558092 Ki = 6700 nM T19567 C2I8VX 155559220 Ki = 8300 nM T19567 CUH07S 155560032 IC50 = 25000 nM T19567 CC5FE7 155564581 Ki > 3000 nM T19567 CB1V8A 155564612 Ki > 3000 nM T84621 D02STN 132971 IC50 = 1608 nM T84621 D02YPG 667484 IC50 = 0.5 nM T84621 D07ABV 468595 IC50 = 310 nM T84621 D09LNI 3365 IC50 = 30000 nM T84621 D0C1WH 3902 IC50 = 2620 nM T84621 D0Q9JT 4174 IC50 = 14.6 nM T84621 D0ZX1P 59693 IC50 = 6.3 nM T84621 D03AJU 44139752 IC50 = 2.5 nM T84621 D0D3PF 6918191 IC50 = 95000 nM T84621 D0SX7F 60876 Ki = 35 nM T84621 C9LCD8 3823 IC50 = 127 nM T84621 CFO8Y3 83332 IC50 = 24800 nM T84621 C78IXN 563347 IC50 = 246 nM T84621 CNG05O 571156 IC50 = 779 nM T84621 C5NT4U 583968 IC50 = 24 nM T84621 C1Y5HM 603115 IC50 = 16700 nM T84621 C8HZL4 618231 IC50 = 3 nM T84621 C7XD4N 706178 IC50 = 10200 nM T84621 CJ4FE1 853038 IC50 = 635 nM T84621 CI16RF 867617 IC50 = 500 nM T84621 CC29WP 886929 IC50 = 194 nM T84621 C6S1WJ 955210 IC50 > 1000 nM T84621 CB5KN2 1118253 IC50 = 14300 nM T84621 C83OBD 3021561 IC50 = 763 nM T84621 CBY4W2 3102914 IC50 > 1000 nM T84621 C1JAT6 6539761 IC50 = 715 nM T84621 CTE57C 6539762 IC50 = 1424 nM T84621 CF17BE 6539771 IC50 = 903 nM T84621 CJ7RS8 6539772 IC50 = 206 nM T84621 CQD13Z 6539787 IC50 = 143 nM T84621 CQ0HD5 6539812 IC50 = 58 nM T84621 CQ9XM0 6539813 IC50 = 26 nM T84621 CP51TH 6539814 IC50 = 96 nM T84621 CP4VI2 6540030 IC50 = 31.4 nM T84621 CR6LS8 6540031 IC50 = 3.3 nM T84621 CU3C1Y 6540034 IC50 = 6.9 nM T84621 CXEW82 6540035 IC50 = 15 nM T84621 CBKX32 6540037 IC50 = 18.7 nM T84621 C8MRI7 6540038 IC50 = 20.6 nM T84621 C8JXY1 6540039 IC50 = 11.17 nM T84621 CZK3T4 6540040 IC50 = 28.7 nM T84621 CDS26H 6540041 IC50 = 19.5 nM T84621 CX38PV 9927427 IC50 = 2 nM T84621 C64PHS 10083522 IC50 = 75000 nM T84621 CTH96I 10584844 IC50 = 5 nM T84621 CA13SW 10711620 IC50 = 79 nM T84621 CZW6V4 10828130 IC50 = 13.4 nM T84621 C6G3JV 11032034 IC50 = 47.86 nM T84621 C1TP7W 11232831 IC50 = 72 nM T84621 CN4T0K 11544009 IC50 = 4898 nM T84621 C9IJ3T 11594132 IC50 = 10505 nM T84621 CW2B3A 11738647 IC50 = 933 nM T84621 C27WEU 12229396 IC50 = 32 nM T84621 CCU19N 13045366 IC50 = 61 nM T84621 C4ELY3 13276694 IC50 = 2848 nM T84621 C1F5IT 13688212 IC50 = 40 nM T84621 C8WU6R 14424120 IC50 = 663 nM T84621 C8LSJ6 15182477 IC50 = 76000 nM T84621 CQ03PZ 16654684 IC50 = 816 nM T84621 CY0RV3 18668566 IC50 = 15 nM T84621 CRDM03 18679298 IC50 = 48 nM T84621 CN8IQ3 18785133 IC50 = 30.9 nM T84621 C1R2FU 22406650 IC50 = 253 nM T84621 C6D2NZ 24692916 IC50 = 1000 nM T84621 C07XJP 24696760 IC50 = 7500 nM T84621 CW3C5U 24896569 IC50 = 4329 nM T84621 C29WQM 25033651 IC50 = 291 nM T84621 C1VPF8 25033652 IC50 = 3109 nM T84621 C9Q8ZK 25033657 IC50 > 20000 nM T84621 CWIC10 25033659 IC50 > 10000 nM T84621 CAI47X 25033725 IC50 > 5000 nM T84621 C1XW6O 25033727 IC50 = 2135 nM T84621 CW5A1U 25033730 IC50 = 1159 nM T84621 CV49HP 25033731 IC50 = 686 nM T84621 C86AIT 25033734 IC50 > 10000 nM T84621 CEJ89P 25033804 IC50 = 2748 nM T84621 C3UF1V 25033806 IC50 = 1076 nM T84621 CF46OB 25033808 IC50 > 20000 nM T84621 CBI59C 25033810 IC50 = 1370 nM T84621 CV19DG 25034278 IC50 = 461 nM T84621 CEP93C 25034345 IC50 = 100 nM T84621 CSX16E 25034347 IC50 = 15 nM T84621 CXDF80 25034348 IC50 = 255 nM T84621 C56WJS 25034349 IC50 = 199 nM T84621 CGD93B 25034350 IC50 = 614 nM T84621 CK3L1J 25034351 IC50 = 1760 nM T84621 C9MF8O 25034425 IC50 = 99 nM T84621 CW7V9I 25034428 IC50 = 64 nM T84621 CH6U1E 25034429 IC50 = 248 nM T84621 CLP17I 25034432 IC50 = 875 nM T84621 CTB95M 25034489 IC50 = 41557 nM T84621 CBLS47 25034490 IC50 = 37796 nM T84621 CW82MN 25034491 IC50 = 31 nM T84621 CJ8M0E 25034492 IC50 = 435 nM T84621 COSJ63 25034493 IC50 = 10 nM T84621 C7KAR1 25034657 IC50 > 10000 nM T84621 C0MEI5 25129119 IC50 = 1956 nM T84621 C2QU1N 25129120 IC50 = 3559 nM T84621 C2FE6G 25129122 IC50 = 2452 nM T84621 CJ48LA 25129123 IC50 = 785 nM T84621 CX4GM7 25129462 IC50 = 24003 nM T84621 C9IFV2 25129463 IC50 = 19816 nM T84621 C6D8UQ 25129464 IC50 = 11307 nM T84621 CJCE15 25130854 IC50 = 1811 nM T84621 C9AS7H 25131165 IC50 = 2936 nM T84621 C9G8MJ 25131494 IC50 = 735 nM T84621 CA7OP2 25131495 IC50 = 9639 nM T84621 CZX08M 25142015 Ki = 15 nM T84621 C1WM2B 25147691 IC50 = 6.9 nM T84621 CYT15G 25180102 IC50 = 5970 nM T84621 CGX76Y 25180105 IC50 = 4371 nM T84621 CMU54R 25180107 IC50 = 290 nM T84621 C0XHA2 25180109 IC50 = 742 nM T84621 C9LQJ6 25180110 IC50 = 5177 nM T84621 CHJ2S3 25180298 IC50 = 339 nM T84621 C1HGB6 25180299 IC50 = 1671 nM T84621 C90UKD 25180304 IC50 = 1145 nM T84621 CPQ6A9 25180305 IC50 = 745 nM T84621 C6ZE9H 25180500 IC50 = 191 nM T84621 C6FN2Z 25180502 IC50 = 5402 nM T84621 C9DB1G 25180503 IC50 = 87 nM T84621 CIZ82U 25180504 IC50 = 769 nM T84621 CJS97E 30507078 IC50 = 5920 nM T84621 C70VMZ 44203017 IC50 = 1987 nM T84621 CT3XM4 44206480 IC50 = 116 nM T84621 C9UWB5 44206481 IC50 = 57 nM T84621 CDTS58 44387709 IC50 = 12.3 nM T84621 CT4L0R 44455927 IC50 = 19 nM T84621 C69QUY 44456068 IC50 > 1000 nM T84621 CM8BT1 44456104 IC50 = 110 nM T84621 C68FJH 44456188 IC50 = 167 nM T84621 CP50NM 44456189 IC50 = 329 nM T84621 CVR70K 44456190 IC50 = 782 nM T84621 C9JCL1 44456223 IC50 = 213 nM T84621 C6BE0T 44456226 IC50 = 107 nM T84621 CO4PI7 44479388 IC50 = 715 nM T84621 C1K6QY 44479389 IC50 = 2296 nM T84621 CLPH49 44479390 IC50 = 247 nM T84621 C2EM5N 44479391 IC50 = 13 nM T84621 CNTI30 44479392 IC50 = 545 nM T84621 C40IPE 44479393 IC50 = 34 nM T84621 C8JHS9 44479641 IC50 = 333 nM T84621 C2P4XT 44479643 IC50 = 158 nM T84621 CWP4Y8 44479644 IC50 = 141 nM T84621 C81QJE 44479645 IC50 = 1288 nM T84621 CO8T3N 44479646 IC50 = 2077 nM T84621 C4YN0S 44479648 IC50 = 28546 nM T84621 CF12OV 44479882 IC50 = 58 nM T84621 CCN58W 44479883 IC50 = 103 nM T84621 C7GV6X 44479884 IC50 = 17 nM T84621 CH8RO1 44479885 IC50 = 40 nM T84621 CES96D 44479886 IC50 = 490 nM T84621 CH02ZN 44480128 IC50 = 21 nM T84621 C1LSH2 44480129 IC50 = 1374 nM T84621 C3UQS0 44480130 IC50 = 43 nM T84621 C4KG5O 44480131 IC50 = 4646 nM T84621 COI7E8 44480132 IC50 = 496 nM T84621 C9KS5O 44480133 IC50 = 2058 nM T84621 CLMI41 44480134 IC50 = 128 nM T84621 CYH9A6 44480385 IC50 = 1312 nM T84621 C9V8CH 44480386 IC50 = 28 nM T84621 CL8KQ3 44480387 IC50 = 54 nM T84621 CT50NZ 44480388 IC50 = 796 nM T84621 CKO4N3 44480389 IC50 = 1692 nM T84621 CT3MO9 44480390 IC50 = 15 nM T84621 CN7LT2 44482245 IC50 = 776 nM T84621 CO63LK 44569291 IC50 = 152 nM T84621 CW06BV 45103704 IC50 = 104 nM T84621 C9Z4YB 45103705 IC50 = 123 nM T84621 CB2FC9 45103804 IC50 = 112.2 nM T84621 C4Q2FU 45103806 IC50 = 43.65 nM T84621 CQF56Z 45103807 IC50 = 12.02 nM T84621 C0RY2G 46233602 IC50 = 213 nM T84621 CUV83E 46854605 IC50 = 3100 nM T84621 CIA08B 46854608 IC50 = 37470 nM T84621 CWJ3F1 46854758 IC50 = 7300 nM T84621 CKRQ67 46854759 IC50 = 7180 nM T84621 CZ1YJ0 46854760 IC50 = 5060 nM T84621 CIC9S5 49799473 IC50 = 2000 nM T84621 C3Q6AS 49862488 IC50 = 26.1 nM T84621 CM43HV 49862547 IC50 = 50.2 nM T84621 CFDH59 49862548 IC50 = 103 nM T84621 CNIA98 49862549 IC50 = 544 nM T84621 CKY2J9 49862550 IC50 = 566 nM T84621 C0N4RT 49862551 IC50 = 930 nM T84621 CLI23H 49862552 IC50 = 122 nM T84621 CGU86D 49862599 IC50 = 55.7 nM T84621 CY8WD5 49862600 IC50 = 119 nM T84621 CS4IP9 49862601 IC50 = 76 nM T84621 C63XUS 49862602 IC50 = 204 nM T84621 C6O7JQ 49862603 IC50 = 471 nM T84621 C8G7FR 49862604 IC50 = 340 nM T84621 CP5D8Q 49862650 IC50 = 20.6 nM T84621 C6X0JA 49862651 IC50 = 222 nM T84621 C7BTK9 49862652 IC50 = 245 nM T84621 C79MQZ 49862653 IC50 = 234 nM T84621 CL8DR6 49862654 IC50 = 182 nM T84621 CMXR96 51355428 IC50 = 45 nM T84621 C5KTL3 51355429 IC50 = 40 nM T84621 C4UTM8 51355430 IC50 = 31 nM T84621 CH5C9K 51355431 IC50 = 20 nM T84621 CRK2Q9 51355432 IC50 = 5 nM T84621 CF7RG5 51355433 IC50 = 20 nM T84621 C41SUK 51355703 IC50 = 100 nM T84621 CM6T7H 51355704 IC50 = 80 nM T84621 CZDA87 51355705 IC50 = 25 nM T84621 CO1V0Y 51355706 IC50 = 45 nM T84621 C2OCG3 51355707 IC50 = 50 nM T84621 CIR0L7 51356252 IC50 = 933 nM T84621 CY69GL 52450897 IC50 = 188 nM T84621 CMTX50 52936939 IC50 = 2045 nM T84621 CC7Q8A 52936940 IC50 = 183 nM T84621 CTD3M1 52936941 IC50 = 1748 nM T84621 C98MZS 52937039 IC50 = 44 nM T84621 CZ72GJ 53316510 IC50 = 46 nM T84621 CR7L6V 53317838 IC50 = 80 nM T84621 CD9JL4 53319024 IC50 = 16100 nM T84621 CJBC94 53319146 IC50 > 1000 nM T84621 CYN7S9 53319147 IC50 = 43 nM T84621 C6WXT3 53320325 IC50 = 369 nM T84621 C20LRW 53320468 IC50 = 32 nM T84621 CU80BY 53320469 IC50 > 1000 nM T84621 C1SH0Q 53321768 IC50 > 1000 nM T84621 CEA3Y9 53321769 IC50 > 1000 nM T84621 C90DZC 53322953 IC50 = 5 nM T84621 CU1V2C 53323093 IC50 = 128 nM T84621 CYU1S5 53323094 IC50 > 1000 nM T84621 CS4A9O 53324450 IC50 = 46 nM T84621 C0B7TL 53325759 IC50 = 197 nM T84621 CVG4U6 53325760 IC50 = 4 nM T84621 CO68YD 53326854 IC50 = 75 nM T84621 C4NU2F 53475401 IC50 = 42 nM T84621 CAE25J 53763992 IC50 = 500 nM T84621 C51RVD 56645155 IC50 = 2857 nM T84621 CG06MB 56645361 IC50 = 401 nM T84621 CUS9L4 56645362 IC50 = 3984 nM T84621 C4N0WL 56645363 IC50 = 100 nM T84621 CTO1X9 56645364 IC50 = 370 nM T84621 C57NSZ 56645568 IC50 = 42 nM T84621 C6PUX9 56645570 IC50 = 435 nM T84621 CTW6K2 56645571 IC50 = 258 nM T84621 CX05HC 56645572 IC50 = 723 nM T84621 CPCW12 56645777 IC50 = 374 nM T84621 C32FWC 56645967 IC50 = 251 nM T84621 CXYW61 56645969 IC50 = 334 nM T84621 C2AP7F 56646158 IC50 = 435 nM T84621 CKWB83 56646160 IC50 = 477 nM T84621 CA3VO0 56949328 IC50 > 7500 nM T84621 CH8CP7 57329709 IC50 = 246 nM T84621 CQD5B4 57329785 IC50 = 76 nM T84621 C8GUF0 57329786 IC50 = 29 nM T84621 CE4YX9 57329787 IC50 = 40 nM T84621 CRAD59 57329788 IC50 = 72 nM T84621 CH8FQ9 57329789 IC50 = 101 nM T84621 C4USR5 57329791 IC50 = 62 nM T84621 C2C5PD 57329792 IC50 = 75 nM T84621 C3D8CZ 57329793 IC50 = 16 nM T84621 CKH02M 57329866 IC50 = 61 nM T84621 C30NOK 57329940 IC50 = 33 nM T84621 C37KZO 57329941 IC50 = 28 nM T84621 CZH28K 57329942 IC50 = 12 nM T84621 CR6EH0 57329943 IC50 = 151 nM T84621 CWN9V2 57329944 IC50 = 60 nM T84621 CFLA57 57330005 IC50 = 21 nM T84621 C2JR3S 57330006 IC50 = 11 nM T84621 C1EZM8 57330007 IC50 = 124 nM T84621 C5H2LE 57330008 IC50 = 69 nM T84621 C05XKT 57330009 IC50 = 98 nM T84621 C26GFC 57330010 IC50 = 32 nM T84621 CS38WC 57330011 IC50 = 6 nM T84621 C54EUF 57330012 IC50 = 1122 nM T84621 C4MN9B 57330078 IC50 = 1711 nM T84621 C5K3VT 57330079 IC50 = 240 nM T84621 C3LVG9 57330084 IC50 = 610 nM T84621 CMNH08 57330085 IC50 = 8 nM T84621 CY58ZD 57330086 IC50 = 2 nM T84621 C7OK1X 57775654 IC50 = 149 nM T84621 CB6RN7 58255346 IC50 = 50 nM T84621 CFXY47 58255349 IC50 = 29 nM T84621 C34JIZ 58255359 IC50 = 224 nM T84621 C7ZH6D 58255361 IC50 = 3.4 nM T84621 C2TUJ7 58255382 IC50 = 2.2 nM T84621 CMBV34 58255389 IC50 = 40 nM T84621 C3DPC0 58255407 IC50 = 40 nM T84621 C9DK1X 58255415 IC50 = 3737 nM T84621 CQEW75 58255430 IC50 = 144 nM T84621 CTI0D7 58255435 IC50 = 5399 nM T84621 C7L1NK 58255436 IC50 = 27 nM T84621 CRQ70M 58255438 IC50 = 1.4 nM T84621 C72VNQ 58255447 IC50 = 6.5 nM T84621 CLQ65O 58255479 IC50 = 347 nM T84621 CP6RA9 58255482 IC50 = 11940 nM T84621 C6DHG3 58255496 IC50 = 70 nM T84621 CAJ17Z 58255506 IC50 = 13 nM T84621 C7AX1R 58255531 IC50 = 110 nM T84621 CJX70M 58255566 IC50 = 745 nM T84621 C64JZC 58255572 IC50 = 438 nM T84621 CW71EO 58255581 IC50 = 2487 nM T84621 CYD9N5 58255637 IC50 = 20 nM T84621 CB7N8A 60195126 IC50 = 19 nM T84621 CX4N0I 62707515 IC50 = 790 nM T84621 CH3QU4 62918897 IC50 = 971 nM T84621 CE6L7O 65040275 IC50 > 10000 nM T84621 C0G3LA 66559847 IC50 = 1098 nM T84621 C4RSI6 66559935 IC50 = 1077 nM T84621 CDX7I8 66559936 IC50 = 1167 nM T84621 CF9EQ5 66559939 IC50 = 1422 nM T84621 CQN6D3 66559940 IC50 = 16170 nM T84621 CN4H8G 66559941 IC50 = 4087 nM T84621 CTP6Q4 66559942 IC50 = 4589 nM T84621 C9EGW2 66575742 IC50 = 3570 nM T84621 CMXA10 66575743 IC50 = 1770 nM T84621 CKWB91 66575744 IC50 = 110 nM T84621 C7I3MW 66575745 IC50 = 16990 nM T84621 CPN17S 66575746 IC50 = 12620 nM T84621 CG0ZA7 66575747 IC50 = 16100 nM T84621 C6HF0U 66575748 IC50 = 7900 nM T84621 CEW4O6 66575816 IC50 = 17296 nM T84621 CDI93T 66575817 IC50 = 428 nM T84621 C6B7PN 66576767 IC50 = 407 nM T84621 CYHS25 66576769 IC50 = 1501 nM T84621 CBP6I7 66576773 IC50 = 2198 nM T84621 CM6U5S 66576848 IC50 > 30000 nM T84621 CNB21T 66576849 IC50 > 10000 nM T84621 C2PFB6 66576850 IC50 > 10000 nM T84621 CDU8R7 66576852 IC50 = 6930 nM T84621 C4NYB0 66576930 IC50 = 1810 nM T84621 C3LP5H 66576931 IC50 = 3910 nM T84621 CE03WG 66576932 IC50 = 6970 nM T84621 CVZ4E0 66692998 IC50 > 10000 nM T84621 C1RLT0 67199421 IC50 = 3451 nM T84621 CC34QF 67509960 IC50 = 21 nM T84621 CQL7H6 67510362 IC50 = 167 nM T84621 CN9VU2 67510431 IC50 = 320 nM T84621 C40FEA 67511528 IC50 = 362 nM T84621 C2MH1G 67515607 IC50 = 126 nM T84621 CC4A7Z 67515696 IC50 = 106 nM T84621 CE27NZ 67515801 IC50 = 782 nM T84621 CZCW84 67515869 IC50 = 362 nM T84621 CKJN74 67515874 IC50 = 409 nM T84621 CW20PM 67516106 IC50 = 502 nM T84621 C14VNF 67516160 IC50 = 1000 nM T84621 CL0XQ7 67516179 IC50 = 971 nM T84621 CM7Z1T 67516370 IC50 = 95 nM T84621 CK1LB2 67516475 IC50 = 542 nM T84621 C5VM6T 67516855 IC50 = 139 nM T84621 CQ0NP7 68053462 IC50 > 10000 nM T84621 CV72CY 68053552 IC50 = 1980 nM T84621 CVF40X 68053622 IC50 = 1831 nM T84621 CG0T8B 68053623 IC50 = 2101 nM T84621 CU76KO 68053624 IC50 > 8333 nM T84621 CYZK18 68053631 IC50 > 8333 nM T84621 CSI12Z 68053632 IC50 > 10000 nM T84621 C0N3IK 68053729 IC50 = 17.7 nM T84621 C19JSA 68053730 IC50 = 250 nM T84621 C5N2MQ 68053837 IC50 = 677 nM T84621 CCJT39 68053838 IC50 = 3923 nM T84621 CF32HJ 70680985 IC50 = 500 nM T84621 CPB63L 70680997 IC50 = 73 nM T84621 CE78SM 70683110 IC50 = 168 nM T84621 CM6LN8 70683111 IC50 = 246 nM T84621 CK0DY6 70683112 IC50 = 611 nM T84621 C9E4ZQ 70685192 IC50 = 269 nM T84621 CW5F3G 70691516 IC50 = 500 nM T84621 C1VMF2 70977969 IC50 = 29540 nM T84621 C70TUP 71455138 IC50 = 139 nM T84621 CFG4L5 71456934 IC50 = 44 nM T84621 CI16NC 71520311 IC50 = 1336 nM T84621 CE9A6B 71520312 IC50 > 5000 nM T84621 C03VKJ 71520313 IC50 = 750 nM T84621 C5J7DI 71520314 IC50 = 16 nM T84621 CE0N5C 71520315 IC50 = 41 nM T84621 C4Z6YP 71520316 IC50 = 1230 nM T84621 CC8Z6L 71520431 IC50 = 4 nM T84621 C1DK9P 71520432 IC50 = 140 nM T84621 C9NOQ1 71521632 IC50 = 68 nM T84621 C0OTA2 71521716 IC50 = 2270 nM T84621 CVLE07 71521717 IC50 = 1220 nM T84621 CJKX84 71521718 IC50 = 36 nM T84621 CZ5P9U 71521719 IC50 = 78 nM T84621 C1YCB0 71521720 IC50 = 1420 nM T84621 CE57PM 71521721 IC50 > 5000 nM T84621 C0O2SA 71521798 IC50 = 276 nM T84621 CMEC10 71521799 IC50 = 2539 nM T84621 CR9O5T 71521800 IC50 = 1688 nM T84621 C0JBI3 71521801 IC50 = 532 nM T84621 CE7Z4I 71521802 IC50 = 88 nM T84621 CW2AG4 71521803 IC50 = 646 nM T84621 C6ID7K 71521804 IC50 = 92 nM T84621 CO5BE7 71535395 IC50 = 280 nM T84621 CCF8Z7 71535398 IC50 = 530 nM T84621 CC16AO 71535399 IC50 = 590 nM T84621 CPZ5S8 71535400 IC50 = 100 nM T84621 CI4W5N 71535682 IC50 = 490 nM T84621 CCRS95 71535683 IC50 = 1800 nM T84621 C58SMB 71574941 IC50 = 0.5 nM T84621 CC09FQ 71574942 IC50 = 19.2 nM T84621 CA2T5L 71574943 IC50 = 156.3 nM T84621 C9MFZ7 71574944 IC50 = 80.1 nM T84621 CW73OE 71574945 IC50 = 25.4 nM T84621 C70NHJ 71574946 IC50 = 92.5 nM T84621 CLH83S 71574947 IC50 = 24.4 nM T84621 CF71AB 71575030 IC50 = 13.1 nM T84621 CCG1S5 71575031 IC50 = 5.5 nM T84621 CH9WE7 71575032 IC50 = 268.4 nM T84621 CO4ZQ7 71575033 IC50 = 415.8 nM T84621 CT86GV 71575034 IC50 = 785.3 nM T84621 CKPV51 71621803 IC50 > 100000 nM T84621 CG09JH 71716351 IC50 = 72 nM T84621 C56LUJ 71716957 IC50 = 219 nM T84621 CJE01S 71745100 IC50 = 4520 nM T84621 CX0WV5 71817943 IC50 = 235 nM T84621 CN1LU6 71817944 IC50 = 1609 nM T84621 CGV4U3 71817945 IC50 = 1159 nM T84621 CJ4L5G 71818086 IC50 = 2935 nM T84621 COXA51 71818087 IC50 = 224 nM T84621 CP1A3M 71818088 IC50 = 1415 nM T84621 CPJ42T 71818089 IC50 = 450 nM T84621 CAP03I 71818090 IC50 = 447 nM T84621 CO23PK 71818091 IC50 = 245 nM T84621 CL4X6A 71818092 IC50 = 7099 nM T84621 CL8GK5 71818093 IC50 = 2824 nM T84621 C4ZVG0 71818094 IC50 = 362 nM T84621 CH2GR0 71818232 IC50 = 238 nM T84621 C0VGQ9 71818233 IC50 = 12286 nM T84621 C5QRF2 71818234 IC50 = 2426 nM T84621 CCG7R3 72703685 IC50 = 250 nM T84621 CAU4Z0 72703889 IC50 = 1010 nM T84621 C56KEC 72703890 IC50 = 1480 nM T84621 C4AEX3 73347616 IC50 = 38 nM T84621 CFD46C 73347617 IC50 = 5 nM T84621 C26LJW 73347618 IC50 = 1015 nM T84621 CIHF35 73350707 IC50 = 51 nM T84621 CT26EZ 73355186 IC50 > 5000 nM T84621 C0NXU4 73355187 IC50 = 87 nM T84621 CML29U 73355188 IC50 = 427 nM T84621 CC5TO4 73356735 IC50 = 125 nM T84621 CWZ3A1 73356736 IC50 = 1.3 nM T84621 C9CY3K 73442767 IC50 = 34 nM T84621 CU6IQ9 73603293 IC50 = 4737 nM T84621 C6MQ8L 73603294 IC50 > 5000 nM T84621 CR81XZ 73603295 IC50 = 1423 nM T84621 CJS6Y2 73603296 IC50 > 5000 nM T84621 C1GR7W 73603297 IC50 > 5000 nM T84621 CM4L6N 73603298 IC50 = 1523 nM T84621 CAIB62 73603299 IC50 > 5000 nM T84621 C7G6KZ 73603343 IC50 = 52 nM T84621 CDX9R1 73603344 IC50 = 516 nM T84621 C7KV2S 73603345 IC50 = 6093 nM T84621 CM10ZX 73603346 IC50 = 3723 nM T84621 CJSY07 73603348 IC50 = 1379 nM T84621 CS03UP 73603349 IC50 = 6812 nM T84621 C56LYP 73603350 IC50 = 6642 nM T84621 C9RKH0 73603387 IC50 = 803 nM T84621 CG86BD 73603388 IC50 = 3125 nM T84621 C2R3ZB 73603389 IC50 = 3756 nM T84621 C5ARE7 73603390 IC50 = 160 nM T84621 CTMF86 73603391 IC50 = 366 nM T84621 C5RG4C 75593332 IC50 = 10.74 nM T84621 CMN51L 76286753 IC50 > 8300 nM T84621 C06HYT 76286902 IC50 = 1299 nM T84621 CPU3T6 76317295 IC50 = 7.2 nM T84621 CZ2U9K 76321000 IC50 = 1.5 nM T84621 C4UO5H 76331904 IC50 < 0.1 nM T84621 CP10SN 76335488 IC50 = 0.3 nM T84621 C1YJW0 77846787 IC50 = 32 nM T84621 CV73PD 77846790 IC50 = 82 nM T84621 C0DIH7 77846872 IC50 = 17 nM T84621 COI25M 77846873 IC50 = 67 nM T84621 CJI8R0 77846875 IC50 = 29 nM T84621 CZK4J1 77846962 IC50 = 70 nM T84621 CEK89G 77846963 IC50 = 110 nM T84621 C5BA8Z 77846964 IC50 = 187 nM T84621 C4D6XJ 77847803 IC50 = 63 nM T84621 CF7O4Q 77847804 IC50 = 40 nM T84621 C2ASY0 86730379 IC50 = 880 nM T84621 CA4QV9 86730380 IC50 = 33 nM T84621 C24ZMT 86730381 IC50 = 37 nM T84621 C9W6RO 86730382 IC50 = 600 nM T84621 C3UMP9 89471867 IC50 = 640 nM T84621 CW8TF6 89471869 IC50 = 300 nM T84621 CL30TR 89471870 IC50 = 760 nM T84621 CJ0H5V 89471872 IC50 = 1100 nM T84621 C3BUS8 89471889 IC50 = 930 nM T84621 CI7HY8 89471890 IC50 = 800 nM T84621 CF2AY7 89471891 IC50 > 8700 nM T84621 CQF07X 89471892 IC50 = 830 nM T84621 C62KFZ 89961587 IC50 > 10000 nM T84621 C8XS2I 89961629 IC50 = 317 nM T84621 C75PMO 89961672 IC50 > 8333 nM T84621 CX0M7B 89961716 IC50 = 1357 nM T84621 C3JN5I 89961721 IC50 > 10000 nM T84621 CSJT14 89961765 IC50 = 1473 nM T84621 CR5D6Y 89961785 IC50 > 10000 nM T84621 C7TI3V 89961787 IC50 > 8333 nM T84621 C2QP7I 89961848 IC50 > 10000 nM T84621 C81FEN 89961879 IC50 > 10000 nM T84621 CI6P0R 89961978 IC50 > 8333 nM T84621 C89TEU 89968659 IC50 = 5705 nM T84621 C7BC5N 89968688 IC50 > 10000 nM T84621 C3XIF5 90252771 IC50 = 1.1 nM T84621 CGZ2S1 90252806 IC50 = 470 nM T84621 C4F9VB 90252809 IC50 = 1400 nM T84621 CE2TM0 90252810 IC50 > 8300 nM T84621 CGVL78 90252811 IC50 > 8300 nM T84621 C0S3HV 90252812 IC50 = 916 nM T84621 C4M8TO 90252814 IC50 = 1200 nM T84621 CM0T2X 90252815 IC50 > 8300 nM T84621 CY5IC7 90252834 IC50 = 98 nM T84621 CF05JI 90252835 IC50 = 1000 nM T84621 C72ICB 90252839 IC50 > 8300 nM T84621 C84NVA 90252850 IC50 = 338 nM T84621 CBY46O 90252851 IC50 = 856 nM T84621 CNVA50 90252852 IC50 = 386 nM T84621 C0Z2TI 90252864 IC50 = 47 nM T84621 CV30CD 90252953 IC50 = 535 nM T84621 C3MV7S 90252954 IC50 = 1690 nM T84621 CD5ST8 90252956 IC50 > 8300 nM T84621 C3JH4P 90252957 IC50 > 8300 nM T84621 CCU4F7 90252958 IC50 = 1987 nM T84621 C89BFG 90333640 IC50 = 58 nM T84621 C82YUB 90644545 IC50 = 302 nM T84621 CVFA18 90644546 IC50 = 736 nM T84621 CR50EN 90644547 IC50 = 61 nM T84621 C46ZNM 90644548 IC50 = 435 nM T84621 CS6N1P 90644549 IC50 = 4100 nM T84621 CB5HI4 90644550 IC50 = 2300 nM T84621 CHD21I 90666137 IC50 = 21.2 nM T84621 CLB2E7 91827654 IC50 = 4402 nM T84621 C5GV1L 101882447 IC50 = 5 nM T84621 CMH51N 118496543 IC50 = 779 nM T84621 C3ZPQ1 118496545 IC50 = 149 nM T84621 CJ9Z0S 118496546 IC50 = 22 nM T84621 C7UN3R 118496547 IC50 = 197 nM T84621 CJ54UQ 118618017 IC50 = 872 nM T84621 CLS25A 118714825 IC50 = 111 nM T84621 CT0FH7 118714826 IC50 = 327 nM T84621 CD8T1P 118714827 IC50 = 1674 nM T84621 C85BVO 118714828 IC50 = 690 nM T84621 CYFP62 118714829 IC50 = 499 nM T84621 CE3ZF1 118714830 IC50 = 2003 nM T84621 C5HKE1 118714831 IC50 = 1750 nM T84621 C7BD3X 118714832 IC50 = 587 nM T84621 C9BM7X 118714833 IC50 = 188 nM T84621 CML4K7 118714834 IC50 = 68 nM T84621 CE5L8U 118714835 IC50 = 2001 nM T84621 CD8YA9 118714836 IC50 > 5000 nM T84621 CRNL64 118714837 IC50 = 28 nM T84621 C4F6AY 118714838 IC50 = 65 nM T84621 CZ9L5S 118714839 IC50 = 334 nM T84621 CU3XP2 118714840 IC50 = 26 nM T84621 C0BRP1 118714841 IC50 = 278 nM T84621 C6M5VU 118714842 IC50 = 382 nM T84621 CQ5KI0 118714843 IC50 = 929 nM T84621 C32MDK 118714844 IC50 = 71 nM T84621 C15PAW 118714845 IC50 = 49 nM T84621 CPH51S 118714846 IC50 = 62 nM T84621 C1L4YZ 118714847 IC50 = 137 nM T84621 CLM64U 118714848 IC50 = 309 nM T84621 C5UD3K 118714849 IC50 = 1224 nM T84621 CNW8E3 118714850 IC50 = 65 nM T84621 CMXG03 118714851 IC50 = 114 nM T84621 CTWO23 118714852 IC50 = 60 nM T84621 CAW36P 118714853 IC50 = 663 nM T84621 C4Y2UF 118714854 IC50 = 1167 nM T84621 CJK08Q 118714855 IC50 = 6 nM T84621 CP4O0C 118720463 IC50 = 6712 nM T84621 CV4IC9 118720464 IC50 = 4196 nM T84621 CKG28R 118720465 IC50 = 7315 nM T84621 CGXD81 118720466 IC50 = 1096 nM T84621 CF1W7I 118720467 IC50 = 8947 nM T84621 COZU39 118720468 IC50 = 4797 nM T84621 CWG6L8 118720469 IC50 = 4487 nM T84621 C2HV3Y 118720470 IC50 = 5549 nM T84621 CX56BZ 118720471 IC50 = 6548 nM T84621 CO8H3J 118720472 IC50 = 7427 nM T84621 C7WEQ3 118720473 IC50 = 5812 nM T84621 CG8PB5 118720474 IC50 = 4710 nM T84621 CN2U6B 118720475 IC50 = 6189 nM T84621 CU7FW1 118720476 IC50 = 6674 nM T84621 CCJ17Z 118720477 IC50 = 5076 nM T84621 CB4DS9 118720479 IC50 = 8550 nM T84621 CC9V6K 118720480 IC50 = 8333 nM T84621 CP7X1B 118720481 IC50 = 9346 nM T84621 CPT58L 118720482 IC50 = 4717 nM T84621 C3E7TA 118720483 IC50 = 6534 nM T84621 CS01NU 118720484 IC50 = 6164 nM T84621 CAW5K3 118723935 IC50 = 48 nM T84621 CK8UL1 118723936 IC50 = 111 nM T84621 CIW7O0 118723937 IC50 = 63 nM T84621 C42CEZ 118723938 IC50 = 48 nM T84621 CJQ63E 118723939 IC50 = 258 nM T84621 CCXN71 118723940 IC50 = 57 nM T84621 CS78BD 118723941 IC50 = 50 nM T84621 C9W3QX 118723942 IC50 > 500 nM T84621 COJ2K8 118723943 IC50 = 15 nM T84621 CZ23UL 118723944 IC50 = 24 nM T84621 CIWU64 118723945 IC50 = 30 nM T84621 CZI6A0 118723946 IC50 = 109 nM T84621 COB46M 118723947 IC50 = 518 nM T84621 CYM08W 118726850 IC50 = 120 nM T84621 CR32JU 118726851 IC50 = 4.5 nM T84621 C2OAI6 118726852 IC50 = 7483 nM T84621 CDHI10 118733086 IC50 > 10000 nM T84621 C18PWB 118733087 IC50 > 10000 nM T84621 C8WJ2Y 118733088 IC50 > 10000 nM T84621 C31ZXP 118733089 IC50 > 10000 nM T84621 CHR84E 118733090 IC50 > 10000 nM T84621 CAQ72M 118733091 IC50 > 10000 nM T84621 CIV1Z5 118733092 IC50 > 10000 nM T84621 CU3Y9W 118733093 IC50 > 10000 nM T84621 CF49NU 118733094 IC50 > 10000 nM T84621 CK73VU 118733095 IC50 > 10000 nM T84621 CR1WU5 118733096 IC50 > 10000 nM T84621 C1V7WI 118735163 IC50 = 279 nM T84621 C6YG9R 118735164 IC50 = 1207 nM T84621 C5C4FZ 118735165 IC50 = 540 nM T84621 C1ZLM6 118735166 IC50 = 23 nM T84621 CQXM57 118735167 IC50 = 13 nM T84621 C0RYM4 118735168 IC50 = 6 nM T84621 C0DCB9 118735169 IC50 = 50 nM T84621 CG4QF3 118735170 IC50 = 2 nM T84621 CD3IY5 118735171 IC50 = 8 nM T84621 C0JZ2Y 118735172 IC50 = 508 nM T84621 C2WS7A 118735173 IC50 = 1201 nM T84621 CYEA24 118735174 IC50 = 51 nM T84621 CZ9X4J 118735175 IC50 = 60 nM T84621 CG14RD 118735176 IC50 = 183 nM T84621 CQ3KR4 118735177 IC50 = 46 nM T84621 C1Z9FX 118735178 IC50 = 812 nM T84621 C2VJU4 118735179 IC50 = 26 nM T84621 CXWH51 118735180 IC50 = 38 nM T84621 C3YUS9 118735181 IC50 = 12 nM T84621 CEH97S 118735182 IC50 = 594 nM T84621 C03HKR 118735183 IC50 = 1150 nM T84621 CC38HG 118735184 IC50 = 1665 nM T84621 C8QIC4 118735185 IC50 = 2665 nM T84621 CZET62 118735186 IC50 = 182 nM T84621 CZ8U2C 118735187 IC50 = 6 nM T84621 CUAE09 121004872 IC50 > 8333 nM T84621 C1OT4E 121458684 IC50 = 1552 nM T84621 C9ETN3 121458685 IC50 = 795 nM T84621 C4V2HU 121458987 IC50 = 225 nM T84621 CPGD72 121458994 IC50 = 117 nM T84621 CXW13O 122179553 IC50 > 10000 nM T84621 C3E0VM 122179554 IC50 > 10000 nM T84621 CJVX13 122179555 IC50 > 8333 nM T84621 CWN9K7 122179556 IC50 > 10000 nM T84621 CV2PQ1 122191831 IC50 > 8333 nM T84621 C2AHB5 122191832 IC50 > 8333 nM T84621 CFZH01 122191833 IC50 > 8333 nM T84621 C1XKA8 122191834 IC50 > 8333 nM T84621 CG4S8F 122191835 IC50 = 887 nM T84621 C37NLK 122191836 IC50 > 8333 nM T84621 CVT7A2 127027254 IC50 = 86.9 nM T84621 C5QNG6 127027265 IC50 > 10000 nM T84621 CIZO64 127027266 IC50 > 10000 nM T84621 C9RXH3 127027267 IC50 > 10000 nM T84621 CEM84R 127027569 IC50 = 1600.8 nM T84621 CT83ZE 127027570 IC50 = 326.9 nM T84621 CHZ54G 127027571 IC50 = 29.5 nM T84621 C2ZFR8 127027572 IC50 = 108.9 nM T84621 CV1BD6 127027573 IC50 = 9.7 nM T84621 C0E6DW 127027574 IC50 > 10000 nM T84621 C2MFJ8 127027575 IC50 > 10000 nM T84621 CM8T9G 127028498 IC50 = 612.3 nM T84621 CQO36B 127028499 IC50 = 58.1 nM T84621 C1M7GD 127028500 IC50 = 222.5 nM T84621 CN42BR 127028817 IC50 = 82.7 nM T84621 C3IMJ8 127028818 IC50 = 179.6 nM T84621 CPEM69 127028819 IC50 = 372.1 nM T84621 C70XOB 127030295 IC50 = 3598.4 nM T84621 CZ7L4J 127031191 IC50 > 10000 nM T84621 C49IME 127031799 IC50 = 88.2 nM T84621 CHS8L7 131982520 IC50 = 1900 nM T84621 C95PYQ 131982530 IC50 = 350 nM T84621 C5IWD9 131982539 IC50 = 2400 nM T84621 CSIP72 131982576 IC50 < 100 nM T84621 CS8C7T 131982729 IC50 = 1100 nM T84621 CHDP80 131982862 IC50 = 410 nM T84621 C1BNU6 131982871 IC50 > 10000 nM T84621 C6CB0I 132585204 IC50 = 2 nM T84621 C7SM9W 134129925 IC50 = 387 nM T84621 CB3EL1 134134056 IC50 = 1595 nM T84621 CB79AO 134134186 IC50 = 1308 nM T84621 CPZX32 134135994 IC50 = 10000 nM T84621 CS2P0E 134136577 IC50 = 2192 nM T84621 CH3V9Q 134139925 IC50 = 460 nM T84621 CFUE13 134141128 IC50 = 1573 nM T84621 COUK40 134141967 IC50 = 1996 nM T84621 CX3Y9D 134142597 IC50 = 1674 nM T84621 CQF59S 134143092 IC50 = 787 nM T84621 C1HG8V 134144349 IC50 = 1739 nM T84621 CFC8O6 134145376 IC50 = 220 nM T84621 C31WNO 134145695 IC50 > 8000 nM T84621 C7JEU2 134148873 IC50 = 250 nM T84621 C2JOB5 134152002 IC50 = 1544 nM T84621 CTXL17 134153274 IC50 = 1000 nM T84621 C3OLF2 134153424 IC50 > 8000 nM T84621 C12LPH 134153935 IC50 = 355 nM T84621 C8ROI0 134153997 IC50 = 630 nM T84621 CDV8M5 134155385 IC50 = 4600 nM T84621 C74ONC 134156861 IC50 = 4460 nM T84621 CKL9N7 135185757 IC50 = 4629 nM T84621 C8HTS7 135185761 IC50 > 10000 nM T84621 C1D4CS 135185764 IC50 = 5380 nM T84621 CMQC50 135185766 IC50 = 378 nM T84621 CIS5H8 135185771 IC50 = 4157 nM T84621 CF0EC1 135185786 IC50 = 4325 nM T84621 C8GB5V 135185787 IC50 = 2035 nM T84621 CH30EN 135185789 IC50 = 3330 nM T84621 CMR5C9 135185792 IC50 = 3926 nM T84621 CX97YM 135185793 IC50 = 1907 nM T84621 CS5FX2 135185796 IC50 = 2267 nM T84621 CV9RM5 135185801 IC50 = 4987 nM T84621 C8MF2Z 135185815 IC50 = 390 nM T84621 CX57GP 135185833 IC50 = 4809 nM T84621 CSZA19 135185836 IC50 = 5723 nM T84621 C6G1CH 135185858 IC50 = 4771 nM T84621 C9LU0C 135185886 IC50 = 4171 nM T84621 CZ1JS3 135186252 IC50 > 10000 nM T84621 CWU63C 136008115 IC50 = 17 nM T84621 CAV9U3 136219390 IC50 = 230 nM T84621 CC7LY3 136239517 IC50 = 960 nM T84621 C2V0IM 136244612 IC50 = 75 nM T84621 CYIF59 136245971 IC50 > 5000 nM T84621 CM97FH 137631528 IC50 = 48 nM T84621 C9LY0O 137631806 IC50 = 1 nM T84621 CH05YR 137633095 IC50 = 20 nM T84621 COG72W 137633343 IC50 = 93 nM T84621 C3QE1V 137633417 IC50 = 3 nM T84621 CVM54L 137634483 IC50 = 4 nM T84621 CV2S5Q 137637282 IC50 = 110 nM T84621 CUIX95 137637496 IC50 = 210 nM T84621 C14LXC 137638585 IC50 = 13 nM T84621 C1D0WG 137638612 IC50 = 9 nM T84621 CF1D5C 137639549 IC50 = 11 nM T84621 C8V7CD 137639692 IC50 = 6 nM T84621 C1SH2M 137639834 IC50 = 1.8 nM T84621 CZA2S8 137639890 IC50 = 14 nM T84621 C0N4PJ 137640302 IC50 = 124 nM T84621 COEV02 137642385 IC50 = 16 nM T84621 CH35RE 137642529 IC50 = 0.6 nM T84621 CP1EJ0 137642735 IC50 = 22 nM T84621 C29FMO 137642787 IC50 = 137 nM T84621 COGQ01 137644314 IC50 = 16 nM T84621 CA73KP 137644560 IC50 = 150 nM T84621 C4UP3J 137647900 IC50 = 2 nM T84621 CI31EQ 137649226 IC50 = 516 nM T84621 CS5BW7 137650545 IC50 = 4 nM T84621 CF71RE 137650772 IC50 = 104 nM T84621 CQ54YG 137651298 IC50 = 5 nM T84621 C4CL2W 137651728 IC50 = 42 nM T84621 CK7QJ4 137651744 IC50 = 2 nM T84621 CI5D2P 137652926 IC50 = 5 nM T84621 CIH34U 137653629 IC50 = 520 nM T84621 CV9I5G 137653991 IC50 = 13 nM T84621 C28VRO 137654883 IC50 = 19 nM T84621 CEV94S 137655303 IC50 = 148 nM T84621 CY5IK7 137655531 IC50 = 2 nM T84621 CUL37V 137655879 IC50 = 1 nM T84621 CN2CQ1 137656473 IC50 = 62 nM T84621 C53NVI 137657989 IC50 = 3 nM T84621 CNI0C1 137658011 IC50 = 42 nM T84621 C32WHO 137658276 IC50 = 181 nM T84621 C0G2UI 137658690 IC50 = 58 nM T84621 CLNU74 137659288 IC50 = 57 nM T84621 CA5LI1 137659926 IC50 = 14 nM T84621 C7YI9N 137660712 IC50 = 10 nM T84621 CFU1Z3 145960404 IC50 = 130 nM T84621 C1IU5W 145960520 IC50 = 1200 nM T84621 CQFH90 145960862 IC50 = 590 nM T84621 CNIB73 145960902 IC50 = 480 nM T84621 C0KNY4 145961099 IC50 < 100 nM T84621 CGI39P 145961215 IC50 = 2100 nM T84621 CW84OQ 145961259 IC50 > 10000 nM T84621 C92JOV 145961758 IC50 > 10000 nM T84621 CR6JH8 145961916 IC50 = 2200 nM T84621 CS4EO5 145962296 IC50 = 180 nM T84621 C1O0NQ 145962517 IC50 = 5700 nM T84621 C6VO0A 145962577 IC50 < 100 nM T84621 CY20CQ 145962664 IC50 > 10000 nM T84621 C6F7UE 145962949 IC50 = 58 nM T84621 C5O4RQ 145963242 IC50 > 10000 nM T84621 CGA01F 145963470 IC50 = 470 nM T84621 CH0TM7 145963574 IC50 > 10000 nM T84621 C0TZR1 145964456 IC50 = 19.2 nM T84621 CRJM82 145965429 IC50 = 6.6 nM T84621 CN7B1I 145968025 IC50 = 12.3 nM T84621 C82JTH 145971322 IC50 = 11.4 nM T84621 C5R6SH 145973507 IC50 = 5.8 nM T84621 C41LQE 145976039 IC50 = 4.7 nM T84621 C01TYI 145976345 IC50 = 15.4 nM T84621 CG23BW 145977901 IC50 = 6.5 nM T84621 C65ZFY 145978611 IC50 = 4.1 nM T84621 CI48QV 145979205 IC50 = 77 nM T84621 C9IQK7 145980859 IC50 = 17 nM T84621 CCKL25 145981178 IC50 = 120 nM T84621 CY4G3E 145981780 IC50 = 0.8 nM T84621 CYI3V5 145988023 IC50 = 29 nM T84621 CH6DJ3 155527950 IC50 = 4523 nM T84621 C80XNT 155530085 IC50 = 1668 nM T84621 C5XB1F 155530577 IC50 > 10000 nM T84621 C6DXN8 155559405 IC50 > 10000 nM T84621 C4UQS2 155564575 IC50 > 10000 nM T84621 CXM62E 155566406 IC50 = 9072 nM T84621 D00BVP 11847320 IC50 = 7 nM T84621 D00DSE 49864196 IC50 = 928 nM T84621 D00DUJ 11687499 IC50 = 7553 nM T84621 D00PXF 44206698 IC50 = 32.36 nM T84621 D01JZO 2779191 IC50 = 1000 nM T84621 D01REI 46901610 IC50 = 1400 nM T84621 D01SUE 6539759 IC50 = 888 nM T84621 D01SZX 46867545 IC50 = 99.1 nM T84621 D02ALK 11514074 IC50 = 2671 nM T84621 D02BXS 46901445 IC50 = 902 nM T84621 D02CSU 6539786 IC50 = 931 nM T84621 D02GFK 25034431 IC50 = 1521 nM T84621 D02JUJ 25034344 IC50 = 8925 nM T84621 D02LWB 6540046 IC50 = 2391 nM T84621 D02NAG 6539765 IC50 = 1472 nM T84621 D02PSL 45103913 IC50 = 6.166 nM T84621 D02UZI 6540056 IC50 = 288 nM T84621 D02XHH 6540043 IC50 = 23.5 nM T84621 D02ZQM 25180104 IC50 = 4921 nM T84621 D03CWL 14535954 IC50 = 323.59 nM T84621 D03EXD 49864181 IC50 = 251 nM T84621 D03KLN 11413434 IC50 = 81 nM T84621 D03MKT 6539788 IC50 = 1098 nM T84621 D03TRM 6540032 IC50 = 25.9 nM T84621 D03VRC 2989557 IC50 = 211 nM T84621 D03YHZ 25147692 IC50 = 33 nM T84621 D04CFP 46901927 IC50 = 469 nM T84621 D04CLL 6539775 IC50 = 763 nM T84621 D04ELJ 6539766 IC50 = 270 nM T84621 D04IBH 11616637 IC50 = 4481 nM T84621 D04ISG 11680597 IC50 = 2724 nM T84621 D04PKP 23644953 IC50 = 2896 nM T84621 D04QPK 6539783 IC50 = 774 nM T84621 D04WJN 10588478 IC50 = 70.8 nM T84621 D05FFY 14231155 IC50 = 141 nM T84621 D05IXU 25130517 IC50 = 953 nM T84621 D05MQE 6539785 IC50 = 657 nM T84621 D05QPR 12229388 IC50 = 489.78 nM T84621 D06CWR 24754344 IC50 = 67 nM T84621 D06HFV 6539805 IC50 = 27 nM T84621 D06JYY 25130848 IC50 = 2804 nM T84621 D06NFC 45103808 IC50 = 16 nM T84621 D06RSD 45103911 IC50 = 307 nM T84621 D07CTI 10853186 IC50 = 22.3 nM T84621 D07DQJ 45103810 IC50 = 7 nM T84621 D07EJK 10632289 IC50 = 478 nM T84621 D07IQG 10473365 IC50 = 6.7 nM T84621 D07JCO 12354256 IC50 = 6338 nM T84621 D07JMO 10220337 IC50 = 143 nM T84621 D07NAH 21772021 IC50 = 207 nM T84621 D07PYC 6539760 IC50 = 87 nM T84621 D07SOM 11847316 IC50 = 12 nM T84621 D07VGT 46901929 IC50 = 627 nM T84621 D07WLT 25180108 IC50 = 3964 nM T84621 D08AZK 6539767 IC50 = 1937 nM T84621 D08EZA 11847317 IC50 = 187 nM T84621 D08FAB 11845485 IC50 = 5826 nM T84621 D08HHA 19902087 IC50 = 204.17 nM T84621 D08HPU 6540052 IC50 = 503 nM T84621 D08IDC 24827305 IC50 = 238 nM T84621 D08ORG 10198247 IC50 = 281.84 nM T84621 D08PNF 6539770 IC50 = 790 nM T84621 D08WHC 10397593 IC50 = 206 nM T84621 D08YGW 10444038 IC50 = 4.786 nM T84621 D08ZTZ 11529133 IC50 = 2517 nM T84621 D09CPC 13728862 IC50 = 6746 nM T84621 D09HEA 1236449 IC50 = 368 nM T84621 D09HOE 6539789 IC50 = 34 nM T84621 D09QDY 6540033 IC50 = 6.1 nM T84621 D09VPA 6539794 IC50 = 2640 nM T84621 D09VQZ 46901616 IC50 = 4742 nM T84621 D09YXV 6539769 IC50 = 1448 nM T84621 D09ZHX 11847318 IC50 = 27 nM T84621 D0AK9S 22466877 IC50 = 18 nM T84621 D0AW7Q 46867544 IC50 = 463 nM T84621 D0B2UM 25034430 IC50 = 114 nM T84621 D0C6US 6540055 IC50 = 2529 nM T84621 D0C7YL 6481821 IC50 = 390 nM T84621 D0D7YL 11586681 IC50 = 2452 nM T84621 D0D8KN 45103805 IC50 = 181 nM T84621 D0D8YE 6540048 IC50 = 5684 nM T84621 D0D9FR 6539795 IC50 = 484 nM T84621 D0E0ZS 46901613 IC50 = 307 nM T84621 D0E8DX 25180300 IC50 = 580 nM T84621 D0E9WX 6540042 IC50 = 26.2 nM T84621 D0F5AC 46867542 IC50 = 15.1 nM T84621 D0F5YU 6539793 IC50 = 301 nM T84621 D0G6QL 23644748 IC50 = 1317 nM T84621 D0G9WP 18407230 IC50 = 819 nM T84621 D0HL9S 1265319 IC50 = 234.42 nM T84621 D0I1YH 46901446 IC50 = 342 nM T84621 D0I2UH 44187006 IC50 = 5.754 nM T84621 D0I5NW 6540047 IC50 = 1729 nM T84621 D0I9PA 25180306 IC50 = 13378 nM T84621 D0JE1I 9815923 IC50 = 9.5 nM T84621 D0K2DR 12050204 IC50 = 5952 nM T84621 D0K5KG 6540050 IC50 = 1268 nM T84621 D0L2QD 45103910 IC50 = 72.44 nM T84621 D0L4NG 6540054 IC50 = 1615 nM T84621 D0L8KL 11275595 IC50 = 805 nM T84621 D0LJ9D 46901783 IC50 = 415 nM T84621 D0M7FS 6539764 IC50 = 125 nM T84621 D0M9VK 11514098 IC50 = 849 nM T84621 D0MA9G 6540051 IC50 = 2117 nM T84621 D0N1GH 11601068 IC50 = 691 nM T84621 D0N1PQ 11506923 IC50 = 1577 nM T84621 D0N4VI 3021558 IC50 = 639 nM T84621 D0N5GZ 12229395 IC50 = 258 nM T84621 D0N8QD 15594569 IC50 = 691.83 nM T84621 D0N9PY 6539773 IC50 = 2368 nM T84621 D0NV7W 45103912 IC50 = 19.95 nM T84621 D0NX0M 6540049 IC50 = 578 nM T84621 D0O7TC 25180103 IC50 = 525 nM T84621 D0P1UO 45103914 IC50 = 26.92 nM T84621 D0PH1G 13688208 IC50 = 47.86 nM T84621 D0Q0BK 46901611 IC50 = 850 nM T84621 D0Q3CX 25034343 IC50 = 52 nM T84621 D0Q3JZ 6539774 IC50 = 2697 nM T84621 D0Q5ZZ 25129117 IC50 = 640 nM T84621 D0Q6BJ 25034426 IC50 = 151 nM T84621 D0Q8KM 44206482 IC50 = 28 nM T84621 D0R0TE 11557864 IC50 = 5419 nM T84621 D0RJ6S 11558270 IC50 = 2939 nM T84621 D0S4KP 25034427 IC50 = 843 nM T84621 D0S4WQ 12229386 IC50 = 151.36 nM T84621 D0S8FV 44586852 IC50 = 1047 nM T84621 D0T8JU 45103811 IC50 = 10.96 nM T84621 D0U7RR 6539768 IC50 = 320 nM T84621 D0V3YH 6539784 IC50 = 304 nM T84621 D0V6QN 45103915 IC50 = 128.82 nM T84621 D0V8CR 6539763 IC50 = 311 nM T84621 D0VL3R 25180303 IC50 = 1977 nM T84621 D0W8IZ 45103809 IC50 = 25.12 nM T84621 D0WN9P 46901444 IC50 = 287 nM T84621 D0X0IH 77918 IC50 = 135 nM T84621 D0X1QS 6540053 IC50 = 1291 nM T84621 D0Y3AV 25034346 IC50 = 373 nM T84621 D0Y5KX 46901443 IC50 = 522 nM T84621 D0YD9J 6539792 IC50 = 1515 nM T84621 D0YS2F 6539776 IC50 = 955 nM T84621 D0Z3GX 46901784 IC50 = 422 nM T35173 D03MXK 25022340 Ki = 5.1 nM T35173 D07CLV 46940575 IC50 = 12.9 nM T35173 D09MIN 24737642 IC50 = 11 nM T35173 D08XOV 50913339 IC50 = 1.3 nM T35173 D0YN1X 71661892 Ki = 5.4 nM T35173 CO1ZE4 9927170 IC50 = 690 nM T35173 CY3RV2 17756618 Ki = 2 nM T35173 CBM94F 23646361 Ki = 328 nM T35173 C8XJG1 24754961 Ki > 10000 nM T35173 C3EN8I 24857831 IC50 = 1860 nM T35173 C7XTN2 25138055 Ki = 5.9 nM T35173 CJ2VZ4 25138056 Ki = 4.2 nM T35173 C29PBM 25138057 Ki = 370 nM T35173 CLO6Y8 25138058 Ki = 20 nM T35173 CPN8E5 25138069 Ki = 1 nM T35173 CWH17B 25138070 Ki = 132 nM T35173 C0BJQ6 25173661 Ki = 20800 nM T35173 CW4U0R 25180313 Ki = 3 nM T35173 CAL8M3 25209021 Ki = 0.25 nM T35173 CD29TU 25209022 Ki = 2.09 nM T35173 C2KPJ0 44576646 IC50 = 1890 nM T35173 C96OTK 46830178 Ki = 24 nM T35173 CECL56 46830179 Ki = 393 nM T35173 C8RDC3 46888403 Ki = 292 nM T35173 CP40QG 46929436 Ki = 4.2 nM T35173 CQ0A5I 46929438 Ki = 47 nM T35173 C5FK8W 46929440 IC50 = 5.3 nM T35173 C1TIK8 46930628 Ki = 22.5 nM T35173 CVC3T5 46930723 Ki = 24.8 nM T35173 CNQO70 52951104 Ki = 1.7 nM T35173 C30GIF 53237922 Ki = 6 nM T35173 CW7AF2 53238154 Ki = 2 nM T35173 C5JPH2 53238155 Ki = 1.2 nM T35173 CW71DY 53238387 Ki = 2 nM T35173 C16JNG 53238388 Ki = 3 nM T35173 C3IPJ4 53238615 Ki = 2 nM T35173 CH0L8C 53238616 Ki = 2 nM T35173 CF83PC 53238842 Ki = 2.5 nM T35173 C2HB0C 53238843 Ki = 3 nM T35173 C7SR2W 53239063 Ki = 2.5 nM T35173 CM46PV 53239064 Ki = 4 nM T35173 CNFD80 53239285 Ki = 7 nM T35173 CCL6I5 53239286 Ki = 11 nM T35173 C61NHL 56945169 Ki = 3.3 nM T35173 C2WXP5 56945170 Ki = 6.4 nM T35173 C7YW1J 56945269 Ki = 6.9 nM T35173 CR7TD9 56945270 Ki = 14 nM T35173 CAD3P5 56945392 Ki = 4 nM T35173 CDYL09 56945393 Ki = 11 nM T35173 C7X1ZF 56946798 Ki = 1.7 nM T35173 C05JAE 56946799 Ki = 1.3 nM T35173 CE6SU4 57689264 Ki = 2 nM T35173 C62ZCQ 57689338 Ki = 25.3 nM T35173 C3KDR0 58609608 IC50 = 209 nM T35173 CTYP01 66972671 IC50 = 2.6 nM T35173 CZI6S5 66972777 IC50 = 4 nM T35173 CK0FP7 66972990 IC50 = 2.7 nM T35173 CQ9Y8K 66972994 IC50 = 3.2 nM T35173 CTKN28 66973039 IC50 = 2.5 nM T35173 CR9CO4 66973072 IC50 = 3.4 nM T35173 CKQ68O 66973165 IC50 = 4.9 nM T35173 CAD24O 66973224 IC50 = 7.6 nM T35173 C0R9TP 66973397 IC50 = 14 nM T35173 CQ1O6Z 66973400 IC50 = 2.1 nM T35173 C1NV7Q 71528757 EC50 = 36 nM T35173 C5RD4E 71570901 IC50 = 214 nM T35173 C9IT5Y 71570902 IC50 = 235 nM T35173 CY83OB 71571046 EC50 = 20 nM T35173 CAR8J2 71578011 IC50 = 1320 nM T35173 CVPJ20 71581702 IC50 = 47 nM T35173 CP9G3R 71581703 IC50 = 11 nM T35173 C3F4OT 71581838 IC50 = 40 nM T35173 CLIU93 71582189 IC50 = 16 nM T35173 C1VME6 71582339 IC50 = 10 nM T35173 CZ8DF4 71661893 Ki = 12.6 nM T35173 CB0O2T 71662077 Ki = 7.7 nM T35173 COCI81 71662078 Ki = 9.9 nM T35173 CNU16X 71662256 Ki = 2.1 nM T35173 CJRL34 71662257 Ki = 10 nM T35173 C2UM5A 71662420 Ki = 11 nM T35173 CVZK59 71662421 Ki = 7.4 nM T35173 CW4G0O 71662584 Ki = 13.3 nM T35173 C8AY6G 71662585 Ki = 7.9 nM T35173 C2UVF7 76335647 IC50 = 21 nM T35173 CZQO17 86650974 IC50 = 1.7 nM T35173 C9PHL5 89569624 IC50 = 24 nM T35173 CO0IY8 89570499 IC50 = 232 nM T35173 CD57CO 89570570 IC50 = 1490 nM T35173 C2ARB5 89570664 IC50 = 900 nM T35173 CIH2F9 90657109 IC50 = 366 nM T35173 CIH5V8 90664859 IC50 = 1300 nM T35173 C7APL4 118732792 IC50 = 1360 nM T35173 CDZ6M0 118732793 IC50 = 2880 nM T35173 C64NWU 118732794 IC50 = 180 nM T35173 CI69WD 118732795 IC50 = 17 nM T35173 C14FGL 122187534 IC50 = 3 nM T35173 C6NFD0 134419123 IC50 = 330 nM T35173 C87BOG 138377561 IC50 = 5.7 nM T35173 C0B8GK 138377594 IC50 = 140 nM T35173 CA43ML 142585287 IC50 > 1000 nM T35173 CGF6R2 142585309 IC50 > 1000 nM T35173 C0HC8R 142585337 IC50 > 9000 nM T35173 C0RHF1 142585361 IC50 > 10000 nM T35173 C5AI8Z 142585365 IC50 > 10000 nM T35173 CM7IG2 142585375 IC50 > 1500 nM T35173 CG46IU 145954838 IC50 > 1000 nM T35173 CKEJ30 145979040 IC50 = 353.3 nM T35173 C7XM4Q 145979112 IC50 = 53.5 nM T35173 CLRM52 145979809 IC50 = 304 nM T35173 CL4F9B 145981512 IC50 = 1103 nM T35173 C1K6AY 145982930 IC50 > 1000 nM T35173 C3L1ZW 145985393 IC50 = 56.6 nM T35173 CY8JR0 145986444 IC50 = 364.3 nM T35173 C1HWA3 145988725 IC50 = 212.1 nM T35173 CX7AV2 145991404 IC50 = 30.6 nM T35173 C79EXP 145992527 IC50 = 15 nM T35173 CK8JB2 155512591 IC50 = 40 nM T35173 CEH0W4 155523271 IC50 = 353 nM T35173 C23UZA 155554597 IC50 = 12.5 nM T35173 CR3UQ4 155561157 IC50 = 9 nM T35173 D03KZH 25172871 Ki = 6.3 nM T35173 D0BW7P 44589292 Ki = 4.8 nM T35173 D0Q7TL 24754886 Ki = 1.84 nM T35173 D0VK7M 49847690 IC50 = 21 nM T91442 D05RQB 457964 IC50 = 600 nM T91442 CZP5J2 3415 IC50 < 280 nM T91442 CQ87XE 72187 IC50 = 5800 nM T91442 CU3P0Y 484047 IC50 = 70 nM T91442 C61SXL 492406 IC50 = 370 nM T91442 CZ1A8T 503580 IC50 = 770 nM T91442 C8F1DN 6482394 IC50 = 460 nM T36445 CJ73BT 45486346 Ki = 53 nM T36445 C9ETC4 45486354 Ki = 70 nM T36445 CVPG40 45486356 Ki = 3.65 nM T36445 CSQ2K4 45486357 Ki = 1.7 nM T36445 C0ET8W 137630787 Ki = 2 nM T36445 D0Y9PH 45486355 Ki = 0.75 nM T82467 CL80QG 11820 IC50 > 100000 nM T82467 C2IJU0 440987 IC50 > 1000000 nM T82467 CV56WH 1637655 IC50 = 23000 nM T82467 CM1AE9 3370466 IC50 = 7943.28 nM T82467 CGE54P 3573716 IC50 = 10000 nM T82467 CS9M8A 3577407 IC50 = 5011.87 nM T82467 CJ4U6Y 3589423 IC50 = 10000 nM T82467 C2U9DI 3657707 IC50 = 31622.78 nM T82467 CPN2V4 3673391 IC50 = 10000 nM T82467 C28EBX 4790771 IC50 > 100000 nM T82467 CXBG75 5125956 IC50 = 50118.72 nM T82467 CL91JP 9452375 IC50 = 79432.82 nM T82467 C1W7TE 16258532 IC50 = 1258.93 nM T82467 C25EUG 16272810 IC50 = 1258.93 nM T82467 CK2ES3 16313990 IC50 > 100000 nM T82467 CZ59FR 16316459 IC50 > 100000 nM T82467 CEN83U 16323492 IC50 = 12589.25 nM T82467 CM1R8O 16344932 IC50 > 100000 nM T82467 CO8M7K 17405877 IC50 = 31622.78 nM T82467 C9IP3Q 17446910 IC50 > 100000 nM T82467 CLP9S1 24687782 IC50 = 12589.25 nM T82467 CEL5F7 26851836 IC50 > 1000000 nM T82467 CG3PR6 52912222 IC50 > 31622.78 nM T82467 CF8B4E 60498769 IC50 > 100000 nM T82467 CHOS65 91820723 IC50 = 100000 nM T82467 C0TNJ7 91820724 IC50 = 12589.25 nM T82467 CAZ9M0 91826677 IC50 = 2511.89 nM T82467 CEN52P 91826678 IC50 = 1000 nM T82467 C3BR8O 118021718 IC50 > 80000 nM T82467 CC14FI 118933132 IC50 > 100000 nM T82467 CWC98G 121499171 IC50 = 2700 nM T82467 CO9J5W 122179607 IC50 = 15848.93 nM T82467 C3WOE8 122179608 IC50 = 50118.72 nM T82467 CW03JY 122179609 IC50 = 3981.07 nM T82467 CHNS18 122179610 IC50 = 1258.93 nM T82467 C2Q0OY 122179611 IC50 = 5011.87 nM T82467 C9GPL4 122179612 IC50 = 1995.26 nM T82467 CZX41C 122179613 IC50 = 1258.93 nM T82467 CJDK15 122179614 IC50 = 1584.89 nM T82467 CSF76G 122179615 IC50 = 794.33 nM T82467 CY7U0Z 122179616 IC50 = 1258.93 nM T82467 C1MV9L 122179617 IC50 = 1584.89 nM T82467 CJ81BV 122179618 IC50 = 3981.07 nM T82467 CZ69QO 122180530 IC50 > 100000 nM T82467 C7D5VP 122180531 IC50 > 100000 nM T82467 CRY84E 122180532 IC50 > 100000 nM T82467 C0J1AY 122180533 IC50 > 100000 nM T82467 CPIV02 122180534 IC50 > 100000 nM T82467 CC9XH7 122180535 IC50 > 100000 nM T82467 C0IWE1 122180536 IC50 = 501187.23 nM T82467 CEF19P 122180537 IC50 = 25118.86 nM T82467 C20LOD 122180538 IC50 = 63095.73 nM T82467 C73OMU 122180539 IC50 = 19952.62 nM T82467 CZSB51 122180540 IC50 = 31622.78 nM T82467 CJ4LO2 122180541 IC50 = 79432.82 nM T82467 C4TB0F 122180542 IC50 = 12589.25 nM T82467 CTXL15 122180543 IC50 = 15848.93 nM T82467 CUDY80 122180544 IC50 > 100000 nM T82467 C0SC2Y 122180545 IC50 > 100000 nM T82467 CR6T4G 122180546 IC50 = 50118.72 nM T82467 CHJG86 122180547 IC50 > 100000 nM T82467 CYZV97 122180548 IC50 > 100000 nM T82467 C0AIU8 122180549 IC50 = 50118.72 nM T82467 CPUS31 122180550 IC50 = 31622.78 nM T82467 CD62RB 122180551 IC50 = 39810.72 nM T82467 C8UCV9 122180552 IC50 = 7943.28 nM T82467 C72NLB 122180553 IC50 = 5011.87 nM T82467 CR0K5P 122180554 IC50 = 15848.93 nM T82467 CZ6L2N 122180555 IC50 = 6309.57 nM T82467 CKH49I 122180556 IC50 = 25118.86 nM T82467 CS4PD6 122180557 IC50 = 10000 nM T82467 CWC9I4 122180558 IC50 = 3162.28 nM T82467 CE7SL5 122180559 IC50 = 2511.89 nM T82467 CR6YD4 122180560 IC50 = 1258.93 nM T82467 C8HCK6 122180561 IC50 = 1258.93 nM T82467 CX9C6Y 122180562 IC50 = 3162.28 nM T82467 CPZ67Y 122180563 IC50 = 19952.62 nM T82467 CN1LE0 122180564 IC50 = 39810.72 nM T82467 CGLF82 122181547 IC50 = 199.53 nM T82467 CZGK74 122181548 IC50 = 125.89 nM T82467 C9P3GX 122181549 IC50 = 316.23 nM T82467 C3QJ5L 122181550 IC50 = 31.62 nM T82467 C3NC4V 122181552 IC50 = 125.89 nM T82467 C41ZXJ 122181555 IC50 = 199.53 nM T82467 C6I3VJ 122181557 IC50 = 39.81 nM T82467 C7CJR2 122181559 IC50 = 5011.87 nM T82467 CP5Z1C 122181560 IC50 = 1584.89 nM T82467 C61RTG 122181561 IC50 = 63095.73 nM T82467 CT62FG 122181571 IC50 = 79.43 nM T82467 C8F9VG 129196931 IC50 = 166 nM T82467 CO3A0E 134817551 IC50 = 251.19 nM T82467 CP4X5W 134817552 IC50 = 100 nM T82467 CA40QW 135535536 IC50 = 10000 nM T82467 CQT3A9 137636309 IC50 > 100000 nM T82467 CQ6XB7 139030526 IC50 = 316.23 nM T82467 CJ3FL8 145982835 IC50 = 251.19 nM T82467 CA2W8M 145984295 IC50 = 199.53 nM T82467 CE05ZV 145984432 IC50 = 25118.86 nM T82467 CV4GH7 145984467 IC50 = 251.19 nM T82467 CT6V0I 145985751 IC50 = 39.81 nM T82467 C0GHY5 145986052 IC50 = 125.89 nM T82467 CK98QJ 146035912 IC50 = 100 nM T82467 C2D1SB 155512075 IC50 = 1995.26 nM T82467 CD3LA9 155512613 IC50 = 1995.26 nM T82467 CE13CA 155515130 IC50 = 3981.07 nM T82467 CPM43N 155516232 IC50 > 100000 nM T82467 C23BXS 155517049 IC50 = 3162.28 nM T82467 C6Q3JK 155517968 IC50 = 1000 nM T82467 CFP24B 155518498 IC50 = 1995.26 nM T82467 CB49NL 155521254 IC50 = 63.1 nM T82467 CC30UG 155521851 IC50 = 1258.93 nM T82467 CL1P4M 155523233 IC50 = 1258.93 nM T82467 C1W8JL 155523577 IC50 = 50118.72 nM T82467 C2K9NI 155523694 IC50 = 2511.89 nM T82467 C0VS8H 155523850 IC50 = 1258.93 nM T82467 C3NYK0 155523937 IC50 = 1000 nM T82467 CW8O7G 155525483 IC50 = 794.33 nM T82467 CKR6V3 155528325 IC50 = 1584.89 nM T82467 COX8K5 155529510 IC50 = 1995.26 nM T82467 CVMC06 155529991 IC50 = 630.96 nM T82467 CL93CM 155530154 IC50 = 1000 nM T82467 CEI09V 155530332 IC50 = 251.19 nM T82467 CY7ST9 155530616 IC50 = 1000 nM T82467 CJ93LE 155531635 IC50 = 1995.26 nM T82467 C82UPM 155532741 IC50 = 3162.28 nM T82467 CAEQ29 155534550 IC50 = 1000 nM T82467 CY08SU 155535485 IC50 = 2511.89 nM T82467 CAL2G4 155538392 IC50 > 1000000 nM T82467 C9ISB5 155538742 IC50 = 2511.89 nM T82467 C1MQP2 155539283 IC50 = 1995.26 nM T82467 C45FSO 155539489 IC50 = 15848.93 nM T82467 CXTO91 155541586 IC50 = 2511.89 nM T82467 CSVH67 155541704 IC50 > 1000000 nM T82467 CNSP97 155542781 IC50 = 501.19 nM T82467 C6FHM8 155543582 IC50 = 630.96 nM T82467 CEA1C5 155545659 IC50 = 30 nM T82467 CM51BF 155546089 IC50 = 12589.25 nM T82467 CFTR89 155546746 IC50 = 1584.89 nM T82467 CRBT87 155547095 IC50 > 1000000 nM T82467 CQNO46 155548910 IC50 = 2511.89 nM T82467 C4VKR0 155551851 IC50 = 1258.93 nM T82467 C2FWB9 155551946 IC50 = 25.12 nM T82467 CT35SU 155553650 IC50 = 6309.57 nM T82467 C0SYN6 155554629 IC50 = 3162.28 nM T82467 CDO08V 155555578 IC50 = 3981.07 nM T82467 C12QHG 155555950 IC50 = 1584.89 nM T82467 C7S8GF 155556284 IC50 > 100000 nM T82467 C6N1CG 155557122 IC50 = 1000 nM T82467 CYM3K9 155557522 IC50 = 2511.89 nM T82467 CSGH17 155559412 IC50 = 1995.26 nM T82467 C1YWF9 155559659 IC50 > 1000000 nM T82467 C3IDR8 155559983 IC50 > 1000000 nM T82467 C5X6EL 155560182 IC50 = 251.19 nM T82467 CS1C5W 155560567 IC50 = 3162.28 nM T82467 C3UC7H 155560671 IC50 = 10000 nM T82467 C7EDG4 155564694 IC50 = 3162.28 nM T82467 C6MX5G 155564795 IC50 > 1000000 nM T82467 CXRJ70 155566441 IC50 = 1258.93 nM T82467 C2PIK0 155567275 IC50 = 1000 nM T82467 CM5FL1 155567534 IC50 = 2511.89 nM T82467 C7C9DH 155568184 IC50 = 6309.57 nM T82467 CZ2VN0 155569163 IC50 = 1258.93 nM T82467 D00XRH 91820725 IC50 = 1258.93 nM T82467 D0F5TZ 91827383 IC50 = 1258.93 nM T82467 D0O6XT 91827373 IC50 > 100000 nM T13260 D00AXJ 4189 IC50 = 600 nM T13260 D00ZFP 5870 Ki = 2500 nM T13260 D02STN 132971 IC50 > 5000 nM T13260 D04DJN 10635 Ki = 220 nM T13260 D06XMU 6013 Ki = 600 nM T13260 D07ABV 468595 IC50 = 8400 nM T13260 D09GOS 2812 IC50 = 1.8 nM T13260 D09LNI 3365 IC50 = 22000 nM T13260 D0B4IF 456201 IC50 = 951.48 nM T13260 D0C1WH 3902 Ki = 0.02 nM T13260 D0C7JF 13769 Ki = 35000 nM T13260 D0D2VS 60198 Ki = 10.2 nM T13260 D0G2MW 446284 IC50 = 53200 nM T13260 D0K8KX 5280343 IC50 = 12 nM T13260 D0M6DO 2145 IC50 = 5.2 nM T13260 D0Q5XX 445580 IC50 = 33200 nM T13260 D0W0BF 2187 Ki = 0.13 nM T13260 D0ZX1P 59693 Ki = 0.05 nM T13260 D03AJU 44139752 IC50 = 856 nM T13260 D05NJI 5287541 IC50 = 300 nM T13260 D08UGX 60652 IC50 = 44.67 nM T13260 D09NST 449459 IC50 = 530000 nM T13260 D0B4VE 10251 IC50 = 8000 nM T13260 D0G5CS 68071 IC50 = 900 nM T13260 D0L4FS 5280961 Ki = 100000 nM T13260 D0U3EP 445154 IC50 > 40 ug.mL-1 T13260 D0W4EB 10090750 IC50 = 6000 nM T13260 D0DK4I 4534 IC50 = 11 nM T13260 D03YPJ 5163 IC50 > 100000 nM T13260 D06JUR 56487 Ki = 1100 nM T13260 D09BKE 4553 IC50 = 680 nM T13260 D0C0JT 4495 IC50 = 27000 nM T13260 D0D3PF 6918191 IC50 = 1.38 nM T13260 D0SX7F 60876 Ki = 7.6 nM T13260 D0Y2OG 177865 IC50 = 0.5 nM T13260 C9LCD8 3823 IC50 = 60 nM T13260 C9NZY3 12452 Ki = 17 nM T13260 C2L1YD 22458 IC50 = 4110 nM T13260 CPY1G9 59694 Ki = 1.5 nM T13260 C87SRA 60796 IC50 = 1.4 nM T13260 CQ0IC4 63062 IC50 = 530000 nM T13260 CLJB07 65544 IC50 = 840 nM T13260 CHI68V 66425 Ki = 100 nM T13260 CG5ZC1 66842 Ki = 100 nM T13260 CMV4R6 67343 Ki = 100 nM T13260 C5JLH9 69088 IC50 > 125700 nM T13260 CRGU58 86488 IC50 = 19000 nM T13260 CR0XY7 88598 IC50 > 10000 nM T13260 CKN0O5 92267 IC50 > 16200 nM T13260 C2Q3LF 92775 IC50 = 9600 nM T13260 CEOP93 100332 IC50 > 40 ug.mL-1 T13260 C1D3WF 101928 IC50 = 1733 nM T13260 C56OAF 104880 Ki = 2.5 nM T13260 C1U3VY 124075 IC50 = 3920 nM T13260 CX30LQ 124600 IC50 = 4000 nM T13260 C64SKJ 125502 Ki = 60.9 nM T13260 CC1ES3 125503 Ki = 172 nM T13260 CPU8L1 125637 Ki = 18 nM T13260 CHWM72 125921 IC50 = 230 nM T13260 CV7MN1 126221 Ki = 17.6 nM T13260 CW45IU 126253 IC50 = 4600 nM T13260 C5E0PO 126735 IC50 = 61.66 nM T13260 CZW26T 128011 Ki = 5 nM T13260 C7CRO3 128300 Ki = 90 nM T13260 CV2KS6 129500 Ki = 5.8 nM T13260 C4UV3D 130636 Ki = 9.9 nM T13260 C7MK6N 131078 IC50 = 310 nM T13260 C9KN0L 131099 Ki = 170 nM T13260 C0JR2M 131426 Ki = 2220 nM T13260 CL0T6W 131798 IC50 = 5.754 nM T13260 C7N1EF 132907 Ki = 5 nM T13260 CL9ZS8 138203 IC50 = 11880 nM T13260 CF83MK 146141 Ki = 34 nM T13260 CPVI09 146142 Ki = 1 nM T13260 C1RTX5 146485 IC50 = 2700 nM T13260 C9H4TV 147045 Ki = 120 nM T13260 CWJ40O 151432 Ki = 120 nM T13260 C5AS9H 155976 IC50 > 40 ug.mL-1 T13260 C3Y7WX 158280 IC50 > 40 ug.mL-1 T13260 C9DTE4 160767 IC50 = 29000 nM T13260 CT5E1S 165184 IC50 > 50000 nM T13260 CYWS98 185848 IC50 > 40 ug.mL-1 T13260 CL5U9T 190972 Ki = 9.8 nM T13260 C0EOM6 193441 Ki = 1000 nM T13260 C1S9AI 196342 Ki = 15 nM T13260 CE4U0D 198531 IC50 > 50000 nM T13260 C36VAO 199390 IC50 > 50000 nM T13260 CU9BQ6 219377 IC50 = 46700 nM T13260 CAD54R 239595 IC50 = 250 nM T13260 C5WUK4 256446 IC50 = 4810 nM T13260 CQ6A8P 266151 IC50 = 800 nM T13260 COA9C7 280309 IC50 = 9000 nM T13260 C1C5TO 281901 Ki = 180 nM T13260 CS86KD 283391 IC50 = 20 nM T13260 CD8E9U 313177 IC50 = 37600 nM T13260 CE9R4U 316687 IC50 = 130 nM T13260 CNP1J9 334704 IC50 > 40 ug.mL-1 T13260 CU7L1E 343584 IC50 = 126000 nM T13260 CHL4T1 387487 IC50 = 95300 nM T13260 CA9B4J 390805 IC50 = 176000 nM T13260 C3AJN7 396930 IC50 = 100 nM T13260 CD2UN0 432882 IC50 = 11000 nM T13260 C7HME8 439246 IC50 = 2.9 nM T13260 CK2EB0 461948 IC50 = 6 nM T13260 CDM69B 484455 IC50 = 2160 nM T13260 CQ59RG 484458 IC50 = 580 nM T13260 CZO45T 484460 IC50 = 9230 nM T13260 CB2DY7 484461 IC50 = 1520 nM T13260 CS2RK5 484470 IC50 = 4000 nM T13260 CRED51 484475 IC50 = 3650 nM T13260 CLR9O8 492641 IC50 = 4590 nM T13260 CL21UY 508444 IC50 = 350 nM T13260 CQSN41 508446 IC50 = 300 nM T13260 CUWG73 508447 IC50 = 460 nM T13260 CQ4KL6 508448 IC50 = 2960 nM T13260 CS7DT2 508449 IC50 = 1510 nM T13260 C3GNC0 508450 IC50 = 1180 nM T13260 C7TVD8 508451 IC50 = 190 nM T13260 CW8JE3 508452 IC50 = 2200 nM T13260 CLAW60 508453 IC50 = 1530 nM T13260 C8L5OZ 510041 IC50 = 1240 nM T13260 CNB76G 510042 IC50 = 260 nM T13260 CH95MB 510043 IC50 = 1090 nM T13260 C9NGK0 510044 IC50 = 1370 nM T13260 CEZW17 510045 IC50 = 1040 nM T13260 CTLY25 510046 IC50 = 510 nM T13260 C7X6RO 510048 IC50 = 110 nM T13260 CX65UW 510049 IC50 = 1320 nM T13260 CXC2M7 510050 IC50 = 1680 nM T13260 CM23DG 510051 IC50 = 1000 nM T13260 C7TYH9 585624 IC50 = 3200 nM T13260 C5LJK2 591809 IC50 = 260 nM T13260 CI5FK2 591810 IC50 = 41000 nM T13260 C2QEF8 596715 IC50 > 50000 nM T13260 C3P1FA 606677 IC50 = 3050 nM T13260 CG72HV 622979 Ki = 58 nM T13260 CQ90BJ 623313 Ki = 140 nM T13260 CU4V9W 623696 Ki = 3000 nM T13260 CZ0AH3 638278 IC50 = 3800 nM T13260 CHV1X7 638701 IC50 = 3980 nM T13260 CM9IU5 641375 IC50 = 31100 nM T13260 CO28QU 641376 IC50 = 31100 nM T13260 CZ14PX 641378 IC50 > 40 ug.mL-1 T13260 CS2IQ3 715186 IC50 = 10600 nM T13260 CE4JQ8 782123 IC50 > 105800 nM T13260 C8EDM5 838923 IC50 = 39710 nM T13260 CFZ7C3 882273 IC50 = 5030 nM T13260 CP25US 1009065 IC50 = 50 nM T13260 CJQK73 1027647 IC50 = 529663443.9 nM T13260 CE9SH3 1291064 IC50 = 11600 nM T13260 C48SKB 1292107 IC50 = 2190 nM T13260 CEOM25 1294577 IC50 = 780 nM T13260 C6B9RE 1481465 IC50 = 22810 nM T13260 C1SH3T 1548910 IC50 > 50000 nM T13260 C7VE1Z 1548995 IC50 = 370000 nM T13260 CB93KS 1550302 IC50 = 9200 nM T13260 C3T8GZ 1831259 IC50 > 10000 nM T13260 CF18YS 2313447 IC50 = 1100 nM T13260 COYU39 2475352 IC50 = 200 nM T13260 CB4N3X 2725996 Ki = 234.3 nM T13260 C8SYF6 2725997 IC50 = 4 nM T13260 C68PUH 2725998 Ki = 63.38 nM T13260 CO84NG 2827372 IC50 = 16.5 nM T13260 CPXD41 2843385 IC50 = 1000 nM T13260 C3M7VX 2939932 IC50 = 10600 nM T13260 C8XJ1B 2992689 IC50 = 172 nM T13260 C3H1DE 2998104 IC50 = 1500 nM T13260 CUVM41 3035832 IC50 = 190 nM T13260 CZ1LD9 3298129 IC50 > 25000 nM T13260 C2SE4A 3346379 IC50 = 4300 nM T13260 C2OS4U 3361302 IC50 = 1100 nM T13260 CCD73S 3399276 IC50 = 3880 nM T13260 CBKQ75 3418244 IC50 = 370 nM T13260 C7O2MH 3943788 IC50 = 80 nM T13260 C40QVD 3964390 IC50 > 40 ug.mL-1 T13260 C7LX0V 4083407 IC50 = 59979107.63 nM T13260 C0WA7C 4103051 Ki = 830 nM T13260 CJ1U7P 4369413 IC50 = 100 nM T13260 CK17YZ 4369414 IC50 = 0.82 nM T13260 C1WIR4 4499193 IC50 > 31622.78 nM T13260 CXNH97 4993111 IC50 = 3670 nM T13260 C5OAR6 5121919 IC50 > 50000 nM T13260 CG0C4J 5281255 IC50 > 40 ug.mL-1 T13260 CM9Z0B 5312198 IC50 = 761 nM T13260 CF67ON 5314722 IC50 > 25000 nM T13260 CEW6B3 5315503 IC50 > 40 ug.mL-1 T13260 C3KDP7 5325467 IC50 = 16310 nM T13260 CW1UM5 5357488 IC50 > 351700 nM T13260 CBF75X 5376779 IC50 > 250000 nM T13260 CUV49J 5472143 IC50 = 5200 nM T13260 CR6N4L 5481966 IC50 > 40 ug.mL-1 T13260 C7VSM2 5702471 IC50 = 9332.54 nM T13260 CST49O 5702960 IC50 > 250000 nM T13260 C84XUK 6035693 IC50 = 5495.41 nM T13260 C3F7JB 6159604 IC50 = 12022.64 nM T13260 C1HZJ2 6438825 IC50 > 40 ug.mL-1 T13260 C2B1RH 6450879 IC50 > 40 ug.mL-1 T13260 CR8IB1 6457965 IC50 = 21700 nM T13260 C26KXD 6458748 IC50 = 2500 nM T13260 C39IEC 6461420 IC50 = 119 nM T13260 CP3O0B 6463551 IC50 = 61.6 nM T13260 CE93VI 6473542 IC50 = 100 nM T13260 C73LCV 6475119 IC50 = 42.7 ug.mL-1 T13260 C21BZK 6493479 IC50 = 63.7 nM T13260 CCO4Q3 6493484 IC50 = 440 nM T13260 CI13SQ 6523638 IC50 = 25000 nM T13260 C1JAT6 6539761 IC50 = 6580 nM T13260 CTE57C 6539762 IC50 = 3790 nM T13260 CF17BE 6539771 IC50 = 1130 nM T13260 CJ7RS8 6539772 IC50 = 4000 nM T13260 CP02JW 6539778 IC50 = 979489.99 nM T13260 CW1U8J 6539779 IC50 > 36000 nM T13260 CQD13Z 6539787 IC50 = 650 nM T13260 CQB1U5 6539798 IC50 = 800 nM T13260 C79FTC 6539799 IC50 = 1010 nM T13260 C5Z9KY 6539802 IC50 = 90 nM T13260 C7CAB8 6539809 IC50 > 36000 nM T13260 COU5D2 6539810 IC50 > 36000 nM T13260 CQ0HD5 6539812 IC50 = 720 nM T13260 CQ9XM0 6539813 IC50 = 1940 nM T13260 CF1R9J 6539815 IC50 > 36000 nM T13260 CMA37K 6539816 IC50 > 36000 nM T13260 CP4VI2 6540030 IC50 = 226 nM T13260 CR6LS8 6540031 IC50 = 190 nM T13260 CU3C1Y 6540034 IC50 = 125 nM T13260 CXEW82 6540035 IC50 = 119 nM T13260 CBKX32 6540037 IC50 = 120 nM T13260 C8MRI7 6540038 IC50 = 218 nM T13260 C8JXY1 6540039 IC50 = 20 nM T13260 CZK3T4 6540040 IC50 = 330 nM T13260 CDS26H 6540041 IC50 = 39 nM T13260 C2FRW5 6540044 IC50 = 970 nM T13260 C2JBQ1 6540045 IC50 = 810 nM T13260 CV0FA1 7330517 IC50 = 40950 nM T13260 CG9RF6 7515053 IC50 > 250000 nM T13260 C1DZ2H 7537616 IC50 = 150 nM T13260 C8VJ4X 8963350 IC50 > 50000 nM T13260 C0J1AS 9794431 IC50 = 10000 nM T13260 CS23XK 9797346 Ki = 10 nM T13260 C9QVL1 9816909 IC50 = 8900 nM T13260 CJ37SX 9818699 IC50 = 1.38 nM T13260 C2YB9F 9819524 IC50 = 12 nM T13260 CF7Z3J 9837392 IC50 = 2.9 nM T13260 C56CLB 9838063 IC50 = 680 nM T13260 CKJ1I6 9838340 IC50 = 580 nM T13260 CF3Z5V 9839853 Ki = 1.4 nM T13260 C35UMF 9890209 IC50 > 500000 nM T13260 CZ15MX 9908653 Ki = 36 nM T13260 CWL3O1 9926844 IC50 = 40000 nM T13260 C9Y3CA 9928113 IC50 = 12 nM T13260 CF24CV 9947889 Ki = 100 nM T13260 C0PHJ6 9948207 Ki = 70 nM T13260 C9BIH0 9948368 IC50 = 95.5 nM T13260 CZFV57 9949484 Ki = 1 nM T13260 CXH81D 9951467 IC50 = 0.12 nM T13260 CO1Z0A 9971194 IC50 = 5600 nM T13260 CBLP75 9972072 IC50 = 42.66 nM T13260 CDT6N2 9972577 IC50 = 8.8 nM T13260 C46LXP 9973019 Ki = 3.4 nM T13260 CB9DF4 9973046 IC50 = 20 nM T13260 C9JPT7 9974683 Ki = 1.4 nM T13260 CW1KO5 9976841 Ki = 36 nM T13260 C6W9NM 9978572 Ki = 16.5 nM T13260 C6Z0WQ 9991753 IC50 = 5000 nM T13260 CR16JI 9991838 IC50 = 530 nM T13260 CZV57I 9992344 IC50 = 6300 nM T13260 CQH4B7 9992433 IC50 = 14000 nM T13260 C2B4RF 9992450 IC50 = 4300 nM T13260 CVU3L0 9993026 IC50 = 3019.95 nM T13260 C85AUN 9998048 IC50 = 38.02 nM T13260 C0J8VR 10000064 IC50 = 78.5 nM T13260 C49HDL 10013868 IC50 = 170 nM T13260 C1FX2N 10014477 IC50 = 9300 nM T13260 C1KAV4 10015136 IC50 = 230 nM T13260 CPG39R 10018603 Ki = 3.4 nM T13260 C58EOH 10019839 IC50 = 130 nM T13260 CX7H2S 10020109 IC50 = 44 nM T13260 C0RP1F 10020714 IC50 = 44 nM T13260 CU12IF 10022210 IC50 = 130 nM T13260 CI7V2F 10023315 Ki = 36 nM T13260 C5PUD9 10026826 IC50 = 210 nM T13260 C5NAU2 10036028 IC50 = 600 nM T13260 C5Y0MK 10036693 IC50 = 380 nM T13260 CU7CI9 10042609 IC50 = 55 nM T13260 CV1K0G 10046399 IC50 = 51.8 nM T13260 C8MC0P 10051115 IC50 = 1650 nM T13260 C6W9NL 10060155 IC50 = 4200 nM T13260 C30LGM 10060824 IC50 = 3400 nM T13260 C64YSN 10064550 IC50 = 62 nM T13260 C9UMW8 10064832 IC50 = 600 nM T13260 C6Y1OT 10067777 Ki = 2.8 nM T13260 CI3S7F 10069029 IC50 = 220 nM T13260 CR13PX 10069113 Ki = 36 nM T13260 CX3FH6 10069477 Ki = 2.8 nM T13260 CR1V5S 10082665 IC50 = 93000 nM T13260 C64PHS 10083522 IC50 = 30 nM T13260 CR13LC 10084738 IC50 = 8700 nM T13260 CB65ED 10086187 Ki = 1.4 nM T13260 CL9X0W 10087126 Ki = 5000 nM T13260 C9YRP5 10087312 IC50 = 57 nM T13260 CPH49E 10087422 IC50 = 61.5 nM T13260 CD0MQ9 10088785 Ki = 1.4 nM T13260 CZB62D 10089657 Ki = 2.8 nM T13260 CNI2R6 10091150 IC50 = 102 nM T13260 C4JM1P 10104524 IC50 = 2400 nM T13260 C92KBY 10105573 IC50 > 19000 nM T13260 C7W5GI 10171354 IC50 = 14000 nM T13260 CD6JG2 10228895 IC50 = 500 nM T13260 CG2U1S 10242773 IC50 = 1000 nM T13260 CC08OX 10243987 IC50 = 590 nM T13260 CG24IZ 10247264 IC50 > 20000 nM T13260 CTK8F5 10248614 Ki = 9.3 nM T13260 C3YC9I 10263082 IC50 = 1900 nM T13260 C4CDG7 10264163 IC50 = 23000 nM T13260 CO2LT5 10286610 IC50 = 860 nM T13260 CD39LQ 10291777 IC50 = 100 nM T13260 CL6WE9 10295791 IC50 = 24000 nM T13260 C5LRW4 10298511 IC50 = 25100 nM T13260 CE2Z5S 10313881 IC50 = 41 nM T13260 C3PYH4 10317448 IC50 = 280 nM T13260 C6AOP4 10317522 IC50 = 530 nM T13260 CMO02D 10317756 Ki = 67000 nM T13260 C65BFK 10317931 IC50 = 400 nM T13260 C64YEQ 10318379 Ki = 9.8 nM T13260 CTUL01 10331100 IC50 = 185 nM T13260 CM81OX 10332392 IC50 = 3715.35 nM T13260 CZ4W0C 10332529 IC50 = 41 nM T13260 CQGS52 10334324 Ki = 1000 nM T13260 CQX4C8 10335739 Ki = 3.4 nM T13260 CT69PQ 10336071 IC50 = 100 nM T13260 C9RX2D 10338362 Ki = 9.3 nM T13260 CUDL75 10340374 Ki = 13.1 nM T13260 C0EO5N 10340839 Ki = 9.3 nM T13260 C07JGF 10355617 IC50 = 3300 nM T13260 CH5DS4 10358509 Ki = 5000 nM T13260 CWY9D0 10360147 Ki = 40 nM T13260 CELR79 10360875 IC50 = 63 nM T13260 CO69BI 10361506 IC50 = 49 nM T13260 CN7JK2 10368162 IC50 = 1650 nM T13260 CYNM04 10376335 IC50 = 260 nM T13260 CWY1X4 10379617 IC50 = 190 nM T13260 C5IZ0X 10380012 IC50 = 35000 nM T13260 CTX86G 10381606 IC50 = 233 nM T13260 COK7N8 10382166 IC50 = 1230 nM T13260 C06BMI 10384926 Ki = 13.1 nM T13260 C8CW6Y 10385742 Ki = 9.8 nM T13260 CP8G9A 10398594 IC50 = 13000 nM T13260 CXY9P7 10398686 IC50 = 1200 nM T13260 C1HZC5 10399349 IC50 = 240 nM T13260 CIJ01W 10400011 IC50 = 170 nM T13260 C3UN8Z 10400778 IC50 = 7900 nM T13260 CJ31WC 10403482 Ki = 42 nM T13260 C9LW2Z 10403903 IC50 = 49 nM T13260 CC5YT4 10404407 IC50 = 3000 nM T13260 CG7P5I 10404636 IC50 = 130 nM T13260 C9Q7CT 10407320 Ki = 36 nM T13260 C8KUR2 10421663 IC50 = 22000 nM T13260 C59NEQ 10426743 IC50 = 4300 nM T13260 CRV19P 10444266 IC50 = 1300 nM T13260 CR0O6C 10447478 IC50 = 20000 nM T13260 CTYP51 10448246 Ki = 5.1 nM T13260 CPAE70 10449017 IC50 = 1460 nM T13260 CUM3X2 10449331 IC50 = 2400 nM T13260 CQWX01 10450499 IC50 > 20000 nM T13260 C4L6ED 10450517 IC50 = 600 nM T13260 CM1IU9 10466775 IC50 = 6400 nM T13260 CT0H4G 10466776 IC50 = 750 nM T13260 C7TL6U 10467336 IC50 = 4786.3 nM T13260 C3YI0N 10467502 IC50 = 17000 nM T13260 C5DP9Z 10471817 IC50 = 10 nM T13260 CSM4H0 10472175 IC50 = 60 nM T13260 CIG25U 10474687 Ki = 10 nM T13260 C9W6YH 10488782 IC50 = 160 nM T13260 CYR2O4 10489655 IC50 = 680 nM T13260 CH7IA3 10489983 IC50 = 38000 nM T13260 CTW6A7 10494334 Ki = 17 nM T13260 CP8F4R 10495337 Ki = 4.7 nM T13260 CG0A6X 10513321 IC50 = 18000 nM T13260 CH2R0N 10513661 IC50 = 3900 nM T13260 C5RHY3 10538018 IC50 = 200 nM T13260 C7I6JP 10562688 IC50 = 239.88 nM T13260 CH8FS5 10565166 Ki = 3.1 nM T13260 C4L8OX 10566080 IC50 = 51000 nM T13260 C9PMK8 10566304 Ki = 12 nM T13260 C43DIK 10571994 Ki = 17 nM T13260 CN2RF5 10585362 IC50 > 250000 nM T13260 C7S5RV 10586086 IC50 = 220 nM T13260 CTI0R2 10587179 IC50 > 250000 nM T13260 CU5GI9 10594307 Ki = 5 nM T13260 C3RM0Y 10595083 Ki = 2.5 nM T13260 C3DH9W 10608774 IC50 = 920 nM T13260 CZ2H3N 10610950 IC50 > 250000 nM T13260 C02GMY 10617003 Ki = 2.5 nM T13260 CNR3V1 10618506 IC50 > 10000 nM T13260 C1F9IE 10636984 Ki = 5.3 nM T13260 C5TVC0 10637984 Ki = 12 nM T13260 CC39RI 10644237 Ki = 7 nM T13260 C04DNA 10656613 IC50 > 250000 nM T13260 C5ION6 10660701 IC50 = 3100 nM T13260 C9QN4J 10660816 IC50 = 36000 nM T13260 CJYQ87 10661641 Ki = 2.5 nM T13260 C8MOG9 10662151 Ki = 12 nM T13260 C8D0PV 10662758 Ki = 2.5 nM T13260 CUA2P0 10663766 Ki = 2.5 nM T13260 C8OUR1 10663913 Ki = 17 nM T13260 CPKA25 10665849 Ki = 17 nM T13260 CAYD96 10667894 Ki = 8.5 nM T13260 CP98RW 10680142 IC50 = 6000 nM T13260 CE12OS 10682353 IC50 = 24000 nM T13260 C0N2BV 10684551 IC50 = 9100 nM T13260 C01ZPW 10684552 IC50 = 10800 nM T13260 C1CGU5 10686589 Ki = 17 nM T13260 COB2W4 10690043 IC50 = 50 nM T13260 C0SIE5 10691220 Ki = 2.5 nM T13260 CMN02T 10708503 Ki = 1100 nM T13260 C1OME3 10710388 IC50 = 5200 nM T13260 CA13SW 10711620 IC50 = 549.54 nM T13260 CUQN16 10714213 IC50 > 10000 nM T13260 CO3JR0 10727176 IC50 = 51000 nM T13260 CBG72H 10729611 IC50 > 250000 nM T13260 CFE87L 10729612 IC50 = 27000 nM T13260 CYW4V9 10731755 IC50 > 10000 nM T13260 CKD29U 10738189 Ki = 9 nM T13260 CHL74J 10752290 IC50 = 103000 nM T13260 CU5W7P 10752634 IC50 = 350 nM T13260 CM3GX1 10753431 IC50 > 250000 nM T13260 C7U3ZR 10755577 IC50 = 4600 nM T13260 C4EXR1 10761806 IC50 = 1100 nM T13260 CZSA79 10774377 IC50 = 111000 nM T13260 CCD9R4 10774996 IC50 = 2400 nM T13260 C9GC0A 10775929 IC50 = 2600 nM T13260 CG27MD 10776192 IC50 > 250000 nM T13260 CNGQ30 10800145 IC50 = 1100 nM T13260 CJ5LW6 10806186 IC50 = 18100 nM T13260 CR25UM 10806331 Ki = 1100 nM T13260 C7P8IX 10810323 Ki = 10 nM T13260 CO53EU 10811011 Ki = 7 nM T13260 C0EAP2 10823139 IC50 = 700 nM T13260 C94PCN 10826001 IC50 = 8000 nM T13260 CN7I8H 10827014 IC50 = 16000 nM T13260 CZW6V4 10828130 IC50 = 2290.87 nM T13260 CM8WH3 10846478 IC50 = 3340 nM T13260 CU3I7B 10847200 IC50 = 440 nM T13260 CLZ5Q7 10853458 Ki = 37 nM T13260 C6RWM5 10854674 Ki = 17 nM T13260 C3UJ7E 10859502 Ki = 68 nM T13260 C26ARU 10859572 Ki = 22 nM T13260 CM5B1D 10883602 IC50 = 12 nM T13260 CVD0E9 10895435 IC50 > 40 ug.mL-1 T13260 CW9Z8X 10900865 IC50 > 40 ug.mL-1 T13260 CP85BH 10902291 Ki = 100 nM T13260 CWZC05 10903498 IC50 = 6.9 nM T13260 C59BGC 10904721 IC50 = 1.1 nM T13260 CXD1M3 10913975 IC50 > 40 ug.mL-1 T13260 C9UJN5 10914511 Ki = 60 nM T13260 CHX8K0 10927303 Ki = 70 nM T13260 CR6CX8 10957235 Ki = 170 nM T13260 C7QXL8 10958364 IC50 > 40 ug.mL-1 T13260 CX9N0T 10990534 IC50 > 40 ug.mL-1 T13260 C0VSL5 11001084 IC50 = 4500 nM T13260 CE3YX7 11015855 IC50 > 40 ug.mL-1 T13260 C04SCF 11023115 Ki = 110 nM T13260 CU5B1T 11033539 Ki = 58 nM T13260 CUQP81 11034900 Ki = 60 nM T13260 CZR21O 11066682 Ki = 250 nM T13260 CRE6W0 11078050 Ki = 90 nM T13260 CWR14N 11079165 IC50 = 39 nM T13260 C9IE5F 11085889 IC50 = 1600 nM T13260 CC2NG5 11109070 IC50 = 23 nM T13260 C52NIS 11140706 IC50 = 1800 nM T13260 CMB40V 11140772 IC50 = 2400 nM T13260 CDI1L7 11141249 Ki = 800 nM T13260 CZ31ND 11141567 IC50 = 5500 nM T13260 C5LS1V 11153057 Ki = 900 nM T13260 C63APE 11164320 IC50 = 610 nM T13260 C7TKN9 11164739 IC50 = 9200 nM T13260 CM59ZA 11176755 Ki = 1160 nM T13260 C1A9IY 11179136 IC50 = 530 nM T13260 C2KJ6H 11196148 IC50 = 168 nM T13260 CTA9B3 11197738 IC50 = 50 nM T13260 CFQ8X5 11213800 IC50 > 100000 nM T13260 C0IC8T 11218132 IC50 = 13900 nM T13260 CQ0IG4 11219074 IC50 = 3600 nM T13260 C1TP7W 11232831 IC50 = 150 nM T13260 CQGN76 11241635 IC50 = 31622.78 nM T13260 CR9UT3 11243132 IC50 = 100000 nM T13260 CC9X2S 11244229 IC50 > 100000 nM T13260 CD15BO 11244509 IC50 = 32 nM T13260 CFYD58 11246736 Ki = 1690 nM T13260 C8PJ7G 11265329 IC50 = 31622.78 nM T13260 C2A0GX 11276968 IC50 = 3380 nM T13260 C0V4IO 11288325 IC50 = 280 nM T13260 CR1JS5 11310894 IC50 = 9770 nM T13260 CRW74G 11322098 IC50 = 144 nM T13260 CI9H7S 11347268 Ki = 3.4 nM T13260 C8SK0O 11356920 IC50 = 1122.02 nM T13260 C9AO5H 11381850 IC50 > 50000 nM T13260 CXDT28 11392371 IC50 = 250 nM T13260 C5X7KI 11402766 IC50 = 26915.35 nM T13260 CH4VM5 11413971 IC50 = 2818.38 nM T13260 CX63YZ 11417114 IC50 = 3600 nM T13260 CF7J8A 11426612 IC50 = 5128.61 nM T13260 CAU8M0 11448232 IC50 = 2820 nM T13260 CO7U8R 11485667 IC50 > 100000 nM T13260 CA90VB 11493223 Ki = 100 nM T13260 CXP5I7 11493374 IC50 = 440 nM T13260 C8P4VL 11493892 IC50 = 960 nM T13260 CEFC74 11495013 IC50 = 12 nM T13260 CV02WR 11515409 IC50 = 1210 nM T13260 C3XAL1 11522408 IC50 = 15.3 nM T13260 CV58AY 11522728 IC50 = 470 nM T13260 CV3U7F 11530377 Ki = 100 nM T13260 CN4T0K 11544009 IC50 = 970 nM T13260 CDG7N4 11544414 IC50 = 110 nM T13260 CSW1P3 11551000 IC50 = 2810 nM T13260 CL5E7M 11558482 IC50 = 870 nM T13260 CAEQ30 11565696 IC50 = 300 nM T13260 CHJB42 11567631 IC50 = 0.92 nM T13260 CF51ZE 11568594 IC50 = 3.9 nM T13260 CX6OV1 11572776 Ki = 100 nM T13260 CVK75E 11572824 IC50 = 760 nM T13260 C5KNY1 11573432 IC50 = 630.96 nM T13260 COX19Z 11581191 IC50 = 176 nM T13260 C9IJ3T 11594132 IC50 = 1252 nM T13260 CBV48A 11595426 IC50 = 95.5 nM T13260 CKTA53 11603462 IC50 = 0.77 nM T13260 C3VHL8 11611589 IC50 = 99 nM T13260 CAM20K 11624089 Ki = 75 nM T13260 CB2L9J 11624690 IC50 = 160 nM T13260 C5Y6MN 11633212 IC50 = 25.5 nM T13260 C2UBZ0 11639518 IC50 = 290 nM T13260 C7SYX1 11644772 IC50 = 5870 nM T13260 C0ZD2V 11645369 IC50 = 230 nM T13260 C2WF8E 11653632 IC50 = 3960 nM T13260 C9QOK8 11654142 IC50 = 17.5 nM T13260 C1OU0F 11667385 IC50 = 2.291 nM T13260 CP6TI4 11681050 Ki = 147 nM T13260 CZA7U6 11687547 IC50 > 25000 nM T13260 CWH82Z 11696602 IC50 = 49 nM T13260 CZ50DQ 11708478 IC50 > 2000 nM T13260 C7WN6I 11716932 IC50 = 4490 nM T13260 CTHL93 11722357 Ki = 1.4 nM T13260 C59DIH 11723061 Ki = 4.9 nM T13260 CS4AR9 11723111 Ki = 3.4 nM T13260 CZH43C 11725276 IC50 = 1800 nM T13260 C0MD6A 11732219 IC50 = 2.3 nM T13260 CFB08O 11737365 IC50 = 0.06 nM T13260 CW2B3A 11738647 IC50 = 51 nM T13260 CD0KR5 11739060 IC50 = 107.15 nM T13260 CUTV09 11758702 IC50 > 16100 nM T13260 CLND03 11758964 IC50 = 150000 nM T13260 CG79IH 11760852 IC50 = 1800 nM T13260 CM2LK4 11774754 IC50 > 100000 nM T13260 CA7S0C 11779699 Ki = 5000 nM T13260 CIJQ20 11784241 IC50 > 50000 nM T13260 C83WAR 11792329 Ki = 2.5 nM T13260 C0LM8Q 11793414 Ki = 17 nM T13260 CIU5X2 11807837 Ki = 50 nM T13260 CZC18Q 11824496 IC50 = 1500 nM T13260 C3V9LP 11833981 IC50 = 420 nM T13260 C7W4TJ 11842924 IC50 = 910 nM T13260 CTCY19 11843079 IC50 = 2500 nM T13260 C81VMW 11843080 IC50 = 10000 nM T13260 C9YK3J 12137521 IC50 > 100000 nM T13260 CY0A2H 12846880 IC50 > 50000 nM T13260 CW7EC6 12854713 IC50 = 38300 nM T13260 CP94EZ 13257279 IC50 = 170000 nM T13260 CNKO41 13288738 IC50 = 54 nM T13260 C70ESC 13437151 IC50 > 50000 nM T13260 CW02LQ 13537950 IC50 = 245000 nM T13260 C90PFA 13537951 IC50 = 6000 nM T13260 CJ05FQ 13537952 IC50 = 2500 nM T13260 C6OQT1 13537953 IC50 = 3600 nM T13260 CAQK75 13537954 IC50 = 3200 nM T13260 CK6AZ4 13537955 IC50 = 330 nM T13260 C6RM8P 13537956 IC50 = 2400 nM T13260 C9XFJ0 13596071 Ki = 1750 nM T13260 C29SJW 13633181 Ki = 41 nM T13260 CY8V7Z 13633182 Ki = 36 nM T13260 C9LM0A 13633183 Ki = 73 nM T13260 CZP9U6 13633184 Ki = 36 nM T13260 CUX8Y6 13660214 IC50 > 300000 nM T13260 CJ41AQ 13660215 IC50 = 135000 nM T13260 CT0A6S 13660217 IC50 = 16000 nM T13260 CMR8V5 13660219 IC50 = 3000 nM T13260 C7YMZ1 13660220 IC50 = 3000 nM T13260 C9ZAK2 13660222 IC50 = 400 nM T13260 C6CVT0 13660223 IC50 = 1100 nM T13260 CL0B9C 13660224 IC50 = 600 nM T13260 CM26OE 13686727 IC50 = 1150 nM T13260 CB1XD6 13688211 IC50 = 3.2 nM T13260 C1F5IT 13688212 IC50 = 3.2 nM T13260 CA6Z5U 13688213 IC50 = 21 nM T13260 C0D4XQ 13688215 IC50 > 1000 nM T13260 CG0KB9 13688216 IC50 = 17.6 nM T13260 C3D8YA 13688218 IC50 = 14.3 nM T13260 CNF97R 13833941 IC50 = 880 nM T13260 C8LRB9 13900578 IC50 = 385000 nM T13260 CT1EY3 13900579 IC50 = 31000 nM T13260 C7IM0K 13900580 IC50 = 40000 nM T13260 CNC7F2 13900581 IC50 = 21000 nM T13260 CXLQ60 13900582 IC50 = 6600 nM T13260 C3HEP2 13900583 IC50 = 1500 nM T13260 C3DM0W 13900584 IC50 = 3000 nM T13260 C3TLJ9 13900585 IC50 = 10000 nM T13260 CS5G4U 13900586 IC50 = 30000 nM T13260 CG7O6E 13964844 Ki = 10000 nM T13260 C28GTK 13990942 Ki = 55 nM T13260 CS82TI 13990943 Ki = 53 nM T13260 CAY1C9 13991369 Ki = 100 nM T13260 C7LKS8 14055913 Ki = 690 nM T13260 CE6L1R 14055915 Ki = 260 nM T13260 CVU6D4 14068934 Ki = 1200 nM T13260 C27JCM 14068935 IC50 = 2500 nM T13260 C9X6BY 14068936 Ki = 50 nM T13260 CQO06Z 14068937 Ki = 1.5 nM T13260 CEK04X 14068938 Ki = 20 nM T13260 CY8M0H 14068939 IC50 = 4000 nM T13260 C7G8AL 14068940 IC50 = 200 nM T13260 C4WV0N 14068941 IC50 = 200 nM T13260 CYM3T7 14068942 IC50 = 2000 nM T13260 C8PIS0 14068943 IC50 = 7000 nM T13260 CNG31F 14068944 IC50 = 700 nM T13260 CDIY35 14077737 Ki = 45 nM T13260 C8GXN7 14097196 IC50 = 7.6 nM T13260 CLZ6B8 14097212 IC50 = 2 nM T13260 CN48CH 14097214 IC50 = 14.1 nM T13260 C0G6FZ 14131679 IC50 > 10000 nM T13260 CG3QI0 14166614 IC50 = 1180 nM T13260 C98EGQ 14196997 IC50 = 100 nM T13260 CL74NV 14213544 IC50 > 40 ug.mL-1 T13260 CI3FX8 14231148 IC50 = 47.86 nM T13260 CC8A0Q 14231150 IC50 = 10.96 nM T13260 CVG0J5 14231162 IC50 = 37.15 nM T13260 C67SBC 14231174 IC50 = 58.88 nM T13260 C58ATZ 14236566 IC50 > 40 ug.mL-1 T13260 CX17LO 14311671 Ki = 670 nM T13260 CDT9L8 14442755 Ki = 260 nM T13260 CJ2CW1 14442756 Ki = 103000 nM T13260 CJX8L5 14442758 Ki = 1198000 nM T13260 CL23QM 14442760 Ki = 130000 nM T13260 CY1G3T 14442762 Ki = 893000 nM T13260 CBI6E0 14442764 Ki = 13000 nM T13260 CI93VX 14442766 Ki = 8560 nM T13260 CKI1V2 14442768 Ki = 3980 nM T13260 C1LZV9 14442770 Ki = 45000 nM T13260 C2TWN4 14442772 Ki = 97000 nM T13260 CQ47RM 14542252 IC50 > 40 ug.mL-1 T13260 C91JNH 14607641 Ki = 100 nM T13260 CM4J5C 14670839 IC50 > 20000 nM T13260 C6CX1G 14732022 Ki = 46 nM T13260 C9OIP8 14777454 Ki = 12 nM T13260 CM52ZO 14777455 Ki = 12 nM T13260 CGE64N 14777478 Ki = 610 nM T13260 CB78FM 14852902 IC50 = 95.5 nM T13260 C3L8RM 14860771 Ki = 170 nM T13260 CYJU57 14860774 Ki = 289 nM T13260 CD6GC9 14860775 Ki = 170 nM T13260 C5EL2K 14860776 IC50 = 38000 nM T13260 CJ47KS 14860787 IC50 = 44000 nM T13260 C86IZO 14860791 IC50 = 100000 nM T13260 CUK4V7 14860794 Ki = 228 nM T13260 CUC7R6 14860795 Ki = 455 nM T13260 CT8X3G 14860799 Ki = 443 nM T13260 CQ2KA6 14860801 IC50 = 26000 nM T13260 CG41LP 14860811 Ki = 7750 nM T13260 C3TC1N 14872622 IC50 = 111 nM T13260 CIX71V 14872623 IC50 = 225 nM T13260 CLSM38 14872624 IC50 = 13 nM T13260 CN3O6Y 14872625 IC50 = 97 nM T13260 CY9G4S 14872626 IC50 = 240 nM T13260 CKW32M 14872634 IC50 = 2000 nM T13260 CK94GY 14872635 IC50 = 62 nM T13260 CD30OJ 14872636 IC50 = 31 nM T13260 C2OL5D 14872637 IC50 = 49 nM T13260 CLAX71 14890692 IC50 = 150 nM T13260 C62CXN 14890719 IC50 = 2100 nM T13260 C71PWS 14890720 IC50 = 13000 nM T13260 C92AQW 14927492 Ki = 1410 nM T13260 C92OWZ 14929519 IC50 > 98400 nM T13260 CP9F8I 14939800 IC50 = 17000 nM T13260 CS26UK 15068090 Ki = 926 nM T13260 C19BZH 15068091 Ki = 870 nM T13260 C3WMI4 15072946 IC50 = 6300 nM T13260 CRHI64 15072947 IC50 = 8912.51 nM T13260 CVU3M9 15072948 IC50 = 691.83 nM T13260 CD06BM 15072949 IC50 = 8600 nM T13260 CFM3T0 15072950 IC50 = 3000 nM T13260 C39GNY 15072951 IC50 = 2200 nM T13260 CBC15T 15072952 IC50 = 6200 nM T13260 CI2QF0 15072953 IC50 = 4900 nM T13260 CAM0B5 15079867 IC50 = 7.2 nM T13260 C69EXT 15079869 IC50 = 43.65 nM T13260 CB0HE6 15079883 IC50 = 95.5 nM T13260 C8KQE9 15180664 IC50 = 290 nM T13260 C3RQS5 15182462 IC50 = 3350 nM T13260 CJ09IM 15182464 IC50 = 69 nM T13260 C9KTC2 15182466 IC50 = 10000 nM T13260 C0H2MI 15182467 IC50 = 30.2 nM T13260 CQM9J1 15182468 IC50 = 370 nM T13260 C7D1CO 15182471 IC50 = 2800 nM T13260 CL7C3M 15182472 IC50 = 2818.38 nM T13260 C5YCE7 15182473 IC50 = 933.25 nM T13260 CB0K4F 15182475 IC50 = 330 nM T13260 C8LSJ6 15182477 IC50 = 66 nM T13260 C07YXF 15192231 IC50 = 96 nM T13260 CSR6T4 15250744 IC50 = 650 nM T13260 CL4E7S 15250885 Ki = 38 nM T13260 CRBA42 15250961 Ki = 100 nM T13260 CX03MI 15250962 Ki = 100 nM T13260 CG28BA 15341075 Ki = 6 nM T13260 CV05SR 15341076 Ki = 12 nM T13260 C30CFK 15383327 Ki = 58 nM T13260 CY5D3M 15485639 IC50 > 50000 nM T13260 C4E5CF 15516845 IC50 > 242400 nM T13260 C6W1EU 15541561 IC50 = 1700 nM T13260 C6FW0G 15658944 IC50 = 2700 nM T13260 CCEG42 15658945 IC50 = 800 nM T13260 C5FH9P 15658946 IC50 = 940 nM T13260 CS97IP 15658947 Ki = 36 nM T13260 CMZ08Y 15658949 Ki = 169 nM T13260 CXQG31 15680919 IC50 = 23000 nM T13260 C1OD2W 15680920 IC50 > 200000 nM T13260 CJ80RP 15680922 IC50 = 4100 nM T13260 C0NHV8 15680923 IC50 = 26000 nM T13260 CMD4C5 15703577 IC50 = 1200 nM T13260 C2CZB1 15710342 IC50 = 10000 nM T13260 CN4H6E 15754992 Ki = 2200 nM T13260 C2TB7G 15765776 IC50 = 42300 nM T13260 CZ32OY 15801213 Ki = 8.8 nM T13260 CV3N8J 15819093 Ki = 143 nM T13260 CTQK31 15926847 Ki = 1424 nM T13260 C7ZF5H 15926848 Ki = 1424 nM T13260 CK90YW 15926849 Ki = 61 nM T13260 CT7KD6 15926850 Ki = 60.9 nM T13260 C1T5KN 15926851 Ki = 174 nM T13260 CX7EL3 15926852 Ki = 60.9 nM T13260 CATK37 15926853 Ki = 94 nM T13260 C6FX8Y 15926855 Ki = 95 nM T13260 CYKA87 15926857 Ki = 88 nM T13260 CIN54V 15926859 Ki = 88 nM T13260 C31YEX 15949288 IC50 = 3000 nM T13260 CWIH26 16004744 IC50 = 180 nM T13260 CDO2P0 16051602 IC50 = 180 nM T13260 CA2MG0 16051603 IC50 = 700 nM T13260 CR0V1J 16051604 IC50 = 1100 nM T13260 CN05YL 16051605 IC50 = 1340 nM T13260 CBR91V 16051709 IC50 = 550 nM T13260 CI7AB0 16059386 IC50 = 20000 nM T13260 C4IX5G 16063410 IC50 = 12630 nM T13260 CAJ31C 16078976 IC50 = 3680 nM T13260 CU32JA 16114920 IC50 = 28300 nM T13260 C1WMH9 16124988 IC50 = 2170 nM T13260 C43QWJ 16124989 IC50 = 330 nM T13260 C0CA7G 16125055 IC50 = 2330 nM T13260 C9PM6N 16125056 IC50 = 7820 nM T13260 CG8R9J 16125059 IC50 = 580 nM T13260 CAT4J7 16125061 IC50 = 330 nM T13260 C30WQC 16125062 IC50 = 850 nM T13260 CY6T7B 16125116 IC50 = 230 nM T13260 CQI2W7 16125118 IC50 = 1170 nM T13260 C0A1WJ 16125119 IC50 = 370 nM T13260 CVG37K 16125176 IC50 = 810 nM T13260 CF93LW 16125180 IC50 = 400 nM T13260 C9JBA6 16125181 IC50 = 260 nM T13260 CDG07Z 16125182 IC50 = 490 nM T13260 CR9SW1 16125242 IC50 = 2680 nM T13260 C42SBM 16125249 IC50 = 1750 nM T13260 C4H7BV 16125314 IC50 = 7450 nM T13260 C9FQU1 16125315 IC50 = 5850 nM T13260 CXD90Z 16125316 IC50 = 5740 nM T13260 C8OYB6 16125317 IC50 = 470 nM T13260 CK1YQ5 16125318 IC50 = 1780 nM T13260 C3M9OJ 16125319 IC50 = 2400 nM T13260 C38VAJ 16125320 IC50 = 650 nM T13260 CU3X2I 16125321 IC50 = 520 nM T13260 CBL30A 16126879 IC50 = 70 nM T13260 C9BC0L 16732000 IC50 > 100000 nM T13260 C6G0AI 16737077 IC50 > 261500 nM T13260 C03XMV 16737078 IC50 > 261500 nM T13260 CI6AJ9 16737167 IC50 > 271400 nM T13260 CUB9P7 16737277 IC50 = 3670 nM T13260 C3IJ8X 16737837 IC50 = 13950 nM T13260 C6ITS8 16738014 IC50 = 4670 nM T13260 CZ7PO3 16738015 IC50 = 28650 nM T13260 C4VB7R 16738021 IC50 = 4080 nM T13260 C5B7NL 16738022 IC50 = 4750 nM T13260 CX5QL0 16738023 IC50 = 12100 nM T13260 CC9XH1 16738210 IC50 = 54670 nM T13260 CJNP76 16738212 IC50 = 82940 nM T13260 CEIO82 16738409 IC50 > 283750 nM T13260 CB79UM 16738411 IC50 = 7670 nM T13260 CCE5G1 16738412 IC50 = 25140 nM T13260 C8QEL7 16738421 IC50 > 295500 nM T13260 CF9ZR8 16738422 IC50 > 310200 nM T13260 CG3F9E 16747839 IC50 = 0.6 nM T13260 CUX1Q4 16747937 IC50 = 560 nM T13260 CN43EH 16747938 IC50 = 7.3 nM T13260 C19REJ 16747939 IC50 = 260 nM T13260 CFI2P7 16747940 IC50 = 5.3 nM T13260 CBZE53 16747941 IC50 = 31 nM T13260 C6RB8S 16747942 IC50 = 25.9 nM T13260 CC5OW7 16748063 IC50 = 17.7 nM T13260 C6H2YB 16748064 IC50 = 400 nM T13260 CVHS73 16748915 IC50 = 0.33 nM T13260 CFX0I7 16749017 IC50 = 1.5 nM T13260 C23CUO 16749018 IC50 = 2.8 nM T13260 CEB09A 16749022 IC50 = 27 nM T13260 C03MDH 16749112 IC50 = 0.88 nM T13260 C6L3DF 16749115 IC50 = 0.51 nM T13260 CS7G6V 16749118 IC50 = 7.6 nM T13260 C0C8HL 16749219 IC50 = 159 nM T13260 CZV59A 16749224 IC50 = 0.18 nM T13260 CNG1F9 16749332 IC50 = 0.5 nM T13260 CQNA43 16749333 IC50 = 1.2 nM T13260 CNHX39 16749336 IC50 = 0.4 nM T13260 CBU08D 16749337 IC50 = 42 nM T13260 C6U7AF 16749441 IC50 = 2.9 nM T13260 CG5KQ0 16749446 IC50 = 24 nM T13260 CC2YU9 17255947 IC50 = 28.7 nM T13260 CHUA83 17966236 Ki = 2400 nM T13260 CKQJ89 18599501 Ki = 8.2 nM T13260 C6WT3S 18628989 IC50 = 913 nM T13260 CZ7PK3 18632820 IC50 = 1000 nM T13260 CT85EY 18731901 IC50 > 50000 nM T13260 CK3SA5 19043020 IC50 = 288.4 nM T13260 C4YOJ7 19043038 IC50 = 147.91 nM T13260 CKX53Q 19043046 IC50 = 870.96 nM T13260 CNS3K1 20757276 IC50 = 750 nM T13260 CK87YW 20841680 Ki = 106 nM T13260 CSKO15 21044501 IC50 = 0.51 nM T13260 CVA07N 21044507 IC50 = 0.73 nM T13260 CA7ZH9 21121774 Ki = 610 nM T13260 C16NDX 21142052 IC50 > 12500 nM T13260 CWPF92 21278956 IC50 = 2300 nM T13260 C3K1MC 21682806 IC50 = 300 nM T13260 C9WKT3 21976841 IC50 = 2.8 nM T13260 CK2ZS8 21976856 IC50 = 43 nM T13260 CE7PI2 21976872 IC50 = 2.5 nM T13260 CN5FM4 21976888 IC50 = 15 nM T13260 C9CG8L 21976892 IC50 = 10 nM T13260 C6WC7P 21976903 IC50 = 2.9 nM T13260 C75VCH 21976905 IC50 = 178 nM T13260 CR9C7D 21976908 IC50 = 0.28 nM T13260 C1KU7Z 22278552 Ki = 150 nM T13260 CR73VN 22809920 Ki = 100 nM T13260 C25LBI 23220724 IC50 = 4580 nM T13260 CLV8H7 23365315 IC50 = 18.2 nM T13260 C9ALK0 23383196 IC50 = 270 nM T13260 CHL65N 23585513 IC50 = 14.4 nM T13260 CHW5O3 23585518 IC50 = 275 nM T13260 CMN52Q 23585571 IC50 = 0.2 nM T13260 CN3CK2 23585671 IC50 = 0.5 nM T13260 CWR42I 23585720 IC50 = 0.15 nM T13260 C43IUA 23585722 IC50 = 0.2 nM T13260 CVFG27 23585723 IC50 = 0.1 nM T13260 CVJ95M 23585770 IC50 = 6 nM T13260 C30WOI 23585773 IC50 = 74 nM T13260 C5VWK3 23644932 Ki = 1820 nM T13260 CT8BJ4 23644933 Ki = 250 nM T13260 C6D9MC 23644934 Ki = 4400 nM T13260 COB81D 23644935 IC50 = 18000 nM T13260 C91ZAQ 23644936 IC50 > 50000 nM T13260 CWX70I 23644937 IC50 > 50000 nM T13260 C2I1BV 23644938 IC50 > 50000 nM T13260 C13NZL 23644951 IC50 = 85 nM T13260 CKBT84 23644968 Ki = 54 nM T13260 CC7FB8 23644969 Ki = 19 nM T13260 CJ3FX4 23644970 Ki = 22 nM T13260 C40DSL 23644971 Ki = 16 nM T13260 C8LJ4B 23644972 Ki = 11 nM T13260 C38VLD 23644973 Ki = 25 nM T13260 CNQ12D 23644974 Ki = 20 nM T13260 CR8VS6 23644975 Ki = 43 nM T13260 CF47DK 23644976 Ki = 4.7 nM T13260 CH5L6T 23644977 Ki = 7 nM T13260 CY1EL0 23644978 Ki = 14 nM T13260 C20LOE 23644979 Ki = 5 nM T13260 CDZN28 23644980 Ki = 8 nM T13260 CBVS04 23644981 Ki = 7.8 nM T13260 CO26RY 23644982 IC50 = 0.037 nM T13260 C4BPW5 23644983 IC50 = 0.11 nM T13260 CYV81F 23644984 IC50 = 0.23 nM T13260 CGF0J4 23644985 IC50 = 9 nM T13260 CVX82D 23644986 IC50 > 50 nM T13260 CG98LY 23644987 IC50 = 0.049 nM T13260 C9JD7L 23644988 IC50 = 0.32 nM T13260 C9JHP1 23644989 IC50 = 0.44 nM T13260 C7ZTD4 23644990 IC50 = 12 nM T13260 COF70P 23644991 IC50 > 50 nM T13260 CYG5P8 23644992 IC50 = 0.19 nM T13260 C74ILW 23644993 IC50 = 0.16 nM T13260 C5T6NR 23644994 IC50 = 0.12 nM T13260 C6FK7A 23644995 IC50 = 0.05 nM T13260 CIN07U 23644996 IC50 = 0.26 nM T13260 C8NY5J 23644997 IC50 = 0.13 nM T13260 C6EZ5V 23644998 Ki = 0.38 nM T13260 C0KZA5 23644999 Ki = 0.18 nM T13260 CKH5D2 23645000 Ki = 2.9 nM T13260 C27FSX 23645001 Ki = 44 nM T13260 CIQ42N 23645002 IC50 > 50 nM T13260 CX8Q9F 23645003 Ki = 0.14 nM T13260 C50OAY 23645004 Ki = 0.34 nM T13260 C5I6RZ 23645005 Ki = 5.5 nM T13260 C6PFS4 23645006 IC50 > 50 nM T13260 CIKQ38 23645007 IC50 > 50 nM T13260 C2DK6T 23645008 Ki = 0.045 nM T13260 CM2JR9 23645024 IC50 = 7400 nM T13260 C0HD7V 23645025 IC50 = 22 nM T13260 C73XCN 23645026 IC50 = 870 nM T13260 CTU28I 23645027 IC50 > 10000 nM T13260 CTUW15 23645028 IC50 > 10000 nM T13260 CL35CQ 23645029 IC50 = 10000 nM T13260 C2P7DG 23645030 IC50 > 10000 nM T13260 C89VHK 23645031 IC50 > 10000 nM T13260 CGKW86 23645032 IC50 > 1000 nM T13260 C2I9XH 23645033 IC50 = 400 nM T13260 C3J6KZ 23645034 IC50 > 10000 nM T13260 CEM21C 23645035 IC50 > 1000 nM T13260 CQ1KF8 23645036 IC50 > 1000 nM T13260 C1IT7Q 23645037 IC50 > 1000 nM T13260 CM81SC 23645038 IC50 > 1000 nM T13260 CA7DX4 23645039 IC50 > 1000 nM T13260 C1CQ4N 23645040 IC50 = 1000 nM T13260 CJV60Q 23645041 IC50 = 570 nM T13260 CQH8D4 23645042 IC50 = 270 nM T13260 C9L5EJ 23645043 IC50 = 50 nM T13260 C1X5NC 23645044 IC50 > 1000 nM T13260 CA76DP 23645045 IC50 > 1000 nM T13260 CLK43G 23645046 IC50 > 1000 nM T13260 C74MFK 23645047 IC50 = 330 nM T13260 CF48RD 23645048 IC50 = 50 nM T13260 C3A5VO 23645049 IC50 > 1000 nM T13260 CS2T8L 23645050 IC50 > 1000 nM T13260 CB24PD 23645051 IC50 > 1000 nM T13260 CLCA31 24204030 IC50 = 3100 nM T13260 CQ41JU 24204037 IC50 = 2400 nM T13260 CPJ8Z9 24205803 IC50 = 4400 nM T13260 CRH52Y 24205804 IC50 = 9100 nM T13260 C2PYN1 24420563 IC50 = 160 nM T13260 CP1YO7 24424201 IC50 = 800 nM T13260 CGVM50 24431784 IC50 > 50000 nM T13260 C6D2NZ 24692916 IC50 = 3715.35 nM T13260 CBU73T 24806841 IC50 > 25000 nM T13260 CA0YQ2 24806842 IC50 > 25000 nM T13260 CC92RE 24806843 IC50 > 25000 nM T13260 C17MET 24807041 IC50 > 25000 nM T13260 C9CMI7 24807042 IC50 > 25000 nM T13260 CZ6I0R 24807043 IC50 > 25000 nM T13260 CMY75P 24807044 IC50 > 25000 nM T13260 CJO96W 24807045 IC50 > 25000 nM T13260 CS8GB3 24807046 IC50 = 2170 nM T13260 C2B4HN 24807239 IC50 = 17370 nM T13260 C39TNQ 24807240 IC50 = 1100 nM T13260 C3PRI8 24807241 IC50 = 16670 nM T13260 CM4P0V 24807242 IC50 = 1770 nM T13260 CS01MP 24807243 IC50 = 250 nM T13260 C3BSZ8 24807244 IC50 = 690 nM T13260 CNTI27 24807245 IC50 = 690 nM T13260 C18DIO 24807434 IC50 = 440 nM T13260 C6CA8F 24807435 IC50 = 1070 nM T13260 C8NR1Y 24807436 IC50 = 120 nM T13260 CC73NY 24873506 IC50 = 1370 nM T13260 CAX9V3 24873507 IC50 = 1540 nM T13260 CS2IG5 24873508 IC50 = 610 nM T13260 C5TA7V 24873509 IC50 = 630 nM T13260 CW3C5U 24896569 IC50 = 38 nM T13260 CS5H2A 24896701 IC50 > 15300 nM T13260 CBZ10U 24901645 IC50 = 13 nM T13260 CY27CS 24901646 IC50 = 12 nM T13260 CD9IV7 24901647 IC50 = 3 nM T13260 CMFU23 24901648 IC50 = 3.2 nM T13260 CTJ76G 24901649 IC50 = 14.3 nM T13260 CJ7R6C 24901650 IC50 = 2457 nM T13260 CVS08H 24901651 IC50 = 169 nM T13260 C2H8EA 24901652 IC50 = 215 nM T13260 CUF1O4 24901653 IC50 = 5.5 nM T13260 C9C0AB 24901654 IC50 = 1.8 nM T13260 CEB6G1 24901655 IC50 = 0.6 nM T13260 CE5QO1 24901656 IC50 = 3.4 nM T13260 C23PCS 25022806 IC50 = 13.7 nM T13260 CF02OB 25071641 IC50 = 11.5 nM T13260 CMXL59 25111668 Ki = 2100 nM T13260 C35FYQ 25111796 IC50 > 500000 nM T13260 C8J2AP 25111799 IC50 > 500000 nM T13260 C06ECA 25111909 Ki = 1530 nM T13260 CON29S 25141424 IC50 = 0.45 nM T13260 CZX08M 25142015 Ki = 13 nM T13260 CV2DP9 25180002 IC50 = 6500 nM T13260 C0XHA2 25180109 IC50 = 426 nM T13260 CS8YW6 25227426 IC50 = 33000 nM T13260 CC1S3T 25256841 IC50 = 24400 nM T13260 CA4G8Y 42597583 IC50 = 13 nM T13260 C5N9MC 42611455 IC50 = 5300 nM T13260 C93BZJ 42618027 IC50 = 1250 nM T13260 C4YXR5 42618028 IC50 = 31500 nM T13260 CVLR83 42618034 IC50 = 5680 nM T13260 CUWO14 42618035 IC50 = 760 nM T13260 CZW8L2 43137984 IC50 = 289 nM T13260 CCZY29 44266320 IC50 = 620 nM T13260 C1BGQ4 44266331 IC50 = 1600 nM T13260 CEHD28 44266353 IC50 = 800 nM T13260 C79VFZ 44275189 Ki = 12 nM T13260 CQ31TG 44275201 Ki = 22 nM T13260 C83QEP 44275202 Ki = 6.7 nM T13260 CDK2T1 44275250 Ki = 5.1 nM T13260 CJ48ZL 44275251 Ki = 63 nM T13260 C78OQW 44275252 Ki = 31 nM T13260 CG4FB5 44275253 Ki = 10 nM T13260 C0OE3W 44275268 Ki = 21 nM T13260 CZ9K6I 44275269 Ki = 11 nM T13260 CP29RM 44275270 Ki = 37 nM T13260 CP2QV1 44275283 Ki = 5.6 nM T13260 C1A6OS 44275328 Ki = 4.7 nM T13260 CLN69H 44275329 Ki = 62 nM T13260 C1LQC6 44275331 Ki = 1.4 nM T13260 CZWI57 44275351 Ki = 8.8 nM T13260 C9R1OJ 44275355 Ki = 4.6 nM T13260 CC30JG 44276238 IC50 = 777000 nM T13260 CN9W6A 44276773 Ki = 75 nM T13260 C7GMW1 44277065 Ki = 1 nM T13260 C76XWA 44277083 Ki = 7 nM T13260 C3SU7M 44286352 IC50 = 170 nM T13260 CH4TJ0 44286353 IC50 = 2900 nM T13260 C74AKY 44286427 IC50 = 200 nM T13260 C0KVR6 44286475 IC50 = 70 nM T13260 C4WE8P 44286839 IC50 = 110 nM T13260 C2T1CJ 44286840 IC50 = 90 nM T13260 CZO6F2 44287464 Ki = 30 nM T13260 C8D9XI 44287465 Ki = 27 nM T13260 CK76RT 44287659 IC50 = 4400 nM T13260 C08POV 44287660 IC50 = 10000 nM T13260 CMA78S 44287741 IC50 = 4400 nM T13260 CGUX54 44287754 IC50 = 1200 nM T13260 CNF17L 44287801 Ki = 30 nM T13260 C5F6MV 44294033 Ki = 63 nM T13260 CHNJ98 44294100 Ki = 27 nM T13260 C7T9RN 44294311 Ki = 926 nM T13260 C5U1JS 44294312 Ki = 870 nM T13260 CMW32B 44294314 Ki = 11 nM T13260 C5JHW7 44294332 Ki = 190 nM T13260 C4TY5K 44306234 IC50 = 200 nM T13260 CCE7A4 44306491 IC50 = 52020 nM T13260 CUQ6L9 44306493 IC50 = 2170 nM T13260 CGU34E 44306494 IC50 = 3000 nM T13260 C9GRJ2 44306526 IC50 = 590 nM T13260 CN34EP 44306915 IC50 = 190 nM T13260 C8RQ5W 44306929 IC50 = 880 nM T13260 C80ZJS 44307719 Ki = 47 nM T13260 C76BWU 44307720 Ki = 28 nM T13260 CM52NG 44307837 Ki = 100 nM T13260 CF1K2N 44310044 Ki = 3000 nM T13260 CB30FN 44310045 Ki = 1800 nM T13260 C0QZ5L 44310046 Ki = 7000 nM T13260 C3QWV2 44310077 Ki = 13000 nM T13260 C32AUZ 44310078 Ki = 2000 nM T13260 CLJ45R 44310148 Ki = 1400 nM T13260 CEOU45 44310393 Ki = 5500 nM T13260 CZMQ71 44310410 Ki = 11000 nM T13260 CKNF03 44310411 Ki = 45000 nM T13260 C6X7WP 44310412 Ki = 9800 nM T13260 C90SJZ 44310767 Ki = 5300 nM T13260 C8W3VA 44310768 Ki = 11000 nM T13260 CO2SE0 44323417 IC50 = 3200 nM T13260 CRW0C1 44323482 IC50 = 2400 nM T13260 C0FAY8 44323523 IC50 = 2500 nM T13260 CRG1T9 44323592 IC50 = 31000 nM T13260 CQM56K 44323610 IC50 = 10000 nM T13260 C63FUL 44323664 IC50 = 3000 nM T13260 CVF86M 44323741 IC50 = 245000 nM T13260 CZIS73 44323756 IC50 = 21000 nM T13260 C0J6ZI 44323759 IC50 = 3600 nM T13260 CQC0G4 44323760 IC50 = 30000 nM T13260 CADY94 44323768 IC50 = 800 nM T13260 CGK6B2 44323782 IC50 = 1500 nM T13260 CQT35R 44323783 IC50 = 6600 nM T13260 CR5S8Z 44323807 IC50 = 40000 nM T13260 C87RGX 44323808 IC50 = 385000 nM T13260 CY1OB4 44323813 IC50 = 4000 nM T13260 CI0H9D 44323814 IC50 = 6000 nM T13260 CLE87R 44328597 Ki = 18.9 nM T13260 CX8DV2 44328668 Ki = 13.1 nM T13260 CXS8N4 44330891 Ki = 25000 nM T13260 C38YFI 44330892 Ki = 1100 nM T13260 C09VTC 44330997 Ki = 12 nM T13260 CFW8Q5 44330998 Ki = 3000 nM T13260 C5CF2O 44331012 Ki = 4.7 nM T13260 CQ85VL 44331071 Ki = 1 nM T13260 CL1YN0 44331102 Ki = 35000 nM T13260 CJIW38 44331119 Ki = 56 nM T13260 CHY39A 44331123 Ki = 1.3 nM T13260 C2MZO4 44331205 Ki = 2.3 nM T13260 CZHI57 44331221 Ki = 3 nM T13260 CXY2W3 44331222 Ki = 9 nM T13260 C28YNW 44331250 Ki = 33000 nM T13260 CR1YC8 44331322 IC50 = 30 nM T13260 CQR2U5 44333942 IC50 = 340 nM T13260 CL4Q0F 44333943 IC50 = 97 nM T13260 CX6Q1N 44334361 IC50 = 89 nM T13260 CB2D4V 44334394 IC50 = 9700 nM T13260 CSO4C8 44334411 IC50 = 11800 nM T13260 CCZ60G 44334579 IC50 = 310 nM T13260 CBZV02 44334580 IC50 = 120 nM T13260 CSR90W 44334594 IC50 = 2000 nM T13260 C8GAF6 44334595 IC50 = 3200 nM T13260 CIB4F8 44339828 Ki = 37 nM T13260 CS2F5B 44340058 Ki = 10 nM T13260 C7PT2A 44340059 Ki = 47.6 nM T13260 C9YAC2 44340330 Ki = 65.8 nM T13260 C0SC3B 44341451 IC50 = 5400 nM T13260 CAD1S9 44341468 IC50 = 238 nM T13260 CKE5L8 44353429 IC50 = 236 nM T13260 CYO3B6 44353430 IC50 = 245 nM T13260 C0UDL7 44353435 IC50 = 342 nM T13260 C3XP8T 44353437 IC50 = 950 nM T13260 C0KIV8 44353626 IC50 = 800 nM T13260 CME45Q 44353627 IC50 = 658 nM T13260 CX43HZ 44353643 IC50 = 490 nM T13260 CQ5UK0 44354378 IC50 = 530 nM T13260 CO8XJ3 44354706 IC50 = 120 nM T13260 C7YDP6 44354757 IC50 = 1320 nM T13260 C1W6IR 44354758 IC50 = 3960 nM T13260 C4AXM5 44354773 IC50 = 440 nM T13260 CZN1X8 44354907 IC50 = 30000 nM T13260 CN8M5U 44354930 IC50 = 5600 nM T13260 CCA28Y 44354942 IC50 = 55000 nM T13260 CNRO38 44354943 IC50 = 3850 nM T13260 CQIP34 44354944 IC50 = 80500 nM T13260 CO1W4F 44355172 IC50 = 8900 nM T13260 CX2R3P 44355187 IC50 > 20000 nM T13260 CCF7G1 44355188 IC50 = 1700 nM T13260 C64IWU 44358640 IC50 = 7100 nM T13260 CR5M1D 44369877 Ki = 18 nM T13260 C3BDK1 44369898 Ki = 65 nM T13260 CKNO08 44369927 Ki = 59 nM T13260 CL19DY 44376315 IC50 = 92.9 nM T13260 CZE46J 44378054 IC50 = 42 nM T13260 C1I0NW 44381001 IC50 > 250000 nM T13260 CDTS58 44387709 IC50 = 15 nM T13260 CUNZ83 44394828 IC50 = 1400 nM T13260 C8I1AE 44394829 IC50 = 31600 nM T13260 C2TLS9 44404116 Ki = 50 nM T13260 CLV8R2 44408288 IC50 = 29.7 nM T13260 C9DS0J 44408292 IC50 = 26.3 nM T13260 CTD91Q 44408293 IC50 = 23.7 nM T13260 C5X7TN 44408294 IC50 = 19.3 nM T13260 CIBP08 44421541 IC50 = 57.54 nM T13260 C0WU4A 44421546 IC50 = 93.33 nM T13260 CCIE32 44421551 IC50 = 3715.35 nM T13260 C9A6IF 44421559 IC50 = 47.86 nM T13260 C5FO6U 44424773 IC50 > 310170 nM T13260 C6BE0T 44456226 IC50 > 5000 nM T13260 CY7OD4 44461241 IC50 > 50000 nM T13260 C4BAS8 44462074 Ki = 228 nM T13260 C9BE8F 44462253 Ki = 455 nM T13260 C92QWL 44521066 IC50 = 0.12 nM T13260 CG16BM 44554135 IC50 = 11500 nM T13260 C47OVI 44562528 IC50 > 500000 nM T13260 CY42QT 44562549 IC50 > 500000 nM T13260 CP3T7B 44567161 IC50 > 40 ug.mL-1 T13260 C90PBX 44567164 IC50 > 40 ug.mL-1 T13260 C49DYC 44567218 IC50 = 7500 nM T13260 CO63LK 44569291 IC50 = 2.3 nM T13260 CNZV98 44577912 IC50 = 93.8 nM T13260 CRP8A7 44577913 IC50 = 18.7 nM T13260 CW8XY2 44577949 IC50 = 1620 nM T13260 C5CSL8 44578878 IC50 = 17300 nM T13260 C2ZWD9 44578879 IC50 = 5060 nM T13260 C4F2AM 44578880 IC50 = 1040 nM T13260 C1AT7Y 44578921 IC50 = 1060 nM T13260 C60AKC 44579025 IC50 = 320 nM T13260 C50KAN 44579026 IC50 = 9960 nM T13260 CJQ67H 44579027 IC50 = 2490 nM T13260 CS4JR7 44579028 IC50 = 1070 nM T13260 CHWK61 44579029 IC50 = 870 nM T13260 C8QW4K 44579570 IC50 = 13040 nM T13260 CP53WC 44580785 IC50 = 17000 nM T13260 CGBT61 45028483 IC50 > 10000 nM T13260 CVO41F 45140953 IC50 = 2 nM T13260 CRZ6N5 45140954 IC50 = 0.5 nM T13260 C01WQZ 45141152 IC50 = 2.4 nM T13260 CT5CR6 45141153 IC50 = 0.22 nM T13260 CC3FT1 45141154 IC50 = 0.35 nM T13260 C8PB0I 45141156 IC50 = 146 nM T13260 CL2Y7U 45141157 IC50 = 29.3 nM T13260 CH1LB7 45141158 IC50 = 19 nM T13260 CDE83B 45141365 IC50 = 52 nM T13260 CGA6Y4 45141366 IC50 = 112 nM T13260 CCIP58 45141367 IC50 = 280 nM T13260 C2S5QX 45141368 IC50 = 24 nM T13260 C2YJ8N 45141369 IC50 = 80 nM T13260 CO4UA1 45141370 IC50 = 920 nM T13260 C5CB0P 45141371 IC50 = 284 nM T13260 CTN65F 45141372 IC50 = 380 nM T13260 CGK5O7 45141601 IC50 = 571 nM T13260 C68SZB 45141602 IC50 = 0.8 nM T13260 C0C3AW 45141603 IC50 = 1.9 nM T13260 C0U7CG 45141604 IC50 = 0.3 nM T13260 CQ4JE3 45378299 IC50 = 97000 nM T13260 CUR6C8 45378303 IC50 = 5100 nM T13260 CY2SV8 45379302 IC50 = 44000 nM T13260 CSE09V 46177290 IC50 = 12100 nM T13260 C4XCR3 46177291 IC50 = 12100 nM T13260 C4S2AI 46198256 Ki = 16.1 nM T13260 CT07FB 46204132 IC50 = 6400 nM T13260 CN47GA 46228644 IC50 = 4.6 nM T13260 C6AMH8 46228668 IC50 = 1.7 nM T13260 CLD4Z5 46228698 IC50 = 0.22 nM T13260 CZH36E 46834487 IC50 > 50000 nM T13260 CUV83E 46854605 IC50 = 12000 nM T13260 CIA08B 46854608 IC50 = 9500 nM T13260 CWJ3F1 46854758 IC50 = 5060 nM T13260 CKRQ67 46854759 IC50 = 49500 nM T13260 CZ1YJ0 46854760 IC50 = 48700 nM T13260 CINV65 46867541 IC50 = 101 nM T13260 CL06TP 46887017 IC50 = 17.2 nM T13260 C0KFI6 46887054 IC50 = 17.2 nM T13260 C6R1HA 46887055 IC50 = 6 nM T13260 CD65CW 46887468 IC50 = 71.8 nM T13260 CM0EK7 46887507 IC50 = 200 nM T13260 CGBE96 46887549 IC50 = 210 nM T13260 C74CER 46887577 IC50 = 3.5 nM T13260 C2OMW7 46895138 IC50 = 12000 nM T13260 CYEA34 46913124 IC50 = 70 nM T13260 C5JR7T 46913125 IC50 = 36 nM T13260 CN1CV7 46939057 Ki = 97 nM T13260 CP8HY2 46939058 Ki = 27 nM T13260 CD67MH 46939156 Ki = 23 nM T13260 C1MFE9 46939157 Ki = 75 nM T13260 C0K8YL 46939158 Ki = 39 nM T13260 CX7B9G 46939159 Ki = 30 nM T13260 CL37EV 46939160 Ki = 56 nM T13260 C9CQU0 46953209 IC50 = 59.2 nM T13260 CUQ0Z7 46957695 IC50 = 13200 nM T13260 CU0KW6 46958302 IC50 = 991 nM T13260 CHN2P9 46960541 IC50 = 34.5 nM T13260 CR3OI4 46960542 IC50 = 46.7 nM T13260 CW3V2P 46962897 IC50 = 499 nM T13260 CQ0XE9 46964149 IC50 = 10600 nM T13260 CL0F1J 46964152 IC50 > 25000 nM T13260 CV3UT0 46967737 IC50 = 3100 nM T13260 CBAE65 46968168 IC50 = 248 nM T13260 CKJ9S6 46968847 IC50 = 3100 nM T13260 CO2XL1 46970377 IC50 = 9 nM T13260 C0GZ4Q 46980515 IC50 = 498 nM T13260 C8QCH2 49779539 IC50 = 2.1 nM T13260 C7V2XL 49779540 IC50 = 0.25 nM T13260 CIC9S5 49799473 IC50 = 5750 nM T13260 C5ZNK0 49799653 IC50 = 21860 nM T13260 CZG04F 49799654 IC50 = 8490 nM T13260 CX5LZ9 50915159 IC50 = 0.018 nM T13260 C8N5OK 50991893 IC50 = 0.21 nM T13260 C0RUX1 50994677 IC50 > 10000 nM T13260 CL2O0Y 50994839 IC50 > 16200 nM T13260 CTG6R4 51041013 IC50 = 4400 nM T13260 CGX85M 51042201 IC50 = 30700 nM T13260 CWG69M 51042401 IC50 = 32300 nM T13260 C1AT4L 51042402 IC50 = 26800 nM T13260 C1VF4Z 51346982 IC50 = 0.015 nM T13260 C6Y3EL 51346989 IC50 = 0.015 nM T13260 C8GQS7 51351108 IC50 > 50000 nM T13260 CB8ND9 51354813 IC50 > 16900 nM T13260 CMXR96 51355428 IC50 = 114 nM T13260 C5KTL3 51355429 IC50 = 113 nM T13260 C4UTM8 51355430 IC50 = 130 nM T13260 CH5C9K 51355431 IC50 = 235 nM T13260 CRK2Q9 51355432 IC50 = 207 nM T13260 CF7RG5 51355433 IC50 = 141 nM T13260 C8XHD9 51355434 IC50 = 267 nM T13260 C41SUK 51355703 IC50 = 178 nM T13260 CM6T7H 51355704 IC50 = 127 nM T13260 CZDA87 51355705 IC50 = 481 nM T13260 CO1V0Y 51355706 IC50 = 169 nM T13260 C2OCG3 51355707 IC50 = 165 nM T13260 CGLU79 51355708 IC50 = 72 nM T13260 CL6XD4 51355709 IC50 = 72 nM T13260 C57MWS 51355970 IC50 = 292 nM T13260 CYC86A 51355971 IC50 = 690 nM T13260 CP7V3Q 51355972 IC50 = 112 nM T13260 CR6NH8 51355973 IC50 = 164 nM T13260 C6SD4P 51355974 IC50 = 296 nM T13260 C97MZT 51355975 IC50 = 81 nM T13260 CJU1O7 51355976 IC50 = 70 nM T13260 CIR0L7 51356252 IC50 = 47 nM T13260 C0BW7G 51356253 IC50 = 105 nM T13260 C39RVA 51356254 IC50 = 3750 nM T13260 C3P5LI 51356255 IC50 = 455 nM T13260 CKXR01 51356256 IC50 = 67 nM T13260 CF21EH 51356258 IC50 = 317 nM T13260 C4M5ZT 51356554 IC50 = 532 nM T13260 CS7X3R 51356555 IC50 = 4010 nM T13260 CR7UG9 51356556 IC50 = 313 nM T13260 C87FEB 51520434 IC50 = 600 nM T13260 C42JIQ 52912619 IC50 = 5040 nM T13260 CY0TF7 53237486 IC50 = 510 nM T13260 C5WQX4 53237725 IC50 = 1000 nM T13260 CD7HC1 53305315 IC50 = 91 nM T13260 C5SN8I 53317948 IC50 = 11000 nM T13260 CQZV41 53318733 IC50 = 30000 nM T13260 C9OPT6 53320278 IC50 = 0.75 nM T13260 CDM50Q 53320823 IC50 = 660 nM T13260 CRLJ68 53321508 IC50 = 700 nM T13260 CCNP36 53321604 IC50 = 0.47 nM T13260 CDV3X5 53323228 IC50 = 3600 nM T13260 C4WY6N 53323229 IC50 = 1000 nM T13260 CFC42O 53323677 IC50 > 16800 nM T13260 CFMK70 53324579 IC50 = 280 nM T13260 C48XBG 53325332 IC50 = 860 nM T13260 CA32FG 53325544 IC50 = 0.05 nM T13260 CN0SW9 53326827 IC50 = 0.1 nM T13260 CSQ45A 53326828 IC50 = 0.15 nM T13260 C0AL2O 53482563 IC50 = 11.8 nM T13260 C0P3VM 53637746 Ki = 58 nM T13260 CAE25J 53763992 IC50 = 970 nM T13260 CUXV34 54026593 Ki = 120 nM T13260 C53FSN 54165563 Ki = 7 nM T13260 C8FA6I 54348149 Ki = 58 nM T13260 CA19BF 54513089 Ki = 25 nM T13260 CE0PC5 54576531 IC50 = 4640 nM T13260 CS0NM1 54576532 IC50 = 1360 nM T13260 CA3YL8 54580402 IC50 = 5790 nM T13260 CB5QY9 54583302 IC50 = 34 nM T13260 CB02LJ 54584262 IC50 = 32 nM T13260 C34FYG 54584352 IC50 = 66.5 nM T13260 CLPG92 54586184 IC50 = 36 nM T13260 C91LBU 54597383 IC50 = 3300 nM T13260 C6G8HK 54597384 IC50 = 1800 nM T13260 CV2NS6 54729584 IC50 = 220 nM T13260 C70EIF 54756790 IC50 > 50000 nM T13260 CZU5L8 54768666 IC50 = 17340 nM T13260 C4C1ZY 54768667 IC50 = 10700 nM T13260 C5AVO9 54770656 IC50 = 12200 nM T13260 C2RW0G 54770885 IC50 = 12010 nM T13260 CW6EK4 54770886 IC50 = 4700 nM T13260 CTP0G9 54770887 IC50 = 5070 nM T13260 CHY71M 54770888 IC50 = 10600 nM T13260 CS42BX 54770889 IC50 = 16020 nM T13260 CU07HL 54770890 IC50 = 19320 nM T13260 CD2JA7 54770891 IC50 = 10330 nM T13260 CD1V8X 54771121 IC50 = 79980 nM T13260 CMX14D 54771122 IC50 = 10970 nM T13260 CVED14 54771123 IC50 = 16110 nM T13260 CPJW41 54771124 IC50 = 7730 nM T13260 C8JEH4 54771125 IC50 = 10950 nM T13260 CA4JF1 54771126 IC50 = 12160 nM T13260 C6Y8ND 54771341 IC50 = 10960 nM T13260 C7E3KS 54771342 IC50 = 14830 nM T13260 C6NRM1 54771343 IC50 = 19360 nM T13260 C3MR9N 54771344 IC50 = 13540 nM T13260 CI5QD9 54771345 IC50 = 13720 nM T13260 C7KBU3 54771346 IC50 = 12940 nM T13260 C7LOA4 54771347 IC50 = 31260 nM T13260 C8OI5N 54771563 IC50 = 13350 nM T13260 CUF4O0 54771564 IC50 = 13370 nM T13260 CP1UM5 54771565 IC50 = 16410 nM T13260 C3ZKB4 54771566 IC50 = 11610 nM T13260 C3YD8A 54771567 IC50 = 26770 nM T13260 C3URW8 54771568 IC50 = 15210 nM T13260 C2BYD3 54771787 IC50 = 4370 nM T13260 CUY87L 54771788 IC50 = 5260 nM T13260 C3WVO7 54771789 IC50 = 3070 nM T13260 CYM98K 54771790 IC50 = 7880 nM T13260 CV5S9D 54771791 IC50 = 10700 nM T13260 C2G6DW 54771792 IC50 = 6090 nM T13260 CHOT94 54771793 IC50 = 3910 nM T13260 CA49SQ 54771794 IC50 = 9160 nM T13260 CN2ES5 54772014 IC50 = 15480 nM T13260 C38PQF 54772015 IC50 = 5620 nM T13260 C3Q9YI 54772016 IC50 = 4170 nM T13260 C76QVG 54772017 IC50 = 2340 nM T13260 C5KI4U 54772018 IC50 = 11570 nM T13260 CR1YL2 54772019 IC50 = 7470 nM T13260 C1OQ4B 54772020 IC50 = 9530 nM T13260 CL7XJ4 54772021 IC50 = 7980 nM T13260 C06PFH 56598207 IC50 = 10500 nM T13260 CL4KT8 56610874 Ki = 8.2 nM T13260 C78MXU 56612673 Ki = 8.2 nM T13260 CV1ZO2 56632357 Ki = 90 nM T13260 C4N0WL 56645363 IC50 = 1021 nM T13260 C57NSZ 56645568 IC50 = 1268 nM T13260 C6PUX9 56645570 IC50 = 4513 nM T13260 CM94ZH 56664989 IC50 = 2780 nM T13260 CMU51H 56681975 IC50 = 2270 nM T13260 C7G5IR 56835177 Ki = 790 nM T13260 C5US1Z 56835178 Ki = 60 nM T13260 C3IZU1 56835179 Ki = 50 nM T13260 CRGX16 56837844 IC50 > 50000 nM T13260 C7M1OX 56837845 IC50 > 50000 nM T13260 CHCM56 56837846 IC50 > 50000 nM T13260 CX19AT 57327815 IC50 = 93 nM T13260 C0I2DY 57327816 IC50 = 59 nM T13260 CY58ZD 57330086 IC50 > 5000 nM T13260 C1C0FZ 57384102 Ki = 0.06 nM T13260 CLJ8A1 57384103 Ki = 0.65 nM T13260 C6I3AN 57390179 IC50 > 50000 nM T13260 C1ZB3N 57390180 IC50 > 50000 nM T13260 CH19RM 57390181 IC50 > 50000 nM T13260 CG2J7F 57390275 IC50 = 64500 nM T13260 C0VRP8 57391308 Ki = 12560 nM T13260 C3BKO8 57391309 Ki = 1482 nM T13260 CW3P7T 57391581 Ki = 100 nM T13260 CI1R4S 57391583 Ki = 250 nM T13260 CB02XQ 57391954 IC50 > 50000 nM T13260 C94BSM 57392056 IC50 = 63200 nM T13260 CJA4L1 57393085 Ki = 1722 nM T13260 CS6V8A 57393681 IC50 > 50000 nM T13260 CPN7Q2 57393682 IC50 > 50000 nM T13260 CV4S6C 57393683 IC50 > 50000 nM T13260 CR5I9O 57393684 IC50 > 50000 nM T13260 C5VDL7 57395400 IC50 > 50000 nM T13260 CC53MX 57395527 IC50 = 47300 nM T13260 CV08LN 57395659 IC50 = 986 nM T13260 CI6Q5O 57395660 IC50 = 304 nM T13260 CQ06KW 57395661 IC50 = 229 nM T13260 C48VIY 57396573 Ki = 5321 nM T13260 C2NML8 57396574 Ki = 8.2 nM T13260 C83ZIP 57396575 Ki = 82.54 nM T13260 C2F1TI 57397238 IC50 > 50000 nM T13260 C4O5DT 57397345 IC50 = 68100 nM T13260 CBL9Z1 57397346 IC50 = 58600 nM T13260 CXP68J 57397347 IC50 = 72000 nM T13260 C5VLB1 57398353 Ki = 35.12 nM T13260 C4DE6B 57398582 Ki = 1000 nM T13260 CW2J6Z 57398927 IC50 > 50000 nM T13260 CP65RI 57398928 IC50 > 50000 nM T13260 CHB0A3 57398929 IC50 > 50000 nM T13260 C81RCO 57398930 IC50 > 50000 nM T13260 CD4BN7 57400011 Ki = 285.1 nM T13260 CJT2G9 57400012 Ki = 100 nM T13260 CJZX60 57400626 IC50 > 50000 nM T13260 CV8KD9 57400627 IC50 > 50000 nM T13260 C3G4RJ 57400766 IC50 = 44800 nM T13260 C2WJ7Y 57400842 IC50 = 57400 nM T13260 C5OYK8 57400879 IC50 = 114 nM T13260 CHVG47 57401821 Ki = 15000 nM T13260 C1MF0V 57402418 IC50 > 50000 nM T13260 CQ9C3L 57402419 IC50 = 26500 nM T13260 CUD85V 57402656 IC50 = 523 nM T13260 CD2U9L 57403526 Ki = 1160 nM T13260 CFI0L8 57403527 Ki = 3.17 nM T13260 C10SAL 57403795 Ki = 79.43 nM T13260 CRL10W 57413872 Ki = 86 nM T13260 C04MZQ 57520593 IC50 = 17000 nM T13260 CX8Q7H 57520594 IC50 = 5800 nM T13260 CYHS09 57679076 IC50 >= 200000 nM T13260 C7OK1X 57775654 IC50 = 4490 nM T13260 CQ0M7J 58215635 IC50 = 3400 nM T13260 C34JIZ 58255359 IC50 = 2130 nM T13260 C2TUJ7 58255382 IC50 = 228 nM T13260 C3DPC0 58255407 IC50 = 43 nM T13260 C9DK1X 58255415 IC50 = 488 nM T13260 CTI0D7 58255435 IC50 = 880 nM T13260 CRQ70M 58255438 IC50 > 500 nM T13260 CLQ65O 58255479 IC50 > 5000 nM T13260 CP6RA9 58255482 IC50 = 3073 nM T13260 CJX70M 58255566 IC50 = 105 nM T13260 CW71EO 58255581 IC50 = 447 nM T13260 C6XPA7 59356082 IC50 = 24000 nM T13260 CX2US1 59356084 IC50 = 35000 nM T13260 CD31PM 59356085 IC50 = 99000 nM T13260 CVRT12 59356087 IC50 = 41000 nM T13260 CLP2O3 60151424 IC50 = 6200 nM T13260 C9M4QI 60156307 IC50 = 112.3 nM T13260 CZ1WU8 60166590 IC50 = 169.3 nM T13260 CB7N8A 60195126 IC50 = 17 nM T13260 CE18JH 60202715 Ki = 48 nM T13260 CX4N0I 62707515 IC50 = 48 nM T13260 C0G3LA 66559847 IC50 = 49 nM T13260 C4RSI6 66559935 IC50 = 162 nM T13260 CDX7I8 66559936 IC50 = 22 nM T13260 CF9EQ5 66559939 IC50 = 2901 nM T13260 CQN6D3 66559940 IC50 = 394 nM T13260 CN4H8G 66559941 IC50 = 954 nM T13260 CTP6Q4 66559942 IC50 = 275 nM T13260 C9EGW2 66575742 IC50 > 10000 nM T13260 CMXA10 66575743 IC50 > 10000 nM T13260 CKWB91 66575744 IC50 > 10000 nM T13260 C7I3MW 66575745 IC50 > 10000 nM T13260 CPN17S 66575746 IC50 > 10000 nM T13260 CG0ZA7 66575747 IC50 > 10000 nM T13260 C6HF0U 66575748 IC50 > 10000 nM T13260 CDI93T 66575817 IC50 > 10000 nM T13260 CBP6I7 66576773 IC50 > 10000 nM T13260 C4NYB0 66576930 IC50 > 10000 nM T13260 C3LP5H 66576931 IC50 > 10000 nM T13260 CE03WG 66576932 IC50 > 10000 nM T13260 C9XYA1 67205290 Ki = 700 nM T13260 CO8IZ3 67854245 IC50 = 590 nM T13260 C2F5TS 68037237 Ki = 442 nM T13260 C97FZU 68561433 IC50 = 31 nM T13260 CK05PZ 68668617 Ki = 7 nM T13260 CC75HS 69198620 IC50 = 160000 nM T13260 CI6U5W 69649421 IC50 = 160 nM T13260 CZN04V 69828765 Ki = 45 nM T13260 CSUX85 70178310 Ki = 55 nM T13260 CBM80I 70354859 Ki = 77 nM T13260 COGQ93 70680979 IC50 = 30000 nM T13260 C96QKR 70683101 IC50 = 61000 nM T13260 CBNF56 70689398 IC50 = 20000 nM T13260 CPNR72 70689399 IC50 = 32000 nM T13260 CCG0U6 70691503 IC50 = 18000 nM T13260 CKE71B 70691504 IC50 = 11000 nM T13260 CA36IC 70695715 IC50 = 29000 nM T13260 CHEJ23 70748349 IC50 = 20900 nM T13260 C1VMF2 70977969 IC50 > 10000 nM T13260 CUV23H 71449132 Ki = 22 nM T13260 C37CSD 71450101 IC50 = 181.1 nM T13260 C7EDZ9 71452741 Ki = 753 nM T13260 CFKO73 71453732 IC50 = 2180 nM T13260 CI6B9U 71454429 IC50 > 50000 nM T13260 C70TUP 71455138 IC50 = 11 nM T13260 CH70RK 71456229 IC50 = 11000 nM T13260 CFG4L5 71456934 IC50 = 35 nM T13260 C8NPL7 71457257 IC50 = 83 nM T13260 CJCY84 71457258 IC50 = 20 nM T13260 C1KY3Q 71458062 Ki = 86 nM T13260 CK5TV7 71461661 Ki = 206 nM T13260 CI16NC 71520311 IC50 = 32 nM T13260 CE9A6B 71520312 IC50 = 246 nM T13260 C03VKJ 71520313 IC50 > 5000 nM T13260 C5J7DI 71520314 IC50 = 3340 nM T13260 CE0N5C 71520315 IC50 > 5000 nM T13260 C4Z6YP 71520316 IC50 = 565 nM T13260 CC8Z6L 71520431 IC50 > 5000 nM T13260 C1DK9P 71520432 IC50 = 1500 nM T13260 C9NOQ1 71521632 IC50 = 2130 nM T13260 C0OTA2 71521716 IC50 = 3660 nM T13260 CVLE07 71521717 IC50 > 5000 nM T13260 CJKX84 71521718 IC50 = 1350 nM T13260 CZ5P9U 71521719 IC50 = 140 nM T13260 C1YCB0 71521720 IC50 = 889 nM T13260 CE57PM 71521721 IC50 = 74 nM T13260 C0O2SA 71521798 IC50 = 81 nM T13260 CMEC10 71521799 IC50 = 59 nM T13260 CR9O5T 71521800 IC50 = 273 nM T13260 C0JBI3 71521801 IC50 = 74 nM T13260 CE7Z4I 71521802 IC50 = 116 nM T13260 CW2AG4 71521803 IC50 = 19 nM T13260 C6ID7K 71521804 IC50 = 55 nM T13260 CPZ5S8 71535400 IC50 = 790 nM T13260 CCRS95 71535683 IC50 = 2200 nM T13260 C9V7KW 71568307 IC50 = 9.01 nM T13260 CZGA56 71568308 IC50 = 148.93 nM T13260 C0E3WP 71568309 IC50 = 77.36 nM T13260 C3IX0R 71568310 IC50 = 4.93 nM T13260 C1B6UY 71568311 IC50 = 16.58 nM T13260 CF6DO2 71568312 IC50 = 21.39 nM T13260 CNBX98 71568313 IC50 = 164.01 nM T13260 CLD9N8 71568314 IC50 = 138.72 nM T13260 C7YVC9 71568442 IC50 = 56.83 nM T13260 C2ZS4G 71568443 IC50 = 27.01 nM T13260 C2BD6R 71568444 IC50 = 6.23 nM T13260 C03WJE 71568445 IC50 = 48.93 nM T13260 CXH93O 71568446 IC50 = 25.56 nM T13260 C0N6UG 71568447 IC50 = 46.92 nM T13260 C3PZG5 71568448 IC50 = 57.43 nM T13260 CPI06S 71568584 IC50 = 111.09 nM T13260 CL4YR2 71568585 IC50 = 203.34 nM T13260 C7ZCL4 71568586 IC50 = 235.33 nM T13260 CTQ79Z 71568587 IC50 = 217.43 nM T13260 C58SMB 71574941 IC50 = 480 nM T13260 CC09FQ 71574942 IC50 = 460 nM T13260 CA2T5L 71574943 IC50 = 300 nM T13260 C9MFZ7 71574944 IC50 = 1100 nM T13260 CW73OE 71574945 IC50 = 1973 nM T13260 C70NHJ 71574946 IC50 = 400 nM T13260 CLH83S 71574947 IC50 = 837 nM T13260 CF71AB 71575030 IC50 = 575 nM T13260 CCG1S5 71575031 IC50 = 565 nM T13260 CH9WE7 71575032 IC50 = 260 nM T13260 CO4ZQ7 71575033 IC50 = 170 nM T13260 CT86GV 71575034 IC50 = 6393 nM T13260 CHC8L4 71614085 IC50 = 0.2 nM T13260 CKPV51 71621803 IC50 > 100000 nM T13260 CG72JK 71681355 IC50 = 9257 nM T13260 C56LUJ 71716957 IC50 = 11160 nM T13260 CJE01S 71745100 IC50 > 10000 nM T13260 C54KVE 71748876 IC50 = 670 nM T13260 CT5Q9N 71812321 IC50 = 750 nM T13260 CBL42N 71812322 IC50 = 450 nM T13260 C9IOA1 71812324 Ki = 45 nM T13260 CX0WV5 71817943 IC50 > 2000 nM T13260 CN1LU6 71817944 IC50 > 2000 nM T13260 CGV4U3 71817945 IC50 > 2000 nM T13260 CJ4L5G 71818086 IC50 > 2000 nM T13260 COXA51 71818087 IC50 > 2000 nM T13260 CP1A3M 71818088 IC50 > 2000 nM T13260 CPJ42T 71818089 IC50 > 2000 nM T13260 CAP03I 71818090 IC50 > 2000 nM T13260 CO23PK 71818091 IC50 > 2000 nM T13260 CL4X6A 71818092 IC50 > 2000 nM T13260 CL8GK5 71818093 IC50 > 2000 nM T13260 C4ZVG0 71818094 IC50 > 2000 nM T13260 CH2GR0 71818232 IC50 > 2000 nM T13260 C0VGQ9 71818233 IC50 > 2000 nM T13260 C5QRF2 71818234 IC50 > 2000 nM T13260 C09VHD 72194216 IC50 = 5500 nM T13260 C4POE7 72546693 Ki = 80 nM T13260 CKI39Q 72546694 Ki = 20 nM T13260 C2SE6Q 72546935 Ki = 111 nM T13260 C49MBW 72546936 Ki = 160 nM T13260 CJCU54 72546937 Ki = 70 nM T13260 CN1Z5U 72546938 Ki = 20 nM T13260 CD6I2S 72546939 Ki = 330 nM T13260 CKE4O3 72546940 Ki = 170 nM T13260 CW5H8C 72546941 Ki = 820 nM T13260 C74PHD 72547200 Ki = 200 nM T13260 CDC4P8 72547201 Ki = 130 nM T13260 CZNW37 72547202 Ki = 841 nM T13260 CFLU42 72547203 Ki = 110 nM T13260 C76AZT 72547204 Ki = 90 nM T13260 C1IP7G 72547205 Ki = 237 nM T13260 C62CNP 72547206 Ki = 350 nM T13260 CG0LT8 72547452 Ki = 647 nM T13260 CU76NM 72703468 IC50 > 10000 nM T13260 C9PRT7 72703681 IC50 > 10000 nM T13260 CCG7R3 72703685 IC50 = 5.3 nM T13260 CU27CK 72703887 IC50 > 10000 nM T13260 CFR2V8 72703888 IC50 > 10000 nM T13260 CAU4Z0 72703889 IC50 = 3.1 nM T13260 C56KEC 72703890 IC50 = 13.3 nM T13260 CB7PR0 72704087 IC50 = 1472 nM T13260 C5SNU6 72708597 IC50 = 3200 nM T13260 CSB7R2 73055580 IC50 = 15000 nM T13260 CG37VI 73055876 IC50 = 20000 nM T13260 CU5DC1 73055877 IC50 = 190000 nM T13260 C5M7RH 73055879 IC50 = 2500 nM T13260 C53JKM 73055880 IC50 = 67100 nM T13260 CR8V7S 73055881 IC50 = 800 nM T13260 C72LFY 73346265 IC50 = 2700 nM T13260 C5F2VZ 73347760 IC50 = 3400 nM T13260 C5QTA7 73349312 IC50 = 3400 nM T13260 CPU7N5 73350879 IC50 = 12500 nM T13260 CT1J5B 73350882 IC50 = 12500 nM T13260 C9Y5FN 73353441 IC50 = 9257 nM T13260 CT9SN8 73353827 IC50 = 4600 nM T13260 CD13BV 73353828 IC50 = 8000 nM T13260 CGWY15 73355361 IC50 = 1800 nM T13260 C1YT7X 73355362 IC50 = 9400 nM T13260 CKEY08 73355363 IC50 = 7900 nM T13260 CGF87Z 73355403 IC50 = 3900 nM T13260 C0OY5P 73356914 IC50 = 1300 nM T13260 CX12ML 73356915 IC50 = 2900 nM T13260 C0UQ3M 73356955 IC50 = 29100 nM T13260 CKG8J2 73357190 IC50 = 590 nM T13260 C9WY3B 73386689 IC50 = 45 nM T13260 CK4NQ1 76186646 IC50 = 0.9 nM T13260 CM52SI 76308995 IC50 = 11900 nM T13260 CS80JY 76310075 IC50 = 50 nM T13260 CB1V2S 76311295 IC50 = 10700 nM T13260 C7XH3E 76314886 IC50 = 80 nM T13260 CPU3T6 76317295 IC50 = 1100 nM T13260 CAM49B 76318503 IC50 = 90 nM T13260 CFJ8G5 76322165 IC50 = 40 nM T13260 C7KEG3 76322166 IC50 = 150 nM T13260 CHBR20 76325787 IC50 = 1010 nM T13260 CXD53T 76327865 IC50 = 160 nM T13260 CS8D4U 76328231 IC50 = 3000 nM T13260 C3F0JZ 76329384 IC50 > 300000 nM T13260 C3JID2 76331906 IC50 = 650 nM T13260 C1YJW0 77846787 IC50 = 790 nM T13260 CV73PD 77846790 IC50 = 10000 nM T13260 C0DIH7 77846872 IC50 = 10000 nM T13260 COI25M 77846873 IC50 = 1000 nM T13260 CJI8R0 77846875 IC50 = 3800 nM T13260 CZK4J1 77846962 IC50 = 2800 nM T13260 CEK89G 77846963 IC50 = 10000 nM T13260 C5BA8Z 77846964 IC50 = 1240 nM T13260 C4D6XJ 77847803 IC50 = 1600 nM T13260 CF7O4Q 77847804 IC50 = 1200 nM T13260 CEC49D 85863219 IC50 = 1610 nM T13260 CZ5PM0 86277538 IC50 = 0.42 nM T13260 CHV8R6 86307678 IC50 = 620 nM T13260 C3X6MJ 86792466 IC50 = 21700 nM T13260 CL30TR 89471870 IC50 = 2300 nM T13260 C3BUS8 89471889 IC50 = 420 nM T13260 CI7HY8 89471890 IC50 = 120 nM T13260 CX0M7B 89961716 IC50 = 21 nM T13260 CR5D6Y 89961785 IC50 > 10000 nM T13260 C89TEU 89968659 IC50 > 10000 nM T13260 CY5IC7 90252834 IC50 = 4600 nM T13260 C84NVA 90252850 IC50 = 6300 nM T13260 CBY46O 90252851 IC50 = 5400 nM T13260 CNVA50 90252852 IC50 = 6200 nM T13260 C89BFG 90333640 IC50 = 1820 nM T13260 CJ8NI5 90655716 Ki = 57 nM T13260 COF02L 90655717 Ki = 62 nM T13260 CO9K2W 90655718 Ki = 31 nM T13260 CX8L7D 90655719 Ki = 69 nM T13260 CHD21I 90666137 IC50 = 14.4 nM T13260 C4A7JU 90677206 IC50 = 12500 nM T13260 C3T5BI 90677209 IC50 = 12500 nM T13260 CV96EW 90677213 IC50 = 12500 nM T13260 C3Y8AQ 90677215 IC50 = 12500 nM T13260 C6PJL5 90677216 IC50 = 12500 nM T13260 CFI3J8 90677218 IC50 = 12500 nM T13260 CQ91ZO 90677219 IC50 = 12500 nM T13260 CQS8C9 91664365 IC50 = 1000 nM T13260 CM9U7B 91758284 Ki = 20 nM T13260 CLB2E7 91827654 IC50 > 30000 nM T13260 C0KDB6 91983064 Ki = 32 nM T13260 CYL1S3 97191385 IC50 = 5100 nM T13260 CXRB41 101152219 IC50 > 10000 nM T13260 C3P9ZY 101199629 IC50 = 41 nM T13260 CL3UQ9 101354484 Ki = 10 nM T13260 C26AKT 101354485 Ki = 14 nM T13260 CZXS85 101354486 Ki = 81 nM T13260 CWXT16 101378163 Ki = 45 nM T13260 C8VZC7 101378164 Ki = 45 nM T13260 C4G5MB 101378165 Ki = 670 nM T13260 C5HLB7 101378166 Ki = 670 nM T13260 C0TOW6 101433013 Ki = 8.2 nM T13260 CLI59T 101579737 IC50 = 160 nM T13260 C18UTF 101587707 Ki = 150 nM T13260 C2SUC3 101587708 Ki = 1180 nM T13260 CI0N8C 101592374 Ki = 24.1 nM T13260 CV87DF 101592375 Ki = 24.1 nM T13260 C1ZN6O 101592376 Ki = 24.1 nM T13260 C5WGQ7 101620856 Ki = 5000 nM T13260 CC01NA 101650066 Ki = 12 nM T13260 CE9T0K 101650068 Ki = 12 nM T13260 CUDV46 101650069 Ki = 12 nM T13260 CBN09G 101651130 Ki = 2 nM T13260 C9CZN6 101668720 Ki = 11100 nM T13260 C9TID7 101701780 Ki = 5000 nM T13260 C0RN1M 101927481 Ki = 25 nM T13260 C9E7GV 102068512 Ki = 7 nM T13260 C63RAU 102068514 Ki = 7 nM T13260 C8YJK2 102068516 Ki = 7 nM T13260 C57AZV 102068518 Ki = 7 nM T13260 C4J1SX 102279741 Ki = 95 nM T13260 CE90MX 102346108 IC50 = 6870 nM T13260 CED87Z 102439715 Ki = 5000 nM T13260 C0DYC5 102532604 Ki = 5000 nM T13260 C9KZ5G 102533756 Ki = 16 nM T13260 CB1Z8U 102533759 Ki = 16 nM T13260 CMO84S 110730849 IC50 = 490 nM T13260 CJ9Z0S 118496546 IC50 = 6900 nM T13260 C2BMT8 118708021 IC50 = 34400 nM T13260 C8NES2 118711691 Ki = 630.96 nM T13260 CKT4A8 118711692 Ki = 707.95 nM T13260 COD91Y 118711693 Ki = 707.95 nM T13260 CGJ93V 118711694 Ki = 25.12 nM T13260 C0WLI2 118711695 Ki = 354.81 nM T13260 CXDE52 118711696 Ki = 144.54 nM T13260 CAW5K3 118723935 IC50 = 549 nM T13260 CK8UL1 118723936 IC50 = 387 nM T13260 CIW7O0 118723937 IC50 = 477 nM T13260 C42CEZ 118723938 IC50 = 584 nM T13260 CJQ63E 118723939 IC50 = 639 nM T13260 CCXN71 118723940 IC50 = 445 nM T13260 CS78BD 118723941 IC50 = 349 nM T13260 C9W3QX 118723942 IC50 = 17464 nM T13260 COJ2K8 118723943 IC50 = 5855 nM T13260 CZ23UL 118723944 IC50 = 3708 nM T13260 CIWU64 118723945 IC50 = 4566 nM T13260 CZI6A0 118723946 IC50 = 8299 nM T13260 COB46M 118723947 IC50 = 31813 nM T13260 CJ1HP9 118728223 Ki = 10000 nM T13260 CZR62N 118730170 IC50 = 810 nM T13260 CDHI10 118733086 IC50 > 10000 nM T13260 C18PWB 118733087 IC50 > 10000 nM T13260 C8WJ2Y 118733088 IC50 > 10000 nM T13260 C31ZXP 118733089 IC50 > 10000 nM T13260 CHR84E 118733090 IC50 > 10000 nM T13260 CAQ72M 118733091 IC50 > 10000 nM T13260 CIV1Z5 118733092 IC50 > 10000 nM T13260 CU3Y9W 118733093 IC50 > 10000 nM T13260 CF49NU 118733094 IC50 > 10000 nM T13260 CK73VU 118733095 IC50 > 10000 nM T13260 CR1WU5 118733096 IC50 > 10000 nM T13260 C5C4FZ 118735165 IC50 = 447 nM T13260 C1ZLM6 118735166 IC50 = 146 nM T13260 CQXM57 118735167 IC50 = 75 nM T13260 C0RYM4 118735168 IC50 = 137 nM T13260 C0DCB9 118735169 IC50 = 2425 nM T13260 CG4QF3 118735170 IC50 = 1894 nM T13260 CD3IY5 118735171 IC50 = 4993 nM T13260 C2VJU4 118735179 IC50 = 2090 nM T13260 CXWH51 118735180 IC50 = 165 nM T13260 C3YUS9 118735181 IC50 = 1546 nM T13260 CZET62 118735186 IC50 = 128 nM T13260 CZ8U2C 118735187 IC50 = 157 nM T13260 COJ81W 118735362 IC50 = 1020 nM T13260 C8VFT2 118735363 IC50 = 1320 nM T13260 CZE92I 118735364 IC50 = 53.1 nM T13260 CFB1G7 118735365 IC50 = 48.1 nM T13260 CX4V1E 118735366 IC50 = 6290 nM T13260 CW60ZD 118735367 IC50 = 337 nM T13260 C6ULM1 118735368 IC50 = 143 nM T13260 CE50LC 118735369 IC50 = 261 nM T13260 CMCW85 118735370 IC50 = 328 nM T13260 C6Y2NQ 118735371 IC50 = 1930 nM T13260 CVEQ39 118735372 IC50 = 48.9 nM T13260 C4LK0C 118735373 IC50 = 16.9 nM T13260 C93CNO 118735374 IC50 = 174 nM T13260 C4YR6E 118735375 IC50 = 715 nM T13260 CS3ZJ8 118735376 IC50 = 699 nM T13260 CV83KA 118735377 IC50 = 493 nM T13260 C0BP6M 118735378 IC50 = 30500 nM T13260 CG9RB4 118735379 IC50 = 1240 nM T13260 CGT60X 118735380 IC50 = 7340 nM T13260 CY6L8W 118735381 IC50 = 491 nM T13260 C3NB6I 122181247 IC50 = 12500 nM T13260 CYCG69 122181248 IC50 = 200 nM T13260 CME27L 122181249 IC50 = 1800 nM T13260 C0KHC3 122191579 IC50 = 0.26 nM T13260 CO7E3N 122191580 IC50 = 0.42 nM T13260 CML6C5 122191581 IC50 = 5.2 nM T13260 CYC63O 122191582 IC50 = 2.7 nM T13260 CP7S0B 122191583 IC50 = 2.3 nM T13260 C61IRT 122191584 IC50 = 4 nM T13260 CYJ32S 122191585 IC50 = 2.3 nM T13260 CAQ5S2 122191586 IC50 = 3.5 nM T13260 C03SBU 122191587 IC50 = 4.2 nM T13260 CLG6J4 122191588 IC50 = 5 nM T13260 CI42KY 122191589 IC50 = 20.7 nM T13260 C9GQP6 122191591 IC50 = 3.4 nM T13260 C0WN2U 122191592 IC50 = 5.5 nM T13260 C0WI6K 122191772 IC50 = 29 nM T13260 C5C2EM 122192355 IC50 = 250 nM T13260 C4HIF8 122192356 IC50 = 220 nM T13260 C0SJU6 122192359 IC50 = 100 nM T13260 C3T9CZ 122192360 IC50 = 41 nM T13260 C58OCL 122192361 IC50 = 0.1 nM T13260 C15NCI 122439267 IC50 = 10000 nM T13260 CX4T7L 122439274 IC50 = 10000 nM T13260 C3YG1J 122443028 IC50 > 19952.62 nM T13260 CW3K8X 122462796 IC50 > 19952.62 nM T13260 C80OLS 122462854 IC50 > 31622.78 nM T13260 CR4YC2 124012328 Ki = 38 nM T13260 C10TQU 124351848 Ki = 1 nM T13260 CCX94N 124351849 Ki = 75 nM T13260 C36AXJ 127025738 Ki = 100 nM T13260 CM2NC0 127025739 Ki = 100 nM T13260 CW5AZ0 127025740 Ki = 100 nM T13260 CY9Q8T 127025741 Ki = 100 nM T13260 C0X8HP 127026020 Ki = 24.1 nM T13260 C4LWG3 127026653 IC50 = 120500 nM T13260 C3ZQ5Y 127026654 IC50 = 1889 nM T13260 CZDU19 127026655 IC50 = 18570 nM T13260 CIT8S3 127026966 IC50 = 1820 nM T13260 CJTB10 127026967 IC50 = 1820 nM T13260 C2ZFR8 127027572 IC50 = 7900 nM T13260 CV1BD6 127027573 IC50 = 3100 nM T13260 C1L9TB 127027959 IC50 = 26000 nM T13260 CPX6K3 127028274 Ki = 100 nM T13260 CQO36B 127028499 IC50 = 5000 nM T13260 CCR07G 127028593 IC50 = 1820 nM T13260 CH6PU4 127028608 Ki = 100 nM T13260 C9WIB4 127028609 Ki = 100 nM T13260 CN42BR 127028817 IC50 > 10000 nM T13260 CIE4Q7 127028911 IC50 = 1820 nM T13260 C49IME 127031799 IC50 = 6100 nM T13260 CGEO60 127035149 IC50 = 245 nM T13260 CJ30BZ 127035150 IC50 = 236 nM T13260 C3MN9I 127035661 Ki = 5 nM T13260 CX3TB1 127035807 Ki = 5 nM T13260 CE6T8A 127035808 Ki = 5 nM T13260 C7JNM3 127036045 Ki = 75000 nM T13260 CS72ZI 127036174 Ki = 100 nM T13260 C9AFT8 127036253 IC50 = 6400 nM T13260 CQS2U0 127036843 IC50 = 2800 nM T13260 C7SM8Y 127037253 Ki = 31 nM T13260 CW08IP 127037254 IC50 = 1700 nM T13260 CXWJ74 127037557 Ki = 36 nM T13260 CK5N0X 127037559 Ki = 10000 nM T13260 CMQD16 127037560 Ki = 10000 nM T13260 CI6S7D 127037561 Ki = 10000 nM T13260 CTE51A 127047976 IC50 = 110 nM T13260 C1IBC5 127048009 IC50 = 530 nM T13260 CWE96C 127048149 IC50 = 12310 nM T13260 CDX0L1 127048499 IC50 = 51 nM T13260 CWD0J9 127048833 IC50 = 7 nM T13260 C9OEW2 127048838 IC50 = 46 nM T13260 CCJ3F0 127048839 IC50 = 6 nM T13260 CQ10PX 127048840 IC50 = 42 nM T13260 CWAH54 127048841 IC50 = 48 nM T13260 CD2O0K 127049168 IC50 = 129 nM T13260 C7ZHU6 127049169 IC50 = 48 nM T13260 CQN95D 127049828 IC50 = 36 nM T13260 C20LNJ 127050749 IC50 = 43 nM T13260 CH6E4C 127050950 IC50 = 168 nM T13260 CQ8PA9 127050951 IC50 = 512 nM T13260 C4Q6RA 127050952 IC50 = 800 nM T13260 C92CDW 127051351 IC50 = 14 nM T13260 CCR94D 127051352 IC50 = 13 nM T13260 CPL7A6 127051353 IC50 = 54 nM T13260 C7T2JR 127051680 IC50 = 339 nM T13260 CEJ1B8 127051681 IC50 = 131 nM T13260 CW3B0L 127051682 IC50 = 79 nM T13260 CE04JD 127052583 IC50 = 16 nM T13260 C48EUT 127052584 IC50 = 45 nM T13260 CT73HY 127052585 IC50 = 21 nM T13260 CL4ZK7 127052586 IC50 = 59 nM T13260 C1EI2R 127052880 IC50 = 22 nM T13260 CU9FI0 127052881 IC50 = 14 nM T13260 C01SHM 127052902 IC50 = 53 nM T13260 C09AZE 127052903 IC50 = 24 nM T13260 CH85FP 127052904 IC50 = 14 nM T13260 CYVM52 127052905 IC50 = 9 nM T13260 C12WOQ 129137247 IC50 = 62.2 nM T13260 C4O3QV 129137260 IC50 = 177.1 nM T13260 CJB4M3 129137266 IC50 = 230 nM T13260 CWVE96 129137276 IC50 = 13.4 nM T13260 CJ1N2M 129137280 IC50 = 220.8 nM T13260 CH42QX 129137285 IC50 = 8.8 nM T13260 CEH4N6 129750903 IC50 = 2600 nM T13260 CD7BX2 132601756 IC50 = 57.54 nM T13260 C5XSM4 132601757 IC50 = 12.11 nM T13260 CC2X1M 132601758 IC50 = 9.016 nM T13260 C8U1VZ 132601759 IC50 = 17.38 nM T13260 CH3V9Q 134139925 IC50 = 7700 nM T13260 CZV71F 134140768 IC50 = 6070 nM T13260 CVS3Q5 134142034 IC50 = 9724 nM T13260 CK4GS1 134142054 IC50 = 4660 nM T13260 C4B3MJ 134142750 IC50 = 9520 nM T13260 C2PT7N 134146686 IC50 = 12530 nM T13260 CK1BE9 134155077 IC50 = 286.9 nM T13260 C8QEA7 134155257 IC50 = 5089 nM T13260 C2BK3Z 134155779 IC50 = 645.3 nM T13260 C6G1CH 135185858 IC50 = 6445 nM T13260 CVR24H 135461648 IC50 = 29800 nM T13260 COWK61 135926058 IC50 > 50000 nM T13260 C7MP6W 135967555 Ki = 2548 nM T13260 CAV9U3 136219390 IC50 = 11.4 nM T13260 C59TUZ 136239410 IC50 > 10000 nM T13260 CH0O1B 136239411 IC50 > 10000 nM T13260 C52CVP 136239516 IC50 = 4152 nM T13260 CC7LY3 136239517 IC50 = 454 nM T13260 CSQR53 136239518 IC50 = 2112 nM T13260 C1N2WP 136244527 IC50 = 6195 nM T13260 C2V0IM 136244612 IC50 = 6 nM T13260 CLU5W1 136244613 IC50 = 922 nM T13260 C5LFY4 136245940 IC50 > 10000 nM T13260 CF07BL 136245941 IC50 > 10000 nM T13260 CYIF59 136245971 IC50 > 10000 nM T13260 CM6GS7 137632939 IC50 = 8900 nM T13260 CD7J1Z 137635610 IC50 = 5670 nM T13260 C4FYB7 137650013 IC50 = 9670 nM T13260 C2OC5D 137660208 IC50 = 6700 nM T13260 C3UK1Z 137660483 IC50 > 10000 nM T13260 C6VX2G 137662301 IC50 = 30.3 nM T13260 CEG7C9 140993853 IC50 = 1092.68 nM T13260 CY9QN0 145949171 IC50 = 2700 nM T13260 C0R6GF 145949298 IC50 = 237.6 nM T13260 C51BOX 145949540 IC50 = 700 nM T13260 C8T1HG 145949588 IC50 = 677.4 nM T13260 CBR4W8 145950208 IC50 = 2700 nM T13260 CVIW14 145950556 IC50 = 2800 nM T13260 C3L5IO 145950622 IC50 = 2300 nM T13260 C2EN9P 145950803 IC50 = 2500 nM T13260 CH80BF 145951156 IC50 = 32.3 nM T13260 CE8S3P 145951478 IC50 = 11900 nM T13260 CF2JT9 145951520 IC50 = 51.2 nM T13260 CD9G1O 145951806 IC50 = 2635 nM T13260 CL7V8M 145952266 IC50 = 11200 nM T13260 C9J0MP 145952426 IC50 = 1058 nM T13260 C4RX0H 145952545 IC50 = 276.8 nM T13260 CAD1R5 145953186 IC50 = 82.9 nM T13260 CGTW16 145953426 IC50 = 9800 nM T13260 C3PG4W 145953645 IC50 = 9800 nM T13260 CCF34U 145954042 IC50 = 8300 nM T13260 C8AR7H 145954077 IC50 = 5500 nM T13260 C5J7MO 145954302 IC50 = 4400 nM T13260 C6LU3T 145954433 IC50 = 7600 nM T13260 CRZ51Q 145954497 IC50 = 217.4 nM T13260 CEU5V2 145955100 IC50 = 4200 nM T13260 CGH62B 145955360 IC50 = 3900 nM T13260 CV49CR 145955375 IC50 = 11900 nM T13260 CYZ7R9 145955426 IC50 = 1400 nM T13260 C04FSJ 145955438 IC50 = 4600 nM T13260 CV5CZ7 145955551 IC50 = 207.5 nM T13260 CO3P9B 145955618 IC50 = 1300 nM T13260 CPS1E4 145956015 IC50 = 14.1 nM T13260 CCVP89 145956394 IC50 = 108.7 nM T13260 CR79QW 145956423 IC50 = 3400 nM T13260 CH8KZ4 145956588 IC50 = 260.8 nM T13260 CF4X3A 145956605 IC50 = 5400 nM T13260 CP65IV 145957520 IC50 = 8800 nM T13260 C7VQ6H 145958289 IC50 = 3500 nM T13260 CW8K2X 145958349 IC50 = 196.5 nM T13260 C8COZ7 145958369 IC50 = 4000 nM T13260 CC7UM6 145958531 IC50 = 36.1 nM T13260 C7TS3W 145958716 IC50 = 7772 nM T13260 C1FBC3 145958737 IC50 = 58.3 nM T13260 C0X5WO 145958928 IC50 = 96.9 nM T13260 C5IEV3 145958952 IC50 = 800 nM T13260 CTGM23 145959211 IC50 = 2300 nM T13260 CV1N0L 145959349 IC50 = 3800 nM T13260 C62HPO 145959622 IC50 = 2800 nM T13260 C4NYX7 145959688 IC50 = 210.6 nM T13260 CCW9R3 145959703 IC50 = 4100 nM T13260 C90VNG 145960023 IC50 = 3200 nM T13260 C7HA8N 145960331 IC50 = 3500 nM T13260 CK71RV 145963932 IC50 > 31622.78 nM T13260 C79FGQ 145965325 IC50 > 31622.78 nM T13260 CI56TJ 145967693 IC50 = 935.46 nM T13260 CKWV62 145967722 IC50 = 3591.14 nM T13260 C7XT0Z 145967929 IC50 = 3482.15 nM T13260 CHA9G8 145967940 IC50 = 3045.68 nM T13260 C0HP1U 145968036 IC50 = 2600.71 nM T13260 C5BM1L 145968186 IC50 = 999.74 nM T13260 C8XB7E 145968768 IC50 = 3253.28 nM T13260 C4JM2H 145968847 IC50 = 5715.79 nM T13260 C74IZW 145969198 IC50 = 3187.68 nM T13260 CNV0K1 145969871 IC50 = 1181.36 nM T13260 C4MQL6 145970012 IC50 = 1984.4 nM T13260 CDZV35 145970043 IC50 = 176.82 nM T13260 CEKI13 145970456 IC50 = 3321.79 nM T13260 C2Q1CO 145970604 IC50 = 1804.56 nM T13260 CW7XA4 145970723 IC50 = 3565.19 nM T13260 CE6P4U 145971254 IC50 = 1700 nM T13260 CGBW36 145972890 IC50 = 15300 nM T13260 CR50XP 145974563 IC50 = 54.4 nM T13260 CTB32X 145987737 IC50 = 3000.88 nM T13260 CJQ23A 145988166 IC50 = 3345.23 nM T13260 CAS5W8 145988425 IC50 = 3409.25 nM T13260 CZBY26 145988625 IC50 = 1703.22 nM T13260 C8I5JY 155511774 IC50 = 3200 nM T13260 C8ZYW2 155512683 Ki = 100 nM T13260 CWL61G 155513859 IC50 = 2750 nM T13260 COUZ40 155515111 Ki = 8 nM T13260 CQ0RX1 155519734 IC50 = 3300 nM T13260 CN8R0W 155521581 IC50 = 405 nM T13260 CS79RV 155522275 Ki = 24 nM T13260 CX9CY6 155523438 Ki = 97 nM T13260 C42DVB 155524075 Ki = 450 nM T13260 C7DX4M 155524253 IC50 = 110 nM T13260 CZCD39 155524316 Ki = 180 nM T13260 CO73MH 155528129 IC50 = 175 nM T13260 C9KHR3 155528792 IC50 = 210 nM T13260 C3PKZ1 155531378 IC50 = 0.2 nM T13260 CE2F1S 155532984 Ki = 81 nM T13260 C65EOC 155533109 Ki = 74 nM T13260 C2YTO1 155533392 IC50 = 520 nM T13260 C57SRY 155539404 IC50 = 105 nM T13260 CA01UF 155542148 IC50 = 210 nM T13260 C05WZC 155544203 Ki = 79 nM T13260 C1CJ3W 155544206 IC50 = 43.55 nM T13260 CZ48QO 155544544 IC50 = 660 nM T13260 C8NOR7 155548567 IC50 = 39.77 nM T13260 CO2G9W 155552576 IC50 = 73.17 nM T13260 C5CKA6 155553716 IC50 = 90.73 nM T13260 CAK73M 155557092 IC50 = 430 nM T13260 CA2H5K 155557102 IC50 = 17.42 nM T13260 C04ZVY 155557805 IC50 > 12500 nM T13260 CAY1Z7 155558257 IC50 = 14.52 nM T13260 CH3N8S 155558347 IC50 = 280 nM T13260 CJX17H 155558789 Ki = 57 nM T13260 CO6W0R 155559106 Ki = 125 nM T13260 C47PER 155559543 IC50 = 19.66 nM T13260 CH3IK5 155559681 IC50 = 8720 nM T13260 C3SWX8 155559867 IC50 = 58.85 nM T13260 CXT67R 155559873 IC50 = 560 nM T13260 CQU6N2 155562191 Ki = 290 nM T13260 C20AJK 155564333 IC50 = 55 nM T13260 CZ1OQ8 155569008 IC50 = 30.19 nM T13260 CH20CY 3114838 IC50 = 441 nM T13260 D00BVP 11847320 IC50 = 79.43 nM T13260 D00EMF 3644637 IC50 > 100000 nM T13260 D00HVZ 5271544 IC50 = 1860 nM T13260 D00RIX 5280443 IC50 = 1000 nM T13260 D00TWK 185914 IC50 > 50000 nM T13260 D00VUO 6539777 IC50 = 6360 nM T13260 D00ZPJ 408350 Ki = 25.5 nM T13260 D01IJX 10537337 IC50 = 3560 nM T13260 D01JZO 2779191 IC50 = 70 nM T13260 D01KKU 5281894 IC50 = 30.5 nM T13260 D01LOU 2238 IC50 = 40 nM T13260 D01MPK 12331302 Ki = 1750 nM T13260 D01REI 46901610 IC50 = 2440 nM T13260 D01SUE 6539759 IC50 = 2040 nM T13260 D01SZX 46867545 IC50 = 150 nM T13260 D01UYI 5281607 IC50 = 1 nM T13260 D02ALK 11514074 IC50 = 2700 nM T13260 D02BGR 9949648 IC50 = 13000 nM T13260 D02BWQ 6539818 IC50 = 2800 nM T13260 D02BXS 46901445 IC50 = 24560 nM T13260 D02CSU 6539786 IC50 = 12735030.81 nM T13260 D02LTV 10019821 IC50 = 110 nM T13260 D02LWB 6540046 IC50 > 36000 nM T13260 D02NAG 6539765 IC50 = 4260 nM T13260 D02QSH 339914 Ki = 1.9 nM T13260 D02SIT 9926623 IC50 = 74 nM T13260 D02XHH 6540043 IC50 = 100 nM T13260 D02XTS 6539811 IC50 = 3630 nM T13260 D03EXD 49864181 IC50 = 3070 nM T13260 D03FBI 49798900 IC50 = 8510 nM T13260 D03KLN 11413434 IC50 = 129 nM T13260 D03LOG 5280450 IC50 = 48000 nM T13260 D03MKT 6539788 IC50 = 1550 nM T13260 D03TRM 6540032 IC50 = 955 nM T13260 D03VRC 2989557 IC50 = 338.84 nM T13260 D04CLL 6539775 IC50 = 4720 nM T13260 D04DZZ 11646165 IC50 = 910 nM T13260 D04ELJ 6539766 IC50 = 4050 nM T13260 D04HVL 364705 IC50 = 2790 nM T13260 D04IBH 11616637 IC50 = 9107 nM T13260 D04IJE 256445 IC50 = 2741574.17 nM T13260 D04ISG 11680597 IC50 > 2000 nM T13260 D04LWL 97252 IC50 > 115600 nM T13260 D04QPK 6539783 IC50 = 1810 nM T13260 D04REX 6539808 IC50 = 790 nM T13260 D04TBB 10354739 IC50 = 2 nM T13260 D04VRY 11847169 IC50 = 467.74 nM T13260 D04WJN 10588478 IC50 = 389.05 nM T13260 D04ZGF 10561174 IC50 = 500 nM T13260 D05FFY 14231155 IC50 = 15 nM T13260 D05HBF 5353357 IC50 = 8.7 nM T13260 D05HRP 13596072 Ki = 800 nM T13260 D05IWY 5464078 IC50 = 4970 nM T13260 D05MQE 6539785 IC50 = 230 nM T13260 D05PXK 11847171 IC50 = 1800 nM T13260 D05QPR 12229388 IC50 = 880 nM T13260 D05YCI 42618032 IC50 = 18470 nM T13260 D05YJR 5495926 IC50 = 5200 nM T13260 D05YNW 6539790 IC50 = 6700 nM T13260 D05ZPO 1890 IC50 = 3800 nM T13260 D06AZC 135494055 IC50 = 1400 nM T13260 D06DDT 5315502 IC50 = 30000 nM T13260 D06FHE 44341253 IC50 = 205 nM T13260 D06GIV 337660 IC50 = 3100 nM T13260 D06HFV 6539805 IC50 = 7447319.74 nM T13260 D06HJB 14355826 IC50 = 55 nM T13260 D06PRC 5281650 IC50 = 20700 nM T13260 D06UQR 15306616 IC50 = 14800 nM T13260 D06WPP 11847170 IC50 = 4073.8 nM T13260 D07CTI 10853186 IC50 = 977.24 nM T13260 D07FGX 6116651 IC50 = 3300 nM T13260 D07IQG 10473365 IC50 = 933.25 nM T13260 D07JKK 11760063 IC50 = 1 nM T13260 D07LUJ 64945 IC50 = 14 ug.mL-1 T13260 D07PHT 324288 Ki = 6.5 nM T13260 D07PHV 10546089 IC50 = 89 nM T13260 D07PYC 6539760 IC50 = 3550 nM T13260 D07SOM 11847316 IC50 = 71 nM T13260 D07TIJ 3828439 IC50 = 2818.38 nM T13260 D07TUX 11230598 IC50 = 31622.78 nM T13260 D07UVN 6440384 IC50 = 3080 nM T13260 D07ZCD 6539804 IC50 = 1710 nM T13260 D07ZYL 6539797 IC50 = 3720 nM T13260 D08ARY 339906 Ki = 5.6 nM T13260 D08AZK 6539767 IC50 = 7830 nM T13260 D08EZA 11847317 IC50 = 45 nM T13260 D08FAB 11845485 IC50 > 2000 nM T13260 D08FHU 42618033 IC50 = 2720 nM T13260 D08FOJ 9898204 IC50 = 4300 nM T13260 D08HPU 6540052 IC50 = 1787 nM T13260 D08IIW 46887422 IC50 = 40 nM T13260 D08ISK 42618030 IC50 > 91290 nM T13260 D08KLN 13580711 IC50 = 3210 nM T13260 D08PKR 10845522 IC50 = 3060 nM T13260 D08PNF 6539770 IC50 = 5570 nM T13260 D08TKB 46889432 IC50 = 389.2 nM T13260 D08UQH 53600 IC50 = 190 nM T13260 D08ZTZ 11529133 IC50 = 1805 nM T13260 D09CPC 13728862 IC50 > 5000 nM T13260 D09DRS 42618031 IC50 = 960 nM T13260 D09HEA 1236449 IC50 = 1096.48 nM T13260 D09HGK 6539796 IC50 = 3960 nM T13260 D09HOE 6539789 IC50 = 800 nM T13260 D09HQH 13308 Ki = 260 nM T13260 D09MQF 15696376 IC50 = 900 nM T13260 D09MYQ 261365 Ki = 266 nM T13260 D09OPA 44593508 IC50 = 3400 nM T13260 D09QDY 6540033 IC50 = 130 nM T13260 D09TUB 11099375 IC50 > 308300 nM T13260 D09VPA 6539794 IC50 = 3400 nM T13260 D09VQM 442428 IC50 = 5000 nM T13260 D09XKH 10356745 IC50 = 2200 nM T13260 D09YXV 6539769 IC50 = 4310 nM T13260 D09ZHX 11847318 IC50 = 436.52 nM T13260 D09ZIW 10143276 IC50 = 7100 nM T13260 D0A0JL 2052 IC50 = 70600 nM T13260 D0A2FO 2825024 IC50 = 8000 nM T13260 D0A2GB 13660221 IC50 = 1300 nM T13260 D0A4EA 445639 IC50 = 32700 nM T13260 D0A4XA 25093379 IC50 > 50000 nM T13260 D0A7PA 49799639 IC50 = 11140 nM T13260 D0AH1B 6539782 IC50 = 12618275.35 nM T13260 D0AM2Z 13660216 IC50 = 11000 nM T13260 D0AW7Q 46867544 IC50 = 7900 nM T13260 D0AY4E 6539780 IC50 = 3930 nM T13260 D0B5MZ 13660218 IC50 = 2300 nM T13260 D0B8PE 10355761 IC50 = 3500 nM T13260 D0BH2T 10107266 IC50 > 40 ug.mL-1 T13260 D0C3XU 46887018 IC50 = 7 nM T13260 D0C5SV 5280934 IC50 = 44200 nM T13260 D0C5ZP 16125122 IC50 = 2140 nM T13260 D0C8EO 6539806 IC50 = 4330 nM T13260 D0C8KC 1504717 IC50 = 960 nM T13260 D0CR6B 11847319 IC50 = 69 nM T13260 D0D0DR 10081625 IC50 = 310 nM T13260 D0D7GG 510040 IC50 = 950 nM T13260 D0D8GU 6539803 IC50 = 1280 nM T13260 D0D8YE 6540048 IC50 = 5700 nM T13260 D0D9FR 6539795 IC50 = 3962780.34 nM T13260 D0DJ3R 10585323 IC50 = 100 nM T13260 D0DO1T 9819080 Ki = 10.3 nM T13260 D0DY5G 443389 IC50 > 100000 nM T13260 D0E2RV 360578 IC50 = 1700 nM T13260 D0E3IK 11680642 IC50 = 2510 nM T13260 D0E5FV 5318585 IC50 = 100 nM T13260 D0E9WX 6540042 IC50 = 27 nM T13260 D0F4MF 49799640 IC50 = 980 nM T13260 D0F4WQ 46867547 IC50 = 5.59 nM T13260 D0F5AC 46867542 IC50 = 17 nM T13260 D0F5YU 6539793 IC50 = 1990 nM T13260 D0F8IB 25256842 IC50 = 16500 nM T13260 D0F9MQ 11493409 IC50 = 2670 nM T13260 D0G2JV 49799657 IC50 = 2280 nM T13260 D0G6QL 23644748 IC50 = 2800 nM T13260 D0GL0L 11232117 IC50 = 3981.07 nM T13260 D0H1LK 161760 IC50 = 10200 nM T13260 D0HC9U 46867416 IC50 = 53 nM T13260 D0HD9P 444899 IC50 = 28200 nM T13260 D0HR9S 388623 Ki = 15.1 nM T13260 D0I1SI 49799655 IC50 = 760 nM T13260 D0I1YH 46901446 IC50 = 663 nM T13260 D0I2UE 46867543 IC50 = 3.98 nM T13260 D0I5NW 6540047 IC50 = 4073 nM T13260 D0I5PY 23585406 IC50 = 210 nM T13260 D0I7GE 11790 Ki = 20 nM T13260 D0J2WW 6539801 IC50 = 770 nM T13260 D0J3PK 11779089 IC50 = 41 nM T13260 D0J4VR 46191176 IC50 = 5000 nM T13260 D0J8FS 5377857 IC50 = 8330 nM T13260 D0JE1I 9815923 IC50 = 680 nM T13260 D0K2SE 10703161 IC50 = 6400 nM T13260 D0K3CE 6539800 IC50 = 280 nM T13260 D0K4PY 114829 IC50 = 2100 nM T13260 D0K5GG 49799652 IC50 = 3570 nM T13260 D0K5JU 46867417 IC50 = 1900 nM T13260 D0K5KG 6540050 IC50 = 6045 nM T13260 D0K8QD 63059 IC50 = 24880 nM T13260 D0L1JF 6539791 IC50 = 180 nM T13260 D0L3AJ 5324988 IC50 = 2020 nM T13260 D0L9BT 10823163 IC50 = 3700 nM T13260 D0M0FE 3317166 IC50 = 160 nM T13260 D0M2IB 9904788 Ki = 4 nM T13260 D0M4CX 356713 Ki = 385 nM T13260 D0M5EW 11276192 IC50 = 2089.3 nM T13260 D0M7FS 6539764 IC50 = 2490 nM T13260 D0M8RO 6128 Ki = 20 nM T13260 D0MA9G 6540051 IC50 = 1507 nM T13260 D0N1GH 11601068 IC50 > 36000 nM T13260 D0N1PQ 11506923 IC50 = 586 nM T13260 D0N5GZ 12229395 IC50 = 24500 nM T13260 D0N7QV 11819989 IC50 = 0.7 nM T13260 D0N9PY 6539773 IC50 = 7080 nM T13260 D0NB8V 49799650 IC50 = 16420 nM T13260 D0NH6T 14218027 IC50 = 400 nM T13260 D0NX0M 6540049 IC50 = 814 nM T13260 D0O0BL 44394887 IC50 = 430 nM T13260 D0O1ZM 13660225 IC50 = 1500 nM T13260 D0O4YS 42618026 IC50 > 98490 nM T13260 D0O6ZM 14256024 IC50 = 670 nM T13260 D0OY1J 11401873 IC50 = 676.08 nM T13260 D0P3ND 46887506 IC50 = 160 nM T13260 D0P5ZV 261861 IC50 = 9800 nM T13260 D0PU5V 10750911 IC50 = 1380 nM T13260 D0Q0BK 46901611 IC50 = 1670 nM T13260 D0Q3JZ 6539774 IC50 = 7680 nM T13260 D0Q6XB 5844100 IC50 = 7470 nM T13260 D0Q8UZ 18785180 IC50 = 590 nM T13260 D0QL1V 508445 IC50 = 1200 nM T13260 D0R0TE 11557864 IC50 = 6638 nM T13260 D0R2YN 5994480 IC50 = 15500 nM T13260 D0R4FM 122850 IC50 > 40 ug.mL-1 T13260 D0R4WW 44265823 Ki = 10.3 nM T13260 D0RJ6S 11558270 IC50 > 36000 nM T13260 D0S0EP 585819 IC50 = 28.18 nM T13260 D0S0OV 10267149 IC50 = 91 nM T13260 D0S0RK 10680 IC50 = 8 nM T13260 D0S1AY 269167 IC50 = 26800 nM T13260 D0S7VY 49798801 IC50 = 2940 nM T13260 D0S8MJ 337743 IC50 = 2100 nM T13260 D0S9YX 5280373 IC50 = 10.2 nM T13260 D0SY2M 5281708 Ki = 100000 nM T13260 D0SY6C 5282073 IC50 = 2 nM T13260 D0T0CK 49799648 IC50 = 14510 nM T13260 D0T3ED 44580826 Ki = 33.4 nM T13260 D0T3PW 5281672 IC50 = 10000 nM T13260 D0T5NO 15306617 IC50 = 100 nM T13260 D0TM4K 6539817 IC50 = 3680 nM T13260 D0U4BB 10748 IC50 > 10000 nM T13260 D0U6IT 6539807 IC50 = 4830 nM T13260 D0U6NJ 11311402 IC50 = 758.58 nM T13260 D0U7RR 6539768 IC50 = 7370 nM T13260 D0U8JC 9862769 IC50 = 4600 nM T13260 D0U9QB 73440 IC50 = 15 nM T13260 D0UI8Q 10566470 IC50 = 2089.3 nM T13260 D0V0DB 46887421 IC50 = 20 nM T13260 D0V1UY 133966 IC50 = 3 nM T13260 D0V3MV 46867546 IC50 = 11.45 nM T13260 D0V3YH 6539784 IC50 = 130 nM T13260 D0V8CR 6539763 IC50 = 2540 nM T13260 D0V8SM 10659706 IC50 = 1096.48 nM T13260 D0W3LG 9866908 IC50 = 9700 nM T13260 D0W3LM 10265122 IC50 = 3700 nM T13260 D0W4IB 23644623 Ki = 680 nM T13260 D0W7GU 5377410 IC50 = 1820 nM T13260 D0W7JA 5273567 IC50 = 35300 nM T13260 D0W9PF 13472 Ki = 43 nM T13260 D0W9ZC 46867540 IC50 = 16.5 nM T13260 D0WK9Q 14256034 IC50 = 2760 nM T13260 D0WN9P 46901444 IC50 = 2830 nM T13260 D0X0IH 77918 IC50 = 150 nM T13260 D0X1QS 6540053 IC50 = 3551 nM T13260 D0X8UK 10751574 IC50 = 350 nM T13260 D0XQ6T 42618029 IC50 = 5760 nM T13260 D0XS6T 53602 IC50 = 1840 nM T13260 D0Y0CT 6539819 IC50 = 4060 nM T13260 D0Y0EK 620596 IC50 = 3400 nM T13260 D0Y0QI 10774864 IC50 = 170 nM T13260 D0Y4TE 340000 Ki = 13.1 nM T13260 D0Y5KX 46901443 IC50 = 24500 nM T13260 D0Y7HG 5281616 Ki = 100000 nM T13260 D0Y7RB 6539781 IC50 = 4600 nM T13260 D0Y8XJ 5497182 IC50 = 16800 nM T13260 D0Y9HD 361928 Ki = 52.7 nM T13260 D0YD9J 6539792 IC50 = 5432503.31 nM T13260 D0YS2F 6539776 IC50 = 9740 nM T13260 D0Z1OI 124662 Ki = 1000 nM T13260 D0Z4GR 4594970 IC50 = 100 nM T13260 D0Z7EL 5280647 IC50 = 11000 nM T93509 D00MXN 25019940 Ki = 0.024 nM T93509 D0G5ME 11319053 Ki = 0.78 nM T93509 D0L5GH 6918509 Ki = 0.014 nM T93509 CXZA43 457930 Ki = 7300 nM T93509 C6W7AM 9847811 Ki = 2700 nM T93509 CANV26 10030220 Ki = 710 nM T93509 CH2NR6 11178760 Ki = 1700 nM T93509 C1LX9V 11397043 Ki = 1800 nM T93509 C8GB7A 11419496 Ki = 1900 nM T93509 CQT6I4 16728074 Ki = 16000 nM T93509 C5RC3J 44563430 IC50 >= 1000 nM T93509 C2BKH7 44563440 EC50 = 0.05 nM T93509 CQ1VU2 57392038 Ki = 26000 nM T93509 CF8R4H 57392039 Ki > 100000 nM T93509 C9T7IA 57393753 Ki = 8000 nM T93509 C6UID4 57393754 Ki = 5200 nM T93509 C1O0EL 57393755 Ki > 100000 nM T93509 C6B2JK 57395477 Ki = 14000 nM T93509 CD91MC 57395478 Ki = 45000 nM T93509 CV87FO 57397325 Ki > 100000 nM T93509 CK6L0F 57400721 Ki = 8 nM T93509 C6GF8M 57402496 Ki > 100000 nM T93509 CL85VH 57402497 IC50 > 10000 nM T93509 CPYG07 73345650 IC50 = 0.85 nM T93509 CH9LP4 73345651 IC50 = 3.45 nM T93509 CJ2V8U 73347156 IC50 = 29.73 nM T93509 C4DWG3 73347157 IC50 = 79.34 nM T93509 C8F9IO 73353230 IC50 = 4.15 nM T93509 CC5Q0Y 73354735 Ki = 0.73 nM T93509 CH7GY0 73354736 Ki = 3.3 nM T93509 C3LV6M 73356281 IC50 = 1.31 nM T93509 C3WJM4 127026899 IC50 = 130 nM T93509 CAJ24S 127026900 IC50 = 13 nM T93509 C7ZF6X 127026901 IC50 = 170 nM T93509 C6TRP3 127027478 IC50 = 15 nM T93509 C63EQW 127027479 IC50 = 19 nM T93509 C5VS7T 127027480 IC50 = 77 nM T93509 C26QAE 127027481 IC50 = 12 nM T93509 C9TR7O 127027482 IC50 = 22 nM T93509 C8DPY7 127027501 IC50 = 190 nM T93509 C1MW5C 127027502 IC50 = 460 nM T93509 CEK1B2 127027503 IC50 = 9.8 nM T93509 C9N5SC 127027797 IC50 = 44 nM T93509 C23NCY 127027803 IC50 = 33 nM T93509 C6JT4M 127027804 IC50 = 130 nM T93509 CXNT13 127027805 IC50 = 130 nM T93509 CI4Z3K 127027806 IC50 = 8.9 nM T93509 CZD67W 127027807 IC50 = 99 nM T93509 CR8GD0 127027810 IC50 = 110 nM T93509 CJH92D 127027811 IC50 = 44 nM T93509 C1BFU9 127027812 IC50 = 120 nM T93509 C0JIC7 127027814 IC50 = 350 nM T93509 CWS56B 127027815 IC50 = 4.3 nM T93509 CH0S6M 127027816 IC50 = 12 nM T93509 CQ3CR8 127027821 IC50 = 140 nM T93509 C0UGB6 127027822 IC50 = 97 nM T93509 CQ56CX 127027823 IC50 = 150 nM T93509 CT95NM 127027824 IC50 = 41 nM T93509 C3IJR5 127028113 IC50 = 46 nM T93509 CBJ5A4 127028116 IC50 = 7 nM T93509 C8SCZ7 127028121 IC50 = 34 nM T93509 CW1D3C 127028122 IC50 = 2.9 nM T93509 CDU86M 127028128 IC50 = 14 nM T93509 C1VEB4 127028129 IC50 = 0.23 nM T93509 CD70TW 127028130 IC50 = 0.11 nM T93509 C86NMZ 127028438 IC50 = 170 nM T93509 CHO8T2 127028443 IC50 = 92 nM T93509 C4Z1ND 127028444 IC50 = 120 nM T93509 CHM0F8 127028769 IC50 = 240 nM T93509 CM25XZ 127028770 IC50 = 54 nM T93509 C4NR9D 127028771 IC50 = 1.1 nM T93509 CTO2K3 127028772 IC50 = 19 nM T93509 CJ4IZ2 127028773 IC50 = 16 nM T93509 CPE3B1 127028774 IC50 = 24 nM T93509 CQ9R3C 127028775 IC50 = 430 nM T93509 D05LMD 16134896 Ki = 3.19 nM T93509 D0I2KW 44406785 IC50 = 740 nM T93509 D0U4BO 44563409 IC50 = 0.64 nM T08446 D0ED7U 60648 IC50 = 1670000 nM T08446 D08ESA 198693 IC50 = 300000 nM T08446 D0C9XA 119 IC50 = 2000 nM T08446 CJ9V4G 40598 IC50 = 290000 nM T08446 CXSD61 155246 IC50 = 3000 nM T08446 CHV0G9 639062 IC50 > 1000000 nM T08446 C97FYX 702501 IC50 = 100000 nM T08446 C8X9TQ 1069892 IC50 = 2884.03 nM T08446 C1A0UL 1502074 IC50 = 7943.28 nM T08446 C3DR8J 1502075 IC50 = 3981.07 nM T08446 C9EI4M 1530639 IC50 > 1000000 nM T08446 CU23IC 4531494 IC50 = 208000 nM T08446 CG1ZF6 5311322 Ki = 1600 nM T08446 CN2C7Q 6604883 IC50 = 630000 nM T08446 C4A6SU 8181355 IC50 = 180000 nM T08446 CQ64IH 9797818 IC50 = 7210000 nM T08446 C31HNE 9884272 Ki = 42000 nM T08446 CY2IS7 9888224 IC50 = 39000 nM T08446 CTZ5Q7 9983570 IC50 = 2660000 nM T08446 C75BDY 10031163 IC50 = 201000 nM T08446 CZ4PO2 10050339 IC50 = 1270000 nM T08446 CP2WF1 10072112 IC50 = 27000 nM T08446 CG1A4H 10073933 IC50 = 151000 nM T08446 C4S1CO 10096504 IC50 = 382000 nM T08446 C0XI3N 10252046 IC50 = 920000 nM T08446 CXJR61 10252950 IC50 = 655000 nM T08446 CC8V4E 10412575 IC50 = 109000 nM T08446 CZ8FQ2 10481573 IC50 = 88000 nM T08446 CU40KP 11743493 IC50 = 435000 nM T08446 CH6GX1 13314232 IC50 = 91000 nM T08446 C6VK4E 17173775 IC50 > 1000000 nM T08446 CE92MX 17174058 IC50 > 1000000 nM T08446 C3OQD7 17250318 IC50 = 170000 nM T08446 CME93B 43345728 IC50 > 1000000 nM T08446 C5JUW9 47058964 IC50 > 1000000 nM T08446 CLIK30 50941729 IC50 > 100000 nM T08446 CQ4XJ7 55285849 IC50 = 5480 nM T08446 CY9O8W 55285850 IC50 = 5480 nM T08446 C8UTR2 67642717 IC50 = 7300 nM T08446 C6ME5H 70684991 IC50 = 335000 nM T08446 C79CYX 70689234 IC50 = 2900000 nM T08446 CD9EV5 70691307 IC50 = 809000 nM T08446 CJ7P8C 70691309 IC50 = 436000 nM T08446 C53QGB 118711599 IC50 = 590 nM T08446 CO18BS 137635197 IC50 = 8000 nM T08446 CQL64H 137637846 IC50 > 1000000 nM T08446 CZ73DV 137638595 IC50 > 100000 nM T08446 CARI53 137638617 IC50 > 100000 nM T08446 CUM2T0 137638836 IC50 > 100000 nM T08446 C3PY5G 137638838 IC50 > 50000 nM T08446 CP7OV5 137639241 IC50 > 100000 nM T08446 C21IZT 137639281 IC50 > 1000000 nM T08446 CP24OX 137642163 IC50 > 100000 nM T08446 CK2VU3 137650102 IC50 > 1000000 nM T08446 C52PYO 137650910 IC50 > 1000000 nM T08446 CS6FX4 137651374 IC50 > 1000000 nM T08446 CPLJ94 137651669 IC50 > 1000000 nM T08446 CN04QK 137652511 IC50 > 1000000 nM T08446 CGC1Z4 137654858 IC50 > 50000 nM T08446 CADN74 137657292 IC50 > 100000 nM T08446 C4NK1W 137658990 IC50 > 50000 nM T08446 CPI4S8 137659917 IC50 > 50000 nM T08446 CI7S8H 155516242 IC50 > 100000 nM T08446 C4U8QT 155524561 IC50 > 100000 nM T08446 CJ4OV6 155530359 IC50 > 100000 nM T08446 C4RL9X 155535776 IC50 > 100000 nM T08446 CL2Q6G 155567178 IC50 > 100000 nM T08446 D02ANG 5216267 IC50 = 47400 nM T08446 D03IWW 6575389 IC50 = 6410000 nM T08446 D08YGM 92409 IC50 = 7210000 nM T08446 D0D2EF 1796510 IC50 = 2310000 nM T08446 D0H7WK 10458835 IC50 = 71700 nM T08446 D0P3KI 9888030 IC50 = 5100 nM T08446 D0RF2M 4498 IC50 = 2370000 nM T08446 D0V5OY 16725912 Ki = 15000 nM T08446 D0V7RG 3532 IC50 = 1870000 nM T97537 CQ5T2C 2837573 Ki = 7700 nM T97537 CIBH72 3834735 Ki > 100000 nM T97537 CA1ZC4 4188970 Ki = 5000 nM T97537 C4EBQ6 8823441 IC50 = 1100 nM T97537 CT45FK 24828324 Ki = 147.91 nM T97537 C1WKD6 24828325 Ki = 20.42 nM T97537 CJ6RS7 24828326 Ki = 5754.4 nM T97537 C98VUW 24828598 Ki = 5370.32 nM T97537 CW64AC 24828600 Ki = 144.54 nM T97537 CFP01R 24828743 Ki = 100 nM T97537 C9LUM1 24828881 Ki = 27.54 nM T97537 CER36P 24828882 Ki = 2137.96 nM T97537 C0VL7B 24890303 Ki = 10715.19 nM T97537 CJ6G0Y 42601512 Ki = 480 nM T97537 CL2A3I 42610322 Ki = 20 nM T97537 C12CDQ 44254309 Ki = 3019.95 nM T97537 C8EI1G 44254310 Ki = 8511.38 nM T97537 CD3L0N 44254402 Ki = 794.33 nM T97537 CHT0Z1 44254404 Ki = 2454.71 nM T97537 CW7LB9 44254495 Ki = 2041.74 nM T97537 C5FDC2 44254496 Ki = 2951.21 nM T97537 CE40ON 44277843 Ki = 52 nM T97537 CID3S9 44450222 Ki = 177.83 nM T97537 CCJ39L 44450246 Ki = 1071.52 nM T97537 CX05EH 44450286 Ki = 173.78 nM T97537 C87BVH 44450320 Ki = 165.96 nM T97537 C98XEN 44450334 Ki = 1318.26 nM T97537 CD7UO5 44450345 Ki = 630.96 nM T97537 CH02ZM 44450376 Ki = 81.28 nM T97537 CD85RG 44450377 Ki = 109.65 nM T97537 CZ4H7R 44560401 Ki = 1200 nM T97537 C70AIZ 44560402 Ki = 12000 nM T97537 C63VWA 44560403 Ki = 7400 nM T97537 CRX2G5 44560404 Ki = 2500 nM T97537 CA4IF6 44560405 Ki = 1400 nM T97537 C57LTE 44560406 Ki = 3700 nM T97537 C2F3TI 44560407 Ki = 3100 nM T97537 CC3GY2 44560408 Ki = 1300 nM T97537 C9YE7J 44560409 Ki = 1300 nM T97537 C1OEW5 44560410 Ki = 1800 nM T97537 CU4G1S 44560411 Ki = 1000 nM T97537 C2Y0OT 44560412 Ki = 97000 nM T97537 CG7BQ8 44560457 Ki = 16000 nM T97537 C1RK3C 44560557 Ki = 35000 nM T97537 C42VEQ 44560558 Ki = 76000 nM T97537 CMLG10 46882676 Ki = 4786.3 nM T97537 CTO1Q8 46882677 Ki = 3981.07 nM T97537 CP9WB0 49840768 Ki = 282 nM T97537 C51YRX 49840770 Ki = 54.8 nM T97537 CJ3Z7V 49840772 Ki = 1752 nM T97537 CS3I8G 49840774 Ki = 3.3 nM T97537 C3IT5V 49840844 Ki = 242 nM T97537 CYBW37 49840846 Ki = 18.5 nM T97537 CFEC23 49840848 Ki = 93.7 nM T97537 C64XMG 49840850 Ki = 5.2 nM T97537 CNU1Q7 49840921 Ki = 34.9 nM T97537 CQ90FE 52941108 Ki = 5506 nM T97537 CU4HK1 52943524 Ki = 196 nM T97537 C9HRG4 52946764 Ki = 22.5 nM T97537 C89EGH 52947188 Ki = 9.3 nM T97537 CU58OG 53257413 Ki = 4.1 nM T97537 C6XY5R 53259047 Ki = 50 nM T97537 C7AXD8 53259048 Ki = 41.1 nM T97537 CX51OK 53259216 Ki = 697 nM T97537 CBS92H 53259217 Ki = 351 nM T97537 C8RZW7 53259219 Ki = 5845 nM T97537 C4KZ7R 53259403 Ki = 4011 nM T97537 CA0Q2E 53259404 Ki = 12000 nM T97537 C6FU2G 53259405 Ki = 10800 nM T97537 CLSC37 53261358 Ki = 25 nM T97537 CXMC12 53261359 Ki = 64.2 nM T97537 C3Q4ZR 53261360 Ki = 193 nM T97537 CGF98A 54585162 Ki = 30.4 nM T97537 CG46AV 71817662 IC50 = 38300 nM T97537 C7P2UD 71817806 IC50 = 3900 nM T97537 CW85UH 71817807 IC50 > 100000 nM T97537 CO8K1H 71817808 IC50 = 46000 nM T97537 CMQN63 71817809 IC50 = 10300 nM T97537 CPNL07 71817811 IC50 = 9600 nM T97537 C1N7QD 71817963 IC50 = 2800 nM T97537 CMBJ36 71817964 IC50 = 1300 nM T97537 CK2T9X 71817965 IC50 = 16300 nM T97537 CE7VJ4 71817966 IC50 > 100000 nM T97537 C74CNV 72193911 IC50 = 30 nM T97537 C8ZGB7 118734158 IC50 = 10000 nM T97537 C0T8FC 118734159 IC50 = 10700 nM T97537 CU5F3O 118734160 IC50 = 57000 nM T97537 CB67XZ 118734161 IC50 = 10900 nM T97537 CJ19XY 118734162 IC50 = 2100 nM T97537 C67EIN 118734163 IC50 = 12000 nM T97537 C5HV4G 118734165 IC50 = 7200 nM T97537 CB7W1N 118734166 IC50 = 14600 nM T97537 CVQ9B5 118734167 IC50 = 34000 nM T97537 CTE28S 118734169 IC50 > 100000 nM T97537 C3VMB4 118734170 IC50 = 3800 nM T97537 C5B3AO 118734171 IC50 = 4800 nM T97537 CR02XN 118734172 IC50 = 10700 nM T97537 CYQ61P 118734173 IC50 = 5700 nM T97537 CG1NJ3 118734176 IC50 = 4100 nM T97537 CTL4C9 118734177 IC50 > 100000 nM T97537 CWK18R 118734179 IC50 = 12000 nM T97537 CED26H 118734180 IC50 > 100000 nM T97537 C24VOF 118734181 IC50 = 22000 nM T97537 C3KJR9 118734182 IC50 > 100000 nM T97537 CMWH70 118734252 IC50 = 7100 nM T97537 CS1R6T 118734253 IC50 > 100000 nM T97537 CK3NV4 118734254 IC50 = 933 nM T97537 C4VK6O 118734255 IC50 = 4400 nM T97537 C7AH4D 118734256 IC50 = 1300 nM T97537 CZ04FM 118734257 IC50 > 100000 nM T97537 CZ97HL 118734258 IC50 = 1200 nM T97537 C1DKP8 118734259 IC50 = 105 nM T97537 CET0D8 118734260 IC50 = 296 nM T97537 C4N7KF 118734261 IC50 = 31000 nM T97537 C2M4UZ 118734262 IC50 = 3300 nM T97537 C3PL1T 118734263 IC50 = 966 nM T97537 C3OS1H 118734264 IC50 = 655 nM T97537 C9NWC0 118734265 IC50 = 31000 nM T97537 C3PW9J 118734266 IC50 = 1700 nM T97537 CX0OA9 118734267 IC50 = 8300 nM T97537 CU8I4F 118734268 IC50 = 3300 nM T97537 CI6S8L 118734269 IC50 = 39600 nM T97537 C6IB5P 118734270 IC50 > 100000 nM T97537 CUGM56 118734271 IC50 = 9900 nM T97537 CH2LO8 118734272 IC50 = 22500 nM T97537 CI9RT3 118734273 IC50 > 100000 nM T97537 CK32TS 118734274 IC50 = 2500 nM T97537 CT5F3Q 118734275 IC50 = 20600 nM T97537 C3KLH4 118734276 IC50 = 14400 nM T97537 CPUI84 118734277 IC50 = 20200 nM T97537 C96PKA 118734278 IC50 = 1300 nM T97537 C4AL9Z 118734279 IC50 = 2400 nM T97537 C71TGN 118734280 IC50 = 4700 nM T97537 C8V9EB 118734281 IC50 = 2900 nM T97537 CIZ3Q6 118734282 IC50 = 3700 nM T97537 CJ64ZC 118734283 IC50 = 3800 nM T97537 C1K7AN 118734284 IC50 = 1300 nM T97537 C6XY9M 118734285 IC50 = 70000 nM T97537 CY8X0V 118734286 IC50 = 3400 nM T97537 CO4F3Y 118734287 IC50 = 5200 nM T97537 C9CN6S 118734288 IC50 = 3700 nM T97537 CI3R0S 118734289 IC50 > 100000 nM T97537 CN7SR4 118734290 IC50 = 3900 nM T97537 C57ZSG 118734291 IC50 > 100000 nM T97537 CKST54 118734292 IC50 = 3600 nM T97537 C9XDY5 118734293 IC50 = 438 nM T97537 C01PYL 118734294 IC50 = 1700 nM T97537 CO6PR7 118734295 IC50 = 35700 nM T97537 C4ZPC8 118734296 IC50 = 2200 nM T97537 CJ40TN 118734297 IC50 = 7600 nM T97537 CA9X0N 118734298 IC50 = 4900 nM T97537 C7FMV5 126456392 Ki = 18 nM T97537 C8QO7V 135554374 IC50 = 28000 nM T97537 CXLS30 137633011 IC50 = 381 nM T97537 CMC5E8 137634250 IC50 = 18 nM T97537 CER06G 137637900 IC50 = 577 nM T97537 C97XKO 137638141 IC50 = 16 nM T97537 CMTG53 137639983 IC50 = 1754 nM T97537 CH6DQ2 137640549 IC50 = 281 nM T97537 C9SWV7 137640590 IC50 = 46 nM T97537 CG0ED2 137641900 IC50 = 14 nM T97537 C3SP9K 137642894 IC50 = 317 nM T97537 C1U3ZM 137642974 IC50 = 1800 nM T97537 CYN9Z5 137646376 IC50 = 41 nM T97537 CDU93R 137646849 IC50 = 13 nM T97537 C96EWT 137647165 IC50 = 32 nM T97537 CJM57W 137648545 IC50 = 13 nM T97537 CC9T7O 137650040 IC50 = 9 nM T97537 CN9F2A 137650752 IC50 = 185 nM T97537 CB9VI7 137652734 IC50 = 102 nM T97537 CSM3V5 137653412 IC50 = 221 nM T97537 CVI87E 137654495 IC50 = 21 nM T97537 C8DV5C 137655020 IC50 = 4024 nM T97537 C2RIG6 137655030 IC50 = 4 nM T97537 CMT56C 137655972 IC50 = 434 nM T97537 C13POW 137656080 IC50 = 561 nM T97537 CCTK37 137657323 IC50 = 34 nM T97537 C4VS2D 137658289 IC50 = 20 nM T97537 CKHE71 137659752 IC50 = 10 nM T97537 C0ID7T 137660529 IC50 = 2 nM T97537 C8E6UD 137661774 IC50 = 29 nM T97537 CV2U0Z 137662110 IC50 = 41 nM T97537 D02MNM 71817810 IC50 = 6000 nM T97537 D04DTE 53259050 Ki = 1.8 nM T97537 D0L3PY 123814 Ki = 7 nM T88415 COQ0J9 9846486 IC50 = 3500 nM T88415 CSH73Q 43230121 IC50 = 5000 nM T88415 C09TSQ 145978898 IC50 = 100 nM T88415 CFX8E2 145979186 IC50 > 100000 nM T88415 CS9M7U 145990033 IC50 = 800 nM T88415 CS2HG5 145991728 IC50 = 100 nM T88415 C4K2YT 145992615 IC50 > 10000 nM T40488 D05VZE 119031 IC50 = 10000 nM T40488 D03BOZ 3342298 IC50 = 0.54 nM T40488 CN6E3U 2366268 IC50 = 83000 nM T40488 CR7T3J 10009978 Ki > 2000 nM T40488 C1LCH3 10016964 IC50 = 62000 nM T40488 CR5H6E 10163627 IC50 = 1600 nM T40488 CK0P3F 10186536 IC50 > 10000 nM T40488 C4K1MJ 10208262 IC50 = 4600 nM T40488 CBM0Y4 10252411 Ki < 100 nM T40488 CY08WJ 10322755 Ki = 1650 nM T40488 CFKA79 10395015 Ki > 2000 nM T40488 C5WV1N 10439082 Ki > 2000 nM T40488 C8C5AV 11294179 IC50 > 10000 nM T40488 CO8QT0 11753905 Ki = 240 nM T40488 C8YWV5 11778852 IC50 = 53000 nM T40488 C02BWA 11967143 Ki > 2000 nM T40488 CQS0F5 16719301 IC50 = 55 nM T40488 C75XDI 16730519 IC50 = 2400 nM T40488 C1MCG7 22004293 Ki = 335 nM T40488 CAQ9Z1 25022681 Ki > 5346 nM T40488 CHQG04 44576676 Ki = 23000 nM T40488 CR65DO 44576708 Ki = 1600 nM T40488 C2QFY7 44576710 Ki = 4570 nM T40488 CU2IP7 44576753 Ki = 22000 nM T40488 C93LDF 44576807 Ki = 372000 nM T40488 CJ41MB 44576851 Ki = 337000 nM T40488 CU2SX3 51355576 Ki > 10000 nM T40488 C6Y2EV 53374826 IC50 > 100000 nM T40488 C1PHI6 57708731 IC50 = 820 nM T40488 CF2Z7W 57708783 IC50 = 140 nM T40488 C9KV2W 57708792 IC50 = 460 nM T40488 CE36GP 57708799 IC50 = 270 nM T40488 C23QGY 57708843 IC50 > 1000 nM T40488 C2J5CW 57708880 IC50 > 1000 nM T40488 C1K6AP 57708886 IC50 = 30 nM T40488 C61NKZ 72720906 IC50 = 21 nM T40488 C7XWM5 72948626 IC50 = 17 nM T40488 CR70EY 72948808 IC50 = 12 nM T40488 C2WV4D 72948991 IC50 = 7810 nM T40488 CA76TR 72948995 IC50 = 18 nM T40488 CZ95GN 72949172 IC50 = 16 nM T40488 CSH7A5 90033597 IC50 = 11400 nM T40488 CYZP25 91824169 IC50 > 10000 nM T40488 C0M3QS 118179775 IC50 = 42 nM T40488 C0XML2 118179776 IC50 = 62 nM T40488 C0W3NG 118179777 IC50 = 435 nM T40488 CX9YG0 118179779 IC50 = 7 nM T40488 CW1TU9 118179786 IC50 = 54 nM T40488 CRG2W5 118179799 IC50 = 189 nM T40488 CH35NR 118179800 IC50 = 9 nM T40488 CK54UB 118179801 IC50 = 739 nM T40488 CP8QO0 118179807 IC50 = 13 nM T40488 CT4G5D 118179817 IC50 = 68 nM T40488 CIU02H 118179819 IC50 = 4 nM T40488 CD9TG2 118179830 IC50 = 103 nM T40488 CN72KV 118179833 IC50 = 184 nM T40488 CZ01AH 118179837 IC50 = 713 nM T40488 C6TR4O 118179845 IC50 = 25400 nM T40488 C5TZ1D 118179847 IC50 = 14 nM T40488 CVWR97 118179850 IC50 = 20700 nM T40488 CT8U1K 118179865 IC50 = 8700 nM T40488 CR64FW 118179867 IC50 = 84 nM T40488 CIXQ34 118179870 IC50 = 3 nM T40488 C27XIK 118225133 IC50 > 10000 nM T40488 C58KIN 118233723 IC50 > 10000 nM T40488 CU6ES2 118233724 IC50 > 10000 nM T40488 C8ET1Z 118233725 IC50 > 10000 nM T40488 C9P0LC 118233726 IC50 > 10000 nM T40488 C8SIM0 118233727 IC50 > 10000 nM T40488 CQTE52 118233728 IC50 > 10000 nM T40488 CEVI64 118233730 IC50 > 10000 nM T40488 C08CPE 118233731 IC50 > 10000 nM T40488 C8Q5XC 118233733 IC50 > 10000 nM T40488 CZQO42 118233734 IC50 > 10000 nM T40488 CCDG68 118233743 IC50 > 10000 nM T40488 C25TYU 118233744 IC50 > 10000 nM T40488 CL5UV6 118233745 IC50 > 10000 nM T40488 C8XWB9 118233746 IC50 > 10000 nM T40488 CC7K9R 118233747 IC50 > 10000 nM T40488 CGA7J1 118233748 IC50 > 10000 nM T40488 CVIG81 118233749 IC50 > 10000 nM T40488 CTU81Y 118233750 IC50 > 10000 nM T40488 CCA6W2 118233751 IC50 > 10000 nM T40488 C60QIZ 118233752 IC50 > 10000 nM T40488 CS5G9T 118233753 IC50 > 10000 nM T40488 CGKD16 118734983 IC50 = 32 nM T40488 C84NEC 118734984 IC50 = 89 nM T40488 CX7H5Q 118734985 IC50 = 17 nM T40488 CNF86U 121493953 Ki = 1.4 nM T40488 CH1GT7 123144081 IC50 > 10000 nM T40488 CKNI84 127050262 IC50 = 8400 nM T40488 CN9D7G 134155756 IC50 = 6300 nM T40488 CHV2U1 135438561 IC50 = 160 nM T40488 C6GR3K 135567051 IC50 = 140 nM T40488 CYH23I 136054468 IC50 = 220 nM T40488 CZ8DW1 136054472 IC50 = 34 nM T40488 C9H0DL 136054473 IC50 = 460 nM T40488 CX7MI0 136054475 IC50 = 64 nM T40488 CA5JR6 136054481 IC50 = 240 nM T40488 CO2VU9 136054484 IC50 < 10 nM T40488 CV47JN 136054485 IC50 = 6.2 nM T40488 CZ48WO 136054487 IC50 = 150 nM T40488 CR9CY5 136054490 IC50 < 10 nM T40488 C8FGT0 136054495 IC50 = 930 nM T40488 CGH39U 136054498 IC50 < 10 nM T40488 C2TO7Y 136054508 IC50 = 640 nM T40488 CG70BZ 136054516 IC50 = 0.35 nM T40488 CSM57W 136054520 IC50 = 2.6 nM T40488 CIEW62 136380958 IC50 = 2.4 nM T40488 C9HS7J 137287436 IC50 = 0.3 nM T40488 CAZ87R 137631621 IC50 = 676.08 nM T40488 C0R5ZT 137635841 IC50 = 436.52 nM T40488 CU5G8I 137636679 IC50 = 635 nM T40488 C1RID9 137636861 IC50 = 2050 nM T40488 CNM8J4 137638970 IC50 = 29.51 nM T40488 C7Y0FB 137642170 IC50 = 1210 nM T40488 CDOQ29 137644394 IC50 = 1698.24 nM T40488 C04KVQ 137647395 IC50 = 705 nM T40488 CHI2E1 137648744 IC50 = 112.2 nM T40488 C1U2QR 137651063 IC50 = 141.25 nM T40488 C5Y8RP 137654086 IC50 = 7380 nM T40488 CRD46H 137658344 IC50 = 347 nM T40488 C3ER5O 137658673 IC50 = 506 nM T40488 CEQ8I9 137659945 IC50 = 588.84 nM T40488 CHO70T 137660954 IC50 = 751 nM T40488 C1IF6L 137661809 IC50 = 131 nM T40488 CYFQ54 144883303 IC50 > 10000 nM T40488 CA2EI4 144883305 IC50 > 10000 nM T40488 CX80ML 144883318 IC50 > 10000 nM T40488 CQYH92 145949456 IC50 > 10000 nM T40488 C2SM0T 145950300 IC50 > 10000 nM T40488 C85BXD 145951133 IC50 > 10000 nM T40488 C6JP8O 145955500 IC50 > 10000 nM T40488 CXT3I5 145958912 IC50 > 10000 nM T40488 CQN59P 145959729 IC50 > 10000 nM T40488 CX6R5D 145959924 IC50 > 10000 nM T40488 C0K4JW 145972664 IC50 > 10000 nM T40488 CF64GH 155518335 Ki = 983 nM T40488 D03AMR 9849669 Ki = 190 nM T40488 D04VPH 45376872 IC50 = 16000 nM T40488 D07SPC 24857837 Ki = 356 nM T40488 D0B3UN 44580458 Ki = 149 nM T40488 D0OR6O 91623362 IC50 = 12 nM T40488 D0Y5IQ 44255320 IC50 = 5000 nM T10877 D04AIT 5280445 IC50 = 8200 nM T10877 D0K8KX 5280343 IC50 = 37900 nM T10877 D0E3LP 5113032 IC50 > 100000 nM T10877 D0U3EP 445154 IC50 > 100000 nM T10877 CU12QE 1203 IC50 > 100000 nM T10877 CEM9Q1 128853 IC50 = 14600 nM T10877 CNMW58 159287 IC50 = 17000 nM T10877 CAB1I4 440832 IC50 = 16300 nM T10877 CT2S6P 441667 IC50 = 6300 nM T10877 CG5OR9 441697 IC50 = 14200 nM T10877 CHE81U 441701 IC50 = 6000 nM T10877 CXB75J 441773 IC50 = 20900 nM T10877 CXG1I8 441774 IC50 = 39200 nM T10877 CLY6K3 661302 IC50 > 100000 nM T10877 CJ0T4E 3612016 IC50 > 100000 nM T10877 CY9C4T 5281680 IC50 = 48600 nM T10877 C4KG0A 5403988 IC50 = 296000 nM T10877 CKC79O 10053069 IC50 = 276000 nM T10877 C5J6HV 11170346 IC50 = 158000 nM T10877 CU7Y3S 12309895 IC50 = 70300 nM T10877 C5VH6T 14842007 IC50 = 32100 nM T10877 C4DQJ9 24285123 IC50 = 120000 nM T10877 C36ILR 44532635 IC50 = 1210 nM T10877 CLX72I 59474759 IC50 > 30000 nM T10877 C5GB8X 91827499 IC50 = 76 nM T10877 C64QCZ 91827500 IC50 = 7200 nM T10877 CM01EG 101886781 IC50 = 27000 nM T10877 CWC1Q3 101886782 IC50 = 6400 nM T10877 C5G1LT 101886783 IC50 = 33000 nM T10877 CDT01C 101886784 IC50 = 3300 nM T10877 CQUF15 118736849 IC50 = 58 nM T10877 C5KPU3 118736852 Ki = 14 nM T10877 CG7I6Z 118736853 IC50 = 52 nM T10877 CDR8M7 118736855 IC50 = 3.9 nM T10877 C3M6IP 118736856 Ki = 0.3 nM T10877 CZSB48 118736857 Ki = 0.7 nM T10877 CIE3W9 118736858 IC50 = 54 nM T10877 CH26AO 118736859 IC50 = 3.8 nM T10877 CAQM69 118736860 IC50 = 13 nM T10877 CEL48B 118736861 Ki = 0.45 nM T10877 C7JQ3Y 118736862 IC50 = 14 nM T10877 C6MZ9V 118736863 IC50 = 10773 nM T10877 C0U5DA 118736864 IC50 = 498 nM T10877 CZVT62 118736865 IC50 = 959 nM T10877 CE21BJ 118736866 IC50 = 1960 nM T10877 C30BIV 118736867 IC50 = 11400 nM T10877 CC10IV 118736868 IC50 = 3350 nM T10877 CXO8F1 118736869 IC50 = 2300 nM T10877 CAYX13 118736870 IC50 = 23400 nM T10877 CDW94Q 118736871 IC50 > 30200 nM T10877 CY4LA6 118736872 IC50 = 4710 nM T10877 CTCH72 118736873 IC50 = 1160 nM T10877 C3ARY5 118736874 IC50 = 1590 nM T10877 CW4O7N 118736875 IC50 = 263 nM T10877 CL51QY 118736876 IC50 = 206 nM T10877 CKMD80 118736877 IC50 = 28 nM T10877 CY93JQ 118736878 IC50 = 26 nM T10877 C73EMV 118736879 IC50 = 64 nM T10877 C1B2JZ 118736880 IC50 = 53 nM T10877 C5KGR7 118736881 IC50 = 42 nM T10877 CVM02C 118736882 IC50 = 245 nM T10877 CCH64S 118736883 IC50 = 50 nM T10877 CB6S3J 118736884 IC50 = 3.4 nM T10877 C2SWZ4 118736886 IC50 = 4.8 nM T10877 CXEC56 118736887 IC50 = 5.3 nM T10877 C9LJ0B 118736888 IC50 = 298 nM T10877 C06HDY 118736889 IC50 = 840 nM T10877 CT8G1K 118736890 IC50 = 1200 nM T10877 CUN41C 118736891 IC50 = 1320 nM T10877 CGJW47 118736892 IC50 = 700 nM T10877 CAU39P 118736893 IC50 = 3610 nM T10877 CT5A7R 118736894 IC50 = 2330 nM T10877 C1YMX6 118736895 IC50 = 970 nM T10877 C0RD2H 118736896 IC50 = 4680 nM T10877 CO70TW 118736897 IC50 = 1230 nM T10877 C8HC3W 118736898 IC50 = 1160 nM T10877 CK2LV7 118736899 IC50 = 12800 nM T10877 CXQ37E 118736900 IC50 = 2150 nM T10877 CRT50V 118736901 IC50 = 700 nM T10877 CPAE18 118736902 IC50 = 970 nM T10877 CUPZ76 118736903 IC50 = 2690 nM T10877 CA87UE 118736904 IC50 = 560 nM T10877 CS59UX 118736905 IC50 = 840 nM T10877 CL7CR9 118736906 IC50 = 460 nM T10877 CT0EM6 118736907 IC50 = 1460 nM T10877 C3AJ1K 118736908 IC50 = 12300 nM T10877 CXJQ24 118736909 IC50 = 3940 nM T10877 CL0OQ1 118736910 IC50 = 950 nM T10877 C8TWX1 118736911 IC50 = 7830 nM T10877 C4OW8Z 118736912 IC50 = 1930 nM T10877 C6W4EN 118736913 IC50 = 281 nM T10877 C4FY6U 118736914 IC50 = 132 nM T10877 C6M7KH 118736915 IC50 = 1680 nM T10877 C3U9ZQ 118736916 IC50 = 1060 nM T10877 CN3DE6 118736989 IC50 = 1030 nM T10877 C3A5TU 118736990 IC50 > 30200 nM T10877 C7USD5 118736991 IC50 > 30200 nM T10877 CH1XL4 118736992 IC50 = 149 nM T10877 C2U9HL 118736993 IC50 = 1220 nM T10877 CI24RE 118736994 IC50 = 117 nM T10877 CDC8E7 118736995 IC50 = 140 nM T10877 CND2U1 118736996 IC50 = 49 nM T10877 C1BGP6 118736997 IC50 = 142 nM T10877 CMO4B9 118736998 IC50 = 406 nM T10877 C0Y4VE 118736999 IC50 = 78 nM T10877 CDV30H 118737000 IC50 = 971 nM T10877 C0XI5O 118737001 IC50 = 92 nM T10877 CQD48J 122185943 IC50 > 30000 nM T10877 C6Y2MI 122185944 IC50 = 22000 nM T10877 CR9G7S 122185945 IC50 = 22000 nM T10877 CD64IJ 122185946 IC50 = 3300 nM T10877 CE9OP1 122185947 IC50 > 30000 nM T10877 CBEL62 122185948 IC50 > 30000 nM T10877 CYM8D4 122185949 IC50 = 19000 nM T10877 CE1ZO9 122185950 IC50 > 30000 nM T10877 CE6VJ3 122185951 IC50 > 30000 nM T10877 CX76QZ 122185952 IC50 = 17000 nM T10877 CZ8N9B 122185953 IC50 = 25000 nM T10877 CHE12L 122185954 IC50 = 3300 nM T10877 CL94EM 122185955 IC50 = 2300 nM T10877 CJ17HX 122185956 IC50 > 30000 nM T10877 CI01XG 122185957 IC50 = 18000 nM T10877 CR9AX0 122185958 IC50 = 620 nM T10877 C79BPI 122185959 IC50 > 30000 nM T10877 CZL15G 122185960 IC50 = 4500 nM T10877 CJOV10 122185961 IC50 > 30000 nM T10877 CY2W1Z 122185962 IC50 = 11000 nM T10877 CEV6S8 122185963 IC50 = 990 nM T10877 CM9A0O 122185964 IC50 > 30000 nM T10877 C6D9YZ 122185965 IC50 = 15000 nM T10877 C9CA8T 122185966 IC50 > 30000 nM T10877 C9KAB4 122185967 IC50 > 30000 nM T10877 CLJ1R3 122185968 IC50 = 16000 nM T10877 C6OA7C 122185969 IC50 = 4000 nM T10877 CH16FN 122185970 IC50 = 9600 nM T10877 C8V0WI 122185971 IC50 = 24000 nM T10877 C1FB8D 122185972 IC50 = 6200 nM T10877 CX89LW 122185973 IC50 = 780 nM T10877 CK0UN1 122185974 IC50 = 1200 nM T10877 CQ1WJ8 122185975 IC50 = 510 nM T10877 CKD43Z 122185976 IC50 = 150 nM T10877 CV73WF 122185977 IC50 = 4700 nM T10877 CS7YJ2 122185978 IC50 = 170 nM T10877 CEIT53 122185979 IC50 = 3600 nM T10877 C3ZNU8 122185980 IC50 = 130 nM T10877 CN5P3Q 122185981 IC50 = 280 nM T10877 CIU0M2 122185982 IC50 = 8500 nM T10877 C13TYI 122185983 IC50 = 7300 nM T10877 CSZ0K1 122185984 IC50 > 30000 nM T10877 C8OL5C 122185985 IC50 = 2100 nM T10877 CU47TS 122185986 IC50 = 4900 nM T10877 CVUP84 122185987 IC50 > 30000 nM T10877 CM47OU 122185988 IC50 = 11000 nM T10877 C1DVY8 122185989 IC50 > 30000 nM T10877 CI01VG 122185990 IC50 > 30000 nM T10877 C0M9EL 122185991 IC50 > 30000 nM T10877 CM4S0B 122185992 IC50 > 30000 nM T10877 CO2R4W 122185993 IC50 = 6600 nM T10877 CN4B2Y 122185994 IC50 = 2700 nM T10877 C8WPN3 122185995 IC50 > 30000 nM T10877 CUG8B4 122185996 IC50 > 30000 nM T10877 COYI82 122185997 IC50 > 30000 nM T10877 CSC4B7 122185998 IC50 > 30000 nM T10877 CSOI57 122185999 IC50 = 24000 nM T10877 CGAB47 122186000 IC50 > 10000 nM T10877 CB2H6L 122186001 IC50 > 30000 nM T10877 CZ3R6F 122186002 IC50 > 30000 nM T10877 C6DN9H 122186003 IC50 > 30000 nM T10877 CD0QV5 122186004 IC50 > 30000 nM T10877 CEHN13 122186005 IC50 > 30000 nM T10877 CKFD41 122186006 IC50 > 30000 nM T10877 CU87NS 122186007 IC50 > 30000 nM T10877 CSZ5T7 122186008 IC50 > 30000 nM T10877 C5DU6F 122186009 IC50 > 30000 nM T10877 CQB19L 122186010 IC50 = 9200 nM T10877 C46EGM 135900947 IC50 = 430000 nM T10877 C61OBZ 135949782 IC50 = 103000 nM T10877 C6MF7P 136124133 IC50 = 109000 nM T10877 C0E3AH 136198640 IC50 = 14000 nM T10877 CACG84 136198641 IC50 = 26000 nM T10877 C4Z1WR 137442659 IC50 = 1900 nM T10877 CN09RB 137442681 IC50 = 450 nM T10877 C9G6IA 137442708 IC50 = 630 nM T10877 C9PUZ4 137442715 IC50 = 620 nM T10877 C7DP2S 137442862 IC50 = 92 nM T10877 CW8LT6 137442987 IC50 = 2300 nM T10877 CK26ZH 145967624 IC50 = 7.8 nM T10877 C0YGC8 145967690 IC50 = 1600 nM T10877 CV90MY 145967850 IC50 = 110 nM T10877 C0KJD1 145967861 IC50 = 21 nM T10877 COYK91 145968096 IC50 = 370 nM T10877 CC4P8J 145968138 IC50 = 72 nM T10877 CIW3B1 145968359 IC50 = 3400 nM T10877 C6F4SD 145968563 IC50 = 4100 nM T10877 COA4B0 145968763 IC50 = 170 nM T10877 CX4GA2 145968779 IC50 = 310 nM T10877 C9YRW1 145968807 IC50 = 1900 nM T10877 C4D1JT 145968829 IC50 = 8000 nM T10877 C9SV6Y 145969196 IC50 = 17 nM T10877 CS70GC 145969309 IC50 = 82 nM T10877 CNH7O5 145969326 IC50 = 51 nM T10877 CHZ7N3 145969706 IC50 = 42 nM T10877 CN56YO 145969928 IC50 = 330 nM T10877 C4CDN0 145969972 IC50 = 83 nM T10877 C1I3TK 145970025 IC50 = 6800 nM T10877 C6A0HJ 145970175 IC50 = 140 nM T10877 CJC43R 145970183 IC50 = 5500 nM T10877 CMKZ95 145970214 IC50 = 4200 nM T10877 CB2NU1 145970392 IC50 = 1600 nM T10877 CJR21T 145970400 IC50 = 410 nM T10877 CQ82EI 145970446 IC50 = 4300 nM T10877 CORE90 145970461 IC50 = 230 nM T10877 C4GR7E 145970630 IC50 = 71 nM T10877 CB4RP9 145970636 IC50 = 160 nM T10877 C3LD1Y 145970800 IC50 = 20 nM T10877 C7N2ZY 145970856 IC50 = 45 nM T10877 CUSO84 145970885 IC50 = 110 nM T10877 CKDZ10 145971093 IC50 = 19000 nM T10877 CW6ER8 145987053 IC50 = 4 nM T10877 CYT73F 145987735 IC50 = 2500 nM T10877 D07NAY 5281692 IC50 = 37900 nM T10877 D0E1QP 4262314 IC50 > 100000 nM T10877 D0O0VZ 667639 IC50 > 100000 nM T10877 D0T3PW 5281672 IC50 = 24800 nM T10877 D0V3PG 128861 IC50 = 21800 nM T69912 D0T9TJ 3034010 IC50 = 50 nM T69912 D05GZD 9918381 IC50 = 0.2512 nM T69912 D0CW8S 71657619 IC50 > 10000 nM T69912 D09NBM 10417440 Ki = 0.03 nM T69912 D0L5UO 9939609 IC50 = 0.035 nM T69912 CN1K3D 5699 IC50 > 100000 nM T69912 CZI2U1 6491 IC50 > 1000000 nM T69912 CYFU26 130606 IC50 > 100000 nM T69912 CZ3R1F 669158 IC50 = 1000000 nM T69912 C2KRB1 973435 IC50 = 44000 nM T69912 CMN1P8 1217803 IC50 = 3431 nM T69912 C2F7OG 2412772 IC50 = 1000000 nM T69912 C9VZ3F 3638243 IC50 > 100000 nM T69912 C1FHP8 4811752 IC50 = 14000 nM T69912 CG0F8O 9808838 IC50 = 1 nM T69912 CC5Y0A 9809899 IC50 = 533 nM T69912 C4TB5Y 9831072 IC50 = 0.6 nM T69912 C4VH8G 9840384 IC50 = 850 nM T69912 CB0EP8 9850883 IC50 = 26 nM T69912 C4R6CU 9851531 IC50 = 20 nM T69912 C89RJZ 9852438 IC50 = 0.5 nM T69912 CTJO81 9893629 IC50 = 85 nM T69912 C9FWY2 9895919 IC50 = 2 nM T69912 C6MD8O 9917136 IC50 = 8 nM T69912 C19SKN 9917325 IC50 = 0.7 nM T69912 CX23UG 9917667 IC50 = 9 nM T69912 CMBO57 9917750 IC50 = 0.4 nM T69912 CSB71L 9938151 IC50 = 18 nM T69912 CFH61N 9938577 IC50 = 26 nM T69912 CMN74S 9938642 IC50 = 12 nM T69912 CGL13H 9939495 IC50 = 0.4 nM T69912 C2EF8Q 9939518 IC50 = 2 nM T69912 CQEN19 9959703 IC50 = 24 nM T69912 C8C0HB 9961561 IC50 = 1 nM T69912 CSW8T3 9961700 IC50 = 0.3 nM T69912 C8X7KP 9961715 IC50 = 9 nM T69912 C1DB0X 10055750 IC50 = 0.17 nM T69912 C1TY3F 10122289 IC50 = 0.25 nM T69912 C0KOC5 10122452 IC50 = 3 nM T69912 C1LSI8 10122657 IC50 = 0.1 nM T69912 CJ4R2U 10168216 IC50 = 0.4 nM T69912 CAK3E1 10189993 IC50 = 0.8 nM T69912 CPG87K 10189998 IC50 = 38 nM T69912 CG65NB 10190629 IC50 = 1 nM T69912 CIK7C8 10211722 IC50 = 1.5 nM T69912 CA4EF3 10211894 IC50 = 2 nM T69912 CFQ5L2 10232552 IC50 = 5 nM T69912 CB72SI 10233112 IC50 = 1 nM T69912 C9UIX5 10233517 IC50 = 0.8 nM T69912 C61ZEV 10282620 IC50 = 1 nM T69912 CQV98P 10305047 IC50 = 0.5 nM T69912 COAR34 10305066 IC50 = 19 nM T69912 CZA96C 10305422 IC50 = 0.8 nM T69912 C7W2NF 10305573 IC50 = 1 nM T69912 C8OPC6 10305637 IC50 = 6 nM T69912 C03CJA 10320992 IC50 = 64 nM T69912 C0JB9D 10394633 IC50 = 0.7 nM T69912 CD3MH2 10411777 IC50 = 54 nM T69912 CU78FP 11521655 IC50 = 25000 nM T69912 CZRT87 11543912 IC50 = 38000 nM T69912 CJW8M7 11564757 IC50 = 26000 nM T69912 C09ASJ 11764593 IC50 = 0.2 nM T69912 CU0Y2Z 12051594 IC50 = 2 nM T69912 C6O8ID 14490158 IC50 = 1000000 nM T69912 CS5CV2 16126765 IC50 = 120 nM T69912 CGN9S6 17899989 IC50 = 640 nM T69912 CK14ET 17899991 IC50 = 210 nM T69912 C8C4LK 18470089 IC50 = 110 nM T69912 C0EU2T 18470090 IC50 = 0.3 nM T69912 C63DZQ 18470117 IC50 = 19 nM T69912 C7FV0Y 18470125 IC50 = 850 nM T69912 CRS63W 18470138 IC50 = 90 nM T69912 CJ0Q9T 18470140 IC50 = 17000 nM T69912 CFI50Y 18470152 IC50 = 34 nM T69912 C1WJ5A 18470163 IC50 = 1000 nM T69912 CZJ25E 18470168 IC50 = 19 nM T69912 CK47RM 18470169 IC50 = 200 nM T69912 C69SCV 18470191 IC50 = 4 nM T69912 C38OXW 18470208 IC50 = 1400 nM T69912 C68IDK 18470209 IC50 = 1000 nM T69912 CYF0B8 18470218 IC50 = 4400 nM T69912 C24HOS 18470241 IC50 = 2 nM T69912 C1Q8NP 18470244 IC50 = 11 nM T69912 CIEQ59 18470251 IC50 = 780 nM T69912 CE69PL 18470253 IC50 = 210 nM T69912 CP5S1M 18470258 IC50 = 650 nM T69912 C1NLE8 18470267 Ki = 41 nM T69912 CA38TG 18470272 IC50 = 430 nM T69912 C9Z0PI 18470273 IC50 = 660 nM T69912 CUTF18 18470282 IC50 = 12000 nM T69912 C9BRG5 18470283 IC50 = 250 nM T69912 CBZ1V0 18470296 IC50 = 12600 nM T69912 CT10SU 18470303 IC50 = 19 nM T69912 CJ35LB 18470304 IC50 = 4400 nM T69912 CV2Q4O 18470306 IC50 = 150 nM T69912 C2EGW7 18470314 IC50 = 16 nM T69912 C6CVW9 18470315 IC50 = 7 nM T69912 CR6S2P 18470316 IC50 = 1300 nM T69912 CT1G0Z 18470322 IC50 = 285 nM T69912 CU3QI1 18470341 IC50 = 960 nM T69912 CEIF53 18470354 IC50 = 450 nM T69912 CS93WA 18470361 IC50 = 2900 nM T69912 C0BE4O 18470368 IC50 = 110 nM T69912 CLS52M 18470371 IC50 = 1000 nM T69912 C8HNR6 18470375 IC50 = 450 nM T69912 C7VK9N 18470385 IC50 = 300 nM T69912 CX6EC7 18470390 IC50 = 250 nM T69912 C45GTM 18470395 IC50 = 0.1 nM T69912 C2EL5G 18470399 IC50 = 55000 nM T69912 C60DVF 18470400 IC50 = 1200 nM T69912 CXW4D9 18470406 IC50 = 200 nM T69912 C07FGB 18470420 IC50 = 330 nM T69912 CPE8J7 18470422 IC50 = 5700 nM T69912 CE1Y8Q 18470432 IC50 = 1400 nM T69912 CL0GA7 18470436 IC50 = 1200 nM T69912 CUA07V 18470440 IC50 = 1100 nM T69912 C0TQ3E 18470452 IC50 = 1100 nM T69912 C5GC2U 18470455 IC50 = 1 nM T69912 CHN74T 18470468 IC50 = 70 nM T69912 C15KXN 18470470 IC50 = 2 nM T69912 CLGR76 18470474 IC50 = 2300 nM T69912 C14IMQ 18470482 IC50 = 630 nM T69912 CR50VA 18470483 IC50 = 1100 nM T69912 C78SLA 18470487 IC50 = 39 nM T69912 CDY3G7 18470494 IC50 = 230 nM T69912 CMFK89 18470498 IC50 = 36 nM T69912 CPI0Y6 18470516 IC50 = 250 nM T69912 CV47NE 18470522 IC50 = 110 nM T69912 C0FYD2 18470524 IC50 = 1100 nM T69912 CG18YS 18470527 IC50 = 7 nM T69912 CI9JK7 18470549 IC50 = 14000 nM T69912 C8Y9TC 18470552 IC50 = 140 nM T69912 CE83XT 18470555 IC50 = 3300 nM T69912 CJY4G6 18470556 IC50 = 1100 nM T69912 COIL12 18470582 IC50 = 2850 nM T69912 C1QV9I 18470585 IC50 = 990 nM T69912 CB95IU 18470590 IC50 = 0.4 nM T69912 CD2G1X 18470595 IC50 = 780 nM T69912 CH63UY 18540820 IC50 = 1 nM T69912 CRC64I 18768423 IC50 = 52.4 nM T69912 CY4AF7 21936103 IC50 = 0.1 nM T69912 C4VY5P 21936114 IC50 = 4 nM T69912 CMS86P 21936124 IC50 = 0.5 nM T69912 CDT3Y6 21936140 IC50 = 0.3 nM T69912 COEI56 21936146 IC50 = 5 nM T69912 C9C3JG 21936169 IC50 = 1 nM T69912 CN5ZP0 21936176 IC50 = 1 nM T69912 C4P8MH 21936183 IC50 = 0.2 nM T69912 C8U3FQ 21936197 IC50 = 8 nM T69912 C9PUJ0 21936206 IC50 = 15 nM T69912 CMR0P1 21936209 IC50 = 5 nM T69912 CB1W0U 21936229 IC50 = 4 nM T69912 CM8NF3 21936243 IC50 = 0.8 nM T69912 CV49NU 21936282 IC50 = 0.6 nM T69912 C6JX0D 21936319 IC50 = 0.2 nM T69912 CCU98M 21936326 IC50 = 3 nM T69912 CB5M3Q 21936345 IC50 = 0.2 nM T69912 CV8QT9 21936398 IC50 = 0.2 nM T69912 C0B2MU 21936403 IC50 = 4 nM T69912 CA4X5J 21936407 IC50 = 5 nM T69912 CEC2B6 22294074 IC50 = 0.5 nM T69912 C2BJY9 23395723 IC50 = 1 nM T69912 CW7FL6 23395729 IC50 = 0.6 nM T69912 C3CZL1 23395731 IC50 = 2.7 nM T69912 C02MBF 23395732 IC50 = 17 nM T69912 CDH5N2 23395748 IC50 = 8 nM T69912 C6Y9DO 23395749 IC50 = 4 nM T69912 CH3RP0 23395766 IC50 = 2 nM T69912 C0G8KF 23395772 IC50 = 0.7 nM T69912 C79IXE 23395774 IC50 = 0.12 nM T69912 CMQ2X3 23395778 IC50 = 1 nM T69912 CH7S9G 23395784 IC50 = 1.6 nM T69912 CXP67J 23395785 IC50 = 0.6 nM T69912 CFN51M 23395786 IC50 = 4.5 nM T69912 CVM86Y 23395788 IC50 = 1.4 nM T69912 C32CYB 23395790 IC50 = 0.8 nM T69912 C8A9OF 23395792 IC50 = 2 nM T69912 C4PL8S 23395794 IC50 = 5 nM T69912 CL2CM7 23395795 IC50 = 1 nM T69912 CW9G8Y 23395798 IC50 = 5 nM T69912 CE1J3W 23395801 IC50 = 0.7 nM T69912 CNDH71 23395803 IC50 = 0.2 nM T69912 CV9H3P 23395804 IC50 = 0.12 nM T69912 CH0G9B 23395805 IC50 = 0.2 nM T69912 CUXA85 23395806 IC50 = 0.35 nM T69912 C01DHS 23395807 IC50 = 0.5 nM T69912 CU2J0M 23395808 IC50 = 0.2 nM T69912 CET9J2 23395809 IC50 = 1.5 nM T69912 C73WNR 44266749 IC50 = 50 nM T69912 C4XW9G 44266800 IC50 = 3 nM T69912 C6OWG4 44300071 IC50 = 34 nM T69912 CKU80A 44300072 IC50 = 21 nM T69912 CLU67B 44300088 IC50 = 97 nM T69912 CD41MI 44300109 IC50 = 140 nM T69912 C6LK3F 44300123 IC50 = 66 nM T69912 C4CG6Q 44300126 IC50 = 1280 nM T69912 C1HYF9 44300132 IC50 = 460 nM T69912 CJE5Y8 44300187 IC50 = 39 nM T69912 CZ6M8X 44300263 IC50 = 350 nM T69912 CHR95L 44300266 IC50 = 260 nM T69912 C72MUZ 44300268 IC50 = 51 nM T69912 CZS4T9 44300303 IC50 = 44 nM T69912 CKNC02 44300306 IC50 = 70 nM T69912 C3WJC0 44300307 IC50 = 29 nM T69912 CUB07K 44300374 IC50 = 3 nM T69912 CD02LG 44300390 IC50 = 410 nM T69912 CQ7M6U 44300414 IC50 = 89 nM T69912 C3FAV2 44300418 IC50 = 6700 nM T69912 CX56UK 44300444 IC50 = 530 nM T69912 C8HPB9 44300446 IC50 = 720 nM T69912 C34HVB 44300478 IC50 = 130 nM T69912 C01MXK 44300573 IC50 = 10 nM T69912 CI2EA3 44300574 IC50 = 69 nM T69912 CK4D5X 44300578 IC50 = 5 nM T69912 CG5HW3 44300752 IC50 = 120 nM T69912 CXQI32 44300753 IC50 = 176 nM T69912 C4ZDS7 44319598 IC50 = 235 nM T69912 CVYP89 44319686 IC50 = 12 nM T69912 CFJD61 44319860 IC50 = 350 nM T69912 CH1TP7 44319861 IC50 = 300 nM T69912 CUV80P 44319972 IC50 = 250 nM T69912 COD96J 44319974 IC50 = 25 nM T69912 CJBU28 44319998 IC50 = 260 nM T69912 CCU1J0 44320037 IC50 = 3 nM T69912 C9UZM1 44320070 IC50 = 15 nM T69912 CL2A8D 44367433 IC50 = 1.6 nM T69912 C0BM7X 44367434 IC50 = 0.5 nM T69912 C0CNE9 44367483 IC50 = 1.6 nM T69912 C8HM0C 44367519 IC50 = 0.2 nM T69912 CGS4E6 44367542 IC50 = 1.7 nM T69912 C04WGR 44367559 IC50 = 5 nM T69912 C0Q9NA 44367560 IC50 = 2.6 nM T69912 CG7AQ0 44367583 IC50 = 0.9 nM T69912 CVB27E 44367645 IC50 = 194 nM T69912 CNK0A7 44367647 IC50 = 5 nM T69912 CQ6S3B 44367648 IC50 = 24 nM T69912 CP2GU1 53299144 IC50 > 100000 nM T69912 CCR5A9 56927662 IC50 = 59 nM T69912 CAG1J5 56927666 IC50 = 23 nM T69912 C6GKE8 56950525 IC50 = 16 nM T69912 C21HQB 57336782 IC50 = 3.4 nM T69912 C5WQ8S 57392555 IC50 = 96 nM T69912 CITS38 57394279 IC50 = 170 nM T69912 CR8GA1 57396026 IC50 = 31 nM T69912 CKN4Q7 57396027 IC50 = 55 nM T69912 C83CEW 57397828 IC50 = 64 nM T69912 CX65FQ 57397830 IC50 = 92 nM T69912 C89RKP 57397831 IC50 = 56 nM T69912 CN5L8A 57397832 IC50 = 91 nM T69912 CMBI04 57397833 IC50 = 2900 nM T69912 CK2C8H 57401254 IC50 = 61 nM T69912 CN9TM3 57401255 IC50 = 130 nM T69912 C4PC1W 57402997 IC50 = 4100 nM T69912 CF23GK 57402999 IC50 = 48 nM T69912 C5SE6Y 57403000 IC50 = 360 nM T69912 CLQ5P8 59900388 IC50 = 1 nM T69912 CL0FU7 63334771 IC50 = 100000 nM T69912 C59VAN 71181474 IC50 = 0.55 nM T69912 C13KJW 71181477 IC50 = 0.23 nM T69912 CI1Y9Z 71181626 IC50 = 1.6 nM T69912 CPXJ23 71181632 IC50 = 0.96 nM T69912 CML2I0 71181668 IC50 = 0.24 nM T69912 CU8YK1 71181747 IC50 = 1.72 nM T69912 C9B7MX 71181764 IC50 = 0.91 nM T69912 CO7K5M 71181859 IC50 = 0.46 nM T69912 C1FGZ5 71181861 IC50 = 0.81 nM T69912 CBG0P3 71181874 IC50 = 0.89 nM T69912 CO0W1H 71476859 IC50 = 0.14 nM T69912 CJPF24 71486715 IC50 = 0.86 nM T69912 C9DA6W 71562486 IC50 = 14000 nM T69912 C40WLD 71562487 IC50 = 230 nM T69912 C0N4SW 71562488 IC50 = 55 nM T69912 CS41XO 71562489 IC50 = 38 nM T69912 CB8E0O 71562597 IC50 = 370 nM T69912 CU02DS 71562598 IC50 = 86000 nM T69912 CX62RJ 71562599 IC50 = 820 nM T69912 CH5GA2 71562600 IC50 = 29000 nM T69912 C2XRB6 71562601 IC50 = 32 nM T69912 CL0KT3 71562602 IC50 = 9700 nM T69912 C6N7RZ 71562603 IC50 = 100 nM T69912 CT64JI 71562727 IC50 = 150 nM T69912 C8AOX0 71562728 IC50 = 150 nM T69912 CRX2Q4 71562729 IC50 = 16 nM T69912 CMWV34 71562730 IC50 = 70 nM T69912 CU4Z2Q 71562731 IC50 = 87 nM T69912 CJU1L8 71562732 IC50 = 44 nM T69912 CQ4AN0 71562733 IC50 = 240 nM T69912 CN15BR 71562848 IC50 = 3000 nM T69912 CY37JA 71562849 IC50 = 41000 nM T69912 C7APK1 71562850 IC50 = 31 nM T69912 CA1C8N 71562851 IC50 = 26 nM T69912 C4OBN3 71562852 IC50 = 13 nM T69912 C6PQG5 71562853 IC50 = 14 nM T69912 C50DMA 71562854 IC50 = 39 nM T69912 CCK65O 71562973 IC50 = 49 nM T69912 CUW2X3 71562974 IC50 = 52 nM T69912 CU2K4F 71562975 IC50 = 120 nM T69912 C1YI9V 71562976 IC50 = 250 nM T69912 C80IKC 71562977 IC50 = 450 nM T69912 CZEX42 71562978 IC50 = 100 nM T69912 C0TQ5W 71562979 IC50 = 39 nM T69912 CO8XE5 71563093 IC50 = 26 nM T69912 C71VWC 71563094 IC50 = 4 nM T69912 C42RMU 71563095 IC50 = 55 nM T69912 CQ39RC 71563096 IC50 = 28 nM T69912 CJU20T 71563097 IC50 = 3 nM T69912 CDJ92S 71563098 IC50 = 3 nM T69912 CUO97N 71563099 IC50 = 80 nM T69912 CC3LF8 71563229 IC50 = 22 nM T69912 C6G8OV 71614098 IC50 = 0.67 nM T69912 CPQ5H2 71614498 IC50 = 0.95 nM T69912 CYO64A 71656315 IC50 > 1000 nM T69912 C50OAM 71656796 IC50 = 210 nM T69912 C2TO5C 71656797 IC50 > 10000 nM T69912 CN89IX 71656798 IC50 = 93 nM T69912 C49OFR 71656799 IC50 = 26 nM T69912 C92YGU 71657082 IC50 = 5000 nM T69912 CV5PM2 71657185 IC50 = 10000 nM T69912 CPT0H5 71657290 IC50 = 10000 nM T69912 CM2ZB8 71657292 IC50 = 810 nM T69912 CBSW63 71657395 IC50 > 10000 nM T69912 CVUD47 71657398 IC50 > 10000 nM T69912 CV24SL 71716432 IC50 = 4 nM T69912 CTH15K 71717661 IC50 = 23 nM T69912 C1AYH2 71718263 IC50 = 32 nM T69912 CTPL54 71718264 IC50 > 100000 nM T69912 CS7WK3 74889411 IC50 > 100 nM T69912 C2KHF7 89677087 IC50 = 1400 nM T69912 CXT5C7 89682527 IC50 = 1500 nM T69912 CPF01Q 89682653 IC50 = 580 nM T69912 CY7PD2 89682704 IC50 = 930 nM T69912 CNU8L7 89682719 IC50 = 1800 nM T69912 C2JS9A 119057479 IC50 = 500000 nM T69912 CZL6P8 119057480 IC50 = 230 nM T69912 C1S6CA 119057481 IC50 = 2000 nM T69912 CV8MY3 119057482 IC50 = 1700 nM T69912 CGN2X5 119057483 IC50 = 230 nM T69912 CW6T2I 121005813 IC50 = 1.7 nM T69912 CL70DK 121448333 IC50 = 8.3 nM T69912 C3N6DK 121448334 IC50 = 1.8 nM T69912 CM4S9R 121448337 IC50 = 4.2 nM T69912 C9U7WD 121448368 IC50 = 1.6 nM T69912 CI86GD 121448372 IC50 = 1.9 nM T69912 C1A5GV 121448374 IC50 = 2.2 nM T69912 CKM5Z4 121448380 IC50 = 2.7 nM T69912 CW0V2U 121448402 IC50 = 4 nM T69912 CG9H1O 121448406 IC50 = 3.7 nM T69912 CRE5L4 121448411 IC50 = 2.2 nM T69912 CF65PJ 121448417 IC50 = 2.6 nM T69912 CX1LF9 121448418 IC50 = 8 nM T69912 C3OBQ9 121448429 IC50 = 4.6 nM T69912 CJ4F7G 121448430 IC50 = 1.2 nM T69912 CZM7L3 121448431 IC50 = 3.5 nM T69912 CSCG90 121448433 IC50 = 1.8 nM T69912 C8TVD7 121448459 IC50 = 1.1 nM T69912 COU74T 121448460 IC50 = 3.9 nM T69912 CIW92J 122196130 IC50 = 11.1 nM T69912 CY4XR8 122196132 IC50 = 10.6 nM T69912 CIY90U 122196137 IC50 = 19.3 nM T69912 C5AFS0 122196138 IC50 = 16 nM T69912 C32FMN 122196204 IC50 = 13.4 nM T69912 CJGP91 122196205 IC50 = 16.9 nM T69912 CKA4Y1 122196208 IC50 = 3.7 nM T69912 CCWJ26 122196209 IC50 = 2.9 nM T69912 C9WZI8 122196212 IC50 = 2.3 nM T69912 CEL90A 122196214 IC50 = 6.5 nM T69912 CQBA39 122196215 IC50 = 10.9 nM T69912 CI3CW8 122196216 IC50 = 6.3 nM T69912 C7JU5Q 122530045 IC50 = 6300 nM T69912 C5BW4Z 122707116 IC50 = 15000 nM T69912 CX92RI 122707117 IC50 = 1600 nM T69912 C23EKP 122707118 IC50 = 1000 nM T69912 CU95PT 122707120 IC50 = 32 nM T69912 CK05FL 127050954 IC50 = 3.6 nM T69912 C8TUI5 127050955 IC50 = 2.4 nM T69912 C7DA4S 127050956 IC50 = 18 nM T69912 C01RCH 127050977 IC50 = 30000 nM T69912 CJW7D2 127051244 IC50 = 560 nM T69912 C1GSK5 127053040 IC50 = 180 nM T69912 CRC6Z1 127053472 IC50 = 1.1 nM T69912 CU0D3S 130346049 IC50 = 1400 nM T69912 CH7EL8 132427687 IC50 = 14 nM T69912 CW74SC 134133758 IC50 = 75 nM T69912 CM5R6E 134135433 IC50 = 10000 nM T69912 CYXB84 134136689 IC50 = 39000 nM T69912 CM98WH 134137624 IC50 = 7900 nM T69912 C1SP0U 134138704 IC50 = 620 nM T69912 CJG9M7 134140857 IC50 = 1500 nM T69912 CP3HL5 134143019 IC50 = 860 nM T69912 CFQ13X 134144083 IC50 = 2700 nM T69912 C1GZ9U 134145078 IC50 = 2000 nM T69912 CUV5B0 134145387 IC50 = 5400 nM T69912 CSN0D4 134146496 IC50 = 1900 nM T69912 C5YD1G 134147073 IC50 = 6200 nM T69912 C8WF9X 134147739 IC50 = 20000 nM T69912 C69BXV 134148543 IC50 = 160 nM T69912 CCE7M2 134150004 IC50 = 0.3981 nM T69912 C36ZHN 134150110 IC50 = 11000 nM T69912 CXV2M9 134150242 IC50 = 4300 nM T69912 C58MQS 134152799 IC50 = 110 nM T69912 C8MA0Z 134153116 IC50 = 980 nM T69912 CZGB70 134154962 IC50 = 160 nM T69912 CA85UF 134155224 IC50 = 86 nM T69912 C16NSU 134155260 IC50 = 660 nM T69912 CHL74N 134156788 IC50 = 10000 nM T69912 CEW49V 134157408 IC50 = 72 nM T69912 C3SVZ5 134693749 IC50 = 355 nM T69912 C3DE5Y 134693750 IC50 = 5 nM T69912 CZ3F5D 135239539 IC50 = 844 nM T69912 C0U9TO 137546866 IC50 = 430 nM T69912 CH4MR3 137633945 IC50 = 902 nM T69912 CTD75A 137633962 IC50 = 9 nM T69912 CRCU09 137634263 IC50 = 236 nM T69912 CH05MV 137636050 IC50 = 613 nM T69912 CG3K6U 137637253 IC50 = 12 nM T69912 CMNT10 137638920 IC50 = 23 nM T69912 CK70BJ 137641309 IC50 = 42 nM T69912 C6LIG7 137642017 IC50 = 222 nM T69912 CZ3F7X 137642755 IC50 = 2477 nM T69912 CJP45C 137643198 IC50 = 924 nM T69912 CS4W0J 137643921 IC50 = 13 nM T69912 CA50JV 137645485 IC50 = 1027 nM T69912 C4F5GR 137647910 IC50 = 322 nM T69912 CFL68S 137649687 IC50 = 1070 nM T69912 CL61YI 137651817 IC50 = 152 nM T69912 CX3AJ9 137652098 IC50 = 17 nM T69912 CJ73YS 137654141 IC50 = 65 nM T69912 CSR0J2 137655061 IC50 = 57 nM T69912 CGBL78 137655982 IC50 = 232 nM T69912 CTU98S 137658155 IC50 = 100 nM T69912 C9X3WS 137658880 IC50 = 1915 nM T69912 CLVM39 137660910 IC50 = 45 nM T69912 C4JV2G 137661511 IC50 = 1418 nM T69912 CO67DI 137661556 IC50 = 45 nM T69912 CEQ7G4 155510849 IC50 > 10000 nM T69912 C9CD3Q 155511585 IC50 = 430 nM T69912 C25OAR 155512542 IC50 = 2000 nM T69912 CI2WL8 155513853 IC50 > 1000 nM T69912 CBG4Q8 155521008 IC50 > 1000 nM T69912 CL6Z1R 155526799 IC50 = 750 nM T69912 CW7N6K 155533489 IC50 = 1000 nM T69912 CQ67EK 155543660 IC50 = 1800 nM T69912 C8XZ7V 155545255 IC50 = 330 nM T69912 C9WGK1 155547201 IC50 = 1300 nM T69912 CH78YM 155549832 IC50 > 1000 nM T69912 C4U9WO 155550747 IC50 = 10000 nM T69912 D05LXG 5063 IC50 = 11000 nM T69912 D09QHC 7370 IC50 > 1000000 nM T69912 D0A1SO 11206881 IC50 = 3800 nM T69912 D0D7AS 11701397 IC50 = 11200 nM T69912 D0FO2B 1923 IC50 > 100000 nM T69912 D0JI8S 11470979 IC50 = 2000 nM T69912 D0WW7A 9939109 IC50 = 8 nM T69912 D0X6UV 11368513 IC50 = 4400 nM T89826 D04AIT 5280445 IC50 = 20000 nM T89826 D07EXH 359 IC50 > 200000 nM T89826 D07MGA 72281 IC50 = 8300 nM T89826 D0J9ZR 4477 IC50 = 40000 nM T89826 D0K8KX 5280343 IC50 = 8100 nM T89826 C5H9TY 14697 IC50 = 207000 nM T89826 C3I7VB 102678 IC50 = 24500 nM T89826 CL5Y4J 159516 Ki = 3100 nM T89826 CV0B7W 442027 IC50 = 49600 nM T89826 C1E2FR 442048 IC50 = 283500 nM T89826 CZ3MD8 647122 IC50 = 16100 nM T89826 C2C8QU 948801 Ki = 27500 nM T89826 CXA4P6 1265413 IC50 = 90720 nM T89826 CUD4A1 1328543 IC50 = 58350 nM T89826 C3ZP4U 2131972 Ki = 9110 nM T89826 CA1N3H 2131982 Ki = 9930 nM T89826 CKL8B2 2219105 IC50 = 29900 nM T89826 CN43XQ 2806068 IC50 = 160 nM T89826 C5J6MO 2849659 IC50 = 28800 nM T89826 CN3P7A 2911959 IC50 = 74500 nM T89826 CZDG23 2947583 IC50 = 186000 nM T89826 CBIP72 2986413 IC50 = 76700 nM T89826 CCU3P7 3635406 IC50 = 2200 nM T89826 CZF0R5 4004950 IC50 = 500 nM T89826 C3AN7C 4117477 IC50 = 1180 nM T89826 CS2WB7 4236803 IC50 = 29800 nM T89826 C0AW3N 4378077 IC50 = 13860 nM T89826 CO3Y0T 4614896 IC50 = 9910 nM T89826 CY68ZT 4788586 IC50 = 940 nM T89826 CTR4Q1 5320532 IC50 = 13300 nM T89826 CVG47I 5958938 IC50 = 10500 nM T89826 CD8ZT2 6026688 IC50 > 50000 nM T89826 C3LZX9 8027611 IC50 = 12660 nM T89826 CJ4C5K 9180583 IC50 = 10800 nM T89826 CYQ8Z4 9882716 IC50 > 50000 nM T89826 C8K2NO 10062715 IC50 = 800000 nM T89826 C49CMU 10411574 IC50 = 21700 nM T89826 C6GN2F 11642725 IC50 = 870000 nM T89826 CHYP53 12310492 IC50 = 233400 nM T89826 C65EOH 15949840 IC50 = 7500 nM T89826 C9V8EM 15956553 IC50 = 300000 nM T89826 C3WYR4 16061499 IC50 = 2000 nM T89826 CTO43V 16085283 Ki = 116000 nM T89826 CU35DQ 21582568 IC50 = 220800 nM T89826 CN45FL 23427055 IC50 = 164700 nM T89826 CK3AF8 25256829 IC50 = 5400 nM T89826 C2SZ7L 42624533 IC50 = 14000 nM T89826 CYP8V1 44404067 IC50 > 50000 nM T89826 CD20PF 44433696 IC50 = 80000 nM T89826 CI4P2V 44433697 IC50 = 10000 nM T89826 CW7B0J 44433698 IC50 = 15000 nM T89826 C8DWL3 44433699 IC50 = 200000 nM T89826 C0ZPE2 44517748 IC50 = 2700 nM T89826 C0OH2T 44584893 IC50 = 5400 nM T89826 C0NZ5E 44584944 IC50 = 7300 nM T89826 CT70DZ 44590821 IC50 = 22500 nM T89826 C0SW2K 45266425 IC50 = 2500 nM T89826 C5WBP2 45266482 IC50 = 3800 nM T89826 CA4K8F 45266488 IC50 = 6600 nM T89826 C3BHZ4 45268445 IC50 > 50000 nM T89826 CC05NI 45268452 IC50 = 15400 nM T89826 C6QD9E 45269292 IC50 > 50000 nM T89826 CY7RV4 45269761 Ki = 21000 nM T89826 CO80TH 45269762 Ki = 297000 nM T89826 CU34ZK 45269763 Ki = 584000 nM T89826 C9P3LZ 45269764 Ki = 478000 nM T89826 CXS19V 45269765 Ki = 45200 nM T89826 C3DY4T 45270971 IC50 > 50000 nM T89826 CR4WA8 45270979 IC50 = 20900 nM T89826 CM78GO 45271412 Ki = 462000 nM T89826 CC90BU 45271826 IC50 = 5200 nM T89826 C0B6KX 45271831 IC50 = 9300 nM T89826 CN85IQ 45271832 IC50 = 8100 nM T89826 C7IF2O 45272299 Ki = 363000 nM T89826 CZRV73 45272304 Ki = 34100 nM T89826 CGV14L 45272305 Ki = 112000 nM T89826 CVTL97 45272306 Ki = 2200 nM T89826 CAM89I 45273174 Ki = 135000 nM T89826 CZT67B 45273179 Ki = 614000 nM T89826 CHF4M5 45273180 Ki = 49300 nM T89826 CND1R3 45273184 Ki = 159000 nM T89826 C0V5WT 45273625 IC50 > 50000 nM T89826 C6OE7V 46784066 IC50 = 28300 nM T89826 C6LH5I 46881919 Ki = 800 nM T89826 CI2FO1 49870840 IC50 = 5500 nM T89826 CF2D0I 49870841 IC50 = 8400 nM T89826 CM52SZ 49870842 IC50 = 6800 nM T89826 C8Q2CZ 50885062 IC50 > 50000 nM T89826 CJ6KV7 52941131 IC50 = 13900 nM T89826 C8M2QD 52943127 IC50 = 24300 nM T89826 CQ84MD 52945913 IC50 = 12000 nM T89826 CJ1LG2 52945915 IC50 = 42000 nM T89826 CZ35DX 52945977 IC50 = 128900 nM T89826 CAB1Y3 52946772 IC50 = 163200 nM T89826 CO4R1B 52947200 IC50 = 18000 nM T89826 CC4X1O 52948928 IC50 = 137700 nM T89826 CMG4U7 52949213 IC50 = 10800 nM T89826 C0X5BL 58589722 IC50 = 76740 nM T89826 CY3CL6 71544384 IC50 = 610 nM T89826 CV3P2U 71544385 IC50 = 230 nM T89826 CJS60O 71571220 IC50 = 49000 nM T89826 C1AY0M 71571221 IC50 = 49000 nM T89826 CY21XB 71571222 IC50 = 4600 nM T89826 C1DX9H 71571223 IC50 = 39000 nM T89826 CKE2C3 73056463 IC50 > 100000 nM T89826 C9S8ZH 73056464 IC50 > 100000 nM T89826 CK9OI0 73056465 IC50 = 31710 nM T89826 C4D8LK 73056466 IC50 = 32080 nM T89826 CRY86G 73056467 IC50 = 34910 nM T89826 C3VS4F 73056760 IC50 = 10070 nM T89826 CYH1F4 73056761 IC50 = 51330 nM T89826 C2CRZ8 73056762 IC50 = 2250 nM T89826 CD4YR3 73056763 IC50 = 11830 nM T89826 C3P2OZ 73056764 IC50 = 67200 nM T89826 C1H8PX 73056765 IC50 = 82910 nM T89826 C8JO7B 73056766 IC50 = 13860 nM T89826 CCYE63 73057087 IC50 = 5520 nM T89826 C54JWM 73057088 IC50 = 39870 nM T89826 C8RBU6 73057089 IC50 = 1040 nM T89826 CEBH65 73057090 IC50 = 1690 nM T89826 C8M2DX 73057091 IC50 = 17820 nM T89826 CQ42AZ 73057092 IC50 = 2820 nM T89826 CPLJ64 73057388 IC50 = 4700 nM T89826 CIN5V0 76320984 IC50 = 4300 nM T89826 C05AYV 102341658 IC50 = 16400 nM T89826 C8S3CR 102341659 IC50 = 37500 nM T89826 C2G9CP 127043455 IC50 = 20200 nM T89826 CVZ4I3 127043641 IC50 = 6000 nM T89826 C7BST4 127043642 IC50 = 5800 nM T89826 CGO01F 127043643 IC50 > 50000 nM T89826 C2TU5A 127043644 IC50 = 6400 nM T89826 C0Y9IT 127043645 IC50 = 41200 nM T89826 CF3B1Z 127045220 IC50 = 11700 nM T89826 CIXJ94 127045221 IC50 = 8600 nM T89826 CQ1CT5 127045222 IC50 = 18700 nM T89826 CKRX04 127045227 IC50 = 30700 nM T89826 CDZ2E1 127045228 IC50 > 50000 nM T89826 CG3E9B 127045229 IC50 = 6700 nM T89826 CG6VR3 127045386 IC50 = 15700 nM T89826 CK9JE3 127045387 IC50 > 50000 nM T89826 CY1E4Z 127045392 IC50 > 50000 nM T89826 CK5PA4 127045393 IC50 = 44700 nM T89826 C34TWD 127045394 IC50 > 50000 nM T89826 C97MQC 127048409 IC50 = 20000 nM T89826 C41VRM 127048410 IC50 = 7500 nM T89826 CZ0B1R 127052510 IC50 = 10000 nM T89826 CRW05E 127052511 IC50 > 50000 nM T89826 CC3TX0 127052512 Ki = 72000 nM T89826 CIQ1U9 127052513 Ki = 41000 nM T89826 CI13JZ 135452883 IC50 = 10000 nM T89826 CG1KW5 135470831 IC50 = 77090 nM T89826 CH4Q6A 145964401 IC50 = 5500 nM T89826 CHU61S 145964420 IC50 = 42100 nM T89826 C6YCA8 145964710 IC50 = 28800 nM T89826 CV6F7L 145966788 IC50 = 2100 nM T89826 CBWX17 145967285 IC50 = 4300 nM T89826 COR9X3 145972736 IC50 = 3900 nM T89826 CQ0M2X 145972809 IC50 = 4100 nM T89826 CF95RZ 145972878 IC50 = 3200 nM T89826 CXI0D1 145975081 IC50 = 6300 nM T89826 CG84ZR 145975487 IC50 = 5100 nM T89826 C91FOT 145976006 IC50 = 5200 nM T89826 C3F4UH 145978039 IC50 = 8800 nM T89826 CL7FB0 2919450 IC50 = 62790 nM T89826 D00RIX 5280443 IC50 = 280800 nM T89826 D01XMM 4117383 IC50 = 4450 nM T89826 D08MZY 145937 Ki = 8200 nM T89826 D08UYP 3008868 Ki = 2400 nM T89826 D09BUG 10207 IC50 = 132000 nM T89826 D0L7AT 10480940 Ki = 19300 nM T89826 D0S0BN 130976 Ki = 10600 nM T89826 D0SY2M 5281708 IC50 = 105000 nM T89826 D0UQ6U 10569 IC50 = 189100 nM T89826 D0WA9S 10429214 IC50 = 146500 nM T90961 C3VRO9 44557921 IC50 > 10000 nM T90961 C67OJG 44588117 Ki = 4400 nM T90961 C4YWO9 134812845 Ki = 17 nM T90961 CG15PY 134812846 Ki > 100000 nM T90961 C9O8CQ 137348448 Ki = 13 nM T90961 C63TGO 137349551 Ki = 17 nM T90961 C6I5ME 137349552 Ki = 19 nM T90961 CRC8D2 155489850 Ki = 95000 nM T90961 CG8J5X 155518911 Ki = 27 nM T90961 CAN08J 155534113 Ki = 36 nM T90961 C16JRL 155535406 Ki = 74 nM T90961 C3XR8O 155536206 Ki = 51 nM T90961 CX68YN 155541385 Ki > 100000 nM T90961 CWU67H 155543077 Ki = 59 nM T90961 CD8K3O 155543384 Ki = 42 nM T90961 CUTW39 155546618 Ki = 20 nM T90961 C4E0HB 155546757 Ki = 120 nM T90961 C49UVQ 155547733 Ki = 17 nM T90961 CI2J4O 155551330 Ki = 37 nM T90961 CP2K8O 155554487 Ki = 30 nM T90961 CS8MC1 155562025 Ki = 33 nM T90961 C8UW4P 155562878 Ki = 17 nM T90961 CDP94M 155569521 Ki = 53 nM T88806 D0BN9X 60947 IC50 > 300000 nM T88806 D01TJY 53340771 IC50 = 7.7 nM T88806 D09ZXO 176873 IC50 = 13.2 nM T88806 D0Q5LF 9961766 IC50 > 100000 nM T88806 D08LIG 153986 IC50 > 3 nM T88806 D0P8JX 177831 IC50 > 5 nM T88806 C7CL3Y 107775 IC50 = 2200 nM T88806 CE19HD 132605 IC50 = 27000 nM T88806 CDOC86 303776 IC50 > 1000 nM T88806 C4U0BM 1878893 IC50 > 20000 nM T88806 C2E9ZX 3080994 IC50 = 1546000 nM T88806 C42AWQ 3797164 IC50 = 20500 nM T88806 CI51MD 9807891 IC50 > 500000 nM T88806 C68UYS 9808123 IC50 = 64 nM T88806 CK6A0I 9808598 IC50 > 500000 nM T88806 CB8GP1 9828375 IC50 = 26 nM T88806 CJ9HV0 9828819 IC50 = 20 nM T88806 C1OP9I 9828979 EC50 > 100000 nM T88806 C87ADQ 9830626 IC50 = 421 nM T88806 C13KPA 9848051 Ki < 10000 nM T88806 C04PAT 9849697 IC50 > 500000 nM T88806 CTM7V0 9851337 IC50 = 316 nM T88806 C2XD7P 9851886 IC50 > 100000 nM T88806 CN1R0K 9852055 IC50 > 500000 nM T88806 CR38MP 9853559 IC50 = 2200 nM T88806 C6E3OL 9863046 IC50 > 100000 nM T88806 C2ZAK6 9870468 IC50 > 800000 nM T88806 CHC56Q 9870640 IC50 = 640 nM T88806 C5EJN9 9884317 IC50 > 20000 nM T88806 CV4T6H 9885053 IC50 = 7800 nM T88806 CME97S 9894966 IC50 = 930 nM T88806 C04INH 9895205 IC50 > 100000 nM T88806 CNX29T 9907082 IC50 = 70000 nM T88806 C9QN4D 9919094 IC50 = 1100000 nM T88806 CF4J2Z 9923982 IC50 = 15000 nM T88806 CUBV32 9924032 IC50 > 20000 nM T88806 CCPD70 9927009 IC50 = 180000 nM T88806 CDU79H 9957105 IC50 = 95 nM T88806 C2R7TW 10069591 IC50 > 500000 nM T88806 C71AIN 10077862 IC50 > 30000 nM T88806 CO8D9C 10196873 IC50 = 133 nM T88806 C7U5CM 10336795 IC50 = 8000 nM T88806 C0IA8K 10455265 IC50 > 450000 nM T88806 CTZC60 10461016 IC50 > 100000 nM T88806 CY1JM2 11024622 IC50 = 1300000 nM T88806 CZO3H7 11399588 IC50 = 3.7 nM T88806 CX9G5B 11534748 IC50 = 25 nM T88806 CFZ2O9 11613998 IC50 = 1.6 nM T88806 CD87UQ 11627754 IC50 = 286 nM T88806 CXA2U4 11671832 IC50 = 670 nM T88806 CWU71P 11699824 IC50 = 15 nM T88806 CGU84F 11721315 IC50 = 1.7 nM T88806 C2ONX6 11721442 IC50 = 6 nM T88806 CT4D1K 11799915 IC50 > 100000 nM T88806 CS24BW 11973730 IC50 > 10000 nM T88806 CZTJ02 12795460 EC50 = 1031 nM T88806 CW41XZ 16663331 IC50 > 10000 nM T88806 CDUC32 16665100 IC50 = 2.5 nM T88806 CTGC60 16678135 IC50 = 2.3 nM T88806 C4T7ZE 16724119 IC50 = 1500 nM T88806 CU8YQ3 16756502 IC50 = 1.1 nM T88806 C9LF8T 16756503 IC50 = 445 nM T88806 CJUK37 16756504 IC50 = 155 nM T88806 C0KW3V 16756505 IC50 = 3.5 nM T88806 C04JOX 16756621 IC50 = 0.54 nM T88806 C4CU7T 16756622 IC50 = 0.55 nM T88806 CFH96E 16756623 IC50 = 0.8 nM T88806 CXK79J 16756847 IC50 = 231 nM T88806 CB15RX 16756849 IC50 = 86 nM T88806 CM18ZN 16756955 IC50 = 1.4 nM T88806 CL38IU 16756956 IC50 = 0.9 nM T88806 CW5P8L 16756957 IC50 = 0.55 nM T88806 CX6AR9 23627460 IC50 = 2 nM T88806 CAVY89 23636144 IC50 > 10000 nM T88806 C1VUH4 23636254 IC50 > 10000 nM T88806 C6LR7V 23636255 IC50 > 10000 nM T88806 C5MSF6 23636502 IC50 > 10000 nM T88806 CYND24 23729562 IC50 > 20000 nM T88806 C96PUZ 23729563 IC50 > 20000 nM T88806 CZ17YE 23731146 IC50 = 3900 nM T88806 CHXT18 23731243 IC50 = 4300 nM T88806 CEA9Z8 23731244 IC50 = 1200 nM T88806 CNK5O6 23731245 IC50 > 20000 nM T88806 C6W9OS 23731246 IC50 = 20000 nM T88806 C79OBD 24864541 IC50 = 82 nM T88806 CR72IF 24864718 IC50 = 11 nM T88806 CFRX87 24864719 IC50 = 710 nM T88806 C9L0QD 24864721 IC50 < 1 nM T88806 CXH2G0 24864898 IC50 < 1 nM T88806 CF23RY 24865076 IC50 = 8 nM T88806 CO3I0M 24865264 IC50 = 69 nM T88806 CPD30N 24865443 IC50 = 480 nM T88806 C17IUE 24865620 IC50 = 8 nM T88806 C7TPO5 24865624 IC50 = 2 nM T88806 C5DVB6 24865625 IC50 = 3 nM T88806 C5DYT6 24865999 IC50 = 24 nM T88806 C5JB3F 24866187 IC50 = 220 nM T88806 C8G2FE 24866358 IC50 = 2 nM T88806 C6I1OF 24866515 IC50 < 1 nM T88806 CZ7QL8 24866516 IC50 = 90 nM T88806 CNCH18 24866519 IC50 = 3 nM T88806 CY6WR2 24872066 IC50 = 2.1 nM T88806 CUM4E3 24872070 IC50 = 2 nM T88806 CG09DH 24872646 IC50 = 1.6 nM T88806 CRS65Q 24873110 IC50 = 2.2 nM T88806 C0HZ7E 24873345 IC50 = 2.7 nM T88806 C28KAH 24873465 IC50 = 43 nM T88806 C1PB6T 25025343 IC50 = 12 nM T88806 CDA2B9 25025730 IC50 = 130 nM T88806 CD2L7Z 25025937 IC50 < 1 nM T88806 C43TCR 25183860 IC50 = 5 nM T88806 CR92LD 25184415 IC50 = 7 nM T88806 C3J7GQ 28510125 IC50 = 136 nM T88806 CLX6T9 28510811 IC50 > 1000 nM T88806 C2SLU4 44286634 IC50 = 3100000 nM T88806 C7B6FS 44286652 IC50 = 65000 nM T88806 C47DUX 44320508 IC50 = 1000000 nM T88806 CX46NY 44343237 IC50 = 6100 nM T88806 C08QPE 44350169 IC50 = 3000 nM T88806 CELV48 44350342 IC50 = 0.18 nM T88806 CP4R1A 44350344 IC50 = 230 nM T88806 C14OBS 44350379 IC50 = 2700 nM T88806 CDE56C 44350392 IC50 = 18 nM T88806 C0W9CT 44350404 IC50 = 1500 nM T88806 CEP6G1 44350415 IC50 = 0.39 nM T88806 CR83VC 44350419 IC50 = 670 nM T88806 CX3MK8 44350425 IC50 = 4700 nM T88806 C4U0XW 44350427 IC50 = 310 nM T88806 CJ47ZT 44350428 IC50 = 13 nM T88806 CX09AV 44350435 IC50 = 1800 nM T88806 CX28UF 44350441 IC50 = 170 nM T88806 C7J9NH 44350447 IC50 = 21 nM T88806 CH6UX8 44350448 IC50 = 14 nM T88806 C4C2PF 44350449 IC50 = 39 nM T88806 CP4TD3 44350450 IC50 = 1.4 nM T88806 CR51ID 44378699 IC50 = 6000 nM T88806 CAO29R 44378701 IC50 = 100 nM T88806 CWP41H 44378720 IC50 = 4300 nM T88806 C2U6ZA 44378747 IC50 = 2100 nM T88806 CT9H2B 44378748 IC50 = 4500 nM T88806 CNS75M 44378858 IC50 = 830 nM T88806 CENU52 44378961 IC50 = 4300 nM T88806 C3UQT1 44378995 IC50 = 1560 nM T88806 CHC7N5 44379066 IC50 = 1200 nM T88806 CVYB52 44393453 IC50 > 20000 nM T88806 CAD12L 44393517 IC50 > 1000 nM T88806 C6G7RF 44436701 IC50 > 1000000 nM T88806 CZ1L9O 44436703 IC50 > 1000000 nM T88806 C7CAJ3 44436705 IC50 > 1000000 nM T88806 CR6XE2 44436707 IC50 = 18 nM T88806 CYOC34 44436708 IC50 > 1000000 nM T88806 CSF3V2 44436709 IC50 > 1000000 nM T88806 C67VHW 44436710 IC50 > 1000000 nM T88806 CBW09N 44436711 IC50 > 1000000 nM T88806 CRNQ31 44436712 IC50 > 1000000 nM T88806 C1YMJ2 44436713 IC50 = 170 nM T88806 CF4UR2 44436714 IC50 > 1000000 nM T88806 C52DMG 44436715 IC50 > 1000000 nM T88806 CLU84X 44436716 IC50 = 35100 nM T88806 CRO80K 44436717 IC50 = 57 nM T88806 CVGW76 44549110 IC50 = 0.3 nM T88806 CWL7J1 44549224 IC50 = 0.7 nM T88806 CO8EM6 44550577 IC50 = 0.1 nM T88806 CX1C4T 44552445 IC50 = 151.6 nM T88806 CCFW92 44605870 IC50 = 220 nM T88806 CM9VI1 44626482 IC50 = 1300 nM T88806 CBO95I 44626483 IC50 > 100000 nM T88806 CS36GK 44627949 IC50 = 520 nM T88806 CX6LM3 44628051 IC50 = 24 nM T88806 CVTO84 44628052 IC50 = 4700 nM T88806 CJQ37N 44628053 IC50 > 100000 nM T88806 CV4P3J 44628054 IC50 > 100000 nM T88806 CTU9W0 44628055 IC50 > 100000 nM T88806 C89ZFA 46224777 IC50 = 0.92 nM T88806 C5X1NZ 46224858 IC50 = 0.9 nM T88806 CDG6B1 46224859 IC50 = 351 nM T88806 CKM2X1 46224860 IC50 = 70 nM T88806 CL39GY 46224861 IC50 = 234 nM T88806 C56PVC 46226894 IC50 = 1.6 nM T88806 CVXH79 46226896 IC50 = 1.6 nM T88806 CBKZ57 46226897 IC50 = 1.5 nM T88806 C30JXH 46226899 IC50 = 13 nM T88806 C2WHK1 46226900 IC50 = 46 nM T88806 C5H9YT 46226901 IC50 = 65 nM T88806 CV8W7P 46226902 IC50 = 887 nM T88806 C83EWD 46226903 IC50 = 79 nM T88806 CRVU54 46226904 IC50 = 87 nM T88806 CE85AX 46226905 IC50 = 6.1 nM T88806 CP7U9T 50907449 IC50 = 19 nM T88806 CK7ZI0 56838719 IC50 = 1050 nM T88806 CG2NY0 57819421 IC50 = 466 nM T88806 CEG3V7 59665282 IC50 = 5900 nM T88806 C5MA9U 59665328 IC50 < 41 nM T88806 CR71ZG 59665343 IC50 = 150 nM T88806 CJ84CU 59665347 IC50 = 83 nM T88806 CTP16I 59665394 IC50 = 76 nM T88806 C5DJB3 59665402 IC50 = 140 nM T88806 C60EVZ 59665407 IC50 = 3 nM T88806 C4UH8X 59665418 IC50 = 6 nM T88806 C5RDW1 59665480 IC50 < 1 nM T88806 CSRE10 59665495 IC50 = 49 nM T88806 C1C0UT 68898764 IC50 = 21 nM T88806 CN93KB 68898863 IC50 = 39 nM T88806 CD10PM 68899361 IC50 = 9 nM T88806 CBF0K8 68899684 IC50 = 1900 nM T88806 C9LB1Y 68900219 IC50 = 1 nM T88806 C74UPO 68900657 IC50 = 9 nM T88806 CD4N6F 68901257 IC50 = 180 nM T88806 CK8UT9 68901290 IC50 = 110 nM T88806 CF4BZ9 68901306 IC50 = 1 nM T88806 CI0AL7 69244056 IC50 = 4 nM T88806 C31IUF 69863577 IC50 = 2807 nM T88806 CPF6S0 70681588 IC50 = 890 nM T88806 CQ4G2O 70683715 IC50 = 5 nM T88806 CVCJ03 70687988 IC50 = 2200 nM T88806 CX73MA 70689988 IC50 = 130 nM T88806 C92FXR 70690012 IC50 = 150 nM T88806 CPA07E 70694227 IC50 = 360 nM T88806 C8NZ7A 70694228 IC50 = 1 nM T88806 CM2AD4 70696326 IC50 < 1 nM T88806 C48NIF 70696327 IC50 = 970 nM T88806 CGMR28 71450831 IC50 = 1200 nM T88806 C8EM7Y 71550913 IC50 = 126.5 nM T88806 CY1MD5 71574157 IC50 = 7.3 nM T88806 C02ZBI 71574158 IC50 = 111 nM T88806 C16JKI 71574159 IC50 = 7 nM T88806 CU95LC 71574160 IC50 = 94 nM T88806 COJ8Y4 71574161 IC50 = 8.7 nM T88806 C5SG9H 71574261 IC50 = 115 nM T88806 C3C9QK 71574262 IC50 = 92 nM T88806 CTZU49 71574263 IC50 = 11 nM T88806 C4HB7F 71574264 IC50 = 39 nM T88806 C3S9QJ 71574355 IC50 = 72 nM T88806 C8V4UB 71574356 IC50 = 5.5 nM T88806 CX0SQ1 71574452 IC50 = 8.7 nM T88806 C1QE0K 71716365 IC50 = 197 nM T88806 CFYM81 71720633 IC50 = 27 nM T88806 CA9K6E 72204688 IC50 = 19 nM T88806 CLC7R0 72204689 IC50 = 9800 nM T88806 CCW43J 72204873 IC50 = 2100 nM T88806 CQ6TF8 72204875 IC50 = 9800 nM T88806 CC49AN 72204878 IC50 > 100000 nM T88806 C0N3SX 72205060 IC50 = 170 nM T88806 CZ2P8U 73345565 IC50 = 6600 nM T88806 CQAE56 73345568 IC50 > 10000 nM T88806 CU1VZ5 73345570 IC50 = 6400 nM T88806 CPT7S8 73345576 IC50 > 10000 nM T88806 C4P3JC 73346588 IC50 = 3650 nM T88806 CZ6Y9R 73347081 IC50 = 4190 nM T88806 CZ35TD 73347085 IC50 = 440 nM T88806 CGM9F7 73347087 IC50 = 7720 nM T88806 C89ENA 73347090 IC50 = 6800 nM T88806 CN1A2D 73347092 IC50 = 5190 nM T88806 CO9L2V 73348591 IC50 = 6240 nM T88806 C43LWV 73348592 IC50 = 1810 nM T88806 CM37AE 73348593 IC50 = 7200 nM T88806 C5BQ6R 73349139 IC50 = 57 nM T88806 CQ5D7B 73350175 IC50 = 870 nM T88806 CJEH13 73350177 IC50 = 6800 nM T88806 C20AJB 73350179 IC50 = 10000 nM T88806 C19PJE 73350181 IC50 = 4790 nM T88806 C2F3YZ 73351673 IC50 = 9200 nM T88806 CJA25I 73351674 IC50 = 2300 nM T88806 C6NCQ1 73351675 IC50 = 440 nM T88806 C46ULG 73351676 IC50 = 10000 nM T88806 C8B6NV 73351677 IC50 = 5100 nM T88806 CIYV49 73351678 IC50 = 1500 nM T88806 C20FGN 73353141 IC50 = 8700 nM T88806 CP6AJ3 73353143 IC50 = 8500 nM T88806 CUPR57 73353147 IC50 = 1200 nM T88806 C83RAM 73353150 IC50 = 8200 nM T88806 CAJ27W 73354663 IC50 = 7720 nM T88806 CT4A5S 73354664 IC50 = 4700 nM T88806 C6XTP9 73354667 IC50 > 10000 nM T88806 CZ1BL4 73354668 IC50 = 1230 nM T88806 C4EJK0 73356213 IC50 = 980 nM T88806 CH8G5C 73356216 IC50 > 10000 nM T88806 CPG36Q 73356217 IC50 = 6000 nM T88806 CD1S3N 73356221 IC50 = 840 nM T88806 C5ALQ2 76285468 IC50 = 74 nM T88806 CI07FE 90645591 IC50 = 66000 nM T88806 C8N6OE 90654504 IC50 = 108 nM T88806 C8TWH9 90654505 IC50 > 10000 nM T88806 CDVB75 90654506 IC50 > 10000 nM T88806 C5HG9N 90654507 IC50 = 64.2 nM T88806 CLCN89 117977916 IC50 = 63 nM T88806 CJO3B6 117978172 IC50 > 10000 nM T88806 C7ANO1 118709464 IC50 = 0.39 nM T88806 CY1IS6 118718872 IC50 = 10000 nM T88806 CV7DK0 122181680 IC50 > 1000 nM T88806 CWY3V2 122181682 IC50 > 1000 nM T88806 CRG07Q 124155531 IC50 > 10000 nM T88806 C69XPN 124163720 IC50 > 10000 nM T88806 C4R3BT 124163838 IC50 = 3200 nM T88806 CS2QR4 124163840 IC50 = 3200 nM T88806 C93HFX 127025140 IC50 = 15 nM T88806 CEU4X3 127025441 IC50 = 26 nM T88806 CTX71B 127025442 IC50 = 1500 nM T88806 C21ACR 133633869 IC50 > 1000 nM T88806 CPU86F 135438774 IC50 > 20000 nM T88806 C3JVT0 136152923 IC50 > 20000 nM T88806 C85WBP 137634338 IC50 = 95.8 nM T88806 C4IX7Z 137649002 IC50 = 30.7 nM T88806 C6NVW5 137652892 IC50 = 101.3 nM T88806 C0X8ER 145949722 IC50 = 20 nM T88806 C2MO7K 145951845 IC50 = 13 nM T88806 CG80FB 145951878 IC50 = 48 nM T88806 C1P0NL 145952828 IC50 = 22 nM T88806 CJA7N9 145953608 IC50 = 41 nM T88806 CZ4SK6 145954275 IC50 = 18 nM T88806 CTA08K 145956036 IC50 = 76 nM T88806 CY5I1O 145956101 IC50 = 45 nM T88806 C8RAG3 145956154 IC50 = 36 nM T88806 CCB51L 145956802 IC50 = 40 nM T88806 CTS5R3 145959048 IC50 = 28 nM T88806 CQ4ET5 145959752 IC50 = 31 nM T88806 CO0W4J 145961652 IC50 = 22 nM T88806 C23HZY 145971531 IC50 = 22 nM T88806 C75GFR 154734316 IC50 = 158 nM T88806 CR9DN2 154734318 EC50 = 9.9 nM T88806 C8ZUJ5 154734319 IC50 = 41.5 nM T88806 C17RZG 155515221 IC50 = 547 nM T88806 CHT1J6 155515540 IC50 = 72.9 nM T88806 CQ5C4M 155516533 IC50 = 689 nM T88806 CQNC74 155517321 IC50 > 10000 nM T88806 CRIA18 155519034 IC50 > 10000 nM T88806 C3S2YZ 155519712 IC50 = 563 nM T88806 CZY8F6 155520344 IC50 = 325 nM T88806 C9HB1M 155526953 IC50 = 5669 nM T88806 C2GJ5V 155527654 IC50 = 835 nM T88806 CQ1G0D 155528127 IC50 = 419 nM T88806 C2GSD7 155528224 IC50 = 3660 nM T88806 CPIL79 155528977 IC50 = 2722 nM T88806 C58JIQ 155530986 IC50 = 1.92 nM T88806 CJZU81 155532583 IC50 = 9287 nM T88806 C9T6SE 155533508 IC50 = 983 nM T88806 CJ7O2X 155534687 IC50 > 1000 nM T88806 C6TCP5 155546837 IC50 = 409 nM T88806 C6D2SM 155550380 IC50 > 10000 nM T88806 CWF98D 155552156 IC50 > 1000 nM T88806 CC64PJ 155561080 IC50 = 8029 nM T88806 C80PGY 155563043 IC50 = 5944 nM T88806 CEF3T8 155563936 IC50 = 38.4 nM T88806 C0SZJ1 155564443 IC50 = 1110 nM T88806 C98UME 155566748 IC50 = 2161 nM T88806 CY8S2L 155569251 IC50 = 11.9 nM T88806 C9NH4F 155569254 IC50 = 154 nM T88806 CZ9D2V 90645090 EC50 = 12 nM T88806 CWA6N4 90645092 EC50 = 763 nM T88806 CA8W7Q 90645094 EC50 = 365 nM T88806 D01AXA 11764797 IC50 = 259000 nM T88806 D06LUT 44379110 IC50 = 3440 nM T88806 D07WDB 104802 IC50 = 830000 nM T88806 D0A0KS 9851104 IC50 = 34700 nM T88806 D0B4JU 15409414 IC50 = 740 nM T20251 D00FGR 3599 IC50 > 100000 nM T20251 D00JAU 3749 IC50 = 194984.46 nM T20251 D00JVR 2267 IC50 = 100 nM T20251 D00KHM 16362 IC50 = 3.02 nM T20251 D00PEH 135449332 IC50 = 630.96 nM T20251 D00SBN 4746 IC50 = 7762.47 nM T20251 D00STL 644241 IC50 = 125.89 nM T20251 D00UVA 11556711 IC50 = 92100 nM T20251 D00UYE 4058 IC50 = 323.59 nM T20251 D00YLW 3033818 IC50 = 6025.6 nM T20251 D01AXB 60835 IC50 = 10000 nM T20251 D01AZG 5073 IC50 = 148 nM T20251 D01FGR 3100 IC50 = 2570.4 nM T20251 D01KPV 3348 IC50 = 21379.62 nM T20251 D01UTL 2995 IC50 = 1380.38 nM T20251 D01ZII 2726 IC50 = 1470 nM T20251 D01ZSO 4235 IC50 = 79432.82 nM T20251 D02EYG 10096344 IC50 > 30000 nM T20251 D02KOF 3948 IC50 = 2398832.92 nM T20251 D02MLW 60753 IC50 = 20 nM T20251 D02YIZ 12560 IC50 = 39 nM T20251 D03CJL 3168 IC50 = 32.2 nM T20251 D03CQE 5379 IC50 = 128824.96 nM T20251 D03DAP 3356 IC50 = 3890.45 nM T20251 D03DIG 5284371 IC50 = 301995.17 nM T20251 D03FLC 3878 IC50 = 251188.64 nM T20251 D03HFG 5324346 IC50 = 3100 nM T20251 D03IGH 213039 IC50 = 100000 nM T20251 D03MIR 3157 IC50 = 588.84 nM T20251 D03NHW 4583 IC50 = 1412537.54 nM T20251 D03QWT 73303 IC50 = 5011872.34 nM T20251 D04AAN 4078 IC50 = 320 nM T20251 D04CRN 54841 IC50 = 2100 nM T20251 D04FVU 6337614 IC50 = 1995.26 nM T20251 D04JCN 47811 IC50 = 120.23 nM T20251 D04JEE 4946 IC50 = 2828 nM T20251 D04LVK 57379345 IC50 = 1250 nM T20251 D04MSM 2554 IC50 = 104712.85 nM T20251 D04OSE 4485 IC50 = 50118.72 nM T20251 D04XGT 31593 IC50 > 100000 nM T20251 D04XPW 446220 IC50 = 4.4 nM T20251 D05CPV 208898 IC50 = 3000 nM T20251 D05EAM 4735 IC50 = 18800 nM T20251 D05LYX 3488 IC50 = 74000 nM T20251 D05MQK 110635 IC50 = 79432.82 nM T20251 D05OFX 219078 IC50 = 50118723.36 nM T20251 D05PIZ 15130 IC50 = 2187.76 nM T20251 D05SBO 46220502 IC50 = 10900 nM T20251 D05XGO 11154555 IC50 = 20720 nM T20251 D06ABF 3957 IC50 = 169.82 nM T20251 D06BCB 443955 IC50 = 39 nM T20251 D06GKN 2099 IC50 = 3235.94 nM T20251 D06MAJ 65906 IC50 = 350 nM T20251 D06MQM 6437380 IC50 = 8100 nM T20251 D06PZN 119584 IC50 = 4800 nM T20251 D06ZUK 3696 IC50 = 3388.44 nM T20251 D07KSG 2733526 IC50 = 1584.89 nM T20251 D07MVK 37393 IC50 = 40 nM T20251 D08CDI 208908 IC50 = 630957.34 nM T20251 D08JZS 4992 IC50 = 1100 nM T20251 D08VXO 6834 IC50 = 891.25 nM T20251 D08YIN 1727 IC50 = 4400000 nM T20251 D09EGZ 2719 IC50 = 2500 nM T20251 D09GOS 2812 IC50 = 3019.95 nM T20251 D09HNR 3002190 IC50 = 40000 nM T20251 D09KTS 24821094 Ki = 1100 nM T20251 D09MWJ 2092 IC50 = 125892.54 nM T20251 D09OJQ 4095 IC50 = 9772.37 nM T20251 D09QUQ 92253 IC50 = 20892.96 nM T20251 D09SGV 25154714 IC50 = 29200 nM T20251 D0AO5H 5578 IC50 = 239883.29 nM T20251 D0AR3J 439501 IC50 = 5800 nM T20251 D0AV3G 3151 IC50 = 162 nM T20251 D0B3UJ 115237 IC50 = 1000 nM T20251 D0B5LF 448042 Ki = 79432.82 nM T20251 D0B7NG 2725 IC50 = 1100 nM T20251 D0BD8D 6917698 IC50 = 12 nM T20251 D0BP9C 193962 IC50 = 25118.86 nM T20251 D0BZ7W 443879 IC50 = 125.89 nM T20251 D0C3SW 53465279 IC50 > 30000 nM T20251 D0C9SY 135400189 IC50 = 79432.82 nM T20251 D0CL9S 159269 IC50 = 5011872.34 nM T20251 D0CS2F 3955 IC50 = 33 nM T20251 D0D1AL 3559 IC50 = 10 nM T20251 D0D7KC 5488548 IC50 = 63095734.45 nM T20251 D0D9FV 4601 IC50 = 851.14 nM T20251 D0DK8V 2678 IC50 = 30199.52 nM T20251 D0DV3O 3241 IC50 = 100000 nM T20251 D0E1WI 3345 IC50 = 1819.7 nM T20251 D0E4DW 1775 IC50 = 100000 nM T20251 D0E6XR 3062316 IC50 = 15848.93 nM T20251 D0E7PQ 5311 IC50 > 30000 nM T20251 D0F0YZ 4737 IC50 = 22800000 nM T20251 D0G9YH 2179 IC50 = 208.93 nM T20251 D0GQ7K 4046 IC50 = 2600 nM T20251 D0GV8J 135565082 IC50 > 100000 nM T20251 D0H0KB 5070 IC50 > 25000 nM T20251 D0H3HM 60795 Ki = 598 nM T20251 D0H7AV 4820 IC50 = 20417.38 nM T20251 D0H7KF 5002 IC50 = 5754.4 nM T20251 D0I0DL 3689 IC50 = 100 nM T20251 D0I1FQ 54671008 IC50 > 50000 nM T20251 D0J0BU 10275777 Ki = 1800 nM T20251 D0J2KV 4932 IC50 = 440 nM T20251 D0JL2K 72474 IC50 = 50000 nM T20251 D0K3QS 6442177 IC50 = 15848931.92 nM T20251 D0K6GZ 60464 IC50 = 21700 nM T20251 D0K7WK 4595 IC50 = 812.83 nM T20251 D0L0ZF 5663 IC50 = 1096.48 nM T20251 D0L4YD 154059 IC50 = 251.19 nM T20251 D0L5WM 2157 IC50 = 10000 nM T20251 D0L7VL 3926 IC50 = 15.85 nM T20251 D0M4YC 3114 IC50 = 91201.08 nM T20251 D0N3VR 71616 IC50 > 40000 nM T20251 D0NJ3V 4680 IC50 = 7244.36 nM T20251 D0NR6S 3002977 IC50 = 79432.82 nM T20251 D0NS6H 3152 IC50 = 1995.26 nM T20251 D0NW3X 71329 IC50 = 5 nM T20251 D0O1WX 2764 IC50 > 30000 nM T20251 D0O3FG 125017 IC50 = 251188.64 nM T20251 D0O3OS 104850 IC50 = 4800 nM T20251 D0O8GK 71496458 IC50 = 16200 nM T20251 D0OB1J 39186 IC50 = 17300 nM T20251 D0P9RF 5401 IC50 = 17782.79 nM T20251 D0Q5UQ 214348 IC50 = 3981071.71 nM T20251 D0Q9EV 11965427 IC50 > 20000 nM T20251 D0R0FE 2520 IC50 = 10 nM T20251 D0R0MW 5329102 IC50 = 500 nM T20251 D0R1JV 60854 IC50 = 120.23 nM T20251 D0R1RS 3715 IC50 = 301995.17 nM T20251 D0RM9Q 68778 IC50 = 851.14 nM T20251 D0S5CU 4499 IC50 = 23000 nM T20251 D0T6WN 6451164 IC50 = 500 nM T20251 D0T8GD 89594 IC50 = 245470.89 nM T20251 D0T8XB 44513473 IC50 > 500000 nM T20251 D0TR5X 3386 IC50 = 10 nM T20251 D0U0VU 5312125 IC50 = 7943.28 nM T20251 D0U1OE 5452 IC50 = 33.2 nM T20251 D0U2JP 4369359 IC50 = 501187.23 nM T20251 D0U2OO 2477 IC50 = 3981.07 nM T20251 D0U3SY 49806720 IC50 > 30000 nM T20251 D0U5FS 3396 IC50 = 2300 nM T20251 D0U5GB 92727 IC50 = 8511.38 nM T20251 D0U5SI 4913 IC50 = 138038.43 nM T20251 D0V4QS 135398745 IC50 = 181.97 nM T20251 D0V8HJ 11671467 IC50 > 1000 nM T20251 D0W8WB 2353 IC50 = 3100 nM T20251 D0W9LX 2585 IC50 = 350 nM T20251 D0WE3O 5288826 IC50 = 1000000 nM T20251 D0WO8W 4062 IC50 = 154881.66 nM T20251 D0WV3U 4893 IC50 = 1584.89 nM T20251 D0X0RI 4178 IC50 = 10000 nM T20251 D0X4RN 3676 IC50 = 263026.8 nM T20251 D0X5ZI 6918493 IC50 = 501187.23 nM T20251 D0Y4JJ 2351 IC50 = 33 nM T20251 D0Y4QG 5388906 IC50 = 0.2 ug.mL-1 T20251 D0Y5AM 444031 IC50 = 79.43 nM T20251 D0Y5DO 2771 IC50 = 3981.07 nM T20251 D0Y5UG 2160 IC50 = 3280 nM T20251 D0Y7RW 4763 IC50 = 3019951.72 nM T20251 D0Z1RV 135398737 IC50 = 191 nM T20251 D0Z1UA 71301 IC50 = 316.23 nM T20251 D0Z1ZM 84029 IC50 = 33113.11 nM T20251 D0Z7ZM 135398744 IC50 = 3300 nM T20251 D00AUX 25230266 IC50 > 20000 nM T20251 D00BUR 216327 IC50 > 1000 nM T20251 D00DRL 44137946 IC50 > 30000 nM T20251 D00FHR 9865515 IC50 > 30000 nM T20251 D00IFR 58423153 IC50 > 30000 nM T20251 D00NZL 11955855 IC50 = 28100 nM T20251 D00RYA 16750271 IC50 > 10000 nM T20251 D00SWQ 10429242 IC50 > 100000 nM T20251 D00WDY 53477157 IC50 = 1400 nM T20251 D00XKB 57406537 IC50 = 2800 nM T20251 D01HLO 58438464 IC50 = 6900 nM T20251 D01NUR 118169620 IC50 = 69000 nM T20251 D01QSO 16654980 IC50 > 30000 nM T20251 D01UBY 46208367 IC50 > 50000 nM T20251 D01UUD 9948102 IC50 = 1700 nM T20251 D01ZAQ 25227436 IC50 > 100000 nM T20251 D02AIN 122678117 IC50 > 33000 nM T20251 D02AYL 456199 IC50 > 30000 nM T20251 D02DTQ 24745335 Ki = 3467.37 nM T20251 D02QWY 24785538 IC50 > 10000 nM T20251 D02WFN 46207733 IC50 = 60000 nM T20251 D03GNI 2166 IC50 = 3900 nM T20251 D03ISJ 135564632 IC50 > 30000 nM T20251 D03KHO 52934180 IC50 = 141000 nM T20251 D03KKR 3547 Ki = 25118.86 nM T20251 D03QAO 25008769 IC50 = 233000 nM T20251 D03QHC 49856296 IC50 = 13400 nM T20251 D03QIE 47953 IC50 = 44668.36 nM T20251 D03RIO 24743758 IC50 = 460 nM T20251 D04COD 25101874 IC50 = 588 ug.mL-1 T20251 D04JZH 11659955 IC50 = 30000 nM T20251 D04LOR 51030730 IC50 = 1900 nM T20251 D04LSD 9818903 Ki = 400 nM T20251 D04OSA 46202416 IC50 = 4800 nM T20251 D04QKU 11438771 IC50 = 7100 nM T20251 D04WUA 219101 IC50 = 10000 nM T20251 D05EXN 58298316 IC50 = 33000 nM T20251 D05LPW 25022354 IC50 = 79600 nM T20251 D05LRD 59286554 IC50 > 30000 nM T20251 D05UYQ 15984937 IC50 = 15848.93 nM T20251 D06DMQ 59472121 IC50 = 3000 nM T20251 D06ENM 66553195 IC50 = 6200 nM T20251 D06EPO 11192346 IC50 = 20000 nM T20251 D06TQR 76287260 IC50 = 26800 nM T20251 D06WHY 16747683 IC50 = 3200 nM T20251 D07EHV 44814409 IC50 = 12000 nM T20251 D07HPJ 11476171 IC50 = 130 nM T20251 D07HZG 11516136 IC50 = 126000 nM T20251 D07LWK 9811357 IC50 = 10000 nM T20251 D08AAV 46893585 IC50 > 100000 nM T20251 D08AOZ 86582336 IC50 = 5500 nM T20251 D08HOM 46207586 IC50 = 1000 nM T20251 D08QGT 17755052 IC50 = 64000 nM T20251 D08UUL 46700756 IC50 = 20000 nM T20251 D09NAW 60195662 Ki > 15857 nM T20251 D09OTX 89741565 IC50 = 1800 nM T20251 D09RVI 23649154 IC50 = 794.33 nM T20251 D0A3CL 49801838 IC50 = 22000 nM T20251 D0A7ZK 56944144 IC50 = 6100 nM T20251 D0B3FV 6445533 IC50 = 10300 nM T20251 D0B5HF 44476893 IC50 > 100000 nM T20251 D0C9UF 155805 IC50 = 1 nM T20251 D0CE6C 135565042 IC50 = 6300 nM T20251 D0DH5X 44472635 IC50 > 30000 nM T20251 D0E0JO 117857370 EC50 > 33000 nM T20251 D0EQ9T 24771368 IC50 > 10000 nM T20251 D0EY0A 42636350 IC50 > 32000 nM T20251 D0F0JJ 11560787 IC50 = 1200 nM T20251 D0F6YM 3035000 IC50 = 20000 nM T20251 D0F7PZ 53316710 IC50 = 12000 nM T20251 D0FD6D 11751922 IC50 = 20000 nM T20251 D0G6QV 208952 IC50 = 34860 nM T20251 D0H9DA 54761306 IC50 = 166000 nM T20251 D0HS5V 11234052 IC50 = 18000 nM T20251 D0HZ2E 5311271 Ki = 1100 nM T20251 D0I2XM 3038500 IC50 = 220 nM T20251 D0I3LO 91933883 IC50 > 10000 nM T20251 D0I3TU 45268455 Ki > 39000 nM T20251 D0I4PW 60164925 IC50 > 30000 nM T20251 D0IZ8X 90111638 IC50 > 10000 nM T20251 D0JU5X 400769 IC50 > 200000 nM T20251 D0K4FP 44548240 IC50 > 33000 nM T20251 D0K4HW 135409468 IC50 = 4466.84 nM T20251 D0K9IF 71666749 IC50 > 30000 nM T20251 D0L9KH 44623998 IC50 > 30000 nM T20251 D0L9QM 59568713 IC50 = 22000 nM T20251 D0LI1C 44469321 IC50 = 30440 nM T20251 D0LQ3L 77108121 IC50 = 195000 nM T20251 D0M3XR 46209133 IC50 = 39000 nM T20251 D0M4TJ 44219292 IC50 > 30000 nM T20251 D0M7CB 9919680 IC50 = 65700 nM T20251 D0M8FD 4261 IC50 > 30000 nM T20251 D0M8OC 16061509 IC50 > 10000 nM T20251 D0M9RQ 11697697 IC50 = 10000 nM T20251 D0MR0B 54766013 IC50 = 31040 nM T20251 D0N6NM 71721648 IC50 > 10000 nM T20251 D0N8QK 24743471 Ki = 8830 nM T20251 D0NU8J 117947097 IC50 > 50000 nM T20251 D0O0BM 44156901 IC50 = 8500 nM T20251 D0O1IM 58298318 IC50 > 33000 nM T20251 D0O1ZI 25006684 IC50 > 100000 nM T20251 D0O8BS 16039797 IC50 > 100000 nM T20251 D0O9XN 11691484 IC50 = 13000 nM T20251 D0OW9L 11973780 IC50 > 10000 nM T20251 D0P5CM 56945146 IC50 = 12589.25 nM T20251 D0PM5U 135564890 IC50 > 40000 nM T20251 D0PM7Q 11152667 IC50 = 15000 nM T20251 D0PW4N 6851740 IC50 = 4810 nM T20251 D0Q7RE 16007391 IC50 > 30000 nM T20251 D0QX8X 71479709 Ki = 3100 nM T20251 D0R0LB 91668194 IC50 > 100000 nM T20251 D0R2OU 25070031 IC50 = 13800 nM T20251 D0R3VK 42642654 IC50 = 4400 nM T20251 D0R8IU 24946280 IC50 > 100000 nM T20251 D0R9IU 44462758 IC50 = 8600 nM T20251 D0R9KG 11604525 IC50 = 11000 nM T20251 D0S1XX 134821691 IC50 > 80000 nM T20251 D0S5IR 86294073 IC50 > 30000 nM T20251 D0SG7B 49831257 IC50 = 85000 nM T20251 D0T0PN 9821217 Ki = 1800 nM T20251 D0T4QA 90456533 IC50 > 10000 nM T20251 D0U4FF 10437018 IC50 = 4000 nM T20251 D0U7KH 86567195 IC50 > 30000 nM T20251 D0U8QH 59239165 IC50 > 100000 nM T20251 D0V2YJ 11655511 IC50 = 20500 nM T20251 D0VI4N 90409366 IC50 > 10000 nM T20251 D0W8XT 60663 Ki = 190 nM T20251 D0XD4I 118502708 IC50 > 33000 nM T20251 D0XT0W 66555680 IC50 = 6900 nM T20251 D0XT6W 6918638 IC50 > 30000 nM T20251 D0Y3ZP 23480 IC50 = 500 nM T20251 D0Y5NA 118435360 IC50 = 9900 nM T20251 D0Y7NA 49871007 IC50 = 4500 nM T20251 D0Z2UQ 25262792 IC50 = 47500 nM T20251 D08IMD 16755780 IC50 = 23000 nM T20251 D0E2FZ 10149311 IC50 > 30000 nM T20251 D0HM5J 118253852 IC50 > 33000 nM T20251 D0IY0R 11591505 IC50 = 23600 nM T20251 D0X5OV 42609962 IC50 > 30000 nM T20251 D01KIJ 72545600 IC50 >= 18500 nM T20251 D02NRD 9865421 IC50 > 10000 nM T20251 D03GTM 118485599 IC50 = 69 nM T20251 D04MAZ 71731606 IC50 = 100000 nM T20251 D0AF0O 54670056 IC50 = 590 nM T20251 D0CV8T 874670 IC50 > 10000 nM T20251 D0D3GL 137662068 IC50 = 15000 nM T20251 D0D4OW 57338826 Ki > 100000 nM T20251 D0F8KE 71059525 Ki = 41.3 nM T20251 D0HG2S 86294663 IC50 = 67000 nM T20251 D0J1LK 118485649 IC50 = 490 nM T20251 D0LU9X 74221950 IC50 = 19000 nM T20251 D0NG8Q 75203906 IC50 = 20900 nM T20251 D0PJ8X 71562840 IC50 = 61700 nM T20251 D0PO8N 117881270 IC50 > 33000 nM T20251 D0V8FC 60169096 IC50 = 25000 nM T20251 D0WS3T 72706254 IC50 = 2700 nM T20251 D0YN2T 86302836 IC50 > 10000 nM T20251 D00PDG 44454750 IC50 = 800 nM T20251 D00PXQ 60785 Ki = 200 nM T20251 D02NGR 9934294 IC50 = 670 nM T20251 D03KWN 11373432 IC50 > 100000 nM T20251 D03OFO 9851380 IC50 = 6000 nM T20251 D04BQR 4342 IC50 = 100000 nM T20251 D06BPG 4528 IC50 > 27000 nM T20251 D06TGE 11226090 IC50 = 14200 nM T20251 D06VXY 9845214 IC50 = 420 nM T20251 D07BUO 25067561 IC50 = 19000 nM T20251 D07GIB 11614352 IC50 = 11000 nM T20251 D07KIJ 10008367 IC50 = 13000 nM T20251 D08AWI 11430856 Ki > 2000 nM T20251 D08SOF 5405 IC50 = 22 nM T20251 D09EVZ 507806 IC50 > 80000 nM T20251 D09RGW 11753159 IC50 > 15848.93 nM T20251 D09XHI 9879103 IC50 = 6350 nM T20251 D0A1NU 16049769 Ki > 45100 nM T20251 D0AQ3H 11505444 IC50 > 10000 nM T20251 D0B4TT 17747460 IC50 = 50.12 nM T20251 D0B7SP 11292933 Ki = 12589.25 nM T20251 D0E2PX 3087190 IC50 = 18.1 nM T20251 D0E3SD 9838729 IC50 > 33000 nM T20251 D0E6OA 65941 IC50 = 251.19 nM T20251 D0G1RH 6918446 IC50 = 194 nM T20251 D0H9GQ 9795276 IC50 = 10000 nM T20251 D0I5UU 123618 IC50 = 27.54 nM T20251 D0J0AE 10052040 IC50 > 3000 nM T20251 D0J9UI 9807238 Ki > 10000 nM T20251 D0K1VK 25262965 IC50 = 30400 nM T20251 D0N8NK 11641563 IC50 = 40000 nM T20251 D0OS6O 60149 IC50 ~ 3 nM T20251 D0Q3ES 11705608 IC50 = 3000 nM T20251 D0W7IR 9887884 IC50 = 32000 nM T20251 D0Y2HR 2247 IC50 = 0.9 nM T20251 D0Y6SN 5311096 IC50 = 630.96 nM T20251 D0Z0CH 3033962 IC50 = 5 nM T20251 C9H6CG 1287 IC50 = 6025.6 nM T20251 CXUC05 2215 IC50 = 2398.83 nM T20251 CCNZ53 2340 IC50 = 3981071.71 nM T20251 CPJ0C2 2747 IC50 = 8800 nM T20251 CZUI83 2769 IC50 = 6.457 nM T20251 CCW9O8 2825 IC50 = 1202.26 nM T20251 CYO1K2 2826 IC50 = 7244.36 nM T20251 C2AXN5 3148 IC50 = 12022.64 nM T20251 CDR20M 3185 IC50 = 1.2 nM T20251 C0H8GR 3191 IC50 = 331.13 nM T20251 C2XP5J 3255 IC50 = 72443.6 nM T20251 CY4WG9 3793 IC50 > 40000 nM T20251 C9LCD8 3823 IC50 = 1905.46 nM T20251 CP4RM6 4486 IC50 = 10000 nM T20251 C5ZC4S 5977 IC50 = 4365158.32 nM T20251 CP1QC0 9801 IC50 = 65 nM T20251 CBHG51 9822 IC50 > 10000 nM T20251 CZXE86 15330 IC50 = 2754.23 nM T20251 CN0WP7 15630 IC50 < 10000 nM T20251 CKCT41 28292 IC50 = 50118.72 nM T20251 CA12TG 38911 IC50 > 40000 nM T20251 C6GN7M 40692 Ki = 1900 nM T20251 CI93MP 51106 IC50 = 9100 nM T20251 C8ODZ3 56069 IC50 > 25000 nM T20251 CV4S2E 62969 IC50 = 200 nM T20251 CP8F7B 64143 IC50 = 12589.25 nM T20251 CD9TC8 64737 IC50 = 22000 nM T20251 C92TML 65014 IC50 > 100000 nM T20251 C97NOS 68634 IC50 = 2100 nM T20251 C1O4FS 73400 IC50 = 16000 nM T20251 CU1H3J 83952 IC50 = 316227.77 nM T20251 C7SXL6 87152 IC50 > 25000 nM T20251 C36LYP 104904 IC50 = 416869.38 nM T20251 C09TNA 107927 IC50 = 40000 nM T20251 CL4IR8 115159 IC50 = 50118.72 nM T20251 CR91WU 117964 IC50 = 84000 nM T20251 CZ48UK 117965 IC50 = 13000 nM T20251 CJ1XF0 119478 IC50 = 169824.37 nM T20251 CEP43C 122068 IC50 = 9500 nM T20251 C6SRK5 123942 IC50 = 1047.13 nM T20251 CMN95P 127718 IC50 = 20.89 nM T20251 CM01FR 128820 IC50 = 44000 nM T20251 CU0C6S 131698 IC50 = 491.4 nM T20251 CIG7L1 160023 IC50 = 8 nM T20251 CGSA42 163906 IC50 = 6100 nM T20251 CDB9P5 170922 IC50 < 10000 nM T20251 C7AV9Z 175533 Ki = 0.4 nM T20251 CLY60V 187063 IC50 = 6606.93 nM T20251 C97DNP 194450 IC50 = 4.3 nM T20251 CI2WO8 219099 IC50 = 120.23 nM T20251 C2V5FA 398712 IC50 = 5000 nM T20251 CLD6J9 441074 IC50 = 323.59 nM T20251 C1Z4HP 441362 IC50 = 5623.41 nM T20251 CQ0XH2 467825 IC50 = 10370 nM T20251 CKC8U4 507751 IC50 > 80000 nM T20251 CPXL01 507783 IC50 > 80000 nM T20251 CM40AT 507791 IC50 > 80000 nM T20251 CFY12E 516173 Ki > 10000 nM T20251 CNCR59 516203 Ki = 30000 nM T20251 C9MVL1 516212 Ki = 16000 nM T20251 CJUT37 516217 Ki = 5700 nM T20251 CRG4W0 516223 Ki = 3800 nM T20251 C2WHI5 516226 Ki = 22000 nM T20251 C9UOI0 516233 Ki = 8100 nM T20251 C67BKT 516235 Ki = 3000 nM T20251 CWTN29 516239 Ki > 10000 nM T20251 C6L1BX 516246 Ki = 3400 nM T20251 C4MQR0 516247 Ki = 5600 nM T20251 C1LB4X 516254 Ki = 37000 nM T20251 CQ52IA 516260 Ki = 14000 nM T20251 C65AZI 516264 Ki = 1000 nM T20251 COA04U 516275 Ki = 3500 nM T20251 C59YWP 516276 Ki = 9600 nM T20251 C9XU6R 516280 Ki = 6000 nM T20251 CHN28A 516284 Ki = 11000 nM T20251 CBYO78 516292 Ki = 2100 nM T20251 C4XN2D 516293 Ki = 2300 nM T20251 CUAO78 516314 Ki = 400 nM T20251 CF2J7U 592280 IC50 = 169824.37 nM T20251 C4TY8B 607867 IC50 = 74 nM T20251 C8WX7B 621620 IC50 = 109647.82 nM T20251 C2M9UC 656771 IC50 = 20 nM T20251 CP7U6Y 667468 IC50 = 6456.54 nM T20251 CN5CJ7 688803 IC50 = 99300 nM T20251 CZN6S9 743974 IC50 > 50118.72 nM T20251 CSMB29 759456 IC50 = 12400 nM T20251 C3LM4S 821286 IC50 > 100000 nM T20251 C90NZF 853261 IC50 > 10000 nM T20251 C79YAJ 1034176 IC50 = 1350 nM T20251 CT2VP9 1471775 IC50 > 32000 nM T20251 CK0JI9 1548955 IC50 = 181.97 nM T20251 C8JLO0 2243267 IC50 = 6300 nM T20251 CTZ4R5 2730286 IC50 = 1500 nM T20251 CD28JA 2735964 IC50 = 10000 nM T20251 CHTM19 2747356 Ki = 1538 nM T20251 C2J9ML 2781852 IC50 > 10000 nM T20251 CORX94 2804997 IC50 > 26302.68 nM T20251 CMRX81 2811640 IC50 > 10000 nM T20251 C9LDS2 2971413 Ki = 5418 nM T20251 C0F4YK 2980278 Ki > 40000 nM T20251 C14NBG 3008866 IC50 > 80000 nM T20251 CUY7J9 3008902 IC50 = 550 nM T20251 CE3Q4V 3008904 IC50 = 1300 nM T20251 CZ1V8Q 3008913 IC50 = 670 nM T20251 C1IS9G 3008917 IC50 = 150 nM T20251 CZV0O6 3008927 IC50 = 570 nM T20251 C8KY7B 3008930 IC50 = 1200 nM T20251 CSED31 3011729 IC50 = 13000 nM T20251 C3U7EZ 3035784 IC50 = 100 nM T20251 C2YQ0B 3082684 IC50 = 14000 nM T20251 CS5F1I 3083481 Ki = 1200 nM T20251 C3HJK8 3525815 IC50 = 2500 nM T20251 C8KN4J 3876755 IC50 > 10000 nM T20251 CO23EI 3959338 IC50 = 27300 nM T20251 C0TV9U 4227718 IC50 > 10000 nM T20251 C9INQ8 4390854 IC50 > 33000 nM T20251 CWE45H 4497898 IC50 = 27000 nM T20251 CO2SY7 4630909 Ki = 870 nM T20251 CE1CP8 4663848 IC50 = 33113.11 nM T20251 C3JHM8 4687521 IC50 = 100000 nM T20251 C16EGI 4961254 IC50 > 10000 nM T20251 CJP1K5 4987129 IC50 > 14790 nM T20251 CZ32RC 5230270 IC50 = 1445.44 nM T20251 CLNI10 5281408 IC50 = 773000 nM T20251 CJB7T6 5288494 IC50 > 33000 nM T20251 CW38FP 5311047 IC50 < 1000 nM T20251 C8EG4K 5326625 IC50 = 8100 nM T20251 C1OZS6 5436342 IC50 > 100000 nM T20251 C3Q2XB 5495793 IC50 > 80000 nM T20251 C0ZAM9 5495818 IC50 > 80000 nM T20251 C6SON9 5837004 IC50 = 36307.81 nM T20251 C95DOH 6098167 IC50 = 12000 nM T20251 CPV72R 6102824 IC50 = 3500 nM T20251 CGL87W 6483572 IC50 = 10500 nM T20251 CO9NP6 6890860 IC50 = 43620 nM T20251 CFTO93 6918704 IC50 = 710 nM T20251 CU68IK 7141881 IC50 > 10000 nM T20251 CZAN92 7472794 IC50 > 25000 nM T20251 C5J8HN 8902499 IC50 = 12700 nM T20251 CL9O2G 9390285 IC50 = 30000 nM T20251 C9IFX8 9390560 IC50 = 13000 nM T20251 CJ07ZA 9800555 IC50 = 32000 nM T20251 C5Z2KM 9805944 IC50 = 245 nM T20251 C2H4ZK 9806118 IC50 = 24 nM T20251 C1W2VB 9814248 IC50 = 5230 nM T20251 CAD92E 9815159 IC50 = 900 nM T20251 CTR6H5 9817349 IC50 = 1995.26 nM T20251 CJS5L9 9819317 IC50 > 30000 nM T20251 C71XRT 9821510 IC50 = 7199.99 nM T20251 CE6NF9 9823363 IC50 = 3100 nM T20251 CEL3C9 9824630 IC50 = 480 nM T20251 C0PQT8 9824969 IC50 = 39800 nM T20251 CZV60D 9825288 Ki = 26400 nM T20251 C97VAE 9825776 Ki = 22700 nM T20251 C8EC9B 9828617 IC50 = 2511.89 nM T20251 CWM26G 9830364 IC50 = 25118.86 nM T20251 C1FQ5A 9835490 IC50 = 8290 nM T20251 C0E7YV 9836903 IC50 > 30000 nM T20251 CU0HE4 9839392 Ki = 18 nM T20251 C30IAQ 9840150 IC50 = 5300 nM T20251 CXE1Y8 9842436 IC50 = 3200 nM T20251 CG3U7J 9843049 IC50 = 1100 nM T20251 CA6N0H 9843867 IC50 = 4700 nM T20251 C7VSU2 9845018 IC50 = 440 nM T20251 CT4E5Z 9846543 IC50 = 210 nM T20251 CKD2H4 9848990 IC50 = 7585.78 nM T20251 C9XY6D 9849838 Ki = 1180 nM T20251 CH57DZ 9850318 IC50 = 1413 nM T20251 CF72XZ 9860561 IC50 = 1600 nM T20251 CRBW42 9861124 IC50 = 5570 nM T20251 C3EX7S 9862272 IC50 = 204 nM T20251 CGC0F7 9864462 IC50 = 2760 nM T20251 CXZ6Q7 9866918 IC50 = 8200 nM T20251 CAOK24 9867098 IC50 = 80 nM T20251 CN9YD5 9868131 IC50 = 3000 nM T20251 C7T3VS 9870145 IC50 = 70 nM T20251 CK7FJ6 9870185 IC50 = 6309.57 nM T20251 CR0EG2 9879772 IC50 = 692 nM T20251 CQJ5X2 9879974 IC50 = 1240 nM T20251 CPS24V 9880847 IC50 = 27460 nM T20251 CS6FN7 9883254 IC50 > 100000 nM T20251 C9IR5L 9884379 IC50 = 90 nM T20251 C2TV9M 9884543 IC50 = 1100 nM T20251 CZ8C7G 9885279 Ki = 6800 nM T20251 C64EOU 9885465 Ki = 1000 nM T20251 CO84WK 9885754 Ki = 62000 nM T20251 C9I8ZU 9887120 IC50 = 10000 nM T20251 CUF35J 9887834 IC50 = 12600 nM T20251 C85BQG 9890458 IC50 = 14000 nM T20251 C2P3GS 9899500 IC50 = 2500 nM T20251 CE28TW 9900179 IC50 = 3020 nM T20251 C2Z9BL 9908431 Ki = 560 nM T20251 CYZ5N4 9909089 EC50 = 7.943 nM T20251 CHB5G9 9909904 IC50 = 199.53 nM T20251 CVJ7I8 9910573 IC50 = 176 nM T20251 C4B2QY 9913339 IC50 = 25000 nM T20251 CF4VO1 9914506 IC50 = 25118.86 nM T20251 CIW81R 9923839 IC50 = 3400 nM T20251 CQF2X8 9925089 IC50 = 974 nM T20251 C10VOI 9930235 IC50 = 3600 nM T20251 CANK40 9931593 IC50 = 10000 nM T20251 C1F4WB 9932192 IC50 = 6960 nM T20251 C9FZO7 9932679 IC50 = 10499.99 nM T20251 C5HQM7 9932974 IC50 = 150 nM T20251 C6RF9U 9933928 IC50 = 1000 nM T20251 CDY39E 9934161 IC50 > 5000 nM T20251 COP96L 9936388 IC50 = 1600 nM T20251 CV5X7E 9938284 Ki = 1000 nM T20251 CS58EO 9944019 IC50 = 3850 nM T20251 CX3ZK9 9946374 IC50 = 1190 nM T20251 CZ4X5D 9946965 IC50 = 101 nM T20251 CV1T2W 9947009 IC50 = 1620 nM T20251 CH6IJ8 9947172 IC50 = 1120 nM T20251 C8T1HO 9948670 Ki = 1300 nM T20251 CLR78W 9952894 Ki = 35000 nM T20251 CKF9X1 9953268 Ki = 1300 nM T20251 CMI58L 9956563 IC50 = 1.7 nM T20251 CJ6BV9 9959777 IC50 = 36 nM T20251 C1NPJ7 9965169 IC50 = 7390 nM T20251 CT7BR0 9965311 IC50 > 1000 nM T20251 C3KTF6 9965610 IC50 = 4670 nM T20251 C6CXJ3 9966330 IC50 = 4560 nM T20251 C0ORJ4 9966331 IC50 = 1310 nM T20251 C49MPX 9966437 IC50 = 3390 nM T20251 CJ2DK6 9966438 IC50 = 1480 nM T20251 C7ZK5J 9966516 IC50 > 10000 nM T20251 CC35UV 9966603 IC50 = 6830 nM T20251 CPX92V 9979309 Ki = 794.33 nM T20251 C7TPF5 9983233 Ki = 445 nM T20251 CGO70N 9983801 IC50 = 82 nM T20251 CJOV70 9983904 IC50 = 54000 nM T20251 CGEJ24 9985625 IC50 = 5100 nM T20251 CRYX90 9986337 IC50 = 9000 nM T20251 C7OAK1 9986346 IC50 = 25.12 nM T20251 CD86AJ 10000396 Ki = 85000 nM T20251 CUQF40 10003657 IC50 = 6309.57 nM T20251 CQL12P 10004545 IC50 > 5000 nM T20251 CGY63T 10004877 IC50 = 85000 nM T20251 CZW1M7 10005242 IC50 > 31622.78 nM T20251 C4Y8TH 10006938 IC50 = 14000 nM T20251 CE7IB5 10007642 IC50 = 11000 nM T20251 CCO68X 10008352 IC50 = 100 nM T20251 CUN7T8 10019811 Ki = 10000 nM T20251 C3NPS8 10025899 Ki = 1750 nM T20251 CA06TQ 10028888 IC50 = 6600 nM T20251 CI3Q9B 10030247 IC50 = 130 nM T20251 CWD3B7 10030344 IC50 = 400 nM T20251 C6V8MF 10032207 IC50 = 8300 nM T20251 C1WH8Q 10042344 IC50 > 10000 nM T20251 C90AVX 10044868 Ki = 51000 nM T20251 C04HZE 10046270 IC50 > 10 nM T20251 CA42DO 10047196 IC50 = 3000 nM T20251 C02OIU 10047339 IC50 = 2250 nM T20251 C73QBA 10047509 IC50 > 10 nM T20251 CR6NW9 10054055 IC50 = 5400 nM T20251 CH5SZ3 10073306 IC50 = 70000 nM T20251 CF7OC8 10073954 IC50 = 21000 nM T20251 CRQL64 10075375 Ki = 120 nM T20251 CR01QE 10076802 IC50 = 1800 nM T20251 C2BG6C 10085660 IC50 > 10000 nM T20251 C8G1PU 10087576 Ki = 2900 nM T20251 CH14BN 10089061 Ki = 480 nM T20251 CR17PA 10093856 IC50 = 2200 nM T20251 CS5K6Q 10095195 IC50 = 2000 nM T20251 C83ZDL 10096130 Ki = 2800 nM T20251 CTN9C2 10097082 IC50 = 3000 nM T20251 C9D5FP 10099787 Ki = 730 nM T20251 C3L9IN 10110435 IC50 = 34000 nM T20251 CBUX03 10113183 IC50 = 8950 nM T20251 CFY9M8 10115569 IC50 = 23000 nM T20251 CVK61T 10116047 IC50 = 26000 nM T20251 CD9EV1 10126599 Ki = 3600 nM T20251 C1WYS8 10127169 Ki = 46 nM T20251 C6N2TK 10131545 IC50 = 2150 nM T20251 CVZ3S9 10132138 IC50 = 10100 nM T20251 C26HWK 10132572 IC50 = 1310 nM T20251 CV67NU 10136016 IC50 = 16700 nM T20251 C09XVI 10144709 IC50 = 54 nM T20251 CLBD08 10144909 Ki = 850 nM T20251 CQM6E2 10149720 Ki = 20000 nM T20251 CLW3J6 10151756 IC50 = 5011.87 nM T20251 CB6V1X 10162604 Ki = 58400 nM T20251 C7JP1A 10163439 Ki = 610 nM T20251 C75JIV 10167216 Ki = 38100 nM T20251 CSHY89 10172243 Ki = 39000 nM T20251 CQ6JH8 10173083 Ki = 15000 nM T20251 CR80BV 10175126 IC50 > 30000 nM T20251 CW0OK6 10178465 IC50 = 6100 nM T20251 C85DYP 10183035 IC50 = 13600 nM T20251 C5K2GS 10185181 Ki = 200 nM T20251 C3DM7B 10186910 IC50 = 12200 nM T20251 CW98JD 10187118 IC50 = 400 nM T20251 C73LXY 10188021 Ki = 11 nM T20251 CK7UT9 10188786 Ki = 290 nM T20251 CLJ02H 10194468 Ki = 240 nM T20251 COV97M 10199905 IC50 = 18600 nM T20251 CCE6H8 10203632 IC50 = 36600 nM T20251 CO51ZR 10205659 Ki = 420 nM T20251 CISE26 10206059 IC50 = 89400 nM T20251 C51SKM 10209082 Ki = 25 nM T20251 CK72XG 10209108 Ki = 490 nM T20251 CCG65P 10210026 Ki = 1200 nM T20251 CT2N1Z 10222208 Ki = 840 nM T20251 C18FMW 10237542 Ki = 320 nM T20251 CQGN38 10237827 Ki = 29 nM T20251 C2PLB1 10239891 IC50 > 30000 nM T20251 C8PJ1V 10248119 IC50 > 10000 nM T20251 CZ90LD 10250452 IC50 = 4600 nM T20251 C24QZK 10256734 IC50 = 4000 nM T20251 CXJ2O5 10256826 IC50 = 2000 nM T20251 C3OE5Z 10257392 IC50 = 2100 nM T20251 C67GCK 10258336 Ki = 43 nM T20251 CF2M9O 10268223 IC50 = 234 nM T20251 CGRQ23 10274114 IC50 = 2700 nM T20251 CHY71P 10274246 IC50 = 960 nM T20251 CM6SE7 10280445 IC50 = 4400 nM T20251 CMNH04 10286136 IC50 = 3300 nM T20251 CUQC81 10287415 Ki = 9400 nM T20251 C9K0SA 10288761 IC50 = 5000 nM T20251 CT89LX 10297708 IC50 = 4000 nM T20251 CV10CU 10297977 Ki = 100 nM T20251 C90DYG 10297996 IC50 = 50100 nM T20251 C1AP6H 10298858 Ki = 2100 nM T20251 CAX9W2 10302405 Ki = 34 nM T20251 C1W5ZD 10308681 Ki = 8050 nM T20251 C3M1VR 10309552 Ki = 225 nM T20251 CZ18PL 10316203 IC50 = 7500 nM T20251 C26EKI 10316979 IC50 = 31000 nM T20251 CF1S8U 10320144 IC50 = 86000 nM T20251 C03ZKG 10324551 IC50 = 5000 nM T20251 CBA2C6 10325032 IC50 = 224 nM T20251 CLKX29 10335984 Ki = 4500 nM T20251 CEZ95L 10342016 Ki = 52000 nM T20251 C5MH7Y 10343434 IC50 = 300 nM T20251 CW50TU 10345610 IC50 = 35200 nM T20251 CIYQ04 10358984 Ki = 6300 nM T20251 CGQN51 10359235 IC50 > 30000 nM T20251 CT6Y9I 10365686 IC50 = 38000 nM T20251 CFH29X 10367570 IC50 = 300 nM T20251 CDA5F7 10369999 IC50 = 6200 nM T20251 C2KO8V 10388264 IC50 = 29000 nM T20251 CP7CH6 10389946 IC50 = 38000 nM T20251 C3H9SB 10390717 IC50 = 19700 nM T20251 CJQV19 10391684 IC50 > 80000 nM T20251 CM9R2K 10391877 IC50 = 1200 nM T20251 CCZ17H 10392978 IC50 = 844 nM T20251 C9WC5D 10393066 IC50 > 8900 nM T20251 CU6X7E 10393880 IC50 = 130 nM T20251 C59QRY 10393962 Ki = 950 nM T20251 C76WZF 10401439 Ki = 11000 nM T20251 CG1T4B 10405623 IC50 = 2700 nM T20251 C6EJ8D 10410012 IC50 = 6.2 nM T20251 C56SLV 10412648 IC50 = 38 nM T20251 CV60SK 10413034 IC50 > 30000 nM T20251 CBN4H0 10415698 IC50 = 1300 nM T20251 CW80YU 10415870 Ki = 710 nM T20251 CUZE30 10416011 IC50 = 100 nM T20251 C6GXW2 10426299 Ki = 1200 nM T20251 C6KR8Z 10428027 Ki = 5100 nM T20251 CS7FG5 10429706 IC50 = 2570.4 nM T20251 C5ZXU8 10433753 IC50 = 25000 nM T20251 C5GQF1 10436125 IC50 = 22700 nM T20251 CWCA76 10439426 IC50 = 76000 nM T20251 C80TCL 10450279 Ki = 5000 nM T20251 CQ4C7Y 10450926 IC50 = 28600 nM T20251 CHW2U1 10451701 IC50 > 33000 nM T20251 C1T7QW 10456093 IC50 = 11000 nM T20251 CVSP85 10456367 IC50 = 29000 nM T20251 C8DWH6 10456892 IC50 = 30700 nM T20251 C38VGA 10457264 IC50 = 2000 nM T20251 C10NHR 10457710 IC50 = 2000 nM T20251 CMDU71 10460463 IC50 = 100 nM T20251 CWFK56 10461282 IC50 = 660 nM T20251 CGXY36 10482372 IC50 = 18100 nM T20251 CEW7C9 10482996 IC50 = 400 nM T20251 C7YPV6 10483558 IC50 = 250 nM T20251 CB52TQ 10495305 Ki = 3000 nM T20251 CPG8U3 10495787 Ki = 1500 nM T20251 C7W9LB 10498834 IC50 = 400 nM T20251 CI0PU7 10518508 IC50 = 10.96 nM T20251 CUQ03E 10520440 Ki = 1600 nM T20251 C2B9PT 10522146 Ki = 930 nM T20251 CV57XZ 10546579 Ki = 110 nM T20251 CMK39Q 10553487 IC50 > 10000 nM T20251 C8E1UH 10570940 IC50 = 3000 nM T20251 CKYT25 10597785 IC50 = 8800 nM T20251 C74NSJ 10615016 Ki = 7000 nM T20251 CQ75TL 10640054 Ki = 1400 nM T20251 C8C2GN 10640055 Ki = 2100 nM T20251 CY9A6G 10689687 IC50 = 790 nM T20251 CG0M4S 10697284 IC50 = 2400 nM T20251 COQ25N 10697363 IC50 = 100 nM T20251 C49IUL 10708935 Ki > 1100 nM T20251 C52SWI 10711404 Ki > 7000 nM T20251 C7PDA6 10713670 Ki = 500 nM T20251 C18ZBG 10758132 Ki = 238 nM T20251 CDK53W 10763704 IC50 = 1000 nM T20251 CFH1Q4 10805130 Ki = 2500 nM T20251 CDOH18 10851309 Ki = 8200 nM T20251 C0VQ3C 10853014 Ki = 5400 nM T20251 CV6ZN3 10861900 Ki = 710 nM T20251 C9QUV7 10863652 Ki = 25000 nM T20251 CX3RT7 10874250 IC50 = 180 nM T20251 C6KW8J 10884405 IC50 = 4300 nM T20251 C4QZ2E 10895064 IC50 = 5800 nM T20251 CLI84D 10895869 IC50 = 9900 nM T20251 C5L2FR 10896860 IC50 = 110 nM T20251 CZFJ03 10899797 IC50 > 60000 nM T20251 CAB0O8 10906012 IC50 = 2700 nM T20251 CDR7G5 10925892 Ki = 69 nM T20251 C9OI8S 10927262 Ki = 1900 nM T20251 CD10XK 10928028 IC50 = 4700 nM T20251 CR8NL2 10950878 IC50 = 870 nM T20251 C4PK7X 10971209 Ki = 570 nM T20251 C6HI0W 10971692 IC50 = 8399.99 nM T20251 C0BUR1 10991521 Ki = 110 nM T20251 CE6XI4 10993905 IC50 = 190 nM T20251 C3WI1P 11004853 IC50 = 4400 nM T20251 CH2A4Z 11016041 IC50 = 4900 nM T20251 C0A7DI 11017241 Ki = 39000 nM T20251 C1N5EF 11026589 IC50 = 9099.99 nM T20251 CG9JC8 11036563 Ki = 4000 nM T20251 C5P8RW 11048955 Ki = 22400 nM T20251 C0EWV4 11056631 Ki = 47 nM T20251 CEPM03 11068867 IC50 = 5870 nM T20251 C56YON 11069321 IC50 = 77 nM T20251 CKBM74 11070099 IC50 = 220 nM T20251 CG2WF1 11111531 Ki = 251 nM T20251 CHX96W 11133309 Ki = 7143 nM T20251 C0VBZ4 11144668 IC50 = 11999.99 nM T20251 CLU8C6 11145028 IC50 = 10000 nM T20251 C7HM0O 11152739 IC50 = 9200 nM T20251 C4NAJ5 11154544 IC50 = 1600 nM T20251 C76YFB 11155030 IC50 = 3300 nM T20251 C3X0AC 11155482 IC50 = 65000 nM T20251 C9AT4X 11163693 IC50 > 20000 nM T20251 CDY8S7 11165745 IC50 = 1650 nM T20251 CK67YW 11166256 Ki > 150000 nM T20251 C6FX8E 11166272 IC50 = 7700 nM T20251 C7OEX0 11174494 IC50 = 17200 nM T20251 CI7L1C 11176908 IC50 = 10000 nM T20251 C1QWM8 11178027 IC50 = 27000 nM T20251 CPEV03 11178961 IC50 = 466 nM T20251 C3TW2O 11187225 IC50 = 2700 nM T20251 C6EWJ9 11188910 IC50 = 13000 nM T20251 C3CAP9 11189372 IC50 = 1000 nM T20251 CUBX19 11189444 IC50 = 1300 nM T20251 CAN73X 11189693 IC50 = 730 nM T20251 CDOC09 11199458 IC50 = 33500 nM T20251 CE6HS7 11200189 IC50 = 56700 nM T20251 CC25EY 11200344 IC50 = 9900 nM T20251 CP6UL9 11200377 IC50 = 9800 nM T20251 CIAE47 11211122 IC50 = 44113 nM T20251 CS5ET8 11212373 IC50 = 1800 nM T20251 CY57AG 11212679 Ki = 794.33 nM T20251 CQ1E8L 11213136 IC50 = 1000 nM T20251 C20HPU 11220991 IC50 = 2300 nM T20251 C5TAN7 11223519 IC50 = 15000 nM T20251 C1VM2S 11225043 IC50 = 200 nM T20251 C0FSV9 11225074 IC50 = 1400 nM T20251 CP9Z1V 11225445 IC50 = 440 nM T20251 CHC3F8 11226573 IC50 = 820 nM T20251 CU75LJ 11227168 IC50 = 26000 nM T20251 CA39QR 11227406 IC50 = 400 nM T20251 C6D3UR 11237434 IC50 = 17900 nM T20251 CC62PB 11238080 IC50 = 52 nM T20251 CTS6F4 11238521 IC50 = 460 nM T20251 C8J5KI 11238580 IC50 = 750 nM T20251 CP8EW3 11245596 IC50 > 10000 nM T20251 C8TD3U 11247946 IC50 = 900 nM T20251 CX43IH 11248146 IC50 = 700 nM T20251 CW1O5V 11256620 IC50 = 220 nM T20251 CP0C2Q 11257803 IC50 > 11000 nM T20251 CZ98EU 11259253 IC50 = 3.6 nM T20251 C7XI0R 11260032 IC50 = 794.33 nM T20251 C92CYH 11265950 Ki > 3000 nM T20251 CRZ3V0 11269310 IC50 = 11784 nM T20251 C2U7OP 11270012 IC50 = 1800 nM T20251 C3N1MF 11270500 IC50 > 24000 nM T20251 C26HWL 11270869 IC50 = 560 nM T20251 CRDU42 11271947 IC50 = 12000 nM T20251 CL0DP6 11272440 IC50 = 501.19 nM T20251 CK36XS 11273324 IC50 = 83.18 nM T20251 CZ8DU0 11273379 IC50 = 10000 nM T20251 C53DQM 11273508 IC50 = 100 nM T20251 COV2U9 11281200 IC50 = 1700 nM T20251 C83KDF 11281738 Ki > 150000 nM T20251 C8CS5F 11282651 IC50 = 6900 nM T20251 CP27SY 11283686 IC50 = 1300 nM T20251 C9X0TH 11291017 IC50 = 15000 nM T20251 CNE3Z7 11296572 IC50 = 700 nM T20251 CV1LG4 11301893 IC50 = 1100 nM T20251 C9BLC7 11304596 Ki = 1995.26 nM T20251 CIMB79 11305766 IC50 = 199.53 nM T20251 C9L0IK 11313056 IC50 = 300000 nM T20251 C30MLR 11313946 IC50 > 31600 nM T20251 CNT19Q 11315446 IC50 = 11000 nM T20251 CVB45M 11315811 IC50 = 24000 nM T20251 C8S4FU 11317045 IC50 = 600 nM T20251 C5DBK1 11326750 IC50 > 50000 nM T20251 CWT28O 11328029 IC50 = 11.5 nM T20251 CP8Y7T 11328449 IC50 = 1800 nM T20251 C5M3ZN 11329138 IC50 = 6100 nM T20251 CQ1CG9 11330529 IC50 = 30000 nM T20251 CIT2Y7 11330837 IC50 > 30000 nM T20251 C7O0ER 11337925 IC50 = 5094 nM T20251 CKZ20A 11353843 IC50 = 9000 nM T20251 CX6C2M 11353855 IC50 = 28000 nM T20251 C0PUK5 11360073 IC50 = 20500 nM T20251 C9L7AT 11364901 IC50 = 40 nM T20251 CZ82WH 11365166 IC50 > 30000 nM T20251 C4BZ1C 11372427 IC50 = 20000 nM T20251 COH57K 11373894 Ki = 1000 nM T20251 C25ZCN 11374110 IC50 > 30000 nM T20251 C36OES 11374857 IC50 = 3.6 nM T20251 CWO2A7 11382160 IC50 = 62000 nM T20251 C2E8MJ 11382472 IC50 = 11989 nM T20251 CEKP86 11383454 IC50 = 501.19 nM T20251 CO1I8H 11384634 Ki = 885 nM T20251 CL1W3C 11387497 IC50 = 100 nM T20251 CE2M9F 11387511 IC50 = 13000 nM T20251 CCK08I 11388055 IC50 = 650 nM T20251 C53ANS 11393281 IC50 > 30000 nM T20251 C9AOM3 11397017 IC50 = 470 nM T20251 CF4OX6 11397149 Ki = 316.23 nM T20251 C7M3XJ 11397742 IC50 = 22600 nM T20251 C82ERW 11397777 IC50 = 350 nM T20251 CQE92F 11406708 IC50 = 21079 nM T20251 CE5ZK6 11409228 IC50 > 30000 nM T20251 CMW42X 11416123 IC50 > 20000 nM T20251 C6I0YP 11416924 IC50 = 3000 nM T20251 C6BE9Q 11417954 IC50 = 78000 nM T20251 CFX98O 11418182 Ki = 5561 nM T20251 C2N0AG 11421712 IC50 > 30000 nM T20251 CML2H3 11428837 IC50 = 7900 nM T20251 CREQ51 11429654 IC50 > 30000 nM T20251 C1YV6P 11442292 IC50 > 100000 nM T20251 CKU8Y3 11442383 IC50 = 18000 nM T20251 CG58SO 11444350 IC50 = 6309.57 nM T20251 CC9D4O 11444936 IC50 = 100 nM T20251 C07VBT 11445050 IC50 = 1900 nM T20251 CY7HT3 11452117 IC50 = 766 nM T20251 CQTM82 11452706 Ki > 150000 nM T20251 CE42DM 11453673 Ki = 1000 nM T20251 CP1WH5 11461365 Ki = 1100 nM T20251 CF6DQ2 11462727 IC50 = 40000 nM T20251 CKU5J7 11464405 IC50 = 4 nM T20251 C39QNY 11464915 IC50 = 500 nM T20251 CO95HP 11474838 IC50 = 19750 nM T20251 C3GMQ1 11477018 IC50 = 794.33 nM T20251 CH6X2L 11478011 IC50 = 6400 nM T20251 CRJ90F 11478858 IC50 = 870 nM T20251 C69PFD 11484605 IC50 > 30000 nM T20251 C8BY4A 11489501 IC50 = 501.19 nM T20251 CA8KE0 11492902 Ki > 20000 nM T20251 C1O9XD 11493620 IC50 = 240 nM T20251 CV41ER 11494867 IC50 = 2400 nM T20251 CXW96U 11495012 IC50 = 18000 nM T20251 CMQ86R 11495432 IC50 = 2530 nM T20251 C7H9AB 11495849 IC50 > 100000 nM T20251 CPX26I 11496746 IC50 = 50118.72 nM T20251 C5Z7GQ 11497411 IC50 = 251.19 nM T20251 CL17QT 11497455 IC50 > 10000 nM T20251 C9YU1O 11497679 IC50 = 1000 nM T20251 CQT5U8 11497680 IC50 = 1995.26 nM T20251 C9JD4N 11497924 IC50 = 1000 nM T20251 C69AMJ 11500781 IC50 = 910 nM T20251 C3B0LO 11501191 IC50 = 760 nM T20251 C6HM0U 11501983 IC50 > 10000 nM T20251 CZIE58 11502008 IC50 = 8.1 nM T20251 CI62OX 11502343 IC50 = 1800 nM T20251 CPO8S1 11502381 IC50 = 7900 nM T20251 CGB8M5 11502401 Ki = 30 nM T20251 C2TVA0 11502638 IC50 = 3800 nM T20251 C3ME1U 11502912 IC50 = 20000 nM T20251 C3ROH5 11504077 IC50 = 2511.89 nM T20251 COD9Z2 11504477 IC50 = 1300 nM T20251 CFSH67 11504490 IC50 = 10000 nM T20251 C10FVQ 11505089 IC50 = 800 nM T20251 C97WGN 11505187 IC50 = 7700 nM T20251 CHX56T 11508058 IC50 = 20200 nM T20251 CLPO39 11508317 Ki = 1100 nM T20251 CH75CA 11508844 IC50 = 4000 nM T20251 C7G4VM 11508924 IC50 = 12000 nM T20251 CV4IZ7 11509189 IC50 = 3036 nM T20251 CCP2Z0 11510399 IC50 = 1370 nM T20251 C72BCW 11510887 IC50 = 13.5 nM T20251 C1LCD7 11510932 IC50 = 560 nM T20251 CF45XR 11511026 Ki = 10 nM T20251 COT4H9 11511117 IC50 = 10000 nM T20251 CE62TB 11511267 IC50 = 1500 nM T20251 C2T8YD 11511361 IC50 > 10000 nM T20251 CP8B7T 11511719 IC50 > 10000 nM T20251 C9DE5V 11511776 IC50 = 490 nM T20251 CDQ18N 11515125 IC50 > 5000 nM T20251 CP9RB7 11515387 Ki > 3000 nM T20251 C23DKS 11516307 Ki = 160 nM T20251 CO0T6Q 11516310 Ki = 910 nM T20251 CS24AX 11516386 IC50 = 2800 nM T20251 CNM42D 11516387 IC50 = 5000 nM T20251 C6X1AJ 11516392 Ki = 710 nM T20251 CZ4OM7 11516508 IC50 = 1730 nM T20251 CVNP35 11517292 IC50 > 3200 nM T20251 C20FMG 11517340 IC50 = 10000 nM T20251 CPQN50 11517341 IC50 = 10000 nM T20251 CTA7M3 11517739 IC50 = 4600 nM T20251 CG3BZ9 11517980 IC50 = 137000 nM T20251 CW68BJ 11518143 IC50 = 14500 nM T20251 CLGO54 11518300 IC50 = 9190 nM T20251 C1KL7T 11518341 IC50 = 4000 nM T20251 CZ3D5Y 11518933 IC50 > 10000 nM T20251 C0WU7G 11518972 IC50 = 125.89 nM T20251 CM4B3J 11519133 IC50 = 6309.57 nM T20251 C08JSL 11519134 IC50 = 5011.87 nM T20251 CY47AQ 11519784 IC50 > 10000 nM T20251 C04RCG 11519858 IC50 = 7943.28 nM T20251 CM09RF 11524148 Ki = 690 nM T20251 CL09JW 11524225 IC50 = 2000 nM T20251 CBRO68 11524900 Ki = 4100 nM T20251 CU7B8I 11525190 IC50 = 110000 nM T20251 CR83WI 11525569 IC50 = 2500 nM T20251 CTNX29 11526451 IC50 = 1000 nM T20251 CR9NA7 11526531 IC50 = 1000 nM T20251 C0O3XD 11527019 IC50 = 58500 nM T20251 CEX8Y5 11527102 IC50 > 10000 nM T20251 CNL15V 11527195 IC50 = 10000 nM T20251 C0BF5R 11527661 IC50 > 30 nM T20251 C75FPD 11529874 Ki = 2840 nM T20251 C0BC6Y 11530223 Ki > 5000 nM T20251 C7NO5X 11531213 Ki = 1000 nM T20251 CZ93HX 11531536 Ki = 710 nM T20251 C94AGK 11531634 Ki = 5000 nM T20251 CS7Q6G 11532065 Ki = 70 nM T20251 CDX19H 11532153 Ki = 42 nM T20251 C89JTB 11532924 IC50 = 1800 nM T20251 C4W2IN 11533195 IC50 = 23900 nM T20251 CFU5V9 11533398 Ki = 800 nM T20251 CJF92G 11533429 IC50 = 3981.07 nM T20251 C2EQ1U 11533448 IC50 = 3981.07 nM T20251 C4LOQ9 11533473 IC50 = 1258.93 nM T20251 CZW9U3 11534726 IC50 = 1995.26 nM T20251 CR53ZL 11537871 IC50 = 18000 nM T20251 C29LCK 11537876 IC50 > 63000 nM T20251 C7R3HN 11538251 Ki = 2200 nM T20251 C8GZ1I 11539020 IC50 = 10000 nM T20251 CIR9M2 11539598 Ki = 16 nM T20251 CSN91H 11539722 IC50 = 6309.57 nM T20251 CJGL17 11539751 IC50 = 19054.61 nM T20251 C0J9NF 11539823 Ki = 3800 nM T20251 CIJ51X 11539903 IC50 = 38000 nM T20251 C0X6CJ 11540474 IC50 = 5011.87 nM T20251 CFS7T8 11540675 IC50 = 17100 nM T20251 CBR9K8 11541314 IC50 > 100000 nM T20251 C8P5GF 11541506 Ki > 10000 nM T20251 CY0JX9 11541985 IC50 = 8428 nM T20251 C5JEZ9 11544171 IC50 < 31622.78 nM T20251 C9UG2V 11544758 Ki > 40000 nM T20251 CS0B4G 11544795 IC50 = 940 nM T20251 CX0DJ3 11545423 Ki = 8252 nM T20251 CF52ZB 11545686 IC50 = 5940 nM T20251 CGE5W7 11546121 Ki = 2800 nM T20251 CFNG56 11546387 Ki = 430 nM T20251 CHT8D7 11547260 IC50 > 30000 nM T20251 CD14OF 11547466 IC50 = 1000 nM T20251 C61LDE 11548217 IC50 = 630.96 nM T20251 CKZ9B0 11548239 IC50 = 158.49 nM T20251 CPA7K8 11548755 IC50 = 251.19 nM T20251 C34JAV 11551351 Ki > 5000 nM T20251 C3DG8U 11552010 IC50 = 340 nM T20251 CCLR26 11552773 IC50 = 19000 nM T20251 CKGI84 11553070 IC50 = 2100 nM T20251 CH0E4A 11553554 Ki = 3100 nM T20251 CKT1O8 11554040 Ki = 2600 nM T20251 CA16WP 11554165 IC50 > 90000 nM T20251 CZD24Q 11554412 IC50 = 47400 nM T20251 CMC79Y 11554762 Ki = 4200 nM T20251 C0VMG7 11555265 IC50 = 251.19 nM T20251 C64NID 11555572 IC50 = 16000 nM T20251 C3Y4GR 11555971 IC50 = 5011.87 nM T20251 CNWU65 11556070 IC50 = 1750 nM T20251 C3RMI1 11559300 IC50 = 5030 nM T20251 C5WKO2 11559625 IC50 > 10 nM T20251 CXR53E 11561126 IC50 = 30 nM T20251 CX1VD8 11562113 IC50 = 1258.93 nM T20251 C0JU9T 11562199 IC50 = 5011.87 nM T20251 CD9SM0 11562361 IC50 > 10000 nM T20251 CQ8CJ9 11562662 IC50 = 10000 nM T20251 C7B4YX 11563243 Ki > 10000 nM T20251 C1VF0P 11566266 IC50 = 1080 nM T20251 CDP9Z0 11566316 IC50 > 20000 nM T20251 C8C1VW 11566318 IC50 > 18700 nM T20251 CCQ8O9 11567495 IC50 = 4300 nM T20251 CZMB92 11567596 IC50 = 2900 nM T20251 CP7W6H 11567952 IC50 = 4300 nM T20251 CJ3FH6 11568363 IC50 = 80 nM T20251 C52PDV 11568714 IC50 = 3162.28 nM T20251 CMFZ35 11568741 IC50 = 10000 nM T20251 CNV08X 11569158 IC50 = 14000 nM T20251 C0J3VR 11569300 IC50 = 2.5 nM T20251 CU6EY8 11569996 IC50 = 1000 nM T20251 CB59HM 11570626 IC50 > 10000 nM T20251 CZD62R 11572546 Ki = 8000 nM T20251 C18BAJ 11572597 IC50 = 27700 nM T20251 C12VCK 11573765 IC50 = 20000 nM T20251 CMX60P 11573849 IC50 > 6870 nM T20251 C3UQL8 11573971 IC50 = 3500 nM T20251 C86YFM 11575878 IC50 < 25118.86 nM T20251 CFC7D3 11576079 IC50 = 9000 nM T20251 CTVX46 11576269 IC50 > 10000 nM T20251 CASH81 11576387 IC50 = 1258.93 nM T20251 C8JW7U 11577059 IC50 = 11000 nM T20251 C8YLD3 11577158 IC50 = 3162.28 nM T20251 CN87ZF 11577588 IC50 = 1550 nM T20251 CR8E2F 11578028 IC50 = 3162.28 nM T20251 CXP2M0 11580426 Ki > 5000 nM T20251 CW7G3X 11580427 Ki > 5 nM T20251 C7I5KM 11581252 Ki = 5200 nM T20251 CE0U8J 11581337 IC50 = 2900 nM T20251 CN1I8D 11581636 IC50 = 6300 nM T20251 CZ28HJ 11581919 IC50 = 6600 nM T20251 CICM46 11582059 Ki = 1600 nM T20251 CVIP95 11582321 IC50 = 2000 nM T20251 C2DG4A 11582651 IC50 = 930 nM T20251 CM0H2R 11583049 IC50 = 6.2 nM T20251 CZ6C8H 11583193 IC50 = 51100 nM T20251 CP53LK 11583743 IC50 > 10000 nM T20251 CP07QN 11583835 IC50 = 450 nM T20251 C0HFP7 11584185 IC50 = 398.11 nM T20251 C6D1MA 11584660 IC50 = 1995.26 nM T20251 CU4J2W 11584694 IC50 = 31.62 nM T20251 CN5DQ9 11585034 IC50 = 2511.89 nM T20251 C73UHS 11585248 IC50 = 1584.89 nM T20251 CR78YS 11585375 IC50 < 1200 nM T20251 CY3A4K 11587772 IC50 = 2270 nM T20251 C5JBF8 11589054 IC50 < 25118.86 nM T20251 COE14C 11589812 IC50 = 6080 nM T20251 CA2KX0 11590078 IC50 > 10000 nM T20251 C7A3OZ 11590444 IC50 < 31622.78 nM T20251 CC75MD 11590828 IC50 = 3981.07 nM T20251 CK4E6V 11591222 IC50 = 12000 nM T20251 CYX50J 11591601 IC50 = 1000 nM T20251 CIUL60 11591633 IC50 = 251.19 nM T20251 CD6Y3F 11592099 IC50 = 11000 nM T20251 C47TZG 11595633 IC50 = 14000 nM T20251 C1A3PZ 11595635 IC50 = 31600 nM T20251 CMAF85 11596311 IC50 = 9.8 nM T20251 COS24N 11596426 IC50 = 8100 nM T20251 C5NRD9 11596521 Ki = 390 nM T20251 CAU85E 11597758 IC50 = 2400 nM T20251 C3LO6F 11597868 IC50 = 7079.46 nM T20251 CH0OD8 11598084 IC50 < 300 nM T20251 C1TOP5 11598123 IC50 = 2511.89 nM T20251 C6KVY0 11598137 IC50 = 9600 nM T20251 CP56DO 11599295 IC50 > 10000 nM T20251 CKI9D5 11599973 IC50 > 31600 nM T20251 CY72UC 11602409 IC50 > 1500 nM T20251 C1GL6E 11602780 IC50 = 3698.63 nM T20251 C7T3WI 11603194 Ki = 480 nM T20251 CRDU82 11603367 IC50 = 11600 nM T20251 C8GVH9 11603554 IC50 = 22387.21 nM T20251 C04ORX 11603648 Ki = 5000 nM T20251 CPXV24 11603996 IC50 > 100000 nM T20251 CH4AE5 11604196 Ki = 6400 nM T20251 C3V9LT 11604824 IC50 = 70000 nM T20251 COI0G2 11605470 Ki = 89 nM T20251 C9DI6R 11606176 IC50 = 19952.62 nM T20251 CO1A5Z 11606378 IC50 = 2511.89 nM T20251 CL04ZJ 11606435 IC50 = 1000 nM T20251 CJC5N8 11606456 IC50 = 3981.07 nM T20251 C83DCU 11609760 IC50 = 2800 nM T20251 C6HLN8 11610150 IC50 = 2810 nM T20251 CC5R1Q 11610423 Ki = 200 nM T20251 CAU61Q 11610483 IC50 = 3550 nM T20251 CD2PU0 11610816 IC50 > 10000 nM T20251 CTF7J8 11611218 IC50 > 30000 nM T20251 COW93C 11611844 IC50 > 63000 nM T20251 C1WI4H 11611859 IC50 = 6100 nM T20251 CZ4B9T 11612643 IC50 = 7500 nM T20251 C6LUG4 11612700 IC50 > 10000 nM T20251 CT16JP 11613587 IC50 = 199.53 nM T20251 CQL5S8 11613750 IC50 = 16000 nM T20251 CN91SZ 11613873 IC50 = 2511.89 nM T20251 C3FQP1 11614515 IC50 = 2100 nM T20251 C8JAM4 11616357 Ki = 12000 nM T20251 CD28IH 11618024 IC50 = 5600 nM T20251 CA5W9R 11618060 EC50 = 9000 nM T20251 C36OSA 11618702 IC50 = 1100 nM T20251 C1GB6K 11618861 Ki = 1500 nM T20251 CA6X1R 11619076 IC50 < 25118.86 nM T20251 CG1RP5 11619850 IC50 = 1.4 nM T20251 CJ73BI 11619909 IC50 = 10000 nM T20251 CKB59U 11620847 IC50 = 3981.07 nM T20251 CXY07A 11621352 IC50 = 251.19 nM T20251 C79OMR 11623756 Ki > 5 nM T20251 C1KD4Z 11623823 IC50 = 40200 nM T20251 CSB9O5 11623845 Ki > 5000 nM T20251 CD2H3T 11624832 IC50 = 18000 nM T20251 C9WMX4 11624970 IC50 = 500 nM T20251 CX1M6Z 11625277 IC50 = 1800 nM T20251 C34OQC 11626062 IC50 = 1000 nM T20251 C6EGB7 11626833 IC50 = 54000 nM T20251 C7C8FX 11626984 Ki = 42 nM T20251 CIO53A 11627085 IC50 > 31600 nM T20251 C3CP2G 11627368 IC50 > 3200 nM T20251 C9FSA8 11627847 IC50 = 1995.26 nM T20251 C51IBH 11627879 IC50 = 5011.87 nM T20251 CEK0Z8 11628328 IC50 > 31600 nM T20251 CE8W1Z 11628452 IC50 = 501.19 nM T20251 CFJN71 11628631 IC50 = 100 nM T20251 C95RDI 11631662 IC50 > 30000 nM T20251 C0G6PN 11632103 IC50 > 10000 nM T20251 CPV49C 11632254 IC50 = 1000 nM T20251 CNS5P7 11632418 IC50 = 1600 nM T20251 C9HCM6 11632711 Ki = 340 nM T20251 CK34LS 11632737 IC50 = 16600 nM T20251 C7H0AV 11633028 Ki = 1500 nM T20251 C1R2BZ 11633045 IC50 = 12600 nM T20251 CWE63G 11633344 IC50 < 25118.86 nM T20251 CD83GL 11634069 IC50 = 36000 nM T20251 CJBR83 11634073 IC50 = 17000 nM T20251 COB0P4 11634166 Ki = 5100 nM T20251 CO68YB 11634336 IC50 = 31000 nM T20251 CYL45U 11634544 IC50 > 10000 nM T20251 C52ZKM 11634651 IC50 > 10000 nM T20251 C75FNR 11634886 IC50 = 1730 nM T20251 CDE1G8 11635187 IC50 > 31600 nM T20251 C8Y9AL 11635230 IC50 > 31600 nM T20251 CUN3R9 11635332 IC50 > 31600 nM T20251 C23XSL 11638166 Ki = 1800 nM T20251 CCE90V 11638319 IC50 > 60000 nM T20251 CQ1U9W 11638962 IC50 = 7570 nM T20251 COLF16 11639342 IC50 = 213000 nM T20251 CR5QB1 11640354 Ki = 930 nM T20251 CIMW51 11640376 Ki = 3800 nM T20251 CY3IN5 11640515 IC50 = 8300 nM T20251 CMNV51 11640588 Ki = 400 nM T20251 CI2KZ1 11641036 IC50 = 170 nM T20251 CWHK19 11641315 IC50 = 11000 nM T20251 C0XC2N 11641596 IC50 = 3981.07 nM T20251 C25KGE 11641641 IC50 = 251.19 nM T20251 C8DXS0 11642163 IC50 = 794.33 nM T20251 CSE96X 11645396 Ki = 3000 nM T20251 CDP23M 11645473 IC50 = 6400 nM T20251 C0M9NX 11646364 Ki = 2100 nM T20251 CW42YV 11646372 IC50 = 7400 nM T20251 CLR3P8 11646541 IC50 = 10000 nM T20251 C24DVX 11647025 Ki = 2600 nM T20251 C9IOM8 11647276 IC50 = 1300 nM T20251 CJQK24 11647458 IC50 = 34600 nM T20251 C6Y4HR 11647548 IC50 > 30000 nM T20251 CPO25R 11647576 IC50 = 4000 nM T20251 C83VLD 11648483 Ki = 1200 nM T20251 CYQB50 11648990 IC50 = 794.33 nM T20251 C0WAT8 11649549 IC50 = 42000 nM T20251 CXG1B4 11649741 IC50 > 100000 nM T20251 CZPG34 11650178 IC50 > 10000 nM T20251 CM5PG0 11653478 Ki = 10000 nM T20251 CEXK54 11653686 IC50 = 15190 nM T20251 C8I7UT 11654412 IC50 = 9 nM T20251 C2R9QT 11654739 Ki = 300 nM T20251 CGU87J 11654962 IC50 = 6300 nM T20251 C0EF3I 11655513 IC50 = 36900 nM T20251 CPH9X5 11655664 IC50 = 4100 nM T20251 CX7FR8 11655728 IC50 > 10000 nM T20251 C48HCV 11656243 IC50 = 2511.89 nM T20251 CVY3H4 11656753 IC50 = 5610 nM T20251 CPE83G 11656848 IC50 = 1258.93 nM T20251 CT14BC 11657494 IC50 = 251.19 nM T20251 CH3N1I 11659592 IC50 = 490 nM T20251 CF92SM 11659664 IC50 = 24700 nM T20251 CC36GP 11660512 Ki = 10000 nM T20251 CR92TH 11660563 IC50 = 3450 nM T20251 CN6Y7D 11661294 IC50 = 7900 nM T20251 C4G9CM 11661358 IC50 > 10000 nM T20251 CMC02O 11661752 Ki = 8700 nM T20251 CXPC31 11662060 IC50 > 100000 nM T20251 CEL15N 11662194 IC50 > 63095.73 nM T20251 C1F9VA 11662657 IC50 = 15600 nM T20251 CKP76R 11662966 IC50 = 10000 nM T20251 CT2AZ4 11663315 Ki = 380 nM T20251 CBU0L8 11663504 IC50 = 5011.87 nM T20251 C69RQX 11663526 IC50 = 2511.89 nM T20251 C3SJO5 11663578 IC50 = 794.33 nM T20251 C1PB0O 11663999 IC50 = 1258.93 nM T20251 C16UWH 11664328 IC50 = 5011.87 nM T20251 CO15KF 11664409 IC50 > 10000 nM T20251 CG3W2T 11666681 Ki = 31000 nM T20251 CPW3A8 11667985 IC50 = 6600 nM T20251 CJSN27 11668594 IC50 = 3000 nM T20251 C64GUF 11668827 Ki = 7900 nM T20251 CFEQ23 11669001 Ki = 5100 nM T20251 C5SJ9K 11669355 Ki = 700 nM T20251 CNE2K5 11669953 IC50 = 25118.86 nM T20251 CU9P5O 11670029 Ki = 900 nM T20251 CPVR45 11670647 IC50 = 794.33 nM T20251 CE6A2S 11671079 IC50 = 780 nM T20251 CX1GS0 11672017 IC50 = 1220 nM T20251 CON70D 11672049 IC50 = 7900 nM T20251 CT3BP5 11674529 IC50 > 10000 nM T20251 CD9XU6 11675152 IC50 < 25118.86 nM T20251 C7A0WS 11675333 IC50 > 10000 nM T20251 C0V7SU 11675388 IC50 = 5235 nM T20251 C29PWK 11675645 IC50 = 1300 nM T20251 CXB59V 11676220 IC50 = 1.7 nM T20251 CX04MA 11676364 IC50 > 150000 nM T20251 CFQP90 11676381 Ki = 62 nM T20251 C3US8X 11676399 Ki = 720 nM T20251 CY5UB8 11676600 Ki = 260 nM T20251 C6GVU2 11676790 IC50 = 31600 nM T20251 CWQ3M4 11677768 IC50 = 1584.89 nM T20251 C6C4BJ 11678080 IC50 = 1995.26 nM T20251 C34RDZ 11678857 Ki = 364 nM T20251 C7JVX2 11681378 Ki > 5000 nM T20251 C7T9ES 11681588 IC50 = 27000 nM T20251 C8RA5V 11682068 IC50 > 10000 nM T20251 C2JSO8 11683474 IC50 < 31622.78 nM T20251 CEHG64 11683903 IC50 = 15.9 nM T20251 CI6JR2 11684405 IC50 = 6300 nM T20251 C1ZD6V 11685267 IC50 = 1258.93 nM T20251 C9K3EO 11688027 IC50 > 60000 nM T20251 CY36RI 11688223 IC50 = 220 nM T20251 CD1O9I 11688761 IC50 > 1000 nM T20251 C87TCD 11689687 IC50 = 1700 nM T20251 C6S2GN 11689802 IC50 = 400 nM T20251 CR91QA 11690139 IC50 = 5000 nM T20251 CRXO13 11690171 Ki = 1200 nM T20251 CG13YQ 11691697 IC50 = 1258.93 nM T20251 CE1KI3 11692214 IC50 = 501.19 nM T20251 CKX65Z 11692293 IC50 = 66000 nM T20251 CGM36K 11692376 IC50 = 1584.89 nM T20251 C7Z0SX 11695591 IC50 = 2300 nM T20251 CFGR63 11695646 IC50 = 15000 nM T20251 CP3G0Q 11695811 IC50 = 1800 nM T20251 CLT3Z7 11695929 EC50 = 5000 nM T20251 CWX2F0 11696319 IC50 = 940 nM T20251 C8QIH0 11696657 IC50 = 2000 nM T20251 CDV58J 11696813 Ki = 930 nM T20251 CX7MT8 11697412 Ki = 500 nM T20251 C8K3OV 11698389 Ki = 150 nM T20251 CT5J9M 11699340 IC50 = 1584.89 nM T20251 CFCB20 11699532 IC50 = 316.23 nM T20251 C4DJ1V 11699804 IC50 > 10000 nM T20251 CBDC74 11702114 IC50 = 590 nM T20251 CQ5P2F 11702115 IC50 = 890 nM T20251 CXFK83 11702578 Ki > 5000 nM T20251 CZ9SY1 11702625 IC50 = 75000 nM T20251 C5UEI7 11703527 Ki = 320 nM T20251 C9SX7H 11704191 Ki = 13000 nM T20251 C3XDB2 11704592 IC50 = 4100 nM T20251 CTZ61B 11704809 IC50 > 95000 nM T20251 CGD80W 11705119 IC50 = 5011.87 nM T20251 CH5B6O 11705343 IC50 = 32000 nM T20251 C2E8BF 11705395 Ki = 30 nM T20251 CLK68A 11705570 IC50 = 1995.26 nM T20251 CPC67X 11705929 IC50 = 501.19 nM T20251 CG2LE3 11706442 IC50 = 3800 nM T20251 CE1FU8 11706443 IC50 = 2300 nM T20251 C04VLB 11706579 Ki > 10000 nM T20251 CG0B5Q 11706981 IC50 = 3300 nM T20251 C3M8DW 11709098 IC50 = 16200 nM T20251 CXMH25 11710453 Ki = 2000 nM T20251 C4M9AU 11710505 IC50 = 2950 nM T20251 CK1FB9 11710573 IC50 < 25118.86 nM T20251 C12EZH 11710694 Ki = 10000 nM T20251 C5FZ1J 11710873 Ki = 3000 nM T20251 C6CM7S 11711078 IC50 = 7900 nM T20251 CIZQ65 11711452 IC50 = 5280 nM T20251 CIUV17 11711973 IC50 = 800 nM T20251 CN8FE3 11712044 IC50 = 15848.93 nM T20251 C9WI7N 11712071 IC50 = 8317.64 nM T20251 CLY3T0 11712237 IC50 = 8000 nM T20251 C5RZ3S 11712530 Ki = 200 nM T20251 CL3H6E 11712583 IC50 = 1200 nM T20251 CHK5I2 11712756 IC50 = 1584.89 nM T20251 C8V9XO 11712898 IC50 = 560 nM T20251 CWQ67V 11713742 IC50 = 9180 nM T20251 C1XYK2 11717025 IC50 = 17000 nM T20251 CI1C4Z 11718272 Ki = 400 nM T20251 C74DRE 11719291 IC50 = 85500 nM T20251 C9R0FW 11719590 IC50 > 10000 nM T20251 CO29BN 11719912 IC50 = 3080 nM T20251 CD9A0J 11720104 IC50 > 10000 nM T20251 C3FP8J 11720191 IC50 = 5600 nM T20251 CX9VH0 11720815 IC50 = 1000 nM T20251 CXUM63 11720838 IC50 = 794.33 nM T20251 C37DMH 11721190 IC50 = 794.33 nM T20251 CIH38K 11723422 Ki = 10000 nM T20251 CP7EV6 11731453 Ki = 21000 nM T20251 CB8N9K 11732098 IC50 = 11000.01 nM T20251 CA7FS4 11732896 IC50 = 2600 nM T20251 CT23IZ 11742071 IC50 = 6.918 nM T20251 CM95SZ 11744578 Ki = 530 nM T20251 CG0YB2 11751828 IC50 = 390 nM T20251 C4L9EC 11752457 IC50 = 24000 nM T20251 C41OBD 11756414 IC50 = 4000 nM T20251 CKW9D4 11756884 IC50 = 17000 nM T20251 C58DMZ 11757696 IC50 = 3200 nM T20251 CZ8E3X 11771731 IC50 < 1000 nM T20251 C7JD4S 11775505 IC50 = 10.5 nM T20251 C5QGC3 11775544 IC50 = 3162.28 nM T20251 CHS9Q3 11785237 IC50 = 5000 nM T20251 CD13QV 11786769 IC50 = 2800 nM T20251 COB43E 11825520 Ki = 150 nM T20251 CG6Q1B 11842628 IC50 = 19700 nM T20251 CD0F5T 11842667 IC50 = 15135.61 nM T20251 CBC08P 11846124 IC50 > 100000 nM T20251 C5LIW2 11846126 IC50 > 100000 nM T20251 CAD8P9 11848624 IC50 < 100 nM T20251 CCT5G7 11848677 IC50 = 3500 nM T20251 CL6B5X 11848835 IC50 = 430 nM T20251 C3UQT0 11853349 IC50 = 2000 nM T20251 C8VK4D 11853588 IC50 = 13000 nM T20251 CYLO43 11854292 Ki = 1900 nM T20251 C1YD8G 11857777 IC50 = 954992586 nM T20251 CXLW54 11948707 Ki > 10000 nM T20251 CP79ZF 11949710 IC50 = 3900 nM T20251 CQSU51 11950826 IC50 = 14125.38 nM T20251 C85VJZ 11950827 IC50 = 1905.46 nM T20251 CQVX45 11950828 IC50 = 208.93 nM T20251 C0WVX4 11951000 IC50 = 8511.38 nM T20251 C0HT7M 11951722 IC50 = 28000 nM T20251 CTR9Z0 11951723 IC50 = 14200 nM T20251 C4EVI9 11951724 IC50 > 30000 nM T20251 CFYK69 11951728 IC50 = 2700 nM T20251 C5M9VQ 11951901 IC50 > 31600 nM T20251 C0GLF5 11952264 IC50 = 11600 nM T20251 CJLB31 11952265 IC50 = 7700 nM T20251 C4JE5Y 11952437 IC50 = 4100 nM T20251 CS3FO8 11952438 IC50 = 6700 nM T20251 CB0LK9 11952439 IC50 = 2400 nM T20251 CK13QD 11953409 IC50 = 6000 nM T20251 C8SZH2 11965686 IC50 = 1995.26 nM T20251 C38ACD 11973711 Ki = 107 nM T20251 CA54WB 11973799 IC50 = 5.4 nM T20251 C09SBY 11973800 IC50 = 21.2 nM T20251 C4G3JS 11973801 IC50 = 14.7 nM T20251 CJ51DI 11973802 IC50 = 47.7 nM T20251 C68TIS 11974129 IC50 = 63.7 nM T20251 CU3J7M 11974130 IC50 = 7.4 nM T20251 CN38YH 11974131 IC50 = 5 nM T20251 C5W7EA 11974229 IC50 = 5.6 nM T20251 C3C2EN 11974230 IC50 = 12.2 nM T20251 CAN81B 11974231 IC50 = 10.4 nM T20251 CNCP71 11974346 IC50 = 20.3 nM T20251 C7W6UZ 11975326 IC50 = 6.7 nM T20251 C3EU8T 11975438 IC50 = 19.9 nM T20251 CN5W3V 11978858 Ki = 10000 nM T20251 C1O8ZJ 11983278 Ki > 9000 nM T20251 CHC85I 11983362 IC50 = 34000 nM T20251 CZ9FS3 11990142 Ki > 9000 nM T20251 C0KM5I 11992827 IC50 = 4500 nM T20251 C56OSH 11995342 IC50 = 21877.62 nM T20251 C0SMQ3 11995420 IC50 = 135000 nM T20251 C9KSG8 11995421 IC50 = 16000 nM T20251 CEYB03 11995422 IC50 > 30000 nM T20251 C58BPD 11995424 IC50 = 21000 nM T20251 CTYE90 11995521 IC50 = 10000 nM T20251 C0DE5H 11995522 IC50 = 76000 nM T20251 CR4YS2 11996303 IC50 = 794.33 nM T20251 C7D1AY 11996304 IC50 = 1258.93 nM T20251 C1A2IB 12001199 IC50 = 1584.89 nM T20251 CNO57E 12001832 IC50 > 50118.72 nM T20251 C1QBK8 12094039 IC50 = 9800 nM T20251 C4CE8D 12111141 Ki = 4000 nM T20251 C5P6ND 12429371 IC50 = 1608 nM T20251 CZ1V4O 12896968 IC50 = 1120 nM T20251 CCS5B1 12951762 IC50 = 506 nM T20251 C7BE0Q 12991318 IC50 = 31600 nM T20251 CM6IO1 14645090 Ki = 24 nM T20251 CIJA82 14645095 Ki = 1.6 nM T20251 C3S8RY 14793784 IC50 = 163.9 nM T20251 C0TO1Z 14921509 IC50 = 17 nM T20251 C0I8GC 14985965 IC50 = 190 nM T20251 CE78SG 15006442 IC50 = 10 nM T20251 C8BF2P 15254720 IC50 = 199.53 nM T20251 C60TVD 15392306 Ki = 3900 nM T20251 C9ZO7G 15604796 IC50 = 19300 nM T20251 CCDX50 15940498 IC50 > 50000 nM T20251 C8JIP7 15940801 IC50 = 16000 nM T20251 CBE59I 15940927 Ki = 5800 nM T20251 CTH2A9 15941083 IC50 = 8400 nM T20251 CF30UM 15941086 IC50 = 10800 nM T20251 CM10PF 15941255 IC50 = 300 nM T20251 CHFW18 15942650 IC50 = 35000 nM T20251 CB8H6M 15947119 IC50 = 250 nM T20251 CPD3V1 15949508 IC50 = 4800 nM T20251 CLD0M2 15949839 IC50 = 33000 nM T20251 CUS3W4 15950258 IC50 = 25000 nM T20251 CM63YP 15950387 IC50 = 14000 nM T20251 C9KJ6D 15950538 IC50 > 80000 nM T20251 C4S7AB 15950540 IC50 > 80000 nM T20251 C3U1VO 15950542 IC50 > 80000 nM T20251 CKX8M6 15950615 IC50 > 80000 nM T20251 C2ZYA6 15951338 IC50 = 39000 nM T20251 C1Q8IV 15951410 IC50 = 23000 nM T20251 C8IJ0O 15952316 IC50 = 1300 nM T20251 CWZM24 15953526 IC50 = 13400 nM T20251 CSA02I 15979148 IC50 = 2778 nM T20251 CBE54Y 15979149 IC50 = 5312 nM T20251 C9QO8U 15979276 IC50 > 10000 nM T20251 C3W8ZL 15981007 IC50 = 290 nM T20251 C8VYW0 15981180 IC50 = 10100 nM T20251 CE4VG5 15981891 IC50 = 24300 nM T20251 C3L4HO 15981894 IC50 = 14800 nM T20251 CB76UT 15981895 IC50 = 49100 nM T20251 C5UOH2 15982018 IC50 = 20000 nM T20251 CI1SK2 15982019 IC50 > 100000 nM T20251 CXD9I3 15982149 IC50 = 50700 nM T20251 CX3M7T 15982150 IC50 > 100000 nM T20251 CP3N4C 15982151 IC50 = 42000 nM T20251 CS9N5F 15982407 IC50 = 40000 nM T20251 CAB1P3 15982533 IC50 = 19000 nM T20251 CD34SB 15982534 IC50 = 35000 nM T20251 CG50BK 15983304 IC50 = 44000 nM T20251 C5OY3I 15983430 IC50 = 29000 nM T20251 CBE59Y 15983549 IC50 = 13000 nM T20251 C6YAJ0 15983550 IC50 = 12900 nM T20251 CUX86I 15983552 IC50 = 6000 nM T20251 CO02BA 15983553 IC50 = 9000 nM T20251 C9TO6J 15983677 IC50 = 3000 nM T20251 CIV82J 15983679 IC50 = 41000 nM T20251 C30OTX 15983680 IC50 = 1400 nM T20251 CT2G7E 15983809 IC50 = 2800 nM T20251 C0GMT8 15983810 IC50 > 100000 nM T20251 CPR25X 15986917 IC50 < 31622.78 nM T20251 CRBP36 15987008 IC50 = 6309.57 nM T20251 C5KW3L 15987108 IC50 = 9332.54 nM T20251 CF6S2D 15987282 IC50 < 63095.73 nM T20251 CXU15Z 15987451 IC50 = 7943.28 nM T20251 C6V3WY 15987452 IC50 < 15848.93 nM T20251 C0HKS9 16004748 IC50 > 10000 nM T20251 CV0YA4 16005493 IC50 = 8410 nM T20251 CG8KR9 16005860 IC50 = 4114 nM T20251 C70KBE 16006079 IC50 = 2220 nM T20251 CCL59Z 16007088 IC50 = 1900 nM T20251 CG5A7W 16013152 IC50 > 30000 nM T20251 CBMF65 16013184 IC50 > 30000 nM T20251 C6V4TG 16013186 IC50 > 30000 nM T20251 CUB5X2 16038385 IC50 > 63095.73 nM T20251 C8AB4L 16039796 IC50 = 18000 nM T20251 CA7QW1 16039834 IC50 = 40000 nM T20251 CPCZ62 16040329 IC50 = 19000 nM T20251 C20CRP 16040587 IC50 > 31622.78 nM T20251 CH8K6G 16040671 IC50 = 31622.78 nM T20251 C8ZP3G 16041292 IC50 > 25118.86 nM T20251 CDU1L0 16041411 IC50 > 30000 nM T20251 CGM4N8 16041594 IC50 > 40000 nM T20251 C1V9EY 16041612 IC50 > 10000 nM T20251 CX9W7Q 16043220 IC50 = 690 nM T20251 CJ78MO 16045297 Ki = 31622.78 nM T20251 CB64EN 16049818 IC50 > 30000 nM T20251 CU27FI 16049886 IC50 = 156666.67 nM T20251 CZC7L2 16049887 IC50 = 115000 nM T20251 CQ9U1Y 16051921 IC50 = 2400 nM T20251 CS8NZ0 16059780 Ki = 6200 nM T20251 C6V4HS 16059786 IC50 = 440 nM T20251 CC2YJ8 16062553 IC50 > 10000 nM T20251 C1LH5T 16062816 IC50 > 10000 nM T20251 C7UCS5 16064456 Ki > 20000 nM T20251 CEZI54 16064872 IC50 = 37153.52 nM T20251 C0V9RI 16064896 Ki > 20000 nM T20251 CM1V6L 16064897 Ki > 20000 nM T20251 C96FEP 16065425 IC50 = 20892.96 nM T20251 CVCJ16 16065428 IC50 = 7762.47 nM T20251 C6MC0Z 16065567 IC50 = 30199.52 nM T20251 CPN9H5 16065569 IC50 = 16595.87 nM T20251 CL1M3W 16065704 IC50 = 16595.87 nM T20251 CF3UG1 16066664 IC50 = 1100 nM T20251 C30UFT 16066811 Ki > 30000 nM T20251 CI1EC9 16068009 Ki = 17000 nM T20251 C3ZKJ5 16068120 Ki = 4400 nM T20251 CPLU48 16068121 Ki = 3800 nM T20251 C9S6QP 16068233 Ki = 13000 nM T20251 CB9Z0L 16068234 Ki = 2600 nM T20251 CW4U7H 16068235 Ki > 20000 nM T20251 CT4JA5 16068236 Ki > 20000 nM T20251 C8SQ5I 16068237 Ki = 6300 nM T20251 CVT0E7 16070046 Ki = 30000 nM T20251 CZ47FJ 16071018 IC50 = 12589.25 nM T20251 CQ06FD 16071731 IC50 = 28000 nM T20251 C3LK2C 16072132 IC50 = 8100 nM T20251 CBM80K 16091080 IC50 = 5319 nM T20251 CX5KI3 16105788 Ki > 10000 nM T20251 CKPQ93 16112836 IC50 = 1584.89 nM T20251 CZC0H1 16116961 IC50 = 25000 nM T20251 CYV05C 16123136 IC50 = 1000 nM T20251 C8C2IW 16123138 IC50 = 100 nM T20251 C7YF8I 16123140 IC50 = 1258.93 nM T20251 C91DQN 16123241 IC50 = 1584.89 nM T20251 CQG7P8 16123247 IC50 = 1258.93 nM T20251 CA6D4S 16123347 IC50 = 1258.93 nM T20251 CBH5P4 16123349 IC50 = 794.33 nM T20251 CPN48R 16123353 IC50 = 1995.26 nM T20251 CK7H2W 16123462 IC50 = 1258.93 nM T20251 C5MY2Q 16123464 IC50 = 10000 nM T20251 CNQ6J2 16123467 IC50 = 3162.28 nM T20251 CWU6P3 16123945 IC50 = 25118.86 nM T20251 CZF23I 16124479 Ki > 100000 nM T20251 C9G8TZ 16124598 IC50 > 31622.78 nM T20251 CYI7J5 16126731 Ki = 16 nM T20251 CTRP20 16190907 IC50 = 15500 nM T20251 CK8Z9L 16220221 IC50 = 2750 nM T20251 CFI8G2 16220223 IC50 = 5300 nM T20251 CTU7J0 16220225 IC50 > 10000 nM T20251 C0ZUH7 16220280 IC50 = 1800 nM T20251 C39SIQ 16220281 IC50 > 10000 nM T20251 C0JA4Q 16220791 IC50 = 5190 nM T20251 CWIT69 16220793 IC50 = 450 nM T20251 CI84RL 16220795 IC50 = 790 nM T20251 C3W1LK 16220874 IC50 = 2590 nM T20251 CUNW89 16220876 IC50 = 3590 nM T20251 C1VUC5 16220877 IC50 = 2500 nM T20251 CN91VO 16220879 IC50 = 3390 nM T20251 CVQ9T5 16220880 IC50 = 4800 nM T20251 C1U9XM 16220882 IC50 = 1750 nM T20251 CZUQ73 16220957 IC50 = 7460 nM T20251 CA5NX6 16220959 IC50 = 1740 nM T20251 C8J3YN 16220960 IC50 = 5870 nM T20251 CPV4G2 16220962 IC50 = 80 nM T20251 C4L7QD 16221024 IC50 = 2100 nM T20251 CAU7E0 16221025 IC50 > 10000 nM T20251 C4GPA2 16221027 IC50 = 1720 nM T20251 C3SH0K 16221088 IC50 > 10000 nM T20251 CM8N1R 16221090 IC50 > 10000 nM T20251 C5E6AC 16221091 IC50 = 1430 nM T20251 CXL6V8 16221092 IC50 > 10000 nM T20251 CW35VX 16221140 IC50 = 1700 nM T20251 C78VJQ 16221258 IC50 = 4870 nM T20251 C9X2GY 16221259 IC50 = 7910 nM T20251 CIA5Y4 16221343 IC50 > 30000 nM T20251 C3P7XC 16221373 IC50 > 10000 nM T20251 CJ8RC1 16221375 IC50 = 53000 nM T20251 C5TV3A 16221425 IC50 > 10000 nM T20251 C8CKV2 16221426 IC50 > 10000 nM T20251 CQE9N1 16221427 IC50 = 2560 nM T20251 CS8W9L 16222361 Ki = 794.33 nM T20251 C2UV9Y 16222392 IC50 > 30000 nM T20251 CA20NM 16222570 Ki = 19952.62 nM T20251 CTH6W4 16292141 IC50 > 25000 nM T20251 CHAY38 16352480 IC50 = 25118.86 nM T20251 CP71ZQ 16389349 IC50 > 50118.72 nM T20251 CX57MU 16648749 IC50 = 6770 nM T20251 C4QU0M 16654984 IC50 = 1200 nM T20251 C6P4BX 16656803 IC50 = 1510 nM T20251 C23NUI 16659197 IC50 = 30000 nM T20251 COC0B8 16659239 IC50 = 25000 nM T20251 CIBY49 16661548 IC50 = 2800 nM T20251 CU9LS2 16661702 IC50 = 780 nM T20251 CYF7U1 16662313 IC50 > 30000 nM T20251 CS90PN 16718565 IC50 = 12600 nM T20251 C7K5AW 16721015 IC50 = 7870 nM T20251 CS14WU 16722242 IC50 > 30000 nM T20251 C8T4JF 16722295 IC50 = 128000 nM T20251 CW62MC 16725327 IC50 = 23000 nM T20251 C4YMP1 16725956 Ki = 206 nM T20251 C92NRU 16727109 IC50 > 80000 nM T20251 COJU37 16727124 IC50 = 200 nM T20251 C4U5XO 16730656 Ki = 18 nM T20251 C8KRM1 16730814 Ki = 4710 nM T20251 C2CRF5 16730815 Ki > 10000 nM T20251 C1D5EW 16733141 Ki = 0.39 nM T20251 CR3W5J 16733265 Ki = 980 nM T20251 C5YWS6 16733266 Ki > 1000 nM T20251 CQO3M8 16733807 Ki = 282 nM T20251 CVI8T4 16735967 IC50 = 27500 nM T20251 CV9US5 16736978 IC50 = 8300 nM T20251 CDG57C 16737679 IC50 = 17000 nM T20251 CHU72I 16738321 IC50 = 11000 nM T20251 CV5F3P 16739263 IC50 > 100000 nM T20251 C6DS7K 16739334 Ki = 4342 nM T20251 CI7Z6F 16741239 Ki = 84 nM T20251 CW2SY5 16750291 IC50 = 7200 nM T20251 CGP40H 16784276 IC50 > 10000 nM T20251 CP69WV 16955923 IC50 = 3000 nM T20251 C5DKZ8 16956771 IC50 = 8000 nM T20251 CU42ZC 17244953 IC50 < 10000 nM T20251 CU05RG 17748274 IC50 > 90000 nM T20251 CAJ0S2 17754557 EC50 > 30000 nM T20251 CN6IP3 17915602 IC50 = 20300 nM T20251 CBNK23 17963226 IC50 > 10000 nM T20251 C5ZT8C 17963227 IC50 = 316.23 nM T20251 CQ7WR1 17963315 IC50 = 10000 nM T20251 C2V6WP 17963332 IC50 > 10000 nM T20251 COCE85 17963334 IC50 > 10000 nM T20251 C2PWS7 17963363 IC50 = 12589.25 nM T20251 C1DVQ9 18004024 IC50 = 562.34 nM T20251 CV5EG7 18727564 Ki > 10000 nM T20251 C1OE8D 18971393 IC50 > 100000 nM T20251 C9JD5Y 19360456 IC50 = 3500 nM T20251 CCA0T1 19958773 IC50 = 2600 nM T20251 C8ICF9 20111627 IC50 = 4300 nM T20251 CES62Q 20299676 IC50 = 300 nM T20251 CSO6R2 20579370 IC50 = 6680 nM T20251 C5S7YM 20579374 IC50 = 1540 nM T20251 C09RQX 20579375 IC50 = 480 nM T20251 CXM1R3 20579392 IC50 = 1480 nM T20251 CWFZ97 20579393 IC50 = 7450 nM T20251 CQAX57 20579471 IC50 = 5920 nM T20251 CFQM24 20664161 IC50 = 2700 nM T20251 C8WSD5 20747478 Ki = 970 nM T20251 CSV2M0 20817761 Ki = 112 nM T20251 C85YPN 20817762 Ki > 2000 nM T20251 CO29QJ 20817763 Ki > 2000 nM T20251 CS4AU1 20817821 Ki = 215 nM T20251 CZC89U 20817846 Ki = 30 nM T20251 CHB01Q 20817864 Ki = 1440 nM T20251 COR4F2 21031286 IC50 > 10000 nM T20251 CMA0D8 21050485 Ki = 4000 nM T20251 C1CA6D 21070989 IC50 = 16000 nM T20251 CAO91K 21099378 Ki = 4000 nM T20251 C9MDU4 21099413 Ki = 8200 nM T20251 C2LMD4 21099424 Ki > 9000 nM T20251 CJB73F 21099433 Ki > 9000 nM T20251 CQU60A 21099448 Ki = 3300 nM T20251 CBCL34 21099463 Ki > 9000 nM T20251 C36INC 21099465 Ki > 9000 nM T20251 C6GRC9 21099470 Ki = 2800 nM T20251 CY75XP 21099472 Ki = 9000 nM T20251 CCO7D2 21099473 Ki > 9000 nM T20251 CP94VE 21099486 Ki > 9000 nM T20251 CF90PJ 21099505 Ki = 7919 nM T20251 CDBY94 21099514 Ki = 6900 nM T20251 CB12UT 21099515 Ki = 9500 nM T20251 C5JCZ6 21193534 Ki = 500 nM T20251 CN85CQ 21252889 IC50 = 2630 nM T20251 CN1XA4 21252891 IC50 = 32500 nM T20251 C18TEI 21303363 IC50 = 8600 nM T20251 COR3F0 21315851 IC50 = 2790 nM T20251 CJV03C 21347732 IC50 < 30000 nM T20251 C6F8SM 21445141 IC50 = 30 nM T20251 CO17PU 21635104 IC50 = 25118.86 nM T20251 C0R5XN 21949788 IC50 = 39000 nM T20251 CCT37S 21949819 IC50 = 9800 nM T20251 C80SEF 21949901 IC50 = 100000 nM T20251 CU0O4K 21955317 Ki = 260 nM T20251 CSZ30L 21998522 Ki = 36870 nM T20251 CSQ2Y0 22017550 Ki = 1268 nM T20251 CJ76FL 22037373 IC50 > 100000 nM T20251 CE65DB 22115679 Ki = 1280 nM T20251 CO32YX 22254068 IC50 > 10000 nM T20251 C0UMW7 22262550 IC50 = 790 nM T20251 C4NO6Y 22315157 IC50 = 23000 nM T20251 C16HAP 22348022 Ki = 355 nM T20251 CCU37W 22348066 Ki = 420 nM T20251 C82XIL 22348140 Ki = 280 nM T20251 CY0WA7 22348155 Ki = 550 nM T20251 C5PS4N 22348219 Ki > 2000 nM T20251 C6KJ0C 22348261 Ki = 778 nM T20251 CMZH62 22391985 IC50 > 94500 nM T20251 CMV28G 22458335 Ki > 10000 nM T20251 CEB1M3 22724580 Ki = 300 nM T20251 CD14YL 23102733 IC50 = 6309.57 nM T20251 CU1T8V 23102749 IC50 = 3981.07 nM T20251 CYW7Q6 23150305 Ki = 8 nM T20251 C5MXI2 23151144 IC50 = 6800 nM T20251 CCES43 23151160 IC50 > 10000 nM T20251 CX6DW5 23151169 IC50 > 10000 nM T20251 C6QC2D 23151199 IC50 = 7900 nM T20251 CGB8I7 23151202 IC50 = 6400 nM T20251 CY8U0D 23151208 IC50 > 10000 nM T20251 C3BP7D 23151209 IC50 > 10000 nM T20251 CT78IA 23151210 IC50 > 10000 nM T20251 C31KDO 23151223 IC50 = 10000 nM T20251 CQ1K7H 23151224 IC50 = 10000 nM T20251 CU24MC 23151229 IC50 > 10000 nM T20251 CM63GT 23151246 IC50 > 10000 nM T20251 C47RDY 23151248 IC50 > 10000 nM T20251 CU4DK0 23151250 IC50 > 10000 nM T20251 C1D0AE 23151312 IC50 > 10000 nM T20251 CE50PJ 23151323 IC50 > 10000 nM T20251 C2KQ6N 23151327 IC50 > 10000 nM T20251 CGJ78I 23151329 IC50 = 8000 nM T20251 COPR89 23151331 IC50 > 10000 nM T20251 C2NYB8 23151337 IC50 > 10000 nM T20251 C12SUL 23151367 IC50 > 10000 nM T20251 C3TVL7 23501721 IC50 > 3000 nM T20251 C7YFT3 23582127 IC50 = 10300 nM T20251 C5E8TY 23582189 Ki = 18540 nM T20251 CL1YH7 23582308 IC50 = 6309.57 nM T20251 C0EJK3 23585071 IC50 > 32000 nM T20251 CW2R4M 23624283 IC50 = 16982.44 nM T20251 C8VD3S 23624312 IC50 = 5400 nM T20251 CMV89L 23625920 IC50 = 2228.44 nM T20251 CW6OB1 23627212 IC50 > 10000 nM T20251 C0R8OI 23628252 IC50 > 10000 nM T20251 CUI9H4 23630215 IC50 = 1200 nM T20251 CK6B7G 23630497 IC50 = 125.89 nM T20251 CH95VG 23630499 IC50 = 63.1 nM T20251 C2XLN1 23630501 IC50 = 10 nM T20251 C1N5TV 23630503 IC50 = 794.33 nM T20251 C7WZJ0 23630505 IC50 = 1258.93 nM T20251 C4MI9Y 23630602 IC50 = 125.89 nM T20251 C24TDZ 23630604 IC50 = 39.81 nM T20251 CU8D0O 23630606 IC50 = 39.81 nM T20251 CKB1E5 23630796 IC50 = 794.33 nM T20251 CJ81PU 23630797 IC50 = 316.23 nM T20251 CV68XN 23630900 IC50 = 39.81 nM T20251 CD61SO 23630901 IC50 = 501.19 nM T20251 CY2RG1 23630902 EC50 = 120 nM T20251 CTJS17 23630998 IC50 = 316.23 nM T20251 CXVR30 23630999 IC50 = 1995.26 nM T20251 CSAT45 23631000 IC50 = 63.1 nM T20251 C6EO1W 23631001 IC50 = 251.19 nM T20251 CE3AM4 23631091 IC50 = 251.19 nM T20251 C9BMW2 23631092 IC50 = 79.43 nM T20251 CKT7B3 23631093 IC50 = 398.11 nM T20251 CM8U1D 23631172 IC50 = 3981.07 nM T20251 CH2I1P 23631366 IC50 = 25.12 nM T20251 C6YS4P 23631368 IC50 = 794.33 nM T20251 C4TV8X 23631454 IC50 = 25.12 nM T20251 CE40PT 23631458 IC50 = 316.23 nM T20251 C09NTA 23631540 IC50 = 794.33 nM T20251 C83QKW 23631544 IC50 = 158.49 nM T20251 C0RPW8 23631636 IC50 = 19.95 nM T20251 CQIG80 23633343 IC50 > 300000 nM T20251 CU1LK3 23633350 IC50 = 100 nM T20251 CC8JL7 23634277 IC50 = 289000 nM T20251 CVF78O 23634281 IC50 = 4200 nM T20251 CEB67J 23644676 IC50 = 4600 nM T20251 C2Q5IK 23645581 Ki = 49000 nM T20251 C07DVE 23646575 IC50 = 2900 nM T20251 CKSD05 23646576 IC50 = 2600 nM T20251 CUJ0D3 23646577 IC50 = 8300 nM T20251 CZ0QF1 23648867 IC50 > 30000 nM T20251 C7MZX9 23649185 IC50 = 3382.98 nM T20251 CE29IW 23650547 IC50 = 9800 nM T20251 CGI6M2 23658492 IC50 = 6200 nM T20251 CM7C4W 23661708 IC50 = 100000 nM T20251 CO6L9F 23661716 IC50 = 100000 nM T20251 CHR14F 23661718 IC50 = 20300 nM T20251 C9H4WT 23686961 IC50 > 31622.78 nM T20251 CASU54 23696973 IC50 > 31622.78 nM T20251 C9PY4A 23725172 IC50 = 13000 nM T20251 CO01RG 24178536 IC50 = 700 nM T20251 CL4WV2 24180125 IC50 > 10000 nM T20251 CBXC05 24424330 IC50 = 80 nM T20251 CQ0KU9 24738459 Ki = 2060 nM T20251 CC52AB 24743739 IC50 = 4500 nM T20251 CN0A5T 24744322 Ki = 6330 nM T20251 CCPE43 24744323 Ki = 2790 nM T20251 C8RC9P 24744325 Ki > 30000 nM T20251 CC5T6J 24744326 Ki > 30000 nM T20251 CP98HS 24744473 Ki = 3400 nM T20251 CCG05Q 24744793 Ki = 9790 nM T20251 CGS47I 24744797 Ki = 460 nM T20251 C1SDO5 24744977 IC50 > 10000 nM T20251 C0CHJ8 24745269 Ki = 16740 nM T20251 CT2DX6 24745764 Ki = 28500 nM T20251 CVB7J3 24746434 Ki = 790 nM T20251 C8EYH1 24746435 Ki = 21450 nM T20251 C28AWJ 24746436 Ki = 1210 nM T20251 CSA6C8 24746437 Ki = 3810 nM T20251 CRN13C 24748804 IC50 = 31622.78 nM T20251 CTIF10 24748806 IC50 < 63095.73 nM T20251 CMJU59 24748889 IC50 = 39810.72 nM T20251 CB6R3K 24748890 IC50 < 63095.73 nM T20251 C5EQ8T 24748892 IC50 < 63095.73 nM T20251 C1XN4V 24748896 IC50 < 15848.93 nM T20251 CFR1S3 24748988 IC50 = 12589.25 nM T20251 CG43ZS 24748989 IC50 = 12589.25 nM T20251 C96KDH 24748992 IC50 = 19952.62 nM T20251 CH8N1W 24748993 IC50 < 63095.73 nM T20251 CQF29T 24749076 IC50 = 25118.86 nM T20251 CU0GX7 24749078 IC50 = 12589.25 nM T20251 CGD2I7 24749080 IC50 = 31622.78 nM T20251 CKVA89 24749182 IC50 < 63095.73 nM T20251 CRGJ52 24749183 IC50 < 63095.73 nM T20251 C13GRZ 24749184 IC50 < 63095.73 nM T20251 C8ZE6H 24749185 IC50 < 31622.78 nM T20251 CG9I8K 24749186 IC50 < 63095.73 nM T20251 CF8W2P 24749291 IC50 < 63095.73 nM T20251 CTB38H 24749292 IC50 < 63095.73 nM T20251 CET71X 24749293 IC50 = 19952.62 nM T20251 CAE9S7 24749294 IC50 < 63095.73 nM T20251 CKV83Y 24749295 IC50 = 7943.28 nM T20251 C6S0OJ 24749401 IC50 = 25118.86 nM T20251 CWTB59 24749606 IC50 = 63095.73 nM T20251 CHYC87 24749609 IC50 < 63095.73 nM T20251 CY53AF 24749610 IC50 < 63095.73 nM T20251 CT93NP 24749721 IC50 < 63095.73 nM T20251 C7EGL2 24749724 IC50 = 12589.25 nM T20251 CW19JN 24749726 IC50 = 50118.72 nM T20251 CI6W7D 24749841 IC50 = 501.19 nM T20251 CV20EP 24749844 IC50 < 63095.73 nM T20251 CYI79E 24749958 IC50 < 63095.73 nM T20251 CGT53R 24749959 IC50 < 63095.73 nM T20251 C20QND 24749960 IC50 = 31622.78 nM T20251 CSXA65 24749962 IC50 < 63095.73 nM T20251 CNOX23 24750086 IC50 = 3981.07 nM T20251 C1XRY9 24750087 IC50 < 63095.73 nM T20251 C89WKU 24750088 IC50 < 63095.73 nM T20251 C7I4LK 24750278 IC50 = 200 nM T20251 CI0W8A 24755210 IC50 = 19600 nM T20251 CUGR26 24757965 IC50 = 15000 nM T20251 CX79CS 24757966 IC50 > 30000 nM T20251 C25HKJ 24758044 IC50 = 7000 nM T20251 CJ1QB7 24758481 IC50 = 2511.89 nM T20251 C8CWX4 24758715 IC50 = 794.33 nM T20251 CU06GI 24758717 IC50 = 630.96 nM T20251 CPL05Y 24758828 IC50 = 630.96 nM T20251 C7RZ9I 24758830 IC50 = 1258.93 nM T20251 C6JQC4 24758832 IC50 = 6309.57 nM T20251 CBNF87 24758834 IC50 = 1995.26 nM T20251 CGQL10 24758836 IC50 = 1995.26 nM T20251 CGE32Q 24758838 IC50 = 6309.57 nM T20251 CL80CU 24758945 IC50 = 6309.57 nM T20251 C8JQW6 24758947 IC50 = 2511.89 nM T20251 CJL67N 24759089 IC50 > 100000 nM T20251 CDF15M 24759558 IC50 = 8000 nM T20251 C1KQY0 24759785 IC50 = 1500 nM T20251 C6GBU8 24762221 Ki = 3981.07 nM T20251 CJ0C1I 24765309 IC50 > 10000 nM T20251 CBJ9T3 24765959 IC50 > 10000 nM T20251 C7RGV4 24768404 IC50 = 950 nM T20251 CZ4J5K 24768415 IC50 = 285 nM T20251 C4ZRC9 24768418 IC50 = 1670 nM T20251 CI6B4H 24768423 IC50 = 4170 nM T20251 CS0C6Q 24768425 IC50 = 600 nM T20251 CBMC42 24768429 IC50 = 420 nM T20251 CA3UK5 24768431 IC50 = 1860 nM T20251 CG8QK3 24768432 IC50 = 1010 nM T20251 CMT5N1 24768433 IC50 = 650 nM T20251 C6HW8J 24768434 IC50 = 2280 nM T20251 CU7W4F 24768547 IC50 = 7100 nM T20251 CHI83W 24769038 IC50 = 32.7 nM T20251 C0I2HU 24769156 IC50 = 10000 nM T20251 CX8DH1 24769723 IC50 > 30000 nM T20251 CVR27S 24769783 IC50 = 6400 nM T20251 C56EJY 24771419 IC50 = 1600 nM T20251 C6H9WM 24771420 IC50 = 1400 nM T20251 COGS63 24771524 IC50 = 3500 nM T20251 CJ9W6U 24771741 IC50 = 900 nM T20251 CBA2P0 24776663 IC50 = 5300 nM T20251 C4ZP5A 24776667 IC50 > 30000 nM T20251 CTG41H 24778289 IC50 = 5800 nM T20251 C30AKB 24778290 IC50 > 30000 nM T20251 CTDU84 24778294 IC50 = 20200 nM T20251 CHZ16E 24778412 IC50 = 2100 nM T20251 CU9Z8O 24778415 IC50 > 30000 nM T20251 C4C3HR 24780883 IC50 = 5.8 nM T20251 C8ELU9 24782303 IC50 = 7943.28 nM T20251 CJ6SF5 24782306 IC50 = 31622.78 nM T20251 C01UNQ 24782307 IC50 = 3981.07 nM T20251 C7KB8R 24782550 IC50 = 15848.93 nM T20251 C3VF5D 24782552 IC50 = 19952.62 nM T20251 C1BQK0 24782553 IC50 = 3981.07 nM T20251 CSPX91 24782554 IC50 = 15848.93 nM T20251 C7A8DI 24782800 IC50 = 25118.86 nM T20251 C5TOI2 24782801 IC50 = 6309.57 nM T20251 C7FZ2J 24782802 IC50 = 10000 nM T20251 C8S4LC 24782803 IC50 = 3981.07 nM T20251 C4KT6W 24782804 IC50 = 5011.87 nM T20251 C2IXL5 24782805 IC50 = 12589.25 nM T20251 CDEB17 24783056 IC50 = 12589.25 nM T20251 C3J4RX 24785333 IC50 = 15848.93 nM T20251 CMPH82 24785597 IC50 = 7943.28 nM T20251 C7HI4R 24785600 IC50 = 10000 nM T20251 CV7WH3 24785604 IC50 = 12589.25 nM T20251 CTF93A 24785864 IC50 = 7943.28 nM T20251 C1JX7P 24785870 IC50 = 25118.86 nM T20251 CRD90F 24786134 IC50 = 7943.28 nM T20251 C7K1EU 24786138 IC50 = 6309.57 nM T20251 CM2DL3 24795066 IC50 = 11000 nM T20251 CP1WR0 24795070 IC50 < 1000 nM T20251 CUM03S 24798754 IC50 = 23000 nM T20251 CDQ58K 24799187 IC50 = 8700 nM T20251 CTQ59S 24799364 IC50 = 7100 nM T20251 C8LJY2 24799365 IC50 = 80000 nM T20251 CO32ND 24799366 IC50 = 14000 nM T20251 C6X0JS 24799545 IC50 = 6100 nM T20251 CG24KB 24799546 IC50 = 9500 nM T20251 C1QL3V 24799711 IC50 = 9900 nM T20251 CH0Y9J 24800231 IC50 = 13000 nM T20251 C10YFG 24800398 IC50 = 12000 nM T20251 C3FYB5 24800577 IC50 = 16000 nM T20251 C17RDK 24800578 IC50 = 2300 nM T20251 C30UAB 24800743 IC50 = 8400 nM T20251 C6SHG9 24800925 IC50 = 15000 nM T20251 C0L6CF 24800927 IC50 = 28000 nM T20251 CM2K4N 24801101 IC50 = 20000 nM T20251 CP8T1L 24801102 IC50 = 33000 nM T20251 CA8GT1 24801457 IC50 = 6000 nM T20251 CW8GD6 24801458 IC50 = 7400 nM T20251 CE25UP 24801459 IC50 = 33000 nM T20251 CSK49W 24801626 IC50 = 25000 nM T20251 C1NK4A 24801627 IC50 = 12000 nM T20251 C9GK5S 24801792 IC50 = 43000 nM T20251 CWH29M 24801795 IC50 = 7700 nM T20251 C84TEM 24801797 IC50 = 8300 nM T20251 C2AKX9 24804150 IC50 = 158.49 nM T20251 CJ4RO1 24804774 Ki = 794.33 nM T20251 CK84BF 24804775 Ki = 10000 nM T20251 C1Z3OQ 24804941 Ki = 2511.89 nM T20251 C6AE2U 24804942 Ki = 1584.89 nM T20251 C1ZYM4 24804943 Ki = 1258.93 nM T20251 CBS5J4 24804985 IC50 > 100000 nM T20251 CH15KN 24808474 IC50 = 60 nM T20251 C73QEI 24808475 IC50 > 10000 nM T20251 CWE46Z 24810003 IC50 = 3960 nM T20251 C14FOH 24810867 IC50 = 30000 nM T20251 CT53OY 24810870 IC50 = 19000 nM T20251 CL5YW9 24825703 IC50 > 30000 nM T20251 CJSO87 24849206 IC50 > 10000 nM T20251 CEA01P 24852079 IC50 > 30000 nM T20251 CR7X1M 24856034 EC50 = 900 nM T20251 CEW31B 24856362 IC50 > 100000 nM T20251 CB4LY1 24857598 IC50 = 2500 nM T20251 CSR8J4 24857759 IC50 = 13100 nM T20251 C9O5NZ 24857819 IC50 = 1600 nM T20251 CY9W8O 24860300 EC50 = 408000 nM T20251 CIR64L 24860582 IC50 = 24200 nM T20251 CKZ25G 24862861 IC50 = 19000 nM T20251 CRUQ41 24863611 IC50 = 17000 nM T20251 C3UNC4 24864147 IC50 = 20000 nM T20251 CCV9N3 24866867 IC50 = 31000 nM T20251 C4UEM5 24871537 IC50 = 1230 nM T20251 CP2L5B 24871655 IC50 = 4650 nM T20251 C7RE9Q 24872164 IC50 = 122000 nM T20251 C06DKB 24875236 IC50 = 16000 nM T20251 CA18VT 24875749 IC50 = 1400 nM T20251 CGI85O 24875752 IC50 = 3640 nM T20251 CT4EZ5 24875845 IC50 = 1710 nM T20251 CLHP80 24875846 IC50 = 17800 nM T20251 CS0K2J 24875942 IC50 = 1070 nM T20251 CU34QD 24884554 IC50 = 12789.47 nM T20251 CNF2E4 24885663 IC50 = 1411.76 nM T20251 CJO97K 24885890 IC50 = 7344.83 nM T20251 C0FUC5 24886365 IC50 = 3666.67 nM T20251 C5KA0N 24893979 IC50 = 3790 nM T20251 CRAK17 24893993 IC50 = 8200 nM T20251 CNQ6I4 24894028 IC50 = 3100 nM T20251 C5WS6R 24894100 IC50 > 10000 nM T20251 C3C0KP 24894134 IC50 = 500 nM T20251 C2EQR6 24894426 IC50 = 940 nM T20251 CT9EZ4 24894428 IC50 = 1500 nM T20251 CN1E8M 24894430 IC50 = 11000 nM T20251 C9USO6 24894431 IC50 = 11000 nM T20251 C4IDR3 24894531 IC50 > 50000 nM T20251 C2AU5Y 24894647 IC50 = 2300 nM T20251 CC6F9D 24894783 IC50 > 50000 nM T20251 C8ERZ5 24895094 IC50 = 5010 nM T20251 C1N0CZ 24895351 IC50 > 10000 nM T20251 CI2S7Y 24895452 IC50 = 1000 nM T20251 CU31LR 24895550 IC50 > 10000 nM T20251 C2IQ9J 24896791 IC50 > 30000 nM T20251 CJ3W0E 24897476 IC50 = 3100 nM T20251 CI4UX5 24900018 IC50 = 7400 nM T20251 C7J4ZQ 24900259 IC50 = 11000 nM T20251 C2TWC8 24900261 IC50 = 7700 nM T20251 CT8GA0 24901491 IC50 > 10000 nM T20251 CY3C1U 24901492 IC50 = 1300 nM T20251 CC2GE7 24901493 IC50 = 2200 nM T20251 CFM1P2 24901494 IC50 = 2400 nM T20251 CF24OR 24901496 IC50 = 1500 nM T20251 CAUZ61 24901497 IC50 = 11000 nM T20251 C7IQO2 24901498 IC50 = 26400 nM T20251 C7TC3P 24901586 IC50 = 2700 nM T20251 C4YDO0 24901587 IC50 = 500 nM T20251 CENZ09 24901588 IC50 = 9000 nM T20251 C8IP6E 24901589 IC50 = 5000 nM T20251 CSD0O9 24901590 IC50 = 1500 nM T20251 CZEF59 24901591 IC50 = 20000 nM T20251 CRNK57 24901592 IC50 = 30000 nM T20251 C4DN3Q 24905400 IC50 > 100000 nM T20251 CD50AV 24905911 IC50 = 14600 nM T20251 CIXU54 24905912 IC50 = 19200 nM T20251 CTU12K 24905913 IC50 = 13800 nM T20251 CGN65K 24905914 IC50 = 15200 nM T20251 C9OAG1 24906198 IC50 = 16900 nM T20251 C0BP8C 24939244 IC50 = 0.41 nM T20251 CYL4U5 24948945 IC50 = 3900 nM T20251 CQU27P 24948946 IC50 = 1100 nM T20251 CRJ08Z 24948948 IC50 = 6000 nM T20251 CC17EO 24950873 IC50 > 10000 nM T20251 C6Z9PO 24951035 IC50 = 6000 nM T20251 CV0PG1 24951036 IC50 > 10000 nM T20251 CB03UR 24951038 IC50 = 5300 nM T20251 C02ADX 24951191 IC50 = 6700 nM T20251 C7WE9M 24951192 IC50 = 1600 nM T20251 CVT49O 24951193 IC50 > 10000 nM T20251 C7DGE0 24951348 IC50 = 2500 nM T20251 C9GA3W 24951349 IC50 = 2600 nM T20251 COW04Z 24951350 IC50 = 350 nM T20251 CHD86F 24951351 IC50 = 2800 nM T20251 CNP3T1 24951733 IC50 > 100000 nM T20251 C40XUR 24952765 IC50 = 30 nM T20251 CCO20I 24953169 Ki = 60 nM T20251 CC0U6X 24953170 Ki = 130 nM T20251 CO41IK 24953519 Ki = 180 nM T20251 C3AQG0 24957697 IC50 = 27500 nM T20251 C2JZ3S 24957698 IC50 > 30000 nM T20251 CZ3FO0 24958070 IC50 > 30000 nM T20251 C82OXU 24958071 IC50 > 30000 nM T20251 C6IC2O 24958072 IC50 > 30000 nM T20251 CB16FH 24958073 IC50 > 30000 nM T20251 C5H4QV 24958074 IC50 > 30000 nM T20251 CCJ9G0 24958075 IC50 > 30000 nM T20251 C04IDY 24958076 IC50 > 30000 nM T20251 C79TOJ 24958447 IC50 > 30000 nM T20251 CDTJ93 24958448 IC50 > 30000 nM T20251 CSF3J5 24958449 IC50 > 30000 nM T20251 CSZ1F5 24958450 IC50 > 30000 nM T20251 C9QX2O 24958451 IC50 > 30000 nM T20251 CAX05W 24958452 IC50 > 30000 nM T20251 CH4C3E 24958809 IC50 > 30000 nM T20251 CPC58S 24958810 IC50 > 30000 nM T20251 C14FUP 24958811 IC50 > 30000 nM T20251 CM94VS 24958812 IC50 > 30000 nM T20251 C65PZU 24958813 IC50 > 30000 nM T20251 C6YR5K 24958814 IC50 > 30000 nM T20251 CNX41V 24958815 IC50 > 30000 nM T20251 C2UZ5G 24958816 IC50 > 30000 nM T20251 C8BEW0 24959168 IC50 = 5200 nM T20251 CNO0U1 24959169 IC50 = 4800 nM T20251 C5J3SP 24959542 IC50 > 30000 nM T20251 CBM71O 24959543 IC50 = 22000 nM T20251 C5BZE7 24959906 IC50 = 2700 nM T20251 CC76EQ 24961017 IC50 = 14800 nM T20251 CR6C3N 24962469 IC50 = 3200 nM T20251 CW4X0E 24962988 Ki = 2830 nM T20251 C6EQG2 24963293 IC50 = 1790 nM T20251 C02YIQ 24963478 IC50 = 26000 nM T20251 CQ58IV 24964189 IC50 > 33000 nM T20251 CS6XP4 24964190 IC50 > 33000 nM T20251 CDC01R 24965775 IC50 = 54 nM T20251 CDF34R 24966125 IC50 = 320 nM T20251 CY0G1A 24966127 IC50 = 230 nM T20251 C6Z7KY 24967023 IC50 = 15000 nM T20251 C14KJT 24967024 IC50 > 33000 nM T20251 CY02UG 24967383 IC50 > 33000 nM T20251 CV40UK 24967750 IC50 > 32000 nM T20251 C4X1JN 24968454 IC50 = 22000 nM T20251 CYH04T 24968455 IC50 = 27000 nM T20251 C4D2VI 24968798 IC50 = 28000 nM T20251 CQ2Z7T 24985115 IC50 > 50118.72 nM T20251 CM7HQ5 24985395 IC50 > 200000 nM T20251 CEJ74C 24985745 IC50 > 200000 nM T20251 CNYD53 24987709 IC50 = 7900 nM T20251 CNMD47 24990839 IC50 = 2200 nM T20251 CZD3W7 24992427 IC50 = 380 nM T20251 CL83OS 24992519 IC50 > 10000 nM T20251 C16SVM 24992849 IC50 = 9000 nM T20251 C8KIP6 24993178 IC50 = 21000 nM T20251 CD8U2B 24993500 IC50 = 8000 nM T20251 CCDF20 24994127 IC50 > 10000 nM T20251 CK5LM1 24996644 IC50 = 7000 nM T20251 CFDQ56 24996645 IC50 > 30000 nM T20251 CTL2D0 24996647 IC50 = 2000 nM T20251 CPYC89 24998177 IC50 = 17000 nM T20251 C2DT4C 24998178 IC50 > 32000 nM T20251 CZ4OL9 24998808 IC50 = 8000 nM T20251 CVB1P5 24999737 IC50 > 32000 nM T20251 C21VCQ 25001553 IC50 = 11000 nM T20251 C6H4YL 25001554 IC50 = 14000 nM T20251 CUMH07 25001555 IC50 > 30000 nM T20251 CJR70I 25001557 IC50 > 30000 nM T20251 CIWR78 25001850 IC50 > 30000 nM T20251 CWO1V4 25004449 IC50 = 680 nM T20251 CETJ60 25006676 Ki = 19952.62 nM T20251 CN6J3R 25008249 IC50 = 93000 nM T20251 CYE9X4 25008593 IC50 = 176000 nM T20251 C5KNH1 25008765 IC50 = 305000 nM T20251 COE0T4 25008767 IC50 = 172000 nM T20251 CD2VF7 25008771 IC50 = 174000 nM T20251 C0KZ5Q 25008940 IC50 = 27000 nM T20251 CXB5T7 25008941 IC50 = 124000 nM T20251 CJ1HQ5 25009146 Ki = 10250 nM T20251 C7XMO2 25009310 Ki = 1760 nM T20251 CZ6T5Q 25009937 Ki = 3300 nM T20251 CCK8G4 25012362 IC50 = 1800 nM T20251 C0EI7T 25012524 IC50 = 277 nM T20251 C1VRJ3 25014630 IC50 = 13000 nM T20251 CM1H6K 25016328 IC50 > 10000 nM T20251 CV02TA 25017750 IC50 = 17000 nM T20251 CTYD20 25018000 IC50 = 11200 nM T20251 CJNR78 25018002 IC50 = 9100 nM T20251 C9AKD7 25018252 IC50 = 8400 nM T20251 CB36TF 25019018 IC50 = 26700 nM T20251 CUF48R 25019019 IC50 = 15800 nM T20251 C91QFN 25019282 IC50 = 15100 nM T20251 CKR94M 25022356 IC50 = 1000 nM T20251 CQ9LS6 25022704 Ki = 5800 nM T20251 C70MLG 25024304 IC50 = 81000 nM T20251 CA20NZ 25025581 IC50 = 4200 nM T20251 CNW89T 25026445 Ki = 4200 nM T20251 C5V1YO 25029711 IC50 = 4610 nM T20251 C8CIY2 25030810 IC50 > 30000 nM T20251 C6DO4B 25032525 Ki = 2202 nM T20251 C6K4SH 25033519 Ki > 7500 nM T20251 CVQS96 25052767 IC50 = 36000 nM T20251 CHQ86P 25054013 IC50 = 2300 nM T20251 C7EQ5T 25054288 IC50 = 9000 nM T20251 CCEY27 25054289 IC50 = 800 nM T20251 C0PIZ8 25054550 IC50 = 16000 nM T20251 C20JHU 25054551 IC50 > 30000 nM T20251 CG8C7J 25054804 IC50 = 2000 nM T20251 CJS39H 25055504 Ki = 5900 nM T20251 C1PKF0 25056080 IC50 > 10000 nM T20251 C0Z2SQ 25056787 IC50 = 10000 nM T20251 CPAZ91 25056788 IC50 = 7943.28 nM T20251 C2FP5D 25056872 IC50 = 16400 nM T20251 C6Z3CE 25057124 IC50 = 8500 nM T20251 C0TYE6 25057388 IC50 = 1800 nM T20251 CE12CD 25057645 IC50 > 30000 nM T20251 C1K9VQ 25057911 IC50 = 1800 nM T20251 CH4PI7 25057913 IC50 = 3300 nM T20251 C8L6JE 25058425 IC50 = 3 nM T20251 CR5FX4 25059765 IC50 = 0.65 nM T20251 CTI38U 25060119 IC50 = 6950 nM T20251 CMJ1F7 25067546 IC50 = 98000 nM T20251 C7YRG0 25067560 IC50 = 1584.89 nM T20251 CM83VQ 25067563 IC50 = 2800 nM T20251 C7O8YH 25068794 Ki = 779 nM T20251 CZ9SN8 25068797 Ki = 931 nM T20251 CL46IP 25068850 Ki = 1560 nM T20251 CEH7D9 25068903 Ki = 1680 nM T20251 CB03DL 25068905 Ki = 2810 nM T20251 C5ZHN9 25068906 Ki = 3610 nM T20251 C0ZJB7 25068907 Ki = 1290 nM T20251 C9G7EM 25068908 Ki = 439 nM T20251 C16ERI 25069015 Ki = 907 nM T20251 CHZB81 25069180 Ki = 1860 nM T20251 CBY3O2 25070582 IC50 > 22300 nM T20251 COE3T5 25071310 IC50 = 2511.89 nM T20251 CU0SR4 25071931 IC50 = 3981.07 nM T20251 C18XGM 25072242 IC50 = 1995.26 nM T20251 CG71VR 25072244 IC50 = 15848.93 nM T20251 C4RE0M 25072246 IC50 = 7943.28 nM T20251 CTWZ82 25072568 IC50 = 50118.72 nM T20251 CW2H9F 25072875 IC50 = 1995.26 nM T20251 CA4FV9 25072876 IC50 = 3981.07 nM T20251 CPUB18 25072877 IC50 = 1584.89 nM T20251 C6GPL3 25072880 IC50 = 794.33 nM T20251 CDY9Z4 25073188 IC50 = 12589.25 nM T20251 C3AJD0 25073189 IC50 = 6309.57 nM T20251 C9KR8V 25073190 IC50 = 10000 nM T20251 C68FHZ 25073191 IC50 = 2511.89 nM T20251 C98ISN 25073801 IC50 = 3981.07 nM T20251 C3AFU0 25093775 IC50 = 670 nM T20251 CP0IR1 25094630 IC50 > 32000 nM T20251 CKP3J6 25094902 IC50 > 25000 nM T20251 CNOA12 25094903 IC50 = 32000 nM T20251 CC6NZ8 25095678 IC50 > 33000 nM T20251 C2H4VG 25096016 IC50 = 1400 nM T20251 C51OJR 25099115 IC50 > 10000 nM T20251 CUB4W5 25102935 IC50 = 12000 nM T20251 CM0O7N 25102936 IC50 > 32000 nM T20251 C3PKV4 25102938 IC50 > 32000 nM T20251 CPM6S0 25104740 IC50 = 13000 nM T20251 CJW1T2 25104741 IC50 > 32000 nM T20251 C4S5XP 25107560 IC50 = 1390 nM T20251 CF1E3C 25107622 IC50 = 1910 nM T20251 CN7W1T 25107626 IC50 = 1630 nM T20251 C0BW7J 25107695 IC50 = 2400 nM T20251 C1XI8C 25107697 IC50 = 170 nM T20251 CUO18X 25107759 IC50 = 730 nM T20251 CC4YH9 25107761 IC50 = 830 nM T20251 CPL78K 25108016 IC50 = 370 nM T20251 C32VHJ 25108017 IC50 = 130 nM T20251 CN1B5F 25108078 IC50 = 430 nM T20251 COS8G5 25108135 IC50 = 1200 nM T20251 CGV7K5 25108137 IC50 = 1700 nM T20251 C5Q6GA 25108843 IC50 > 30000 nM T20251 CON1U6 25110598 IC50 = 12000 nM T20251 CQ2XF3 25110840 IC50 > 5000 nM T20251 CP03LT 25113806 IC50 = 2511.89 nM T20251 CWO19M 25114846 IC50 = 9970 nM T20251 CSI90H 25114847 IC50 = 85900 nM T20251 CDW2I9 25114850 IC50 = 7180 nM T20251 CS24RM 25115077 IC50 = 14100 nM T20251 C1D7TX 25115962 IC50 > 32000 nM T20251 CJC90O 25115964 IC50 > 32000 nM T20251 C2D9XW 25116186 IC50 = 52000 nM T20251 CMXE76 25116191 IC50 > 32000 nM T20251 C0QOD8 25117760 IC50 > 33000 nM T20251 CH57JF 25118124 IC50 > 33000 nM T20251 C6C0HA 25118125 IC50 > 33000 nM T20251 C4DMZ5 25118127 IC50 > 33000 nM T20251 CXBZ57 25118294 Ki = 400 nM T20251 CXE6T1 25118477 IC50 = 20800 nM T20251 CZ96TL 25118804 IC50 > 100000 nM T20251 C8T7NC 25118805 IC50 > 100000 nM T20251 CJM41E 25119356 Ki = 400 nM T20251 C8HI9Y 25119357 Ki = 500 nM T20251 CGL63Q 25119716 Ki = 500 nM T20251 CQ8Y7T 25120419 Ki = 1000 nM T20251 CS6O1Q 25120608 IC50 > 30000 nM T20251 C2G0BK 25120953 IC50 > 30000 nM T20251 CLV98T 25120954 IC50 > 30000 nM T20251 CXL3Q8 25121114 Ki = 600 nM T20251 C2S1LG 25121469 Ki = 200 nM T20251 CR2D3W 25122009 IC50 = 25000 nM T20251 C1RBQ7 25122183 Ki = 1070 nM T20251 CYWO57 25122184 Ki = 80 nM T20251 C07OMT 25122324 IC50 = 25000 nM T20251 C0KOU6 25123487 IC50 = 161 nM T20251 C0W8IC 25124143 IC50 = 1400 nM T20251 CL4XY0 25125138 IC50 = 100 nM T20251 CIYA24 25125139 IC50 = 720 nM T20251 CF54QZ 25129041 IC50 > 100000 nM T20251 CDO26T 25129042 IC50 = 7943.28 nM T20251 CUO63Q 25129091 IC50 = 379 nM T20251 CHK3S8 25129266 IC50 = 5000 nM T20251 CT9CL8 25129432 IC50 = 585 nM T20251 CLW14R 25129434 IC50 < 100 nM T20251 CQ36GH 25129435 IC50 = 663 nM T20251 C2XI7E 25129436 IC50 > 100000 nM T20251 CT30ZV 25129437 IC50 = 303 nM T20251 CM6KY3 25129438 IC50 = 6450 nM T20251 C5AF2Y 25129498 IC50 = 483 nM T20251 CDQ7C1 25129500 IC50 = 655 nM T20251 C5PA3S 25129777 IC50 = 47440 nM T20251 C9ELP5 25129778 IC50 = 1814 nM T20251 C5Q3JF 25129779 IC50 = 18310 nM T20251 C4DL2M 25129780 IC50 = 60000 nM T20251 CV93JO 25129849 IC50 = 2208 nM T20251 CL8YG2 25129850 IC50 = 883 nM T20251 CJ6TD3 25129852 IC50 = 1799 nM T20251 C8PJ6A 25129853 IC50 = 1047 nM T20251 C4SA9U 25129854 IC50 = 4823 nM T20251 C6CB1W 25130210 IC50 = 3674 nM T20251 CXK12T 25130211 IC50 = 1021 nM T20251 C6CF3U 25130212 IC50 = 2047 nM T20251 CS3OY1 25130213 IC50 = 4810 nM T20251 CGC5U6 25130214 IC50 = 4731 nM T20251 CYD2Q3 25130556 IC50 > 10000 nM T20251 CK04RW 25130557 IC50 = 1260 nM T20251 C3I1XJ 25132254 IC50 = 1995.26 nM T20251 C9J1MQ 25138078 IC50 = 24000 nM T20251 CC5O4P 25138090 IC50 = 540 nM T20251 CM03CP 25138344 IC50 > 50118.72 nM T20251 C9DQ8L 25139490 IC50 = 3900 nM T20251 CWL9E2 25139491 IC50 > 10000 nM T20251 C3XJM1 25139625 IC50 = 7300 nM T20251 CKLC61 25139757 IC50 = 5400 nM T20251 C4N1YF 25139758 IC50 = 3300 nM T20251 CFS3N9 25144422 IC50 = 860 nM T20251 CUX49Z 25144536 IC50 = 40900 nM T20251 C2H4KJ 25145553 IC50 = 740 nM T20251 CQR84M 25147644 IC50 = 54000 nM T20251 C35XQI 25150621 IC50 > 10000 nM T20251 CD0QU5 25150624 IC50 > 10000 nM T20251 CIZ1N9 25150625 IC50 > 10000 nM T20251 CE1ND3 25150628 IC50 > 10000 nM T20251 CAVR45 25150711 IC50 > 10000 nM T20251 CYOV03 25150901 IC50 > 30000 nM T20251 CMS9R3 25151607 IC50 > 30000 nM T20251 C0XBY4 25151662 IC50 > 30000 nM T20251 CD70KZ 25151793 IC50 = 2372 nM T20251 CHU1R7 25151849 IC50 > 30000 nM T20251 C7XDZ8 25151850 IC50 = 3580 nM T20251 CC1T8M 25151988 IC50 = 11330 nM T20251 CH9NA3 25151989 IC50 > 30000 nM T20251 C5AY6K 25151990 IC50 > 30000 nM T20251 CT3D7E 25152023 IC50 = 2310 nM T20251 C05HFO 25152653 IC50 > 30000 nM T20251 C8HXD1 25152860 IC50 > 30000 nM T20251 C7N4FW 25152862 IC50 > 30000 nM T20251 C68NWT 25153075 IC50 > 30000 nM T20251 CXC85P 25153077 IC50 = 1188 nM T20251 CZI56N 25153212 IC50 > 30000 nM T20251 CJW29T 25153282 IC50 = 12650 nM T20251 CR0EH4 25153700 IC50 > 30000 nM T20251 CH3M5P 25154041 IC50 = 3000 nM T20251 CI0E2L 25154395 IC50 = 2400 nM T20251 C4I1CJ 25155417 IC50 = 3000 nM T20251 CJVM09 25156194 Ki = 6600 nM T20251 C0TI3Z 25156476 Ki = 10000 nM T20251 CMX1W0 25156477 Ki = 220 nM T20251 C24UVQ 25156478 Ki = 870 nM T20251 C8AYP4 25156480 Ki = 620 nM T20251 C1HG2K 25156481 Ki = 2100 nM T20251 CKP4R2 25156482 Ki = 10000 nM T20251 CBM05I 25156750 Ki = 10000 nM T20251 C3QT7F 25156751 Ki = 10000 nM T20251 CJPO67 25156752 Ki = 10000 nM T20251 C7VC0P 25157642 IC50 > 5000 nM T20251 C7F1GA 25157660 IC50 = 3700 nM T20251 CP72MB 25159060 IC50 > 30000 nM T20251 CUAB05 25160153 IC50 = 1100 nM T20251 CGH08V 25164128 IC50 = 77.62 nM T20251 CW9MX8 25168440 IC50 > 10000 nM T20251 CYQ2X5 25170416 IC50 = 56 nM T20251 CZ28ES 25171661 IC50 > 32000 nM T20251 C5TJD2 25172265 IC50 > 30000 nM T20251 C94BLY 25173349 IC50 = 16000 nM T20251 C6AHF5 25174166 IC50 > 33000 nM T20251 CXG59Q 25175568 IC50 > 32000 nM T20251 C0YOQ7 25176461 IC50 = 9000 nM T20251 C1JL9X 25176462 IC50 = 5500 nM T20251 CL0Z1F 25181502 IC50 = 13000 nM T20251 C5C7GH 25184832 IC50 > 50118.72 nM T20251 C52BNH 25186023 Ki = 210 nM T20251 CJF9H4 25186569 Ki = 200 nM T20251 CG6NC3 25186839 Ki = 160 nM T20251 C3J8FK 25189510 IC50 = 95.5 nM T20251 CX4MV0 25190195 IC50 = 467.74 nM T20251 C1SX2E 25190435 IC50 = 630.96 nM T20251 CRS71Z 25190875 IC50 = 2700 nM T20251 C4AE8F 25190876 IC50 > 3000 nM T20251 CIR2T7 25190877 IC50 > 3000 nM T20251 C4XIE6 25190878 IC50 > 3000 nM T20251 CMZ83A 25190879 IC50 = 350 nM T20251 CG49HK 25190880 IC50 = 630 nM T20251 CHN5O0 25190977 IC50 = 10400 nM T20251 CV3TA6 25192021 IC50 > 3000 nM T20251 C7A8UE 25192471 IC50 > 3000 nM T20251 CH3L6V 25192656 IC50 > 30000 nM T20251 C6NA1J 25194889 IC50 = 178 nM T20251 C08QMV 25195086 Ki = 37.2 nM T20251 CD4L9N 25195087 Ki = 23.9 nM T20251 CNI57D 25195088 Ki > 100 nM T20251 CO8QV5 25195089 Ki > 100 nM T20251 CBK27L 25196164 IC50 > 30000 nM T20251 C19CNW 25196320 IC50 > 33000 nM T20251 C0MQ7R 25196433 IC50 > 33000 nM T20251 CHS15A 25196434 IC50 > 33000 nM T20251 C3F5HA 25196664 IC50 > 33000 nM T20251 CF2O6Z 25196665 IC50 > 33000 nM T20251 C58AOY 25196773 IC50 > 33000 nM T20251 CM5V0Q 25197117 IC50 > 31000 nM T20251 CF0O3T 25197227 IC50 > 33000 nM T20251 CT5P4U 25204216 IC50 = 700 nM T20251 CTQM87 25210756 IC50 > 100000 nM T20251 C2UQJ6 25211598 EC50 > 30000 nM T20251 CKI86X 25211805 EC50 > 30000 nM T20251 CHW2X0 25211910 EC50 > 30000 nM T20251 CK0AM3 25216601 IC50 > 30000 nM T20251 C3PZ7E 25216602 IC50 > 30000 nM T20251 CJ1Z9H 25216680 IC50 = 7400 nM T20251 C6EO8B 25216683 IC50 = 17000 nM T20251 CXK8C2 25217299 IC50 = 32500 nM T20251 CA8RO1 25217406 IC50 = 11300 nM T20251 CLHN01 25217407 IC50 = 8800 nM T20251 CT67WG 25217408 IC50 = 9300 nM T20251 CW7RJ2 25218015 IC50 = 300 nM T20251 CT3LJ6 25218017 IC50 = 140 nM T20251 C0VI2J 25218142 IC50 = 8800 nM T20251 C1T3LR 25218143 IC50 = 8200 nM T20251 C8RCG2 25218267 IC50 = 11000 nM T20251 C6VNQ4 25218268 IC50 = 16000 nM T20251 C0ONJ9 25218269 IC50 = 29000 nM T20251 CU63JR 25218271 IC50 = 6200 nM T20251 CPI03N 25218397 IC50 = 11000 nM T20251 C4GSU5 25218398 IC50 = 2500 nM T20251 CL1R3Q 25218401 IC50 = 9600 nM T20251 CN6XA4 25218555 IC50 = 1597 nM T20251 CL8K9U 25218556 IC50 = 1492 nM T20251 C9WA4B 25218557 IC50 = 183 nM T20251 CRG29Y 25218558 IC50 = 167 nM T20251 CEH71M 25218560 IC50 = 25090 nM T20251 C15YDI 25218563 IC50 = 12390 nM T20251 C9X6YJ 25229646 IC50 > 30000 nM T20251 CNF50T 25229676 Ki > 10000 nM T20251 C6FG0Q 25242540 IC50 > 30000 nM T20251 C53PTZ 25256089 IC50 > 10000 nM T20251 C90OGX 25256781 Ki = 5030 nM T20251 C2XS0Y 25256782 Ki = 903 nM T20251 CW9JM2 25256832 IC50 > 100000 nM T20251 C3GC7P 25256833 IC50 = 52000 nM T20251 C1IW5M 25261456 IC50 > 10000 nM T20251 CM81QH 25262336 IC50 > 32000 nM T20251 C20QHN 25262627 IC50 = 24200 nM T20251 C5E3ZH 25265089 IC50 = 37000 nM T20251 C20SGN 25265312 IC50 = 480 nM T20251 C5BNH3 25265516 IC50 = 18900 nM T20251 C7PK2X 29938807 IC50 > 33000 nM T20251 C60RHJ 30634189 IC50 = 320 nM T20251 CR6Q3D 34598448 IC50 = 24000 nM T20251 CJ8V4H 34681379 IC50 = 22900 nM T20251 C4GSR9 35901875 IC50 = 2238.72 nM T20251 CTI9S6 42601404 Ki = 2990 nM T20251 CQR2J6 42601405 Ki > 7200 nM T20251 CBQO98 42602095 IC50 = 7200 nM T20251 CJ61SE 42602096 IC50 = 6495 nM T20251 CI42XG 42602097 IC50 = 2600 nM T20251 CD2AH4 42602175 IC50 = 57793 nM T20251 CSWA85 42602176 IC50 > 100000 nM T20251 C1LUN4 42602178 IC50 > 100000 nM T20251 C8O3EA 42602260 IC50 > 100000 nM T20251 C93NKL 42602264 IC50 > 100000 nM T20251 C7WPJ5 42602351 IC50 > 33300 nM T20251 C2FZ9P 42606792 IC50 > 80000 nM T20251 CKH3P1 42606928 IC50 = 1900 nM T20251 CIH75Y 42615261 IC50 > 30000 nM T20251 C1YO7H 42618040 EC50 = 12000 nM T20251 CGU3N8 42618068 EC50 = 8000 nM T20251 CY4LG8 42622934 IC50 = 22000 nM T20251 CI1C5U 42623163 IC50 = 4000 nM T20251 CV3FM2 42625548 IC50 = 900 nM T20251 CZ96KC 42625549 IC50 = 2500 nM T20251 C1U5IS 42625550 IC50 = 60 nM T20251 C9GPZ5 42625636 IC50 = 500 nM T20251 C4C5QJ 42625708 IC50 = 1300 nM T20251 C5XVB9 42625945 IC50 = 1200 nM T20251 CZ4V2A 42625948 IC50 = 1200 nM T20251 C2VA7M 42625949 IC50 = 500 nM T20251 CQ1YN9 42626020 IC50 = 40 nM T20251 C7K6PG 42626023 IC50 = 3500 nM T20251 CJ8LY0 42626024 IC50 = 1000 nM T20251 CRQ91B 42626318 IC50 = 380 nM T20251 CNU7P4 42630820 IC50 > 10000 nM T20251 C1CWU0 42631007 IC50 = 6850 nM T20251 CW24IK 42633780 IC50 = 700 nM T20251 C75GFD 42633960 IC50 > 10000 nM T20251 C57VJY 42635854 IC50 = 3400 nM T20251 CP8RA7 42635855 IC50 = 3000 nM T20251 CG0E4V 42635876 IC50 = 17782.79 nM T20251 C05BWT 42635901 IC50 = 8200 nM T20251 CY5E4B 42635983 IC50 = 1700 nM T20251 C8V6IK 42635984 IC50 = 990 nM T20251 C34DCR 42636018 IC50 = 750 nM T20251 C1J4XZ 42636222 IC50 > 30000 nM T20251 C9PL8Z 42641334 Ki = 5000 nM T20251 C6MX0U 42641453 IC50 = 4500 nM T20251 CZM36T 42641892 IC50 = 1400 nM T20251 CA5TW1 42641905 Ki = 2200 nM T20251 CQS4U7 42642010 Ki = 680 nM T20251 CIX54O 42642011 Ki = 1000 nM T20251 CRYH80 42642459 IC50 = 2700 nM T20251 CZF5G9 42916879 IC50 > 50000 nM T20251 C0VC7J 43314210 IC50 = 20000 nM T20251 CYV94L 43314375 IC50 = 4560 nM T20251 CXYI49 44121506 IC50 > 33000 nM T20251 CS40ML 44123747 IC50 = 30000 nM T20251 CD61KH 44125830 IC50 = 95499.26 nM T20251 CPB8S3 44125832 IC50 = 18197.01 nM T20251 C1BT4A 44129293 IC50 = 3162.28 nM T20251 C1HZK2 44135978 IC50 = 3300 nM T20251 C1HRC7 44135979 IC50 = 3300 nM T20251 CA7HI4 44137226 IC50 = 2100 nM T20251 CSX10M 44138030 IC50 = 18000 nM T20251 CXZH39 44138098 Ki = 2511.89 nM T20251 CG73ST 44138103 IC50 > 30000 nM T20251 CUOD42 44138104 Ki = 3981.07 nM T20251 CSM1A0 44138577 IC50 = 490 nM T20251 C4VYG8 44138579 IC50 > 10000 nM T20251 C3WOD7 44138581 IC50 > 10000 nM T20251 C4P8OL 44138706 IC50 > 10000 nM T20251 CW2G7S 44138708 IC50 = 7800 nM T20251 C7H3NP 44138709 IC50 > 10000 nM T20251 CU4XB0 44139234 IC50 = 1730 nM T20251 CDF14X 44139355 IC50 = 490 nM T20251 C4Q9IL 44139356 IC50 > 10000 nM T20251 CG3KU0 44139478 IC50 > 10000 nM T20251 CXR3J2 44139479 IC50 = 4330 nM T20251 CW8J0K 44139480 IC50 > 10000 nM T20251 COJK15 44139481 IC50 = 6930 nM T20251 CX17RC 44139599 IC50 = 6330 nM T20251 CY0GQ3 44139600 IC50 > 10000 nM T20251 CVCH41 44139601 IC50 > 10000 nM T20251 C79OCX 44139602 IC50 > 10000 nM T20251 C9Z0RV 44139603 IC50 > 10000 nM T20251 C2U9ES 44139732 IC50 = 6300 nM T20251 C49YRK 44143406 IC50 = 23 nM T20251 C6U7HP 44143413 IC50 = 23 nM T20251 CAB3T9 44143415 IC50 = 2900 nM T20251 CG3PW7 44143417 IC50 = 23000 nM T20251 CB94OV 44143418 IC50 = 2700 nM T20251 COP5W8 44143419 IC50 = 16000 nM T20251 C3S1PL 44143422 IC50 = 9000 nM T20251 CQE5U4 44143426 IC50 = 1200 nM T20251 CZR49E 44143427 IC50 = 30000 nM T20251 C63RXB 44143428 IC50 = 29000 nM T20251 C8OH4S 44143429 IC50 = 21000 nM T20251 CTE6S1 44143430 IC50 = 23000 nM T20251 CL57VS 44143431 IC50 = 41000 nM T20251 C2C5QW 44143432 IC50 = 1500 nM T20251 C6GDL8 44143433 IC50 > 10000 nM T20251 C3BNV0 44143434 IC50 = 4900 nM T20251 CXV0B8 44143435 IC50 = 3000 nM T20251 CN7HE0 44143436 IC50 = 8500 nM T20251 C9CJN0 44143437 IC50 = 11000 nM T20251 C6INT4 44143438 IC50 = 990 nM T20251 CJ46YA 44143439 IC50 > 10000 nM T20251 C0KB7Y 44143441 IC50 > 10000 nM T20251 C3RF4I 44143442 IC50 > 10000 nM T20251 C5NZM3 44143446 IC50 = 3900 nM T20251 CGSW03 44143448 IC50 > 10000 nM T20251 CBWD06 44143449 IC50 > 10000 nM T20251 C2ST5N 44143450 IC50 > 10000 nM T20251 CF4V5K 44143451 IC50 > 10000 nM T20251 CL3R6D 44143452 IC50 > 10000 nM T20251 C8IG1V 44143453 IC50 = 4400 nM T20251 C2Q3DE 44143454 IC50 = 6300 nM T20251 CZX75A 44143455 IC50 = 380 nM T20251 C02YJQ 44143456 IC50 = 3400 nM T20251 CZV0C7 44143457 IC50 > 10000 nM T20251 C6TND7 44155109 IC50 = 8400 nM T20251 CN5G6U 44156749 IC50 = 100 nM T20251 C2C4NJ 44156750 IC50 = 7400 nM T20251 C6UOJ1 44157408 IC50 > 10000 nM T20251 CAS7T0 44157572 IC50 > 10000 nM T20251 CHI65U 44159530 IC50 > 30000 nM T20251 CE3OF9 44160137 IC50 = 750 nM T20251 CU2PO5 44180522 IC50 = 25118.86 nM T20251 CPF50A 44184875 IC50 = 17000 nM T20251 C2XE7Y 44189733 IC50 = 25000 nM T20251 C1ML3E 44190627 IC50 > 10000 nM T20251 C2AV1K 44190762 IC50 = 3230 nM T20251 CP06EY 44199337 IC50 = 28000 nM T20251 CJ7AF4 44203948 IC50 = 5000 nM T20251 CMR7T1 44204999 IC50 = 79.43 nM T20251 C4TMP9 44205087 IC50 > 30000 nM T20251 CX54AP 44215433 IC50 = 4400 nM T20251 CT29ZS 44216196 Ki = 2702 nM T20251 C2KJB0 44216880 IC50 = 1400 nM T20251 CUQ4T9 44217080 EC50 = 7943.28 nM T20251 CCJ3S4 44222256 Ki = 4650 nM T20251 CE0U8G 44222257 Ki = 7900 nM T20251 CC3XR6 44222258 Ki = 22500 nM T20251 CRNL71 44225654 Ki = 2900 nM T20251 C3MR8P 44229544 IC50 > 10000 nM T20251 CGPI02 44229545 IC50 > 10000 nM T20251 C83NXZ 44229546 IC50 > 10000 nM T20251 CQ4TG8 44229547 IC50 = 8300 nM T20251 CUVJ20 44229621 IC50 = 1600 nM T20251 CB5P7N 44230873 IC50 > 30000 nM T20251 CIBR82 44231149 IC50 > 10000 nM T20251 CX4YL8 44232522 IC50 > 30000 nM T20251 CMKQ59 44233027 IC50 = 19400 nM T20251 CQ13MH 44234032 IC50 > 30000 nM T20251 C7UY5F 44235863 IC50 > 30000 nM T20251 CX2W8Y 44236320 IC50 = 8000 nM T20251 C8LN0U 44236321 IC50 = 25000 nM T20251 CK4S5Y 44236322 IC50 = 6000 nM T20251 C75UQR 44236568 IC50 > 25000 nM T20251 CK7F2E 44240743 IC50 = 1300 nM T20251 C4W0SH 44247585 IC50 = 3200 nM T20251 C7MY2N 44247806 IC50 = 1400 nM T20251 CF9TE1 44247935 IC50 = 1200 nM T20251 CJ8RW5 44249745 IC50 = 7943.28 nM T20251 CLX51J 44249749 IC50 = 50118.72 nM T20251 C7QS6G 44250210 IC50 = 11400 nM T20251 C64ASH 44250211 IC50 = 26600 nM T20251 C85DHY 44250284 Ki = 18 nM T20251 C8P2LE 44250288 IC50 = 4900 nM T20251 C2K0VZ 44253016 IC50 > 63095.73 nM T20251 CY0QB9 44253226 IC50 = 3810 nM T20251 C1O8LH 44253973 IC50 = 12653 nM T20251 CMD87L 44254048 IC50 = 7000 nM T20251 C47RZO 44254057 IC50 = 2543 nM T20251 C41MNG 44254058 IC50 = 1261 nM T20251 C2SVL6 44254059 IC50 = 5132 nM T20251 CVW13I 44254060 IC50 = 3463 nM T20251 C0NZW8 44254061 IC50 = 71666 nM T20251 C3N2KB 44254062 IC50 = 4485 nM T20251 CJW3P2 44254063 IC50 = 4243 nM T20251 CXA10D 44254307 IC50 = 1918.03 nM T20251 C6OJS0 44254504 IC50 = 3190 nM T20251 CSBD48 44254505 IC50 = 23070 nM T20251 C1IPQ6 44254506 IC50 = 10566 nM T20251 CTL57U 44254584 IC50 = 54256 nM T20251 CZY2S1 44254585 IC50 = 1571 nM T20251 C9SQ8D 44254859 IC50 > 100000 nM T20251 CB47EJ 44254954 IC50 = 6809 nM T20251 C79QBX 44254955 IC50 = 3027 nM T20251 CVCP62 44254956 IC50 = 3501 nM T20251 CK7B1Q 44254957 IC50 = 13500 nM T20251 CJH6K5 44255041 IC50 = 6429 nM T20251 C5Z9KH 44255042 IC50 = 18471 nM T20251 C1FE8D 44255043 IC50 > 100000 nM T20251 CGB3A7 44255044 IC50 = 3794 nM T20251 CTY9U6 44255045 IC50 = 418 nM T20251 CZXC86 44267871 IC50 = 4360 nM T20251 CLC2O3 44294224 Ki = 1200 nM T20251 CO37IY 44294481 Ki = 1900 nM T20251 CV80DA 44294519 Ki = 400 nM T20251 C37OCJ 44294535 Ki = 460 nM T20251 CLHM64 44294659 Ki = 2200 nM T20251 CK7E2B 44294660 Ki = 490 nM T20251 CR2W3U 44294689 Ki = 1400 nM T20251 CCB5Y4 44296949 IC50 = 457.09 nM T20251 CE1S8X 44297083 IC50 = 36.31 nM T20251 CDSI60 44297084 IC50 = 10000 nM T20251 CE9H3D 44297095 IC50 = 2200 nM T20251 CP0T8C 44297148 IC50 = 10000 nM T20251 CD74SU 44297164 IC50 = 26000 nM T20251 CG9E7X 44297171 IC50 = 23.44 nM T20251 CR92VP 44297212 IC50 = 10000 nM T20251 CSX1R4 44297356 IC50 = 1947 nM T20251 C1VF2S 44297363 IC50 = 15848.93 nM T20251 C71ZUL 44297364 IC50 = 4570881.9 nM T20251 C96MUT 44297365 IC50 = 1480 nM T20251 C4MRW5 44297377 IC50 = 75000 nM T20251 C2FSL4 44297378 IC50 = 131 nM T20251 C5ZYX2 44297395 IC50 = 575.44 nM T20251 C3PX0Q 44297409 IC50 = 137 nM T20251 C0LT3N 44297410 IC50 = 87.1 nM T20251 C09HMY 44305854 Ki = 600 nM T20251 CMIB37 44306212 Ki > 10000 nM T20251 C70XSQ 44317802 Ki = 42200 nM T20251 C9AV2P 44326600 IC50 = 5888.44 nM T20251 CKSO92 44360724 Ki > 100000 nM T20251 CYED53 44360725 Ki = 5700 nM T20251 C50NME 44360749 Ki = 40000 nM T20251 CXTP74 44360787 Ki > 100000 nM T20251 C5MB1D 44360809 Ki = 17000 nM T20251 C29DTA 44360810 Ki = 29000 nM T20251 CR7Q9N 44360911 Ki = 5900 nM T20251 C6IZ8L 44360955 Ki = 22000 nM T20251 CY8A9K 44361010 Ki = 1900 nM T20251 CMU02Q 44364616 Ki = 20 nM T20251 C1XOB5 44387732 Ki = 1525 nM T20251 CL54KN 44387733 Ki = 398 nM T20251 C80WKC 44387740 Ki = 6800 nM T20251 CROA61 44387743 Ki = 9971 nM T20251 C1M5OY 44387746 Ki = 2446 nM T20251 CK36VZ 44387776 Ki > 9000 nM T20251 CC0WK5 44387777 Ki > 9000 nM T20251 CQ9WS8 44387780 Ki = 397 nM T20251 CY09ES 44396504 IC50 > 30000 nM T20251 C4X2OS 44396541 IC50 = 76800 nM T20251 CY80RP 44396542 IC50 = 800 nM T20251 C16MBG 44401760 IC50 < 10000 nM T20251 CC4O3R 44402387 IC50 = 180 nM T20251 C08LKH 44402452 IC50 = 30 nM T20251 CFA9P3 44402564 IC50 = 151.36 nM T20251 CXJ0Z6 44402597 IC50 = 40 nM T20251 CZI0A4 44405840 IC50 = 3.2 nM T20251 CH7Z3D 44407321 Ki = 4800 nM T20251 CFU2S7 44407325 Ki = 240 nM T20251 CE2R3O 44407331 Ki = 420 nM T20251 CHO57T 44407370 Ki = 190 nM T20251 CS21QZ 44407422 Ki > 5000 nM T20251 CLG2U0 44407427 Ki = 360 nM T20251 CUTS73 44407431 Ki > 6000 nM T20251 CCQX09 44407459 Ki > 6000 nM T20251 C9B4AK 44407467 Ki = 1400 nM T20251 CDPQ01 44407513 Ki = 270 nM T20251 CRB41P 44408123 Ki = 798 nM T20251 CQPK26 44408124 Ki = 1996 nM T20251 C92YHJ 44408144 Ki = 984 nM T20251 C35UHG 44408158 Ki = 3706 nM T20251 CF05TZ 44408176 Ki = 327 nM T20251 CA94TU 44408177 Ki = 947 nM T20251 CK4IB0 44408290 Ki = 1946 nM T20251 CDK7W3 44408291 Ki = 2987 nM T20251 CTM53U 44408295 Ki = 6529 nM T20251 CJE43Y 44408313 Ki = 862 nM T20251 COH25L 44409031 IC50 = 40000 nM T20251 CWX62Y 44409096 IC50 = 21000 nM T20251 CG87PW 44409290 IC50 > 30000 nM T20251 CB91NT 44409718 IC50 = 7800 nM T20251 C5YP1R 44409879 IC50 = 7800 nM T20251 CKI20Y 44409884 IC50 = 15000 nM T20251 C39MWE 44409885 IC50 = 6600 nM T20251 CF8A0Z 44409903 IC50 = 8500 nM T20251 CYO7B5 44409904 IC50 = 5600 nM T20251 C7BM2G 44409905 IC50 = 18000 nM T20251 CP10EK 44410155 Ki = 1300 nM T20251 C3YC0E 44410191 Ki = 1930 nM T20251 C5I4SO 44410193 Ki = 100 nM T20251 CY69JU 44410194 Ki = 1250 nM T20251 C5QG1S 44410207 Ki = 3150 nM T20251 CVB31D 44410278 Ki = 1800 nM T20251 CKWZ76 44410281 Ki = 2800 nM T20251 CQ8T0X 44410283 Ki > 10000 nM T20251 CYT96G 44410317 Ki > 5000 nM T20251 CYP37K 44410821 Ki = 150 nM T20251 CJI8T3 44410823 Ki = 150 nM T20251 C01JXU 44410838 Ki = 160 nM T20251 C1LYC9 44410849 Ki = 88 nM T20251 CGF17I 44410876 Ki = 135 nM T20251 CF0O7N 44410878 Ki = 1800 nM T20251 CL1XV7 44410904 Ki = 310 nM T20251 C4P5TW 44410944 Ki > 2000 nM T20251 CAO78Q 44411663 Ki > 9000 nM T20251 C8NVH0 44411664 Ki > 9000 nM T20251 C2Y8VK 44411667 Ki > 9000 nM T20251 C38VWG 44411668 Ki = 4869 nM T20251 C5Z2IY 44411674 Ki > 9000 nM T20251 CU2EY5 44411847 Ki > 9000 nM T20251 CD0OH1 44411864 Ki > 9000 nM T20251 CTLN43 44411929 Ki > 9000 nM T20251 CKX6D2 44411930 Ki > 9000 nM T20251 CQ89KF 44411933 Ki > 9000 nM T20251 CCJ1S9 44411934 Ki > 9000 nM T20251 CL28ZA 44411935 Ki > 9000 nM T20251 CG13DQ 44411936 Ki > 9000 nM T20251 CUB0V6 44412159 Ki > 9000 nM T20251 CO82EW 44412173 Ki = 1800 nM T20251 CACE19 44412207 Ki > 9000 nM T20251 CV4KZ7 44412225 Ki > 9000 nM T20251 CHF80Z 44412226 Ki > 9000 nM T20251 CCD01F 44412235 Ki = 1400 nM T20251 CECW41 44412236 Ki > 9000 nM T20251 C1D7YV 44412245 Ki > 9000 nM T20251 CH04GP 44412373 Ki = 5400 nM T20251 CYK1I6 44412374 Ki = 6700 nM T20251 CK5O6Q 44412445 Ki = 2400 nM T20251 CW71MS 44412453 Ki > 9000 nM T20251 C6R2ID 44412493 Ki = 8500 nM T20251 CDT7U5 44414663 IC50 > 24000000 nM T20251 CQD2S5 44414696 IC50 = 10900 nM T20251 C5Y4NH 44415354 IC50 = 170 nM T20251 C0OG4J 44415524 IC50 = 2600 nM T20251 CG1WM8 44417887 IC50 = 3300 nM T20251 CK76AM 44417889 IC50 = 3300 nM T20251 CPE50S 44417890 IC50 = 5860 nM T20251 CQS6G2 44417891 IC50 = 1700 nM T20251 CAK9U7 44417893 IC50 = 4000 nM T20251 C35KLS 44417895 IC50 = 5000 nM T20251 CL5XO4 44417897 IC50 = 25000 nM T20251 CM9QI8 44417899 IC50 = 14600 nM T20251 CI16UJ 44417902 IC50 = 26700 nM T20251 C8GK5Q 44417904 IC50 = 1800 nM T20251 C9BDI1 44417906 IC50 = 20000 nM T20251 C3GW2E 44417908 IC50 = 24000 nM T20251 CN2G7U 44417910 IC50 = 25000 nM T20251 CPDW02 44417913 IC50 = 10000 nM T20251 CY46AB 44417914 IC50 = 25000 nM T20251 C5HA7X 44417916 IC50 = 14000 nM T20251 CW1D3V 44417919 IC50 = 2600 nM T20251 C3CM4J 44417922 IC50 = 5100 nM T20251 CH0T1F 44417923 IC50 = 11000 nM T20251 C4WU0N 44417924 IC50 = 13000 nM T20251 CE96RJ 44417926 IC50 = 5200 nM T20251 C27PHW 44417927 IC50 = 13200 nM T20251 CT0B1U 44417929 IC50 = 2000 nM T20251 CH08OA 44417936 IC50 = 85200 nM T20251 CH3QM1 44417938 IC50 = 60700 nM T20251 CP1U0Z 44417939 IC50 = 5790 nM T20251 C7CP8I 44417993 IC50 = 20000 nM T20251 C6Q7ZM 44418004 IC50 = 6700 nM T20251 CVF74L 44418464 IC50 = 5151.52 nM T20251 C04THX 44418471 IC50 = 28461.54 nM T20251 CS6PZ7 44418472 IC50 = 19411.76 nM T20251 C9XDL2 44418473 IC50 = 52500 nM T20251 C49MQF 44418477 IC50 = 12222.22 nM T20251 CQ2D0O 44418482 IC50 = 101111.11 nM T20251 CPTD84 44418489 IC50 = 37619.05 nM T20251 CX09NV 44418490 IC50 = 66923.08 nM T20251 C68QUP 44418491 IC50 = 115000 nM T20251 CV5PD9 44418497 IC50 = 115000 nM T20251 CU8B2E 44418498 IC50 = 52500 nM T20251 C6YX3F 44418499 IC50 = 22258.06 nM T20251 CUH08F 44418511 IC50 = 40000 nM T20251 CR9EN2 44418522 Ki = 5100 nM T20251 C2S4RW 44418978 Ki = 1800 nM T20251 C93VJL 44418979 Ki = 6500 nM T20251 C16FUK 44418980 Ki = 510 nM T20251 CS08LV 44418981 Ki = 530 nM T20251 CP9VN3 44418982 Ki = 2500 nM T20251 CS5EY1 44418983 Ki = 8000 nM T20251 CHF36T 44418984 Ki = 2000 nM T20251 CF1A6T 44418985 Ki > 9000 nM T20251 C85GLF 44418986 Ki > 9000 nM T20251 CHS73F 44418998 Ki = 3000 nM T20251 C1FM8H 44419014 Ki = 8900 nM T20251 C5MT2W 44419015 Ki = 880 nM T20251 C7GY8W 44419017 Ki = 520 nM T20251 CW1DP9 44419019 Ki = 8200 nM T20251 C9H0DC 44419033 Ki > 9000 nM T20251 CT9U3N 44419048 Ki = 370 nM T20251 CR4SW2 44419049 Ki = 51 nM T20251 CP92ZY 44419050 Ki = 600 nM T20251 CO78NZ 44419051 Ki > 10000 nM T20251 CP85IH 44419052 Ki > 10000 nM T20251 C7OI8A 44419059 Ki = 4900 nM T20251 CCY70M 44419061 Ki = 840 nM T20251 C8PJ6U 44419062 Ki = 320 nM T20251 CCIF05 44419082 Ki = 71 nM T20251 CZNH91 44419083 Ki = 17 nM T20251 CRM0E4 44419084 Ki > 10000 nM T20251 CUI95V 44419085 Ki > 10000 nM T20251 C9LPR4 44419087 Ki > 10000 nM T20251 CQR29N 44419088 Ki = 880 nM T20251 CSQ5G8 44419089 Ki > 10000 nM T20251 COJ27C 44419090 Ki = 1400 nM T20251 CJ0W7B 44419091 Ki = 1400 nM T20251 C8LV0Y 44419092 Ki = 140 nM T20251 CDN8K7 44419097 Ki > 2000 nM T20251 C1A0LP 44419098 Ki = 1000 nM T20251 C3LE0S 44419101 Ki = 1600 nM T20251 C1VCN7 44419103 Ki = 89 nM T20251 CQ7PD9 44419104 Ki > 10000 nM T20251 C06ELF 44419105 Ki = 71 nM T20251 C7XKO9 44419106 Ki > 6600 nM T20251 CPL39F 44419108 Ki = 4600 nM T20251 CID32E 44419109 Ki = 200 nM T20251 C7HDX0 44419112 Ki = 570 nM T20251 C54KZH 44419113 Ki > 10000 nM T20251 C0J4HZ 44419117 Ki > 10000 nM T20251 CX5NU8 44419120 Ki = 790 nM T20251 CSIJ84 44419121 Ki > 10000 nM T20251 COV56X 44419122 Ki > 10000 nM T20251 CXZ2L3 44421702 IC50 = 5360 nM T20251 CT0J7Z 44421703 IC50 = 1410 nM T20251 CT03MH 44424972 Ki = 3.6 nM T20251 CEA35L 44424973 Ki = 7300 nM T20251 C3U2GQ 44424974 Ki = 160 nM T20251 CRV85N 44424975 Ki = 18 nM T20251 C4IRD2 44424976 Ki = 13 nM T20251 C7HW6E 44424977 Ki = 7 nM T20251 CDXQ90 44424979 Ki = 19 nM T20251 CXS4T5 44424981 Ki = 10 nM T20251 CIH6L7 44424983 Ki = 15 nM T20251 C53YCH 44424984 Ki = 89 nM T20251 C42IGZ 44424985 Ki > 1000 nM T20251 C6JW9A 44425428 Ki = 24000 nM T20251 CU43XH 44425429 Ki = 106000 nM T20251 C1JS6T 44425430 Ki > 150000 nM T20251 C2OSP1 44425431 Ki > 150000 nM T20251 CSR6M2 44425432 Ki = 64000 nM T20251 C02HMN 44425433 Ki > 100000 nM T20251 CUWC08 44425434 Ki > 100000 nM T20251 CZ7IT9 44425435 Ki > 150000 nM T20251 CI94RJ 44425436 Ki = 72000 nM T20251 CH6B9Z 44425437 Ki > 100000 nM T20251 C5Y6CS 44425438 Ki > 150000 nM T20251 C8OR0K 44425439 Ki > 150000 nM T20251 C56HGJ 44425440 Ki = 112000 nM T20251 CL0DM4 44425441 Ki > 150000 nM T20251 C53ELI 44425442 Ki = 45000 nM T20251 CCRH08 44428207 IC50 = 251.19 nM T20251 CTD5N2 44430312 IC50 > 30000 nM T20251 CON04H 44430571 IC50 = 7100 nM T20251 CCBR69 44430578 IC50 = 15900 nM T20251 C9GIE3 44433617 IC50 > 100000 nM T20251 C6VLC5 44433700 IC50 > 30000 nM T20251 CM0FX1 44433701 IC50 > 30000 nM T20251 CN24TK 44433702 IC50 > 10000 nM T20251 C1QH9B 44433704 IC50 > 30000 nM T20251 CWL6Z1 44433706 IC50 > 30000 nM T20251 C3CS8V 44433710 IC50 > 30000 nM T20251 C6UVW9 44433711 IC50 > 30000 nM T20251 CKVG69 44433749 IC50 > 30000 nM T20251 CEX75D 44435377 IC50 = 15900 nM T20251 CJ1ST3 44437610 Ki = 56 nM T20251 CY9IK3 44438461 Ki = 98.1 nM T20251 C6W2EZ 44438462 Ki = 261 nM T20251 C9IFR5 44438464 Ki = 205 nM T20251 CUB30F 44438465 Ki = 693 nM T20251 CE36YV 44438467 Ki = 709 nM T20251 CLWE65 44438469 Ki = 525 nM T20251 CI93VE 44438472 Ki = 1300 nM T20251 CXD9B1 44438473 Ki = 410 nM T20251 C0QEB9 44438474 Ki = 222 nM T20251 C9T7JL 44438740 IC50 = 65000 nM T20251 CB9S3W 44438741 IC50 = 4300 nM T20251 CL20OD 44438742 IC50 = 1600 nM T20251 CG3PZ7 44438744 IC50 = 34000 nM T20251 C71UWM 44438745 IC50 = 740 nM T20251 CBJ5R9 44438747 IC50 = 3200 nM T20251 C5VFD8 44438748 IC50 = 450 nM T20251 CW8GU6 44438753 IC50 = 6300 nM T20251 CS9D3H 44438755 IC50 = 6600 nM T20251 CQ18PR 44439374 Ki > 9000 nM T20251 CN9RH5 44439375 Ki > 9000 nM T20251 C2X1FS 44439377 Ki > 9000 nM T20251 CW2KQ1 44439378 Ki = 4200 nM T20251 C2J9LG 44439379 Ki = 4800 nM T20251 COKH57 44439380 Ki = 5000 nM T20251 CO20GU 44439381 Ki = 1500 nM T20251 C4KQ8C 44439384 Ki = 1400 nM T20251 CQXS03 44439385 Ki = 2900 nM T20251 C1R0DN 44441341 Ki > 7500 nM T20251 C2GAV7 44441348 IC50 = 2900 nM T20251 C61VKY 44441350 IC50 = 1600 nM T20251 CF4A8D 44441351 IC50 = 2400 nM T20251 CD30KT 44441353 IC50 = 1200 nM T20251 CG5KW9 44442083 IC50 > 30000 nM T20251 COX3Q2 44442283 IC50 = 3300 nM T20251 C2X7NQ 44442481 IC50 = 2600 nM T20251 CAC7V9 44442482 IC50 = 2400 nM T20251 CVO5Z2 44442483 IC50 = 1600 nM T20251 CJPR25 44442484 IC50 = 7400 nM T20251 C9NMQ3 44442485 IC50 = 3100 nM T20251 CLX76D 44442486 IC50 = 16000 nM T20251 CZF32M 44442487 IC50 = 3300 nM T20251 C8S9AX 44442488 IC50 = 10000 nM T20251 C01RSY 44442489 IC50 < 1500 nM T20251 CGM63L 44442490 IC50 < 1000 nM T20251 C83FXU 44442491 IC50 = 11000 nM T20251 C52VPZ 44443347 IC50 = 1800 nM T20251 C7M0HV 44443354 IC50 = 165000 nM T20251 CUG6X5 44443360 IC50 = 10000 nM T20251 CP7WL5 44443363 IC50 = 28900 nM T20251 CPN7J9 44443420 IC50 > 300000 nM T20251 CXQP15 44443798 IC50 = 5300 nM T20251 CUHO63 44443803 IC50 = 13200 nM T20251 CIH69B 44445848 IC50 = 800 nM T20251 C5RVE0 44446999 Ki = 101 nM T20251 C9E0FL 44447001 Ki = 616 nM T20251 CSJ4U5 44447002 Ki = 164 nM T20251 CL87PU 44447003 Ki = 196 nM T20251 CCD6B5 44447005 Ki = 35 nM T20251 CBH65G 44447007 Ki = 278 nM T20251 C8CF7X 44447008 Ki = 272 nM T20251 CN3EH7 44447010 Ki = 194 nM T20251 CYWP06 44447012 Ki = 166 nM T20251 C41KNM 44447013 Ki = 78 nM T20251 CE12BC 44447015 Ki = 358 nM T20251 CUD31L 44447018 Ki = 201 nM T20251 CNLX79 44447028 Ki = 511 nM T20251 CM8K1H 44447039 Ki = 35 nM T20251 C5IJW2 44447059 Ki = 150 nM T20251 CHXF10 44447061 Ki = 143 nM T20251 CG93OH 44447063 Ki = 184 nM T20251 C9KJR2 44447065 Ki = 269 nM T20251 C5QK8Z 44447067 Ki = 137 nM T20251 C7A6RP 44447068 Ki = 219 nM T20251 CM8P9A 44447070 Ki = 135 nM T20251 CK4HA6 44447072 Ki = 202 nM T20251 C9EM8Q 44447733 IC50 = 410 nM T20251 CX89DC 44447734 IC50 = 2000 nM T20251 CI8Q9M 44447766 IC50 = 16 nM T20251 C50JFH 44447775 IC50 = 45 nM T20251 CWY54R 44447782 IC50 = 217 nM T20251 C2UGM9 44447783 IC50 = 67 nM T20251 CSLU08 44447786 IC50 = 2786 nM T20251 CRV6F7 44447789 IC50 = 19720 nM T20251 CDI1F4 44447815 IC50 = 186 nM T20251 C5K8ZM 44447866 IC50 > 100000 nM T20251 C8W5YG 44447872 IC50 > 100000 nM T20251 CRO52K 44448053 Ki = 180 nM T20251 CJC38Z 44449333 Ki > 7500 nM T20251 COP8A3 44449880 IC50 = 5610 nM T20251 CGR0B6 44452775 IC50 > 20000 nM T20251 CDS52W 44453970 IC50 = 47000 nM T20251 CB1MX2 44454118 IC50 = 6309.57 nM T20251 CR3IC6 44454120 IC50 = 31622.78 nM T20251 C5B0IF 44454150 IC50 = 1584.89 nM T20251 CRD82N 44454166 IC50 = 3981.07 nM T20251 CMVS90 44454167 IC50 > 15848.93 nM T20251 C7FY1E 44454168 IC50 = 6309.57 nM T20251 CW4S3P 44454190 IC50 = 1995.26 nM T20251 C7H3CL 44454192 IC50 = 12589.25 nM T20251 CU0N1E 44454217 IC50 = 398.11 nM T20251 C9DBA3 44454218 IC50 = 12589.25 nM T20251 CK01QH 44454219 IC50 = 2511.89 nM T20251 CLO6X0 44454223 IC50 = 10000 nM T20251 CECR53 44454247 IC50 = 630.96 nM T20251 CD4ZU7 44454248 IC50 = 2511.89 nM T20251 CS2N1D 44454275 IC50 = 6309.57 nM T20251 CJ5XB1 44454278 IC50 = 63.1 nM T20251 C4GON0 44454309 IC50 = 6.31 nM T20251 C91PHS 44454318 IC50 = 1995.26 nM T20251 CT50UC 44454320 IC50 = 5011.87 nM T20251 C35WYK 44454339 IC50 = 2511.89 nM T20251 CZO96M 44454340 IC50 = 39810.72 nM T20251 C2CIO7 44454351 IC50 = 251.19 nM T20251 C9AH1O 44454352 IC50 = 794.33 nM T20251 CM8H2G 44454353 IC50 = 2511.89 nM T20251 C1EZP7 44454358 IC50 = 12589.25 nM T20251 CEB84V 44454371 IC50 = 50118.72 nM T20251 C5EV7Z 44454381 IC50 = 2511.89 nM T20251 CWC92Y 44454382 IC50 = 1584.89 nM T20251 CH0S2F 44454384 IC50 = 251.19 nM T20251 C32LHE 44454400 IC50 = 31622.78 nM T20251 CG18KC 44454401 IC50 = 251.19 nM T20251 CI0CJ9 44454402 IC50 = 50118.72 nM T20251 CP34QH 44454403 IC50 > 3981.07 nM T20251 CW4OX5 44454418 IC50 = 3162.28 nM T20251 CW1I4Z 44454420 IC50 = 12589.25 nM T20251 CXA7W2 44454458 IC50 = 398.11 nM T20251 CBGJ08 44454459 IC50 = 1258.93 nM T20251 C32WLZ 44454571 IC50 = 5700 nM T20251 C2Q0EH 44454597 IC50 = 6800 nM T20251 CL6KS1 44454834 IC50 > 3000 nM T20251 C6YQU9 44455589 Ki = 1590 nM T20251 C9PG3H 44455590 Ki = 7250 nM T20251 C1BR2G 44455619 Ki > 7500 nM T20251 CO1X6Z 44455620 Ki = 3751 nM T20251 C8F5CI 44455622 Ki = 3866 nM T20251 C4Z0WX 44455645 IC50 = 11000 nM T20251 C0EM9R 44455651 Ki = 1556 nM T20251 C3W1EZ 44455653 Ki = 2213 nM T20251 CI4K0E 44455654 Ki > 7500 nM T20251 CZV45C 44455655 Ki = 1757 nM T20251 C0L9YB 44455677 Ki > 7500 nM T20251 CV10IJ 44455678 Ki > 7500 nM T20251 CIW6A1 44455707 Ki = 5932 nM T20251 C3CXW8 44455739 Ki > 7500 nM T20251 CO4B1F 44455740 Ki = 4380 nM T20251 CBID06 44455782 IC50 = 12000 nM T20251 C02DNS 44456907 IC50 = 100000000 nM T20251 C3LQ5I 44456908 IC50 = 20417379.45 nM T20251 C05PZX 44456916 IC50 = 512861384 nM T20251 CG7E3Q 44456934 IC50 = 2951209.23 nM T20251 CB46NK 44456935 IC50 = 97723722.1 nM T20251 CVA46I 44456948 IC50 = 1412.54 nM T20251 COF1S4 44456951 IC50 = 85113803.82 nM T20251 CJ4NR1 44456970 IC50 = 645654229 nM T20251 CVB17U 44456974 IC50 = 66069344.8 nM T20251 CI71FO 44456993 IC50 = 446.68 nM T20251 C2MN1I 44456997 IC50 = 64565422.9 nM T20251 CT5H0R 44457009 IC50 = 100 nM T20251 C7VG4S 44457011 IC50 = 512861384 nM T20251 CNBT41 44457012 IC50 = 37153522.91 nM T20251 CX5IE3 44457029 IC50 = 758577575 nM T20251 CM0IE4 44457030 IC50 = 33113112.15 nM T20251 CTCQ07 44457046 IC50 = 81.28 nM T20251 C6HN4F 44457047 IC50 = 251188643.2 nM T20251 CRSI16 44457089 IC50 = 537031796.4 nM T20251 C2XZN7 44457090 IC50 = 45.71 nM T20251 CE6U0F 44457093 IC50 = 20.89 nM T20251 CW06YM 44457095 IC50 = 28183829.31 nM T20251 CPK1J7 44457105 IC50 = 2.512 nM T20251 CZEY35 44457108 IC50 = 43651583.22 nM T20251 CRPN60 44457141 IC50 = 158489319.3 nM T20251 CM65QS 44457156 IC50 = 6165950.02 nM T20251 CBSZ02 44458521 Ki = 43000 nM T20251 CIA6J1 44458523 Ki = 37000 nM T20251 C6LKZ7 44458534 Ki = 42000 nM T20251 CM65HC 44458548 Ki = 5300 nM T20251 CKM0F5 44458549 Ki = 6000 nM T20251 CC7I6Y 44458573 Ki = 73000 nM T20251 CF7I9V 44458586 Ki = 39000 nM T20251 CW7QX0 44458587 Ki = 16000 nM T20251 CJ7Y6A 44458592 Ki = 5500 nM T20251 C9QMB2 44458594 Ki > 90000 nM T20251 CPJW14 44458603 Ki > 90000 nM T20251 C0K2SV 44458617 Ki > 90000 nM T20251 CSIL15 44458629 Ki = 19000 nM T20251 C3EZ1V 44458770 Ki = 28000 nM T20251 CGT38B 44462719 Ki = 18000 nM T20251 CL9O8M 44462783 IC50 = 1970 nM T20251 C8WM0Z 44467183 IC50 = 44000 nM T20251 C5ETU8 44467185 IC50 = 19000 nM T20251 C7UDS1 44467360 IC50 = 1900 nM T20251 CQ0WM7 44469273 IC50 = 4200 nM T20251 C2KMI6 44469322 IC50 > 30000 nM T20251 C2QK4J 44472590 IC50 = 11200 nM T20251 CQ8C3F 44472591 IC50 = 2000 nM T20251 CC2TA5 44472592 IC50 > 30000 nM T20251 CWN95E 44472610 IC50 > 30000 nM T20251 C1H2ZT 44472612 IC50 > 30000 nM T20251 C9G5ID 44472613 IC50 > 30000 nM T20251 C5N4KE 44472633 IC50 > 30000 nM T20251 CJ39UE 44473168 Ki = 6800 nM T20251 C3CX0V 44475155 IC50 > 33000 nM T20251 C5RNK0 44476261 IC50 = 8600 nM T20251 CXY7T9 44476436 IC50 = 54200 nM T20251 C6V2YR 44476607 IC50 = 500 nM T20251 C6O0ZQ 44476624 IC50 = 34000 nM T20251 C6AK3W 44476911 IC50 > 30000 nM T20251 CLDQ43 44476913 IC50 > 30000 nM T20251 CG3R4T 44477000 IC50 = 14000 nM T20251 CDZP10 44479308 Ki = 950 nM T20251 CXJN29 44479309 Ki > 29000 nM T20251 C4Y5GO 44479310 Ki = 23000 nM T20251 CJDX78 44479549 IC50 > 10000 nM T20251 CJ25FS 44479563 Ki > 29000 nM T20251 C4CPX0 44479566 Ki = 15000 nM T20251 CI7EX6 44479809 Ki > 29000 nM T20251 C7C1HW 44481057 IC50 = 8100 nM T20251 C1FTA7 44481065 Ki > 29000 nM T20251 CVW53Z 44481067 Ki = 13000 nM T20251 C5COJ1 44481316 Ki = 4800 nM T20251 C8TIN9 44481318 Ki = 28000 nM T20251 CC2Q0J 44481321 Ki = 11000 nM T20251 C3NI0V 44481584 IC50 > 10000 nM T20251 C9U1KA 44481856 IC50 > 10000 nM T20251 CCA93X 44481857 IC50 > 10000 nM T20251 C13ZGK 44481860 Ki > 29000 nM T20251 CR3TH8 44481861 Ki = 17000 nM T20251 CW1ZR7 44481862 Ki = 7600 nM T20251 C8O9PY 44482139 Ki = 18000 nM T20251 CB0O7Y 44482409 Ki = 5000 nM T20251 C7XV2J 44512857 Ki = 28000 nM T20251 C5PI4H 44515310 Ki = 14 nM T20251 C1H8NX 44516817 IC50 > 30000 nM T20251 CFAZ41 44517710 IC50 = 16000 nM T20251 C68NXC 44517723 IC50 > 10000 nM T20251 C9OY3U 44517726 IC50 = 3162.28 nM T20251 C83JWO 44517778 IC50 = 3100 nM T20251 CS9H0L 44517795 IC50 > 100000 nM T20251 CSO35V 44520546 IC50 = 31622.78 nM T20251 C3Q5LP 44525560 IC50 = 3000 nM T20251 C9N1BU 44539192 IC50 > 15000 nM T20251 C01UWF 44540282 IC50 > 33000 nM T20251 CWP9Q3 44540283 IC50 = 17000 nM T20251 CKCG52 44540374 IC50 = 11000 nM T20251 C46HBA 44540470 IC50 = 23000 nM T20251 C2MF7Z 44540754 IC50 = 14000 nM T20251 C5O4TM 44540839 IC50 = 22000 nM T20251 CV92IJ 44541354 IC50 = 38.5 nM T20251 C6IK7J 44541892 IC50 = 33000 nM T20251 C16HIP 44542338 IC50 = 8700 nM T20251 C2B6OY 44542339 IC50 = 14100 nM T20251 CQ4W7V 44542340 IC50 = 14300 nM T20251 CD4LN9 44543781 IC50 = 21000 nM T20251 CS10AL 44543784 IC50 = 9300 nM T20251 C17LUC 44543889 IC50 = 14000 nM T20251 C9X2SL 44543890 IC50 = 26000 nM T20251 CE6HW8 44543891 IC50 > 33000 nM T20251 C27TZY 44543970 IC50 > 30000 nM T20251 CB83EJ 44544123 IC50 = 31000 nM T20251 CN64WQ 44544347 IC50 = 4600 nM T20251 CQ79RB 44544349 IC50 = 8600 nM T20251 CSV3F9 44544441 IC50 = 9200 nM T20251 C0RI5Z 44544444 IC50 = 7300 nM T20251 CK8T7U 44544546 IC50 = 8900 nM T20251 COJ7H6 44544644 IC50 = 5100 nM T20251 CYJB15 44544645 IC50 = 5500 nM T20251 C8RAF0 44544851 IC50 = 5500 nM T20251 CWKZ36 44544853 IC50 = 16000 nM T20251 C6AX2C 44544950 IC50 = 3300 nM T20251 CGB50M 44545053 IC50 = 9700 nM T20251 CU16DA 44545166 IC50 = 3600 nM T20251 CW78UO 44545168 IC50 = 4300 nM T20251 CNZ12F 44545169 IC50 = 5600 nM T20251 C5KZ2M 44545289 IC50 = 6600 nM T20251 C9JK4V 44545402 IC50 = 8200 nM T20251 C6L8QO 44545403 IC50 = 5600 nM T20251 CK1Z8P 44545482 IC50 > 30000 nM T20251 CX13MK 44547414 IC50 > 100000 nM T20251 CGLQ31 44552634 IC50 = 20000 nM T20251 CTX13C 44555196 IC50 = 16000 nM T20251 CUQ0J7 44555369 Ki > 13000 nM T20251 CJE2Q6 44555375 IC50 = 280 nM T20251 CT5N4E 44555481 IC50 = 11900 nM T20251 C4LJ6X 44557554 IC50 > 31600 nM T20251 C1EVH2 44560678 IC50 = 2143 nM T20251 CI58CZ 44560679 IC50 = 2500 nM T20251 CC4Z5M 44560681 IC50 = 10000 nM T20251 CWOM65 44560715 IC50 > 10000 nM T20251 C7YCO3 44560716 IC50 > 10000 nM T20251 C5X7PO 44560717 IC50 = 4800 nM T20251 COTH35 44560718 IC50 = 6100 nM T20251 C6J0ZC 44560719 IC50 = 7400 nM T20251 CL0A2D 44560720 IC50 = 3500 nM T20251 CR8K0X 44560724 IC50 = 9800 nM T20251 CE08JD 44560725 IC50 > 10000 nM T20251 CSX84T 44560726 IC50 = 9100 nM T20251 C1O0IG 44560727 IC50 = 6000 nM T20251 CB7X4S 44560728 IC50 = 8300 nM T20251 C94LIO 44560729 IC50 > 10000 nM T20251 C3UQ8C 44560730 IC50 > 10000 nM T20251 C8OD4F 44560731 IC50 = 4700 nM T20251 CLB20U 44560732 IC50 > 10000 nM T20251 CC01KM 44561020 IC50 = 13000 nM T20251 C4SVU2 44561370 IC50 = 740 nM T20251 CRJM24 44561454 IC50 = 7800 nM T20251 CXJK43 44561493 IC50 = 13000 nM T20251 CY14MD 44561518 IC50 = 86 nM T20251 CR8OX1 44562611 IC50 = 1780 nM T20251 CL64BM 44562612 IC50 = 2110 nM T20251 CVB0Q6 44562613 IC50 = 3040 nM T20251 C02CWF 44562614 IC50 = 2110 nM T20251 C7CSF8 44562615 IC50 = 873 nM T20251 CNJM41 44562616 IC50 = 1230 nM T20251 C3VP6N 44562943 IC50 = 1740 nM T20251 C7DS0M 44562944 IC50 = 10400 nM T20251 C4XL2E 44562989 IC50 = 3880 nM T20251 C5J6HU 44563054 IC50 = 3010 nM T20251 CZW0B1 44563061 IC50 = 4700 nM T20251 CT9S4L 44563063 IC50 = 460 nM T20251 C2HJ9Z 44563066 IC50 = 7000 nM T20251 C83CZN 44563067 IC50 > 32000 nM T20251 C97AJO 44563111 IC50 = 20000 nM T20251 CL3MW0 44563112 IC50 = 11000 nM T20251 C6B2FI 44563127 IC50 = 4800 nM T20251 CL0DS9 44563128 IC50 = 5440 nM T20251 CDTB89 44563137 IC50 = 350 nM T20251 C51TLU 44563144 IC50 = 10000 nM T20251 CNR1B2 44563145 IC50 = 3000 nM T20251 C0D1LO 44563146 IC50 = 20000 nM T20251 C0J2GS 44563163 IC50 = 3210 nM T20251 C67TOD 44563164 IC50 = 3030 nM T20251 CL5HW8 44563165 IC50 = 2690 nM T20251 CJV9S8 44563177 IC50 = 6000 nM T20251 CV90NH 44563178 IC50 > 32000 nM T20251 CDX3R8 44563203 IC50 = 785 nM T20251 C5QX2S 44563204 IC50 = 5110 nM T20251 CF4ZK8 44563205 IC50 = 1640 nM T20251 C3ZUH6 44563206 IC50 = 1150 nM T20251 CJ9O6U 44563238 IC50 = 645 nM T20251 CB8P3I 44563239 IC50 = 3690 nM T20251 CB9NG8 44563240 IC50 = 2470 nM T20251 CN5U4V 44563241 IC50 = 5230 nM T20251 CLJ7C2 44563242 IC50 = 3120 nM T20251 C2OX9D 44563243 IC50 = 4790 nM T20251 C1VQ5X 44563244 IC50 = 1060 nM T20251 CU9J5W 44564565 IC50 > 100000 nM T20251 C3MNR0 44565080 IC50 > 10000 nM T20251 CF6JG1 44565081 IC50 > 10000 nM T20251 CA0FC1 44565082 IC50 = 2300 nM T20251 C6DI0T 44565083 IC50 = 2100 nM T20251 CV1IL5 44565796 IC50 = 70000 nM T20251 C9SL5D 44565872 IC50 > 10000 nM T20251 COA7X5 44565892 IC50 = 54000 nM T20251 C3YE7P 44567441 IC50 = 11 nM T20251 C46KUB 44568231 IC50 = 1200 nM T20251 COTQ47 44568792 IC50 = 3034 nM T20251 CWLT20 44570180 IC50 > 63000 nM T20251 C1W9AF 44570584 IC50 = 15700 nM T20251 CXHT91 44571305 IC50 = 6000 nM T20251 CR32XZ 44571307 IC50 = 17000 nM T20251 CIV48S 44572053 IC50 = 2018 nM T20251 CZM8O6 44573159 Ki = 3410 nM T20251 CVSJ62 44573160 Ki = 3690 nM T20251 CF0A2J 44573161 Ki = 2090 nM T20251 C13LFI 44573162 Ki = 3430 nM T20251 C7HZJ6 44573224 Ki = 5240 nM T20251 CO4NI2 44573249 Ki = 17 nM T20251 C9OF8P 44573250 Ki = 169 nM T20251 CPJ27Z 44573251 Ki = 35 nM T20251 CIK5T2 44573291 Ki = 201 nM T20251 CM89KA 44573292 Ki = 82 nM T20251 CI6F0Y 44573293 Ki = 343 nM T20251 CL6C7B 44573294 Ki = 548 nM T20251 CBM82T 44573332 Ki > 10000 nM T20251 CMSV07 44573403 Ki = 1840 nM T20251 CLX14F 44573404 Ki > 10000 nM T20251 C0PD8L 44573405 Ki = 9690 nM T20251 CA03TK 44573444 Ki > 10000 nM T20251 CZ26TO 44573445 Ki = 865 nM T20251 CQ9WA5 44573446 Ki = 518 nM T20251 CKJ2O8 44573447 Ki = 746 nM T20251 CNUJ50 44574003 IC50 > 10000 nM T20251 C1T4QN 44574053 IC50 = 2000 nM T20251 C5LJ0D 44577963 IC50 = 1380 nM T20251 CFJB16 44578266 Ki > 2700 nM T20251 CML90U 44578389 IC50 = 710 nM T20251 CD1U2S 44578570 IC50 = 5500 nM T20251 C1MC0I 44578615 IC50 = 18000 nM T20251 CFAW91 44578616 IC50 = 8400 nM T20251 CYPJ70 44578617 IC50 > 24000 nM T20251 CR0F7I 44578649 IC50 > 32000 nM T20251 C9E6QP 44579079 IC50 = 5770 nM T20251 C7CKG9 44579080 IC50 = 1455 nM T20251 CH5B0N 44579120 IC50 = 420 nM T20251 CN42GY 44579121 IC50 = 710 nM T20251 CDUJ10 44579122 IC50 = 360 nM T20251 CQJ0L6 44579123 IC50 = 540 nM T20251 CO13BP 44579170 IC50 = 890 nM T20251 CP0X4D 44579171 IC50 = 2340 nM T20251 CS60PG 44579172 IC50 = 5040 nM T20251 CY2E6M 44579173 IC50 > 30000 nM T20251 C4RNV0 44580338 Ki = 26 nM T20251 CE87QS 44580381 Ki = 94 nM T20251 C9B2LH 44580383 Ki = 49 nM T20251 C3L5ER 44583033 IC50 = 11800 nM T20251 CTO9G3 44583367 IC50 > 30000 nM T20251 CL62PK 44588589 IC50 = 198 nM T20251 CMI7N1 44588590 IC50 = 680 nM T20251 CP9QH1 44588591 IC50 = 71500 nM T20251 CLZ05M 44588592 IC50 = 740 nM T20251 C09TKD 44589077 IC50 = 31800 nM T20251 CKU85Z 44589520 Ki = 14560 nM T20251 C9RA0C 44589548 EC50 > 30000 nM T20251 CT7F0N 44589856 Ki = 590 nM T20251 C3C6WU 44589911 Ki = 19250 nM T20251 CVA4I9 44589912 Ki > 10000 nM T20251 CVQ83W 44589913 Ki = 9800 nM T20251 CNBO74 44589970 EC50 = 3300 nM T20251 C0GQ2C 44589971 Ki = 760 nM T20251 C9OL3W 44590015 Ki = 1900 nM T20251 C5AWD8 44590016 Ki = 170 nM T20251 C0MLS4 44590017 Ki = 3200 nM T20251 CGP0W8 44590018 Ki = 97 nM T20251 C4C5AQ 44590111 Ki = 6300 nM T20251 CVZ23T 44590151 Ki > 10000 nM T20251 CDC86A 44590152 Ki = 9420 nM T20251 CJ0U5K 44590153 Ki = 8620 nM T20251 CB67HK 44590208 Ki = 10980 nM T20251 CRG54L 44590209 Ki = 8699 nM T20251 C1G2VQ 44590210 Ki = 9070 nM T20251 CJK1Q3 44590211 Ki = 7540 nM T20251 CU71HW 44590230 IC50 = 849 nM T20251 CE5U9X 44590439 IC50 = 3410 nM T20251 CS8ZR6 44590583 IC50 = 248 nM T20251 CRN4U5 44590696 IC50 = 86000 nM T20251 CIH56J 44590864 IC50 = 4.7 nM T20251 CZ5HT9 44590865 IC50 = 117 nM T20251 CAC12Y 44590943 IC50 = 3100 nM T20251 C2EB4O 44590944 IC50 < 5280 nM T20251 CHQM54 44590946 IC50 = 1650 nM T20251 C1OCI9 44591315 IC50 = 237 nM T20251 C7GL4H 44591704 Ki = 1020 nM T20251 C91FTW 44591848 IC50 = 85000 nM T20251 CY78PR 44591849 IC50 = 55000 nM T20251 CE2LW5 44591850 IC50 = 59000 nM T20251 CI6R1Z 44592120 Ki = 4500 nM T20251 C1QO8J 44592121 Ki = 10300 nM T20251 CVT6R5 44592123 Ki = 716 nM T20251 CV8E7O 44592155 Ki = 412 nM T20251 CMS5I2 44592158 Ki > 5000 nM T20251 C4EH6O 44592207 Ki = 100 nM T20251 CZ5I1N 44592208 Ki = 3162.28 nM T20251 CKM8T7 44592209 Ki = 7943.28 nM T20251 CJO9K5 44592245 Ki = 10100 nM T20251 CDJ32U 44592249 Ki = 5011.87 nM T20251 CS2FL4 44592250 Ki = 1584.89 nM T20251 CL17WU 44592251 Ki = 1584.89 nM T20251 CJCL64 44592252 Ki = 398.11 nM T20251 CO6ES5 44592257 IC50 = 7300 nM T20251 CM0I3E 44592294 Ki = 10000 nM T20251 CQ04EG 44592295 Ki = 12589.25 nM T20251 C65XQL 44592296 Ki = 3981.07 nM T20251 CEB2S1 44592297 Ki = 3162.28 nM T20251 CP51QS 44592332 Ki = 5011.87 nM T20251 CD2Z4J 44592333 Ki = 6309.57 nM T20251 C7NCT2 44592334 Ki = 6309.57 nM T20251 CHY20X 44592335 Ki = 3162.28 nM T20251 C5H7XK 44592371 Ki = 630.96 nM T20251 CI7G1T 44592534 IC50 = 7800.01 nM T20251 C69VSL 44592535 IC50 = 6000 nM T20251 COE58F 44592580 IC50 = 190 nM T20251 CP1U5K 44592598 IC50 = 1100 nM T20251 CCQ73Z 44592962 IC50 = 5800 nM T20251 C6HA0L 44592987 IC50 = 50000 nM T20251 CDP7R8 44592988 IC50 = 50000 nM T20251 CE62VG 44592989 IC50 = 20999.99 nM T20251 C21FGX 44592990 IC50 = 11000.01 nM T20251 CUX2C0 44593418 IC50 = 88 nM T20251 CDC59A 44593419 IC50 = 135 nM T20251 CSD5Z3 44593420 IC50 = 1930 nM T20251 CQ12YR 44593444 IC50 = 2120 nM T20251 C2U5KV 44593866 IC50 > 1000 nM T20251 CKTZ17 44594174 IC50 = 52000 nM T20251 C3CJW9 44595244 Ki = 637 nM T20251 C96MTQ 44595526 Ki = 5214 nM T20251 CF4YN8 44598057 IC50 = 1905.46 nM T20251 C9MT0V 44598058 IC50 = 1905.46 nM T20251 C71QNY 44598059 IC50 = 229.09 nM T20251 C9TH0G 44598060 IC50 = 11220.18 nM T20251 CZWY54 44598061 IC50 = 19498.45 nM T20251 CP27OH 44598062 IC50 = 38018.94 nM T20251 CS76XZ 44598121 IC50 = 16982.44 nM T20251 C0L4FZ 44598124 IC50 = 30902.95 nM T20251 CGQT32 44598769 IC50 = 19054.61 nM T20251 CG2SD8 44598819 IC50 = 2344.23 nM T20251 C27GZB 44598820 IC50 = 5128.61 nM T20251 CV9G1H 44598821 IC50 = 70.79 nM T20251 CM2UG7 44598902 IC50 = 6000 nM T20251 C84NFS 44599828 IC50 = 2400 nM T20251 CVJG25 44600846 IC50 = 4600 nM T20251 C89VRG 44605616 IC50 > 50118.72 nM T20251 CZD25I 44605617 IC50 > 50118.72 nM T20251 CEQN62 44609163 IC50 > 30000 nM T20251 C7G4FT 44609164 IC50 > 30000 nM T20251 CH9FO5 44609165 IC50 > 30000 nM T20251 CLPY85 44609168 IC50 > 30000 nM T20251 CU0QT2 44609322 IC50 = 23000 nM T20251 CQ06VN 44609327 IC50 > 30000 nM T20251 CE9GN6 44609485 IC50 > 30000 nM T20251 C9GWF1 44609645 IC50 = 7000 nM T20251 CI10GR 44610722 Ki = 1600 nM T20251 CW84TH 44610723 Ki = 3200 nM T20251 CPIB93 44610724 Ki = 11000 nM T20251 CDX2H1 44621189 IC50 = 15800 nM T20251 CO3I5F 44622849 Ki > 22000 nM T20251 C8B0HO 44622872 IC50 = 396 nM T20251 CZHP95 44626357 IC50 = 3700 nM T20251 C9N4MQ 44626527 IC50 = 1995.26 nM T20251 CSJ9F1 44626530 IC50 = 630.96 nM T20251 CCLQ67 44626632 IC50 = 794.33 nM T20251 CA93OY 44626637 IC50 = 251.19 nM T20251 CPML65 44626639 IC50 = 125.89 nM T20251 CDA90T 44626641 IC50 = 630.96 nM T20251 C2TBL0 44626734 IC50 = 630.96 nM T20251 C7LUV5 44626738 IC50 = 630.96 nM T20251 CRCL97 44626740 IC50 = 199.53 nM T20251 CZ25SY 44626744 IC50 = 630.96 nM T20251 C5DM7T 44626835 IC50 = 251.19 nM T20251 C85ZIF 44626928 IC50 = 158.49 nM T20251 C4BYG5 44626929 IC50 = 1000 nM T20251 CK5BG2 44626935 IC50 = 630.96 nM T20251 CWL84Q 44627022 IC50 = 1584.89 nM T20251 CGXJ71 44627023 IC50 = 630.96 nM T20251 CBP18J 44627024 IC50 = 398.11 nM T20251 C30KEM 44627025 IC50 = 398.11 nM T20251 CV1DO3 44627033 IC50 = 1258.93 nM T20251 CAH6O1 44627120 IC50 = 3981.07 nM T20251 CUE56O 44627123 IC50 = 110 nM T20251 CDY32E 44627127 IC50 = 1258.93 nM T20251 CJ4ZQ0 44627129 IC50 = 1995.26 nM T20251 CN1O6P 44627131 IC50 = 1000 nM T20251 CQE59L 44627133 IC50 = 3162.28 nM T20251 C4QV9Y 44627238 IC50 = 6309.57 nM T20251 C1D5FJ 44627240 IC50 = 199.53 nM T20251 CNK4P0 44627242 IC50 = 501.19 nM T20251 CY3LE2 44627245 IC50 = 398.11 nM T20251 C5LN9E 44627351 IC50 = 501.19 nM T20251 CLUN07 44627353 IC50 = 1258.93 nM T20251 CZ1FY5 44627355 IC50 = 3162.28 nM T20251 C3ZWA4 44627357 IC50 = 630.96 nM T20251 CY1TE0 44627358 IC50 = 1995.26 nM T20251 CG97OK 44627359 IC50 = 1000 nM T20251 C65RAG 44627466 IC50 = 1000 nM T20251 C06TJC 44627468 IC50 = 398.11 nM T20251 CBV8I6 44627470 IC50 = 1258.93 nM T20251 C7NIU3 44628133 IC50 = 50 nM T20251 CE6M8G 44628198 IC50 = 9960 nM T20251 CERD02 44628200 IC50 = 20 nM T20251 CIM8C4 44628201 IC50 = 10 nM T20251 C1XQ8G 44629350 IC50 = 1220 nM T20251 CMO1Z6 44631854 IC50 > 30000 nM T20251 CIX15W 44631974 IC50 > 90000 nM T20251 C37AQP 44815590 IC50 = 8500 nM T20251 CU8P7K 44815806 Ki = 28540 nM T20251 C4C9LB 44815976 Ki = 2500 nM T20251 C0LRQ2 45101475 IC50 = 19000 nM T20251 CSEP-69 45102708 IC50 > 15848.93 nM T20251 C32YHG 45102733 Ki = 200 nM T20251 C45PUQ 45102745 Ki = 4200 nM T20251 C4XAC1 45103619 IC50 > 30000 nM T20251 C4G7PQ 45104756 IC50 = 5740 nM T20251 CVCQ85 45104767 IC50 = 95000 nM T20251 C0DLU3 45109862 IC50 = 100 nM T20251 C40BIM 45139151 IC50 = 17700 nM T20251 C4KRT0 45254002 IC50 = 29300 nM T20251 CJ0Y1O 45254127 Ki > 10000 nM T20251 C8FQ9P 45254130 Ki > 10000 nM T20251 CQB45G 45254505 Ki > 10000 nM T20251 C1R3PL 45254506 Ki > 10000 nM T20251 C2JD1Y 45254508 Ki > 10000 nM T20251 C2YE7A 45254510 Ki > 10000 nM T20251 C2M9RC 45254900 Ki = 3280 nM T20251 CUL8G3 45255106 Ki > 15000 nM T20251 C43HDC 45256109 Ki = 660 nM T20251 C2Q3MJ 45256294 Ki = 1840 nM T20251 C5RQ2B 45256296 Ki = 410 nM T20251 C0Q2WV 45256478 Ki = 4980 nM T20251 C8H4SQ 45256479 Ki > 15000 nM T20251 CV32EW 45256653 Ki = 10700 nM T20251 C5LYK1 45256654 Ki = 1420 nM T20251 CE9IU1 45256823 Ki = 150 nM T20251 CI70YH 45256826 Ki = 1160 nM T20251 CT41IW 45256827 Ki > 15000 nM T20251 C1K0ZH 45259193 IC50 = 2511.89 nM T20251 C0C4FV 45265850 IC50 > 14000 nM T20251 CAHW68 45267251 IC50 = 5011.87 nM T20251 CW1S6B 45267254 IC50 = 3162.28 nM T20251 CD47IO 45267261 IC50 = 794.33 nM T20251 CJPS81 45267262 IC50 = 1995.26 nM T20251 C4HOR6 45267270 IC50 = 1995.26 nM T20251 CUT2B4 45267348 IC50 > 30000 nM T20251 CF4PM0 45267382 IC50 = 900 nM T20251 C1N5ZL 45267385 IC50 = 800 nM T20251 C4AZD3 45267386 IC50 = 3500 nM T20251 C8LPF5 45267399 IC50 = 2340 nM T20251 C8PR5X 45267430 IC50 > 31600 nM T20251 C3T5PI 45267459 IC50 = 2900 nM T20251 CPD18Y 45267471 IC50 = 12589.25 nM T20251 CL0WP4 45267480 IC50 = 63.1 nM T20251 C2H4ZX 45267491 IC50 = 794.33 nM T20251 C0KTX2 45267492 IC50 = 794.33 nM T20251 C2R9HN 45267503 IC50 = 2511.89 nM T20251 CEY87M 45267504 IC50 = 1584.89 nM T20251 CFY4R2 45267593 IC50 > 10000 nM T20251 CP7XE6 45267597 IC50 > 10000 nM T20251 CK58HY 45267611 IC50 = 9210 nM T20251 CM23AU 45267709 IC50 = 19600 nM T20251 CGB32I 45267714 IC50 = 3080 nM T20251 CO3Y0N 45267724 IC50 > 31600 nM T20251 CI7KZ2 45267735 IC50 = 5340 nM T20251 CC5OP0 45267739 IC50 = 12700 nM T20251 CXJ8H3 45267746 IC50 = 25800 nM T20251 CUEY48 45267808 IC50 = 14600 nM T20251 CF2R3T 45268112 IC50 = 1584.89 nM T20251 C3S5ZP 45268113 IC50 = 630.96 nM T20251 C0UG9Z 45268119 IC50 = 19952.62 nM T20251 C37TAV 45268120 IC50 = 1000 nM T20251 CP1TV2 45268127 IC50 = 31622.78 nM T20251 C79VFY 45268141 IC50 = 3981.07 nM T20251 C64NZQ 45268142 IC50 = 25118.86 nM T20251 CENZ75 45268148 IC50 = 6309.57 nM T20251 CJH3A2 45268206 IC50 > 30000 nM T20251 CTB32R 45268225 IC50 = 400 nM T20251 CP85WO 45268247 IC50 = 31000 nM T20251 C0XAR6 45268283 IC50 = 12 nM T20251 C7V1WF 45268290 IC50 = 4.4 nM T20251 C9RCS2 45268299 IC50 = 1000 nM T20251 CLF90U 45268300 IC50 = 1700 nM T20251 C2T0ZC 45268315 IC50 = 1300 nM T20251 CM1SA7 45268333 IC50 = 1000 nM T20251 CH53XO 45268345 IC50 = 7.943 nM T20251 CHB5U0 45268346 IC50 = 251.19 nM T20251 COCN89 45268373 IC50 = 6309.57 nM T20251 C4MU3C 45268438 IC50 = 3162.28 nM T20251 C4DZO1 45268459 IC50 > 10000 nM T20251 CRP90V 45268466 IC50 > 16300 nM T20251 CQ7J4A 45268477 IC50 > 10000 nM T20251 CSJ4L2 45268478 IC50 > 20000 nM T20251 C9IJK8 45268483 IC50 = 7400 nM T20251 C7UG6Q 45268498 IC50 = 15000 nM T20251 C7VZR5 45268637 IC50 = 20900 nM T20251 CV1IR5 45268644 IC50 > 31600 nM T20251 C9B5EH 45268653 Ki = 116 nM T20251 C18EGU 45268687 IC50 = 530 nM T20251 CUQ23Z 45268922 IC50 > 10000 nM T20251 CEK21M 45268987 IC50 = 10000 nM T20251 CHB76Z 45268990 IC50 = 3981.07 nM T20251 CR3YU9 45268999 IC50 = 3981.07 nM T20251 CW57CP 45269000 IC50 = 7943.28 nM T20251 CYQ1I7 45269020 IC50 = 199.53 nM T20251 C4WR0V 45269087 IC50 > 30000 nM T20251 CRPS25 45269096 IC50 = 27000 nM T20251 C7BNY6 45269104 IC50 = 6000 nM T20251 CC8P5K 45269117 IC50 = 480 nM T20251 C6ETI8 45269118 IC50 = 910 nM T20251 CX53RU 45269119 IC50 = 7000 nM T20251 CRN8Y1 45269121 IC50 = 1600 nM T20251 CVH8S4 45269235 IC50 = 3162.28 nM T20251 CED18G 45269300 IC50 > 10000 nM T20251 CZC09M 45269305 IC50 > 10000 nM T20251 CFJ17A 45269306 IC50 > 10000 nM T20251 CCQ8W4 45269310 IC50 = 6700 nM T20251 CNA70T 45269316 IC50 > 10000 nM T20251 C1SB8A 45269317 IC50 > 10000 nM T20251 C5OED7 45269318 IC50 > 20000 nM T20251 CF2P9H 45269325 IC50 > 20000 nM T20251 CQ03ZU 45269337 IC50 > 20000 nM T20251 CXE36D 45269351 IC50 > 7460 nM T20251 C78UOX 45269357 IC50 = 9900 nM T20251 C4WT5J 45269358 IC50 = 15000 nM T20251 C97ZET 45269449 IC50 = 780 nM T20251 CU02ZQ 45269860 IC50 = 1995.26 nM T20251 CS1Q2X 45269947 IC50 > 30000 nM T20251 C1BE5U 45269948 IC50 > 30000 nM T20251 CG1H9N 45269950 IC50 = 8200 nM T20251 CA3MZ6 45269996 IC50 = 14000 nM T20251 C5DIS2 45270014 IC50 = 1000 nM T20251 C8C2AK 45270025 IC50 = 25 nM T20251 C2L8JN 45270044 IC50 = 7000 nM T20251 CDM73H 45270136 IC50 = 2100 nM T20251 C2Q4SM 45270142 IC50 > 10000 nM T20251 CX31KD 45270149 IC50 = 1440 nM T20251 CLPB92 45270153 IC50 = 9000 nM T20251 CGXC75 45270156 IC50 > 10000 nM T20251 C3GA6N 45270158 IC50 > 18200 nM T20251 C3KI7Q 45270163 IC50 > 20000 nM T20251 C0QR1E 45270171 IC50 > 17600 nM T20251 C6YI5N 45270172 IC50 > 18500 nM T20251 CZ9DA3 45270173 IC50 = 2350 nM T20251 CA38NB 45270184 IC50 = 31000 nM T20251 CPG7D6 45270273 IC50 > 31600 nM T20251 C0J6BO 45270297 IC50 > 31600 nM T20251 C23PMF 45270302 IC50 > 31600 nM T20251 C9WNG1 45270303 IC50 = 7330 nM T20251 C4SXQ3 45270319 IC50 = 6900 nM T20251 C8GQ7J 45270330 Ki = 1461 nM T20251 C48BMQ 45270339 Ki > 7500 nM T20251 CS67XW 45270376 IC50 = 460 nM T20251 COFD89 45270589 IC50 = 6610 nM T20251 CEX26T 45270595 IC50 = 950 nM T20251 CF43XE 45270678 IC50 = 31622.78 nM T20251 CK01NU 45270702 IC50 = 12589.25 nM T20251 C1NT2M 45270771 IC50 > 30000 nM T20251 CA05IG 45270778 IC50 = 9000 nM T20251 CZ7MK9 45270788 IC50 = 7000 nM T20251 C0R5NB 45270796 IC50 = 4300 nM T20251 C3A0NB 45270802 IC50 = 630 nM T20251 C35TNH 45270803 IC50 = 1090 nM T20251 C3GLV8 45270841 IC50 = 2170 nM T20251 CD5OS6 45270850 IC50 > 31600 nM T20251 CUV67Q 45270855 IC50 = 11 nM T20251 C5UP2J 45270862 IC50 = 470 nM T20251 CEM4Z0 45270863 IC50 = 6300 nM T20251 C9GK5C 45270870 IC50 = 4800 nM T20251 CO0P8H 45270903 IC50 = 398.11 nM T20251 C7OM4D 45270916 IC50 = 50118.72 nM T20251 CZ9OC8 45270973 IC50 = 530 nM T20251 CB94YA 45270992 IC50 = 4700 nM T20251 C13QSU 45270993 IC50 > 16800 nM T20251 CU9HV3 45271001 IC50 = 2210 nM T20251 CBW87K 45271004 IC50 = 1300 nM T20251 C71AON 45271011 IC50 > 19000 nM T20251 C2G5XK 45271015 IC50 = 19000 nM T20251 CO05CL 45271041 IC50 = 3200 nM T20251 C42GYR 45271095 IC50 = 1810 nM T20251 C1F5RT 45271103 IC50 = 3000 nM T20251 CCN0F4 45271111 IC50 = 11700 nM T20251 CS9M8B 45271114 IC50 = 4120 nM T20251 CY70FL 45271134 IC50 = 1300 nM T20251 C18WQE 45271166 Ki > 5000 nM T20251 CMQ25P 45271491 IC50 = 1000 nM T20251 CEQ19M 45271499 IC50 = 2511.89 nM T20251 CESN63 45271510 IC50 = 1584.89 nM T20251 CMDC23 45271511 IC50 = 15848.93 nM T20251 C8TXI5 45271516 IC50 = 6309.57 nM T20251 C5P3FX 45271520 IC50 = 1584.89 nM T20251 CF9I3G 45271548 IC50 = 794.33 nM T20251 C9TM2P 45271593 IC50 > 30000 nM T20251 C06YAD 45271599 IC50 > 30000 nM T20251 CG0I8P 45271610 IC50 > 30000 nM T20251 C6FBH0 45271618 IC50 = 2600 nM T20251 C08OEP 45271626 IC50 = 830 nM T20251 C13PCQ 45271633 IC50 = 1600 nM T20251 C3OA8C 45271642 IC50 = 1550 nM T20251 CP7CX1 45271647 IC50 = 28000 nM T20251 CH1PS3 45271663 IC50 > 31600 nM T20251 CM4ZX1 45271673 IC50 = 1700 nM T20251 CN4W1B 45271701 IC50 = 440 nM T20251 CW0JQ7 45271712 IC50 = 2500 nM T20251 CAO92B 45271713 IC50 = 14000 nM T20251 C6R3LQ 45271737 IC50 = 1258.93 nM T20251 CM5Q8S 45271738 IC50 = 63.1 nM T20251 C42EJD 45271753 IC50 = 2511.89 nM T20251 CT3DP1 45271760 IC50 = 1584.89 nM T20251 CE8Z1K 45271821 IC50 = 520 nM T20251 C1L4DN 45271828 IC50 > 10000 nM T20251 CLD3T9 45271838 IC50 > 10000 nM T20251 C1S6TI 45271840 IC50 > 20000 nM T20251 C3QAP5 45271853 IC50 > 20000 nM T20251 CP7K0V 45271861 IC50 > 10000 nM T20251 CFG5Z3 45271864 IC50 > 20000 nM T20251 C36SRE 45271994 IC50 = 3870 nM T20251 C73LNM 45272006 IC50 = 3330 nM T20251 CMYT82 45272014 IC50 = 4890 nM T20251 C60DPZ 45272024 IC50 > 31600 nM T20251 C2MKZ1 45272040 IC50 > 31600 nM T20251 CU9C4I 45272046 Ki = 40 nM T20251 CAY8I7 45272070 Ki = 3536 nM T20251 C5U7LD 45272411 IC50 = 10000 nM T20251 CM9W5B 45272412 IC50 = 25118.86 nM T20251 CG9CO5 45272414 IC50 = 6309.57 nM T20251 C4W9NG 45272415 IC50 = 398.11 nM T20251 C12WFN 45272425 IC50 = 1258.93 nM T20251 CK67XC 45272426 IC50 = 3162.28 nM T20251 CQ2ZS6 45272434 IC50 = 12589.25 nM T20251 CGKZ21 45272435 IC50 = 19952.62 nM T20251 CH0MA8 45272437 IC50 = 63095.73 nM T20251 CW2MD0 45272438 IC50 = 3981.07 nM T20251 C71VIG 45272510 IC50 = 2000 nM T20251 C05EDY 45272511 IC50 = 27000 nM T20251 C5R7OL 45272520 IC50 = 540 nM T20251 C6FCW0 45272539 IC50 = 10000 nM T20251 CGV7P0 45272576 IC50 = 5 nM T20251 CR1F7A 45272583 IC50 = 1300 nM T20251 C1TLM4 45272592 IC50 = 3800 nM T20251 CE1P8L 45272616 IC50 = 1258.93 nM T20251 CEO57P 45272634 IC50 = 3162.28 nM T20251 CI7C1L 45272635 IC50 = 6309.57 nM T20251 C5DE4U 45272692 IC50 = 9600 nM T20251 CN3G7M 45272695 Ki = 130000 nM T20251 CPM1U3 45272720 IC50 > 20000 nM T20251 CJ52PS 45272816 IC50 = 2030 nM T20251 CT5KW9 45272826 IC50 = 6500 nM T20251 CD6FR7 45272837 IC50 = 2160 nM T20251 C3GUS5 45272853 IC50 > 31600 nM T20251 C62IGT 45272875 Ki = 57 nM T20251 C3GUK4 45272876 Ki = 73 nM T20251 CBE0M8 45272877 Ki = 158 nM T20251 CR04WH 45272878 Ki = 102 nM T20251 CZ7N8Q 45272889 Ki = 426 nM T20251 CK2B5U 45272890 Ki = 776 nM T20251 C8TC4R 45272894 Ki = 137 nM T20251 CA0SD1 45272895 IC50 = 809 nM T20251 CH17KU 45272913 IC50 = 65600 nM T20251 CPUR70 45272936 IC50 = 2200 nM T20251 CQ98IX 45272939 IC50 = 3800 nM T20251 CX1QY9 45273266 IC50 = 3162.28 nM T20251 C62LGY 45273272 IC50 = 1995.26 nM T20251 CZ2OL1 45273273 IC50 = 7943.28 nM T20251 CBM9R2 45273292 IC50 = 1258.93 nM T20251 CS04AC 45273293 IC50 = 15848.93 nM T20251 CS95IU 45273334 IC50 = 5011.87 nM T20251 CD62AH 45273373 IC50 > 30000 nM T20251 CMN39U 45273380 IC50 = 10000 nM T20251 C9JQT2 45273392 IC50 = 1020 nM T20251 CPTE06 45273401 IC50 = 11700 nM T20251 CG4YS2 45273406 IC50 = 4200 nM T20251 C0GK4R 45273485 IC50 = 6200 nM T20251 CFY94G 45273510 IC50 = 5011.87 nM T20251 CRSF80 45273522 IC50 = 1584.89 nM T20251 C3DB8P 45273523 IC50 = 199.53 nM T20251 CM10UD 45273529 IC50 = 79.43 nM T20251 CRD9C8 45273530 IC50 = 630.96 nM T20251 CNQJ09 45273545 IC50 = 1995.26 nM T20251 C7XC3T 45273551 IC50 = 3981.07 nM T20251 C1JLQ3 45273630 IC50 > 10000 nM T20251 C27VWT 45273649 IC50 = 900 nM T20251 C7HQ9B 45273656 IC50 > 10000 nM T20251 CT3V0B 45273663 IC50 > 13500 nM T20251 C58HQB 45273679 IC50 = 34000 nM T20251 CLFN69 45273777 IC50 = 4700 nM T20251 CP7OZ1 45273778 IC50 = 14700 nM T20251 COD72W 45273783 IC50 = 7930 nM T20251 CCJR41 45273790 IC50 = 3960 nM T20251 C3TZ8X 45273801 IC50 = 4040 nM T20251 CX9T5I 45273802 IC50 = 2840 nM T20251 C5E2XR 45273828 Ki = 157 nM T20251 CN4IE3 45275362 IC50 > 100000 nM T20251 C2GKC7 45278576 IC50 > 80000 nM T20251 C2J0GO 45278647 IC50 = 6800 nM T20251 CZ71RN 45278805 IC50 = 140 nM T20251 CZN6M7 45278882 IC50 = 540 nM T20251 C3NW0C 45279216 IC50 = 500 nM T20251 C7DXG1 45279490 IC50 = 5500 nM T20251 CR0N4Z 45279585 IC50 = 3000 nM T20251 C7XI9W 45279680 IC50 > 10000 nM T20251 C84XIH 45279772 IC50 = 3300 nM T20251 CJO30G 45279869 IC50 = 2000 nM T20251 CLX86A 45380509 IC50 = 11000 nM T20251 CL41HJ 45380693 IC50 = 3200 nM T20251 C9NCV4 45380694 IC50 = 3700 nM T20251 C6SZ8A 45380791 IC50 = 4800 nM T20251 CEM0V9 45380893 IC50 = 10000 nM T20251 CU7Z8X 45381216 IC50 > 33000 nM T20251 CWA35Y 45381330 IC50 = 16000 nM T20251 C5I3OG 45381546 IC50 = 5900 nM T20251 C9UF1Z 45381640 IC50 > 33000 nM T20251 CP3HD2 45381723 IC50 > 33000 nM T20251 C4AM7K 45381799 IC50 = 9100 nM T20251 CG1QY5 45381801 IC50 = 4600 nM T20251 CO4BT1 45381802 IC50 = 2700 nM T20251 CT21WU 45381890 IC50 = 12000 nM T20251 CWJM09 45381983 IC50 > 33000 nM T20251 C91UWI 45482679 IC50 = 204.08 nM T20251 CP1YN5 45482680 IC50 = 1363.64 nM T20251 CV56HF 45482684 IC50 = 6949.15 nM T20251 C2C1XZ 45482685 IC50 = 204.08 nM T20251 CA45ZR 45482686 IC50 = 2658.23 nM T20251 CGP38T 45482687 IC50 = 7543.86 nM T20251 CHV1Q5 45482688 IC50 = 323333.33 nM T20251 CK2G6S 45482693 IC50 = 6666.67 nM T20251 C9L4FG 45482694 IC50 = 1111.11 nM T20251 CEY8O1 45482699 IC50 = 989.01 nM T20251 C7W0DZ 45482705 IC50 = 19411.76 nM T20251 CP2ZT9 45482708 IC50 = 1111.11 nM T20251 CRL9I4 45482709 IC50 = 8181.82 nM T20251 C9UE0Y 45482713 IC50 = 101.01 nM T20251 C3P5TG 45482727 IC50 = 40000 nM T20251 CZM43G 45482728 IC50 = 190000 nM T20251 CB8E2S 45482734 IC50 = 196000 nM T20251 CDM1L4 45482735 IC50 = 80000 nM T20251 CEM05T 45482739 IC50 = 43000 nM T20251 C2LU1K 45482740 IC50 = 140000 nM T20251 CHQ4M5 45482745 IC50 = 23333.33 nM T20251 CJ3X8T 45482746 IC50 = 190000 nM T20251 C3NC6W 45482751 IC50 = 1235.96 nM T20251 CX9RG6 45482752 IC50 = 40000 nM T20251 C28XSF 45482753 IC50 = 8518.52 nM T20251 CZLA81 45482756 IC50 = 9607.84 nM T20251 CIH4Z3 45482757 IC50 = 6393.44 nM T20251 C4EIV8 45482763 IC50 = 132857.14 nM T20251 CE0H4S 45482770 IC50 = 1764.71 nM T20251 CLKA86 45482775 IC50 = 101.01 nM T20251 C2ED8W 45482783 IC50 = 309.28 nM T20251 C0CHF4 45482789 IC50 > 30000 nM T20251 C8YIM9 45483679 IC50 = 411 nM T20251 CE4LA5 45483880 IC50 = 11220.18 nM T20251 CX12QY 45483901 IC50 = 3467.37 nM T20251 C0TED2 45483913 IC50 = 4168.69 nM T20251 CMQ17N 45484111 IC50 = 5600 nM T20251 C5YT2N 45484113 IC50 = 4400 nM T20251 C85XBW 45484115 IC50 = 12200 nM T20251 C9D6SC 45484116 IC50 = 33000 nM T20251 CO42HZ 45484117 IC50 = 28300 nM T20251 CC8X7E 45485452 Ki = 431 nM T20251 C3AT2W 45485462 IC50 > 100000 nM T20251 CSQ1J5 45487336 IC50 > 10000 nM T20251 C3QU2C 45487384 IC50 = 5100 nM T20251 C24WVU 45487513 IC50 = 6309.57 nM T20251 CMX27T 45487640 IC50 = 530 nM T20251 C5NO1K 45487641 IC50 > 10000 nM T20251 CR10DI 45487647 IC50 = 17 nM T20251 CS17WK 45487652 IC50 = 24 nM T20251 CAQ2D8 45487653 IC50 = 3670 nM T20251 C3A7QW 45487657 IC50 = 23 nM T20251 CB9K2G 45487660 IC50 = 25 nM T20251 CJ8R3S 45487668 IC50 = 250 nM T20251 CN1V0Y 45487671 IC50 = 140 nM T20251 CWH0O7 45487673 IC50 = 520 nM T20251 CCZR81 45487674 IC50 = 1790 nM T20251 C80FMT 45487762 Ki = 4200 nM T20251 CR0X4I 45487870 Ki = 1600 nM T20251 CL32NJ 45488686 IC50 = 19000 nM T20251 C32YDN 46175430 IC50 = 50118.72 nM T20251 CH5Y4W 46175432 IC50 > 100000 nM T20251 C6MI2B 46175433 IC50 = 36000 nM T20251 CZ8SI1 46175518 IC50 = 19952.62 nM T20251 CR9J1S 46175520 IC50 = 62000 nM T20251 CZKB10 46175521 IC50 = 10000 nM T20251 CA6G8I 46175610 IC50 = 50118.72 nM T20251 C2L3HT 46175611 IC50 > 100000 nM T20251 C7CK6V 46178246 IC50 = 4800 nM T20251 CP12AF 46179404 IC50 > 30000 nM T20251 CS8TU3 46179405 IC50 > 30000 nM T20251 CR0I3A 46180744 IC50 = 8700 nM T20251 C7W2LJ 46180746 IC50 = 2200 nM T20251 CL7F3D 46187355 IC50 > 30000 nM T20251 CNDF17 46187356 IC50 > 80000 nM T20251 CZ8N7D 46197576 IC50 = 27600 nM T20251 CF9QB5 46197577 IC50 = 13400 nM T20251 CMK3H7 46197578 IC50 = 9100 nM T20251 C7IGB2 46197685 IC50 = 29300 nM T20251 C9T7FD 46197686 IC50 = 28400 nM T20251 C8IQ5Z 46197687 IC50 = 13500 nM T20251 CJZ3X6 46197795 IC50 = 19300 nM T20251 C7Z6JK 46197796 IC50 = 30000 nM T20251 C9Z6UF 46197797 IC50 = 9900 nM T20251 CFKV19 46197898 IC50 = 15300 nM T20251 CYAI40 46198106 IC50 = 20000 nM T20251 CTI0F8 46198107 IC50 > 80000 nM T20251 CJ9OY8 46198108 IC50 = 10000 nM T20251 CI9QH8 46198109 IC50 > 80000 nM T20251 CU3VQ1 46198110 IC50 = 7300 nM T20251 C2P9ST 46198216 IC50 = 38000 nM T20251 CSEL57 46198325 IC50 = 53000 nM T20251 C2VIF3 46198326 IC50 = 8600 nM T20251 C6JWH5 46198327 IC50 = 25900 nM T20251 C13RUW 46198329 IC50 = 26000 nM T20251 CRLM46 46201983 IC50 = 1000 nM T20251 C7VR2G 46202081 IC50 = 3500 nM T20251 C56SZE 46202415 IC50 = 7200 nM T20251 C38LWQ 46202743 IC50 = 3800 nM T20251 C4A5NH 46203391 IC50 = 2100 nM T20251 CFYP54 46203897 IC50 < 400 nM T20251 CBQ31T 46205018 IC50 > 100000 nM T20251 C9L4KT 46205341 IC50 > 333000 nM T20251 C4OK3I 46205343 IC50 > 333000 nM T20251 C1A5VL 46205345 IC50 > 333000 nM T20251 CX8OB9 46205674 IC50 = 174000 nM T20251 C9MPG6 46205967 IC50 = 5700 nM T20251 CNVX45 46205968 IC50 = 3100 nM T20251 CL41FE 46206000 IC50 > 333000 nM T20251 CR9A5G 46206291 IC50 = 16000 nM T20251 C9B1CG 46206292 IC50 = 7900 nM T20251 CSX8P1 46206294 IC50 = 1600 nM T20251 CD0R7T 46206296 IC50 = 500 nM T20251 C3X4KZ 46206324 IC50 > 333000 nM T20251 CR1X0F 46206642 IC50 = 11000 nM T20251 C8JYQ3 46206643 IC50 = 6400 nM T20251 C0R1YT 46206645 IC50 = 1700 nM T20251 CH8Y7D 46206977 IC50 = 2200 nM T20251 C9FI2Z 46208126 IC50 = 13000 nM T20251 CE45XW 46208354 IC50 = 360 nM T20251 CUHB49 46208355 IC50 = 7700 nM T20251 CW38GO 46208357 IC50 = 17000 nM T20251 C43COY 46208358 IC50 = 8100 nM T20251 CE4Q7D 46208596 IC50 = 4800 nM T20251 CM9UN7 46208601 IC50 > 100000 nM T20251 CMG47W 46208633 IC50 = 7500 nM T20251 CLUF01 46208857 IC50 = 6400 nM T20251 CO3Y7Q 46208858 IC50 = 12000 nM T20251 CH7JB4 46209051 IC50 > 100000 nM T20251 C0SNL2 46209134 IC50 = 21000 nM T20251 C5KFD3 46212800 IC50 > 33000 nM T20251 CB04XO 46212809 IC50 > 33000 nM T20251 C6U0CX 46212866 IC50 > 33000 nM T20251 CU6X8G 46213054 Ki = 690 nM T20251 CL51NF 46216732 Ki = 2560 nM T20251 CZJL95 46216733 Ki = 4910 nM T20251 C8BN4H 46216788 IC50 = 11000 nM T20251 C57OFD 46216800 IC50 = 12000 nM T20251 C3JUH5 46216812 IC50 = 8000 nM T20251 CPI8M7 46224242 IC50 = 5800 nM T20251 C0TYK4 46224262 IC50 = 8900 nM T20251 C26LPQ 46225987 IC50 = 9500 nM T20251 CHO7G1 46226010 IC50 = 15800 nM T20251 CDS61T 46226025 IC50 = 40100 nM T20251 CARU41 46226027 IC50 = 135000 nM T20251 CA2L5H 46227092 Ki = 4620 nM T20251 CLS58Y 46227093 Ki = 300 nM T20251 CH5VD2 46227102 Ki = 3000 nM T20251 C1DO4U 46230960 Ki = 3310 nM T20251 C59XOB 46230961 Ki = 1650 nM T20251 C9EGU1 46230962 Ki > 4760 nM T20251 C2FVA8 46231075 IC50 = 1540 nM T20251 CA3R5W 46231076 IC50 = 1720 nM T20251 CSZ2F6 46231077 Ki = 2110 nM T20251 CVL6C0 46231146 Ki > 5190 nM T20251 C8W4VL 46231147 Ki = 4530 nM T20251 CRTO63 46231148 Ki = 177 nM T20251 CZ6C0S 46231149 Ki = 3810 nM T20251 C8RP5H 46232900 IC50 > 90000 nM T20251 C7OB2G 46235733 IC50 = 6400 nM T20251 CZK5E9 46238536 IC50 = 7500 nM T20251 CY2A9C 46240380 IC50 = 22500 nM T20251 CIG71O 46240381 IC50 > 50000 nM T20251 CFY3L5 46240481 IC50 = 43800 nM T20251 CPHB87 46240482 IC50 = 32000 nM T20251 C8R1QX 46240484 IC50 = 28000 nM T20251 CR0NX3 46240582 IC50 = 15000 nM T20251 CF9O5C 46240584 IC50 = 6200 nM T20251 CV2X5E 46240585 IC50 > 50000 nM T20251 CD1M3J 46240687 IC50 = 6000 nM T20251 C63QWF 46240785 IC50 > 50000 nM T20251 C3YU2T 46240895 IC50 = 24000 nM T20251 CEH6U9 46241010 IC50 = 28000 nM T20251 C43MLP 46241011 IC50 > 50000 nM T20251 CJ7L3Z 46241120 IC50 = 27000 nM T20251 C7PVU1 46241121 IC50 > 50000 nM T20251 CDZ3V6 46241509 IC50 = 37000 nM T20251 CH8F5U 46241608 IC50 = 11200 nM T20251 CD1H3B 46241609 IC50 = 25000 nM T20251 CXJ7C5 46241610 IC50 = 5500 nM T20251 C35CXM 46241611 IC50 = 17500 nM T20251 C5Y8ZT 46241717 IC50 = 14500 nM T20251 C8EX9T 46241718 IC50 = 9800 nM T20251 CZK4H8 46241719 IC50 = 10000 nM T20251 CK9H6B 46241720 IC50 = 12500 nM T20251 CA05ZH 46241826 IC50 = 35000 nM T20251 C3LD6V 46241827 IC50 = 21600 nM T20251 CRJD47 46241829 IC50 = 35000 nM T20251 CL7C2K 46244173 IC50 > 100000 nM T20251 C2NH0A 46244259 IC50 > 33000 nM T20251 CVJM38 46244260 IC50 > 33000 nM T20251 C31PAF 46700737 IC50 = 17000 nM T20251 CJ2D3O 46701015 IC50 = 5280 nM T20251 CM04ZI 46701016 IC50 = 5640 nM T20251 C0JWP5 46701017 IC50 = 5430 nM T20251 C5H0MJ 46701086 IC50 = 6480 nM T20251 C9HWI7 46701087 IC50 = 3640 nM T20251 CVE5O1 46701088 IC50 = 2320 nM T20251 C1VPM0 46701089 IC50 = 4140 nM T20251 CQ8B6R 46701090 IC50 = 4330 nM T20251 C6C0FS 46701091 IC50 = 4730 nM T20251 C2ILJ9 46701790 Ki = 1258.93 nM T20251 C2SOY1 46785920 IC50 > 30000 nM T20251 CCJ08W 46830055 IC50 = 39900 nM T20251 CC68WI 46830289 IC50 = 2000 nM T20251 CC3UF9 46830325 IC50 = 5100 nM T20251 C5TC2S 46830335 IC50 > 10000 nM T20251 C1K7FL 46830336 IC50 > 10000 nM T20251 C2ZGO0 46830791 IC50 = 8000 nM T20251 CL7XJ8 46831392 IC50 = 13000 nM T20251 CEV89K 46831395 IC50 = 20000 nM T20251 CICY27 46833073 IC50 = 4100 nM T20251 C6G1DY 46833075 IC50 = 900 nM T20251 C7MU0O 46835136 IC50 = 500 nM T20251 C9CR0E 46835922 IC50 = 18000 nM T20251 CGS4F2 46836713 IC50 = 30000 nM T20251 C0GY1V 46837247 IC50 > 40000 nM T20251 CQ41PO 46837248 IC50 > 40000 nM T20251 CN1EK8 46837249 IC50 > 40000 nM T20251 C6IXU7 46837365 IC50 = 10000 nM T20251 C0M8AW 46839029 IC50 = 2000 nM T20251 C1ZDW9 46839030 IC50 = 3000 nM T20251 C21ILB 46839164 IC50 = 1200 nM T20251 C1OIG5 46839165 IC50 = 10000 nM T20251 C9S4IH 46839298 IC50 = 6900 nM T20251 C1EPB3 46839300 IC50 = 20000 nM T20251 C1N4KX 46842383 IC50 > 10000 nM T20251 CIM53K 46847263 IC50 = 13800 nM T20251 CO7G8Z 46851863 IC50 = 4040 nM T20251 C4S6YJ 46853439 IC50 = 170 nM T20251 CO31WX 46861576 IC50 = 8500 nM T20251 CC5IO9 46861756 IC50 > 10000 nM T20251 C19ZCY 46861765 IC50 = 4970 nM T20251 CP6DN0 46861858 Ki = 5291 nM T20251 C5VOF1 46861859 Ki = 1373 nM T20251 CW1FS9 46861860 Ki > 10000 nM T20251 C2QH7O 46865650 Ki > 3000 nM T20251 CC2O9R 46865656 IC50 = 19952.62 nM T20251 CQN2H4 46865774 IC50 > 80000 nM T20251 CPV2L4 46865775 IC50 = 30000 nM T20251 CC5KR7 46865978 Ki > 3000 nM T20251 CC7DG3 46866398 IC50 = 1100 nM T20251 CO3P0J 46866604 IC50 > 30000 nM T20251 CS9LD5 46867516 IC50 > 30000 nM T20251 C1XGZ8 46867925 IC50 > 30000 nM T20251 CZQ57K 46868086 IC50 = 2300 nM T20251 C9NGO7 46869046 IC50 = 18000 nM T20251 C8BT1F 46869326 IC50 = 12000 nM T20251 C97JEP 46871671 IC50 = 120 nM T20251 C8JZ2A 46871848 IC50 > 30000 nM T20251 CLS29B 46872626 IC50 = 77000 nM T20251 CFZ75O 46880148 IC50 > 30000 nM T20251 C0PXY7 46880628 IC50 > 10000 nM T20251 C2MC4K 46881463 IC50 = 7943.28 nM T20251 CSQ4C9 46881468 IC50 = 15848.93 nM T20251 C4BH9E 46882458 IC50 = 2511.89 nM T20251 CAH31I 46882578 IC50 = 180 nM T20251 CMS27C 46882857 IC50 > 40000 nM T20251 CM45ZP 46882858 IC50 = 7920 nM T20251 C3IGF1 46882859 IC50 = 19800 nM T20251 CHLZ97 46882860 IC50 > 10000 nM T20251 C4B8EX 46882909 IC50 = 4120 nM T20251 CFY95C 46882910 IC50 = 52400 nM T20251 C0SQX2 46882912 IC50 > 10000 nM T20251 CJ82WI 46882913 IC50 > 10000 nM T20251 CM5Z4G 46882938 IC50 = 12900 nM T20251 C60YMF 46883462 IC50 > 20000 nM T20251 C7J6GU 46883497 IC50 > 18600 nM T20251 C3F5AS 46883498 IC50 = 7140 nM T20251 CRSE34 46883499 IC50 = 16800 nM T20251 C0CX3O 46883500 IC50 = 7740 nM T20251 C15KEH 46883819 IC50 = 12700 nM T20251 C3J5IG 46883820 IC50 = 7880 nM T20251 CGKP83 46883876 IC50 = 3810 nM T20251 CJ39QM 46883878 IC50 = 384 nM T20251 CXIM81 46883917 IC50 = 12000 nM T20251 C3OBL5 46883918 IC50 = 2310 nM T20251 CR6FO1 46883919 IC50 = 13800 nM T20251 CW6A9I 46884062 Ki > 5000 nM T20251 C04JMO 46884063 Ki = 0.73 nM T20251 CR1Z8E 46884119 Ki > 5000 nM T20251 CR0CQ9 46884120 IC50 = 3000 nM T20251 C9OYT5 46884152 IC50 = 330 nM T20251 CCI32B 46884153 Ki > 5000 nM T20251 C2JQE7 46884154 Ki > 5000 nM T20251 C20HET 46884155 Ki > 5000 nM T20251 C0HYN3 46884200 IC50 = 1500 nM T20251 CM6A8S 46884201 IC50 = 1700 nM T20251 CW94IK 46884202 Ki > 5000 nM T20251 C3QT0U 46884239 Ki > 5000 nM T20251 CYC64I 46884402 IC50 = 61 nM T20251 CF7HD6 46884426 IC50 = 178 nM T20251 C9M4RX 46884427 IC50 = 188 nM T20251 CT9K2R 46884428 IC50 = 202 nM T20251 CWK75U 46884462 IC50 = 6650 nM T20251 C82IYB 46884463 IC50 = 9190 nM T20251 COPQ16 46884600 Ki > 3000 nM T20251 C85MOA 46884637 Ki > 3000 nM T20251 C36NKV 46884638 Ki > 3000 nM T20251 CQ84IF 46884639 Ki > 3000 nM T20251 CZGS15 46884640 Ki > 3000 nM T20251 CZ72SW 46884641 Ki > 3000 nM T20251 CA3Z6G 46884666 Ki > 3000 nM T20251 C8DBY0 46884667 IC50 = 1900 nM T20251 CU3BG6 46884668 IC50 = 520 nM T20251 CPG14Q 46884669 IC50 = 2100 nM T20251 C7R9AK 46884670 IC50 = 110 nM T20251 C64KNW 46884698 IC50 = 230 nM T20251 C0ASK4 46884699 IC50 = 360 nM T20251 CYNU85 46884731 Ki > 3000 nM T20251 CJ6O8D 46884732 Ki > 3000 nM T20251 C9QT7G 46884733 Ki > 3000 nM T20251 CL6Z7Q 46884734 IC50 = 1800 nM T20251 C6PRX8 46884735 Ki = 1200 nM T20251 CWK8I4 46884736 IC50 = 620 nM T20251 CB8GE1 46884818 IC50 > 10000 nM T20251 C4MQ0A 46884856 IC50 = 10000 nM T20251 CCNT25 46884898 IC50 > 10000 nM T20251 C3MSG2 46885027 IC50 > 10000 nM T20251 CB7XI0 46885213 IC50 > 10000 nM T20251 CD3E4C 46885323 Ki = 6.65 nM T20251 CNW43Y 46885367 Ki > 9.17 nM T20251 CV23JL 46885415 Ki = 5.87 nM T20251 CHPS01 46885417 Ki > 5.27 nM T20251 C4SVE1 46885480 Ki = 4.65 nM T20251 C5QI7J 46885481 Ki = 5.07 nM T20251 COU5X2 46885482 Ki > 10 nM T20251 C1TXI0 46885514 IC50 > 60000 nM T20251 CS90MN 46885524 Ki > 10 nM T20251 CQ94VM 46885526 Ki > 10 nM T20251 C90ABZ 46885558 Ki > 10 nM T20251 CKF74T 46885587 IC50 > 60000 nM T20251 CKH5W7 46885611 IC50 = 2300 nM T20251 C0Y9NF 46885711 Ki > 10 nM T20251 C3O5BR 46885712 Ki = 7.91 nM T20251 CK8D6G 46885760 Ki = 5 nM T20251 CY30PG 46885815 Ki = 5.84 nM T20251 CFC5L1 46885972 Ki > 7.88 nM T20251 CF8N0U 46886536 IC50 = 3000 nM T20251 CZ59HO 46886537 IC50 > 80000 nM T20251 C28IHA 46886538 IC50 = 4000 nM T20251 C0UDN9 46886539 IC50 = 22000 nM T20251 CO2PM3 46887855 IC50 = 1320 nM T20251 C8EOA7 46887961 IC50 = 3000 nM T20251 C0XR8B 46887962 IC50 = 7800 nM T20251 CE4X6C 46887963 IC50 = 2000 nM T20251 CVB6C0 46887993 IC50 = 7200 nM T20251 C0U3CX 46887994 IC50 > 10000 nM T20251 CG8I9K 46887995 IC50 = 2900 nM T20251 CVY2T4 46888365 IC50 = 2000 nM T20251 CO7M5J 46888366 IC50 = 4600 nM T20251 CLS1G3 46888367 IC50 = 630 nM T20251 CGD6T5 46888386 IC50 > 30000 nM T20251 C13SVO 46888387 IC50 = 540 nM T20251 C9G2HI 46888388 IC50 = 2660 nM T20251 C5D2CK 46888389 IC50 > 30000 nM T20251 CAE10V 46888443 IC50 > 10000 nM T20251 C9QO6J 46888468 IC50 > 10000 nM T20251 C6DB3K 46888487 IC50 > 10000 nM T20251 CM76UZ 46888550 IC50 > 10000 nM T20251 CQ5B2F 46888578 IC50 = 2800 nM T20251 CDUM26 46888645 IC50 = 300 nM T20251 CTN16E 46888688 IC50 = 600 nM T20251 C4SX5W 46888719 IC50 = 80 nM T20251 CT8E9F 46888720 IC50 > 30000 nM T20251 CP75RD 46888721 IC50 > 30000 nM T20251 C9Z2CO 46888748 IC50 = 1200 nM T20251 CR7HN9 46888749 IC50 = 5300 nM T20251 C06HUF 46888750 IC50 = 8700 nM T20251 CEMZ98 46888775 IC50 > 30000 nM T20251 CYT7P0 46888776 IC50 = 380 nM T20251 CJDH10 46888777 IC50 = 1100 nM T20251 CM6S8Z 46888778 IC50 = 1600 nM T20251 CZBL19 46888785 Ki > 5000 nM T20251 CK3B2R 46888786 Ki = 1262 nM T20251 C46QKX 46888787 Ki > 10000 nM T20251 CJS87P 46888788 Ki > 10000 nM T20251 C98ROS 46888789 Ki = 638 nM T20251 C9RXL8 46888825 Ki = 926 nM T20251 CHN7W1 46888826 Ki = 2649 nM T20251 C46PXH 46888827 Ki = 1840 nM T20251 CR42EN 46888828 Ki > 10000 nM T20251 C3B2QN 46888853 Ki > 10000 nM T20251 C94FRI 46888854 Ki > 3000 nM T20251 C30FVT 46888855 Ki = 1183 nM T20251 C4Q2MA 46888856 Ki > 3000 nM T20251 CJK1Z5 46888857 IC50 = 720 nM T20251 C4U3CN 46888882 Ki = 6515 nM T20251 C61GZW 46888883 Ki > 10000 nM T20251 C6KOP3 46888884 Ki > 10000 nM T20251 C4AFL7 46888885 Ki = 10336 nM T20251 CC8G6T 46888886 Ki > 10000 nM T20251 C3V4ZN 46888887 IC50 = 2100 nM T20251 CX92WH 46889257 IC50 = 492 nM T20251 C01DMO 46889258 IC50 = 233 nM T20251 C2CI9O 46889753 IC50 = 7500 nM T20251 C3J5IQ 46889754 IC50 = 35000 nM T20251 CX18GT 46889932 IC50 = 3000 nM T20251 CM12LB 46889933 IC50 = 2300 nM T20251 CL51ME 46890090 Ki = 440 nM T20251 C2XCK5 46890181 Ki = 1200 nM T20251 CTS04G 46890283 Ki = 4500 nM T20251 CV8C4E 46890347 Ki = 5600 nM T20251 CH56AN 46890391 IC50 = 6370 nM T20251 CPDX34 46890392 IC50 = 6400 nM T20251 C0YGP2 46890393 IC50 = 2960 nM T20251 C61INJ 46890394 IC50 = 21400 nM T20251 C4XLV0 46890430 Ki = 5600 nM T20251 CI14SE 46890441 IC50 = 20800 nM T20251 CP4GD3 46890442 IC50 = 8550 nM T20251 CQI2Y8 46890443 IC50 = 10400 nM T20251 CZ2MG7 46890444 IC50 = 40100 nM T20251 CP6A8K 46890445 IC50 > 22500 nM T20251 CD5J8B 46890446 IC50 = 16000 nM T20251 C4IK6F 46890475 Ki = 2100 nM T20251 CK08VN 46890476 Ki = 6200 nM T20251 CYK9D2 46890489 IC50 = 6500 nM T20251 CCR04L 46890490 IC50 = 8240 nM T20251 CT4O9M 46890491 IC50 = 9120 nM T20251 CGPM19 46890493 IC50 = 6110 nM T20251 CM56CG 46890523 Ki = 6900 nM T20251 C2K4HZ 46890562 Ki = 780 nM T20251 C89ZNE 46890564 Ki = 54000 nM T20251 CT4Q8R 46890603 Ki = 1700 nM T20251 C6XPD3 46890638 Ki = 4400 nM T20251 CQLS54 46890639 Ki = 4200 nM T20251 CP7ZS3 46890640 Ki = 1500 nM T20251 CU3O0K 46890688 Ki = 10000 nM T20251 CZ0A7U 46890769 Ki = 5.3 nM T20251 C1AK8C 46890770 Ki = 1.2 nM T20251 CB6T3M 46890771 Ki > 65 nM T20251 CP8FW2 46890772 Ki = 14 nM T20251 CX7I3Y 46890773 Ki = 1.9 nM T20251 C3MPJ7 46890808 Ki > 9000 nM T20251 C2I9CM 46890824 Ki > 51 nM T20251 C6RB1V 46890825 Ki = 9 nM T20251 C5JT1D 46890826 Ki = 22 nM T20251 CC0E7P 46890827 Ki = 1.3 nM T20251 CT6UY7 46890828 Ki = 0.56 nM T20251 C9QFU5 46890891 Ki > 35 nM T20251 CS74RA 46890892 Ki = 4.3 nM T20251 CNQ26O 46890893 Ki = 1.85 nM T20251 CZQ25U 46890894 Ki = 13 nM T20251 CJ8YV7 46890895 Ki = 10 nM T20251 CWDG43 46890952 Ki = 2.7 nM T20251 CIC32L 46890953 Ki = 0.55 nM T20251 C4ZYM8 46890954 Ki = 46 nM T20251 C0P4GM 46890955 Ki = 11 nM T20251 CK94BQ 46890956 Ki = 2 nM T20251 CEW98A 46891012 Ki = 32 nM T20251 C3CPE9 46891013 Ki = 2.9 nM T20251 C51IBN 46891527 Ki = 8.8 nM T20251 CQ34CV 46891528 Ki = 1.8 nM T20251 CH91DV 46891529 Ki > 55 nM T20251 C7LS0J 46891530 Ki = 21 nM T20251 CCE34G 46891585 Ki = 2.2 nM T20251 CMJ93X 46891586 Ki > 57 nM T20251 CHGA57 46891587 Ki = 12 nM T20251 C2FOK8 46891588 Ki = 12 nM T20251 C4ZXM7 46891589 Ki = 26 nM T20251 CZ7C1J 46893145 Ki = 2900 nM T20251 CS8XC4 46893453 IC50 = 29512.09 nM T20251 C5F1CH 46893542 IC50 > 100000 nM T20251 C90NYX 46896338 IC50 = 10000 nM T20251 CC9FZ0 46898063 IC50 = 10500 nM T20251 C1JSH9 46899637 Ki = 199.53 nM T20251 C3MSL0 46899638 Ki = 501.19 nM T20251 CV3LP2 46899639 Ki = 1258.93 nM T20251 CGHZ15 46899640 Ki = 1000 nM T20251 CN9FC3 46900150 Ki = 1584.89 nM T20251 C40ZJO 46900451 Ki = 398.11 nM T20251 CNC02A 46900453 Ki = 398.11 nM T20251 CTCH14 46900455 Ki = 25.12 nM T20251 CP41AQ 46900457 Ki = 1000 nM T20251 CR3L4I 46900459 Ki = 12589.25 nM T20251 CK17PA 46900606 Ki = 2511.89 nM T20251 CQ2K1C 46900608 Ki = 501.19 nM T20251 C5ZT1B 46900610 Ki = 7943.28 nM T20251 C1NAX4 46900612 Ki = 6309.57 nM T20251 CT0SQ2 46900614 Ki = 2511.89 nM T20251 CXD9S3 46900776 Ki = 3981.07 nM T20251 C8I7SJ 46900778 Ki = 1000 nM T20251 C7QDM9 46900782 Ki = 2511.89 nM T20251 C15FMY 46900954 Ki = 630.96 nM T20251 C8W1FU 46900956 Ki = 501.19 nM T20251 CH35BV 46900958 Ki = 199.53 nM T20251 C7T2GX 46909057 IC50 = 37000 nM T20251 CZ46AH 46911015 IC50 = 1690 nM T20251 C3JCB1 46911060 IC50 > 100000 nM T20251 CA2JU7 46911115 IC50 = 4000 nM T20251 C73VYX 46911116 IC50 = 6000 nM T20251 C1MEW3 46911124 IC50 > 300000 nM T20251 C4DTN2 46911175 IC50 = 5900 nM T20251 C5XAF7 46912235 IC50 = 9000 nM T20251 CE7KZ8 46914881 IC50 = 170 nM T20251 CI0Y4F 46914882 IC50 > 30000 nM T20251 C8HWO7 46914883 IC50 > 30000 nM T20251 C6FN4G 46914884 IC50 > 30000 nM T20251 CY3O2C 46915043 IC50 = 29 nM T20251 CR5OZ8 46916382 IC50 = 2000 nM T20251 C0HZ4C 46916514 IC50 > 10000 nM T20251 CDBM59 46916519 IC50 > 10000 nM T20251 CW6Y2D 46916520 IC50 > 10000 nM T20251 CK9E8N 46927116 IC50 = 10000 nM T20251 C82HXR 46927117 IC50 = 2800 nM T20251 C8GAI9 46927903 IC50 = 1995.26 nM T20251 C3D7FL 46931619 Ki = 1100 nM T20251 CW3L9K 46931735 IC50 = 4200 nM T20251 CKO76R 46931815 IC50 = 1000 nM T20251 C3M4LT 46931848 IC50 = 9800 nM T20251 C9EG4R 46931852 IC50 = 2800 nM T20251 CB84WK 46931947 IC50 = 10300 nM T20251 CJMS30 46931948 IC50 = 3200 nM T20251 C2M1KO 46932044 Ki = 1700 nM T20251 C3QLC4 46932045 Ki = 2800 nM T20251 CC91MK 46932046 Ki = 3400 nM T20251 CQ91FA 46932047 Ki = 3900 nM T20251 CYCF24 46932049 Ki = 6200 nM T20251 C3O4MA 46932136 Ki = 6000 nM T20251 CF9YV2 46932138 Ki = 4200 nM T20251 COL7J6 46932139 Ki = 10500 nM T20251 CSMK50 46932141 Ki = 3300 nM T20251 C29RXO 46932234 Ki = 21200 nM T20251 CC0F4D 46932235 Ki = 13700 nM T20251 C8QB4Z 46932237 Ki = 9800 nM T20251 CG2J9V 46932512 Ki = 15300 nM T20251 C2VZ7Q 46932514 Ki = 19500 nM T20251 C4PW3A 46932704 Ki > 60000 nM T20251 C82QKP 46932796 IC50 = 4800 nM T20251 COY21M 46935743 IC50 = 69000 nM T20251 CU90MG 46938037 IC50 > 1000000000 nM T20251 CX2U5I 46938097 IC50 > 1000000000 nM T20251 C47QBL 46938101 IC50 > 1000000000 nM T20251 CV28ZU 46944853 IC50 = 6200 nM T20251 CT9P5G 46944854 IC50 = 8200 nM T20251 CWH4K6 46944855 IC50 = 23000 nM T20251 CC3O0S 46945254 IC50 = 44000 nM T20251 C1UB8E 46945255 IC50 = 37000 nM T20251 C4RZG5 46945857 IC50 = 12000 nM T20251 CAK5J0 46946058 IC50 = 9800 nM T20251 CY09UB 46946452 IC50 = 2400 nM T20251 C6J4TV 46946859 Ki = 1850 nM T20251 CFH87K 46947816 IC50 = 10000 nM T20251 CVEF51 49763568 IC50 = 2800 nM T20251 C43LAE 49763569 IC50 = 2800 nM T20251 CI6AR9 49763571 IC50 = 4000 nM T20251 C78ICP 49763574 IC50 = 3300 nM T20251 C65RMG 49763575 IC50 = 6200 nM T20251 CQLN97 49763682 IC50 = 3000 nM T20251 CY5ME3 49763685 IC50 = 1300 nM T20251 C0ADU9 49763686 IC50 = 23000 nM T20251 C1GVM0 49763804 IC50 = 7900 nM T20251 C94ARN 49763931 IC50 = 2500 nM T20251 C68SFM 49764196 IC50 = 13500 nM T20251 CSW83Q 49764322 IC50 = 8900 nM T20251 C1Z0UD 49764446 IC50 = 25000 nM T20251 C5AD0E 49764447 IC50 = 4100 nM T20251 C20WNR 49764700 IC50 = 2800 nM T20251 CIZ86P 49764701 IC50 = 1500 nM T20251 CABL63 49765080 IC50 = 2 nM T20251 CIXN24 49767138 IC50 = 1600 nM T20251 CR13SJ 49767146 IC50 = 4300 nM T20251 CZWN54 49767224 IC50 = 6900 nM T20251 CDM18G 49768863 IC50 = 4230 nM T20251 CWU2R3 49773361 IC50 = 12400 nM T20251 CYWX19 49780808 IC50 = 7943.28 nM T20251 C9RI3L 49780809 IC50 = 251.19 nM T20251 C39KWP 49781039 IC50 = 2511.89 nM T20251 C9O2RB 49781040 IC50 = 630.96 nM T20251 C7T3KS 49781255 IC50 = 316.23 nM T20251 CYL65E 49781476 IC50 = 158.49 nM T20251 CFQN89 49781477 IC50 = 501.19 nM T20251 CL82ES 49781478 IC50 = 501.19 nM T20251 CAFW31 49783666 IC50 = 26000 nM T20251 CNI1P6 49783903 IC50 > 33000 nM T20251 CGF65B 49783985 IC50 > 33000 nM T20251 CZ7A9E 49796933 IC50 = 9700 nM T20251 C5RF0Y 49796938 IC50 > 90000 nM T20251 CE0C3Y 49796939 IC50 = 79000 nM T20251 CI25XP 49796945 IC50 = 870 nM T20251 C8WYA5 49796953 IC50 = 76000 nM T20251 CQH86V 49796955 IC50 > 100000 nM T20251 CBMV50 49796972 Ki = 1100 nM T20251 CX74RG 49796999 IC50 = 4600 nM T20251 C7B5DY 49797060 IC50 = 59000 nM T20251 CA2U4Y 49797089 IC50 > 100000 nM T20251 CBS36X 49797110 IC50 > 100000 nM T20251 C0STP5 49797111 IC50 > 100000 nM T20251 C2OI0Y 49797114 IC50 = 8300 nM T20251 CW20FJ 49797115 IC50 > 100000 nM T20251 CY1OJ5 49797177 Ki > 50000 nM T20251 C25ZSD 49797191 IC50 = 36700 nM T20251 C6ZGL5 49797198 IC50 > 100000 nM T20251 CON0A6 49797232 IC50 = 26100 nM T20251 CA4E8M 49797242 IC50 = 9900 nM T20251 C37MDP 49797244 IC50 = 8100 nM T20251 CUMH43 49797248 IC50 = 33200 nM T20251 C93VJO 49797347 IC50 > 90000 nM T20251 C1Z8HB 49797353 IC50 = 49000 nM T20251 CTYO37 49797358 IC50 > 90000 nM T20251 C1K4FR 49797359 IC50 = 78000 nM T20251 CA3Q2W 49797361 IC50 > 90000 nM T20251 CNMF62 49797362 IC50 = 39000 nM T20251 C76KMB 49797451 IC50 = 37000 nM T20251 CU72EZ 49797596 IC50 = 17000 nM T20251 C6DJX7 49797605 IC50 = 38000 nM T20251 CK3ZI1 49797607 IC50 = 2500 nM T20251 CV6I0O 49797630 IC50 = 7500 nM T20251 CQVG17 49798349 IC50 = 7943.28 nM T20251 C62VRQ 49798437 IC50 > 63095.73 nM T20251 CY90CD 49798461 IC50 > 31622.78 nM T20251 C5I1HQ 49798777 IC50 = 20000 nM T20251 C02EUQ 49800098 IC50 = 8130 nM T20251 CM75QU 49801042 IC50 = 2400 nM T20251 C8LFB9 49801043 IC50 = 9000 nM T20251 C8IYR7 49801044 IC50 = 3500 nM T20251 C8A0LD 49801837 IC50 = 28000 nM T20251 CP91TS 49802222 IC50 = 16000 nM T20251 CIFZ02 49803320 IC50 = 28000 nM T20251 CEP3B7 49803607 IC50 > 30000 nM T20251 C1BLY0 49804185 IC50 = 40000 nM T20251 C97LZE 49804478 IC50 = 5200 nM T20251 C2IGB7 49804777 IC50 = 2200 nM T20251 C73PSQ 49805872 IC50 > 3000 nM T20251 CML8Z5 49805873 IC50 > 10000 nM T20251 C41TPM 49806128 IC50 > 3000 nM T20251 C4O0QK 49821278 Ki = 13000 nM T20251 CDAB96 49836026 IC50 = 1995.26 nM T20251 CI8FT3 49836033 IC50 > 33000 nM T20251 CO20JE 49836187 IC50 > 63095.73 nM T20251 CT7CV0 49836295 IC50 > 39810.72 nM T20251 CYJW87 49836299 IC50 > 63095.73 nM T20251 C8E6WA 49836410 IC50 > 39810.72 nM T20251 CNM9X8 49836528 IC50 > 39810.72 nM T20251 COK75S 49836633 IC50 > 50118.72 nM T20251 CB71TA 49837867 IC50 = 700 nM T20251 CZQC64 49837869 IC50 > 20000 nM T20251 CVNA15 49837870 IC50 > 20000 nM T20251 C9L3XR 49838879 IC50 > 160000 nM T20251 CL64TH 49842175 IC50 > 10000 nM T20251 C3T6NH 49843555 Ki = 3700 nM T20251 CU63QR 49847377 IC50 = 22000 nM T20251 CZT4I8 49847378 IC50 = 22000 nM T20251 CA72PE 49847379 IC50 = 46000 nM T20251 C4V7EW 49848258 IC50 = 19000 nM T20251 C4BXP1 49848557 IC50 > 50118.72 nM T20251 CP8TS6 49848895 IC50 = 6400 nM T20251 C9COF5 49848896 IC50 = 23000 nM T20251 CK0B1G 49848897 IC50 = 13000 nM T20251 CP61VJ 49849002 IC50 = 31000 nM T20251 CBM62Z 49849007 IC50 = 54000 nM T20251 C05SEW 49849008 IC50 = 7200 nM T20251 CF64IJ 49849120 IC50 = 38000 nM T20251 CC9EB4 49849122 IC50 = 21000 nM T20251 C2ORV5 49849123 IC50 = 2000 nM T20251 CTR7Q0 49850345 IC50 > 50118.72 nM T20251 CSGQ38 49850568 Ki = 316.23 nM T20251 C07JTU 49850570 Ki = 630.96 nM T20251 CR4EZ0 49850870 Ki = 501.19 nM T20251 C5K4EC 49850872 Ki = 3981.07 nM T20251 C8AW0R 49850874 Ki = 50.12 nM T20251 CL59YO 49852191 IC50 > 30000 nM T20251 C7ZUF5 49852192 IC50 > 30000 nM T20251 C6KX1V 49852195 IC50 > 30000 nM T20251 CN2V8R 49854681 IC50 = 5700 nM T20251 C65YMH 49855492 IC50 > 33000 nM T20251 C12FKR 49855495 IC50 = 19000 nM T20251 CP3M8H 49855496 IC50 > 33000 nM T20251 CKT38C 49855683 IC50 > 33000 nM T20251 C8KA3J 49855886 IC50 > 33000 nM T20251 C9TO2S 49856484 IC50 = 4800 nM T20251 C6UO5Y 49857245 IC50 = 1500 nM T20251 C0UOW3 49857439 IC50 = 11100 nM T20251 CQ3LC1 49857440 IC50 = 2300 nM T20251 CW9NX3 49858377 IC50 > 33000 nM T20251 C1EMQ2 49861348 Ki > 10 nM T20251 CR53VH 49862169 Ki = 2160 nM T20251 CT3WH4 49862215 Ki = 1580 nM T20251 CC97JM 49862219 Ki = 1780 nM T20251 C6IW4Q 49862238 Ki > 1000 nM T20251 CB13XF 49863795 IC50 = 700 nM T20251 C18ICN 49863958 IC50 = 11800 nM T20251 CMRQ30 49863961 IC50 = 6900 nM T20251 CLOY62 49864459 IC50 > 10000 nM T20251 CR8JK9 49864483 IC50 > 10000 nM T20251 C0Y5ZU 49865137 IC50 > 10000 nM T20251 CG98LM 49865191 IC50 > 10000 nM T20251 CKWA93 49865589 IC50 > 63095.73 nM T20251 CXWL20 49865623 IC50 = 1584.89 nM T20251 CXW97O 49865703 IC50 > 33000 nM T20251 CRG60N 49865732 IC50 > 33000 nM T20251 CZY2T3 49865733 IC50 = 0.61 nM T20251 CI2W0D 49865783 IC50 = 250 nM T20251 CUK35O 49865784 IC50 = 1100 nM T20251 CLD4P0 49865785 IC50 = 20000 nM T20251 CFZ39O 49865822 IC50 = 3100 nM T20251 CL0DR3 49865859 IC50 = 1100 nM T20251 CE15WQ 49865860 IC50 = 1000 nM T20251 C4EM1X 49865861 IC50 = 1600 nM T20251 CEF3O1 49865862 IC50 = 1500 nM T20251 C5YP2L 49865863 IC50 = 1000 nM T20251 CK7O1S 49865875 IC50 > 10000 nM T20251 C8V3NG 49865877 IC50 > 10000 nM T20251 CEK89Q 49865878 IC50 > 10000 nM T20251 CZA5X4 49865879 IC50 > 10000 nM T20251 CD4LO5 49865880 IC50 > 10000 nM T20251 CNGL32 49865918 IC50 = 15000 nM T20251 C9HEP1 49865919 IC50 = 680 nM T20251 CL6ZG8 49865920 IC50 = 660 nM T20251 CHYN61 49865922 IC50 = 1100 nM T20251 C3YJ4G 49865936 IC50 > 10000 nM T20251 CB5WR8 49865937 IC50 = 5900 nM T20251 C5NJ6K 49865969 IC50 = 340 nM T20251 C3CJ4R 49865970 IC50 = 680 nM T20251 CP8VQ6 49865971 IC50 = 1000 nM T20251 CAI09G 49865972 IC50 = 1400 nM T20251 C5TMG9 49865973 IC50 = 1300 nM T20251 CFT26X 49866025 IC50 = 1600 nM T20251 CN9PI1 49867423 Ki = 120 nM T20251 CMV6Y2 49868651 IC50 = 4100 nM T20251 C8AJ5K 49869035 IC50 = 16700 nM T20251 C1WM9N 49869037 IC50 > 33000 nM T20251 CAPI06 49869040 IC50 = 28800 nM T20251 CG5IV6 49869041 IC50 = 21000 nM T20251 C1WYF9 49869172 IC50 > 33000 nM T20251 CR0D3P 49869174 IC50 > 33000 nM T20251 C19EDA 49869312 IC50 = 12400 nM T20251 CD62TH 49869313 IC50 = 14400 nM T20251 CMB32F 49869877 IC50 = 24500 nM T20251 C07DIE 49870853 IC50 > 63000 nM T20251 C7GR0H 49872381 IC50 = 7900 nM T20251 CD1X3U 49872384 IC50 > 10000 nM T20251 C60RMP 49872483 IC50 > 10000 nM T20251 CD5J7W 50898619 IC50 = 4100 nM T20251 CX5V7B 50898694 IC50 = 15400 nM T20251 C90UKY 50899643 IC50 = 16000 nM T20251 CYGD56 50899654 IC50 > 10000 nM T20251 CBLK68 50899745 IC50 = 5400 nM T20251 CU7TK4 50899749 IC50 > 10000 nM T20251 C1R5UC 50905013 Ki = 27000 nM T20251 C67IRJ 50908804 Ki = 2511.89 nM T20251 CLOB24 50908805 Ki = 1995.26 nM T20251 CL01TJ 50913783 IC50 = 3800 nM T20251 C1YF6I 50915132 IC50 > 30000 nM T20251 CD0G9L 50915507 IC50 = 10000 nM T20251 C4IOV5 50916528 IC50 > 30000 nM T20251 C7JB8Z 50925394 IC50 < 1000 nM T20251 CP2N7E 50925496 Ki = 14000 nM T20251 CX3NI6 50925497 Ki = 16000 nM T20251 C64HTN 50925513 IC50 = 3500 nM T20251 C2GTE4 50938548 IC50 = 1600 nM T20251 C90ANW 50939489 IC50 = 6900 nM T20251 CJ43IF 50941460 IC50 = 7800 nM T20251 C2HJL6 50942025 IC50 = 2230 nM T20251 CP7B9V 50942696 IC50 = 3900 nM T20251 COJ32C 50942806 IC50 >= 10000 nM T20251 CWK9X2 50942874 IC50 >= 10000 nM T20251 CX8N4D 50990920 IC50 = 8000 nM T20251 CXF4V3 50990921 IC50 = 65000 nM T20251 C2T4IC 50991056 IC50 = 31300 nM T20251 CI32TR 50992246 IC50 = 1700 nM T20251 C4IFR9 50992499 IC50 = 2000 nM T20251 CFG8M7 50992643 IC50 = 10 nM T20251 C41QJN 50992719 IC50 = 1000 nM T20251 C4BP6M 50992720 IC50 = 5000 nM T20251 CIO9B5 50992721 IC50 = 6000 nM T20251 C2ST3V 50992722 IC50 = 5000 nM T20251 C2SHO8 50993865 IC50 = 1600 nM T20251 CLY9W1 50994950 IC50 = 8300 nM T20251 C2CH1R 50995330 IC50 > 30000 nM T20251 C0X9OY 50997095 IC50 = 49 nM T20251 CS9G6E 50997096 IC50 = 460 nM T20251 C4UPJ2 51030637 IC50 = 10000 nM T20251 CP6NI2 51030711 IC50 > 9800 nM T20251 CSE2G4 51030732 IC50 = 500 nM T20251 CM1F2R 51030830 IC50 = 1900 nM T20251 CWQ20B 51030833 IC50 = 2000 nM T20251 C15LDS 51030834 IC50 = 800 nM T20251 C1P9UY 51030897 IC50 = 5900 nM T20251 CW06HL 51030898 IC50 = 11600 nM T20251 C4QW2B 51030901 IC50 = 7600 nM T20251 C48USP 51030919 IC50 = 1900 nM T20251 C0QP3A 51030920 IC50 = 80000 nM T20251 C70OGS 51030984 IC50 = 12000 nM T20251 CX28ZP 51030985 IC50 = 10000 nM T20251 CXB2Q6 51031001 IC50 > 30000 nM T20251 CUY1S2 51033690 IC50 = 17000 nM T20251 CVE0J3 51033997 IC50 > 20000 nM T20251 CAU5Y8 51038251 IC50 = 1820 nM T20251 CBA1X5 51039205 IC50 = 32100 nM T20251 C96AQN 51346908 IC50 = 28900 nM T20251 C2W8LE 51346934 IC50 > 10000 nM T20251 CA3Y7Q 51347395 IC50 = 0.66 ug.mL-1 T20251 C3MWD8 51349244 IC50 = 2630 nM T20251 CO7U5C 51355838 IC50 = 15000 nM T20251 CIXL91 51355841 IC50 > 30000 nM T20251 C3XQE2 52337837 IC50 = 5 nM T20251 C8K6CQ 52916803 IC50 = 68000 nM T20251 CIRP71 52917998 IC50 = 2 nM T20251 CT0B1S 52917999 IC50 = 290 nM T20251 CFX76G 52918016 IC50 = 140 nM T20251 C47RHB 52918017 IC50 = 1260 nM T20251 CUQ53T 52918018 IC50 = 10000 nM T20251 CTP6U5 52918019 IC50 > 10000 nM T20251 CTJ28K 52918135 IC50 > 20000 nM T20251 CCP0V7 52920236 IC50 = 4000 nM T20251 CKDE49 52933949 IC50 = 21000 nM T20251 CL2Q9F 52934178 IC50 = 23000 nM T20251 CDI09M 52934690 IC50 = 5100 nM T20251 CUV9B4 52934924 IC50 = 12900 nM T20251 CEMS67 52938764 IC50 > 100000 nM T20251 CJ19FP 52940753 IC50 = 199.53 nM T20251 CCDZ51 52940788 IC50 = 1258.93 nM T20251 CH5S0P 52940936 Ki > 10000 nM T20251 C2RW5A 52940961 IC50 = 5011.87 nM T20251 CKP92N 52941058 Ki = 500 nM T20251 C8FZL4 52941427 IC50 = 794.33 nM T20251 COK7Q1 52941460 Ki > 20000 nM T20251 C1M3SD 52941462 IC50 = 0.38 nM T20251 CUV8I6 52941526 IC50 = 12100 nM T20251 C58ART 52941549 IC50 = 15 nM T20251 CVT1A7 52941563 Ki = 11000 nM T20251 C7N6RA 52941564 Ki > 20000 nM T20251 CP8BI3 52941601 IC50 = 1200 nM T20251 C1FX6A 52941684 IC50 > 63000 nM T20251 CE26GV 52941856 IC50 = 5900 nM T20251 C5JAY6 52941880 IC50 > 10000 nM T20251 CU7A2Y 52941972 IC50 = 1000 nM T20251 C51MIQ 52942095 Ki = 710 nM T20251 C0OU8I 52942126 IC50 = 740 nM T20251 C3E5WI 52942171 Ki = 2510 nM T20251 CL65FB 52942200 Ki = 560 nM T20251 C3WH6F 52942248 Ki = 1120 nM T20251 CYLC29 52942529 IC50 = 4.6 nM T20251 CX9AF4 52942551 Ki = 3162.28 nM T20251 CPOQ82 52942580 IC50 = 1.9 nM T20251 C3YF5D 52942581 IC50 = 7.3 nM T20251 CR0G5U 52942644 Ki > 31622.78 nM T20251 CKN2U6 52942810 IC50 = 3.7 nM T20251 CX2E5H 52942854 Ki = 969 nM T20251 C8N4AB 52943069 IC50 > 10000 nM T20251 C5V4DW 52943162 IC50 = 0.14 nM T20251 C2DOU4 52943195 IC50 = 400 nM T20251 CXD0O1 52943196 IC50 = 20000 nM T20251 CNI79L 52943227 Ki = 370 nM T20251 C0F3LG 52943305 IC50 = 3200 nM T20251 CJWI80 52943409 Ki > 10000 nM T20251 C71MDG 52943756 IC50 < 1000 nM T20251 CNK14O 52943803 IC50 = 0.62 nM T20251 CCF97B 52943811 Ki = 25118.86 nM T20251 C2FG9O 52943861 Ki = 31622.78 nM T20251 C9G4CI 52943891 Ki = 7943.28 nM T20251 CRH1Q5 52943993 IC50 = 4.8 nM T20251 CBW0A9 52944041 IC50 = 1.8 nM T20251 CE7K2D 52944154 IC50 = 260 nM T20251 C25NCO 52944522 Ki = 3980 nM T20251 C89GIK 52944552 IC50 = 3.5 nM T20251 CO85FM 52944637 Ki = 400 nM T20251 CCVP06 52944840 Ki = 5011.87 nM T20251 CP5A3T 52944907 IC50 = 13 nM T20251 C54ZBG 52944974 IC50 = 3 nM T20251 CQJ7C0 52945023 IC50 = 1000 nM T20251 CV48KS 52945118 IC50 = 0.72 nM T20251 C1G0IP 52945138 IC50 = 6 nM T20251 C34ZMB 52945520 IC50 > 30000 nM T20251 CSZ4R3 52945588 IC50 = 0.25 nM T20251 CNGU78 52945626 IC50 = 0.52 nM T20251 C1Z9HY 52945786 Ki > 10000 nM T20251 C5RAX8 52945794 IC50 > 100000 nM T20251 CF46DK 52945849 Ki = 320 nM T20251 CNQF49 52945978 IC50 = 63095.73 nM T20251 CJ49MX 52946290 Ki = 5011.87 nM T20251 CG8CN4 52946340 IC50 > 33 nM T20251 CK5VU2 52946383 IC50 > 63000 nM T20251 COZ9J3 52946432 IC50 = 2511.89 nM T20251 C4K6BH 52946883 Ki > 10000 nM T20251 C2GVW6 52947078 Ki > 10000 nM T20251 CK5ER0 52947414 Ki = 3981.07 nM T20251 CFD18K 52947437 IC50 > 33 nM T20251 CI5V3X 52947507 IC50 = 5011.87 nM T20251 CFN7I8 52947509 IC50 = 3.3 nM T20251 C6ZSQ8 52947516 IC50 = 1995.26 nM T20251 C41AYU 52947523 IC50 > 33 nM T20251 CEU2N1 52947551 IC50 = 12600 nM T20251 CY06OH 52947573 IC50 = 1.6 nM T20251 CY72CQ 52947593 IC50 = 4.9 nM T20251 CAVB03 52947615 Ki = 10000 nM T20251 CCIG41 52947616 IC50 = 1400 nM T20251 CGCK63 52947618 IC50 > 63000 nM T20251 C1HRK4 52947622 Ki = 6309.57 nM T20251 CN32PV 52947694 IC50 = 1584.89 nM T20251 CFI96N 52947735 IC50 = 0.62 nM T20251 CI63UL 52948240 IC50 = 1.5 nM T20251 CZ01DH 52948653 IC50 = 6309.57 nM T20251 C15KNW 52948655 IC50 = 13 nM T20251 C4ZC1K 52948697 Ki = 3981.07 nM T20251 C48RBH 52948719 IC50 = 0.43 nM T20251 CZX5B9 52948735 IC50 = 6.6 nM T20251 CDN06O 52948827 IC50 > 63000 nM T20251 CE0R3S 52948850 IC50 = 4.7 nM T20251 C25FAX 52948924 Ki = 3160 nM T20251 CPN4Z8 52948969 IC50 = 2.8 nM T20251 CN85WP 52949210 IC50 = 4800 nM T20251 CH02CI 52949290 IC50 = 800 nM T20251 C9OSI0 52949300 IC50 = 630.96 nM T20251 C9YWD1 52949393 Ki > 10000 nM T20251 CROV43 52949411 Ki > 10000 nM T20251 C0AZH4 52949420 Ki = 630 nM T20251 CVWY23 52949439 IC50 = 2.8 nM T20251 CRL18H 52949508 Ki = 1580 nM T20251 C9V6GB 52950007 IC50 = 0.95 nM T20251 C4OAP3 53234015 IC50 > 5000 nM T20251 CT3F0N 53235532 Ki = 700 nM T20251 C8ETM0 53237536 IC50 = 390 nM T20251 CYHS15 53237773 IC50 = 2000 nM T20251 C8EW1X 53239080 IC50 < 30000 nM T20251 CFI32H 53239287 Ki = 11600 nM T20251 CMYJ58 53239519 IC50 < 30000 nM T20251 CMQZ70 53242178 IC50 > 100000 nM T20251 CKNJ47 53245660 IC50 > 33000 nM T20251 CW9IQ0 53248730 IC50 > 33000 nM T20251 CQIY23 53248846 IC50 > 60000 nM T20251 C9MHR0 53248847 IC50 = 25000 nM T20251 CG3LA9 53248849 IC50 = 1890 nM T20251 CNB90W 53257735 IC50 = 19054.61 nM T20251 CW0M1K 53259021 IC50 = 1000 nM T20251 C70QNI 53260398 IC50 = 1000 nM T20251 C9NF0C 53302364 IC50 > 30000 nM T20251 CRB6N5 53307604 IC50 > 26302.68 nM T20251 CWQ8Y2 53307787 IC50 = 390 nM T20251 CR7TD8 53307788 IC50 > 10000 nM T20251 CQ87XN 53307874 Ki = 800 nM T20251 CW4S5E 53307875 Ki = 250 nM T20251 C7V1YI 53307876 Ki = 1100 nM T20251 C6QY4D 53307877 Ki = 1900 nM T20251 C68TEC 53307957 Ki = 970 nM T20251 CY92LZ 53310757 IC50 > 10000 nM T20251 CDT9H2 53310826 IC50 = 4300 nM T20251 CLZ60N 53310827 IC50 > 30000 nM T20251 C06JVE 53310828 IC50 > 30000 nM T20251 CZ6T1A 53310829 IC50 = 7100 nM T20251 CE9UD4 53310977 IC50 > 30000 nM T20251 C1O8DZ 53310978 IC50 > 30000 nM T20251 CCV51N 53310979 IC50 > 30000 nM T20251 C38JFV 53310980 IC50 > 30000 nM T20251 CR97IC 53310981 IC50 > 30000 nM T20251 CI6J2A 53310982 IC50 > 30000 nM T20251 C19ZEA 53311068 IC50 = 20500 nM T20251 CQ7B4Z 53311133 IC50 = 3000 nM T20251 CRI92N 53311230 IC50 > 50118.72 nM T20251 CJ83EB 53311393 IC50 = 4700 nM T20251 CG5WV2 53312065 IC50 = 9700 nM T20251 C89ETA 53312066 IC50 > 11000 nM T20251 CZ5IB8 53312148 IC50 > 11000 nM T20251 CVW9A8 53312150 IC50 > 11000 nM T20251 C9P4YV 53316457 IC50 = 3830 nM T20251 CW7TF1 53316459 IC50 = 1160 nM T20251 C1-MAY-02 53317017 IC50 > 10000 nM T20251 CPS12B 53317097 IC50 > 10000 nM T20251 CHNX58 53317305 IC50 = 4.3 nM T20251 CDH87Y 53317306 IC50 = 2.9 nM T20251 CK3MZ0 53317307 IC50 = 0.67 nM T20251 C9RK8W 53317504 IC50 = 1120 nM T20251 CNZ84M 53317555 IC50 = 6025.6 nM T20251 CK27PC 53317643 IC50 = 7300 nM T20251 CXV3W2 53317718 Ki > 60000 nM T20251 CP14EK 53317957 Ki = 35000 nM T20251 CL45CT 53318503 IC50 = 4300 nM T20251 C13SNK 53318592 IC50 > 10 nM T20251 CGWD27 53318593 IC50 = 2.4 nM T20251 C54SRN 53318594 IC50 = 7 nM T20251 C74CVF 53318595 IC50 = 1.7 nM T20251 C37ZAQ 53318697 IC50 = 4730 nM T20251 CBLD50 53318698 IC50 = 390 nM T20251 CK1ZI3 53318801 IC50 > 10 nM T20251 CB09MA 53318910 IC50 = 21000 nM T20251 CK2G3D 53319480 IC50 = 2000 nM T20251 CTA23R 53319654 IC50 = 7800 nM T20251 CUG7V3 53320013 IC50 = 990 nM T20251 CS04NZ 53320014 IC50 = 300 nM T20251 CTJ59M 53320020 Ki = 1621 nM T20251 CWLQ84 53320117 IC50 = 9.3 nM T20251 CVU69D 53320143 IC50 = 251.19 nM T20251 CGZX46 53320144 IC50 = 17.78 nM T20251 CXF1S4 53320328 IC50 = 1610 nM T20251 CB84NG 53320778 IC50 = 2320 nM T20251 CML70D 53321223 IC50 = 0.81 nM T20251 CQD62W 53321323 IC50 = 980 nM T20251 COT69M 53321324 IC50 = 510 nM T20251 CAJ4L7 53321331 Ki = 119 nM T20251 CJ9BK7 53321473 IC50 = 83176.38 nM T20251 C7Y2AB 53321474 IC50 = 74131.02 nM T20251 CRY96M 53321650 Ki = 3162.28 nM T20251 C4X3IS 53321979 IC50 = 3500 nM T20251 CMH54U 53322279 IC50 = 7600 nM T20251 C3YWZ5 53322451 IC50 = 40000 nM T20251 C98PDX 53322555 IC50 = 1.9 nM T20251 C5G8RQ 53322642 Ki = 7080 nM T20251 C1WA2E 53322643 Ki = 3802 nM T20251 C35XLW 53322810 IC50 = 4900 nM T20251 C01ILC 53322949 IC50 = 3162.28 nM T20251 CGN6Z3 53323531 Ki = 1.3 nM T20251 CR57HN 53323639 IC50 = 1400 nM T20251 CX54CT 53323813 IC50 = 23000 nM T20251 CDRV76 53323814 IC50 = 23000 nM T20251 C8ZHY7 53323979 IC50 = 310 nM T20251 C0HC8D 53324076 IC50 = 1.2 nM T20251 C1VNZ9 53324198 IC50 = 5000 nM T20251 CC08MY 53324265 IC50 > 20000 nM T20251 C2XT7J 53324382 IC50 = 107.15 nM T20251 C4ZO1H 53324408 IC50 = 2270 nM T20251 CS3L5G 53325164 IC50 = 4.3 nM T20251 CUO1R8 53325274 IC50 > 10000 nM T20251 CZB7M2 53325275 IC50 = 140 nM T20251 C3QNR2 53325463 IC50 = 3250 nM T20251 CZN8B4 53325581 IC50 = 5270 nM T20251 COS87G 53325596 IC50 = 102329.3 nM T20251 CY15EU 53325639 IC50 = 3900 nM T20251 CZ1SE0 53325908 Ki > 60000 nM T20251 C1N7XO 53325966 IC50 = 8600 nM T20251 CYA3F1 53325983 IC50 = 1500 nM T20251 C28HNA 53326213 IC50 > 10000 nM T20251 C9ZF4V 53326457 IC50 = 5.8 nM T20251 C3KWC5 53326627 IC50 > 10000 nM T20251 C5O1VT 53326682 IC50 = 537031.8 nM T20251 C0K7AS 53326693 IC50 = 218776.16 nM T20251 C18TPG 53326909 IC50 = 40000 nM T20251 C1KYR9 53326941 IC50 = 2600 nM T20251 CUF26V 53326945 IC50 = 501.19 nM T20251 C7J8ZY 53327611 IC50 = 13600 nM T20251 CQ7LB1 53327841 IC50 > 30000 nM T20251 CC6ME0 53327888 IC50 > 30000 nM T20251 C9F7ED 53341130 Ki = 1254 nM T20251 CCX7M5 53353847 IC50 > 30000 nM T20251 CS4HK7 53354783 IC50 = 170 nM T20251 C8PJ6E 53354789 IC50 = 40000 nM T20251 CYMP74 53354793 IC50 = 20000 nM T20251 C8ZRE3 53356518 IC50 > 80000 nM T20251 C6O7VL 53357600 IC50 = 25900 nM T20251 CYG6Q1 53358318 IC50 = 2600 nM T20251 C3B5AJ 53361011 IC50 > 30000 nM T20251 C9H5YE 53361128 IC50 > 10000 nM T20251 C23WVS 53361524 IC50 > 10000 nM T20251 CX83CK 53362097 IC50 = 5600 nM T20251 C54YUZ 53362500 IC50 > 10000 nM T20251 C6CR4I 53362501 IC50 = 1930 nM T20251 CJW0B3 53362502 IC50 = 440 nM T20251 CBAC86 53362558 IC50 = 4100 nM T20251 CYX87Q 53362559 IC50 = 2600 nM T20251 C8B1ZY 53362973 IC50 = 3800 nM T20251 COG5K0 53363092 IC50 = 7520 nM T20251 CCZW39 53363093 IC50 = 8160 nM T20251 CU59EZ 53363442 IC50 = 10000 nM T20251 C1PVA2 53363480 Ki = 6309.57 nM T20251 CU7VZ1 53363805 IC50 = 5770 nM T20251 C4D9RH 53363970 IC50 = 8480 nM T20251 C6N8KX 53363971 IC50 = 31240 nM T20251 C3WBV5 53364352 IC50 > 30000 nM T20251 CSV85J 53364356 IC50 = 10400 nM T20251 C2PHM7 53364357 IC50 = 10030 nM T20251 CNI7P9 53372541 IC50 = 10000 nM T20251 CA6H2P 53372668 IC50 = 398.11 nM T20251 CFM7W8 53372672 IC50 = 31622.78 nM T20251 C9GYZ3 53372790 IC50 = 3162.28 nM T20251 CT6K2O 53373472 IC50 = 15000 nM T20251 CL37YO 53380288 IC50 > 10000 nM T20251 C4ORN7 53380491 IC50 > 30000 nM T20251 CK52GI 53380818 IC50 > 30000 nM T20251 CZWO31 53387025 EC50 = 4700 nM T20251 C87NKH 53387026 IC50 = 4700 nM T20251 CCUH12 53387402 IC50 > 30000 nM T20251 CJ39QE 53387563 IC50 = 5700 nM T20251 CI15GW 53387564 IC50 = 21000 nM T20251 CS7X9W 53387565 IC50 = 5600 nM T20251 CIGM78 53389570 IC50 > 30000 nM T20251 CVG90B 53389651 IC50 > 10000 nM T20251 C47VGW 53393916 IC50 > 20000 nM T20251 C1QYU2 53464257 Ki = 5600 nM T20251 C6KC5V 53464567 Ki > 15000 nM T20251 C4Q0JV 53464571 Ki > 15000 nM T20251 CPE0Q3 53464695 Ki > 10000 nM T20251 CG7NH3 53464819 Ki = 2770 nM T20251 CC7P2U 53464882 Ki > 15000 nM T20251 CPRZ03 53464941 Ki > 10000 nM T20251 CRA3L0 53464942 Ki > 15000 nM T20251 CYE6O4 53464943 Ki > 10000 nM T20251 C3I8KD 53464944 Ki > 15000 nM T20251 C6K5JY 53464945 Ki > 10000 nM T20251 CK8YI4 53465003 Ki > 15000 nM T20251 C9K6FT 53465005 Ki > 15000 nM T20251 CH9CX8 53465067 Ki > 10000 nM T20251 CVM91G 53465142 Ki > 15000 nM T20251 C24FQU 53465297 IC50 = 9100 nM T20251 CHN72W 53469852 IC50 = 4200 nM T20251 CK1C9O 53472113 IC50 = 1400 nM T20251 CH5A9S 53484202 IC50 = 12080 nM T20251 CG3FA9 53492750 IC50 = 12882.5 nM T20251 C4U5IX 53493001 EC50 = 15000 nM T20251 CE9K7U 53494972 IC50 = 53000 nM T20251 C7TR2W 53497131 IC50 = 25100 nM T20251 CWA14L 53802926 IC50 = 6309.57 nM T20251 CP24ZC 54579002 IC50 = 8700 nM T20251 CTA9K1 54579972 IC50 = 45 nM T20251 C1GXF9 54579973 IC50 = 370 nM T20251 CQ8AZ0 54580065 Ki = 1584.89 nM T20251 CYM8N2 54580066 Ki = 794.33 nM T20251 CT2FB8 54580068 Ki = 1995.26 nM T20251 C4KGT2 54580069 Ki = 2511.89 nM T20251 CL5V4H 54580071 Ki = 316.23 nM T20251 CG86QM 54580083 IC50 = 56234.13 nM T20251 C4RH7W 54580091 IC50 = 18197.01 nM T20251 CC0R4A 54580092 IC50 > 31622.78 nM T20251 C73HNQ 54580097 IC50 = 41686.94 nM T20251 C89MEB 54580190 IC50 = 8600 nM T20251 CMDO43 54580283 Ki = 80 nM T20251 C6M4ND 54580284 Ki = 40 nM T20251 CB58LO 54580324 IC50 = 8912.51 nM T20251 CLW26Q 54580457 IC50 = 160 nM T20251 CRV6M8 54580555 IC50 = 900 nM T20251 C2YWA6 54580845 IC50 = 8620 nM T20251 C6R3MZ 54580973 IC50 = 790 nM T20251 C4GAB9 54581050 Ki = 1584.89 nM T20251 CP7HC3 54581052 Ki = 2511.89 nM T20251 CF9L7B 54581072 IC50 = 44668.36 nM T20251 C54SOM 54581080 IC50 > 50118.72 nM T20251 CC3J5L 54581190 IC50 = 7600 nM T20251 C8S1LG 54581286 Ki = 80 nM T20251 CQ6V1E 54581466 IC50 = 1030 nM T20251 C4EH1F 54581551 IC50 = 440 nM T20251 CBT56Y 54581676 IC50 = 2300 nM T20251 CJV9G1 54581702 IC50 = 3200 nM T20251 CQ0YA3 54581861 IC50 = 1890 nM T20251 CHJK47 54581904 IC50 = 6230 nM T20251 C7QWE4 54581905 IC50 = 9400 nM T20251 C8CTD7 54581962 IC50 = 1200 nM T20251 CUN59X 54582014 IC50 = 28 nM T20251 C5S1ZK 54582015 IC50 = 1960 nM T20251 CWKA42 54582019 IC50 = 2000 nM T20251 CL52TN 54582094 Ki = 251.19 nM T20251 CB6DW8 54582096 Ki = 630.96 nM T20251 C10TMQ 54582108 IC50 = 31622.78 nM T20251 C69IDP 54582109 IC50 = 1995.26 nM T20251 C5Y1OZ 54582114 IC50 > 50118.72 nM T20251 CG3HB9 54582215 IC50 = 2100 nM T20251 C4KMX1 54582216 IC50 = 8900 nM T20251 CD1AE2 54582217 IC50 = 6500 nM T20251 CAG68L 54582303 Ki = 200 nM T20251 C51QIK 54582357 IC50 = 7943.28 nM T20251 C1HBD8 54582798 IC50 = 16000 nM T20251 CB8JV7 54582823 IC50 = 7110 nM T20251 CZ71VB 54582892 IC50 > 30000 nM T20251 C2CAO0 54582957 IC50 = 200 nM T20251 CZ3DW2 54582958 IC50 = 47 nM T20251 CS3P4K 54582960 IC50 = 29 nM T20251 CD0WT4 54582961 IC50 = 16 nM T20251 CP8TG1 54583028 Ki = 251.19 nM T20251 CHT78R 54583030 Ki = 630.96 nM T20251 CUHW91 54583050 IC50 = 1584.89 nM T20251 CX24KS 54583051 IC50 = 50118.72 nM T20251 CB8S6F 54583055 IC50 > 31622.78 nM T20251 C14MKQ 54583056 IC50 = 794.33 nM T20251 CUC32E 54583059 IC50 = 52480.75 nM T20251 CLX7U9 54583111 IC50 = 17000 nM T20251 C3WZ9I 54583112 IC50 = 52800 nM T20251 CYD20W 54583185 IC50 = 42600 nM T20251 COQD25 54583186 IC50 = 1200 nM T20251 CC19ZA 54583187 IC50 = 300 nM T20251 CEOZ15 54583522 IC50 = 12500 nM T20251 CXLA39 54583624 IC50 = 30000 nM T20251 C9OB1C 54583833 IC50 = 6670 nM T20251 CE61RX 54583834 IC50 = 5200 nM T20251 CG78OW 54583895 IC50 = 5400 nM T20251 CSCE48 54583896 IC50 = 1500 nM T20251 C6UED1 54583954 IC50 = 56 nM T20251 CU10AQ 54584056 IC50 = 79432.82 nM T20251 CUKW62 54584057 IC50 = 63095.73 nM T20251 CDV2Z9 54584068 IC50 = 30902.95 nM T20251 C90AHI 54584164 IC50 = 3900000 nM T20251 C7MP0S 54584254 Ki = 4168.69 nM T20251 CY80OU 54584273 Ki = 500 nM T20251 C8YEA3 54584294 IC50 = 30199.52 nM T20251 C4LN8M 54584295 IC50 = 12882.5 nM T20251 CVUI69 54584296 IC50 = 100000 nM T20251 CJV94T 54584501 IC50 = 3400 nM T20251 CPS93U 54584537 IC50 < 200 nM T20251 CTM3D4 54584797 IC50 = 3850 nM T20251 CF49IN 54584798 IC50 = 18800 nM T20251 C3C8QF 54584905 IC50 = 34 nM T20251 C7UY2T 54584908 IC50 = 28 nM T20251 CR7UW2 54584957 IC50 = 31622.78 nM T20251 C8P6MI 54584991 Ki = 1000 nM T20251 CI0P4H 54585005 IC50 = 125892.54 nM T20251 CZ4S0B 54585107 IC50 > 90000 nM T20251 C3TAR4 54585108 IC50 = 35900 nM T20251 C8RTU2 54585109 IC50 < 300 nM T20251 CL7P1G 54585233 Ki = 5011.87 nM T20251 C9PB7S 54585251 IC50 = 36307.81 nM T20251 C30LYP 54585371 Ki = 630.96 nM T20251 C2A6ER 54585480 IC50 < 200 nM T20251 CY5LT9 54585737 IC50 = 18600 nM T20251 C0C2BE 54585833 IC50 = 600 nM T20251 CPX76L 54585862 IC50 = 20300 nM T20251 CW31VH 54585863 IC50 = 120 nM T20251 C2M9RO 54585864 IC50 = 4620 nM T20251 C8OR2E 54585941 Ki = 3981.07 nM T20251 C4V8AE 54585969 IC50 = 25118.86 nM T20251 CN8E3L 54585970 IC50 = 6025.6 nM T20251 CJ4QK6 54585971 IC50 = 63095.73 nM T20251 CH6X1P 54585974 IC50 > 31622.78 nM T20251 CC6HY7 54586021 IC50 = 1100 nM T20251 C3MLH7 54586172 Ki = 1584.89 nM T20251 CSX84E 54586210 IC50 = 10000 nM T20251 CSC0H3 54586414 IC50 = 16400 nM T20251 C7HD0U 54586415 IC50 = 1500 nM T20251 C8TLD6 54586719 IC50 = 2150 nM T20251 CYVZ19 54586720 IC50 = 2180 nM T20251 C67NFK 54586780 IC50 = 10600 nM T20251 C4ACJ8 54586781 IC50 = 4000 nM T20251 C59FXV 54586919 Ki = 1258.93 nM T20251 CTK5S1 54586921 Ki = 794.33 nM T20251 CCL0M3 54586940 IC50 = 25118.86 nM T20251 C6VQT3 54587171 Ki = 150 nM T20251 CSX1R5 54587172 Ki = 3700 nM T20251 CO19MR 54587173 Ki = 2300 nM T20251 CLAJ60 54587208 Ki = 1258.93 nM T20251 C09OSL 54587230 IC50 = 12022.64 nM T20251 C0UYD7 54587231 IC50 = 8912.51 nM T20251 CD06RB 54587434 IC50 = 24400 nM T20251 C8MH6B 54587759 IC50 = 27000 nM T20251 CH3US7 54587760 IC50 > 33000 nM T20251 CZ5IY9 54587813 IC50 = 2600 nM T20251 C30XLO 54592009 IC50 > 100000 nM T20251 C57DQW 54670057 IC50 = 100 nM T20251 C7L5YB 54670058 IC50 = 39 nM T20251 CM7FC6 54670152 IC50 = 780 nM T20251 CF7XA0 54674257 IC50 = 21000 nM T20251 C3S9EC 54674292 IC50 = 12140 nM T20251 C9JCZ5 54675567 IC50 = 2780 nM T20251 C0ZG2V 54709839 IC50 = 20000 nM T20251 CO75TL 54712015 IC50 > 50000 nM T20251 CLT3Q8 54716246 IC50 > 10000 nM T20251 C28RDF 54746913 IC50 > 60000 nM T20251 C5OBC3 54753437 IC50 > 10000 nM T20251 CGIP16 54754722 IC50 = 32000 nM T20251 CX4LK5 54754723 IC50 = 5600 nM T20251 C6LZ8B 54754724 IC50 = 5000 nM T20251 CSA9I6 54754844 IC50 = 24000 nM T20251 CEGJ53 54754845 IC50 = 32000 nM T20251 C9NV8L 54754967 IC50 = 32000 nM T20251 CI78YZ 54754968 IC50 = 2500 nM T20251 CV3K8U 54754969 IC50 = 1100 nM T20251 C6T8XS 54755079 IC50 = 9500 nM T20251 CL2AU5 54755081 IC50 = 9100 nM T20251 C2R6KO 54755083 IC50 = 34000 nM T20251 C5LT0A 54755193 IC50 = 6200 nM T20251 C3SD6W 54755560 IC50 = 7600 nM T20251 C4GBT5 54755562 IC50 = 2500 nM T20251 C0KZ4M 54755801 IC50 = 7600 nM T20251 C2QP4W 54755919 IC50 = 1900 nM T20251 CPWZ05 54756038 IC50 = 5600 nM T20251 CJBW64 54756045 IC50 = 20000 nM T20251 C0ZWL2 54756156 IC50 = 3700 nM T20251 CI20JA 54756906 IC50 = 6760.83 nM T20251 CCG08B 54756907 IC50 = 12589.25 nM T20251 CK50BF 54756908 IC50 = 19952.62 nM T20251 CILG27 54758399 IC50 = 17782.79 nM T20251 C8AB1J 54759606 IC50 = 18830 nM T20251 C80STN 54761221 IC50 > 10000 nM T20251 C0Y9ZG 54761473 IC50 = 15000 nM T20251 CU62DN 54764919 IC50 > 10000 nM T20251 C0T3KY 54765285 IC50 = 3700 nM T20251 CFHI34 54768835 IC50 = 8300 nM T20251 CLY35F 54768836 IC50 = 2100 nM T20251 C9U4YQ 54768838 IC50 = 25700 nM T20251 CO4FY1 54769305 IC50 = 5200 nM T20251 CFC91M 54769914 IC50 = 9000 nM T20251 CWN90Q 54771978 IC50 = 32900 nM T20251 CUM4B5 54771980 IC50 = 7500 nM T20251 CL7UD5 54772203 IC50 = 16000 nM T20251 CH7K6J 54772204 IC50 = 12900 nM T20251 C4E5YQ 54772205 IC50 = 6600 nM T20251 C7Y8KR 54772206 IC50 = 20200 nM T20251 C8WHT5 56593934 IC50 = 7943.28 nM T20251 C8KO5T 56595054 IC50 = 720 nM T20251 CW89BT 56595402 IC50 > 10000 nM T20251 C4C3XQ 56595529 IC50 > 10000 nM T20251 CXEH21 56595883 IC50 > 10000 nM T20251 C7G4FQ 56596230 IC50 > 50000 nM T20251 CCG6D9 56597407 IC50 = 5500 nM T20251 CAC5B2 56597542 IC50 = 9800 nM T20251 CTK41N 56597689 IC50 = 8600 nM T20251 CN54TH 56597851 IC50 = 10000 nM T20251 CZNV53 56597988 IC50 = 15000 nM T20251 CI6B8D 56597990 IC50 > 33000 nM T20251 CSU5C1 56597991 IC50 > 33000 nM T20251 CJ4V0G 56598130 IC50 = 21000 nM T20251 CCR0Z1 56598517 IC50 > 25000 nM T20251 CK6VF3 56598528 IC50 = 8500 nM T20251 C91PGO 56603115 IC50 = 14700 nM T20251 C5ES6P 56603116 IC50 = 5400 nM T20251 CVI51O 56603118 IC50 = 19500 nM T20251 C2IM6T 56603174 IC50 = 4900 nM T20251 CH05TN 56603175 IC50 = 4400 nM T20251 CDL94H 56603301 IC50 = 1200 nM T20251 C9D1MV 56603353 IC50 = 16000 nM T20251 C60YTB 56603356 IC50 = 560 nM T20251 C9ZF6B 56643412 IC50 = 1200 nM T20251 CGX06Z 56643450 IC50 = 5000 nM T20251 CQ18BI 56643478 IC50 = 3700 nM T20251 CXI5V1 56643481 IC50 = 4840 nM T20251 CH3BN6 56643486 IC50 = 3460 nM T20251 CNB76L 56643505 IC50 > 30000 nM T20251 CS5P3M 56643544 IC50 = 24000 nM T20251 C6XI4W 56647652 IC50 = 4310 nM T20251 CUGA78 56649284 IC50 = 15500 nM T20251 C94RZF 56657929 IC50 = 10000 nM T20251 COST81 56657930 IC50 = 12000 nM T20251 CP2B8C 56657939 Ki = 5 nM T20251 CJ93HB 56657949 IC50 = 360 nM T20251 C13WTO 56658050 IC50 = 24000 nM T20251 C71XNV 56658572 IC50 = 2300 nM T20251 C21NEQ 56659196 IC50 > 50000 nM T20251 C7B9TW 56659197 IC50 = 25000 nM T20251 CL2YE8 56659224 IC50 = 4600 nM T20251 C5F1TD 56659225 IC50 = 10000 nM T20251 CUM53N 56659295 IC50 = 8.7 nM T20251 CVG04B 56659303 IC50 = 501.19 nM T20251 CRTE61 56659304 IC50 = 1000 nM T20251 C3R8ZJ 56659305 IC50 = 2511.89 nM T20251 CXBH95 56659572 Ki = 7200 nM T20251 CS4N2M 56659870 IC50 > 10000 nM T20251 CI1Z4B 56659871 IC50 = 8100 nM T20251 C0PSG1 56659872 IC50 = 2150 nM T20251 CJZS68 56660076 Ki = 27000 nM T20251 C4IZL5 56661444 IC50 = 4700 nM T20251 CQ25TB 56661451 IC50 = 18000 nM T20251 CM6A3K 56661468 Ki = 190 nM T20251 CC3XP8 56661559 IC50 = 25000 nM T20251 CCA76B 56661560 IC50 = 9400 nM T20251 C4H3VZ 56661561 IC50 = 17000 nM T20251 C43ICJ 56661679 IC50 = 4300 nM T20251 CJ0VW5 56662035 IC50 = 1300 nM T20251 CXFL76 56662692 IC50 > 33000 nM T20251 C7K4TJ 56662695 IC50 = 23000 nM T20251 CO3I1H 56662705 IC50 = 10000 nM T20251 CF45CH 56662780 IC50 = 4730 nM T20251 CP2LW0 56662936 IC50 = 316 nM T20251 CME1K7 56663526 Ki = 15000 nM T20251 CMI4D9 56663528 Ki = 12000 nM T20251 C9T2JQ 56663564 IC50 = 9900 nM T20251 C1KDU3 56663565 IC50 = 12000 nM T20251 CO1E6D 56663566 IC50 = 9400 nM T20251 CED2I5 56663567 IC50 = 4300 nM T20251 C3XW6G 56664901 Ki = 818 nM T20251 C9WDB6 56664902 IC50 = 8400 nM T20251 C7SJH2 56664979 IC50 = 840 nM T20251 CMY64U 56665506 IC50 = 45000 nM T20251 CL4XG3 56666171 IC50 = 7200 nM T20251 C6B7WR 56666236 IC50 = 2511.89 nM T20251 CVBA49 56666237 IC50 = 2511.89 nM T20251 C45XIM 56666238 IC50 > 50118.72 nM T20251 CHB63V 56666239 IC50 = 40000 nM T20251 CMZ6K8 56666240 IC50 = 8400 nM T20251 CYA27T 56666252 IC50 = 920 nM T20251 CL0BX9 56666253 IC50 = 310 nM T20251 C6I7DL 56666254 IC50 = 480 nM T20251 C0QOY7 56666255 IC50 = 2350 nM T20251 C4MFS5 56666758 IC50 = 320 nM T20251 CF0KZ2 56666759 IC50 > 10000 nM T20251 C62JDU 56666760 IC50 > 10000 nM T20251 CZG61M 56666868 IC50 = 4730 nM T20251 CLF45N 56666970 Ki > 29000 nM T20251 CUL0F4 56667010 IC50 = 8800 nM T20251 C9G1FY 56667011 IC50 = 14000 nM T20251 CA6K8E 56667012 IC50 = 8100 nM T20251 C2HXG3 56667013 IC50 = 1300 nM T20251 CC5S6K 56667036 IC50 = 3800 nM T20251 CF2N5W 56668309 IC50 = 12000 nM T20251 C4SP2W 56668313 IC50 = 4100 nM T20251 CT37LU 56668326 Ki = 13 nM T20251 C31SKP 56668413 IC50 > 50000 nM T20251 CJ95CA 56668427 Ki = 14 nM T20251 CX4Z9G 56668494 IC50 > 30000 nM T20251 CF7LR5 56668542 IC50 = 7100 nM T20251 CVGX27 56668837 Ki > 29000 nM T20251 CRVH74 56668949 IC50 > 100000 nM T20251 CKO8M6 56669554 IC50 > 33000 nM T20251 CI5Y4E 56669631 IC50 > 50 nM T20251 C5OF9G 56669642 IC50 = 3981.07 nM T20251 C4NR8W 56669644 IC50 = 16800 nM T20251 C5LE0N 56669662 IC50 = 1500 nM T20251 C36RHL 56669664 IC50 = 1570 nM T20251 C2HW9M 56669665 IC50 = 1900 nM T20251 CF06GH 56669910 Ki > 29000 nM T20251 CZO49F 56670192 IC50 = 2490 nM T20251 C5K4NS 56670257 IC50 = 8181.82 nM T20251 C9P6EQ 56670309 IC50 = 1500 nM T20251 CF23IK 56670310 IC50 = 4760 nM T20251 CRE51K 56670312 IC50 = 1570 nM T20251 CC7FH3 56670429 Ki = 1200 nM T20251 C76KFA 56670457 IC50 > 33000 nM T20251 C0I6AP 56670458 IC50 = 5300 nM T20251 C9Y8PV 56670459 IC50 = 10000 nM T20251 C5E7OB 56670460 IC50 = 16000 nM T20251 CCPY59 56670461 IC50 = 14000 nM T20251 CUP61N 56671791 IC50 = 1584.89 nM T20251 C34WPT 56671792 IC50 = 36000 nM T20251 CXUJ14 56671793 IC50 = 24000 nM T20251 C4UHW2 56671794 IC50 = 12000 nM T20251 CG1JX9 56671795 IC50 > 50000 nM T20251 CY0GX2 56671810 Ki = 10000 nM T20251 C2GFT1 56671811 Ki = 230 nM T20251 CCI1K3 56671812 Ki = 2220 nM T20251 C9GRW8 56671830 IC50 = 920 nM T20251 CXIQ98 56671923 IC50 = 1200 nM T20251 C19LWV 56671924 IC50 = 3100 nM T20251 CE3Y0C 56671925 IC50 = 8000 nM T20251 CX3LP4 56672008 IC50 = 22700 nM T20251 CET7K4 56672021 IC50 > 50 nM T20251 C29OYU 56672433 IC50 > 100000 nM T20251 CK9L4C 56672570 IC50 = 47300 nM T20251 CGAF01 56673075 IC50 = 14000 nM T20251 CP9Z2L 56673090 IC50 = 2000 nM T20251 C83MQK 56673091 IC50 = 2900 nM T20251 C6E7WM 56673153 IC50 = 794.33 nM T20251 C2Z1LP 56673154 IC50 = 3981.07 nM T20251 CC04NV 56673156 IC50 = 6000 nM T20251 C6FPR7 56673157 IC50 = 4800 nM T20251 C5G0ID 56673158 IC50 = 2480 nM T20251 C04ZUP 56673173 IC50 = 2800 nM T20251 C39ADI 56673420 Ki = 8400 nM T20251 C1E4CX 56673467 IC50 > 30000 nM T20251 C4G0YE 56673715 IC50 = 2190 nM T20251 CWZV47 56673716 IC50 = 390 nM T20251 C1KW9Z 56673717 IC50 = 5430 nM T20251 C19GOU 56673914 Ki = 17000 nM T20251 CW4J1Y 56673944 IC50 > 30000 nM T20251 CK5HP1 56673946 IC50 > 33000 nM T20251 C2D4JW 56673947 IC50 = 9400 nM T20251 CPU13M 56673948 IC50 = 4800 nM T20251 CY26SL 56675205 IC50 = 27000 nM T20251 CN3UM2 56675220 IC50 = 890 nM T20251 C03LOT 56675300 IC50 = 30000 nM T20251 CK9JX5 56675301 IC50 = 4500 nM T20251 CU0H6Z 56675302 IC50 = 7400 nM T20251 CJEA89 56675420 IC50 = 28000 nM T20251 C8JX6T 56675817 IC50 > 100000 nM T20251 CC73NZ 56676392 IC50 = 620 nM T20251 CP41OM 56676397 IC50 = 10000 nM T20251 CWS95P 56676398 IC50 = 5108.11 nM T20251 C0KG7I 56676474 IC50 = 11 nM T20251 CF3G7P 56676480 IC50 = 1584.89 nM T20251 CN4US8 56676481 IC50 = 3162.28 nM T20251 C49LUC 56676482 IC50 = 25118.86 nM T20251 CW86SU 56676730 Ki > 29000 nM T20251 CV79CF 56677248 Ki = 11000 nM T20251 CTW73X 56677275 IC50 = 1500 nM T20251 CHG64Z 56677276 IC50 = 9500 nM T20251 CBTG12 56677288 IC50 = 11700 nM T20251 CU35WX 56677289 IC50 = 7600 nM T20251 CE3T1U 56677296 IC50 = 1500 nM T20251 CP14LU 56678505 IC50 = 2511.89 nM T20251 CD8IZ5 56678506 IC50 = 25000 nM T20251 C7QW5F 56678507 IC50 = 44000 nM T20251 C7MXE5 56678508 IC50 = 27000 nM T20251 C5M0AS 56678518 Ki = 10000 nM T20251 C7IWP6 56678519 Ki = 1194 nM T20251 C0IGC6 56678520 Ki = 841 nM T20251 CT7BE0 56678521 Ki = 76 nM T20251 CUM2R9 56678534 IC50 = 160 nM T20251 C2O4SY 56678640 IC50 = 23000 nM T20251 CO9AX8 56678641 IC50 = 5800 nM T20251 C8QOB7 56678653 Ki = 90 nM T20251 CY5HJ2 56678654 Ki = 2747 nM T20251 CSHO51 56679737 IC50 = 10000 nM T20251 CDS09F 56679795 IC50 = 6309.57 nM T20251 CU04BI 56679796 IC50 = 7943.28 nM T20251 CTEK36 56679797 IC50 = 7943.28 nM T20251 COSK12 56679817 IC50 = 360 nM T20251 CM51TG 56679818 IC50 = 4980 nM T20251 CGCA84 56680098 IC50 > 30000 nM T20251 C9DTH0 56680351 IC50 = 1250 nM T20251 CMR0J9 56680352 IC50 > 10000 nM T20251 CDIZ56 56680456 IC50 = 3210 nM T20251 C67GMA 56680575 IC50 = 5100 nM T20251 C4MH8J 56681858 Ki = 1125 nM T20251 C1A0OH 56681872 IC50 = 130 nM T20251 C6ZOT4 56681873 IC50 = 460 nM T20251 C1XR6E 56681874 IC50 = 290 nM T20251 CPD15R 56681875 IC50 = 13830 nM T20251 C06HAF 56681960 IC50 = 38000 nM T20251 C1Y0MO 56682216 IC50 = 10000 nM T20251 CIW1T6 56683044 IC50 = 31000 nM T20251 CY1QA2 56683053 IC50 = 29000 nM T20251 C7F1JG 56683065 IC50 = 10000 nM T20251 CKVB12 56683116 IC50 = 17000 nM T20251 C9KMN5 56683121 IC50 = 16 nM T20251 CYJ1S0 56683143 IC50 = 3210 nM T20251 CBZG16 56683144 IC50 = 4760 nM T20251 CEYA71 56683146 IC50 = 1290 nM T20251 CP9G8Z 56683392 Ki > 29000 nM T20251 CR0E4M 56683440 IC50 > 30000 nM T20251 C4X7IP 56683681 IC50 = 2700 nM T20251 CIY31D 56683751 IC50 = 420 nM T20251 CH92EZ 56683889 Ki = 1700 nM T20251 CY1W2Q 56683890 Ki = 750 nM T20251 CWBF48 56683908 IC50 = 15000 nM T20251 C0MQ2W 56832511 IC50 = 16000 nM T20251 CE3PY9 56834574 IC50 = 23000 nM T20251 CD2FQ8 56834575 IC50 > 33000 nM T20251 CAJ3G0 56834577 IC50 = 206000 nM T20251 CY0K3F 56834578 IC50 > 33000 nM T20251 CMY23H 56834579 IC50 > 33000 nM T20251 CY92VU 56835087 IC50 > 30000 nM T20251 C0JMA7 56835088 IC50 = 7000 nM T20251 CR7LS4 56835090 IC50 = 20000 nM T20251 C4E6HV 56835171 Ki = 3235.94 nM T20251 CK7HJ8 56837192 Ki = 23000 nM T20251 C73MZW 56924689 IC50 = 13000 nM T20251 C8ZW3O 56927659 Ki = 1701 nM T20251 CV8W4T 56933229 IC50 > 300000 nM T20251 C9KI7Q 56940718 IC50 = 23700 nM T20251 CP5UD4 56944043 IC50 > 10000 nM T20251 C6F3VI 56944044 IC50 = 7700 nM T20251 C6GDX1 56944245 IC50 = 2200 nM T20251 CB0P9N 56944383 IC50 = 4000 nM T20251 C09WRF 56944429 IC50 = 4800 nM T20251 CHRU78 56946423 IC50 = 3300 nM T20251 CDK93W 56946894 IC50 > 100000 nM T20251 C5LJE8 56951456 IC50 > 30000 nM T20251 C6N0ZI 56951457 IC50 > 30000 nM T20251 CL90EM 56951458 IC50 > 30000 nM T20251 CD3V1J 56952775 IC50 = 2800 nM T20251 C8L7SJ 56952776 IC50 = 2540 nM T20251 CR9Q2E 56952777 IC50 = 2890 nM T20251 C0L4QG 56952778 IC50 = 670 nM T20251 CKMG86 56953069 IC50 = 920 nM T20251 C4V6ET 56953070 IC50 = 1480 nM T20251 CAK91L 56955954 IC50 = 17318 nM T20251 CP8H0D 56962365 IC50 = 5800 nM T20251 C1TR4E 56963091 Ki = 10700 nM T20251 C9L6FD 56963908 IC50 = 400 nM T20251 CKN0Z8 56964577 IC50 > 25000 nM T20251 C62OJE 56970264 IC50 = 27400 nM T20251 CJ6DK1 56970422 IC50 = 1600 nM T20251 C7S9ER 56970466 IC50 > 30000 nM T20251 CDH38V 56970630 IC50 = 3000 nM T20251 C67JVW 56970631 IC50 = 670 nM T20251 C4DMU9 56970632 IC50 = 1900 nM T20251 C3RBO8 56970861 IC50 = 430 nM T20251 CJ5O6Y 56970863 IC50 = 670 nM T20251 C1DN0L 56970864 IC50 = 470 nM T20251 CRF6L7 56971088 IC50 = 12 nM T20251 CQ5IH3 56971089 IC50 <= 1000 nM T20251 C9N0LO 56971556 IC50 = 31 nM T20251 CONA69 57065698 IC50 = 4660 nM T20251 CT67IO 57325589 IC50 > 25000 nM T20251 CV5CP4 57326678 IC50 = 6480 nM T20251 CVK5A3 57328247 IC50 = 100000 nM T20251 CQT5I3 57328465 IC50 = 8500 nM T20251 CY3B1Z 57330204 IC50 = 3600 nM T20251 CHN80L 57331188 IC50 = 12000 nM T20251 C4E1NK 57331209 IC50 = 1400 nM T20251 C8PWJ3 57331210 IC50 = 14000 nM T20251 C1E3WV 57331240 IC50 = 160 nM T20251 C4WI9O 57331241 IC50 = 1300 nM T20251 C68CPW 57331268 IC50 = 2700 nM T20251 CD0WM9 57331302 IC50 = 18000 nM T20251 CY0W1H 57331373 IC50 = 1300 nM T20251 CLB5K0 57331386 IC50 = 101700 nM T20251 CGUA26 57331668 IC50 = 17000 nM T20251 C64PSR 57331747 IC50 = 46000 nM T20251 CH30RG 57334102 IC50 = 159 nM T20251 C6DK4O 57334404 IC50 = 820 nM T20251 CD9I4N 57334553 IC50 = 1591 nM T20251 CXQ47N 57334707 IC50 = 226 nM T20251 CEG4N8 57334716 Ki = 470 nM T20251 C0UW5Z 57341142 EC50 = 4500 nM T20251 CS2FH5 57341143 EC50 = 5800 nM T20251 C2AUM9 57341144 EC50 > 30000 nM T20251 CX1FQ0 57341332 EC50 > 30000 nM T20251 CN3Y9D 57341333 EC50 > 30000 nM T20251 C3H1GV 57341334 EC50 = 27500 nM T20251 C0Z3JI 57341335 EC50 > 30000 nM T20251 C83DHY 57341336 EC50 > 30000 nM T20251 CDU9W0 57341337 EC50 > 30000 nM T20251 CL45WN 57345320 IC50 = 8920 nM T20251 CHE2I1 57345500 IC50 = 950 nM T20251 C63TFM 57345501 IC50 = 13300 nM T20251 C8KT2F 57345502 IC50 = 10000 nM T20251 CYZ1S5 57345568 IC50 = 326 nM T20251 CW4QD9 57345597 IC50 = 3200 nM T20251 CBQK82 57345598 IC50 = 16100 nM T20251 C3REK0 57345599 IC50 = 1288.25 nM T20251 CX49PE 57345600 IC50 = 1299.87 nM T20251 CD50GK 57345628 IC50 = 8900 nM T20251 COTF12 57382553 IC50 = 25700 nM T20251 CBF53W 57384005 IC50 = 5500 nM T20251 CF1OM2 57384006 IC50 > 40000 nM T20251 C8X5JG 57384039 IC50 = 8600 nM T20251 CV0GJ4 57384040 IC50 > 33000 nM T20251 C73XBL 57384077 Ki = 369 nM T20251 C34DJP 57384236 IC50 = 17000 nM T20251 CEOC15 57384237 IC50 = 720 nM T20251 CY50WC 57384238 IC50 = 4700 nM T20251 C7S0ZR 57384239 IC50 = 15000 nM T20251 C2XN1G 57384481 IC50 = 370 nM T20251 CR73IZ 57384482 IC50 = 650 nM T20251 CR2M5H 57384483 IC50 = 8500 nM T20251 CQ72HI 57384749 IC50 = 8900 nM T20251 C68KGE 57384750 IC50 = 7100 nM T20251 CQX8J0 57385070 IC50 > 300000 nM T20251 CPS89B 57385071 IC50 > 300000 nM T20251 CNU9C0 57385072 IC50 > 300000 nM T20251 CG5MT6 57385073 IC50 > 300000 nM T20251 CMC8H6 57386782 IC50 > 30000 nM T20251 CCT5D4 57386783 IC50 = 7000 nM T20251 CC30XZ 57386784 IC50 = 2400 nM T20251 C79BXP 57386785 IC50 > 60000 nM T20251 CM6DV7 57387028 IC50 = 5700 nM T20251 C0GS4F 57387282 IC50 = 12000 nM T20251 C0TL9C 57387283 IC50 = 8000 nM T20251 CRV2P5 57387539 IC50 = 1400 nM T20251 CAU3G9 57387540 IC50 = 7800 nM T20251 CL2AO8 57387541 IC50 = 23000 nM T20251 C0XWL8 57387542 IC50 = 16000 nM T20251 CC4DK0 57387775 IC50 = 2500 nM T20251 CSH7D9 57390216 IC50 = 5400 nM T20251 CLN2F8 57390217 IC50 = 11000 nM T20251 CM37LJ 57390221 Ki = 600 nM T20251 C58KFP 57390222 Ki = 900 nM T20251 CSCB73 57390223 Ki = 620 nM T20251 CVO05U 57390547 IC50 = 7900 nM T20251 CP8D5L 57390807 Ki = 43000 nM T20251 CDJC72 57390808 Ki = 24000 nM T20251 CE03ZS 57390809 Ki = 29000 nM T20251 CR8MW2 57391205 IC50 > 100000 nM T20251 CI9UT0 57391292 IC50 = 13489.63 nM T20251 C78LTO 57391294 IC50 = 1300 nM T20251 C2AR3V 57391609 IC50 = 900 nM T20251 CCA7D3 57391720 IC50 = 5800 nM T20251 C5QD2I 57391722 IC50 = 7900 nM T20251 CBEO41 57391765 IC50 > 30 nM T20251 CK9L1O 57391766 IC50 > 30 nM T20251 CN1Q4Y 57391767 IC50 > 30 nM T20251 CC53ND 57391768 IC50 > 30 nM T20251 CKPB03 57391802 IC50 = 2800 nM T20251 C8SW9E 57391803 IC50 = 4300 nM T20251 C5UWC6 57391804 IC50 = 9000 nM T20251 C78QEY 57391805 IC50 = 16900 nM T20251 CYAQ83 57391806 IC50 = 21700 nM T20251 CZ1EH9 57391826 IC50 = 33000 nM T20251 COL58X 57391831 IC50 = 12000 nM T20251 C6SGK0 57391843 Ki > 3000 nM T20251 C3MUQ4 57392006 IC50 = 15000 nM T20251 C4S7ET 57392007 IC50 = 18000 nM T20251 CT96ZS 57392011 Ki = 4500 nM T20251 CB6C4T 57392012 Ki = 910 nM T20251 CCZJ34 57392013 Ki = 1300 nM T20251 CP48ZB 57392014 Ki = 880 nM T20251 CHSW27 57392492 IC50 < 1000 nM T20251 CX89LJ 57392493 IC50 = 1300 nM T20251 C16PSG 57392623 Ki = 20000 nM T20251 CFM8E5 57392624 Ki = 8200 nM T20251 CGB71E 57393073 IC50 = 2398.83 nM T20251 CPQC75 57393451 IC50 = 7900 nM T20251 CJTY79 57393468 IC50 > 30000 nM T20251 CKS3X9 57393534 IC50 = 28200 nM T20251 CM2EH0 57393535 IC50 > 30000 nM T20251 CVO5M3 57393573 IC50 = 450 nM T20251 C9K0MG 57393724 IC50 = 13000 nM T20251 C2V7SB 57393725 IC50 > 33000 nM T20251 CH97QF 57393726 Ki = 460 nM T20251 CM80PV 57393727 Ki = 250 nM T20251 CJE1N0 57393728 Ki = 160 nM T20251 CWC2E8 57393729 Ki = 340 nM T20251 C13XZY 57394046 IC50 = 52000 nM T20251 C2XNP7 57394056 IC50 = 200000 nM T20251 C6D7UA 57394195 IC50 = 3900 nM T20251 CHA2Q7 57394339 Ki = 20000 nM T20251 CS8M9I 57394340 Ki = 1800 nM T20251 CLP4Z8 57394341 Ki = 12000 nM T20251 C8PWV4 57394342 Ki = 10000 nM T20251 C16OJD 57394343 Ki = 5700 nM T20251 C0AJM8 57394344 Ki = 55000 nM T20251 C6HR3Q 57394345 Ki = 47000 nM T20251 C0XDZ8 57394407 IC50 = 2600 nM T20251 CNOH63 57394711 IC50 > 100000 nM T20251 CRE41N 57394797 IC50 = 9400 nM T20251 CGV90O 57395178 IC50 = 3200 nM T20251 C9G6OJ 57395179 IC50 = 32000 nM T20251 CGR9F3 57395184 IC50 = 6500 nM T20251 CTG35L 57395190 IC50 > 30000 nM T20251 C3QCD9 57395216 IC50 > 30 nM T20251 C94MZO 57395217 IC50 > 30 nM T20251 CDIF34 57395218 IC50 > 30 nM T20251 C81ASJ 57395219 IC50 > 30 nM T20251 C5USX7 57395248 IC50 = 1600 nM T20251 CJ80BU 57395249 IC50 = 1800 nM T20251 CSO4Z0 57395278 IC50 = 1000 nM T20251 C01VOH 57395286 Ki = 2600 nM T20251 CB09IO 57395287 IC50 = 2300 nM T20251 C9CI3A 57395445 IC50 = 20000 nM T20251 CZ9G4Q 57395446 IC50 = 8700 nM T20251 C6SUR4 57395447 IC50 > 33000 nM T20251 C6VQ7I 57395454 Ki = 300 nM T20251 CFE6D4 57395455 Ki = 300 nM T20251 C0CGK5 57395838 IC50 = 3000 nM T20251 CHX4Z7 57396095 Ki = 19000 nM T20251 CRS39Y 57396096 Ki = 6400 nM T20251 CLEH95 57396097 Ki > 60000 nM T20251 C4NVE2 57396098 Ki = 12000 nM T20251 C7PT9Q 57396099 Ki = 22000 nM T20251 C23WQH 57396100 Ki = 7700 nM T20251 CTI36W 57396117 IC50 > 30000 nM T20251 C6HBG0 57396813 IC50 = 3300 nM T20251 CWU1I0 57396950 IC50 = 1200 nM T20251 CR41GU 57396951 IC50 > 32 nM T20251 C9YT0S 57396952 IC50 = 14000 nM T20251 CTH3P5 57396953 IC50 = 4000 nM T20251 C3L4ED 57396970 IC50 = 1000 nM T20251 CO37CB 57396999 IC50 > 30 nM T20251 C0P8KM 57397016 IC50 = 6700 nM T20251 CE85SV 57397017 IC50 = 4400 nM T20251 CYC1Q5 57397055 Ki > 3000 nM T20251 C25FTZ 57397056 IC50 = 900 nM T20251 C9W6IB 57397288 IC50 = 3600 nM T20251 CP0A2G 57397289 IC50 = 28000 nM T20251 CG8O2H 57397290 IC50 > 30000 nM T20251 CB7XV5 57397291 IC50 = 17000 nM T20251 C9WB0G 57397294 Ki = 1400 nM T20251 C7GJ6H 57397295 Ki = 1100 nM T20251 C7ML8N 57397296 Ki = 850 nM T20251 CLR02T 57397297 Ki = 8400 nM T20251 CEYO28 57397298 Ki = 710 nM T20251 CB20QV 57397299 Ki = 4400 nM T20251 CDQS63 57397589 IC50 = 25000 nM T20251 CNX73U 57397760 IC50 = 1100 nM T20251 CC8EV2 57397761 IC50 = 900 nM T20251 CH4Z3O 57397916 Ki = 7000 nM T20251 C9Y6KG 57397934 IC50 > 30000 nM T20251 CKDZ14 57398339 IC50 = 13598.78 nM T20251 CE5JQ8 57398341 IC50 = 128.82 nM T20251 C8Y4UJ 57398343 IC50 = 33113.11 nM T20251 CYO6T8 57398750 IC50 > 30 nM T20251 CSU2O9 57398779 IC50 = 1100 nM T20251 C5D0RB 57398829 Ki > 3000 nM T20251 CL4I6O 57398830 Ki > 3000 nM T20251 CSW1C3 57398976 IC50 = 9900 nM T20251 C0JIL8 57398977 IC50 = 13000 nM T20251 CH25BK 57398981 Ki = 1800 nM T20251 C4EY3H 57398982 Ki = 1400 nM T20251 CNY94K 57398983 Ki = 240 nM T20251 CG1D3L 57398984 Ki = 1100 nM T20251 C2J7GK 57398992 Ki = 360 nM T20251 CP8KQ7 57399426 IC50 = 12000 nM T20251 C4H6LZ 57399427 IC50 = 4700 nM T20251 CB42RN 57399556 Ki = 12000 nM T20251 CJO70A 57400003 IC50 = 129.99 nM T20251 CR09LY 57400127 IC50 = 5011.87 nM T20251 CK97BJ 57400372 IC50 = 25000 nM T20251 CA5KO3 57400374 IC50 = 25000 nM T20251 CDQ57A 57400458 IC50 = 1900 nM T20251 CED9C4 57400459 IC50 = 2000 nM T20251 CR0BU6 57400501 Ki > 3000 nM T20251 CE82XL 57400502 IC50 = 2100 nM T20251 CWZ50O 57400503 IC50 = 930 nM T20251 CJBU02 57400505 IC50 = 1500 nM T20251 CH13FG 57400694 IC50 = 11000 nM T20251 C6W1SD 57400695 IC50 = 7300 nM T20251 C9IXS8 57400698 Ki = 900 nM T20251 CS0E7F 57401040 IC50 = 113000 nM T20251 CCL98E 57401058 IC50 = 29500 nM T20251 CU2V1C 57401137 IC50 = 15000 nM T20251 CVXU49 57401184 IC50 = 3000 nM T20251 CUYK04 57401306 Ki = 24000 nM T20251 CSQK78 57401307 Ki = 9300 nM T20251 C8GC4D 57401308 Ki = 7600 nM T20251 CFL71K 57401309 Ki = 13000 nM T20251 CJQ89O 57401397 Ki = 2100 nM T20251 CKA34L 57401798 IC50 = 3090.3 nM T20251 CF0CA4 57401801 IC50 = 33113.11 nM T20251 C9X7PT 57401860 IC50 = 6 nM T20251 C3EV5S 57401884 IC50 = 25100 nM T20251 CG0DR6 57402003 IC50 = 330 nM T20251 C5NDS6 57402175 IC50 = 3200 nM T20251 C7CG1T 57402187 IC50 > 30000 nM T20251 CV54BI 57402219 IC50 = 13200 nM T20251 CV2ME6 57402260 IC50 = 5000 nM T20251 CQ1A8P 57402261 IC50 = 1300 nM T20251 CW94QA 57402262 IC50 = 1800 nM T20251 CMJA69 57402263 IC50 = 3400 nM T20251 C5X0LN 57402288 IC50 = 16000 nM T20251 C9D3ZE 57402314 Ki > 3000 nM T20251 CXT2L1 57402315 IC50 = 3400 nM T20251 CJ0E6V 57402465 IC50 = 11000 nM T20251 C6PM9O 57402466 IC50 > 33000 nM T20251 C1G3WE 57402816 IC50 = 63100 nM T20251 C2WT8S 57402817 IC50 = 4900 nM T20251 C65TPY 57403054 IC50 = 27000 nM T20251 CQ1ZV2 57403067 Ki = 11000 nM T20251 CHA41T 57403138 IC50 = 25000 nM T20251 CO94YE 57403139 IC50 = 18000 nM T20251 CX94UQ 57403171 IC50 = 80000 nM T20251 CC0D8X 57403932 IC50 = 35000 nM T20251 CX31VN 57403989 IC50 = 12000 nM T20251 C49JDH 57404030 Ki > 10000 nM T20251 C9SB1D 57404031 Ki > 3000 nM T20251 C1L8YD 57404359 IC50 = 8800 nM T20251 C8SX7A 57404360 IC50 = 6100 nM T20251 C6WU8O 57406717 IC50 = 15000 nM T20251 C0M6NB 57406720 IC50 = 2700 nM T20251 CWCY97 57406911 IC50 > 33000 nM T20251 C5CRJ1 57412107 IC50 = 2380 nM T20251 CUSO25 57414544 IC50 = 62 nM T20251 C8UMR2 57414545 IC50 = 580 nM T20251 CSA3P9 57414546 IC50 = 39.81 nM T20251 CI2TO3 57414547 IC50 = 2.512 nM T20251 CA8K1N 57414548 IC50 = 7860 nM T20251 CX6N9E 57414549 IC50 = 192 nM T20251 C1CUJ7 57441855 IC50 = 4000 nM T20251 CF9Z3R 57441946 IC50 > 32000 nM T20251 CRV53F 57441994 IC50 > 32000 nM T20251 C47QNO 57442001 IC50 = 13200 nM T20251 CR58EY 57442010 IC50 > 32000 nM T20251 C54JSK 57448273 IC50 > 10000 nM T20251 CVNR58 57448274 IC50 = 2500 nM T20251 C5CBG4 57448276 IC50 = 2800 nM T20251 CUWK92 57448281 IC50 > 10000 nM T20251 CY86DR 57448284 IC50 = 8900 nM T20251 C74GKR 57448289 IC50 > 10000 nM T20251 CAE6B5 57448332 IC50 > 10000 nM T20251 CK9TD7 57448346 IC50 > 10000 nM T20251 CA6YR3 57448356 IC50 > 10000 nM T20251 C0I1CB 57448358 IC50 > 10000 nM T20251 CWA9F6 57482815 IC50 = 63095.73 nM T20251 C2QS1Y 57504248 IC50 = 50118.72 nM T20251 CMB2W7 57504266 IC50 = 19952.62 nM T20251 CAY71X 57504268 IC50 > 33000 nM T20251 CBU6N2 57504311 IC50 > 100000 nM T20251 C6S8CV 57504312 IC50 > 79432.82 nM T20251 C0W5QD 57504313 IC50 > 100000 nM T20251 CD85MW 57504320 IC50 = 31622.78 nM T20251 CH79YV 57504325 IC50 = 79432.82 nM T20251 CZ8SF5 57504326 IC50 = 63095.73 nM T20251 CRC5O1 57504327 IC50 = 15848.93 nM T20251 C7JDH2 57504328 IC50 = 50118.72 nM T20251 CM8Z6N 57504345 IC50 = 25118.86 nM T20251 CKE12J 57504346 IC50 = 12589.25 nM T20251 C4UAZ5 57504347 IC50 = 15848.93 nM T20251 CH3Y9K 57504348 IC50 = 63095.73 nM T20251 C9TY4W 57504354 IC50 = 19952.62 nM T20251 CCT08G 57504355 IC50 = 63095.73 nM T20251 C0OIW2 57504356 IC50 > 100000 nM T20251 CPQA09 57504358 IC50 = 10000 nM T20251 CP7BL3 57504360 IC50 = 63095.73 nM T20251 CV20RS 57504361 IC50 = 50118.72 nM T20251 C42OWY 57504362 IC50 > 100000 nM T20251 C8K7TB 57504363 IC50 = 79432.82 nM T20251 CPR02A 57504388 IC50 = 50118.72 nM T20251 CI74AT 57504389 IC50 = 50118.72 nM T20251 COB73U 57504402 IC50 = 15848.93 nM T20251 CLWU10 57504418 IC50 = 63095.73 nM T20251 C8UHW1 57504419 IC50 > 100000 nM T20251 C0BGQ4 57504420 IC50 > 100000 nM T20251 C38YSV 57504421 IC50 > 100000 nM T20251 C1CPF8 57504444 IC50 = 79432.82 nM T20251 CB54GY 57504445 IC50 = 10000 nM T20251 CYHT79 57504446 IC50 = 7943.28 nM T20251 CAV2N7 57504447 IC50 > 100000 nM T20251 C3AOX7 57504450 IC50 = 25118.86 nM T20251 CR0HE5 57504454 IC50 = 6309.57 nM T20251 CV8B0T 57504457 IC50 = 63095.73 nM T20251 CRLJ46 57504462 IC50 > 100000 nM T20251 CNEB25 57504463 IC50 = 31622.78 nM T20251 CR1A8Z 57504467 IC50 = 39810.72 nM T20251 C90OLN 57504474 IC50 = 26000 nM T20251 CB47MQ 57514846 IC50 > 10000 nM T20251 C7I4QD 57519510 IC50 > 30000 nM T20251 C3N4MF 57520842 IC50 > 30000 nM T20251 CEL56T 57520942 IC50 > 30000 nM T20251 C7PLG5 57521314 IC50 = 49800 nM T20251 CWE9J4 57522010 IC50 > 30000 nM T20251 C3I5XK 57522013 IC50 = 21900 nM T20251 C53BGU 57522014 IC50 > 30000 nM T20251 CHU5T7 57523687 IC50 = 27000 nM T20251 C5P3HT 57545640 Ki = 2314 nM T20251 CR34CL 57582353 IC50 > 30000 nM T20251 C7D1JL 57606048 IC50 = 105000 nM T20251 C9I6RO 57606050 IC50 > 33000 nM T20251 C6D3MG 57606067 IC50 > 33000 nM T20251 C3OQ4Z 57606068 IC50 > 33000 nM T20251 CYEQ10 57606070 IC50 > 33000 nM T20251 CY59ML 57606091 IC50 > 33000 nM T20251 C1F2DJ 57606095 IC50 > 33000 nM T20251 CI59LU 57609886 Ki = 498 nM T20251 C6GCQ8 57611057 IC50 = 9100 nM T20251 CYV5K2 57639150 IC50 = 38100 nM T20251 CM32RA 57656640 IC50 = 7100 nM T20251 C0OJA5 57656641 IC50 = 6300 nM T20251 CT8V9X 57656657 IC50 = 890 nM T20251 CH7BO0 57656701 IC50 = 13000 nM T20251 CMI4T3 57656713 IC50 = 400 nM T20251 CB30PQ 57656715 IC50 = 2000 nM T20251 C51DOT 57656719 IC50 = 6300 nM T20251 C2GHC7 57656729 IC50 = 5000 nM T20251 C6W3EJ 57656749 IC50 = 6300 nM T20251 C1KAC6 57656808 IC50 = 8900 nM T20251 CN7O1T 57656825 IC50 = 14000 nM T20251 CHJ87A 57656833 IC50 = 60000 nM T20251 CS6O1V 57656854 IC50 = 19000 nM T20251 CPN5S4 57656869 IC50 = 16000 nM T20251 CU8I2F 57656871 IC50 = 10000 nM T20251 CD5W4E 57656887 IC50 = 28000 nM T20251 CQX1D5 57656921 IC50 = 7100 nM T20251 C1QSF4 57656938 IC50 = 13000 nM T20251 C5V0JI 57656942 IC50 = 14000 nM T20251 CJYS25 57663369 IC50 = 7943.28 nM T20251 C4QG8R 57663382 IC50 = 6309.57 nM T20251 CHQI67 57663405 IC50 > 63095.73 nM T20251 CA9RK8 57663418 IC50 = 7943.28 nM T20251 CM7H9G 57663419 IC50 = 19952.62 nM T20251 C58ERT 57663421 IC50 = 15848.93 nM T20251 CY2S7K 57663434 IC50 = 1995.26 nM T20251 C9A0XM 57663447 IC50 = 25118.86 nM T20251 C18FHN 57663450 IC50 = 12589.25 nM T20251 CPSX03 57663451 IC50 = 7943.28 nM T20251 CMUD63 57663495 IC50 = 12589.25 nM T20251 CVL35Z 57663496 IC50 = 19952.62 nM T20251 CBK0Y1 57663581 IC50 = 63095.73 nM T20251 CSK82C 57663586 IC50 = 15848.93 nM T20251 C5J1QT 57663596 IC50 = 29512.09 nM T20251 CTV29J 57663598 IC50 = 19952.62 nM T20251 C2X7OT 57663610 IC50 = 12589.25 nM T20251 C98CVM 57663630 IC50 = 15848.93 nM T20251 CGA1V2 57663637 IC50 > 63095.73 nM T20251 CV2J9A 57663655 IC50 = 18620.87 nM T20251 CR7S5U 57663666 IC50 = 19952.62 nM T20251 C4GXF1 57663688 IC50 = 12589.25 nM T20251 CZ2UB5 57705473 IC50 > 10000 nM T20251 C35GXV 57720515 EC50 = 6000 nM T20251 CQP7E0 57750290 IC50 = 21030 nM T20251 C1U3YR 57750299 IC50 > 33300 nM T20251 CEY8W0 57750311 IC50 > 33300 nM T20251 CNBO65 57750312 IC50 = 80124 nM T20251 C2F9DS 57750315 IC50 > 100000 nM T20251 CZ08KN 57750321 IC50 > 100000 nM T20251 CUY8T6 57750329 IC50 > 33300 nM T20251 CK4W1L 57750342 IC50 > 33300 nM T20251 CM5X9L 57750343 IC50 = 9092 nM T20251 C0TNP8 57750364 IC50 > 33300 nM T20251 CBY5E4 57750369 IC50 = 74807 nM T20251 CO6P5G 57750381 IC50 > 33300 nM T20251 CSI9Y4 57750382 IC50 = 1600 nM T20251 C6GH7X 57750391 IC50 = 3500 nM T20251 CL7CW0 57750402 IC50 = 9369 nM T20251 CA4G5W 57750407 IC50 = 29367 nM T20251 CM7XL6 57750408 IC50 = 6747 nM T20251 CY4Z8R 57750418 IC50 = 26957 nM T20251 C8OY4I 57750420 IC50 > 33300 nM T20251 CT89JH 57780007 IC50 = 50118.72 nM T20251 CT8RO7 57780008 IC50 = 7943.28 nM T20251 C5RIN4 57780016 IC50 > 63095.73 nM T20251 CE9WC0 57780017 IC50 = 15848.93 nM T20251 C1W4SB 57780018 IC50 = 31622.78 nM T20251 CT96WD 57780020 IC50 = 2511.89 nM T20251 C9FH4B 57790981 IC50 = 5500 nM T20251 CG16CV 57916503 IC50 > 100000 nM T20251 C8E6PG 57927934 IC50 > 33000 nM T20251 C10VYA 57948490 IC50 > 30000 nM T20251 CAU57Q 57969602 IC50 = 3000 nM T20251 C1LZI4 57969746 IC50 > 10000 nM T20251 CXI6A1 57970302 IC50 = 1000 nM T20251 C67MSZ 58017509 IC50 = 14000 nM T20251 CG9V4E 58017514 IC50 = 15000 nM T20251 CN6Z0X 58017523 IC50 = 5600 nM T20251 C7M3DS 58017531 IC50 > 33000 nM T20251 C1EP6I 58024825 IC50 > 29000 nM T20251 C19XQV 58026164 IC50 = 20000 nM T20251 CEWR70 58065681 IC50 = 5200 nM T20251 C9JCL7 58080768 IC50 = 4900 nM T20251 C5B0RJ 58083331 Ki = 33600 nM T20251 C1C6OS 58083336 Ki = 31200 nM T20251 C6DZ0X 58083358 Ki = 23000 nM T20251 CND4G1 58088117 IC50 = 2500 nM T20251 C2EY8P 58109378 IC50 = 5300 nM T20251 CJ07OW 58109450 IC50 = 6300 nM T20251 C4FH0W 58118983 IC50 > 10000 nM T20251 C46AUK 58137055 IC50 > 32000 nM T20251 C7ONC3 58137106 IC50 > 33000 nM T20251 CRPL37 58137176 IC50 > 32000 nM T20251 C2R3IZ 58178960 IC50 = 7200 nM T20251 C1TL8P 58179284 IC50 > 30000 nM T20251 C7AY1J 58190324 IC50 = 11000 nM T20251 CI63UA 58190330 IC50 > 30000 nM T20251 CPQ0Z4 58269588 IC50 > 30000 nM T20251 CD18IU 58269609 IC50 > 30000 nM T20251 C8ILS3 58269629 IC50 = 27000 nM T20251 C5VFQ7 58269655 IC50 = 4000 nM T20251 C2PYB1 58269668 IC50 > 30000 nM T20251 C3CFB8 58269691 IC50 > 30000 nM T20251 CTWG72 58290872 IC50 = 24500 nM T20251 CJ4B6P 58299601 IC50 = 2000 nM T20251 CT78UE 58299836 IC50 = 720 nM T20251 CB3IT1 58302173 Ki > 30000 nM T20251 CW1G9J 58302348 Ki = 740 nM T20251 C0F3BO 58394783 IC50 > 100000 nM T20251 C0X7IK 58394837 IC50 > 100000 nM T20251 CASI81 58395078 IC50 > 100000 nM T20251 CWBM72 58395283 IC50 = 20000 nM T20251 CZ2VK4 58408526 Ki = 8820 nM T20251 CE80UP 58438175 IC50 > 30000 nM T20251 C5DC7T 58438322 IC50 = 1300 nM T20251 C9UK7P 58438475 IC50 = 2900 nM T20251 CC8TK0 58466119 Ki > 10000 nM T20251 C9IRW0 58466120 Ki > 15000 nM T20251 CSU91B 58466122 Ki > 15000 nM T20251 CKSF73 58466243 Ki = 1240 nM T20251 CH9ER4 58466295 Ki = 6900 nM T20251 C6QJX4 58466300 Ki > 10000 nM T20251 C6OJC2 58466301 Ki = 496 nM T20251 CBN9L0 58561169 IC50 = 600 nM T20251 CIJ09G 58576126 IC50 = 58 nM T20251 C4VT6Z 58615686 IC50 = 3180 nM T20251 C6JKM0 58834906 IC50 = 9900 nM T20251 CF9Z0L 58834953 IC50 = 18000 nM T20251 C4PWA9 58835024 IC50 > 30000 nM T20251 CCR4T7 58835217 IC50 > 30000 nM T20251 C9ZE7J 58874273 IC50 > 10000 nM T20251 CCNI49 58920310 IC50 = 22000 nM T20251 CXGW57 58920485 IC50 > 80000 nM T20251 CETS76 59019389 IC50 > 16000 nM T20251 CJS46Y 59086459 IC50 = 7300 nM T20251 CO6TL1 59135478 IC50 = 420 nM T20251 C31KUT 59149763 IC50 = 11220.18 nM T20251 CH41MU 59149828 IC50 > 100000 nM T20251 CCQM76 59153288 IC50 > 30000 nM T20251 C0Z5IL 59173801 IC50 = 3080 nM T20251 CWJT87 59174010 IC50 = 1290 nM T20251 C3L4JY 59176329 IC50 = 3900 nM T20251 CW24YS 59190451 IC50 = 6309.57 nM T20251 CEI8A5 59190544 IC50 = 19952.62 nM T20251 CY54RB 59199467 IC50 = 4800 nM T20251 C94HKZ 59199478 IC50 = 1700 nM T20251 CMSR93 59199482 IC50 = 6300 nM T20251 C30VAF 59199488 IC50 = 3500 nM T20251 CNUT13 59218182 IC50 > 10000 nM T20251 CHVU94 59218184 IC50 > 10000 nM T20251 CY6EB4 59218190 IC50 > 10000 nM T20251 C2PJ4N 59271992 IC50 = 13000 nM T20251 C7XM1P 59272333 Ki > 15000 nM T20251 CWCK45 59272335 Ki = 14000 nM T20251 C9VNB7 59275242 IC50 = 5800 nM T20251 CTF1U6 59275404 IC50 = 18000 nM T20251 C4KU2S 59278286 IC50 > 30000 nM T20251 CEAY32 59278314 IC50 = 30000 nM T20251 CN1Y9X 59279548 IC50 = 39810.72 nM T20251 CC1AN4 59279550 IC50 = 12589.25 nM T20251 CM4XB0 59279551 IC50 = 39810.72 nM T20251 CBWJ84 59291203 IC50 > 33000 nM T20251 CPWM60 59291925 IC50 > 100000 nM T20251 CE6KO4 59291951 IC50 > 100000 nM T20251 CT3EW2 59292007 IC50 > 100000 nM T20251 C2PE0T 59292008 IC50 > 100000 nM T20251 C90EAP 59295914 IC50 = 3162.28 nM T20251 CFX9H8 59295925 IC50 = 6309.57 nM T20251 C5P6UI 59295926 IC50 = 6309.57 nM T20251 C18YQX 59295928 IC50 > 31622.78 nM T20251 C9NMZ2 59295931 IC50 = 251.19 nM T20251 CA8T3Q 59295938 IC50 = 5011.87 nM T20251 C59QBR 59295939 IC50 = 1995.26 nM T20251 COG4S6 59295946 IC50 = 5011.87 nM T20251 CHP65R 59295958 IC50 = 1258.93 nM T20251 C3PCY5 59295968 IC50 > 31622.78 nM T20251 CYG56K 59295969 IC50 = 794.33 nM T20251 C4PYU5 59295974 IC50 > 31622.78 nM T20251 CRZN12 59295978 IC50 = 1995.26 nM T20251 CR2T5D 59295982 IC50 > 6309.57 nM T20251 C17USX 59295994 IC50 > 10000 nM T20251 CJV58T 59296000 IC50 = 501.19 nM T20251 C2K1TV 59296010 IC50 = 398.11 nM T20251 C0KM5W 59296024 IC50 > 31622.78 nM T20251 CE73NG 59296033 IC50 = 1000 nM T20251 CT2P4Z 59296039 IC50 = 251.19 nM T20251 CXK7O5 59296048 IC50 = 1995.26 nM T20251 CPE0B2 59296066 IC50 = 10000 nM T20251 CFR8S7 59296077 IC50 = 1995.26 nM T20251 CMD56H 59296081 IC50 = 1000 nM T20251 CFCE90 59296090 IC50 = 5011.87 nM T20251 CUC57E 59296099 IC50 = 1995.26 nM T20251 C1ZN0M 59296100 IC50 = 1258.93 nM T20251 CX6JS1 59296104 IC50 = 1995.26 nM T20251 C5TMB2 59296111 IC50 = 3162.28 nM T20251 C6E5UG 59366166 Ki < 13 nM T20251 CSF3A7 59394005 IC50 = 7000 nM T20251 CP34RY 59394193 IC50 > 30000 nM T20251 C5IQ4P 59394335 IC50 = 23500 nM T20251 CY9RB5 59394429 IC50 = 15600 nM T20251 CHXC24 59394467 IC50 = 11100 nM T20251 C7A5KZ 59394725 IC50 = 7400 nM T20251 CK4Y8T 59395224 IC50 > 33000 nM T20251 CDA17U 59396249 IC50 = 46100 nM T20251 C80HTM 59396252 IC50 = 78600 nM T20251 CE01DO 59396594 IC50 = 76000 nM T20251 C6IDV0 59396641 IC50 = 50100 nM T20251 CQK9S3 59401826 IC50 = 1000 nM T20251 C53BVH 59401876 IC50 = 480 nM T20251 CNOI48 59401886 IC50 = 1800 nM T20251 C29YCJ 59411406 IC50 = 27100 nM T20251 C03EFU 59440893 IC50 > 30000 nM T20251 CPUZ69 59447115 IC50 > 10000 nM T20251 CK6LX0 59454220 IC50 = 7000 nM T20251 C2SDN1 59454252 IC50 = 5000 nM T20251 C46UHJ 59458228 IC50 = 33000 nM T20251 CSOL31 59458454 IC50 > 80000 nM T20251 C0L2FW 59458459 IC50 = 44000 nM T20251 C83DOJ 59458460 IC50 = 11000 nM T20251 C0ZLU4 59458594 IC50 = 23000 nM T20251 CZ0Q7W 59458647 IC50 > 80000 nM T20251 CV41DL 59458714 IC50 > 80000 nM T20251 C6K0MO 59458732 IC50 = 21000 nM T20251 CFP75N 59458738 IC50 = 16000 nM T20251 CJ5I3Q 59459021 IC50 = 25600 nM T20251 C9XI4D 59459390 IC50 = 63000 nM T20251 CTH04J 59459492 IC50 = 12000 nM T20251 C1E3XT 59472470 EC50 = 15000 nM T20251 C92NPY 59472493 IC50 = 18100 nM T20251 CL4F1U 59472507 IC50 = 800 nM T20251 CG1ZH6 59472511 IC50 = 1580 nM T20251 CHU2S4 59472516 IC50 = 1390 nM T20251 CW4I0H 59472517 IC50 = 2680 nM T20251 C4RZ7E 59472522 IC50 = 17600 nM T20251 CKS31U 59472524 IC50 = 8740 nM T20251 C35EKB 59472530 IC50 = 530 nM T20251 CLB40A 59472544 EC50 = 1300 nM T20251 CL9Y0P 59472546 IC50 = 4030 nM T20251 CXH19J 59472574 IC50 = 2610 nM T20251 C51KUS 59472588 IC50 = 3560 nM T20251 CS87XI 59472603 IC50 = 8960 nM T20251 CI8H4T 59472630 IC50 = 3050 nM T20251 CXO21N 59472637 IC50 = 20800 nM T20251 CH0S6A 59472641 IC50 = 4060 nM T20251 C0LBN5 59472644 IC50 > 10000 nM T20251 C4SR9V 59472646 IC50 > 30000 nM T20251 C6D7LS 59472679 IC50 = 3680 nM T20251 C8UMR6 59472684 IC50 = 1830 nM T20251 C1ME7D 59472698 IC50 = 1010 nM T20251 CYO06N 59472699 IC50 = 870 nM T20251 C6XDH2 59472707 IC50 = 800 nM T20251 CF72WU 59472713 IC50 = 3220 nM T20251 C9L0GJ 59472717 IC50 = 43900 nM T20251 CJR3K7 59472756 IC50 = 1490 nM T20251 C1RUN6 59472765 Ki = 3600 nM T20251 CZ52KP 59472771 IC50 = 10300 nM T20251 CB3X0F 59472773 IC50 = 7570 nM T20251 C6YZR8 59472775 IC50 = 44200 nM T20251 CDOV85 59472789 IC50 > 30000 nM T20251 CWD0K3 59472815 IC50 = 2870 nM T20251 C15JGP 59472849 IC50 = 6220 nM T20251 CM0G7S 59472858 IC50 > 50000 nM T20251 CEP94I 59472861 IC50 = 630 nM T20251 CLH47W 59472872 IC50 = 2220 nM T20251 C2SNL8 59541239 IC50 = 12000 nM T20251 CA9NE4 59548712 IC50 = 8000 nM T20251 CG2V1M 59568650 IC50 = 14000 nM T20251 C7FAN1 59568652 IC50 = 18000 nM T20251 CM1G2P 59568656 IC50 = 33000 nM T20251 CS19JW 59568702 IC50 = 22000 nM T20251 C4W8RH 59651989 IC50 > 30000 nM T20251 CIL17E 59652016 IC50 = 18000 nM T20251 CF8E1J 59764390 IC50 = 400 nM T20251 CC48EN 59764418 IC50 = 5300 nM T20251 C4NBG7 59764433 IC50 = 3020 nM T20251 C40UZT 59764460 IC50 = 2640 nM T20251 C6AQX8 59764524 IC50 = 3350 nM T20251 CJ7E6C 60026483 IC50 = 3800 nM T20251 C45XVN 60142198 Ki = 1980 nM T20251 CJ5M9S 60142200 Ki = 1740 nM T20251 C79ZOY 60142335 Ki = 4800 nM T20251 CNKF60 60143411 IC50 = 27600 nM T20251 CYCN68 60143412 IC50 > 100000 nM T20251 CJP6A3 60143413 IC50 > 100000 nM T20251 CX9PB5 60143414 IC50 > 100000 nM T20251 CGJ5H3 60143415 IC50 > 100000 nM T20251 C7TC5K 60143416 IC50 > 100000 nM T20251 CRFV62 60143588 IC50 > 100000 nM T20251 C7S4PH 60143589 IC50 > 100000 nM T20251 C9EH3R 60143590 IC50 = 78700 nM T20251 CZ3QD9 60143591 IC50 > 100000 nM T20251 CM62NL 60143592 IC50 > 100000 nM T20251 C9ME8V 60143757 IC50 > 100000 nM T20251 CFH4L9 60143758 IC50 > 100000 nM T20251 C4R6PH 60143759 IC50 = 49100 nM T20251 CVA2X8 60143760 IC50 > 100000 nM T20251 CD65CK 60143761 IC50 > 100000 nM T20251 C4TES3 60143762 IC50 > 100000 nM T20251 CR1ZN4 60143921 IC50 > 100000 nM T20251 CD5T7O 60143922 IC50 > 100000 nM T20251 C5DJA6 60143923 IC50 > 100000 nM T20251 CPF6A9 60143924 IC50 > 100000 nM T20251 CRTN28 60143925 IC50 > 100000 nM T20251 CYJ19Q 60143926 IC50 > 100000 nM T20251 C8UQ7D 60144084 IC50 > 100000 nM T20251 CM0C9O 60144086 IC50 > 100000 nM T20251 CN4A8W 60144088 IC50 > 100000 nM T20251 CJ4XM3 60144089 IC50 > 100000 nM T20251 CY4H9Z 60144244 IC50 > 100000 nM T20251 CMQ78O 60144245 IC50 > 100000 nM T20251 CAPO85 60145490 IC50 = 76500 nM T20251 C4KZ3M 60145492 IC50 > 100000 nM T20251 CBP2K4 60145493 IC50 = 13600 nM T20251 C0B7QX 60145494 IC50 = 18800 nM T20251 CDK1O7 60145629 IC50 > 100000 nM T20251 COR56Z 60145630 IC50 > 100000 nM T20251 C03HNY 60145631 IC50 > 100000 nM T20251 C6CE5G 60145632 IC50 > 100000 nM T20251 CJSV45 60145633 IC50 > 100000 nM T20251 CB4ND5 60145634 IC50 = 26100 nM T20251 C0FR9I 60145771 IC50 > 100000 nM T20251 C8S4EL 60145772 IC50 > 100000 nM T20251 CE17ZH 60145773 IC50 > 100000 nM T20251 CHJ03O 60145774 IC50 > 100000 nM T20251 C40GSO 60145775 IC50 > 100000 nM T20251 CQW7A8 60149247 IC50 = 9000 nM T20251 CGF54X 60150483 IC50 = 5600 nM T20251 C3HZ5J 60150507 IC50 = 2500 nM T20251 C30UIB 60150707 IC50 = 5400 nM T20251 CTL97W 60151476 IC50 > 10000 nM T20251 C3D2ZI 60155056 IC50 > 24000 nM T20251 CA4OH9 60155057 IC50 > 23400 nM T20251 CR36EQ 60155058 IC50 > 22700 nM T20251 CT7ID2 60162269 IC50 = 8240 nM T20251 C2D3HQ 60168069 IC50 = 73600 nM T20251 CSN5C8 60170856 IC50 > 10000 nM T20251 CPLU74 60170970 IC50 = 9700 nM T20251 C6U0HA 60194465 IC50 = 14500 nM T20251 CYH8P0 60199250 IC50 > 30000 nM T20251 C4VZ5L 60199310 IC50 = 23990 nM T20251 CSPU20 60199433 IC50 > 30000 nM T20251 CEKA47 60199634 IC50 = 15000 nM T20251 CC8YH1 60199796 IC50 = 75000 nM T20251 C2TY3G 60199965 IC50 = 168000 nM T20251 CR4IL3 60199967 IC50 = 25000 nM T20251 CPK52S 60200126 IC50 = 32000 nM T20251 C29HIU 60200128 IC50 > 333000 nM T20251 COJ18I 60200280 IC50 = 152000 nM T20251 CO5HD0 60201085 IC50 = 5300 nM T20251 CA57OQ 60201086 IC50 = 4900 nM T20251 C5UKQ8 60201087 IC50 = 11000 nM T20251 CA7NI3 60201088 IC50 = 24000 nM T20251 C1YQ8J 60201256 IC50 > 33000 nM T20251 CM92ST 60201265 IC50 = 189000 nM T20251 C5WQ3Z 60201425 IC50 = 88000 nM T20251 CN18KX 60201945 IC50 = 199000 nM T20251 CJ23UN 60201946 IC50 = 57000 nM T20251 C6Z2HF 60201948 IC50 = 75000 nM T20251 C2D0TI 60202105 IC50 = 156000 nM T20251 CK3G6T 60202107 IC50 = 117000 nM T20251 CY04QB 60210882 IC50 > 10000 nM T20251 CL42CH 60509567 IC50 = 0.76 nM T20251 CW3H0V 60634975 IC50 > 25000 nM T20251 C4BZ2N 60637368 IC50 < 10000 nM T20251 CI7DY2 60965486 IC50 > 10000 nM T20251 C02TAQ 62705172 IC50 > 50000 nM T20251 CV0X4K 62705173 IC50 > 50000 nM T20251 CG2VD0 62705174 IC50 > 50000 nM T20251 CWL9J4 62705175 IC50 = 6300 nM T20251 CQ5LS1 62705176 IC50 = 6600 nM T20251 CK2DG6 62705177 IC50 = 9300 nM T20251 CX7Q2A 62705299 IC50 > 10000 nM T20251 C59QUB 62705330 IC50 = 13000 nM T20251 CANL67 62705331 IC50 > 50000 nM T20251 CW19CI 62705332 IC50 = 46000 nM T20251 CK2WS1 62705333 IC50 = 22000 nM T20251 C1SNE7 62705334 IC50 = 5300 nM T20251 C2O6FQ 62705335 IC50 = 3400 nM T20251 CTM29C 62705504 IC50 = 5700 nM T20251 CZHO61 62705505 IC50 = 7900 nM T20251 CT41VY 62705506 IC50 = 6300 nM T20251 CP9HO0 62705507 IC50 = 4400 nM T20251 CSHR51 62705508 IC50 = 1900 nM T20251 CVPW40 62705509 IC50 = 3400 nM T20251 CA4RU3 62706110 IC50 = 1600 nM T20251 CM0Z3B 62707610 IC50 = 7300 nM T20251 CZDW91 65458453 IC50 > 16000 nM T20251 C9SEG5 65458673 IC50 > 16000 nM T20251 CC82DM 65459349 IC50 = 1800 nM T20251 C0JSU4 65459575 IC50 > 16000 nM T20251 CVUT64 66549717 IC50 = 4080 nM T20251 C1MDS9 66549721 IC50 = 13970 nM T20251 C6EJ3F 66551245 IC50 = 25118.86 nM T20251 CBI4P9 66551368 IC50 = 290 nM T20251 C3SCF6 66551759 IC50 = 870 nM T20251 C2LBW7 66551925 IC50 > 30000 nM T20251 CLHX28 66553128 IC50 = 27000 nM T20251 CA42UL 66554658 IC50 = 15848.93 nM T20251 CX25QN 66555696 IC50 > 50118.72 nM T20251 CL0X8S 66555697 IC50 > 50118.72 nM T20251 C2Y7FX 66555698 IC50 = 25118.86 nM T20251 C8PST7 66556032 IC50 = 10000 nM T20251 CV8JO4 66556033 IC50 > 50118.72 nM T20251 CSZ6I5 66556035 IC50 > 50118.72 nM T20251 C6SL1Q 66556036 IC50 > 50118.72 nM T20251 CX6J3B 66556201 IC50 = 25118.86 nM T20251 CHWG72 66556203 IC50 = 39810.72 nM T20251 CVPT78 66556206 IC50 = 50118.72 nM T20251 C0F5HW 66556207 IC50 > 50118.72 nM T20251 C6E7CU 66556365 IC50 = 12589.25 nM T20251 CR7JT9 66556366 IC50 = 31622.78 nM T20251 CSM89V 66556371 IC50 = 5011.87 nM T20251 CK9QI1 66556533 IC50 = 19952.62 nM T20251 CA1Z4Q 66556534 IC50 > 50118.72 nM T20251 CNRZ13 66556535 IC50 > 50118.72 nM T20251 C7MD5X 66556536 IC50 = 15848.93 nM T20251 CL3EN2 66556938 IC50 > 10000 nM T20251 CUC7B3 66557964 IC50 = 45000 nM T20251 C85RBC 66559553 IC50 = 1900 nM T20251 C95GNE 66559554 IC50 = 2700 nM T20251 CKW13M 66559641 IC50 = 4300 nM T20251 CP1BI4 66559642 IC50 = 30000 nM T20251 C3MW0K 66559643 IC50 = 1100 nM T20251 C0TL3Y 66559644 IC50 > 30000 nM T20251 CXS5D6 66590299 Ki = 9520 nM T20251 CHO3M7 66597981 IC50 > 30000 nM T20251 C7W2XF 66597997 IC50 > 30000 nM T20251 C52HRW 66598095 IC50 > 30000 nM T20251 C1ET4P 66598128 IC50 = 1900 nM T20251 C5D3TJ 66598153 IC50 > 30000 nM T20251 CZF76R 66608383 IC50 > 10000 nM T20251 CECR98 66615606 IC50 = 15848.93 nM T20251 C9IQ1Y 66615619 IC50 > 31622.78 nM T20251 CA59FS 66615678 IC50 > 31622.78 nM T20251 CL69HQ 66615705 IC50 > 31622.78 nM T20251 CLA3R9 66645269 IC50 > 33000 nM T20251 COTD35 66667669 Ki > 30000 nM T20251 CXSA80 66671848 IC50 > 10000 nM T20251 CZKV14 66679405 IC50 = 2000 nM T20251 CJ0KL5 66679507 IC50 > 10000 nM T20251 C9RS5B 66679618 IC50 = 1800 nM T20251 CUC7E1 66679703 IC50 > 10000 nM T20251 C4TQP9 66688557 IC50 = 12200 nM T20251 C3FG4T 66688815 IC50 = 10300 nM T20251 CKR1D0 66693299 IC50 = 24900 nM T20251 C9BF6L 66797369 IC50 = 72000 nM T20251 C78XLS 66813470 IC50 = 10000 nM T20251 CAOB97 66813557 IC50 = 6309.57 nM T20251 C89WUE 66813671 IC50 = 12589.25 nM T20251 CPK67V 66813703 IC50 = 3981.07 nM T20251 C7DX6Z 66813839 IC50 = 6309.57 nM T20251 CH2D5F 66813859 IC50 = 25118.86 nM T20251 C90OSR 66813870 IC50 = 15848.93 nM T20251 COZ0U9 66813914 IC50 = 7943.28 nM T20251 C5OTD2 66813927 IC50 = 10000 nM T20251 C39PEZ 66814019 IC50 = 25118.86 nM T20251 CG80RS 66814110 IC50 = 15848.93 nM T20251 C5BU7L 66829310 IC50 > 30000 nM T20251 CPZQ50 66829372 IC50 = 1900 nM T20251 C38BYQ 66829396 IC50 > 30000 nM T20251 CEVJ65 66829417 IC50 > 30000 nM T20251 CBE2J9 66829485 IC50 = 12000 nM T20251 CRI63W 66829595 IC50 = 12700 nM T20251 CD1BQ8 66829616 IC50 > 30000 nM T20251 C8OZR1 66829709 IC50 > 30000 nM T20251 CEQ7A6 66829716 IC50 = 2560 nM T20251 CMAD65 66829757 IC50 = 10200 nM T20251 C95TOQ 66855889 IC50 = 794 nM T20251 C85HLV 67011331 IC50 > 30000 nM T20251 C1HSE0 67035086 IC50 = 420 nM T20251 CWI6K5 67035106 IC50 = 1100 nM T20251 C38RGB 67035556 IC50 = 3600 nM T20251 CFM6H7 67049587 IC50 > 100000 nM T20251 CJMU80 67055888 IC50 > 80000 nM T20251 C3VFY7 67104025 IC50 = 19000 nM T20251 CV6Z2X 67204288 IC50 > 10000 nM T20251 CD3C7S 67204380 IC50 = 29000 nM T20251 C7CDA0 67220645 IC50 = 20000 nM T20251 C7V8QD 67251061 IC50 = 20 nM T20251 C3WJ5C 67260498 IC50 > 10000 nM T20251 CKQ9W2 67264691 IC50 = 7620 nM T20251 C3F2JN 67264841 IC50 = 2230 nM T20251 C38ROH 67264950 IC50 = 22100 nM T20251 C3CAR6 67265132 IC50 > 30000 nM T20251 C3Q6ZA 67282848 IC50 = 2200 nM T20251 C4R1IH 67283149 IC50 > 10000 nM T20251 C9LI0M 67294297 IC50 > 30000 nM T20251 CBK9T7 67325548 IC50 = 2100 nM T20251 C2NEB3 67339181 IC50 = 10715.19 nM T20251 CKMV48 67345882 IC50 > 100000 nM T20251 CO3ND7 67387844 Ki > 15000 nM T20251 C36MVU 67389741 IC50 = 16000 nM T20251 C4R8OG 67401728 IC50 = 1100 nM T20251 CPV39L 67406727 IC50 = 47000 nM T20251 C7XU0T 67425014 IC50 > 10000 nM T20251 CBFE84 67436561 Ki > 15000 nM T20251 CZC9M5 67469084 IC50 = 7445 nM T20251 CX60UI 67472601 IC50 = 27500 nM T20251 C37YHJ 67496729 IC50 > 30000 nM T20251 CL9JR7 67516635 IC50 = 1300 nM T20251 CIB4Y6 67516958 IC50 = 7100 nM T20251 COH79P 67517411 IC50 = 150 nM T20251 C0WAQ6 67517817 IC50 = 3000 nM T20251 C02TCR 67518221 IC50 = 420 nM T20251 CF3GR9 67538211 IC50 = 26000 nM T20251 CNB15W 67607112 IC50 > 10000 nM T20251 COM54X 67775149 IC50 = 8500 nM T20251 C32GEY 67922794 IC50 > 10000 nM T20251 CY3AZ9 67960061 IC50 = 3700 nM T20251 C3ARI1 67972106 IC50 = 46000 nM T20251 CXJ68U 67972107 IC50 = 55000 nM T20251 CB05ID 67972431 IC50 > 60000 nM T20251 C5K7QG 67974411 IC50 > 10000 nM T20251 CC28AD 68003782 IC50 = 28400 nM T20251 CXU2T6 68003962 IC50 = 16900 nM T20251 C7ZA5Y 68003997 IC50 = 35100 nM T20251 CQ4M8Y 68004002 IC50 > 50000 nM T20251 CB7T0X 68004010 IC50 = 37500 nM T20251 C9SZT4 68004011 IC50 = 28500 nM T20251 C9BFS2 68004012 IC50 > 50000 nM T20251 CX0B4G 68004016 IC50 > 50000 nM T20251 C6U9NR 68004034 IC50 > 50000 nM T20251 C8EM6J 68004094 IC50 = 11200 nM T20251 CCO4A2 68004146 IC50 = 13400 nM T20251 CO6W9D 68004741 IC50 > 10000 nM T20251 CB6U7F 68005465 IC50 > 10000 nM T20251 CK83VI 68005486 IC50 > 10000 nM T20251 C1RJ7Y 68005600 IC50 > 10000 nM T20251 COX3U9 68005621 IC50 = 8600 nM T20251 C57DTK 68045182 IC50 > 30000 nM T20251 CBOF40 68046989 IC50 = 2900 nM T20251 CG24FU 68071359 IC50 = 120 nM T20251 CG2QU1 68071450 IC50 = 9 nM T20251 CNS57A 68071672 IC50 = 2800 nM T20251 CJ8Y2W 68071788 IC50 = 25 nM T20251 CR5BI7 68071790 IC50 = 110 nM T20251 C3DZ1N 68071887 IC50 = 460 nM T20251 CTL92R 68083077 IC50 = 5900 nM T20251 C0PQL8 68094634 IC50 > 100000 nM T20251 CKJ13C 68095253 IC50 = 13000 nM T20251 CW23LG 68154393 IC50 = 49100 nM T20251 C4KYJ9 68171468 IC50 = 4900 nM T20251 C8T4IB 68199725 IC50 = 2200 nM T20251 C73IYJ 68199726 IC50 = 690 nM T20251 CV0P7D 68199727 IC50 = 1200 nM T20251 CY41JC 68199728 IC50 = 1000 nM T20251 C80ARK 68199735 IC50 = 1900 nM T20251 C7NM8D 68199737 IC50 = 8400 nM T20251 CZ3LH9 68199741 IC50 = 180 nM T20251 CUZX17 68204888 IC50 = 4600 nM T20251 C3K4RT 68204896 IC50 = 20000 nM T20251 CWTD61 68204898 IC50 = 6200 nM T20251 C5QZG7 68204899 IC50 = 2700 nM T20251 CF59AG 68204902 IC50 = 3100 nM T20251 CLS7H4 68204905 IC50 = 8400 nM T20251 CM58CG 68204907 IC50 = 6700 nM T20251 CNTP78 68204921 IC50 > 80000 nM T20251 C7V2SY 68204942 IC50 = 4600 nM T20251 C32QIB 68204998 IC50 = 4800 nM T20251 C4SWU5 68205000 IC50 > 80000 nM T20251 CZQ8R4 68205062 IC50 > 80000 nM T20251 CVA87O 68230212 IC50 > 30000 nM T20251 CYR38C 68241014 IC50 = 6600 nM T20251 C0DEM2 68254010 IC50 = 15000 nM T20251 C17JAZ 68284084 IC50 > 30000 nM T20251 CO48FM 68287853 Ki > 9182 nM T20251 C06RFV 68288164 Ki > 15219 nM T20251 CO6Z7D 68288263 Ki > 9182 nM T20251 C4M9LX 68289700 IC50 > 50118.72 nM T20251 C07JAL 68290083 IC50 > 50118.72 nM T20251 CC70KY 68290508 IC50 > 50118.72 nM T20251 CV9Q6N 68305341 IC50 = 10400 nM T20251 C8V0QK 68305342 IC50 > 11000 nM T20251 CIB52Q 68309298 IC50 > 50118.72 nM T20251 CBGL83 68309299 IC50 > 50118.72 nM T20251 CWDS89 68310172 IC50 > 50118.72 nM T20251 CI6YC4 68378925 IC50 > 30000 nM T20251 CI7S6T 68378958 IC50 = 25000 nM T20251 CU71NC 68379030 IC50 = 24000 nM T20251 C7CBD4 68379135 IC50 = 19000 nM T20251 CT32VB 68379165 IC50 = 23000 nM T20251 CBD8C9 68379213 IC50 = 2100 nM T20251 CLBY90 68380304 IC50 = 9200 nM T20251 CA9MK4 68432911 IC50 = 12000 nM T20251 CA7UZ6 68434755 IC50 = 9000 nM T20251 CQ38HU 68437484 IC50 > 30000 nM T20251 CGM78B 68472574 IC50 > 33000 nM T20251 CB8O4N 68475743 IC50 > 33000 nM T20251 C52HIW 68483436 IC50 = 9400 nM T20251 CEL85X 68483794 IC50 = 1800 nM T20251 CWE97U 68490431 IC50 > 100000 nM T20251 CM61LR 68495004 IC50 = 6000 nM T20251 C0OPQ6 68495695 IC50 = 2100 nM T20251 CXS64A 68502671 IC50 > 31600 nM T20251 C4XJ6F 68513796 IC50 > 100000 nM T20251 C3H7AJ 68513937 IC50 = 15000 nM T20251 C5QB6P 68528423 IC50 = 6000 nM T20251 C4B8KQ 68529738 IC50 = 3700 nM T20251 C85NIY 68533570 IC50 = 4600 nM T20251 C7MB8R 68591735 IC50 > 10000 nM T20251 CM5ZS8 68592173 IC50 > 10000 nM T20251 C2J0MD 68592299 IC50 > 10000 nM T20251 C8YG7Z 68592484 IC50 = 6835 nM T20251 C54QNY 68592631 IC50 = 7551 nM T20251 C6UW1R 68592632 IC50 > 10000 nM T20251 CP29IA 68592826 IC50 < 1000 nM T20251 C2GSP7 68593153 IC50 = 10000 nM T20251 C2PJN0 68593295 IC50 > 10000 nM T20251 C62QGB 68593458 IC50 = 10000 nM T20251 C1Q2UZ 68593479 IC50 = 7711 nM T20251 CKQ4O9 68593622 IC50 = 4580 nM T20251 CSQY72 68593732 IC50 > 10000 nM T20251 C2VIM9 68593774 IC50 > 10000 nM T20251 CE6X8W 68593871 IC50 > 10000 nM T20251 C0MYB6 68653619 IC50 > 33000 nM T20251 CH3Z7F 68658979 IC50 = 600 nM T20251 CYV20U 68728631 IC50 = 3700 nM T20251 CD3U6K 68731121 IC50 = 10500 nM T20251 CCB1T5 68764898 IC50 = 1800 nM T20251 C70QJS 68767049 IC50 = 14000 nM T20251 C8XT7M 68767109 IC50 > 80000 nM T20251 CP23JT 68767124 IC50 > 80000 nM T20251 CKWJ72 68767577 IC50 > 80000 nM T20251 C8U1DK 68767802 IC50 > 80000 nM T20251 CRM71Y 68768923 IC50 > 80000 nM T20251 C6L3ZT 68769143 IC50 > 80000 nM T20251 CHS3Z2 68769744 IC50 = 77000 nM T20251 CTL0O6 68770301 IC50 > 33000 nM T20251 CUVF59 68770356 IC50 = 24000 nM T20251 CT2D3M 68772321 IC50 = 32000 nM T20251 CX5Q2G 68772765 IC50 > 33000 nM T20251 CM92FU 68773430 IC50 = 27000 nM T20251 CZ07NC 68773726 IC50 > 33000 nM T20251 C16VTD 68774064 IC50 = 45000 nM T20251 CR28FH 68774353 IC50 > 33000 nM T20251 CWV13E 68774423 IC50 = 30000 nM T20251 C5J1XL 68774942 IC50 > 33000 nM T20251 C59FDP 68775014 IC50 > 31000 nM T20251 C23PDV 68775184 IC50 > 33000 nM T20251 CL6N2D 68775231 IC50 > 33000 nM T20251 CC98XW 68775928 IC50 = 56000 nM T20251 C89CQS 68779277 EC50 > 10000 nM T20251 CG46AF 68816399 IC50 = 1200 nM T20251 C9S1NP 68818964 IC50 = 1100 nM T20251 C6FZD0 68846936 IC50 = 25118.86 nM T20251 CZPM30 68849581 IC50 > 31622.78 nM T20251 C3YW1K 68860750 IC50 > 1000 nM T20251 C1UMP9 68867935 IC50 = 60000 nM T20251 C5PY2V 68938028 IC50 > 25118.86 nM T20251 C8Y3PB 68963393 IC50 = 700 nM T20251 C1KAN5 68963686 IC50 = 1600 nM T20251 C52BVJ 68963698 IC50 > 10000 nM T20251 CWZU52 68988296 IC50 > 80000 nM T20251 CBH6T3 69003776 IC50 = 14000 nM T20251 CG6JX0 69010662 IC50 > 31600 nM T20251 C9SFL1 69011426 IC50 = 2100 nM T20251 CYIB47 69012259 IC50 = 5900 nM T20251 CF57OD 69012280 IC50 = 3800 nM T20251 CI8GH6 69013596 IC50 = 4900 nM T20251 C6IP8Q 69082816 IC50 = 12000 nM T20251 C5CB4U 69087439 IC50 = 33000 nM T20251 CJM2Y1 69087440 IC50 = 10000 nM T20251 CZ0IC8 69087441 IC50 = 60000 nM T20251 C08ZXY 69087444 IC50 = 3400 nM T20251 CAIG78 69087446 IC50 = 3400 nM T20251 C57NKJ 69087450 IC50 = 8500 nM T20251 CX2U1Z 69087451 IC50 = 12000 nM T20251 C04OLI 69087452 IC50 = 52000 nM T20251 C59HRV 69087454 IC50 = 4500 nM T20251 C1O4EV 69087469 IC50 = 9100 nM T20251 CXV98R 69087490 IC50 = 31000 nM T20251 C1XE4Q 69087494 IC50 = 8200 nM T20251 CGQ40U 69087495 IC50 = 13000 nM T20251 CCO97X 69087505 IC50 = 27000 nM T20251 CI3A6W 69087537 IC50 = 100000 nM T20251 CMA21H 69087541 IC50 = 49000 nM T20251 CQF9T5 69087543 IC50 = 68000 nM T20251 CVG42E 69087545 IC50 = 22000 nM T20251 CG31FX 69087546 IC50 = 33000 nM T20251 CX3P0T 69087562 IC50 = 17000 nM T20251 CXF5P9 69213151 IC50 = 7943.28 nM T20251 C07YOG 69260079 IC50 = 31622.78 nM T20251 CV7P3D 69260851 IC50 = 31622.78 nM T20251 C4QO7E 69260946 IC50 = 31622.78 nM T20251 CO9U3M 69262172 IC50 = 1584.89 nM T20251 C7HN5L 69272932 IC50 = 31622.78 nM T20251 CJ2D3I 69274365 IC50 = 31622.78 nM T20251 CPGC67 69285465 IC50 > 80000 nM T20251 CM5XA1 69285531 IC50 = 32000 nM T20251 C0QZ4U 69285563 IC50 > 80000 nM T20251 C5T2GC 69285794 IC50 = 360 nM T20251 C8R4LZ 69286108 IC50 = 5300 nM T20251 CNT95I 69286635 IC50 = 2700 nM T20251 COD5Y1 69347575 IC50 = 15848.93 nM T20251 C51DQR 69347707 IC50 = 31622.78 nM T20251 C8F1CY 69347719 IC50 = 12589.25 nM T20251 C93COF 69347980 IC50 = 19952.62 nM T20251 CPW42A 69348078 IC50 = 25118.86 nM T20251 C6Z7UL 69435853 IC50 = 600 nM T20251 C6XQ3C 69439557 IC50 = 600 nM T20251 CGD48T 69513487 IC50 = 2000 nM T20251 C6RV9Y 69513502 IC50 = 110 nM T20251 C0NAD7 69513622 IC50 = 2000 nM T20251 C25HXG 69513678 IC50 = 5000 nM T20251 COSH07 69513688 IC50 = 100 nM T20251 CKE4H3 69513748 IC50 = 5000 nM T20251 C2AZ4X 69787126 IC50 = 3981.07 nM T20251 CC8QU9 70227534 IC50 > 10000 nM T20251 CI0XF8 70274815 IC50 > 100000 nM T20251 CCG16F 70276365 IC50 = 25118.86 nM T20251 CE1J0O 70276811 IC50 = 15848.93 nM T20251 C06WFN 70276830 IC50 > 100000 nM T20251 CDQ85E 70276990 IC50 > 100000 nM T20251 CGET13 70278898 IC50 = 31622.78 nM T20251 C2GT5H 70280758 IC50 > 100000 nM T20251 CA6DM2 70281073 IC50 > 100000 nM T20251 CK26FY 70295607 IC50 = 4400 nM T20251 CV4X5S 70295927 IC50 > 30000 nM T20251 CXD5V6 70297609 IC50 = 260 nM T20251 C5ZSV0 70355830 Ki = 5220 nM T20251 C7VJ6A 70647728 IC50 = 10000 nM T20251 CC63NT 70675147 IC50 = 37000 nM T20251 CYM94S 70676472 IC50 = 2200 nM T20251 C7J0FD 70676474 IC50 = 980 nM T20251 CLTA38 70676476 IC50 = 830 nM T20251 CMN57J 70676478 IC50 = 180 nM T20251 C9QZ7C 70676480 IC50 = 1560 nM T20251 CN12IT 70680969 IC50 = 2500 nM T20251 C0VEM7 70680970 IC50 = 6500 nM T20251 CP8XS4 70681040 Ki = 1400 nM T20251 CF85AB 70681063 Ki = 2460 nM T20251 C9LW7K 70681064 Ki = 950 nM T20251 CS8V7G 70681068 Ki = 730 nM T20251 CA27SR 70681184 IC50 > 10000 nM T20251 C23CRI 70681196 IC50 = 5350 nM T20251 CEP43U 70681217 IC50 = 1200 nM T20251 C4AX2B 70681647 IC50 = 900 nM T20251 C3MBU1 70681648 IC50 = 10 nM T20251 C71XOI 70681872 IC50 > 100000 nM T20251 C4KWV3 70682467 IC50 = 9800 nM T20251 CSM23I 70682523 IC50 > 10000 nM T20251 CZ84UX 70682584 IC50 > 100000 nM T20251 C8D6ZB 70683088 IC50 = 1600 nM T20251 CKM4C2 70683089 IC50 = 13000 nM T20251 C7BPF4 70683090 IC50 = 3600 nM T20251 CRTD40 70683091 IC50 = 2000 nM T20251 CJV64I 70683156 Ki = 160 nM T20251 C9BR3A 70683161 Ki = 2900 nM T20251 CN79ZX 70683165 Ki = 1900 nM T20251 C94GTH 70683168 Ki = 2800 nM T20251 C3ZY6F 70683178 Ki = 1400 nM T20251 C6QC5J 70683184 Ki = 300 nM T20251 CK6JM8 70683187 Ki = 980 nM T20251 C1UBD3 70683285 IC50 = 21900 nM T20251 C3NR1Z 70683781 IC50 = 300 nM T20251 C1ARO8 70684544 IC50 = 15848.93 nM T20251 C6CWV8 70684549 IC50 = 100 nM T20251 C9F5ZM 70684550 IC50 = 3500 nM T20251 CKN95T 70685174 IC50 = 2900 nM T20251 CUQ92A 70685175 IC50 = 1200 nM T20251 CIV4S6 70685239 Ki = 50 nM T20251 CLW68N 70685259 Ki = 2500 nM T20251 C2IDQ6 70685264 Ki = 1500 nM T20251 CO1ZR5 70685266 Ki = 600 nM T20251 CRP7Z1 70685269 Ki = 2900 nM T20251 CWIC42 70685308 IC50 = 28800 nM T20251 CNH04A 70685394 IC50 = 20800 nM T20251 CG1MS3 70685518 IC50 = 28000 nM T20251 C8HF3M 70685675 IC50 = 93200 nM T20251 C3UO2F 70686000 IC50 = 33000 nM T20251 C0NMH8 70686404 IC50 = 13400 nM T20251 C7OX5Z 70686473 IC50 > 33000 nM T20251 CYO5N3 70686766 IC50 > 25000 nM T20251 CL9RE3 70686820 IC50 > 100000 nM T20251 C65EDY 70686822 IC50 > 100000 nM T20251 CY0N4S 70687331 IC50 = 2600 nM T20251 C84GET 70687332 IC50 = 7000 nM T20251 CI0Z9V 70687389 Ki = 320 nM T20251 CEAK85 70687392 Ki = 800 nM T20251 C3E9VJ 70687415 Ki = 1100 nM T20251 C0A3VH 70687418 Ki = 2300 nM T20251 C0YZF1 70687477 IC50 = 3700 nM T20251 C9V6ML 70687502 Ki = 30000 nM T20251 CL8W4C 70687532 IC50 = 1920 nM T20251 C85ORZ 70687534 IC50 = 200 nM T20251 CFO9M4 70687535 IC50 = 5480 nM T20251 CX58LB 70688042 IC50 = 800 nM T20251 CWO02R 70688127 IC50 = 16300 nM T20251 CIS85H 70688149 IC50 = 5600 nM T20251 C4VU7J 70688210 IC50 > 60000 nM T20251 CR80CD 70688263 IC50 = 2100 nM T20251 CD2EW1 70688785 IC50 > 31622.78 nM T20251 C1GN5V 70688791 IC50 = 120 nM T20251 CA7PZ9 70688792 IC50 = 100 nM T20251 C17MXW 70688793 IC50 = 240 nM T20251 C5IYR0 70688897 IC50 > 100000 nM T20251 CL68HK 70689385 IC50 = 4200 nM T20251 CBY8T6 70689386 IC50 = 2800 nM T20251 CTJL92 70689387 IC50 = 15000 nM T20251 C6YJL1 70689452 Ki = 1100 nM T20251 CO89VX 70689473 Ki = 1200 nM T20251 CM3PD8 70689475 Ki = 2200 nM T20251 CIE2O6 70689591 IC50 = 6270 nM T20251 CHAV16 70689592 IC50 = 40800 nM T20251 CMGO80 70689593 IC50 = 13100 nM T20251 CVYC02 70689594 IC50 = 3300 nM T20251 C9RDP5 70689914 IC50 > 30000 nM T20251 C0QUO1 70689915 IC50 > 30000 nM T20251 CV82BX 70690866 IC50 = 7943.28 nM T20251 CVSJ38 70690870 IC50 = 25 nM T20251 CY6E2Q 70691339 IC50 = 1400 nM T20251 CV2T7S 70691408 IC50 = 1040 nM T20251 CJY73E 70691486 IC50 = 3000 nM T20251 CV8QT4 70691487 IC50 = 2000 nM T20251 C8R0SZ 70691558 Ki = 1100 nM T20251 CRXG05 70691559 Ki = 1200 nM T20251 CYJ3F6 70691560 Ki = 100 nM T20251 CK6I2V 70691577 Ki = 1500 nM T20251 C7ET5J 70691581 Ki = 990 nM T20251 CJ85NC 70691582 Ki = 930 nM T20251 C27IPY 70691584 Ki = 1100 nM T20251 C2N1MW 70691706 IC50 = 430 nM T20251 C14ZJR 70691707 IC50 = 840 nM T20251 C27ECJ 70691721 IC50 = 2500 nM T20251 C0XRC9 70691981 IC50 = 76000 nM T20251 C7ASK8 70692129 IC50 > 32000 nM T20251 C2GXN6 70692344 IC50 = 1600 nM T20251 CZOF81 70693115 IC50 = 6309.57 nM T20251 CMFW03 70693116 IC50 = 25118.86 nM T20251 C5RSJ0 70693117 IC50 = 25118.86 nM T20251 CM4P5Z 70693582 IC50 = 2100 nM T20251 CA9R2G 70693583 IC50 = 4500 nM T20251 C35ASU 70693584 IC50 = 1300 nM T20251 C8JUY5 70693585 IC50 = 7600 nM T20251 CX0E3Y 70693586 IC50 = 4700 nM T20251 CLN9F4 70693648 Ki = 900 nM T20251 CM3LU4 70693649 Ki = 2000 nM T20251 C3GVN0 70693667 IC50 = 760 nM T20251 CKP02Q 70693669 Ki = 1200 nM T20251 C6N3DT 70693670 Ki = 2750 nM T20251 C6GCU1 70693673 Ki = 1800 nM T20251 CHUE45 70693674 Ki = 680 nM T20251 C6P3XM 70693710 IC50 = 2700 nM T20251 CR30DQ 70693785 IC50 = 250 nM T20251 C52LMB 70693791 IC50 = 870 nM T20251 C7HW2B 70694179 IC50 > 33000 nM T20251 C1VS0O 70694288 IC50 = 750 nM T20251 C65FHO 70694723 IC50 > 30000 nM T20251 CCQ49A 70695045 IC50 = 12589.25 nM T20251 C63MTE 70695047 IC50 > 31622.78 nM T20251 C2O7WF 70695089 IC50 = 21500 nM T20251 C75YPE 70695115 IC50 > 25000 nM T20251 C01IDC 70695171 IC50 > 100000 nM T20251 C5T6JA 70695705 IC50 = 10000 nM T20251 CEK60M 70695761 Ki = 430 nM T20251 CX6L3G 70695764 Ki = 500 nM T20251 CF4HZ3 70695774 IC50 = 510 nM T20251 CBHD70 70695780 Ki = 3200 nM T20251 CZL9G2 70695782 Ki = 2300 nM T20251 CUL37Y 70695784 Ki = 2400 nM T20251 C26OHM 70695785 Ki = 1000 nM T20251 CD1V2W 70695786 Ki = 320 nM T20251 CFB1W2 70695912 IC50 = 31900 nM T20251 CB50NG 70696261 IC50 > 33000 nM T20251 C3GDX9 70696694 IC50 > 30000 nM T20251 CMS6J5 70697098 IC50 = 730 nM T20251 C84WJI 70697099 IC50 = 5100 nM T20251 CT1GF8 70697151 IC50 > 25000 nM T20251 C34WHG 70697225 IC50 > 100000 nM T20251 CBDL19 70792359 IC50 > 30000 nM T20251 C7DO1N 70817239 IC50 > 30000 nM T20251 C6L7FH 70817382 IC50 > 30000 nM T20251 CKP4O8 70855957 IC50 = 8600 nM T20251 CLKU89 70856302 IC50 = 7000 nM T20251 CUCQ24 70874317 EC50 > 100000 nM T20251 C1H7VK 70874453 EC50 = 23000 nM T20251 CJF91M 70874544 EC50 = 13200 nM T20251 C9EWB8 70874603 EC50 = 65000 nM T20251 CF1G3K 70874916 EC50 = 34000 nM T20251 C30AJI 70914208 EC50 = 16000 nM T20251 C2TC8W 70914230 EC50 = 71000 nM T20251 CM65DI 70980530 IC50 = 9000 nM T20251 CH7J2X 70982568 IC50 = 1000 nM T20251 C61DAP 70983443 IC50 = 1200 nM T20251 C9ASG6 70984064 IC50 = 3600 nM T20251 C0O7XS 71007248 IC50 = 2800 nM T20251 CHC04W 71008131 IC50 >= 10000 nM T20251 CX3H4C 71009783 IC50 = 1000 nM T20251 C57SJO 71041303 IC50 = 9300 nM T20251 CZ3BM6 71041781 IC50 = 600 nM T20251 C6HRK0 71041789 IC50 = 5400 nM T20251 C4A8FE 71041792 IC50 = 4470 nM T20251 CGXQ60 71041800 IC50 > 10000 nM T20251 C1X8VO 71041841 IC50 = 9100 nM T20251 C3J4SN 71041846 IC50 > 10000 nM T20251 C9WRL7 71041848 IC50 = 1800 nM T20251 C6SH7U 71041850 IC50 = 6000 nM T20251 CK2ML7 71041874 IC50 = 5800 nM T20251 CGWL13 71041904 IC50 = 7200 nM T20251 CV7DL8 71041905 IC50 = 5500 nM T20251 C9RX6A 71041917 IC50 = 8100 nM T20251 C18RLK 71072034 IC50 = 6309.57 nM T20251 C4C0SP 71072040 IC50 = 15848.93 nM T20251 C1YNH6 71072044 IC50 > 10000 nM T20251 CVU3G7 71072050 IC50 > 31622.78 nM T20251 C2M1JY 71072052 IC50 = 5011.87 nM T20251 CE6Y8Z 71072057 IC50 > 10000 nM T20251 C0Z3KN 71072081 IC50 = 6309.57 nM T20251 C3FR6X 71072104 IC50 = 10000 nM T20251 C1BEC9 71072113 IC50 = 6309.57 nM T20251 CNY09L 71072115 IC50 = 12589.25 nM T20251 CFNZ23 71072118 IC50 >= 10000 nM T20251 C6HRB4 71077940 Ki = 40700 nM T20251 C6NKY5 71078482 Ki = 11000 nM T20251 C50WGF 71078515 Ki = 7000 nM T20251 CQUR63 71089192 IC50 = 21000 nM T20251 CFK50V 71110267 Ki = 4500 nM T20251 CS4T0U 71110270 Ki = 4000 nM T20251 C3ORQ5 71110347 Ki = 4900 nM T20251 C3G7QB 71110423 Ki = 12000 nM T20251 CD80YI 71110425 Ki = 20500 nM T20251 CAH09S 71110518 Ki = 25700 nM T20251 CZ29NF 71113911 IC50 > 50118.72 nM T20251 CT1L2V 71113915 IC50 > 50118.72 nM T20251 C1XHA8 71116039 IC50 = 13000 nM T20251 CC43QK 71151588 IC50 = 6200 nM T20251 CYDQ07 71152634 IC50 = 14000 nM T20251 CV0O7K 71152643 IC50 = 8000 nM T20251 C1SQ5Y 71152646 IC50 = 2.13 nM T20251 CL2DQ6 71152655 IC50 = 1000 nM T20251 CHW5A1 71152656 IC50 = 6100 nM T20251 C9GD1Z 71152689 IC50 = 7900 nM T20251 CTK5F6 71152708 IC50 = 2700 nM T20251 CDI7Y0 71152709 IC50 = 8.75 nM T20251 C40QZK 71152713 IC50 = 320 nM T20251 C8QRW6 71152722 IC50 = 3.87 nM T20251 CFZS36 71152743 IC50 = 2000 nM T20251 CQ1Y5R 71152751 IC50 = 12200 nM T20251 CN1O5A 71152755 IC50 = 1.21 nM T20251 CUA70R 71152803 IC50 = 2400 nM T20251 C5MD0V 71152806 IC50 = 900 nM T20251 CDZ6I8 71152809 IC50 = 23900 nM T20251 C95POA 71152813 IC50 = 4000 nM T20251 CDW0Q6 71152814 IC50 = 25400 nM T20251 CIYU58 71152816 IC50 = 3300 nM T20251 C1HYG6 71152822 IC50 = 29100 nM T20251 C6AI9L 71152823 IC50 = 3700 nM T20251 C7R5CM 71152828 IC50 = 200 nM T20251 CQ1R7G 71152842 IC50 = 2.9 nM T20251 CV83IB 71152846 IC50 = 4260 nM T20251 CD2ZN8 71152850 IC50 = 9400 nM T20251 CLK89J 71152851 IC50 = 5300 nM T20251 C2LRT0 71152860 IC50 = 3200 nM T20251 C9B0LK 71152871 IC50 = 0.73 nM T20251 C2AP9L 71152878 IC50 = 9200 nM T20251 C21SCA 71152890 IC50 = 2900 nM T20251 CMG8Y1 71152895 IC50 = 800 nM T20251 CAD57T 71152903 IC50 = 1.19 nM T20251 CGVW14 71152905 IC50 = 3000 nM T20251 C50BQR 71152932 IC50 = 2400 nM T20251 CDKF43 71152934 IC50 = 700 nM T20251 CJZM06 71152971 IC50 = 370 nM T20251 C6W3UY 71152975 IC50 = 700 nM T20251 C05ODL 71152981 IC50 = 3300 nM T20251 CW5KQ7 71152985 IC50 = 8.35 nM T20251 C2G9IR 71153003 IC50 > 60000 nM T20251 C08EJQ 71153009 IC50 = 17300 nM T20251 CC42ES 71153030 IC50 = 8900 nM T20251 CI50XB 71153035 IC50 > 60000 nM T20251 CD4N6B 71153053 IC50 = 3.21 nM T20251 CALF50 71153055 IC50 = 6300 nM T20251 C3HZ6D 71153063 IC50 = 400 nM T20251 C84NTK 71153068 IC50 = 17500 nM T20251 CRES81 71153070 IC50 = 1300 nM T20251 CAV03R 71153095 IC50 = 5800 nM T20251 CSU6Y5 71153098 IC50 = 800 nM T20251 CH52AF 71153108 IC50 = 24400 nM T20251 CGI67Z 71153155 IC50 = 7600 nM T20251 CRJL31 71153157 IC50 = 1000 nM T20251 CPEC13 71153160 IC50 = 11.46 nM T20251 CK27UL 71153161 IC50 = 1.66 nM T20251 C21IBW 71153175 IC50 = 43500 nM T20251 CC9H1B 71181325 IC50 = 1200 nM T20251 CYXF24 71181326 IC50 = 11000 nM T20251 CS4O1D 71181328 IC50 = 8400 nM T20251 CJY8L3 71181338 IC50 = 2800 nM T20251 C5QVR4 71181386 IC50 = 4.83 nM T20251 C3A2MI 71181421 IC50 = 1400 nM T20251 CKO9P6 71181433 IC50 = 1600 nM T20251 CS7O9E 71181495 IC50 = 900 nM T20251 CM25RB 71181508 IC50 = 2700 nM T20251 CB98GE 71181529 IC50 = 1.78 nM T20251 CM1PL3 71181535 IC50 = 700 nM T20251 C0M1WO 71181547 IC50 > 60000 nM T20251 CX5P1U 71181567 IC50 = 1300 nM T20251 C9UP3L 71181628 IC50 = 7000 nM T20251 CY6V8S 71181641 IC50 = 5500 nM T20251 C32UMV 71203748 IC50 = 40000 nM T20251 CBKF84 71222614 IC50 = 3500 nM T20251 C87MGT 71226277 IC50 = 16000 nM T20251 CLIH32 71226367 IC50 = 4300 nM T20251 CRSA04 71226374 IC50 = 25700 nM T20251 C4J8MI 71226400 IC50 = 16000 nM T20251 CE4Y8J 71226521 IC50 = 2400 nM T20251 COU73Y 71226944 IC50 = 4500 nM T20251 C1WP5Y 71226964 IC50 = 13000 nM T20251 C1B9KV 71227161 IC50 = 12000 nM T20251 CI8E6U 71227163 IC50 = 8900 nM T20251 C7Y2LB 71230234 IC50 > 100000 nM T20251 CSB2N6 71235464 IC50 = 5800 nM T20251 C40JOZ 71235465 IC50 = 24000 nM T20251 CH29GF 71258526 IC50 > 30000 nM T20251 CIR30L 71263305 IC50 > 30000 nM T20251 C9AT8D 71263621 IC50 = 1600 nM T20251 C6BE5X 71271461 IC50 > 30000 nM T20251 C1MVL0 71273460 IC50 > 30000 nM T20251 C0GL4U 71276387 IC50 = 11400 nM T20251 CV7ZP5 71276437 IC50 = 4100 nM T20251 C47QTF 71279423 IC50 > 10000 nM T20251 CZR37K 71279507 IC50 > 2000 nM T20251 CU4P3X 71279543 IC50 > 3000 nM T20251 C5L8SW 71279563 IC50 > 1000 nM T20251 CV96FO 71279672 IC50 = 4150 nM T20251 CKJ58I 71279693 IC50 = 293 nM T20251 CZY5P7 71279859 IC50 = 414 nM T20251 CXZG59 71280008 IC50 = 4100 nM T20251 C5TXH9 71280067 IC50 > 3000 nM T20251 CW0FK6 71280128 IC50 > 30000 nM T20251 CGI01S 71280152 IC50 = 1440 nM T20251 C61BWN 71280407 IC50 > 2000 nM T20251 C5CTH0 71280416 IC50 < 300 nM T20251 C63EIL 71280539 IC50 = 429 nM T20251 CUP25C 71280634 IC50 = 6320 nM T20251 CT1NU9 71283192 IC50 = 4000 nM T20251 C8OGT4 71283628 IC50 > 30000 nM T20251 C4AP9F 71288434 IC50 > 10000 nM T20251 CNVG06 71304813 IC50 > 50000 nM T20251 CWY4S0 71304814 IC50 > 50000 nM T20251 C5DXK1 71307955 IC50 = 5000 nM T20251 CR37DA 71419478 IC50 = 31622.78 nM T20251 C3QUF4 71449241 EC50 = 4600 nM T20251 CBQ8P4 71449250 IC50 = 1258.93 nM T20251 CCX2W5 71449253 IC50 = 42 nM T20251 CR4L9T 71449282 IC50 = 10000 nM T20251 CHF08N 71449283 IC50 = 19952.62 nM T20251 CVY54C 71449294 IC50 = 3981.07 nM T20251 C5SML3 71449452 IC50 = 31622.78 nM T20251 CH5X6M 71449584 IC50 = 12589.25 nM T20251 CH5PX8 71449585 IC50 = 10000 nM T20251 CBIT41 71449750 IC50 > 100000 nM T20251 CDP7T0 71449813 IC50 > 10000 nM T20251 C92RIS 71449970 IC50 = 8500 nM T20251 CHU5V7 71449971 IC50 = 1300 nM T20251 CL64JH 71449972 IC50 = 5500 nM T20251 C5YX9S 71450146 IC50 = 300 nM T20251 CS2W0I 71450257 IC50 = 5500 nM T20251 CQ41UR 71450379 IC50 = 19000 nM T20251 CFPK62 71450420 IC50 = 11500 nM T20251 C6DIL5 71450436 IC50 = 8000 nM T20251 CPDJ19 71450468 Ki = 462 nM T20251 CB83YL 71451044 IC50 = 79.43 nM T20251 C0B7ZW 71451051 IC50 = 150 nM T20251 C0L8PR 71451052 IC50 = 3.1 nM T20251 CE98WI 71451053 IC50 = 67 nM T20251 C9BK1J 71451073 IC50 = 1810 nM T20251 CIFE14 71451076 IC50 = 12589.25 nM T20251 CLSQ82 71451077 IC50 = 31622.78 nM T20251 C0RL3C 71451078 IC50 = 6309.57 nM T20251 CGJ7K0 71451084 IC50 = 19952.62 nM T20251 CI0B8V 71451085 IC50 > 31622.78 nM T20251 C3FC1H 71451390 IC50 > 100000 nM T20251 C4W6YG 71451391 IC50 > 100000 nM T20251 CI1OL6 71451639 IC50 > 100000 nM T20251 CL7P2A 71451832 IC50 = 19000 nM T20251 CZ7R2Y 71451924 Ki = 950 nM T20251 C9AO0Q 71452203 IC50 = 16000 nM T20251 C03DBO 71452204 IC50 = 5000 nM T20251 CW6C9V 71452241 IC50 = 7000 nM T20251 CL01IH 71452297 Ki = 2206 nM T20251 C5ZKN6 71452298 Ki = 44 nM T20251 CHQ1F0 71452299 Ki = 377 nM T20251 CHEB80 71452520 IC50 = 6300 nM T20251 C0YXD3 71452871 IC50 = 1258.93 nM T20251 CY7NM9 71452872 IC50 = 2511.89 nM T20251 C42GQM 71452880 IC50 = 47 nM T20251 C3JZH1 71452881 IC50 = 280 nM T20251 CKMZ80 71452882 IC50 = 4700 nM T20251 CXT57R 71452899 IC50 = 6309.57 nM T20251 COQ0P1 71453071 IC50 = 31622.78 nM T20251 C8C9JT 71453204 IC50 > 100000 nM T20251 C45PHI 71453617 IC50 = 3100 nM T20251 CP74WT 71453805 IC50 > 33000 nM T20251 CT23NI 71453897 IC50 = 22 nM T20251 C3ZLD5 71453913 IC50 = 19700 nM T20251 CC7PH1 71453987 IC50 = 5100 nM T20251 CB43OI 71454008 IC50 = 24000 nM T20251 CZI84F 71454093 Ki = 1638 nM T20251 CLDP69 71454277 IC50 = 11000 nM T20251 C47GYB 71454279 IC50 > 25000 nM T20251 C02FKR 71454296 IC50 = 12589.25 nM T20251 C4JN5I 71454639 IC50 = 3.981 nM T20251 C8Q0JV 71454645 IC50 = 7 nM T20251 C5WU8L 71454670 IC50 = 3981.07 nM T20251 C7XQZ4 71454678 IC50 = 19952.62 nM T20251 CZ4HI3 71455166 IC50 = 7400 nM T20251 C0YD9K 71455398 IC50 = 15000 nM T20251 C8OD4R 71455430 Ki > 10000 nM T20251 C6LH8Q 71455522 IC50 = 1100 nM T20251 CL9YX8 71455523 IC50 = 1800 nM T20251 C8J0WA 71455643 IC50 = 16300 nM T20251 CS2V3E 71455663 IC50 = 8200 nM T20251 CZT0H5 71455744 IC50 = 9500 nM T20251 C8BRU5 71455750 IC50 = 8000 nM T20251 CB0RN5 71455780 IC50 = 13100 nM T20251 C6VDY5 71456055 IC50 = 8300 nM T20251 CMBU21 71456359 IC50 = 251.19 nM T20251 CVT39B 71456360 IC50 = 5011.87 nM T20251 CK87DI 71456361 IC50 = 1258.93 nM T20251 CT7EN2 71456366 IC50 = 22 nM T20251 C3YOV7 71456368 IC50 = 560 nM T20251 C1X6TY 71456401 IC50 = 6309.57 nM T20251 C7AL1C 71456402 IC50 > 25118.86 nM T20251 CORH12 71456403 IC50 = 19952.62 nM T20251 CC3Q9J 71456413 IC50 = 12589.25 nM T20251 CL9BS3 71456722 IC50 > 100000 nM T20251 CT0OQ6 71456725 IC50 = 31622.78 nM T20251 CE2M1B 71456899 IC50 = 23442.29 nM T20251 C6QVT0 71456917 IC50 > 33113.11 nM T20251 C3M9KC 71456918 IC50 > 33113.11 nM T20251 CCF78E 71456919 IC50 = 24547.09 nM T20251 CLO4B6 71456969 IC50 > 100000 nM T20251 CMB6O8 71457147 IC50 = 2900 nM T20251 C7MNB5 71457264 Ki = 800 nM T20251 CQB9F3 71457442 IC50 = 20200 nM T20251 C6PX9L 71457622 Ki = 2189 nM T20251 C1NH9X 71457850 IC50 > 10000 nM T20251 C1EA6Q 71458069 Ki = 18 nM T20251 C3VMS0 71458203 IC50 = 2511.89 nM T20251 C8T5EJ 71458204 IC50 = 158.49 nM T20251 CZ6BX7 71458205 IC50 = 63.1 nM T20251 CI7B2J 71458215 IC50 = 3.9 nM T20251 CK6S7X 71458227 IC50 = 1200 nM T20251 CPST04 71458774 IC50 > 33113.11 nM T20251 CZW7X0 71458868 IC50 > 19952.62 nM T20251 CJ98EQ 71459165 IC50 > 33000 nM T20251 CYL5C6 71459166 IC50 > 33000 nM T20251 C58BIQ 71459167 IC50 = 26800 nM T20251 CV4ZI2 71459168 IC50 = 17500 nM T20251 CY8G0F 71459407 IC50 = 2500 nM T20251 C1LIN4 71459486 IC50 = 1000 nM T20251 COJ85G 71459516 Ki = 2616 nM T20251 CJ1M6I 71459762 IC50 = 2511.89 nM T20251 C89YUI 71460069 IC50 = 150 nM T20251 CYBR37 71460098 IC50 = 7943.28 nM T20251 CQW3L4 71460099 IC50 = 6309.57 nM T20251 CSB76D 71460108 IC50 = 19952.62 nM T20251 CP26GF 71460416 IC50 = 10000 nM T20251 CH51UB 71460419 IC50 = 3981.07 nM T20251 C9LYM0 71460575 IC50 = 19000 nM T20251 CZH53R 71460636 IC50 > 10000 nM T20251 CR2C6Z 71461172 IC50 = 16000 nM T20251 CU9X6E 71461217 IC50 = 30000 nM T20251 C5UB8I 71461218 IC50 = 6000 nM T20251 CETP14 71461260 Ki = 1403 nM T20251 CBSY93 71461487 IC50 > 10000 nM T20251 CEBC62 71461781 IC50 = 15.85 nM T20251 C9DJ1V 71461782 IC50 = 50.12 nM T20251 CV6QH8 71461787 IC50 = 19 nM T20251 CC92TB 71461788 IC50 = 23 nM T20251 CV7ML5 71461830 IC50 = 19952.62 nM T20251 C9UG2X 71462100 IC50 > 100000 nM T20251 CL4MZ5 71462103 IC50 = 10000 nM T20251 CKYO86 71462283 IC50 > 31622.78 nM T20251 CX97KJ 71462389 IC50 > 10000 nM T20251 CZQ4T0 71462891 IC50 = 16400 nM T20251 COT2V4 71462903 IC50 > 33000 nM T20251 C6HN7D 71462955 IC50 = 1000 nM T20251 CG2KF6 71462956 IC50 = 12000 nM T20251 CH2CE8 71462982 Ki = 385 nM T20251 C9R4EX 71462983 Ki = 543 nM T20251 CQ4WG2 71462984 Ki = 300 nM T20251 C7UVZ5 71463198 IC50 = 9500 nM T20251 C0GBL7 71466345 IC50 = 2000 nM T20251 C3YA7I 71466474 IC50 = 47800 nM T20251 C2PMJ7 71474167 Ki = 530 nM T20251 COI42Y 71478198 Ki = 3000 nM T20251 C7MCJ0 71487141 IC50 = 500 nM T20251 CL3S8Q 71487418 IC50 = 11300 nM T20251 CFA9V1 71494937 IC50 = 16000 nM T20251 CCR8J9 71496459 IC50 > 33000 nM T20251 C8V4GQ 71496460 IC50 = 17500 nM T20251 CD64WC 71500036 IC50 > 33000 nM T20251 C1PC8B 71516677 IC50 = 2000 nM T20251 C24ZPL 71516877 IC50 = 5900 nM T20251 CY83FI 71516959 IC50 = 5000 nM T20251 C1N2HF 71517046 IC50 = 1600 nM T20251 C7GS4P 71517047 IC50 = 13000 nM T20251 CWLO57 71517048 IC50 = 5300 nM T20251 C87CZW 71517049 IC50 > 33000 nM T20251 CY0VJ8 71517192 IC50 = 5800 nM T20251 C5S0XY 71517194 IC50 = 6600 nM T20251 C31DLT 71517195 IC50 = 4100 nM T20251 CRG0P7 71517196 IC50 > 33000 nM T20251 CA07TC 71517197 IC50 > 33000 nM T20251 CLAF67 71517240 IC50 > 50000 nM T20251 CYSI71 71517241 IC50 > 50000 nM T20251 C8SR2Q 71517242 IC50 > 50000 nM T20251 C4TGH7 71517401 IC50 > 50000 nM T20251 CU28ZL 71517402 IC50 > 50000 nM T20251 C0BWE4 71517403 IC50 > 50000 nM T20251 CU2TR7 71517573 IC50 > 50000 nM T20251 C1XWC3 71517574 IC50 > 50000 nM T20251 CZ5QD8 71517575 IC50 > 50000 nM T20251 CGE96J 71517576 IC50 > 50000 nM T20251 CFZ27L 71517577 IC50 > 50000 nM T20251 CK81FA 71517737 IC50 > 50000 nM T20251 CVN31I 71518405 IC50 > 50000 nM T20251 CTL9E5 71518406 IC50 = 33500 nM T20251 C9V5RD 71518407 IC50 = 33600 nM T20251 CW39SU 71518408 IC50 = 14700 nM T20251 CH5UM0 71518570 IC50 = 23100 nM T20251 C6DIG9 71518571 IC50 > 50000 nM T20251 CZ0S5X 71518572 IC50 = 47000 nM T20251 CEJ1O6 71518573 IC50 > 50000 nM T20251 CQC14H 71518574 IC50 > 50000 nM T20251 CXV79I 71518727 IC50 = 38900 nM T20251 CMKZ52 71518728 IC50 = 40900 nM T20251 CL05CZ 71518896 IC50 > 50000 nM T20251 C4UMA0 71518897 IC50 = 33300 nM T20251 C3Y2CP 71518898 IC50 = 48900 nM T20251 CGO9T8 71519050 IC50 > 50000 nM T20251 CSU8J9 71519051 IC50 = 46600 nM T20251 C0E9LJ 71519052 IC50 = 46900 nM T20251 CK1GR7 71519053 IC50 = 23500 nM T20251 CGY45E 71519054 IC50 = 42400 nM T20251 C29BZD 71519055 IC50 = 20300 nM T20251 CR1IO9 71519224 IC50 = 27600 nM T20251 CQ8F3O 71519225 IC50 = 33700 nM T20251 CE07SH 71519226 IC50 = 7400 nM T20251 C2FE7Q 71519227 IC50 > 50000 nM T20251 CP25YK 71519381 IC50 > 50000 nM T20251 CZ03XO 71519496 IC50 > 33000 nM T20251 CLQ31I 71519674 Ki > 100000 nM T20251 CLE21W 71520368 IC50 > 33000 nM T20251 C5S0FT 71520369 IC50 > 33000 nM T20251 CZY20B 71520370 IC50 > 33000 nM T20251 C0T9BG 71520371 IC50 > 33000 nM T20251 C3AKL4 71520372 IC50 > 33000 nM T20251 C4OBM9 71520373 IC50 > 33000 nM T20251 CXT3L0 71520486 IC50 > 33000 nM T20251 CA3B5V 71520487 IC50 > 33000 nM T20251 C1HI9J 71520488 IC50 > 33000 nM T20251 C92QDP 71520489 IC50 > 33000 nM T20251 CM6DZ1 71520490 IC50 > 33000 nM T20251 CD1XT8 71520491 IC50 > 33000 nM T20251 CSQH86 71520575 IC50 > 33000 nM T20251 CM1B0W 71523649 IC50 = 14000 nM T20251 C8JC6A 71525586 Ki = 26915.35 nM T20251 CR9ZE5 71525587 Ki > 100000 nM T20251 CRL42M 71525588 Ki = 12882.5 nM T20251 CRM9Q1 71525678 Ki = 34673.69 nM T20251 C2GK7O 71525679 Ki = 43651.58 nM T20251 C7HR1A 71525680 Ki > 100000 nM T20251 C8A0NC 71525681 Ki > 100000 nM T20251 CKU02X 71527981 IC50 = 800 nM T20251 CG7HA3 71528087 IC50 = 3500 nM T20251 CCVD76 71528088 IC50 = 3900 nM T20251 C3O6EK 71529541 IC50 = 17500 nM T20251 C3CT1R 71530223 IC50 > 50000 nM T20251 CE82HN 71533671 IC50 = 3630 nM T20251 CI71DK 71533675 IC50 = 1600 nM T20251 CN8CM1 71533722 IC50 = 24000 nM T20251 C67ZSQ 71540073 IC50 = 4600 nM T20251 CVG8M5 71540729 IC50 = 4700 nM T20251 CWE32H 71540731 IC50 = 20000 nM T20251 C90TFO 71540846 IC50 = 7700 nM T20251 CK2EY7 71540967 IC50 > 33000 nM T20251 C3WR0T 71541076 IC50 > 33000 nM T20251 C0SKF2 71541077 IC50 = 29000 nM T20251 C45CNE 71541078 IC50 = 13000 nM T20251 C3UR6G 71541079 IC50 > 33000 nM T20251 CQ0D2T 71541080 IC50 > 33000 nM T20251 C9VF1X 71541081 IC50 > 33000 nM T20251 CBN7X9 71541082 IC50 > 33000 nM T20251 CJ89BQ 71541083 IC50 = 7800 nM T20251 C9T1HK 71541084 IC50 = 3600 nM T20251 CO26TC 71541094 IC50 = 10000 nM T20251 CE8YO0 71541095 IC50 = 6100 nM T20251 CN79ZY 71541096 IC50 = 10000 nM T20251 CNCR14 71541097 IC50 = 5300 nM T20251 CW34SU 71541098 IC50 = 7600 nM T20251 CKW24J 71541099 IC50 = 10000 nM T20251 C4PYZ6 71541174 IC50 = 6800 nM T20251 C1RZ5T 71541175 IC50 = 3300 nM T20251 CF1B8U 71541176 IC50 = 6600 nM T20251 CU5E7L 71541177 IC50 = 12000 nM T20251 C9I1QA 71541178 IC50 > 33000 nM T20251 CA5O1N 71541179 IC50 = 13000 nM T20251 CZUV57 71541180 IC50 = 21000 nM T20251 C92PZK 71541187 IC50 = 26000 nM T20251 C0T4RD 71541188 IC50 = 15000 nM T20251 CB91FO 71541189 IC50 = 11000 nM T20251 CY5E0J 71541190 IC50 = 21000 nM T20251 C4XK1S 71541191 IC50 = 13700 nM T20251 C32HNI 71541192 IC50 = 15400 nM T20251 C9C0JU 71541193 IC50 > 27000 nM T20251 CFO05K 71541194 IC50 = 26000 nM T20251 CD1T5J 71541195 IC50 = 23000 nM T20251 CXS47M 71541275 IC50 > 33000 nM T20251 C3AFY4 71541276 IC50 > 33000 nM T20251 C98TJN 71541277 IC50 = 15000 nM T20251 C4AG9L 71541278 IC50 > 33000 nM T20251 CVX93I 71541279 IC50 > 33000 nM T20251 C1J4KM 71541280 IC50 > 33000 nM T20251 CBWZ86 71541287 IC50 > 31000 nM T20251 CK82YE 71541288 IC50 > 33000 nM T20251 CQ81HF 71541289 IC50 = 19000 nM T20251 CU53JE 71541292 IC50 > 33000 nM T20251 CR7E4G 71541370 IC50 = 23000 nM T20251 C9IE3U 71541371 IC50 = 13000 nM T20251 CFO83N 71541372 IC50 = 25000 nM T20251 CI6J5K 71541373 IC50 = 12000 nM T20251 CC7YB2 71541376 IC50 = 29000 nM T20251 CWT0Y3 71541468 IC50 = 26000 nM T20251 CGJ86B 71541469 IC50 = 12000 nM T20251 C0CBT4 71541470 IC50 = 13000 nM T20251 CQ8JN9 71541471 IC50 = 18000 nM T20251 CZV7N9 71541472 IC50 = 34000 nM T20251 CL20CV 71541473 IC50 = 9000 nM T20251 C6J9NY 71541572 IC50 = 4300 nM T20251 CS0J6B 71541573 IC50 = 12000 nM T20251 C5CO8Z 71541574 IC50 = 17000 nM T20251 CI90PK 71541575 IC50 = 17000 nM T20251 C4FS8Z 71541576 IC50 = 3100 nM T20251 CSI37G 71541577 IC50 = 9200 nM T20251 C5D6IE 71541687 IC50 = 9000 nM T20251 C3RQP5 71542927 IC50 > 50000 nM T20251 C9N7YA 71544706 IC50 > 32000 nM T20251 C92NEY 71544707 IC50 > 32000 nM T20251 C83YJF 71544946 IC50 > 13000 nM T20251 C2PC6S 71547342 IC50 = 29000 nM T20251 CD97ZU 71547584 IC50 = 1700 nM T20251 CIRZ76 71547586 IC50 = 600 nM T20251 C7V9SQ 71547699 IC50 = 48000 nM T20251 CC0B1F 71547911 IC50 = 6500 nM T20251 CEV53L 71548006 IC50 > 30000 nM T20251 CI7Q4K 71548718 IC50 > 30000 nM T20251 CED62L 71548719 IC50 = 11000 nM T20251 CKB12X 71549359 IC50 = 27000 nM T20251 C4LZM6 71549637 IC50 = 17000 nM T20251 C6JOB5 71549767 IC50 = 5100 nM T20251 CV47CJ 71549769 IC50 = 8000 nM T20251 C5IV9D 71549913 IC50 = 7300 nM T20251 CSHT69 71550657 IC50 > 6000 nM T20251 C7XGD2 71552097 IC50 = 46000 nM T20251 CQ31YB 71552260 IC50 = 32700 nM T20251 CO3WL9 71552261 IC50 = 36100 nM T20251 CHO7D1 71555244 IC50 > 20000 nM T20251 CM04ZX 71555465 IC50 > 20000 nM T20251 C5HK2E 71555534 IC50 > 20000 nM T20251 COW5E6 71560030 IC50 = 13000 nM T20251 CKP12Z 71560031 IC50 = 17400 nM T20251 C6XBY4 71560280 IC50 = 49500 nM T20251 C0FQS4 71560281 IC50 = 2370 nM T20251 C0C5GA 71560284 IC50 > 32000 nM T20251 CYC2W1 71560403 IC50 = 213320 nM T20251 C1WA7E 71560526 IC50 = 21000 nM T20251 C6TEO9 71562957 IC50 = 65300 nM T20251 C0NFT4 71563078 IC50 = 22700 nM T20251 CY74BK 71570778 IC50 = 3950 nM T20251 C6WFT5 71570924 IC50 = 9200 nM T20251 C6SU2O 71572050 Ki = 37700 nM T20251 C14BCP 71572051 Ki = 23400 nM T20251 CB1YS4 71572385 Ki > 60000 nM T20251 CR0KX9 71572386 Ki = 2700 nM T20251 CN52ZY 71572387 Ki = 8600 nM T20251 C2L8XG 71572646 IC50 = 28000 nM T20251 CB2F3M 71573174 IC50 = 7400 nM T20251 C3R0FO 71575419 IC50 > 30000 nM T20251 CUJT21 71582799 IC50 > 100000 nM T20251 CHEZ52 71583033 IC50 = 6600 nM T20251 CNUV80 71583035 IC50 > 25000 nM T20251 CD0K5I 71583037 IC50 > 25000 nM T20251 CQV96E 71583048 IC50 > 33300 nM T20251 CSPR52 71583049 IC50 > 33300 nM T20251 CNT5F3 71583050 IC50 > 33300 nM T20251 CH7I0W 71583051 IC50 > 100000 nM T20251 CAQR82 71583149 IC50 > 25000 nM T20251 CQ16UM 71584055 IC50 > 33000 nM T20251 CWD2Z5 71585566 IC50 > 10000 nM T20251 CNY52I 71586326 Ki = 2000 nM T20251 C5YL7V 71590612 IC50 >= 10000 nM T20251 CH5LE3 71598532 IC50 = 6309.57 nM T20251 CYW46V 71601091 IC50 = 18350 nM T20251 CZS74H 71601235 IC50 > 40000 nM T20251 CAC2V3 71601378 IC50 > 40000 nM T20251 C3XKL2 71603135 Ki = 3388.44 nM T20251 CQ3Y9W 71603136 Ki = 831.76 nM T20251 CA4GQ7 71603139 Ki = 4677.35 nM T20251 CK4T5Q 71603140 Ki = 3630.78 nM T20251 C70OBY 71603141 Ki = 1513.56 nM T20251 C1HEY4 71603142 Ki = 2454.71 nM T20251 CUW27Q 71603194 Ki = 2754.23 nM T20251 C3YA4C 71603551 IC50 = 14800 nM T20251 C6MZO8 71603797 IC50 > 10000 nM T20251 CKY82R 71603916 IC50 = 25200 nM T20251 C9J0EH 71603917 IC50 = 20300 nM T20251 CT8ZS9 71603918 IC50 = 19900 nM T20251 C2X3AO 71603919 IC50 = 12500 nM T20251 CFTR25 71603920 IC50 = 10000 nM T20251 C7BD6V 71603987 IC50 = 75900 nM T20251 C98YDN 71603990 IC50 > 10000 nM T20251 CQ37SD 71604125 IC50 = 59400 nM T20251 CYLF28 71604550 IC50 = 371 nM T20251 CLQ64Y 71604552 IC50 = 208 nM T20251 C5V7WR 71604554 IC50 = 158 nM T20251 CV02ZN 71604556 Ki = 6 nM T20251 C80SAZ 71604558 IC50 = 60 nM T20251 CU6Y8R 71604699 IC50 = 74 nM T20251 CN1EC9 71604700 Ki = 3.5 nM T20251 C8BEX7 71604701 IC50 = 15 nM T20251 CC8PG6 71604703 IC50 > 10 nM T20251 CJ04ZL 71605375 IC50 = 40 nM T20251 C28ZRB 71605376 IC50 > 10000 nM T20251 CJTH01 71605377 IC50 = 146 nM T20251 C7J1QI 71605382 IC50 = 2908 nM T20251 CMZ9J1 71605546 IC50 > 10 nM T20251 CY4MR9 71605549 IC50 = 346 nM T20251 CL9E4D 71605712 IC50 = 53 nM T20251 CT0K3J 71605714 IC50 = 767 nM T20251 C1VE9A 71605716 IC50 = 107 nM T20251 C7L8SH 71605718 IC50 = 135 nM T20251 C08BKQ 71605894 IC50 = 24 nM T20251 CTX0A3 71605896 Ki > 100000 nM T20251 CD3A6U 71606227 IC50 = 285 nM T20251 CZ9AQ8 71606230 Ki = 1208 nM T20251 C4BP5U 71606232 Ki = 86 nM T20251 CB37JD 71606234 IC50 = 377 nM T20251 CW8YG2 71606394 IC50 = 1159 nM T20251 CLBT68 71606396 IC50 = 4019 nM T20251 CZJ74L 71606398 IC50 = 3901 nM T20251 CXM6Z7 71606400 IC50 > 10000 nM T20251 CZ2DN9 71606402 IC50 = 14426 nM T20251 C6WGD4 71606558 IC50 = 14014 nM T20251 CY7S8Z 71606562 Ki = 2460 nM T20251 CX1Z4A 71606712 IC50 = 1992 nM T20251 CJT3H7 71606718 IC50 = 9.9 nM T20251 CI6C2A 71606877 IC50 = 24 nM T20251 C2N0PZ 71606880 IC50 = 86 nM T20251 CBI53Y 71613516 IC50 > 30000 nM T20251 C1Z6JV 71613522 IC50 = 47600 nM T20251 CVBQ58 71614504 IC50 = 30900 nM T20251 CRD4I9 71625797 IC50 = 5400 nM T20251 C5IKR3 71625970 IC50 = 1000 nM T20251 CC54ZM 71625972 IC50 = 6309.57 nM T20251 C5NA4Y 71625975 IC50 = 3981.07 nM T20251 CW7DI6 71626041 IC50 = 1995.26 nM T20251 CGR3I5 71626043 IC50 = 15848.93 nM T20251 CCQ69B 71626102 IC50 = 7943.28 nM T20251 C2WJX0 71626755 IC50 = 10000 nM T20251 CTRE28 71626822 IC50 = 7943.28 nM T20251 C8TID3 71626894 IC50 = 3981.07 nM T20251 C26TXG 71626895 IC50 = 15848.93 nM T20251 C4DHC9 71626896 IC50 = 19952.62 nM T20251 CJV92N 71626898 IC50 = 3981.07 nM T20251 C3XV8I 71626968 IC50 = 5011.87 nM T20251 C7GZI2 71626969 IC50 = 1258.93 nM T20251 CX0VE7 71626971 IC50 = 7943.28 nM T20251 C46RFP 71655299 IC50 > 17500 nM T20251 CDL35U 71655748 IC50 > 10000 nM T20251 CI0GU8 71660496 IC50 = 10900 nM T20251 CA0N8I 71665696 IC50 = 8100 nM T20251 CGD2R7 71680685 IC50 = 7600 nM T20251 CT5L2D 71680688 IC50 = 1500 nM T20251 C6EDG5 71680844 IC50 = 8600 nM T20251 C4C9OW 71680849 IC50 = 9200 nM T20251 C26UGV 71681009 IC50 = 10000 nM T20251 CG2F5B 71681010 IC50 = 12000 nM T20251 CN7ZH6 71681015 IC50 > 33000 nM T20251 C50DHN 71681166 IC50 = 23000 nM T20251 C79QKU 71681209 IC50 = 195 nM T20251 C10OCG 71681315 IC50 = 5700 nM T20251 CRQ1Y6 71681316 IC50 = 2800 nM T20251 C4OU0Y 71681318 IC50 = 1500 nM T20251 C13RPX 71681468 IC50 = 9000 nM T20251 C86XQA 71681473 IC50 = 6150 nM T20251 CU23DO 71681634 IC50 > 33000 nM T20251 C8H2PC 71681635 IC50 = 11000 nM T20251 CH4R7G 71682752 IC50 = 1600 nM T20251 CBVC07 71682893 IC50 = 6000 nM T20251 CFE3Y7 71683044 IC50 = 8000 nM T20251 C3ISR6 71683048 IC50 = 9000 nM T20251 C8LE5D 71695973 IC50 = 22000 nM T20251 CS62NH 71698376 IC50 = 24200 nM T20251 CI8X1R 71698379 IC50 = 12500 nM T20251 CHGS40 71710904 IC50 = 3990 nM T20251 CF6JR1 71711842 IC50 > 3700 nM T20251 CVMG84 71711917 IC50 = 20200 nM T20251 CD3OY7 71711988 IC50 > 33000 nM T20251 C24DMC 71711989 IC50 = 3700 nM T20251 C4L1VN 71713035 IC50 = 14000 nM T20251 C8I9BS 71713478 IC50 = 3700 nM T20251 C9I3GO 71714121 IC50 = 16000 nM T20251 CW7TD2 71716405 IC50 = 2070 nM T20251 COBD81 71716733 IC50 > 33000 nM T20251 C5GE1T 71716742 IC50 > 50000 nM T20251 CWB3V1 71718136 IC50 > 20000 nM T20251 C0O4ID 71718185 IC50 > 33000 nM T20251 CUWM58 71719137 IC50 = 1300 nM T20251 C6YQ4H 71719475 IC50 = 2400 nM T20251 C02FQE 71719561 IC50 > 100000 nM T20251 CG30CF 71719764 IC50 > 50000 nM T20251 C2EWG5 71719830 IC50 > 33000 nM T20251 C1FYA8 71720426 IC50 = 17000 nM T20251 C8IBF0 71720519 IC50 = 5.1 nM T20251 CMI1V5 71720664 IC50 = 7200 nM T20251 CO7B8C 71720776 IC50 = 13000 nM T20251 C30NBJ 71722055 IC50 > 30000 nM T20251 CIN10C 71727133 IC50 = 14500 nM T20251 C73WPT 71730102 Ki = 11890 nM T20251 C7Z1IR 71730238 Ki = 8140 nM T20251 CF78GV 71730361 Ki = 1360 nM T20251 CFHK37 71730881 Ki = 616 nM T20251 CNH38L 71731010 Ki = 1427 nM T20251 CPB1F0 71731512 Ki = 2250 nM T20251 CQ82DI 71731513 Ki > 60000 nM T20251 C60BIX 71763463 IC50 > 100000 nM T20251 CC80KL 71768688 IC50 > 50000 nM T20251 C4KUV6 71768721 IC50 = 43000 nM T20251 C7ZY1J 71768865 IC50 = 5800 nM T20251 CV53CZ 71768899 IC50 > 50000 nM T20251 CKU6V5 71768931 IC50 = 29000 nM T20251 CTSK68 71811225 IC50 > 10000 nM T20251 CVL54T 71811261 IC50 = 4700 nM T20251 COVS02 71812189 IC50 = 1600 nM T20251 C2QT3H 71812413 IC50 = 4000 nM T20251 CZPJ89 71812414 IC50 > 30000 nM T20251 CU1KS7 71812606 IC50 = 17000 nM T20251 CRAB14 71812607 IC50 = 6000 nM T20251 C5JV1P 71812623 IC50 > 100000 nM T20251 CQD1F2 71812796 IC50 = 21000 nM T20251 C2UOA5 71812797 IC50 = 23000 nM T20251 C9NK1C 71812798 IC50 > 30000 nM T20251 C3RE7M 71812799 IC50 = 16000 nM T20251 CD28XR 71816087 IC50 = 9670 nM T20251 CW20HQ 71818431 IC50 > 50000 nM T20251 C2L7TX 71818575 IC50 > 50000 nM T20251 CZ47NP 71819426 IC50 > 33000 nM T20251 C8S3ON 72163808 IC50 > 33000 nM T20251 CPA03W 72163810 IC50 > 33000 nM T20251 CR4B7C 72163925 IC50 = 19000 nM T20251 CQFI71 72163926 IC50 = 16000 nM T20251 CU64GF 72163928 IC50 > 33000 nM T20251 CYNV72 72163929 IC50 = 19000 nM T20251 CK0TQ3 72163930 IC50 = 11000 nM T20251 CCHA62 72164043 IC50 = 16000 nM T20251 CG4M7N 72164287 IC50 > 33000 nM T20251 CZ7YO2 72164288 IC50 > 33000 nM T20251 CDKV52 72164289 IC50 > 33000 nM T20251 CJP4N6 72164290 IC50 > 33000 nM T20251 CE19XB 72164409 Ki = 3520 nM T20251 CB2NP7 72165228 IC50 = 26000 nM T20251 CH68XV 72188554 IC50 > 30000 nM T20251 CO15AV 72188905 IC50 > 30000 nM T20251 C1ERA6 72192163 IC50 = 5000 nM T20251 CD85OH 72201590 IC50 = 1100 nM T20251 C5KTR3 72201875 IC50 = 9 nM T20251 C1N7LQ 72202249 IC50 > 30000 nM T20251 CKMZ39 72202597 IC50 = 5000 nM T20251 CO5XJ3 72202738 IC50 = 3700 nM T20251 C9XL7F 72202747 IC50 > 10000 nM T20251 CJTS50 72202874 IC50 = 8100 nM T20251 CXLR81 72203284 IC50 > 30000 nM T20251 CA10KU 72205492 IC50 = 10230 nM T20251 C78TDP 72205494 IC50 = 9560 nM T20251 CB19LS 72205495 IC50 = 11490 nM T20251 C2PBS7 72375648 IC50 = 46 nM T20251 C23VDP 72375650 IC50 = 32000 nM T20251 CRZ48N 72375747 IC50 = 2500 nM T20251 C6W8VM 72375748 IC50 = 6500 nM T20251 CU9DR1 72375749 IC50 = 27000 nM T20251 CA0Y6E 72375832 IC50 = 5100 nM T20251 CKS9M4 72375834 IC50 = 1400 nM T20251 CV19HQ 72375835 IC50 = 6900 nM T20251 CJ9T5X 72375921 IC50 = 40000 nM T20251 CCP0Q4 72376019 IC50 = 26000 nM T20251 C3B0CK 72544445 IC50 > 30000 nM T20251 C1A4YW 72545684 IC50 > 30000 nM T20251 CU0NH5 72546987 IC50 = 170 nM T20251 C5WXJ6 72546988 IC50 = 530 nM T20251 CBK6T9 72546989 IC50 = 290 nM T20251 CU80HY 72547065 IC50 = 10600 nM T20251 CE3X8Y 72547066 IC50 = 2300 nM T20251 CCVG84 72547070 IC50 = 4800 nM T20251 CX70JT 72547320 IC50 = 4900 nM T20251 CY19IP 72547496 IC50 = 1500 nM T20251 CO1PV2 72548922 IC50 = 980 nM T20251 C8JTK6 72549156 IC50 > 19000 nM T20251 CT0RY5 72550282 IC50 > 20000 nM T20251 C2Q6YJ 72670421 IC50 > 10000 nM T20251 CN2GV9 72697443 IC50 = 47500 nM T20251 CCT15O 72703033 IC50 = 3700 nM T20251 CPIO30 72706193 IC50 = 350 nM T20251 C1CQG9 72706253 IC50 = 9200 nM T20251 CF4W8Z 72706442 IC50 = 2200 nM T20251 CX6T7A 72706947 IC50 = 29000 nM T20251 CBE48L 72707143 IC50 > 10000 nM T20251 CRNB25 72711191 IC50 > 33000 nM T20251 C1XSU9 72711835 IC50 > 33000 nM T20251 C29YGC 72712370 IC50 = 2300 nM T20251 C7A5EW 72714054 IC50 > 20000 nM T20251 C7SZ3V 72714058 IC50 = 35300 nM T20251 C61NKZ 72720906 IC50 > 100000 nM T20251 C6PLC5 72722131 IC50 = 25900 nM T20251 C8QEJ3 72725792 IC50 > 50000 nM T20251 C7AO4X 72792633 IC50 > 33000 nM T20251 CLK7O4 72792692 IC50 > 33000 nM T20251 CO4EX3 72793304 IC50 = 4080 nM T20251 C0KWR6 72793305 IC50 = 40 nM T20251 C65WZH 72793306 Ki = 1.8 nM T20251 C7YIT5 72793307 IC50 = 7820 nM T20251 CQ0S4C 72793308 IC50 = 3543 nM T20251 CU19BY 72793309 IC50 = 2654 nM T20251 CY42BM 72793378 IC50 = 4.9 nM T20251 C9IHR7 72793379 IC50 = 3470 nM T20251 CM04AY 72793380 IC50 = 5090 nM T20251 CTD8U0 72793381 Ki = 97 nM T20251 C0J2HG 72793383 IC50 = 4394 nM T20251 CW3O4P 72793384 IC50 = 6007 nM T20251 C6VC4N 72793385 IC50 = 53 nM T20251 CJ8RX9 72793386 IC50 = 5590 nM T20251 C6D9FH 72793441 IC50 = 1890 nM T20251 C5IL8C 72793442 IC50 = 473 nM T20251 CMK6T0 72793446 IC50 = 7372 nM T20251 CD5W8J 72793447 IC50 = 834 nM T20251 CPS57O 72793448 IC50 = 4810 nM T20251 C5BX1R 72793512 IC50 = 970 nM T20251 CHG41A 72793513 IC50 = 1050 nM T20251 C9AUO5 72793514 IC50 = 243 nM T20251 CQJF87 72793517 IC50 = 1127 nM T20251 CD5O1Q 72793518 IC50 < 5 nM T20251 C24KXZ 72793520 Ki = 119 nM T20251 CN7R9Y 72793578 IC50 = 1868 nM T20251 CZ57PR 72793579 IC50 = 238 nM T20251 C16GMC 72793580 IC50 = 1178 nM T20251 C13QTN 72793581 IC50 = 1.5 nM T20251 CB4CT7 72793582 IC50 = 2500 nM T20251 CWGK78 72793583 IC50 = 123 nM T20251 CH07SV 72793584 IC50 = 124 nM T20251 CHDB60 72793898 IC50 = 3200 nM T20251 C6R8DI 72943374 IC50 > 50000 nM T20251 C6ZA8H 72945087 IC50 > 10000 nM T20251 C7MS4G 72945112 IC50 = 13100 nM T20251 CXOI39 72945311 IC50 = 4600 nM T20251 C5TS1M 72945313 IC50 = 1000 nM T20251 CH63BO 72945314 IC50 = 700 nM T20251 C2VU8F 72945510 IC50 = 2400 nM T20251 CQ5MD0 72945512 IC50 = 3800 nM T20251 C4EM1B 72945827 IC50 > 50000 nM T20251 C1G5DP 72945830 IC50 > 50000 nM T20251 C8RLE2 72946008 IC50 > 50000 nM T20251 CDG6A2 72946010 IC50 > 50000 nM T20251 C3N7RS 72946013 IC50 = 49600 nM T20251 COEL45 72946092 IC50 > 30000 nM T20251 C37UZP 72946198 IC50 > 50000 nM T20251 CF65HX 72946199 IC50 > 50000 nM T20251 CI8Z0Q 72946200 IC50 > 50000 nM T20251 C9FLS6 72946202 IC50 = 42600 nM T20251 CA4L5S 72946204 IC50 > 50000 nM T20251 CPA9G7 72946205 IC50 = 42100 nM T20251 CF7WR3 72946381 IC50 > 50000 nM T20251 CX82VR 72946384 IC50 > 50000 nM T20251 C7X2ZL 72946387 IC50 > 50000 nM T20251 C16RLM 72946775 IC50 > 50000 nM T20251 CP21YZ 72946982 IC50 > 50000 nM T20251 CB51JH 72947191 IC50 > 50000 nM T20251 CZR9S4 72947193 IC50 > 50000 nM T20251 CMB52G 72947411 IC50 = 24100 nM T20251 CN8U7J 72947413 IC50 > 50000 nM T20251 CU9NB5 72947593 IC50 > 50000 nM T20251 C7TIG1 72947595 IC50 > 50000 nM T20251 CJQ04K 72948000 IC50 > 50000 nM T20251 CO42FH 72948001 IC50 > 50000 nM T20251 CFC70R 72948004 IC50 > 50000 nM T20251 CR70EY 72948808 IC50 = 37000 nM T20251 CA76TR 72948995 IC50 = 63400 nM T20251 CDN18F 72950534 IC50 = 109.1 nM T20251 C8R1CQ 72950535 IC50 = 416.8 nM T20251 CJZW17 72950698 IC50 = 216 nM T20251 CQF4K5 72950786 IC50 = 1000 nM T20251 C9WU2M 72950813 IC50 > 20000 nM T20251 CY9A0D 73211784 IC50 > 10000 nM T20251 CH1JK9 73213123 EC50 > 50000 nM T20251 C62TJC 73254853 EC50 > 30000 nM T20251 CG8RI0 73292361 IC50 = 7100 nM T20251 CBQ72N 73292545 IC50 = 9100 nM T20251 CKA79H 73292924 IC50 = 20000 nM T20251 C95JUO 73293105 IC50 = 600 nM T20251 CRY7G9 73294187 IC50 = 1500 nM T20251 CQV1P0 73294507 IC50 = 4200 nM T20251 C7EW4M 73294791 IC50 = 7330 nM T20251 C31ZVM 73294948 IC50 > 10000 nM T20251 CV2B0K 73294950 IC50 > 10000 nM T20251 CG8T3O 73295804 IC50 > 10000 nM T20251 CG9L2Q 73295805 IC50 > 30000 nM T20251 C5F0XZ 73295967 IC50 > 10000 nM T20251 C46HKB 73295968 IC50 > 10000 nM T20251 CTP8H1 73296128 IC50 > 10000 nM T20251 C7S0QC 73296291 IC50 > 10000 nM T20251 C86WRD 73296431 IC50 > 10000 nM T20251 C7G5OI 73296435 IC50 > 10000 nM T20251 C59TYH 73296577 IC50 > 10000 nM T20251 C9LBA7 73296578 IC50 > 10000 nM T20251 CWJS76 73331695 IC50 > 30000 nM T20251 C57LGA 73349098 IC50 = 44000 nM T20251 CX08AE 73349556 IC50 = 418350 nM T20251 CC5B9P 73351121 IC50 = 18660 nM T20251 CT1XL6 73352589 IC50 = 131 nM T20251 C3EV2U 73352607 IC50 = 5600 nM T20251 CG7R3F 73353420 IC50 = 13000 nM T20251 C0K7WP 73356819 IC50 = 206000 nM T20251 C5LBH4 73357152 IC50 = 42970 nM T20251 C6AN3L 73357170 IC50 = 11 nM T20251 C9ODB8 73387740 IC50 > 30000 nM T20251 CT1E6V 73387743 IC50 = 17300 nM T20251 CU3D9N 73388373 EC50 = 39810.72 nM T20251 CRA5H6 73389570 IC50 > 10000 nM T20251 C6V2TF 73426595 IC50 = 30000 nM T20251 C8JTD0 73442848 IC50 > 60000 nM T20251 CEP9F4 73507167 IC50 = 15800 nM T20251 CVF5P0 73603034 IC50 = 2700 nM T20251 C1SD9O 73670857 IC50 = 300 nM T20251 CJQ8B4 73670858 IC50 = 230 nM T20251 CM3Y6X 73670970 EC50 > 30000 nM T20251 CC3AG1 73670971 EC50 > 30000 nM T20251 C06YDA 73671018 IC50 = 2540 nM T20251 CJOU70 73671602 IC50 = 7200 nM T20251 CNIL19 73671824 IC50 = 1570 nM T20251 C85GVU 73671825 IC50 = 4530 nM T20251 C2K5DS 73672762 IC50 = 1900 nM T20251 C5XM3C 73673377 IC50 = 20 nM T20251 CYX59S 73673505 IC50 > 100000 nM T20251 CGC10B 73777172 IC50 = 6309.57 nM T20251 C5LPC2 73777186 IC50 = 3981.07 nM T20251 C3NDE7 73777188 IC50 = 12589.25 nM T20251 CS71JA 73777210 IC50 = 10000 nM T20251 CK3W5O 73777215 IC50 = 7943.28 nM T20251 CJ86QT 73953235 IC50 = 10000 nM T20251 CMU19S 74221664 IC50 > 30000 nM T20251 CZ3TB5 74221949 IC50 = 64000 nM T20251 CW9N8T 74222036 IC50 = 74000 nM T20251 CZK27X 74627726 IC50 = 26 nM T20251 C7M4FR 75201717 IC50 = 36000 nM T20251 C0OJ7W 75201718 IC50 = 16000 nM T20251 C2S0CO 75201720 IC50 > 80000 nM T20251 C5S2HO 75201785 IC50 = 16000 nM T20251 C4U5MR 75201786 IC50 = 6700 nM T20251 C6S2ZO 75201851 IC50 = 43000 nM T20251 C2E7QW 75201901 IC50 = 12000 nM T20251 CPS18J 75276948 EC50 > 80000 nM T20251 CF1G7P 76070567 IC50 = 3490 nM T20251 CW61JI 76071739 IC50 = 13200 nM T20251 C1W9RS 76072334 IC50 > 10000 nM T20251 CQ71AT 76073628 IC50 = 1700 nM T20251 C0N3RW 76282073 IC50 > 30000 nM T20251 CN2M8A 76284154 IC50 = 7300 nM T20251 C5ALQ2 76285468 IC50 > 10000 nM T20251 CFRU64 76285722 IC50 > 30000 nM T20251 C52KTI 76286498 IC50 = 9300 nM T20251 CZF0N7 76287389 IC50 > 30000 nM T20251 CDM04P 76310604 IC50 = 3960 nM T20251 C18SIP 76310732 IC50 = 8500 nM T20251 CO1TF8 76311072 IC50 = 30000 nM T20251 CL3N7Y 76311099 IC50 < 10 nM T20251 CB2QY6 76311111 IC50 > 33000 nM T20251 CY43DL 76311112 IC50 > 33000 nM T20251 CMF40L 76313439 IC50 = 400 nM T20251 CT2QF9 76314234 IC50 > 50000 nM T20251 CA83KU 76314239 IC50 = 2340 nM T20251 CSFB37 76314242 IC50 = 22900 nM T20251 CJ38IO 76314519 EC50 = 9800 nM T20251 C8HIS3 76314722 IC50 > 33000 nM T20251 C7K2WL 76314723 IC50 > 33000 nM T20251 C1H0GX 76314724 IC50 > 33000 nM T20251 CSL9B8 76317193 Ki > 10000 nM T20251 CEUN37 76317941 IC50 = 2000 nM T20251 CN8Q6E 76318296 IC50 > 33000 nM T20251 C1ZY4T 76318298 IC50 > 33000 nM T20251 CET31O 76318342 IC50 = 176600 nM T20251 CCMW30 76320680 IC50 = 1400 nM T20251 CDE3Y9 76321032 IC50 = 4000 nM T20251 C3TXQ5 76321521 IC50 = 16800 nM T20251 CQT3F1 76321527 IC50 > 50000 nM T20251 CEK3O5 76321713 IC50 = 6000 nM T20251 CNY2D6 76321910 EC50 = 20000 nM T20251 CR05PL 76322043 IC50 = 6100 nM T20251 CQ3CW1 76322044 IC50 = 12000 nM T20251 CYXU43 76322162 IC50 > 100000 nM T20251 C8N9QM 76325121 IC50 > 50000 nM T20251 CD3CE2 76325259 IC50 = 2800 nM T20251 CC79HT 76325260 IC50 = 6800 nM T20251 CHDF36 76325614 IC50 > 33000 nM T20251 CS27NF 76325615 IC50 > 33000 nM T20251 C3C7HE 76325645 IC50 = 48000 nM T20251 C2HCL6 76327886 IC50 = 200 nM T20251 CP9V7B 76328692 IC50 = 1260 nM T20251 CI3U1S 76328815 IC50 = 2700 nM T20251 CF27TB 76328817 IC50 = 1800 nM T20251 C5UMK8 76328829 IC50 > 40000 nM T20251 C8CQ9Y 76328873 IC50 = 14000 nM T20251 C8H9JD 76329183 IC50 > 33000 nM T20251 CAXT31 76329184 IC50 > 33000 nM T20251 C7S0CZ 76329185 IC50 > 33000 nM T20251 CWD5R4 76331595 IC50 = 3 nM T20251 CS7MR5 76331825 IC50 = 58 nM T20251 C2YIP6 76332364 IC50 = 12500 nM T20251 CNA06U 76332366 IC50 = 780 nM T20251 CI2K3T 76332845 IC50 > 33000 nM T20251 CTVI40 76332894 IC50 = 4000 nM T20251 CL7TN0 76332895 IC50 = 5600 nM T20251 CZ93JC 76335400 IC50 = 14443 nM T20251 C3Y0WL 76335990 IC50 > 50000 nM T20251 CGE5S3 76336366 EC50 = 32000 nM T20251 C0VAU9 76336449 IC50 < 10 nM T20251 CD7TI2 76336464 IC50 > 33000 nM T20251 C92WBQ 76336500 IC50 = 12700 nM T20251 C8KBZ1 76336501 IC50 = 1500 nM T20251 CQM69X 76336502 IC50 = 23300 nM T20251 C5PW6K 76683678 IC50 > 10000 nM T20251 CXM51U 76683680 IC50 = 4900 nM T20251 CGE15Z 76683773 IC50 > 10000 nM T20251 CL03DO 76683775 IC50 > 10000 nM T20251 C8HAR3 76683777 IC50 > 10000 nM T20251 CG0TR9 76683781 IC50 = 2200 nM T20251 C95OWP 76683875 IC50 = 3900 nM T20251 C67SLP 76683883 IC50 > 10000 nM T20251 C6IS1X 76683885 IC50 > 10000 nM T20251 CBSD29 76683976 IC50 > 10000 nM T20251 C0WR4O 76684092 IC50 > 10000 nM T20251 CR76SA 76684100 IC50 > 10000 nM T20251 CLD49W 76684104 IC50 = 3100 nM T20251 C08EZV 76684202 IC50 > 10000 nM T20251 C75VCS 76684206 IC50 > 10000 nM T20251 CKC14S 76684208 IC50 > 10000 nM T20251 CV62NT 76684214 IC50 = 5200 nM T20251 C8P7EC 76684296 IC50 = 2200 nM T20251 C6MSH2 76684391 IC50 > 10000 nM T20251 CAT95V 76685067 IC50 = 79750 nM T20251 CR3N1A 76900049 IC50 > 40000 nM T20251 CM73EU 76901852 IC50 = 14800 nM T20251 CQT14W 76955651 IC50 = 10100 nM T20251 C9EP7I 77003908 IC50 > 10000 nM T20251 C51DJB 77050686 IC50 > 10000 nM T20251 C2JTH8 77107528 IC50 > 30000 nM T20251 CPZ92R 77460996 IC50 = 140 nM T20251 C34TAM 77845572 IC50 > 30000 nM T20251 CT6E4H 77846842 IC50 = 700 nM T20251 CX5A7E 77846926 IC50 > 10000 nM T20251 CLC6F8 77938792 IC50 = 6400 nM T20251 CAV9J0 77989921 IC50 = 3600 nM T20251 CQZ0L8 78158242 IC50 >= 10000 nM T20251 C2NCH9 78318214 IC50 > 30000 nM T20251 C2GET7 78318815 IC50 > 30000 nM T20251 CKOU34 78319724 IC50 = 3900 nM T20251 CO0DA2 78320170 IC50 = 10800 nM T20251 C5FP1U 78321115 IC50 > 100000 nM T20251 C43NLO 78322060 IC50 = 9870 nM T20251 CV0P3A 78357783 IC50 = 14800 nM T20251 CDX94E 78426574 IC50 = 5600 nM T20251 C86QLE 81689770 IC50 = 8000 nM T20251 C9GQS2 81689815 IC50 = 50000 nM T20251 C3U0KE 81689842 IC50 > 100000 nM T20251 CHW72V 82556507 IC50 > 25000 nM T20251 CQ74UP 84626694 IC50 = 41000 nM T20251 CQMB31 85470872 IC50 > 10000 nM T20251 CLG83C 86268944 IC50 > 20000 nM T20251 CA1CE3 86270720 IC50 > 10000 nM T20251 C9TE7X 86271008 IC50 > 10000 nM T20251 CMZV56 86271009 IC50 > 10000 nM T20251 CXN93A 86271108 IC50 > 10000 nM T20251 CZL23E 86271138 IC50 > 100000 nM T20251 C5IR2K 86271238 IC50 = 8500 nM T20251 CN9MO7 86271494 IC50 > 3000 nM T20251 C4T3IW 86272102 IC50 = 39000 nM T20251 C30NBD 86272865 IC50 = 12589.25 nM T20251 C3OLB1 86274489 IC50 = 66000 nM T20251 CAB78T 86274732 IC50 = 50000 nM T20251 CCU13T 86275207 IC50 = 50000 nM T20251 CMR27C 86276168 IC50 > 25000 nM T20251 COS71Y 86276169 IC50 > 25000 nM T20251 CK20QY 86276216 IC50 > 100000 nM T20251 CW0ER2 86276224 IC50 = 900 nM T20251 CF4QX9 86278359 IC50 > 10000 nM T20251 CL09JQ 86279005 IC50 = 19560 nM T20251 CQC9M3 86279081 IC50 = 1000 nM T20251 C98IVM 86279102 Ki = 3300 nM T20251 CFJ10Z 86279104 Ki = 28800 nM T20251 CI5N8M 86279145 IC50 = 1200 nM T20251 CXF9Q3 86279146 IC50 = 10000 nM T20251 C4Y3VP 86279147 IC50 > 33000 nM T20251 CSL0I1 86279148 IC50 > 33000 nM T20251 CU70DL 86279235 IC50 = 3600 nM T20251 C38CMG 86279412 IC50 > 10000 nM T20251 C31OGJ 86279928 IC50 > 20000 nM T20251 CH3FN8 86288905 IC50 = 6800 nM T20251 CO74AR 86292101 IC50 = 5000 nM T20251 CF7GZ5 86292750 IC50 = 20800 nM T20251 CF7Y2I 86292753 IC50 = 2600 nM T20251 CV8OI5 86292754 IC50 = 1430 nM T20251 CDV37Y 86292938 IC50 = 15000 nM T20251 CZ97VP 86294733 IC50 = 24900 nM T20251 CN0W9I 86302543 IC50 = 600 nM T20251 C9EMQ0 86304601 IC50 > 30000 nM T20251 C5ZI4L 86341927 EC50 = 22800 nM T20251 CZI4Q8 86342076 EC50 > 30000 nM T20251 C4EQ8X 86342079 EC50 = 14100 nM T20251 CMK19R 86342113 EC50 > 30000 nM T20251 C73LNE 86342141 EC50 = 18800 nM T20251 CK03YC 86342156 IC50 = 2110 nM T20251 CB5F1W 86343364 IC50 = 2100 nM T20251 CKG7N2 86343365 IC50 = 13800 nM T20251 C9IVM5 86343366 IC50 = 4800 nM T20251 CMXZ65 86346192 IC50 > 50000 nM T20251 C6CD1Z 86617892 IC50 > 32000 nM T20251 CH86IJ 86670613 IC50 > 80000 nM T20251 CMG39E 86673884 IC50 > 30000 nM T20251 C9NTP1 86677234 IC50 = 5600 nM T20251 C5YX8T 86677253 IC50 = 15600 nM T20251 CCX1U5 86677265 IC50 = 7400 nM T20251 CZQ1F7 86677270 IC50 = 4300 nM T20251 CDXM47 86677874 IC50 = 75000 nM T20251 CXJA65 86685547 IC50 = 10000 nM T20251 CTG76E 86687532 IC50 > 30000 nM T20251 CR76VN 86694482 IC50 = 1200 nM T20251 CRJ9F2 86699098 IC50 > 72000 nM T20251 C52BXE 86705377 IC50 = 490 nM T20251 CC8I0M 86707711 IC50 = 3000 nM T20251 CMK52I 86721807 Ki = 780 nM T20251 CZ5J3N 86721820 Ki = 1800 nM T20251 COA34E 86721822 Ki = 1300 nM T20251 CNDS02 86722641 IC50 = 8800 nM T20251 CS7T2Z 86722660 IC50 = 8600 nM T20251 CVJ8L5 86728666 IC50 = 3500 nM T20251 C3FE1T 86730519 IC50 = 6500 nM T20251 CJ0V5L 86730522 IC50 = 2100 nM T20251 CA17UE 86732669 IC50 > 30000 nM T20251 C7OIC6 86762648 IC50 = 4300 nM T20251 CQ45XR 86763358 IC50 > 3162.28 nM T20251 CF70JO 86765186 IC50 = 12870 nM T20251 CR7Y9T 86766090 IC50 = 4500 nM T20251 C2U0BG 87055263 IC50 = 4600 nM T20251 C02UGP 87056204 IC50 = 24000 nM T20251 C6FO9E 87152177 IC50 = 13000 nM T20251 CNVS32 87343636 IC50 > 30000 nM T20251 C2EMU3 87509467 IC50 = 1132 nM T20251 CH7N2Y 87509988 IC50 = 2862 nM T20251 CF67AV 88875879 IC50 > 30000 nM T20251 C7QJ8S 88886827 IC50 = 24000 nM T20251 C6JLC2 89315866 IC50 = 1600 nM T20251 CWR09T 89449220 IC50 = 1800 nM T20251 CTC40E 89449230 IC50 = 6400 nM T20251 CW4Z2F 89470642 IC50 = 40000 nM T20251 CBRF87 89470690 IC50 > 60000 nM T20251 C7B8OH 89470730 IC50 > 60000 nM T20251 CHUO79 89471082 IC50 > 60000 nM T20251 CDQ8C6 89471114 IC50 = 40000 nM T20251 C4G5LP 89471136 IC50 > 60000 nM T20251 CX1DZ3 89471497 IC50 = 32000 nM T20251 CX1MA3 89471556 IC50 = 26000 nM T20251 CGY2Z5 89486768 IC50 = 1600 nM T20251 CQCJ02 89512686 Ki > 10000 nM T20251 C1CR9M 89512731 Ki = 2950 nM T20251 CTE1L0 89517065 IC50 = 1600 nM T20251 C56KSC 89517226 IC50 = 26000 nM T20251 CP8X3E 89573118 IC50 > 10000 nM T20251 C71QCV 89582842 Ki = 4100 nM T20251 C47HED 89583208 IC50 > 10000 nM T20251 C83JRE 89583782 IC50 > 60000 nM T20251 C1ZPE2 89583933 IC50 = 2100 nM T20251 CU74LB 89584002 IC50 = 3300 nM T20251 CBQ8J0 89584012 IC50 = 5300 nM T20251 CR0P6K 89584034 IC50 = 9100 nM T20251 C4NZW1 89584050 IC50 = 3300 nM T20251 CZOJ21 89584118 IC50 = 19000 nM T20251 CC94YO 89584863 Ki = 3800 nM T20251 CNZ2I8 89584875 Ki = 26900 nM T20251 CIBL54 89584906 Ki = 3000 nM T20251 CQY4J1 89584935 Ki = 19000 nM T20251 CP4T5E 89619103 IC50 = 5900 nM T20251 C89MLI 89619107 IC50 = 10000 nM T20251 CZ1A3U 89619266 IC50 = 12300 nM T20251 C7T9GQ 89633340 IC50 = 75900 nM T20251 C4D3MX 89633347 IC50 = 41500 nM T20251 CXPV63 89633380 IC50 = 10000 nM T20251 CRWG69 89633382 IC50 > 10000 nM T20251 CX4MP3 89633392 IC50 > 90000 nM T20251 C5FZ4E 89633466 IC50 = 33700 nM T20251 CX90VG 89691439 IC50 > 10000 nM T20251 CXR3A4 89702226 IC50 > 10000 nM T20251 CA49UY 89726151 IC50 > 10000 nM T20251 CIXB02 89738547 IC50 > 10000 nM T20251 C9X3MF 89752438 IC50 = 7600 nM T20251 CF5RQ7 89762819 IC50 = 18000 nM T20251 C8MN9K 89763714 IC50 = 1100 nM T20251 C5MR9K 89777151 IC50 > 33000 nM T20251 CI57QV 89782019 IC50 > 30000 nM T20251 C7TRY9 89844945 IC50 > 80000 nM T20251 CE2Z4C 89845025 IC50 > 80000 nM T20251 CTP94N 89845031 IC50 > 80000 nM T20251 C5RAI0 89907349 IC50 = 17000 nM T20251 CP0GY3 89908140 IC50 = 1800 nM T20251 C0JA2V 89908303 IC50 = 1500 nM T20251 CJW7L6 89908440 IC50 > 30000 nM T20251 CN76VK 89912923 IC50 = 15848.93 nM T20251 C2MPT3 89954418 IC50 > 10000 nM T20251 C54XDY 89975061 IC50 = 110 nM T20251 C5YEP2 89992279 IC50 = 4900 nM T20251 C8P1SX 89992280 IC50 > 10000 nM T20251 C0R6LF 89992295 IC50 = 3200 nM T20251 C63CJN 89992309 IC50 = 8900 nM T20251 CQ5HZ7 89996234 IC50 > 30000 nM T20251 CAKV98 89997377 Ki > 10000 nM T20251 CIBY41 89997417 Ki = 11700 nM T20251 C8Z9QB 89997423 Ki = 2950 nM T20251 C4PT6B 89997503 Ki > 10000 nM T20251 CB7L1N 89997512 Ki > 10000 nM T20251 CE7PH6 89997520 Ki > 10000 nM T20251 C52QPK 89997526 Ki = 145 nM T20251 C90TSY 89997709 Ki > 15000 nM T20251 C2SJY8 89997744 Ki > 10000 nM T20251 CFYO09 89997799 Ki > 10000 nM T20251 C7Z1GY 89997802 Ki > 15000 nM T20251 C89LAZ 89997856 Ki > 15000 nM T20251 C5EQM4 89997906 Ki = 377 nM T20251 C7M5KB 89997911 Ki > 15000 nM T20251 CXP2Q5 89997939 Ki = 797 nM T20251 CX4S6M 89997948 Ki = 90 nM T20251 COR4F3 89997978 Ki > 15000 nM T20251 CDI4P0 89997990 Ki > 15000 nM T20251 C9TG4Q 89998018 Ki > 10000 nM T20251 CN0DA6 89998034 Ki = 210 nM T20251 CD1VM9 89998106 Ki > 10000 nM T20251 CT38QK 89998122 Ki > 10000 nM T20251 CMO1B0 89998184 Ki = 259 nM T20251 CZ5QN1 89998216 Ki = 3810 nM T20251 C7NA0W 89998237 Ki > 10000 nM T20251 CRTP06 90000797 IC50 > 30000 nM T20251 C0NM2P 90001216 IC50 > 30000 nM T20251 C1RDQ2 90043471 IC50 > 30000 nM T20251 C3CYP0 90043482 IC50 > 30000 nM T20251 CAM93E 90043622 IC50 > 10000 nM T20251 CJ4KS1 90043633 IC50 > 10000 nM T20251 CY82BX 90044129 IC50 > 30000 nM T20251 CG5P9A 90153688 IC50 = 2500 nM T20251 CV6H7R 90153809 IC50 = 38000 nM T20251 CE7N6F 90265032 IC50 = 16600 nM T20251 C0M7NI 90268057 IC50 = 1551 nM T20251 CY5P6I 90268061 IC50 = 16940 nM T20251 CP0X1V 90311949 IC50 = 14400 nM T20251 C75FLG 90326903 IC50 = 19700 nM T20251 C26LKW 90341025 IC50 > 30000 nM T20251 C9UZX2 90355303 IC50 = 1700 nM T20251 CTO87I 90355486 IC50 = 8500 nM T20251 CB1P9Y 90355676 IC50 = 2400 nM T20251 C03ZXF 90355716 IC50 = 17700 nM T20251 CDN1X8 90366524 IC50 = 6100 nM T20251 CTV52A 90367281 IC50 = 3000 nM T20251 CA47VK 90408538 IC50 > 10000 nM T20251 CE4IT5 90408860 IC50 > 3000 nM T20251 CB0RP3 90410604 IC50 > 10000 nM T20251 CQ8ZW3 90410911 IC50 > 10000 nM T20251 CD5W6K 90417914 IC50 = 7300 nM T20251 CDJ1R8 90418278 IC50 > 50000 nM T20251 CV9HL2 90420193 IC50 = 15000 nM T20251 CTZY03 90420346 IC50 > 11000 nM T20251 C1X7PZ 90420407 IC50 = 2900 nM T20251 CX3AU6 90420765 IC50 > 33000 nM T20251 CL4WR9 90465846 IC50 = 11700 nM T20251 CJE7P5 90467013 IC50 > 33000 nM T20251 CX6DQ4 90467014 IC50 > 33000 nM T20251 C7D2UK 90467156 IC50 > 33000 nM T20251 CV75ZC 90467159 IC50 > 33000 nM T20251 C3RO1M 90467162 IC50 > 33000 nM T20251 C6BID5 90469437 IC50 > 10000 nM T20251 CW61DN 90488999 IC50 = 7400 nM T20251 CF30KA 90643570 IC50 = 31000 nM T20251 C2CE9A 90643781 Ki = 2000 nM T20251 C05MTO 90643782 Ki = 620 nM T20251 C6RM2B 90643783 Ki > 10000 nM T20251 CPD10X 90643784 Ki > 10000 nM T20251 CUB0Q1 90643785 Ki > 10000 nM T20251 CPN65E 90643787 IC50 > 30000 nM T20251 C1HGB2 90644097 IC50 = 5300 nM T20251 C83UOX 90644098 IC50 = 26000 nM T20251 C3BM4E 90644099 IC50 = 69000 nM T20251 C5VTU0 90644100 IC50 = 50600 nM T20251 CICV18 90644101 IC50 = 10000 nM T20251 CIM7G0 90644102 IC50 = 33000 nM T20251 CFB56D 90644103 IC50 = 2500 nM T20251 C1D4UG 90644104 IC50 = 74000 nM T20251 CV0X9O 90644105 IC50 = 12000 nM T20251 C8Y2XF 90644106 IC50 = 69000 nM T20251 CG48ID 90644107 IC50 = 13000 nM T20251 CZ8BP9 90644108 IC50 > 100000 nM T20251 CKAB34 90644109 IC50 > 100000 nM T20251 C13AEC 90644110 IC50 = 133000 nM T20251 C87MOQ 90644111 IC50 = 90000 nM T20251 CUK9C4 90644112 IC50 = 151000 nM T20251 CW7K6S 90644113 IC50 > 100000 nM T20251 CQJ1C8 90644114 IC50 > 100000 nM T20251 C4MHY0 90644115 IC50 > 100000 nM T20251 C6TR0K 90644116 IC50 > 100000 nM T20251 CCJQ83 90644117 IC50 > 100000 nM T20251 C3JMQ9 90644367 IC50 = 2750 nM T20251 CMV2F4 90644368 IC50 = 17000 nM T20251 CGN7C6 90644461 IC50 > 100000 nM T20251 C7R3QG 90644462 IC50 > 100000 nM T20251 CI62FU 90644463 IC50 > 100000 nM T20251 C9R6LO 90644464 IC50 > 33000 nM T20251 C8TK5D 90644465 IC50 = 16000 nM T20251 CBT08V 90644466 IC50 > 33000 nM T20251 CU9K6R 90644467 IC50 > 33000 nM T20251 CB12SV 90644468 IC50 > 33000 nM T20251 C7WIM0 90644678 IC50 = 18000 nM T20251 C5O8HN 90644762 IC50 > 10500 nM T20251 CZ5YK9 90644763 IC50 > 33300 nM T20251 CUK5T1 90644764 IC50 > 33300 nM T20251 CIHE96 90644765 IC50 > 33300 nM T20251 CY4PB3 90644766 IC50 > 33300 nM T20251 CVUE08 90644767 IC50 > 33300 nM T20251 CV79BJ 90644768 IC50 > 33300 nM T20251 CL5UB3 90644769 IC50 > 33300 nM T20251 C6AMK9 90644770 IC50 = 16600 nM T20251 CK84IG 90644771 IC50 = 3500 nM T20251 CQVY70 90644772 IC50 = 4500 nM T20251 CAVN86 90644773 IC50 = 12200 nM T20251 CPS9I2 90644774 IC50 = 10300 nM T20251 C1VU8Q 90644775 IC50 = 22000 nM T20251 CMQ30B 90644776 IC50 = 25000 nM T20251 C6FL9K 90644777 IC50 > 33300 nM T20251 CXSJ16 90644778 IC50 > 33300 nM T20251 CV3C5H 90644779 IC50 = 60000 nM T20251 C0KQV4 90645474 IC50 = 135 nM T20251 CE8AI2 90654467 IC50 = 920 nM T20251 CV87PR 90655950 IC50 > 40000 nM T20251 C62SML 90655967 IC50 > 33000 nM T20251 CJ7LT3 90655968 IC50 > 33000 nM T20251 CB61WC 90655969 IC50 > 33000 nM T20251 CK6QN4 90656025 IC50 > 50000 nM T20251 CO73FL 90656026 IC50 > 50000 nM T20251 COW7U5 90656027 IC50 = 3100 nM T20251 CV9H8U 90656285 IC50 > 30000 nM T20251 CDF9O2 90656287 IC50 = 8200 nM T20251 CIL2W9 90664452 IC50 = 9800 nM T20251 C4MUI2 90664601 IC50 = 8110 nM T20251 CA79EY 90664683 IC50 = 1700 nM T20251 CTR58M 90664931 IC50 = 1000 nM T20251 CHT7D5 90664962 IC50 > 10000 nM T20251 C01UNB 90665166 Ki = 3760 nM T20251 CXJ62T 90665173 IC50 = 900 nM T20251 CG98QO 90665194 IC50 = 1300 nM T20251 CJCR26 90665456 IC50 = 9670 nM T20251 C71ARQ 90665737 IC50 = 22000 nM T20251 CZOW03 90665738 IC50 = 4000 nM T20251 CVJE69 90665739 IC50 = 59000 nM T20251 CG4E8W 90665845 IC50 = 8700 nM T20251 C1S7YU 90665846 IC50 = 2100 nM T20251 C8B1RN 90665847 IC50 = 3500 nM T20251 CCQ67W 90665848 IC50 = 2100 nM T20251 C2DF8V 90665849 IC50 = 3700 nM T20251 CGB7U8 90665850 IC50 = 2500 nM T20251 C67YNO 90665851 IC50 > 10000 nM T20251 C2E6NI 90665852 IC50 > 8300 nM T20251 C1X2PV 90665949 IC50 = 18000 nM T20251 CKY18S 90665950 IC50 > 28000 nM T20251 CDQ56W 90665987 IC50 > 10000 nM T20251 C97PUB 90666011 IC50 = 11000 nM T20251 CU9OP3 90666012 IC50 = 10000 nM T20251 C8O2ZM 90666013 IC50 = 15000 nM T20251 C3ND7I 90666014 IC50 = 22000 nM T20251 CSJE46 90666015 IC50 = 21000 nM T20251 C6W4GH 90666017 IC50 = 47000 nM T20251 C0D5FT 90666018 IC50 = 43000 nM T20251 CMX8H0 90666019 IC50 > 100000 nM T20251 C4AP0G 90666024 IC50 = 44000 nM T20251 C5WQN4 90666035 IC50 = 2900 nM T20251 C85AMH 90666036 IC50 = 3200 nM T20251 CKF14A 90666037 IC50 = 12000 nM T20251 CM7ED5 90666038 IC50 = 4100 nM T20251 CU2T3C 90666039 IC50 = 14000 nM T20251 C59YXE 90666040 IC50 = 7300 nM T20251 C6QZL4 90666041 IC50 = 6800 nM T20251 CY35OV 90666042 IC50 = 8400 nM T20251 C2IN9R 90666094 IC50 = 1970 nM T20251 CMU2J7 90666098 IC50 = 1700 nM T20251 CU9MV6 90666148 IC50 = 18000 nM T20251 CC07QH 90666256 IC50 = 1200 nM T20251 C6H5CY 90666260 IC50 = 1900 nM T20251 C45NLU 90666267 IC50 = 1700 nM T20251 C5VZC6 90666479 IC50 = 2200 nM T20251 CQ23WR 90667215 IC50 = 13000 nM T20251 CGP3C6 90667419 IC50 = 18300 nM T20251 CF6MO3 90667420 IC50 = 1280 nM T20251 CCO96L 90667421 IC50 = 4920 nM T20251 CIW51L 90667423 IC50 = 86200 nM T20251 CG2J7Y 90667424 IC50 = 92100 nM T20251 CC7G4Q 90667584 IC50 = 210 nM T20251 CW5UZ9 90667585 IC50 = 1280 nM T20251 CGX4S0 90667586 IC50 = 390 nM T20251 CK4GF3 90667587 IC50 = 37 nM T20251 C9XVG4 90667588 IC50 = 174 nM T20251 C08COA 90667590 IC50 = 93600 nM T20251 C7BK1O 90667600 IC50 = 81700 nM T20251 CZL03G 90667602 IC50 = 107 nM T20251 CR59JY 90667603 IC50 = 75800 nM T20251 CGRK73 90667608 IC50 = 1270 nM T20251 C2ZN9Y 90667609 IC50 > 100000 nM T20251 CT5H7A 90667610 IC50 = 160 nM T20251 CTD7C6 90667611 IC50 = 480 nM T20251 CIM1S7 90667868 IC50 > 100000 nM T20251 CT2GU1 91246771 IC50 = 10700 nM T20251 CYHR27 91664373 IC50 > 10000 nM T20251 CUI10E 91666686 IC50 = 19600 nM T20251 C76AKI 91754444 IC50 = 81000 nM T20251 C7EXH8 91755097 IC50 > 80000 nM T20251 C37IZB 91755098 IC50 = 18000 nM T20251 CX4DJ7 91799322 IC50 = 800 nM T20251 C90JVH 91799688 IC50 = 49 nM T20251 CGJ6S0 91801175 IC50 > 60000 nM T20251 CK6E0W 91810397 IC50 = 48000 nM T20251 CC9B6T 91820646 IC50 = 28000 nM T20251 C3L6KU 91820689 IC50 > 40000 nM T20251 CDT6C1 91824787 Ki = 6251 nM T20251 CK5X2M 91826235 IC50 = 23000 nM T20251 C9MO7C 91826722 IC50 = 4300 nM T20251 C64QCZ 91827500 IC50 = 501.19 nM T20251 CL7S4U 91844670 IC50 > 50000 nM T20251 CSK6Z1 91844707 IC50 = 5290 nM T20251 CRX16J 91884611 IC50 = 4050 nM T20251 CBG6E7 91885506 IC50 > 10000 nM T20251 CFT9N5 91885578 IC50 = 20000 nM T20251 CU1G3S 91933941 IC50 > 30000 nM T20251 CQN41K 91938095 Ki = 1732 nM T20251 CWZX73 91971958 IC50 = 5100 nM T20251 CYMH49 92044895 IC50 > 20000 nM T20251 C38ZID 92045057 IC50 > 10000 nM T20251 CEJK10 92135927 IC50 = 21000 nM T20251 CCY0O2 100951644 IC50 > 33300 nM T20251 CNQ6J9 101873336 Ki = 7048 nM T20251 C0QXE2 101882778 IC50 = 400 nM T20251 C05NTY 101884761 IC50 = 4000 nM T20251 CWM71R 101884762 IC50 = 6700 nM T20251 C4KH1V 101886593 IC50 = 210 nM T20251 C2EJK6 101910737 IC50 = 6980 nM T20251 CB5DK1 102004349 IC50 = 400 nM T20251 CQ9PN8 102593934 IC50 > 30000 nM T20251 C4Z1OU 110451319 IC50 > 25000 nM T20251 CN57AX 110451673 IC50 > 25000 nM T20251 C8F6VO 117604931 IC50 > 100000 nM T20251 C6UOT8 117653759 IC50 = 17000 nM T20251 C8ZM9J 117678530 IC50 = 3200 nM T20251 C5CL8X 117684497 IC50 = 3500 nM T20251 C4O3VF 117689963 IC50 = 26800 nM T20251 CT7GW0 117690258 IC50 = 19700 nM T20251 CX0DY2 117690263 IC50 = 17600 nM T20251 CQF32S 117690304 IC50 = 8900 nM T20251 C15QUL 117690396 IC50 = 53400 nM T20251 CFT94I 117700435 IC50 > 10000 nM T20251 CG60JW 117700665 IC50 = 3130 nM T20251 C3GB4X 117715778 IC50 > 50000 nM T20251 C2TG7Y 117715783 IC50 = 6900 nM T20251 CW8RS3 117760464 Ki > 30000 nM T20251 CZC84D 117769161 IC50 = 10200 nM T20251 CE7BZ8 117769174 IC50 = 8500 nM T20251 CBJ07Q 117769217 IC50 > 80000 nM T20251 CXHQ08 117769229 IC50 = 7200 nM T20251 CS9WO4 117769234 IC50 = 7700 nM T20251 C1SA9I 117769244 IC50 = 35000 nM T20251 C0VY7C 117769271 IC50 = 7500 nM T20251 CSR9B0 117769289 IC50 = 5300 nM T20251 C2M9CR 117769307 IC50 = 41000 nM T20251 C7FWS3 117769309 IC50 = 12000 nM T20251 CYWV32 117769339 IC50 = 4100 nM T20251 CZV35K 117769346 IC50 > 80000 nM T20251 C5V6RG 117769349 IC50 > 80000 nM T20251 C4O1PX 117769362 IC50 = 7600 nM T20251 CPV4C8 117769365 IC50 = 13800 nM T20251 CP3MC5 117769379 IC50 = 9600 nM T20251 C8V6LG 117769392 IC50 = 8000 nM T20251 C2NBZ8 117769396 IC50 = 6000 nM T20251 COV59Y 117769408 IC50 = 4900 nM T20251 CXJ3I6 117769409 IC50 = 17000 nM T20251 C8LTZ6 117769464 IC50 > 80000 nM T20251 CSKO30 117769533 IC50 = 5000 nM T20251 C6XC3W 117769575 IC50 = 300 nM T20251 C8Y5ZX 117778486 IC50 = 9500 nM T20251 CDUH09 117809287 IC50 = 30000 nM T20251 C3FY8A 117838708 IC50 = 7800 nM T20251 C7VDL3 117838709 IC50 = 30000 nM T20251 C0BI1C 117838710 IC50 = 13500 nM T20251 CBD0X6 117852205 IC50 = 29600 nM T20251 CN5H7Y 117852210 IC50 = 7900 nM T20251 CB9X7D 117852213 IC50 = 6100 nM T20251 CTKJ90 117852221 IC50 = 1200 nM T20251 C3PST8 117852226 IC50 = 193 nM T20251 CN8G6X 117852236 IC50 = 2400 nM T20251 C3SW9X 117852238 IC50 = 3290 nM T20251 CO3X7N 117852239 IC50 > 60000 nM T20251 C17KYZ 117852241 IC50 = 17400 nM T20251 CI06AN 117852248 IC50 = 10500 nM T20251 C3K8XU 117852302 IC50 = 1800 nM T20251 CMS0A3 117852327 IC50 = 16100 nM T20251 C04UHW 117852380 IC50 = 2400 nM T20251 CQ4FJ5 117852383 IC50 = 8900 nM T20251 C0A4XC 117871929 IC50 = 2900 nM T20251 CV4B2W 117871992 IC50 > 60000 nM T20251 CY5JF0 117872250 IC50 = 6100 nM T20251 COIM28 117872315 IC50 > 60000 nM T20251 C7PM6F 117872316 IC50 = 5200 nM T20251 C6X8VS 117872368 IC50 = 40000 nM T20251 CQ5S7L 117872990 IC50 = 1900 nM T20251 C9OA4U 117873033 IC50 = 25000 nM T20251 CL6QV4 117873045 IC50 = 12000 nM T20251 C6XS8J 117887024 IC50 = 2300 nM T20251 CP0I7M 117887098 IC50 = 1200 nM T20251 CA7Z3W 117887511 IC50 = 1600 nM T20251 CFV23K 117887619 IC50 = 700 nM T20251 C89EQN 117897570 IC50 = 20200 nM T20251 C4CH7J 117955548 IC50 = 240 nM T20251 C07ACT 117955744 IC50 = 3700 nM T20251 CK53MQ 117972250 IC50 = 380 nM T20251 C9KV7L 117993993 Ki > 30000 nM T20251 CNV24M 117993998 Ki > 30000 nM T20251 CS16CJ 118022791 IC50 = 11400 nM T20251 C89WQL 118023142 IC50 = 6800 nM T20251 CFE6M2 118038416 IC50 > 10000 nM T20251 C2WQ4G 118039220 IC50 = 260 nM T20251 CTU3K2 118043167 IC50 > 10000 nM T20251 CPU7C0 118043263 IC50 = 10000 nM T20251 CR2XJ5 118043265 IC50 = 3300 nM T20251 C4HQ5C 118043312 IC50 = 1500 nM T20251 CB4A6H 118043313 IC50 > 10000 nM T20251 C45RCJ 118072307 IC50 > 80000 nM T20251 CH7LT6 118072319 IC50 > 80000 nM T20251 CUQ85I 118102658 IC50 > 30000 nM T20251 CMX3U8 118107483 IC50 = 1400 nM T20251 C5R1XP 118107577 IC50 > 10000 nM T20251 C91QJN 118107589 IC50 > 10000 nM T20251 C9JE0K 118107598 IC50 > 10000 nM T20251 C3ID1F 118111696 IC50 = 300 nM T20251 CD48WH 118121169 IC50 = 4500 nM T20251 C3F6XG 118165440 IC50 = 4000 nM T20251 CDAC50 118165497 IC50 = 6300 nM T20251 CN4O5K 118165763 IC50 = 2800 nM T20251 C0TMZ8 118167692 IC50 = 14000 nM T20251 C68QVN 118167694 IC50 = 24000 nM T20251 CSM69G 118167758 IC50 = 4200 nM T20251 C9EY8L 118167812 IC50 = 6500 nM T20251 CP8QO0 118179807 IC50 > 100000 nM T20251 CT4G5D 118179817 IC50 > 100000 nM T20251 CIU02H 118179819 IC50 = 100000 nM T20251 C4KC7H 118189484 IC50 = 9000 nM T20251 C5DYL3 118189493 IC50 = 7000 nM T20251 CLH8X7 118189551 IC50 = 9500 nM T20251 CAI09J 118195093 IC50 > 30000 nM T20251 CZ5G7W 118195200 IC50 = 4200 nM T20251 C0NM1V 118195331 IC50 = 1500 nM T20251 C3J4UQ 118198923 IC50 = 310 nM T20251 CV67TP 118207324 IC50 = 400 nM T20251 CPZ69K 118207398 IC50 > 30000 nM T20251 CG84LB 118207404 IC50 = 620 nM T20251 C1GH3R 118207538 IC50 = 7800 nM T20251 C91ECG 118217204 IC50 > 5000 nM T20251 CV16QJ 118217208 IC50 > 30000 nM T20251 CL5C4K 118253824 IC50 > 33000 nM T20251 CCH97D 118253857 IC50 = 17000 nM T20251 CCG7Y6 118253883 IC50 = 31000 nM T20251 CA72QZ 118253888 IC50 > 33000 nM T20251 CZ3U4P 118270292 IC50 = 3380 nM T20251 C3E5PL 118307312 IC50 = 3290 nM T20251 C93OPR 118307317 IC50 = 12400 nM T20251 CIY0X1 118307334 IC50 = 20100 nM T20251 CD93MJ 118307348 IC50 = 3510 nM T20251 C89TZG 118307431 IC50 > 30000 nM T20251 CKG4L3 118334971 IC50 = 2100 nM T20251 CRV14T 118334974 IC50 = 500 nM T20251 C7VYK2 118334975 IC50 = 200 nM T20251 CIS2L9 118334979 IC50 = 2000 nM T20251 CKM6L0 118334982 IC50 = 900 nM T20251 CH8PU2 118334995 IC50 = 500 nM T20251 C1TF9K 118368174 IC50 = 22000 nM T20251 CBIR89 118389918 IC50 = 15600 nM T20251 CRHY82 118409479 IC50 > 30000 nM T20251 CO75VB 118409494 IC50 > 30000 nM T20251 C3FVW7 118409564 IC50 > 30000 nM T20251 CW3IC5 118414671 IC50 = 30000 nM T20251 C94WRZ 118435363 IC50 = 9300 nM T20251 C1WL4E 118435382 IC50 = 23600 nM T20251 C5L9VH 118435403 IC50 = 12100 nM T20251 CNXH97 118435407 IC50 = 9000 nM T20251 C8Z2FP 118435412 IC50 = 10700 nM T20251 CJIP45 118435414 IC50 = 10100 nM T20251 CY6EP7 118435506 IC50 = 43000 nM T20251 CPE35X 118435524 IC50 = 9600 nM T20251 CVK6Y8 118435560 IC50 = 11700 nM T20251 CN5L8K 118435601 IC50 = 13100 nM T20251 C37SFM 118435617 IC50 = 17900 nM T20251 CZLJ20 118441559 IC50 = 400 nM T20251 CR9QF7 118441560 IC50 = 11970 nM T20251 CEMZ15 118464420 IC50 > 1000 nM T20251 CRV8S3 118478927 IC50 > 10000 nM T20251 CL32JE 118478933 IC50 > 10000 nM T20251 C5S1HZ 118478972 IC50 > 10000 nM T20251 C8G9HP 118478986 IC50 > 10000 nM T20251 CBV89G 118478994 IC50 > 10000 nM T20251 CK0ER5 118478999 IC50 > 10000 nM T20251 CU25KC 118479000 IC50 > 10000 nM T20251 CW07IS 118479006 IC50 = 6700 nM T20251 C3ZAV0 118479034 IC50 > 10000 nM T20251 C4W6ZS 118479038 IC50 > 10000 nM T20251 CRG24C 118479053 IC50 > 10000 nM T20251 CD4ME1 118479123 IC50 > 10000 nM T20251 CB0XM2 118479161 IC50 > 10000 nM T20251 C18NTQ 118479199 IC50 = 10000 nM T20251 CJ0Z1Y 118479222 IC50 > 10000 nM T20251 CP0U6Y 118479229 IC50 > 10000 nM T20251 C3A6HD 118479231 IC50 > 10000 nM T20251 CJ14CR 118479241 IC50 = 9900 nM T20251 C1FO3N 118479293 IC50 = 4300 nM T20251 CF02TZ 118479295 IC50 = 10000 nM T20251 C90TED 118479305 IC50 = 10000 nM T20251 C7I9RC 118479316 IC50 > 10000 nM T20251 CRC4F6 118479354 IC50 > 10000 nM T20251 CRCV51 118479359 IC50 > 10000 nM T20251 CJL5W0 118479428 IC50 > 10000 nM T20251 CS2VA7 118479440 IC50 > 10000 nM T20251 CJ9P0M 118479445 IC50 = 6900 nM T20251 C3U1RB 118479452 IC50 = 4500 nM T20251 CBJ28X 118483320 IC50 > 30000 nM T20251 C0KPH4 118485600 IC50 = 160 nM T20251 C43GZF 118485601 IC50 = 980 nM T20251 C8UT1Z 118485623 IC50 = 610 nM T20251 CC94IQ 118485651 IC50 = 4900 nM T20251 CMK97G 118491864 IC50 = 9000 nM T20251 C62FCZ 118491902 IC50 = 6000 nM T20251 CD57MP 118491918 IC50 > 30000 nM T20251 C05LQH 118498627 IC50 > 33000 nM T20251 CXCF46 118498683 IC50 > 33000 nM T20251 CJA07S 118498727 IC50 > 33000 nM T20251 CG6D1J 118498935 IC50 = 27000 nM T20251 CXR46C 118499887 IC50 > 33000 nM T20251 CFVN15 118500050 IC50 > 33000 nM T20251 CY9NW0 118500097 IC50 > 33000 nM T20251 CXEI18 118500108 IC50 > 33000 nM T20251 CL2Z5Y 118502821 IC50 = 22000 nM T20251 CVY64N 118502892 IC50 > 33000 nM T20251 CO20ET 118502895 IC50 = 14000 nM T20251 CU1X3H 118502919 IC50 > 33000 nM T20251 CK04PJ 118512792 IC50 = 4670 nM T20251 C48PFK 118512802 IC50 = 14500 nM T20251 C76UQN 118512804 IC50 = 1600 nM T20251 CAKI19 118514811 IC50 = 8460 nM T20251 C0R2MP 118519041 IC50 > 30000 nM T20251 CRAF61 118523357 IC50 > 33000 nM T20251 C5P7VH 118523411 IC50 = 18000 nM T20251 CD0EY5 118523423 IC50 > 33000 nM T20251 C7AYV5 118540795 Ki = 1091 nM T20251 CG19TS 118554552 IC50 > 33300 nM T20251 CU02NF 118559124 IC50 = 7570 nM T20251 CB41MH 118560618 IC50 = 5500 nM T20251 C5CDE0 118562359 IC50 = 600 nM T20251 CS63OE 118562362 IC50 = 1100 nM T20251 C60BSA 118562375 IC50 = 1200 nM T20251 CE3D0A 118562384 IC50 = 800 nM T20251 C7IVW9 118562402 IC50 = 8200 nM T20251 CE53DJ 118562440 IC50 = 600 nM T20251 CW26NV 118562451 IC50 = 300 nM T20251 C7G5HO 118562469 IC50 = 200 nM T20251 C5JKQ9 118562510 IC50 = 400 nM T20251 CF6LK7 118562538 IC50 = 1200 nM T20251 C6FOS9 118562556 IC50 = 1000 nM T20251 C25MXS 118562567 IC50 = 100 nM T20251 CJF1E6 118562576 IC50 = 100 nM T20251 C5QB2S 118562584 IC50 = 1200 nM T20251 C6TC3D 118562598 IC50 = 2000 nM T20251 CWA4B2 118562606 IC50 = 100 nM T20251 C2EPN1 118565438 IC50 = 600 nM T20251 C0XIN5 118567313 IC50 = 1900 nM T20251 C6PA1C 118567531 IC50 = 6600 nM T20251 CD4XK8 118567534 IC50 = 500 nM T20251 CLVO18 118567538 IC50 = 3300 nM T20251 C1CP6Z 118567543 IC50 > 10000 nM T20251 C32PGF 118567545 IC50 = 3800 nM T20251 C7G8IT 118567547 IC50 = 1100 nM T20251 CXW0K9 118567604 IC50 = 1200 nM T20251 C4ULH8 118567605 IC50 = 100 nM T20251 C8TP7C 118567608 IC50 = 1000 nM T20251 CI0JY2 118567747 IC50 = 1200 nM T20251 C78LNX 118572065 IC50 > 100000 nM T20251 COYJ84 118575663 IC50 > 25000 nM T20251 CSW92P 118607432 IC50 > 100000 nM T20251 CM93VO 118611725 IC50 = 8000 nM T20251 CE69HN 118613626 IC50 > 100000 nM T20251 C2EQ9X 118613653 IC50 > 100000 nM T20251 C1X8GW 118613658 IC50 > 100000 nM T20251 CVE4S5 118627059 IC50 = 1180 nM T20251 CL74GH 118665602 IC50 = 35000 nM T20251 CP71CK 118665611 IC50 = 38000 nM T20251 CR3F5V 118665613 IC50 = 29000 nM T20251 C60TWO 118665627 IC50 = 42000 nM T20251 CY7T8F 118665628 IC50 = 38000 nM T20251 CBZ59D 118701008 IC50 = 1800 nM T20251 CRS34C 118705500 IC50 > 100000 nM T20251 C2WP6X 118706538 IC50 = 1410 nM T20251 CZE4U0 118706539 IC50 = 1460 nM T20251 CP6O2R 118706799 IC50 = 190 nM T20251 C2O7GE 118707553 IC50 = 31200 nM T20251 C8S9VW 118707562 IC50 = 12900 nM T20251 C9BCT8 118707596 IC50 = 21100 nM T20251 C62JCD 118707597 IC50 = 20700 nM T20251 C8CXM5 118707599 IC50 = 22000 nM T20251 CC0VX1 118707602 IC50 = 59500 nM T20251 CN2IC3 118707603 IC50 = 19900 nM T20251 CH9MA5 118707606 IC50 = 40500 nM T20251 CRNF04 118709230 IC50 = 7000 nM T20251 CARX10 118709238 IC50 > 30000 nM T20251 CQ65IH 118709240 IC50 > 30000 nM T20251 CG96QP 118709241 IC50 = 3300 nM T20251 C8QO1J 118709242 IC50 > 30000 nM T20251 CBK73W 118709243 IC50 > 30000 nM T20251 C35GDB 118709244 IC50 > 30000 nM T20251 CI9Q7O 118709245 IC50 > 30000 nM T20251 CD0B1Z 118709246 IC50 > 30000 nM T20251 CMX6S5 118709259 IC50 > 60000 nM T20251 CM64SW 118709261 IC50 = 4800 nM T20251 C7WY2D 118709262 IC50 = 10000 nM T20251 CN25PF 118709263 IC50 = 7000 nM T20251 CU25HN 118709264 IC50 = 1000 nM T20251 CQOS43 118709267 IC50 = 1000 nM T20251 CXH06J 118709268 IC50 = 4500 nM T20251 CFZV13 118709269 IC50 = 1400 nM T20251 CTJ0H1 118709270 IC50 = 1200 nM T20251 CP9W5U 118709272 IC50 = 10000 nM T20251 C15VXF 118709274 IC50 = 1400 nM T20251 CXFS23 118709275 IC50 > 33000 nM T20251 CJ5C4D 118709276 IC50 = 2000 nM T20251 C7O1JS 118709277 IC50 = 1800 nM T20251 C1CUQ5 118709784 IC50 = 3500 nM T20251 CFN94L 118709786 IC50 = 12700 nM T20251 C32EZA 118709832 IC50 = 21500 nM T20251 CSL13X 118709837 IC50 = 7300 nM T20251 CV26JZ 118709848 IC50 = 8800 nM T20251 CFC1J5 118710523 IC50 = 707 nM T20251 C4X8NC 118710524 IC50 = 625 nM T20251 CK3WG9 118710525 IC50 = 1420 nM T20251 C4NIK8 118710526 IC50 = 1205 nM T20251 C3JAX9 118710527 IC50 = 2257 nM T20251 CXV1C5 118710528 IC50 = 2520 nM T20251 CA5TR0 118710529 IC50 = 1611 nM T20251 CX9Q7Z 118710530 IC50 = 2845 nM T20251 C27IPK 118710531 IC50 = 8703 nM T20251 C9AZ1B 118710534 IC50 = 11990 nM T20251 C0YL9Z 118710536 IC50 = 95600 nM T20251 CD34IY 118710582 IC50 = 1000 nM T20251 CYP20X 118711743 Ki = 7050 nM T20251 C47GVE 118711875 Ki = 6250 nM T20251 C2IUO5 118711883 Ki > 10000 nM T20251 C4MP7C 118711884 Ki > 10000 nM T20251 CD9E1M 118711886 Ki > 10000 nM T20251 C5A4XS 118712578 IC50 = 209000 nM T20251 CP2S6F 118712580 IC50 = 25000 nM T20251 C4T2FY 118712775 IC50 = 97700 nM T20251 C5M3BX 118712788 IC50 = 55300 nM T20251 CN4XM2 118713119 IC50 = 14000 nM T20251 C84GOU 118713773 IC50 = 4710 nM T20251 C2LY9D 118713799 IC50 = 1880 nM T20251 CMO2V7 118713801 IC50 = 5500 nM T20251 C9IXE6 118715640 IC50 = 41000 nM T20251 CMN87B 118716079 IC50 > 33000 nM T20251 CC56DO 118718808 IC50 = 56000 nM T20251 CYX8Z6 118720352 Ki = 624 nM T20251 CF5HV8 118720613 IC50 = 1500 nM T20251 C2UIB7 118720614 IC50 > 30000 nM T20251 CSH50J 118720615 IC50 = 12500 nM T20251 C9Y4EH 118720886 IC50 > 30000 nM T20251 C9SF2E 118720891 IC50 > 30000 nM T20251 CY4G7A 118720929 IC50 > 100000 nM T20251 C3BXY9 118720930 IC50 > 333000 nM T20251 CQ6U9R 118720931 IC50 > 333000 nM T20251 CYO0F9 118720932 IC50 > 100000 nM T20251 CTB1R4 118720940 IC50 = 29000 nM T20251 C9IP0Z 118720958 IC50 = 4000 nM T20251 CDN58A 118720960 IC50 > 33000 nM T20251 C70UZF 118720963 IC50 = 4000 nM T20251 C4M5WY 118720964 IC50 > 33000 nM T20251 CS73GH 118720967 IC50 = 12000 nM T20251 C30QPT 118720970 IC50 > 33000 nM T20251 CQK8L9 118720972 IC50 = 400 nM T20251 C8VYR0 118721373 IC50 = 8300 nM T20251 CE90RQ 118721374 IC50 > 100000 nM T20251 C7MN6D 118721376 IC50 = 54700 nM T20251 CPC71H 118722570 IC50 = 6900 nM T20251 CTL19H 118722571 IC50 = 6400 nM T20251 C2JGB3 118722572 IC50 = 3600 nM T20251 CKD42B 118722573 IC50 = 9400 nM T20251 C6PMQ1 118722574 IC50 > 30000 nM T20251 C3ZL5Y 118722575 IC50 = 11000 nM T20251 CR3UB2 118722576 IC50 = 5700 nM T20251 CX1W8N 118722577 IC50 > 30000 nM T20251 C49DXR 118722578 IC50 = 17000 nM T20251 CW5GK1 118722579 IC50 > 30000 nM T20251 C50GXM 118722580 IC50 > 30000 nM T20251 CEI62G 118722581 IC50 = 3600 nM T20251 C9UG3Z 118722582 IC50 = 28000 nM T20251 C5XH4V 118722583 IC50 > 30000 nM T20251 C6Q3RV 118722584 IC50 > 30000 nM T20251 CCWD82 118722585 IC50 > 30000 nM T20251 CZ0DG2 118722586 IC50 > 30000 nM T20251 CI3R9V 118722587 IC50 = 7400 nM T20251 CSWJ92 118723345 IC50 = 280 nM T20251 CJ6V0G 118723355 IC50 = 3760 nM T20251 C0J7CS 118723360 IC50 = 950 nM T20251 C4X0GY 118723362 IC50 = 2610 nM T20251 CGN4Z9 118723363 IC50 = 1540 nM T20251 CQ3JF0 118723364 IC50 = 1400 nM T20251 C0LUV6 118723826 Ki > 10000 nM T20251 CXE6I5 118723827 Ki > 10000 nM T20251 CKO8P6 118723828 Ki > 10000 nM T20251 CL6CM1 118725606 IC50 = 3000 nM T20251 CUN73P 118725613 IC50 = 1100 nM T20251 CL5K0U 118725614 IC50 = 2000 nM T20251 CXEP50 118725615 IC50 = 2300 nM T20251 C1LTN0 118725864 Ki = 7800 nM T20251 CIR0O4 118725970 Ki > 15000 nM T20251 CS6BC8 118725971 Ki > 15000 nM T20251 CDV7Z0 118725972 Ki > 15000 nM T20251 CVZ9F7 118725973 Ki > 15000 nM T20251 CX9W7R 118725974 Ki > 15000 nM T20251 C1X4CO 118725975 Ki > 15000 nM T20251 C4DVC0 118725976 Ki > 15000 nM T20251 C0SO8I 118725977 Ki > 15000 nM T20251 CXH13A 118727337 IC50 = 1060 nM T20251 C6F5AX 118727347 IC50 = 40000 nM T20251 CF39TB 118727349 IC50 = 12000 nM T20251 CBIJ20 118728075 IC50 = 394000 nM T20251 CL32ES 118728076 IC50 = 12300 nM T20251 CHP59R 118728077 IC50 = 13800 nM T20251 CZY1K8 118728078 IC50 = 7300 nM T20251 COXN68 118728079 IC50 = 24500 nM T20251 C5K6YS 118728080 IC50 > 60000 nM T20251 CQ4TP6 118728081 IC50 > 60000 nM T20251 CRNU85 118728967 IC50 > 60000 nM T20251 CJ7N4U 118728968 IC50 > 60000 nM T20251 CY0GP6 118728969 IC50 > 60000 nM T20251 C46MUV 118728970 IC50 > 60000 nM T20251 CT7AV4 118728971 IC50 > 60000 nM T20251 CGY0L7 118728972 IC50 > 60000 nM T20251 CM7DW9 118728973 IC50 > 60000 nM T20251 CL38UF 118728974 IC50 = 53300 nM T20251 CPR5B4 118728975 IC50 > 60000 nM T20251 CB0AQ3 118728976 IC50 > 60000 nM T20251 CI1L8O 118730350 IC50 = 11500 nM T20251 C6HV3B 118730351 IC50 = 12900 nM T20251 CX50MI 118730679 IC50 > 10000 nM T20251 C1WFY9 118730799 IC50 = 48400 nM T20251 CQC32W 118730800 IC50 = 7600 nM T20251 CJ0IH1 118730801 IC50 = 32600 nM T20251 CN6UX9 118730802 IC50 = 28700 nM T20251 C05UZL 118730803 IC50 = 17600 nM T20251 CTJG53 118730804 IC50 = 11500 nM T20251 CQ48NV 118730805 IC50 = 10400 nM T20251 C26OMX 118730806 IC50 = 9300 nM T20251 CB47AL 118730807 IC50 = 8400 nM T20251 CNTH27 118730808 IC50 = 8400 nM T20251 CX50CM 118730809 IC50 = 45500 nM T20251 CN26ZK 118730810 IC50 = 6800 nM T20251 C2PT0H 118730811 IC50 = 2500 nM T20251 CRUA27 118730812 IC50 = 5700 nM T20251 CKJS86 118730813 IC50 = 4600 nM T20251 CQYK51 118730814 IC50 = 3400 nM T20251 C7TJQ5 118730994 IC50 = 2100 nM T20251 CV4E7S 118730999 IC50 = 1400 nM T20251 CC2I1K 118733347 IC50 = 5200 nM T20251 C1AVK5 118733348 IC50 = 42000 nM T20251 C43XUF 118733349 IC50 > 60000 nM T20251 C7XG3O 118733350 IC50 = 14000 nM T20251 CNYV64 118733351 IC50 = 1000 nM T20251 CLI96Y 118733352 IC50 = 5900 nM T20251 C5Q2VW 118733353 IC50 = 18000 nM T20251 C5YB6G 118733354 IC50 = 44000 nM T20251 CRO7S5 118733755 IC50 > 30000 nM T20251 C2XZN0 118733756 IC50 > 30000 nM T20251 C7MRW8 118733798 IC50 = 3980 nM T20251 C6VO5G 118733806 IC50 = 2000 nM T20251 CGKD16 118734983 IC50 = 50300 nM T20251 CX7H5Q 118734985 IC50 > 30000 nM T20251 CAN90V 118735353 IC50 = 4700 nM T20251 CIY1L8 118735865 IC50 = 730 nM T20251 CLOM28 118735866 IC50 = 1750 nM T20251 C1AI3Y 118735867 IC50 = 1060 nM T20251 C87IQN 118735868 IC50 = 5900 nM T20251 CAU0F9 118735870 IC50 = 1550 nM T20251 C3ES8P 118736031 IC50 = 13.91 nM T20251 CIB75P 118736034 IC50 = 1.7 nM T20251 C8XC3Y 118736035 IC50 = 12.38 nM T20251 C7CER2 118736036 IC50 = 0.89 nM T20251 CHL4E9 118736037 IC50 = 18.37 nM T20251 C0L2KD 118736038 IC50 = 3.27 nM T20251 CWX5Y3 118736039 IC50 = 4.2 nM T20251 C7B2JW 118736040 IC50 = 1.43 nM T20251 C60KVO 118736041 IC50 = 2.49 nM T20251 CV8Y9W 118736042 IC50 = 1.6 nM T20251 CEB0Q6 118736043 IC50 = 5.22 nM T20251 CG4D0N 118736044 IC50 = 4.21 nM T20251 CMK5V7 118736045 IC50 = 0.87 nM T20251 CRW2Y1 118736046 IC50 = 1.96 nM T20251 C0U1NW 118736047 IC50 = 13.09 nM T20251 CK58FE 118736048 IC50 = 2.08 nM T20251 CBMZ68 118736049 IC50 = 6.71 nM T20251 CJ95DR 118736050 IC50 = 2.29 nM T20251 CYQ3N5 118736051 IC50 = 0.99 nM T20251 C9CE2G 118736052 IC50 = 0.39 nM T20251 CUG5T3 118736053 IC50 = 15.62 nM T20251 CYR6Z9 118736054 IC50 = 4.93 nM T20251 CA18KF 118736055 IC50 = 16.75 nM T20251 C7VT6Q 118736056 IC50 = 7.87 nM T20251 CJ4AM8 118736655 IC50 = 25700 nM T20251 C37CTY 118736656 IC50 > 60000 nM T20251 CE3JA4 118736657 IC50 = 126000 nM T20251 C64UZP 118736658 IC50 > 60000 nM T20251 C0U5IX 118736659 IC50 > 60000 nM T20251 CS5WB8 118736662 IC50 = 30500 nM T20251 CPS96F 118736663 IC50 = 11700 nM T20251 CY5SC3 118736664 IC50 = 30000 nM T20251 CE37GC 118736665 IC50 = 7300 nM T20251 CNUS74 118736667 IC50 = 2600 nM T20251 CB42EV 118736668 IC50 > 60000 nM T20251 CP9D1G 118736669 IC50 > 60000 nM T20251 CY8I6E 118736670 IC50 > 60000 nM T20251 C97CJG 118736671 IC50 > 60000 nM T20251 CJH5D7 118736673 IC50 > 60000 nM T20251 C6WQ3N 118736674 IC50 > 60000 nM T20251 CVKD56 118736675 IC50 > 60000 nM T20251 CH0R6U 118736676 IC50 > 60000 nM T20251 C8IEB7 118736677 IC50 > 60000 nM T20251 CKV91L 118736679 IC50 = 16500 nM T20251 C3IM7W 118736680 IC50 > 60000 nM T20251 C1X8EJ 118736681 IC50 > 60000 nM T20251 CG52WO 118736682 IC50 > 60000 nM T20251 C9ZQH1 118736683 IC50 = 30400 nM T20251 C06IYV 118736684 IC50 = 31600 nM T20251 CRJ38C 118736685 IC50 > 60000 nM T20251 C67WJQ 118736760 IC50 > 60000 nM T20251 C8OZ7Q 118736762 IC50 > 60000 nM T20251 C54VYM 118736763 IC50 > 60000 nM T20251 CT28OR 118736765 IC50 = 30600 nM T20251 CL38BF 118736766 IC50 > 60000 nM T20251 C3UF7B 118736767 IC50 = 28200 nM T20251 C34XVR 118736768 IC50 = 33600 nM T20251 CGR7C8 118736770 IC50 = 32 nM T20251 CJ7AU0 118736771 IC50 = 8 nM T20251 CRN35A 118736772 IC50 = 64 nM T20251 C8WD3X 118736773 IC50 = 16 nM T20251 CJ46BO 118736774 IC50 = 16 nM T20251 CB23PD 118736775 IC50 = 64 nM T20251 C9X5JA 118736776 IC50 = 64 nM T20251 C2IB6U 118736777 IC50 = 32 nM T20251 CZDH32 118736778 IC50 = 64 nM T20251 CN1XD6 118736779 IC50 = 16 nM T20251 CVN7J1 118737793 IC50 > 100000 nM T20251 CVH7A9 118737794 IC50 > 100000 nM T20251 CI53XV 118737807 IC50 > 100000 nM T20251 CFM30P 118864208 IC50 = 35000 nM T20251 C6L4OC 118864285 IC50 = 8080 nM T20251 C9DM5W 118864313 IC50 = 4750 nM T20251 CF09GY 118864337 IC50 = 135000 nM T20251 C59NDJ 118864419 IC50 = 3470 nM T20251 C8AR7P 118864437 IC50 = 9560 nM T20251 CS20BC 118864476 IC50 = 52400 nM T20251 C4D9VF 118864482 IC50 = 52600 nM T20251 CELZ36 118866105 IC50 = 6900 nM T20251 CPK47S 118868365 IC50 = 79000 nM T20251 C14DLY 118872292 IC50 > 30000 nM T20251 C5Z0XH 118911481 IC50 = 120000 nM T20251 CM59EQ 118917669 IC50 > 100000 nM T20251 C6J8YF 118917671 IC50 > 100000 nM T20251 C2RBF7 118918048 IC50 = 2340 nM T20251 CW5EM8 118934075 IC50 = 10000 nM T20251 C7VL6I 118949555 IC50 > 10000 nM T20251 CN56FH 118949563 IC50 > 10000 nM T20251 C7CPN2 118950092 IC50 > 10000 nM T20251 CWR8M4 118950147 IC50 > 10000 nM T20251 C9UHO7 118950386 IC50 > 10000 nM T20251 CI9MA2 118950452 IC50 > 10000 nM T20251 CIQ51N 118953858 IC50 = 3200 nM T20251 CHJ70O 118960212 IC50 > 10000 nM T20251 CGJ9O5 118978102 IC50 > 31622.78 nM T20251 CSWO08 119057475 IC50 = 238000 nM T20251 CPS9N3 121245322 IC50 > 63095.73 nM T20251 C8P7OW 121245346 IC50 > 31622.78 nM T20251 CFOM46 121246727 IC50 > 31622.78 nM T20251 CL5Q9G 121246911 IC50 > 31622.78 nM T20251 CAL43C 121246982 IC50 > 31622.78 nM T20251 C6XK2Y 121247103 IC50 = 25118.86 nM T20251 C5S3FA 121292609 IC50 > 10000 nM T20251 COS3K9 121304408 IC50 = 812.83 nM T20251 C9G3ZJ 121304414 IC50 = 7585.78 nM T20251 CVN57T 121304417 IC50 = 2454.71 nM T20251 C4RD9Y 121304424 IC50 = 446.68 nM T20251 CN5YP1 121304426 IC50 < 100 nM T20251 CXL97W 121304430 IC50 = 2089.3 nM T20251 CA8CY5 121304437 IC50 = 295.12 nM T20251 C1PKR0 121304441 IC50 = 2818.38 nM T20251 CWLB20 121304449 IC50 = 467.74 nM T20251 CC3MP6 121304452 IC50 = 151.36 nM T20251 CW68KD 121304458 IC50 = 2884.03 nM T20251 CVA9F4 121304464 IC50 > 10000 nM T20251 CPB58L 121304467 IC50 = 3162.28 nM T20251 CFXN81 121304470 IC50 = 251.19 nM T20251 CTCA98 121304474 IC50 < 100 nM T20251 COB2X5 121304477 IC50 = 6309.57 nM T20251 CZ0BI4 121304484 IC50 = 10000 nM T20251 CW51NQ 121304485 IC50 = 407.38 nM T20251 CX1DQ6 121304488 IC50 = 1318.26 nM T20251 CZ4D2Y 121304493 IC50 = 794.33 nM T20251 CU50JM 121304499 IC50 = 257.04 nM T20251 C7NLV2 121304500 IC50 = 2951.21 nM T20251 C18GSY 121304506 IC50 = 3630.78 nM T20251 C21MEQ 121304510 IC50 < 100 nM T20251 C7F3NO 121304514 IC50 = 691.83 nM T20251 CPNV43 121304527 IC50 = 758.58 nM T20251 CCW3A9 121304532 IC50 = 1230.27 nM T20251 CQ2UM4 121304538 IC50 = 660.69 nM T20251 CR7L0O 121304539 IC50 = 891.25 nM T20251 C2GI6S 121304542 IC50 = 933.25 nM T20251 C1AB6P 121304551 IC50 = 602.56 nM T20251 CTI6Z7 121304565 IC50 = 602.56 nM T20251 CFVP28 121304568 IC50 = 446.68 nM T20251 CO6JN7 121304569 IC50 = 120.23 nM T20251 CN05ZQ 121304574 IC50 = 7943.28 nM T20251 CU0M7B 121304590 IC50 = 190.55 nM T20251 CLZK90 121304596 IC50 = 2511.89 nM T20251 C6YLM8 121304597 IC50 = 2754.23 nM T20251 CX5MO3 121304598 IC50 = 6918.31 nM T20251 C12GJP 121304609 IC50 = 2691.53 nM T20251 C31AEQ 121304649 IC50 = 524.81 nM T20251 C2VTK5 121304654 IC50 = 2754.23 nM T20251 CSYD40 121304673 IC50 = 316.23 nM T20251 C6IB0P 121304685 IC50 > 10000 nM T20251 CU0L6A 121304697 IC50 = 4677.35 nM T20251 CNOW27 121304705 IC50 = 616.6 nM T20251 C6NA0P 121304710 IC50 = 204.17 nM T20251 CXC70Q 121304711 IC50 = 933.25 nM T20251 CE0ND7 121304744 IC50 = 223.87 nM T20251 C1MZ6T 121304754 IC50 > 10000 nM T20251 C6C9EF 121304827 IC50 > 3000 nM T20251 C5HQ4S 121304867 IC50 = 1202.26 nM T20251 C6E2VF 121305983 IC50 = 9000 nM T20251 CL8P4D 121305987 IC50 = 7400 nM T20251 CR0HG1 121313818 IC50 = 4500 nM T20251 CO97HF 121313830 IC50 = 1400 nM T20251 CCUN52 121313839 IC50 = 8000 nM T20251 C4USB9 121313840 IC50 = 5000 nM T20251 C1GPN7 121313866 IC50 > 60000 nM T20251 CML4Z3 121313870 IC50 = 4200 nM T20251 CWC64Z 121313891 IC50 = 36400 nM T20251 C37BWZ 121313899 IC50 = 45000 nM T20251 CC9A1P 121313903 IC50 = 54 nM T20251 CA5L4N 121313914 IC50 = 1500 nM T20251 C0VQ4K 121313943 IC50 = 9.5 nM T20251 CD6Z2S 121313948 IC50 = 10400 nM T20251 C5TJ0N 121313953 IC50 = 12300 nM T20251 C1H8OV 121313959 IC50 = 21900 nM T20251 CTD80X 121313965 IC50 > 60000 nM T20251 CU4CW1 121313969 IC50 = 20000 nM T20251 CFP26R 121313971 IC50 = 17200 nM T20251 CNT7G1 121313972 IC50 > 60000 nM T20251 CC1G3N 121313978 IC50 = 7600 nM T20251 C8ZC5L 121313982 IC50 = 2700 nM T20251 CR74PF 121313995 IC50 = 17600 nM T20251 CTD40H 121314002 IC50 = 4500 nM T20251 CQFC86 121314009 IC50 = 3800 nM T20251 C8I2PZ 121314020 IC50 = 9400 nM T20251 C7QK2C 121314021 IC50 = 12000 nM T20251 CJT43I 121314036 IC50 > 60000 nM T20251 C8PT6Y 121314045 IC50 = 4900 nM T20251 CH8S4J 121314048 IC50 = 4700 nM T20251 CFW68T 121314052 IC50 = 19100 nM T20251 CP13EB 121314068 IC50 = 27000 nM T20251 CAS0Y9 121315197 IC50 = 562.34 nM T20251 CRZ1V0 121315205 IC50 = 263.03 nM T20251 CV3XH6 121315206 IC50 = 1949.84 nM T20251 C4TI7P 121315244 IC50 = 200 nM T20251 CLM9E8 121315259 IC50 = 524.81 nM T20251 C7B3XN 121315293 IC50 = 3981.07 nM T20251 C9U5CV 121315295 IC50 = 134.9 nM T20251 CN39AK 121315339 IC50 = 295.12 nM T20251 C14NCL 121315356 IC50 = 144.54 nM T20251 COG90M 121315374 IC50 = 151.36 nM T20251 CEY62R 121315401 IC50 < 100 nM T20251 C0E6HD 121315586 IC50 < 100 nM T20251 CBAG84 121315634 IC50 < 100 nM T20251 C9Q2ND 121333973 IC50 > 10000 nM T20251 C5BVJ8 121351012 IC50 > 25000 nM T20251 C46DBJ 121362063 IC50 = 30000 nM T20251 COGV39 121362167 IC50 = 2600 nM T20251 CV9TX1 121399281 IC50 = 19900 nM T20251 C7IU8N 121401335 IC50 > 50000 nM T20251 C7NWK8 121401336 IC50 = 44700 nM T20251 C5RXG7 121401340 IC50 > 50000 nM T20251 CV0FH9 121401343 IC50 = 2200 nM T20251 C2WD1Q 121407246 IC50 = 5351 nM T20251 CR5HV8 121410292 IC50 = 16000 nM T20251 CVE96K 121410294 IC50 = 3300 nM T20251 CK9G7V 121410328 IC50 = 2600 nM T20251 CQ3KL4 121410329 IC50 = 1800 nM T20251 CBN62U 121410340 IC50 = 8000 nM T20251 CNF06J 121410352 IC50 = 7200 nM T20251 C91PVZ 121428416 IC50 > 30000 nM T20251 CO9SQ6 121454909 IC50 > 60000 nM T20251 CH0X4Z 121454982 IC50 > 60000 nM T20251 CT0KS4 121455652 IC50 = 54000 nM T20251 CW35TI 121455794 IC50 = 26000 nM T20251 CBL46V 121488126 IC50 > 30000 nM T20251 C3WC9Y 121488127 IC50 = 12000 nM T20251 C7X1BQ 121493987 IC50 > 60000 nM T20251 CHD26A 121596332 IC50 > 33300 nM T20251 CV06MA 122177111 IC50 > 33000 nM T20251 C2DH7M 122177112 IC50 = 29000 nM T20251 CL8GC2 122177113 IC50 = 7800 nM T20251 C0H8AW 122177723 IC50 > 30000 nM T20251 CZ1F4O 122178097 Ki > 9182 nM T20251 C2AWE9 122178128 IC50 = 1600 nM T20251 CO4Y3I 122179072 IC50 = 1170 nM T20251 C92SDF 122179073 IC50 = 22390 nM T20251 C9OQ8P 122179074 IC50 > 50100 nM T20251 C6DA3N 122179075 IC50 > 50100 nM T20251 C4RYS0 122179076 IC50 > 50100 nM T20251 C9WB6E 122179416 IC50 > 40000 nM T20251 CY6C1E 122179442 IC50 = 93560 nM T20251 C5KGV7 122179447 Ki = 290 nM T20251 CFO15B 122179448 Ki = 50 nM T20251 CJP38S 122179449 Ki = 440 nM T20251 C3FP8V 122179450 Ki = 2870 nM T20251 CQGW18 122179451 Ki = 720 nM T20251 CYW75S 122179452 IC50 = 200 nM T20251 COHA53 122179453 IC50 = 190 nM T20251 CI8H9C 122179454 IC50 = 90 nM T20251 CKZ4X8 122179455 IC50 = 340 nM T20251 CZ6U4L 122179456 IC50 = 170 nM T20251 CS12JW 122179457 IC50 = 8544 nM T20251 CEQ5M0 122179459 IC50 = 7300 nM T20251 CNP81Q 122179460 IC50 = 9600 nM T20251 C54KTN 122179461 IC50 = 3200 nM T20251 C8DLB2 122179463 IC50 = 3700 nM T20251 C56TKY 122179464 IC50 = 3200 nM T20251 C49TGA 122179465 IC50 = 4300 nM T20251 CWJ9C7 122179466 IC50 = 8500 nM T20251 CI3L7J 122179467 IC50 = 22400 nM T20251 C41LSM 122179468 IC50 = 10400 nM T20251 C4U2EY 122179469 IC50 = 1600 nM T20251 C24FUL 122179470 IC50 = 35400 nM T20251 CN2FR7 122179471 IC50 = 1100 nM T20251 CJ70OH 122179472 IC50 = 5500 nM T20251 CBAO67 122179474 IC50 = 25800 nM T20251 CQ0D2N 122179475 IC50 = 51500 nM T20251 C7FA8O 122179476 IC50 = 27900 nM T20251 CNGQ19 122179477 IC50 = 27000 nM T20251 C9CLO5 122179478 IC50 = 7700 nM T20251 CY6CB1 122179479 IC50 = 7700 nM T20251 C4MZT8 122179480 IC50 = 5500 nM T20251 CDQ37R 122179481 IC50 = 3400 nM T20251 C6FME8 122179482 IC50 = 30500 nM T20251 CO34VW 122179483 IC50 = 34500 nM T20251 C3OJS0 122180330 IC50 > 10000 nM T20251 C2WV9G 122180336 IC50 > 10000 nM T20251 CJ1AP3 122180337 IC50 = 6000 nM T20251 CBN0J2 122180338 IC50 > 10000 nM T20251 CEA80S 122180339 IC50 > 10000 nM T20251 CTG4B2 122180340 IC50 > 10000 nM T20251 CTCN25 122180342 IC50 > 10000 nM T20251 C35BFD 122180343 IC50 = 6900 nM T20251 C80QZN 122180344 IC50 = 8100 nM T20251 CDZY73 122181598 Ki = 65 nM T20251 C0AM6I 122181599 Ki = 203 nM T20251 C0HR6P 122181600 Ki = 588 nM T20251 CR5T7L 122181601 Ki = 355 nM T20251 C1TA2K 122181602 Ki = 66 nM T20251 C2YMS5 122181603 Ki = 5571 nM T20251 C7L1CN 122181604 Ki = 944 nM T20251 C15JKL 122181605 Ki = 54 nM T20251 C54PWV 122181606 Ki = 60 nM T20251 C7CRS0 122181607 Ki = 48 nM T20251 CF1A6N 122181608 Ki = 3282 nM T20251 CSF5Q3 122181609 Ki = 1196 nM T20251 CP29KL 122181610 Ki = 12 nM T20251 C3GX7Z 122181612 Ki = 0.28 nM T20251 C8IGV9 122181614 Ki = 3.4 nM T20251 CF1A8R 122181616 Ki = 17 nM T20251 C64EZY 122181618 Ki = 108 nM T20251 CK0T8W 122181620 Ki = 1179 nM T20251 C9U0MK 122181622 Ki = 63 nM T20251 CJ3MG7 122181646 Ki = 577 nM T20251 C37YWX 122181648 Ki = 122 nM T20251 C1XF3L 122181650 Ki = 176 nM T20251 C61YUM 122181652 Ki = 139 nM T20251 C29KZA 122181654 Ki = 303 nM T20251 CD9YE3 122181656 Ki = 247 nM T20251 CD6HB2 122181658 Ki = 153 nM T20251 C0TDQ1 122181660 Ki = 71 nM T20251 C8M4CH 122182156 IC50 > 100000 nM T20251 CK4A6L 122182159 IC50 = 28700 nM T20251 C1MA9K 122182829 IC50 = 49970 nM T20251 C06YKW 122182830 IC50 = 23830 nM T20251 CT6L2Q 122182831 IC50 = 21870 nM T20251 CZ45UW 122182832 IC50 = 25460 nM T20251 CA1I5D 122182833 IC50 = 22290 nM T20251 C9S2AG 122182834 IC50 = 2184 nM T20251 C2R5TF 122182835 IC50 > 60000 nM T20251 CQI46V 122182836 IC50 = 47600 nM T20251 CDQ50Z 122182837 IC50 = 21060 nM T20251 CU7NC1 122182838 IC50 = 20750 nM T20251 CGJ4S6 122182839 IC50 > 60000 nM T20251 CKR73I 122182840 IC50 = 47030 nM T20251 CE7M1W 122182841 IC50 = 17880 nM T20251 C8LIP2 122182842 IC50 > 60000 nM T20251 CWE9G8 122182843 IC50 = 24330 nM T20251 C6GTI8 122182881 IC50 = 39190 nM T20251 C0D4IR 122182882 IC50 > 60000 nM T20251 CW8L5K 122184697 IC50 > 10000 nM T20251 C2VO8E 122184845 IC50 > 40000 nM T20251 CGSF80 122184846 IC50 > 40000 nM T20251 CN4H8Q 122184847 IC50 > 40000 nM T20251 CT94PN 122184848 IC50 > 40000 nM T20251 CHW2O8 122185935 IC50 = 4300 nM T20251 C9Q6GP 122185936 IC50 = 300 nM T20251 CUR4T8 122185937 IC50 = 500 nM T20251 CZJ1F9 122185938 IC50 = 1200 nM T20251 CQ1WJ8 122185975 IC50 = 398.11 nM T20251 CKD43Z 122185976 IC50 = 501.19 nM T20251 CV6OS1 122186032 IC50 = 2400 nM T20251 C9U7CE 122186033 IC50 > 30000 nM T20251 CRN80B 122186034 IC50 > 30000 nM T20251 CR8XJ5 122186035 IC50 = 2400 nM T20251 CBNO03 122186196 IC50 = 600 nM T20251 C13DXU 122186197 IC50 > 60000 nM T20251 CZ2T0Y 122186198 IC50 = 500 nM T20251 CA0IQ6 122186199 IC50 > 30000 nM T20251 CUZ16L 122186200 IC50 = 29700 nM T20251 C64MDZ 122186201 IC50 = 39900 nM T20251 CH62CJ 122186268 IC50 > 60000 nM T20251 CEG4I0 122186270 IC50 = 2300 nM T20251 C7CLG6 122186271 IC50 = 10500 nM T20251 C59PMH 122186272 IC50 = 400 nM T20251 CV36HF 122186275 IC50 = 3500 nM T20251 CV7YJ4 122186276 IC50 = 500 nM T20251 CPWB01 122186277 IC50 = 1100 nM T20251 CKD2V7 122186847 Ki = 3300 nM T20251 CQA8B2 122187067 IC50 = 1600 nM T20251 CU4X9L 122187092 IC50 > 33000 nM T20251 CQC2K7 122187093 IC50 > 100000 nM T20251 CV3LK7 122187094 IC50 > 33000 nM T20251 CJ1I2P 122187095 IC50 = 82000 nM T20251 CWE2Q3 122187096 IC50 > 100000 nM T20251 CTHX29 122187097 IC50 > 224000 nM T20251 CAZY54 122187098 IC50 > 100000 nM T20251 C2LRE0 122187099 IC50 > 100000 nM T20251 CLD74S 122187100 IC50 > 100000 nM T20251 CZR97H 122187101 IC50 = 79000 nM T20251 C8M7AW 122187102 IC50 > 100000 nM T20251 C2EN0J 122187103 IC50 > 100000 nM T20251 C45DJR 122187104 IC50 > 100000 nM T20251 CF6U2X 122187105 IC50 > 100000 nM T20251 CGO2U9 122187106 IC50 > 100000 nM T20251 CXEH62 122187107 IC50 > 100000 nM T20251 C1X9PC 122187108 IC50 = 75000 nM T20251 C59JBF 122187726 IC50 = 4450 nM T20251 CC7W9L 122187727 IC50 = 6680 nM T20251 C2N0KO 122187728 IC50 = 4750 nM T20251 CRUK02 122187729 IC50 = 900 nM T20251 C7BF8W 122187730 IC50 = 9000 nM T20251 C9VFM5 122187799 Ki = 1900 nM T20251 C4XCP1 122187801 Ki = 8300 nM T20251 CCU2N7 122187802 Ki = 6500 nM T20251 C52XCY 122188482 IC50 = 9000 nM T20251 C2XJ7S 122188483 IC50 = 1700 nM T20251 CPW3L7 122188565 IC50 = 10000 nM T20251 CSDG34 122188566 IC50 = 5700 nM T20251 C1F2GQ 122188567 IC50 = 7700 nM T20251 C49ACM 122188568 IC50 = 4800 nM T20251 CCQ2U5 122188569 IC50 = 20000 nM T20251 CMV95H 122189010 Ki = 436 nM T20251 COAL50 122189011 Ki = 777 nM T20251 CE1P0S 122189012 Ki > 10000 nM T20251 C2KD1F 122189013 Ki = 4237 nM T20251 C3KFQ6 122189014 Ki = 1666 nM T20251 CUFN73 122190176 IC50 = 1400 nM T20251 C2H7BX 122190180 IC50 > 33000 nM T20251 CNYH67 122190199 IC50 = 900 nM T20251 CJ6FZ9 122190274 IC50 = 2400 nM T20251 CGQF31 122190276 IC50 = 700 nM T20251 CEP27O 122190278 IC50 = 6100 nM T20251 C5AFZ6 122191639 IC50 > 30000 nM T20251 C1XKA8 122191834 IC50 > 30000 nM T20251 C4NUY0 122192382 IC50 = 17000 nM T20251 C1MVP5 122192989 IC50 = 10930 nM T20251 CLHV68 122192990 IC50 = 3051 nM T20251 C4DXM3 122193184 IC50 > 13000 nM T20251 C2EHL1 122193185 IC50 > 13000 nM T20251 CFU6Z1 122193186 IC50 > 13000 nM T20251 CI74XN 122193187 IC50 > 13000 nM T20251 CJ87GI 122193188 IC50 = 32000 nM T20251 C7LU2A 122193256 IC50 = 4800 nM T20251 CJ93YN 122193259 IC50 > 33000 nM T20251 CM69QJ 122193260 IC50 = 1400 nM T20251 CQ0FE9 122193263 IC50 = 500 nM T20251 CSR2O7 122195839 IC50 > 10000 nM T20251 CP7N1K 122196372 IC50 = 850 nM T20251 C7V3BY 122196373 IC50 = 3760 nM T20251 CH7TS1 122196381 IC50 = 5980 nM T20251 C0SM9Q 122196384 IC50 = 630 nM T20251 C9BAO3 122196385 IC50 = 1010 nM T20251 CZR09C 122198706 Ki = 13000 nM T20251 CZ4U5A 122429808 IC50 > 30000 nM T20251 C0AKG9 122433571 IC50 = 17500 nM T20251 CR94XB 122442340 IC50 = 10000 nM T20251 C4CMY5 122442358 IC50 = 370 nM T20251 C4RU7S 122442363 IC50 = 82 nM T20251 CB7EI3 122442376 IC50 > 10000 nM T20251 C0E5TJ 122442379 IC50 = 1700 nM T20251 CJ12FN 122442383 IC50 > 10000 nM T20251 CMW6Q8 122442385 IC50 > 10000 nM T20251 CVO84P 122442392 IC50 > 10000 nM T20251 CO3H6P 122442396 IC50 = 200 nM T20251 C2Q4VX 122442405 IC50 > 10000 nM T20251 C6KZF3 122442410 IC50 > 10000 nM T20251 C7RD0C 122442412 IC50 = 1900 nM T20251 CC05AO 122442428 IC50 > 10000 nM T20251 CI7TA4 122442447 IC50 = 900 nM T20251 CTOZ85 122442455 IC50 > 10000 nM T20251 CHE8U1 122443093 IC50 = 500 nM T20251 CC2EZ8 122443959 IC50 > 30000 nM T20251 CH6VJ4 122453014 IC50 = 10000 nM T20251 COX7E3 122510453 IC50 > 10000 nM T20251 CME91S 122513214 Ki = 2200 nM T20251 C68PHW 122579408 IC50 > 80000 nM T20251 C2HZB8 122604308 IC50 = 20000 nM T20251 C8UL7Y 122657565 IC50 = 6380 nM T20251 C85JKN 122668190 IC50 = 1520 nM T20251 CXP73N 122678088 IC50 > 31622.78 nM T20251 C1YK2E 122678192 IC50 > 33000 nM T20251 CYJX49 123132228 IC50 > 30000 nM T20251 CK7W8B 123132907 IC50 = 3500 nM T20251 CRW0C2 123132915 IC50 = 2600 nM T20251 CKT6V0 123320121 Ki = 426 nM T20251 CBT9C4 123372252 IC50 > 40000 nM T20251 C2CHR3 123471111 IC50 = 25000 nM T20251 C0T6VF 123561371 IC50 > 20000 nM T20251 CA94XD 123818187 Ki = 13040 nM T20251 C7G6IA 123944769 IC50 > 20000 nM T20251 CT9K0V 124000588 IC50 = 8800 nM T20251 CDL2V4 124005596 IC50 > 20000 nM T20251 C5ZY7L 124114343 IC50 > 50000 nM T20251 CPO7N5 124125214 IC50 > 10000 nM T20251 C4VT3O 124127413 IC50 = 15000 nM T20251 CUO46T 124140941 IC50 = 200 nM T20251 C04VCS 124140943 IC50 = 250 nM T20251 C0UAQ6 124147818 IC50 > 30000 nM T20251 C8QAD1 124147824 IC50 = 6600 nM T20251 C9SO3J 124147915 IC50 = 980 nM T20251 CS43YV 124147927 IC50 > 30000 nM T20251 CZEC76 124147932 IC50 = 17000 nM T20251 C5B4UL 124147957 IC50 = 930 nM T20251 C1KFO8 124147973 IC50 > 30000 nM T20251 C70DOJ 124147979 IC50 > 30000 nM T20251 C2VE5C 124148108 IC50 = 7 nM T20251 C3ER2Z 124148120 IC50 = 290 nM T20251 CH7OZ3 124148123 IC50 = 1200 nM T20251 CFR2G7 124148125 IC50 = 1900 nM T20251 CEK31I 124148318 IC50 > 100000 nM T20251 C25IJY 124150428 IC50 > 30000 nM T20251 C04FYJ 124150499 IC50 > 30000 nM T20251 C5H2QB 124150512 IC50 = 4000 nM T20251 CLJ36I 124150528 IC50 > 30000 nM T20251 CE2W0X 124150540 IC50 > 30000 nM T20251 C8N5JR 124150544 IC50 > 30000 nM T20251 C9TB6E 124150550 IC50 > 30000 nM T20251 C58EUN 124150620 IC50 = 9800 nM T20251 C94XQA 124150663 IC50 = 6000 nM T20251 C6FSR3 124175917 Ki > 10000 nM T20251 C7TOU4 124175991 IC50 > 10000 nM T20251 CC1O5L 124176023 IC50 = 5300 nM T20251 C49NHK 124176024 Ki = 1100 nM T20251 C49ONG 124176026 Ki = 1400 nM T20251 CTD7Q0 124176027 Ki = 2400 nM T20251 C53AYP 124176028 Ki = 5900 nM T20251 CM56CN 124176084 Ki > 10000 nM T20251 C9RLT1 124176103 Ki = 900 nM T20251 CT6HB4 124176198 Ki = 2900 nM T20251 CL7K0C 124176200 Ki = 2900 nM T20251 CWMF80 124176201 Ki = 4900 nM T20251 CYD04K 124176232 IC50 > 10000 nM T20251 CMS9P1 124176233 IC50 > 10000 nM T20251 C7EQH8 124176242 IC50 > 10000 nM T20251 C4TQO9 124176277 IC50 > 10000 nM T20251 CGJH79 124176281 IC50 > 10000 nM T20251 CCYK63 124176287 IC50 > 10000 nM T20251 CWF7N2 124176288 IC50 > 10000 nM T20251 CK0B3W 124176291 IC50 > 10000 nM T20251 CR3I7P 124176294 IC50 > 10000 nM T20251 CNC17W 124176295 IC50 > 10000 nM T20251 CO1EA0 124176296 IC50 > 10000 nM T20251 CMG02Z 124176321 IC50 > 10000 nM T20251 C4E7VI 124176804 IC50 = 1800 nM T20251 CS9U3T 126502731 IC50 > 30000 nM T20251 C6TEJ0 126532768 IC50 = 1584.89 nM T20251 CNRI41 126533424 IC50 = 316.23 nM T20251 CG65RM 126533453 IC50 < 100 nM T20251 CRX67M 126533461 IC50 = 316.23 nM T20251 C0OPY6 126533669 IC50 = 794.33 nM T20251 CSN21X 126533798 IC50 = 125.89 nM T20251 CMHY08 126533799 IC50 = 1584.89 nM T20251 CP8W0X 126533801 IC50 = 1995.26 nM T20251 CXM45K 126533810 IC50 < 100 nM T20251 C0E7OY 126533847 IC50 = 5011.87 nM T20251 CPL62Z 126533872 IC50 = 630.96 nM T20251 C1ST0Y 126533877 IC50 = 794.33 nM T20251 CDP5C4 126533939 IC50 = 158.49 nM T20251 CX2A4N 126533957 IC50 = 2511.89 nM T20251 CIV7R0 126533969 IC50 = 3981.07 nM T20251 CC7V5Y 126533978 IC50 = 630.96 nM T20251 CI97TU 126533981 IC50 = 125.89 nM T20251 CON63X 126534012 IC50 = 251.19 nM T20251 C9G1IV 126534022 IC50 < 100 nM T20251 C9AN4B 126534041 IC50 = 158.49 nM T20251 C8JKG0 126534069 IC50 = 125.89 nM T20251 C65OJB 126534075 IC50 = 630.96 nM T20251 CA4QM3 126534084 IC50 = 1258.93 nM T20251 C3SUR8 126534086 IC50 = 199.53 nM T20251 CCX0O5 126534178 IC50 = 398.11 nM T20251 C6NU0Y 126534182 IC50 < 100 nM T20251 CNUA81 126534195 IC50 = 100 nM T20251 CIAD86 126534204 IC50 = 1258.93 nM T20251 C4R7XU 126534291 IC50 = 5011.87 nM T20251 CVBX50 126534373 IC50 = 199.53 nM T20251 CB94HO 126534441 IC50 = 2511.89 nM T20251 CSX9W5 126534443 IC50 = 794.33 nM T20251 CQ39ZD 126534462 IC50 = 199.53 nM T20251 CT75WF 126534466 IC50 = 630.96 nM T20251 C52IHK 126534498 IC50 = 398.11 nM T20251 CFA3D6 126534516 IC50 = 794.33 nM T20251 CX14VB 126534676 IC50 < 100 nM T20251 CIW18V 126534678 IC50 = 125.89 nM T20251 CJPA49 126534738 IC50 < 100 nM T20251 CG7CY3 126534740 IC50 < 100 nM T20251 CQDE96 126534746 IC50 = 1995.26 nM T20251 CIN62J 126534758 IC50 = 199.53 nM T20251 CXI58O 126534764 IC50 = 125.89 nM T20251 C0WUJ5 126534771 IC50 = 1258.93 nM T20251 CFDR90 126534824 IC50 = 158.49 nM T20251 CX9LM7 126534859 IC50 = 6309.57 nM T20251 CKN57U 126534860 IC50 < 100 nM T20251 C3YB2Z 126534863 IC50 < 100 nM T20251 CR70LT 126534933 IC50 = 1000 nM T20251 CKBT37 126534948 IC50 = 1258.93 nM T20251 C6DLR7 126534986 IC50 = 794.33 nM T20251 CR10PO 126534991 IC50 = 1258.93 nM T20251 CFT24J 126535001 IC50 = 100 nM T20251 C58EIM 126535029 IC50 < 100 nM T20251 C5HQB6 126535034 IC50 < 100 nM T20251 C9Q0VB 126535075 IC50 = 251.19 nM T20251 CIZC84 126535109 IC50 > 10000 nM T20251 CMT3Q8 126535410 IC50 = 1000 nM T20251 C5YS6F 126535470 IC50 = 501.19 nM T20251 C4TZ6I 126535517 IC50 < 100 nM T20251 CTAG09 126567264 IC50 = 3380 nM T20251 C5QT4N 126567306 IC50 = 3500 nM T20251 CCH07K 126640345 IC50 = 1750 nM T20251 CR70JL 126641909 IC50 = 8300 nM T20251 CT7M6Q 126641926 IC50 = 13200 nM T20251 CLG67Z 126641948 IC50 = 12000 nM T20251 CVAC39 126641974 IC50 = 340 nM T20251 C1ZTB7 126641995 IC50 = 15800 nM T20251 CA81IH 126642266 IC50 = 19000 nM T20251 CNJL38 126642277 IC50 = 4000 nM T20251 CIW02N 126642282 IC50 = 55000 nM T20251 CY7US6 126715366 IC50 > 33000 nM T20251 CX37RN 126715380 IC50 > 100000 nM T20251 CH6YP0 126715392 IC50 > 100000 nM T20251 C1QB5R 126715400 IC50 = 22000 nM T20251 CO2X6J 126715460 IC50 = 15000 nM T20251 C09PAE 126744799 IC50 > 10000 nM T20251 COJ60B 126744800 IC50 > 10000 nM T20251 C0FKA4 126744972 IC50 = 6300 nM T20251 CT3R2Q 126961699 IC50 = 10000 nM T20251 COF75Z 126970673 IC50 = 29000 nM T20251 CS1B2E 127020968 IC50 > 100000 nM T20251 COWC81 127025601 IC50 > 11100 nM T20251 C1HGA4 127025889 IC50 > 100000 nM T20251 CF61HD 127025890 IC50 > 11100 nM T20251 CM74CE 127025891 IC50 > 100000 nM T20251 C4D9QY 127026491 IC50 > 30000 nM T20251 CBE56W 127026514 IC50 = 2830 nM T20251 C76CNA 127027374 IC50 > 10000 nM T20251 C15EJA 127027375 IC50 = 3701 nM T20251 CK8M1R 127027397 IC50 = 7261 nM T20251 C20XMQ 127027566 IC50 = 19000 nM T20251 C1PZ5S 127027702 IC50 > 10000 nM T20251 CZVP92 127028061 IC50 = 3100 nM T20251 CZ3G8X 127028062 IC50 = 4900 nM T20251 CN32ML 127028362 IC50 = 6600 nM T20251 C8MC1I 127028408 IC50 = 9100 nM T20251 CF1HM4 127028816 IC50 = 42000 nM T20251 CJ61PC 127028946 IC50 > 10000 nM T20251 CG14NR 127029113 IC50 = 21000 nM T20251 C32VER 127029260 IC50 > 5000 nM T20251 COAM29 127029262 IC50 > 5000 nM T20251 CF1MD9 127029702 IC50 = 42000 nM T20251 CL9IY6 127029888 IC50 = 17 nM T20251 C5RFV1 127029889 IC50 = 839 nM T20251 CZDO76 127030069 IC50 > 33000 nM T20251 C8WD7N 127030070 IC50 = 26000 nM T20251 C9GHX6 127030071 IC50 = 10000 nM T20251 CZCQ82 127030226 IC50 = 158 nM T20251 C7FD0M 127030227 IC50 = 467 nM T20251 C80JUT 127030228 IC50 = 69 nM T20251 C7YE3D 127030229 IC50 = 247 nM T20251 CF0S8I 127030230 IC50 = 350 nM T20251 CT9E3O 127030231 IC50 = 634 nM T20251 C0OKZ3 127030367 IC50 = 16000 nM T20251 CEP0T2 127030368 IC50 = 14000 nM T20251 CRV2K4 127030530 IC50 = 130 nM T20251 CJI5T4 127030531 IC50 = 58 nM T20251 C1F4OY 127030547 IC50 = 1742 nM T20251 C3VFN1 127030548 IC50 = 465 nM T20251 C3TQ4U 127030549 IC50 = 1817 nM T20251 C80CHF 127030550 IC50 = 1753 nM T20251 CU5T7O 127030626 IC50 = 26000 nM T20251 CQL8J6 127030928 IC50 = 7900 nM T20251 CH93CT 127030999 IC50 = 24000 nM T20251 CMKT63 127031154 IC50 = 258 nM T20251 CR87FU 127031155 IC50 = 495 nM T20251 C1RF0I 127031156 IC50 = 316.23 nM T20251 C0A5RC 127031270 IC50 > 33000 nM T20251 CF4V0J 127031338 IC50 = 5500 nM T20251 CZ6A2D 127031339 IC50 = 11000 nM T20251 CZ6P7H 127031354 IC50 = 16000 nM T20251 C5BTJ9 127031355 IC50 = 31000 nM T20251 CB7XP0 127031356 IC50 = 24000 nM T20251 CAV6G1 127031432 IC50 = 1025 nM T20251 CMU7D8 127031454 IC50 = 144 nM T20251 C9FR7D 127031456 IC50 = 101 nM T20251 C0A3PY 127031458 IC50 = 251.19 nM T20251 CY0EJ4 127031464 IC50 = 7518 nM T20251 C4GH0Z 127031465 IC50 = 2701 nM T20251 CM89VC 127031576 IC50 > 33000 nM T20251 C98TDU 127031577 IC50 > 33000 nM T20251 C4F3QY 127031621 IC50 = 11000 nM T20251 CB7Y6D 127031622 IC50 = 4200 nM T20251 CUO4V9 127031623 IC50 = 6200 nM T20251 CVGP91 127031694 IC50 = 44900 nM T20251 C2GK1H 127031773 IC50 = 4393 nM T20251 CFG8U2 127031907 IC50 = 5300 nM T20251 CI9ZB4 127031908 IC50 = 3300 nM T20251 C3NE8G 127031909 IC50 = 7500 nM T20251 CYHK91 127032122 IC50 = 44000 nM T20251 CYAR63 127032340 IC50 = 136 nM T20251 C7XI2Z 127032341 IC50 = 2944 nM T20251 C1OE8W 127032342 IC50 = 506 nM T20251 C79DCQ 127032659 IC50 = 146 nM T20251 CDX69E 127032660 IC50 = 522 nM T20251 C2TH8G 127032662 IC50 = 87 nM T20251 CZ9LM1 127032786 IC50 = 7400 nM T20251 CYZH79 127032787 IC50 = 3000 nM T20251 C7AK5Z 127033095 IC50 = 1800 nM T20251 C3UKI0 127033096 IC50 > 33000 nM T20251 CLJ6G9 127033551 IC50 = 4026 nM T20251 C9MD2C 127033672 IC50 > 33000 nM T20251 C1YR3E 127033673 IC50 = 25000 nM T20251 C1HO7F 127033703 IC50 = 970 nM T20251 CB12AP 127033704 IC50 = 6960 nM T20251 C5ITG3 127033945 IC50 = 15000 nM T20251 C4NIU0 127034022 IC50 = 1500 nM T20251 C5NU3M 127034125 IC50 = 530 nM T20251 CLR2J7 127034153 IC50 > 30000 nM T20251 CEWM81 127034292 IC50 = 200 nM T20251 C1FBI6 127034426 IC50 = 5503 nM T20251 CLN17T 127034427 IC50 = 4895 nM T20251 CMYQ47 127034428 IC50 = 6481 nM T20251 CON9I2 127034429 IC50 = 3619 nM T20251 CKS28E 127034802 IC50 = 2650 nM T20251 CKSZ13 127035240 IC50 > 60000 nM T20251 CGV62B 127035655 IC50 = 11200 nM T20251 CZY9R4 127035656 IC50 = 4900 nM T20251 C2KC9W 127035890 IC50 = 6309.57 nM T20251 CQ9ZK4 127036284 IC50 > 12250 nM T20251 C1L7MN 127036387 IC50 = 6000 nM T20251 CZA74X 127036551 IC50 = 18200 nM T20251 CGVD97 127036552 IC50 = 3300 nM T20251 CZG07V 127036553 IC50 = 5400 nM T20251 CE7M4J 127036775 IC50 > 10000 nM T20251 CS4H9O 127037230 IC50 = 3000 nM T20251 CTG43Z 127037413 IC50 = 2500 nM T20251 C15YEC 127037414 IC50 = 1200 nM T20251 C4OZ3F 127037433 IC50 = 6500 nM T20251 CL0IJ7 127037593 IC50 = 60000 nM T20251 C7T3PJ 127037594 IC50 = 36100 nM T20251 CB41IW 127037818 IC50 = 5100 nM T20251 C7L1DB 127037832 IC50 > 30000 nM T20251 CQA4K0 127038376 IC50 = 3810.2 nM T20251 C5I1PX 127038786 EC50 = 4600 nM T20251 CLH0B9 127040096 IC50 > 31622.78 nM T20251 C60HOC 127040550 IC50 = 11000 nM T20251 C6Z9VL 127040695 Ki = 1000 nM T20251 CG74QA 127040713 Ki = 1995.26 nM T20251 C34BGK 127040715 Ki = 5011.87 nM T20251 C0J8HC 127041348 Ki = 1000 nM T20251 CG84RM 127041558 IC50 = 31000 nM T20251 CS20QX 127041559 IC50 > 60000 nM T20251 CGN34V 127041705 IC50 = 1390.1 nM T20251 CN2T3I 127041869 IC50 = 7000 nM T20251 C2BE3M 127041870 IC50 = 36000 nM T20251 CS78AZ 127041951 Ki = 3162.28 nM T20251 CU9C4S 127041952 Ki = 3162.28 nM T20251 C9HPT6 127041953 Ki = 2511.89 nM T20251 C8H1RB 127041988 IC50 = 6309.57 nM T20251 CK6S5V 127042037 EC50 = 12000 nM T20251 C31SDE 127042181 IC50 = 17000 nM T20251 CS2AP8 127042622 IC50 = 6300 nM T20251 CL40ZB 127042623 IC50 > 11100 nM T20251 CJ45OF 127042624 IC50 = 10000 nM T20251 CP9L4A 127042940 IC50 = 5600 nM T20251 CR7QK2 127043679 IC50 = 1400 nM T20251 C79PSH 127044134 IC50 = 3200 nM T20251 CO6ZX5 127045058 IC50 = 26000 nM T20251 C4SFJ8 127045059 IC50 > 30000 nM T20251 C08FHU 127045060 IC50 = 21000 nM T20251 C8FZV7 127045061 IC50 = 8600 nM T20251 C5AXB2 127045351 IC50 = 7700 nM T20251 CY8BX9 127045352 IC50 = 5700 nM T20251 CC6WS4 127045353 IC50 = 9200 nM T20251 CZ0TP1 127045361 IC50 > 30000 nM T20251 CHIN43 127046285 IC50 = 47100 nM T20251 C34REM 127046317 IC50 = 94000 nM T20251 CAG9K7 127046489 IC50 > 100000 nM T20251 CH6W2T 127046982 IC50 = 2100 nM T20251 C6DP7Y 127047275 IC50 > 100000 nM T20251 C3DVM9 127047276 IC50 > 100000 nM T20251 CJH46E 127047680 IC50 = 1400 nM T20251 CM81AR 127047922 IC50 = 48380 nM T20251 C84TQV 127048530 IC50 = 640 nM T20251 CZV7Q0 127049047 IC50 > 79432.82 nM T20251 CB54VQ 127049048 IC50 > 100000 nM T20251 CDWJ67 127049172 IC50 = 2160 nM T20251 C2TKU8 127049173 IC50 = 2680 nM T20251 CJ8SG3 127049204 IC50 = 18000 nM T20251 C7D5QM 127049475 IC50 = 17000 nM T20251 C3V9MD 127049476 IC50 = 23000 nM T20251 C9A2DS 127049825 IC50 = 1890 nM T20251 CZS1L6 127049862 IC50 = 1030 nM T20251 CZD91J 127049863 IC50 = 998 nM T20251 CUT7E8 127050751 IC50 = 1610 nM T20251 CZW39D 127050752 IC50 = 1460 nM T20251 CUVQ34 127050762 IC50 = 97000 nM T20251 C5LVW9 127050783 Ki = 217 nM T20251 CXUH85 127050784 Ki = 12 nM T20251 C4LQ7M 127050803 IC50 = 6340 nM T20251 C25HJR 127050807 IC50 = 980 nM T20251 CS6C8O 127050851 IC50 = 24000 nM T20251 C1HAU4 127050852 IC50 = 23000 nM T20251 CHVU86 127050853 IC50 = 6400 nM T20251 CWDX26 127050854 IC50 = 5200 nM T20251 C7DU0N 127050855 IC50 = 17000 nM T20251 CLX8S5 127050856 IC50 = 9300 nM T20251 C9V4EG 127051045 IC50 = 6400 nM T20251 CH46LU 127051126 IC50 > 33000 nM T20251 C39WXP 127051127 IC50 > 33000 nM T20251 C5J3KY 127051128 IC50 > 33000 nM T20251 C7E4QP 127051129 IC50 > 33000 nM T20251 C35JLQ 127051177 IC50 = 3700 nM T20251 CDJQ32 127051599 IC50 = 5400 nM T20251 C2ISZ9 127051600 IC50 = 6600 nM T20251 C61GFX 127051601 IC50 = 5200 nM T20251 CFQ2X7 127051618 IC50 = 21000 nM T20251 C4DSF7 127051619 IC50 = 27000 nM T20251 C8JMN0 127051620 IC50 = 10000 nM T20251 CTZK49 127051621 IC50 = 7200 nM T20251 C7PZM3 127051622 IC50 > 33000 nM T20251 CZO5C7 127052225 IC50 = 12000 nM T20251 COX90Y 127052226 IC50 = 22000 nM T20251 CW6BR1 127052309 Ki = 91 nM T20251 C75EAL 127052638 IC50 = 600 nM T20251 C2GY5W 127052655 IC50 > 25000 nM T20251 CBYA45 127052869 IC50 = 1450 nM T20251 C5OE2H 127053611 IC50 = 17000 nM T20251 CKIU42 127263150 IC50 = 30 nM T20251 C38WDU 129012089 IC50 = 6700 nM T20251 CJI14M 129072680 IC50 > 100000 nM T20251 COL81P 129085358 IC50 > 100000 nM T20251 CI1H4A 129085361 IC50 > 100000 nM T20251 C5M7AB 129103161 IC50 = 823.7 nM T20251 C3WIA6 129103318 IC50 = 2905.4 nM T20251 C51ZGV 129103322 IC50 = 1899.6 nM T20251 CBSW14 129116690 IC50 = 11000 nM T20251 CS6OA8 129116809 IC50 = 23000 nM T20251 CV98PG 129136448 IC50 = 23000 nM T20251 C6GC0F 129186534 IC50 = 6130 nM T20251 C8KM6N 129186554 IC50 = 2670 nM T20251 CEZT92 129186564 IC50 = 5800 nM T20251 C5KJS8 129259157 IC50 > 25000 nM T20251 CBVS14 129387808 IC50 = 4880 nM T20251 CE8TV5 129893260 IC50 > 25000 nM T20251 CIL0Z5 129907910 IC50 = 130 nM T20251 CD80OM 129909338 IC50 = 186 nM T20251 C0FM1R 130196825 IC50 = 10000 nM T20251 CYA92R 130282633 IC50 > 100000 nM T20251 CO3QE2 130282636 IC50 > 100000 nM T20251 C3M2IV 130344977 IC50 = 3200 nM T20251 CE8Q7I 130345035 IC50 = 25000 nM T20251 C01UGK 130345060 IC50 = 36000 nM T20251 CN9S7B 130345097 IC50 = 51000 nM T20251 C3CH7B 130345110 IC50 = 47000 nM T20251 C7RN8L 130345158 IC50 = 68000 nM T20251 CF20BS 130345178 IC50 = 10000 nM T20251 CMO50A 130345200 IC50 = 4600 nM T20251 C29WVS 130358344 IC50 = 29000 nM T20251 CZM13E 130358354 IC50 = 66000 nM T20251 CRSH41 130391959 IC50 > 40000 nM T20251 CDE38Y 130406760 IC50 = 7800 nM T20251 CQ2K0R 130406834 IC50 > 10000 nM T20251 C47CAY 130421765 IC50 = 19952.62 nM T20251 C84YKI 130422161 IC50 > 31622.78 nM T20251 CY14VE 130449668 IC50 = 6100 nM T20251 C7HB2T 130449692 IC50 = 9600 nM T20251 CZB60C 130449716 IC50 = 7900 nM T20251 C70SUN 130449733 IC50 > 60000 nM T20251 CZCT84 130449749 IC50 > 60000 nM T20251 C9YSZ8 130449791 IC50 = 7900 nM T20251 CK68CA 130453737 IC50 = 15000 nM T20251 CR5X1T 130453989 IC50 = 15848.93 nM T20251 CVT2U3 130454024 IC50 = 7943.28 nM T20251 CT4BY6 130454058 IC50 > 31622.78 nM T20251 CZK41V 130454091 IC50 = 31622.78 nM T20251 C2OJ3C 130454093 IC50 = 12589.25 nM T20251 CDP9S1 130470501 IC50 = 17000 nM T20251 C5U1XV 130470509 IC50 = 24000 nM T20251 CLTQ15 130470516 IC50 = 14000 nM T20251 CUO41K 130470684 IC50 = 22000 nM T20251 CPC2A7 130470749 IC50 > 27000 nM T20251 C0GD9S 131728656 IC50 = 63.1 nM T20251 C96UHE 131728658 IC50 = 128.82 nM T20251 C4Z5MQ 131839619 IC50 > 100000 nM T20251 CY3P7I 131953432 IC50 > 10000 nM T20251 CE26HW 131955087 IC50 = 500 nM T20251 CU73IM 131985420 IC50 > 31622.78 nM T20251 CQEK82 131985476 IC50 = 12589.25 nM T20251 C20ZAT 131985489 IC50 > 50118.72 nM T20251 C1IKD6 131985494 IC50 > 31622.78 nM T20251 CI6W9O 131985523 IC50 > 50118.72 nM T20251 C4A1KN 132014906 IC50 = 4500 nM T20251 CN4RF6 132019596 IC50 > 100000 nM T20251 C93UNX 132041675 IC50 = 4500 nM T20251 CX27OU 132054828 IC50 > 33000 nM T20251 C3HI8S 132141090 IC50 = 371.54 nM T20251 C5P9AV 132153537 IC50 = 223.87 nM T20251 CRH07J 132156331 IC50 = 112.2 nM T20251 CWY58Z 132185302 IC50 > 40000 nM T20251 CQL4B7 132185442 IC50 = 19530 nM T20251 CS3C8P 132471744 IC50 > 100000 nM T20251 CF73XU 132473042 IC50 > 30000 nM T20251 C5U7JM 132473043 IC50 > 30000 nM T20251 CACJ46 132489333 IC50 > 10000 nM T20251 C81YTI 132510857 IC50 > 30000 nM T20251 CX05RI 132515052 IC50 = 21527.82 nM T20251 CES7P6 132517499 IC50 = 12500 nM T20251 CJZ7Y8 132569635 IC50 > 10000 nM T20251 C0Y2TP 132585192 IC50 = 50815.94 nM T20251 CJ04HZ 132585195 IC50 > 40000 nM T20251 C6CB0I 132585204 IC50 = 23000 nM T20251 CRAG89 132609278 IC50 = 14700 nM T20251 C2F6RM 132991430 IC50 > 15000 nM T20251 C39UCD 133080605 IC50 = 2900 nM T20251 C18GQC 134128280 IC50 > 10000 nM T20251 CO1RW6 134132142 IC50 = 54570 nM T20251 C6B1EN 134133066 EC50 > 30000 nM T20251 CQ95LB 134133571 IC50 > 63095.73 nM T20251 CR8HL3 134134147 IC50 = 3467.37 nM T20251 CR6I1X 134134165 IC50 = 22000 nM T20251 CJOQ95 134134229 IC50 > 60000 nM T20251 CTJF87 134134782 IC50 > 30000 nM T20251 CB9T4J 134134906 IC50 > 10000 nM T20251 CC7OQ2 134135307 IC50 = 3400 nM T20251 CE5TV4 134135453 IC50 = 2200 nM T20251 C2OSR5 134135634 IC50 = 3290 nM T20251 C1W4DO 134135721 IC50 = 11500 nM T20251 CG5VL6 134136656 IC50 = 4660 nM T20251 CG9J7V 134136763 IC50 = 1584.89 nM T20251 CD7NA5 134138492 IC50 > 30000 nM T20251 C3W5SM 134139893 IC50 = 1000 nM T20251 CWI1J7 134140478 IC50 = 8730 nM T20251 CHG9Z5 134140686 IC50 = 39810.72 nM T20251 C6B5RW 134141023 IC50 = 5400 nM T20251 CFW7E3 134141385 IC50 = 31622.78 nM T20251 CG7CX5 134141441 IC50 = 2240 nM T20251 CW04KZ 134141466 IC50 = 2700 nM T20251 C0W3JX 134142019 IC50 > 15000 nM T20251 CF41GA 134142277 IC50 > 10000 nM T20251 CYW9L4 134142282 IC50 = 16500 nM T20251 CUZB68 134143422 IC50 = 1140 nM T20251 C2IM4X 134143913 IC50 > 63095.73 nM T20251 CAL5D8 134145302 IC50 > 10000 nM T20251 CS8D9B 134145411 IC50 = 1300 nM T20251 CQ9G7H 134145670 IC50 > 30000 nM T20251 CZXT87 134145806 IC50 = 440 nM T20251 CN35SO 134146628 IC50 > 30000 nM T20251 CX3A0W 134146922 IC50 = 10400 nM T20251 CHN1C9 134147829 IC50 = 6550 nM T20251 CFG60Q 134148895 IC50 = 9100 nM T20251 CM9ZY1 134150199 IC50 > 10000 nM T20251 CA5B2J 134150245 IC50 > 60000 nM T20251 C1PQ5T 134150412 IC50 = 19952.62 nM T20251 C0S2VH 134150637 IC50 = 3311.31 nM T20251 C6NYU2 134150754 IC50 = 9549.93 nM T20251 C4R9EG 134151006 IC50 > 15000 nM T20251 COPA84 134151189 IC50 = 4500 nM T20251 C9Z1VM 134153244 IC50 > 10000 nM T20251 C8SH1L 134154191 IC50 = 3600 nM T20251 C7H8GQ 134157229 IC50 = 7900 nM T20251 C7AFS1 134157353 IC50 > 10000 nM T20251 C80WJP 134157894 IC50 = 3310 nM T20251 CSWE45 134163712 IC50 = 11000 nM T20251 C3TW0A 134374895 IC50 > 10000 nM T20251 CVLH60 134374993 IC50 = 8000 nM T20251 C47TLY 134378796 IC50 = 20000 nM T20251 C3HC0S 134537158 IC50 = 93000 nM T20251 CQC5S9 134539527 IC50 = 1170 nM T20251 C0MV7I 134539764 IC50 = 718 nM T20251 CVR60G 134539903 IC50 = 4160 nM T20251 CLA3C8 134540034 IC50 = 3280 nM T20251 CDFE40 134540190 IC50 > 30000 nM T20251 C20HAT 134585236 IC50 = 22200 nM T20251 C6W3VL 134585536 IC50 > 30000 nM T20251 CRL3O8 134585831 IC50 = 26300 nM T20251 CJXA12 134611894 IC50 = 31622.78 nM T20251 CX0UR7 134694318 IC50 = 4500 nM T20251 CLD78B 134694953 IC50 = 8300 nM T20251 CA89MQ 134813901 IC50 > 10000 nM T20251 C45OIZ 134814269 IC50 > 33300 nM T20251 C3K5PA 134814272 IC50 = 3700 nM T20251 C13ZRU 134817449 IC50 = 3120 nM T20251 CRPH17 134817805 IC50 = 3700 nM T20251 CZB7I6 134821685 IC50 = 5460 nM T20251 CS71IF 135126189 IC50 > 30000 nM T20251 C9FUK2 135151360 IC50 > 198000 nM T20251 C0BLS7 135156185 Ki > 10000 nM T20251 CUI9X6 135156216 Ki > 10000 nM T20251 C1GY2T 135156251 EC50 > 10000 nM T20251 C2HPY7 135156445 Ki > 10000 nM T20251 CCB30F 135179035 IC50 > 198000 nM T20251 CWQ30S 135192932 IC50 = 6100 nM T20251 CQI48P 135192983 IC50 = 16000 nM T20251 CT0GQ6 135197577 IC50 > 10000 nM T20251 C87VKA 135197594 IC50 > 10000 nM T20251 CQXS07 135197635 IC50 > 10000 nM T20251 C7KXF1 135197643 IC50 > 10000 nM T20251 C14FWK 135348858 IC50 > 30000 nM T20251 CWL67T 135397764 IC50 > 50118.72 nM T20251 COK4D6 135401985 IC50 > 30000 nM T20251 C1DM3K 135401987 IC50 = 21000 nM T20251 CMH4G1 135412290 Ki > 15000 nM T20251 C47LAF 135418940 IC50 > 30000 nM T20251 CB1VD9 135426471 Ki > 15000 nM T20251 CWU95A 135445691 IC50 = 133299.95 nM T20251 C6HFC8 135450111 IC50 = 12882.5 nM T20251 C9J4ES 135503073 IC50 > 10000 nM T20251 C4PM9W 135515431 IC50 = 11481.54 nM T20251 CRM4Q8 135518358 IC50 = 28000 nM T20251 CY4MV6 135566354 IC50 > 30000 nM T20251 CYVU41 135566744 IC50 = 53500 nM T20251 CI47VJ 135566923 IC50 > 30000 nM T20251 C61CPM 135570331 IC50 = 26200 nM T20251 CCNH91 135743577 IC50 > 10000 nM T20251 CN2B3D 135747628 IC50 > 30000 nM T20251 CNI90F 135797785 Ki = 2100 nM T20251 CNQ47X 135846033 IC50 = 50.12 nM T20251 CRL10Y 135857967 IC50 > 33000 nM T20251 CI1D7K 135875806 IC50 > 10000 nM T20251 CCK5I3 135883253 IC50 = 16000 nM T20251 CBX90O 135910326 IC50 > 10000 nM T20251 C5EC2O 135910327 IC50 > 10000 nM T20251 CK8XQ2 135981707 IC50 = 1400 nM T20251 C0Y4RD 135983984 IC50 > 32000 nM T20251 C4AI7G 136030608 IC50 > 10000 nM T20251 C2HP1X 136030609 IC50 > 10000 nM T20251 CCZO92 136030610 IC50 = 870 nM T20251 CO0L9T 136056541 IC50 > 30000 nM T20251 CLIE18 136056542 IC50 = 20000 nM T20251 CN1PY3 136056548 IC50 > 30000 nM T20251 CT57ZH 136069450 IC50 = 1500 nM T20251 CFT9R3 136069453 IC50 = 20000 nM T20251 CRPQ42 136069494 IC50 = 220 nM T20251 CK8Z3V 136069521 IC50 = 1000 nM T20251 CPY1B2 136069522 IC50 = 27000 nM T20251 CX0OM4 136069523 IC50 = 7700 nM T20251 C6EU4D 136069524 IC50 = 9000 nM T20251 CQA2Z1 136069531 IC50 = 22000 nM T20251 CCH31A 136069532 IC50 = 950 nM T20251 CQ1FS4 136069563 IC50 > 60000 nM T20251 CA83VQ 136094778 Ki = 5800 nM T20251 C3ZS9L 136099767 IC50 = 6800 nM T20251 CLB4O7 136099768 IC50 = 800 nM T20251 CUG28I 136117980 Ki = 1400 nM T20251 C7GP2R 136123532 IC50 = 67000 nM T20251 C1U8TM 136160538 IC50 > 10000 nM T20251 CGX6C4 136173253 IC50 > 100000 nM T20251 CRO13K 136187001 IC50 = 400 nM T20251 CJM67G 136198642 IC50 = 1960 nM T20251 CQTB32 136205798 IC50 > 30000 nM T20251 CV8QP3 136205832 IC50 = 8100 nM T20251 CB93EM 136205833 IC50 = 13000 nM T20251 CAD80N 136245084 EC50 > 10000 nM T20251 CQ4UT7 136253018 IC50 = 2200 nM T20251 C03JRC 136253041 IC50 = 300 nM T20251 C18IDZ 136253042 IC50 = 300 nM T20251 C6ZQ3M 136253058 IC50 = 80 nM T20251 CJ32EY 136253061 IC50 = 6000 nM T20251 C5KI7Q 136264975 Ki = 1641 nM T20251 C0W8KA 136299435 IC50 = 0.95 nM T20251 C5G4ES 136299436 IC50 = 1.4 nM T20251 CN41IE 136377142 IC50 = 16000 nM T20251 CL6M4I 136377184 IC50 = 2500 nM T20251 C4OVP2 136416802 IC50 > 30000 nM T20251 C7ZCT8 136416815 IC50 > 30000 nM T20251 C94CEV 136598218 IC50 = 6000 nM T20251 C7GX9P 136598247 IC50 = 16000 nM T20251 C62TMK 136598251 IC50 = 17000 nM T20251 C5EW1N 136598257 IC50 = 270 nM T20251 CG1O5Z 136598272 IC50 = 230 nM T20251 C0JQC3 136607508 IC50 = 4500 nM T20251 CO59KS 136607554 IC50 = 14000 nM T20251 C0R2IL 136901416 IC50 > 100000 nM T20251 C91WJF 136947741 Ki = 6800 nM T20251 C4VAQ0 136966273 IC50 = 800 nM T20251 CK4CM2 137028369 IC50 > 60000 nM T20251 CKJY95 137040409 IC50 = 1000 nM T20251 CF27GZ 137062183 IC50 = 1200 nM T20251 CE1G4P 137333984 IC50 > 25000 nM T20251 C8L5PZ 137348437 IC50 = 900 nM T20251 C81LGX 137349435 IC50 > 10000 nM T20251 CW6P2I 137394489 IC50 > 30000 nM T20251 C0PL4B 137434175 IC50 = 1 nM T20251 CXZ16C 137480037 IC50 > 31622.78 nM T20251 CW8QT1 137527725 IC50 = 8100 nM T20251 CS34IR 137628304 IC50 > 25000 nM T20251 C9ACX4 137628305 IC50 > 25000 nM T20251 CP2C1J 137628306 IC50 < 10000 nM T20251 CDGB50 137628309 IC50 > 25000 nM T20251 CW8ZR6 137628310 IC50 > 25000 nM T20251 C48QKY 137628311 IC50 > 25000 nM T20251 CH5AV6 137628312 IC50 > 25000 nM T20251 CU9O3A 137628639 IC50 > 50000 nM T20251 C6B5US 137628648 IC50 > 10000 nM T20251 C3A6PQ 137628670 IC50 = 10940 nM T20251 CNXJ86 137628681 IC50 = 24600 nM T20251 CQF1N6 137631458 IC50 = 131.83 nM T20251 CFB89A 137631484 IC50 > 16000 nM T20251 C2QCA5 137631487 IC50 > 60000 nM T20251 CY6TK1 137631739 IC50 = 4900 nM T20251 C0YMI5 137631826 IC50 = 570 nM T20251 CUYN25 137631834 IC50 = 3700 nM T20251 COQ47K 137631897 IC50 = 9000 nM T20251 C62NAF 137632738 IC50 = 281.84 nM T20251 CBR0X1 137632751 IC50 = 4600 nM T20251 C5N1VU 137632947 IC50 > 30000 nM T20251 C39SCN 137632955 IC50 = 2760 nM T20251 C8JWF7 137633017 IC50 = 14700 nM T20251 CVH35W 137633042 IC50 = 3000 nM T20251 CH43XI 137633091 IC50 > 60000 nM T20251 C6VWP8 137633129 IC50 = 4190 nM T20251 C30SZG 137633174 IC50 = 19000 nM T20251 C75YBS 137633326 IC50 = 251.19 nM T20251 C05ILH 137633336 IC50 = 3200 nM T20251 CHB92M 137633815 IC50 = 4960 nM T20251 CZOD53 137633880 IC50 = 2800 nM T20251 CJLB61 137633993 IC50 = 10200 nM T20251 C8C0OE 137634027 IC50 > 30000 nM T20251 C8HPN4 137634334 IC50 > 60000 nM T20251 CU40QT 137634377 IC50 = 13700 nM T20251 C5A9LK 137634700 IC50 = 87.1 nM T20251 CLK7A3 137635011 IC50 = 13900 nM T20251 CE6ZM1 137635237 IC50 = 12000 nM T20251 CX7GA4 137635351 IC50 = 32100 nM T20251 C3XRW2 137635947 IC50 > 30000 nM T20251 CMN6T7 137636115 IC50 > 40000 nM T20251 C32TPC 137636184 IC50 = 3260 nM T20251 CGOI28 137636189 IC50 = 8230 nM T20251 C7BJY5 137636807 IC50 = 4600 nM T20251 CCE5M7 137636942 IC50 = 45300 nM T20251 C7IL4D 137637204 IC50 = 14000 nM T20251 C2B1MZ 137637375 IC50 = 33000 nM T20251 CJH2V9 137637559 IC50 > 100000 nM T20251 CC8B6T 137637727 IC50 = 398.11 nM T20251 CHI7U2 137638473 IC50 = 900 nM T20251 CC09VU 137638599 IC50 = 1900 nM T20251 C3XT2M 137638639 IC50 = 3800 nM T20251 C52GLN 137638676 IC50 = 27100 nM T20251 CXG42C 137638912 IC50 > 33000 nM T20251 CF8S5N 137639002 IC50 = 1300 nM T20251 CY6VP5 137639127 IC50 = 12100 nM T20251 CF5TI6 137639661 IC50 > 100000 nM T20251 C4DW9S 137639931 IC50 = 1900 nM T20251 C4B7UM 137640060 IC50 > 30000 nM T20251 C5KX6V 137640062 IC50 = 1400 nM T20251 CJX8N5 137640241 IC50 = 13500 nM T20251 CA0QO6 137640453 IC50 > 40000 nM T20251 CVLN62 137640626 IC50 > 30000 nM T20251 CZSJ59 137640675 IC50 > 16000 nM T20251 CX01ER 137640926 IC50 > 30000 nM T20251 C91GMY 137641491 IC50 = 49200 nM T20251 C48UDJ 137642293 IC50 = 25100 nM T20251 CY98CE 137642361 IC50 > 30000 nM T20251 C9N1IG 137642471 IC50 = 1070 nM T20251 C5OXI1 137642484 IC50 > 30000 nM T20251 CBJX42 137642666 IC50 = 400 nM T20251 CYWA72 137643103 IC50 = 3800 nM T20251 C58ISN 137643139 IC50 = 34800 nM T20251 CQ87SJ 137643211 IC50 = 15000 nM T20251 C4MN6W 137643261 IC50 = 3300 nM T20251 C9BF0V 137643369 IC50 = 6100 nM T20251 CHOI53 137643582 IC50 = 1500 nM T20251 C70XZQ 137643636 IC50 = 34010 nM T20251 CU2PD4 137643678 IC50 = 1640 nM T20251 CVP8M6 137643865 IC50 > 20000 nM T20251 CEKO63 137643918 IC50 = 18.2 nM T20251 C6FPZ5 137644016 IC50 = 5480 nM T20251 C0CI4P 137644180 IC50 = 4100 nM T20251 CO7T8B 137644182 IC50 = 3300 nM T20251 CUMA78 137644191 IC50 > 30000 nM T20251 C09FUH 137644619 IC50 = 2460 nM T20251 CHS17L 137644882 IC50 = 16200 nM T20251 CV56QL 137645221 IC50 = 16500 nM T20251 C3K5IV 137645234 IC50 = 15000 nM T20251 CC1Y6W 137645554 IC50 > 31600 nM T20251 C23IRT 137645590 IC50 = 14000 nM T20251 CY1HN6 137645732 IC50 > 30000 nM T20251 C10CBD 137646316 IC50 = 20400 nM T20251 CWG0D6 137646487 IC50 > 10000 nM T20251 CM38TQ 137646827 IC50 = 1659.59 nM T20251 CFPE40 137646880 IC50 > 30000 nM T20251 C6EKO4 137646948 IC50 = 43.65 nM T20251 C8ZB5K 137647001 IC50 > 30000 nM T20251 C4O0JE 137647028 IC50 = 10000 nM T20251 C0NWV1 137647092 IC50 = 3000 nM T20251 C4DB7J 137647113 IC50 = 29000 nM T20251 C1PSL6 137647194 IC50 > 31600 nM T20251 CG9U3X 137647321 IC50 = 6500 nM T20251 CZXR87 137647404 IC50 > 10000 nM T20251 CO5M6C 137647489 IC50 > 200000 nM T20251 C3TXN9 137647591 IC50 = 31700 nM T20251 C19CXJ 137647807 IC50 = 14000 nM T20251 C4W9ED 137647842 IC50 = 28.84 nM T20251 CCIM31 137647884 IC50 > 20000 nM T20251 CTD69B 137647980 IC50 = 1200 nM T20251 CL06NY 137648464 IC50 = 29890 nM T20251 C7UTE8 137648598 IC50 = 2900 nM T20251 CH1J9F 137648789 IC50 = 67 nM T20251 CY8NV3 137648854 IC50 = 10700 nM T20251 CO89DX 137649100 IC50 = 100 nM T20251 COLY80 137649218 IC50 > 60000 nM T20251 CUFO39 137649223 IC50 > 60000 nM T20251 C0J6GS 137649319 IC50 = 900 nM T20251 CG3X9M 137649357 IC50 = 45000 nM T20251 C7SXI2 137649457 IC50 = 11300 nM T20251 C3GP4Y 137649582 IC50 > 30000 nM T20251 C04JSE 137649716 IC50 = 10300 nM T20251 CP6F7W 137650046 IC50 > 40000 nM T20251 CV0J6S 137650114 IC50 = 19300 nM T20251 CI7F1J 137650316 IC50 = 1300 nM T20251 COH10Y 137651081 IC50 = 1800 nM T20251 COCF21 137651256 IC50 > 60000 nM T20251 CB6G5D 137651292 IC50 = 75.86 nM T20251 CANL61 137651426 IC50 > 30000 nM T20251 CVR29E 137651451 IC50 = 28400 nM T20251 CS0PU8 137651464 IC50 > 40000 nM T20251 C3Z7LM 137651481 IC50 = 35000 nM T20251 CZ89GD 137651664 IC50 > 31600 nM T20251 CGXE73 137651731 IC50 > 30000 nM T20251 CRWS26 137652032 IC50 = 5600 nM T20251 CQ96SK 137652235 IC50 = 25000 nM T20251 CLN2U7 137652270 IC50 = 83000 nM T20251 CKW9B5 137652423 IC50 > 25000 nM T20251 CINE03 137652514 IC50 = 15000 nM T20251 CZ2MT3 137652584 IC50 = 26400 nM T20251 CXR6C1 137653051 IC50 >= 100000 nM T20251 CUL85Y 137653097 IC50 = 29000 nM T20251 C65XKJ 137653127 IC50 > 60000 nM T20251 CX0YC9 137653149 IC50 = 302 nM T20251 C38FXZ 137653443 IC50 > 80000 nM T20251 CQ32NO 137653545 IC50 = 11200 nM T20251 C4AQS0 137653772 IC50 = 2900 nM T20251 CVBC79 137653856 IC50 = 2200 nM T20251 C0O5HF 137654037 IC50 > 30000 nM T20251 C46DKN 137654445 IC50 = 200 nM T20251 CU6SM3 137654538 IC50 = 12400 nM T20251 CO9SD0 137654952 IC50 = 8400 nM T20251 CV89YB 137655268 IC50 = 32600 nM T20251 C8BDX5 137655281 IC50 > 60000 nM T20251 CP5S6L 137655441 IC50 = 46000 nM T20251 CSRK73 137655508 IC50 = 5600 nM T20251 C45CQG 137655515 IC50 = 1300 nM T20251 C7HO5N 137655611 IC50 > 16000 nM T20251 C17LIA 137655641 IC50 = 6730 nM T20251 C3LG7W 137655838 IC50 = 39380 nM T20251 C1OXG8 137655944 IC50 > 10000 nM T20251 CA7B5Z 137656105 IC50 > 30000 nM T20251 CVBS03 137656215 IC50 = 13200 nM T20251 CZ4W3T 137656391 IC50 = 4800 nM T20251 CN2UE9 137656598 IC50 > 60000 nM T20251 CW1J7N 137657095 IC50 = 2500 nM T20251 CXV0H7 137657379 IC50 = 5600 nM T20251 CRT86S 137657427 IC50 = 19700 nM T20251 C6C7FX 137657428 IC50 = 2900 nM T20251 C2ME3D 137657693 IC50 = 10300 nM T20251 C1NI7Z 137657872 IC50 = 22300 nM T20251 C8YB3D 137657887 IC50 = 2450 nM T20251 C9JP7K 137657919 IC50 = 14000 nM T20251 COH35U 137657930 IC50 > 30000 nM T20251 C5ZX4W 137657934 IC50 = 390 nM T20251 CB7C5E 137657969 IC50 = 3100 nM T20251 C59BVH 137658028 IC50 = 40000 nM T20251 CF7Q6D 137658206 IC50 > 30000 nM T20251 CLT89J 137658267 IC50 = 8680 nM T20251 CLZ6F9 137658483 IC50 = 20100 nM T20251 CJY5S1 137658512 IC50 = 260 nM T20251 CA72YP 137658615 Ki > 30000 nM T20251 CD87KA 137658644 IC50 > 28700 nM T20251 C45WRB 137659034 IC50 = 75.86 nM T20251 C5PV0M 137659142 IC50 = 5000 nM T20251 C1ZH9J 137659238 IC50 = 3100 nM T20251 CF25MB 137659327 IC50 = 1000 nM T20251 C0UM2I 137659879 IC50 = 4200 nM T20251 CYI45R 137660122 IC50 = 21000 nM T20251 CR41KW 137660124 IC50 = 25000 nM T20251 C5WI8U 137660200 IC50 = 5740 nM T20251 C6GN8Z 137660334 IC50 = 6700 nM T20251 C8A3EK 137660337 IC50 = 36000 nM T20251 C1YB0M 137660460 IC50 = 870 nM T20251 CJZ1A3 137660546 IC50 > 300000 nM T20251 CIMY59 137660725 IC50 = 24200 nM T20251 CXM59Y 137660745 IC50 > 16000 nM T20251 C9QHV0 137660822 IC50 > 40000 nM T20251 C7H2LV 137660844 IC50 = 46000 nM T20251 C2KX3V 137661020 IC50 > 30000 nM T20251 CC42XJ 137661121 IC50 = 19.95 nM T20251 CL8H3R 137661393 IC50 > 10000 nM T20251 C29DMS 137661489 IC50 > 60000 nM T20251 CP4IV9 137661909 IC50 = 5150 nM T20251 CUJ2F0 137662184 IC50 = 91.2 nM T20251 CY07GS 137662191 IC50 > 30000 nM T20251 C6KYD7 137700754 IC50 > 30000 nM T20251 CM3UF7 137700779 IC50 = 4700 nM T20251 CC9K8L 137796790 IC50 = 23000 nM T20251 C3QL4O 138319676 IC50 = 32000 nM T20251 C9MNG4 138319677 IC50 = 13000 nM T20251 C7TAV3 138319685 IC50 > 100000 nM T20251 CPTE92 138319693 IC50 > 30000 nM T20251 CMP8U3 138376515 IC50 = 1900 nM T20251 CE79SV 138377584 IC50 = 45000 nM T20251 CKT7F5 138393065 Ki = 15800 nM T20251 C2QLX3 138393292 IC50 > 40000 nM T20251 CFR0X3 138454761 IC50 > 40000 nM T20251 CA3C4O 138454792 IC50 > 30000 nM T20251 CHQA31 138454800 IC50 > 40000 nM T20251 C81ILP 138471783 IC50 = 8700 nM T20251 CKDZ26 138504497 IC50 = 24000 nM T20251 CBN08I 138544609 Ki = 5400 nM T20251 CSRI06 138547901 IC50 > 40000 nM T20251 CN6M0G 138964067 IC50 > 300000 nM T20251 CV6JY5 139030528 IC50 > 50118.72 nM T20251 CI1D9F 139600335 IC50 = 28000 nM T20251 CG2NH6 139600336 IC50 = 10600 nM T20251 C0HN5J 139600337 IC50 = 3000 nM T20251 CIQ96U 141478757 IC50 = 2900 nM T20251 C9JSZ2 141529337 IC50 = 47980 nM T20251 CSE1D2 141529338 IC50 = 38920 nM T20251 C43LDR 141730928 IC50 > 30000 nM T20251 C2D9TE 141756938 IC50 = 8000 nM T20251 C53UZY 141757055 IC50 = 5300 nM T20251 C7KD9N 142533975 IC50 = 7000 nM T20251 C17XZS 142727681 IC50 > 50000 nM T20251 C3MI8P 142747294 IC50 = 4000 nM T20251 C1W8QR 145865307 IC50 > 30000 nM T20251 C9ISH6 145925685 IC50 = 4700 nM T20251 CL8VT0 145946399 IC50 > 10000 nM T20251 C54ACE 145949595 IC50 = 7943.28 nM T20251 C6P9QW 145949880 IC50 = 12589.25 nM T20251 C85SDC 145949931 IC50 = 8100 nM T20251 C9Q1TH 145950015 IC50 = 15000 nM T20251 CVK2J4 145950020 IC50 = 4700 nM T20251 CTM0N6 145950094 IC50 > 10000 nM T20251 C3ASH6 145950133 IC50 = 80 nM T20251 C91DXZ 145950201 IC50 = 25118.86 nM T20251 CAB3N0 145950456 IC50 = 2620 nM T20251 CXKB09 145950494 IC50 = 4400 nM T20251 CK64FQ 145950570 IC50 > 33000 nM T20251 C6JYA5 145950619 IC50 = 2100 nM T20251 CPE7N3 145950719 IC50 > 33000 nM T20251 CYF32C 145950953 IC50 > 30 nM T20251 CL2OR1 145950976 IC50 = 20300 nM T20251 CW6XJ2 145951187 IC50 = 14000 nM T20251 CRXJ25 145951211 IC50 > 30 nM T20251 C7Q6MF 145951374 Ki > 40000 nM T20251 CCOW60 145952011 IC50 = 27000 nM T20251 CG48IY 145952272 IC50 > 10000 nM T20251 CX2UH4 145952348 Ki > 40000 nM T20251 CVR31U 145952361 IC50 = 24000 nM T20251 CAF83G 145952396 IC50 = 1584.89 nM T20251 CCY29F 145952435 IC50 > 10000 nM T20251 CVS48W 145952572 Ki > 40000 nM T20251 CLQ6T3 145953268 IC50 = 5200 nM T20251 C60XZR 145953297 IC50 > 30 nM T20251 C2WFH6 145953847 IC50 > 33000 nM T20251 CHG09C 145953855 IC50 = 3981.07 nM T20251 CJN63M 145953914 IC50 > 10000 nM T20251 C0V8SM 145954139 IC50 > 30 nM T20251 CJ89WR 145954168 IC50 = 3207 nM T20251 CJ3P0C 145954173 IC50 = 10500 nM T20251 C25NVO 145954311 IC50 = 6309.57 nM T20251 CTRQ36 145954357 IC50 = 8900 nM T20251 CBO52Q 145954980 Ki > 40000 nM T20251 C82RDB 145955110 IC50 > 10000 nM T20251 CQ56XG 145955114 IC50 = 2700 nM T20251 CFG31P 145955509 IC50 > 10000 nM T20251 CWJ0K6 145955642 IC50 > 30000 nM T20251 C3XQ4O 145956183 IC50 = 10000 nM T20251 C4Y9RM 145956261 IC50 > 10000 nM T20251 CJ5GW3 145956273 Ki > 40000 nM T20251 C0LJB1 145956360 Ki > 40000 nM T20251 CR9DQ8 145956659 IC50 > 10000 nM T20251 CL0NH3 145956868 IC50 > 10000 nM T20251 CB74GR 145957221 IC50 > 30 nM T20251 C50ATS 145957391 IC50 = 10000 nM T20251 CLC41T 145957467 IC50 = 4.22 nM T20251 CFZJ34 145957574 IC50 = 31622.78 nM T20251 C9X4EA 145957598 IC50 = 1753 nM T20251 CILC62 145957718 IC50 = 14 nM T20251 C6R0OC 145957812 IC50 = 5700 nM T20251 CB8S9C 145957865 Ki = 28000 nM T20251 CA4C9J 145957925 IC50 = 18000 nM T20251 CTN8V5 145958082 IC50 = 8500 nM T20251 CAQ41N 145958476 IC50 = 6800 nM T20251 CQ19NA 145958506 Ki > 40000 nM T20251 C2FR5D 145958670 IC50 = 21300 nM T20251 CZK51T 145958678 Ki > 40000 nM T20251 CWT43A 145958774 IC50 = 2511.89 nM T20251 C73CBD 145959061 IC50 = 23000 nM T20251 C6T8GR 145959482 IC50 > 10000 nM T20251 CDYO54 145959735 IC50 = 27000 nM T20251 C4MDJ7 145960187 IC50 > 10000 nM T20251 C4N8XW 145960316 IC50 > 10000 nM T20251 CTVX81 145960555 IC50 > 10000 nM T20251 CZ8W1F 145960626 IC50 > 30000 nM T20251 CX3VH5 145960676 IC50 = 13000 nM T20251 C4IT2A 145960697 Ki = 12700 nM T20251 CW5AC7 145960817 Ki = 38400 nM T20251 CJ1O5H 145961103 IC50 > 30000 nM T20251 CTVR05 145961491 IC50 = 7700 nM T20251 C5ZD1H 145961500 Ki = 38200 nM T20251 CG43LE 145961709 Ki > 40000 nM T20251 CRYN14 145961777 IC50 = 25000 nM T20251 CKM9A7 145961840 IC50 > 100000 nM T20251 CTC3O8 145961901 Ki = 34000 nM T20251 CIM9O6 145961922 IC50 > 100000 nM T20251 CH3D1Z 145961966 IC50 > 10000 nM T20251 CX7FC9 145962196 Ki = 16000 nM T20251 C3FB4W 145962568 Ki = 14100 nM T20251 C3GX1E 145962661 Ki = 2200 nM T20251 C5E3RJ 145962891 IC50 = 17000 nM T20251 C6VNH3 145962956 IC50 > 30000 nM T20251 C21LTM 145963134 IC50 = 4500 nM T20251 C8CQX3 145963143 IC50 > 30000 nM T20251 CC1T5Z 145963172 IC50 > 30000 nM T20251 C0QJV2 145963337 IC50 = 4200 nM T20251 CWS86L 145963466 IC50 = 15000 nM T20251 CF7K5G 145963483 IC50 = 8600 nM T20251 CE9Q8L 145963631 IC50 = 1200 nM T20251 CW7DC0 145963634 IC50 > 10000 nM T20251 CB9S3T 145963706 IC50 > 30000 nM T20251 CW62NS 145963795 IC50 > 39810.72 nM T20251 C6NT1H 145963881 IC50 = 21000 nM T20251 CAJQ14 145964002 IC50 = 5300 nM T20251 CIAD71 145964098 IC50 > 30000 nM T20251 C6K9YI 145964252 IC50 = 350 nM T20251 CQ5XM3 145964429 IC50 = 530 nM T20251 CUQ97V 145964493 IC50 = 750 nM T20251 C9FUW4 145964611 IC50 = 2200 nM T20251 CTJI01 145964752 IC50 = 1700 nM T20251 CQZ3F7 145965198 IC50 > 30000 nM T20251 CJP34X 145965420 IC50 = 85600 nM T20251 C2WE1B 145965485 IC50 = 690 nM T20251 CSK8Y1 145965486 IC50 = 4600 nM T20251 CG5C1Y 145965772 IC50 = 5490 nM T20251 CMHZ94 145965813 IC50 = 280 nM T20251 CFP9G3 145965954 IC50 > 39810.72 nM T20251 CVF4M6 145965985 IC50 = 6800 nM T20251 CQE6K0 145966013 IC50 = 430 nM T20251 C2MS3R 145966170 IC50 = 166 nM T20251 C36CZY 145966369 IC50 = 55400 nM T20251 CJ34YW 145966384 IC50 = 1120 nM T20251 CR4AG3 145966633 IC50 = 2100 nM T20251 CS51VC 145966675 IC50 = 5700 nM T20251 C4V5QG 145966727 IC50 = 460 nM T20251 CA5NY2 145966786 IC50 = 410 nM T20251 C1WA0P 145966817 IC50 > 40000 nM T20251 CZ21YN 145967045 IC50 = 760 nM T20251 C2P3YJ 145967230 IC50 = 15000 nM T20251 CDW83M 145967332 IC50 > 40000 nM T20251 C0H5UD 145967429 IC50 = 4800 nM T20251 C3K7QC 145967522 IC50 = 1900 nM T20251 C38BZY 145967590 IC50 > 3000 nM T20251 CS9MZ3 145967758 IC50 = 16000 nM T20251 CTGF42 145967808 IC50 = 800 nM T20251 CPI9S3 145967920 IC50 = 1900 nM T20251 CZKG72 145968038 IC50 = 6309.57 nM T20251 CR36FU 145968121 IC50 = 600 nM T20251 CNR31W 145968279 IC50 = 2500 nM T20251 CNB7G5 145968344 IC50 = 400 nM T20251 C9OU8R 145968403 IC50 > 2000 nM T20251 C0XC7I 145968454 IC50 = 178 nM T20251 CQCY49 145968539 IC50 = 500 nM T20251 C7MAX3 145968702 IC50 > 30000 nM T20251 C1AW2J 145968863 IC50 = 7500 nM T20251 CQU16D 145968894 IC50 = 9500 nM T20251 CK5B1E 145969068 IC50 = 12000 nM T20251 CT4QJ0 145969110 IC50 = 2000 nM T20251 CNH7O5 145969326 IC50 = 3162.28 nM T20251 CIYJ92 145969331 IC50 = 3000 nM T20251 C3KI4V 145969352 IC50 < 1000 nM T20251 CO3QA4 145969383 IC50 = 370 nM T20251 CUI97C 145969471 IC50 > 1000 nM T20251 C6TDW9 145969499 IC50 = 800 nM T20251 C06WLJ 145969520 IC50 > 10000 nM T20251 C9TWE2 145969541 IC50 > 10000 nM T20251 CR4FH0 145969547 IC50 = 1000 nM T20251 CM60DT 145969661 IC50 = 3300 nM T20251 C7T1AN 145969666 IC50 = 940 nM T20251 CHZ7N3 145969706 IC50 = 12589.25 nM T20251 CQU2J7 145969790 IC50 = 810 nM T20251 CSUM19 145969910 IC50 = 6309.57 nM T20251 CDFU92 145969917 IC50 = 1000 nM T20251 CP0YH5 145969933 IC50 = 4800 nM T20251 C5TN8I 145969964 IC50 > 10000 nM T20251 C5J9LU 145969970 IC50 = 1000 nM T20251 CK9C0H 145970062 IC50 = 3800 nM T20251 C0WIZ5 145970221 IC50 = 3800 nM T20251 CPL40F 145970342 IC50 = 1300 nM T20251 CG9BH2 145970410 IC50 = 1000 nM T20251 CM75RU 145970450 IC50 = 1300 nM T20251 CYF0S4 145970568 IC50 < 1000 nM T20251 CMRZ53 145970708 IC50 = 410 nM T20251 C8B4IY 145970709 IC50 = 900 nM T20251 CATQ85 145970768 IC50 = 800 nM T20251 CMO6C2 145970858 IC50 = 2300 nM T20251 C5O2EA 145971149 IC50 = 900 nM T20251 CP6ET4 145971201 IC50 > 10000 nM T20251 C9R2VH 145971456 IC50 = 15000 nM T20251 C53OSI 145971666 IC50 = 18400 nM T20251 C6RS0M 145972161 IC50 = 4310 nM T20251 C64NXT 145972392 IC50 = 29.96 nM T20251 CU13IP 145972573 IC50 = 2300 nM T20251 C1KJ6X 145972784 IC50 = 25118.86 nM T20251 C8RFM3 145973261 IC50 > 33000 nM T20251 C7PTX6 145973283 IC50 = 43000 nM T20251 CS6UG1 145973762 IC50 = 211.7 nM T20251 C6OI3K 145973962 IC50 = 8100 nM T20251 CVK1O7 145974594 IC50 > 100000 nM T20251 CVM02B 145974600 IC50 > 100000 nM T20251 C6XV4Q 145974681 IC50 = 7700 nM T20251 C4UBG5 145974805 IC50 = 2200 nM T20251 CUJ43W 145975270 IC50 = 850 nM T20251 CA7DN0 145975339 IC50 = 2100 nM T20251 C9ME5T 145975612 IC50 = 2300 nM T20251 CPM02H 145975616 IC50 = 2200 nM T20251 CH30YP 145975799 IC50 > 30000 nM T20251 CY7U6W 145976048 IC50 > 39810.72 nM T20251 C9MK4Z 145976157 IC50 = 880 nM T20251 C41FLJ 145976727 IC50 = 5300 nM T20251 CKU21C 145977020 IC50 = 39900 nM T20251 CM27YI 145977049 IC50 > 100000 nM T20251 C5R7ZH 145977058 IC50 = 890 nM T20251 CT5W7C 145977076 IC50 > 30000 nM T20251 CUV49K 145977796 IC50 = 4400 nM T20251 CHD83O 145977889 IC50 = 3050 nM T20251 CWJ46S 145978007 IC50 = 8000 nM T20251 CU2A1M 145978072 IC50 > 100000 nM T20251 CUQ30C 145978119 IC50 = 1400 nM T20251 CH7G2C 145978242 IC50 = 350 nM T20251 CYH46T 145978250 IC50 = 6200 nM T20251 C4DU7J 145978279 IC50 = 380 nM T20251 CY3K9M 145978286 IC50 = 2069 nM T20251 C8UOA3 145978371 IC50 = 3.27 nM T20251 CRC96P 145978494 IC50 > 39810.72 nM T20251 CVK9J5 145978628 IC50 = 85700 nM T20251 CGW6Q5 145978668 IC50 = 16500 nM T20251 CWB3L0 145978768 IC50 = 3270 nM T20251 CJWI69 145979108 IC50 = 6371 nM T20251 COBE14 145979224 IC50 = 210 nM T20251 CQ5E8T 145980370 IC50 = 2300 nM T20251 CV85ZH 145980382 IC50 = 3160 nM T20251 CVE82W 145980394 IC50 < 300 nM T20251 CSEC23 145980764 IC50 = 55300 nM T20251 CW7I0E 145981058 IC50 > 30000 nM T20251 CGA83C 145981271 IC50 = 15000 nM T20251 CNDI08 145981275 IC50 > 10000 nM T20251 CZ70KB 145981598 IC50 > 30000 nM T20251 C0QWN2 145981606 IC50 = 3900 nM T20251 CY8IF4 145981627 IC50 > 10000 nM T20251 CG1AU0 145981699 IC50 = 16000 nM T20251 C4SKG5 145981746 IC50 = 900 nM T20251 C7AE4L 145981787 IC50 > 10000 nM T20251 CD5GI8 145982093 IC50 > 30000 nM T20251 C1BP0G 145982116 IC50 = 27500 nM T20251 CVOU09 145982242 IC50 = 50000 nM T20251 CD6IQ0 145982284 IC50 = 220 nM T20251 CZN0U6 145982478 IC50 > 10000 nM T20251 CX0P5N 145982847 IC50 = 10000 nM T20251 CL13NC 145982905 IC50 = 794.33 nM T20251 C4XQK5 145982959 IC50 = 1600 nM T20251 CF8E5K 145983040 IC50 = 1300 nM T20251 C4N5TW 145983050 IC50 = 25118.86 nM T20251 CND20U 145983060 IC50 = 3300 nM T20251 CC3SD4 145983205 IC50 = 5000 nM T20251 C1DW4U 145983928 IC50 = 7850 nM T20251 C8UI5J 145984101 IC50 = 3000 nM T20251 C7CUB1 145984146 IC50 = 26000 nM T20251 CJ70YV 145984499 IC50 = 1995.26 nM T20251 CJ8K4G 145984512 IC50 = 5600 nM T20251 C4R5NQ 145984560 IC50 = 10000 nM T20251 C4HAP0 145984727 IC50 = 2060 nM T20251 C9VMD1 145985361 IC50 = 6700 nM T20251 CI9QP2 145985779 IC50 = 6000 nM T20251 COG61P 145985793 IC50 = 3100 nM T20251 CRA6D0 145985939 IC50 = 1258.93 nM T20251 CNK1M7 145986171 IC50 = 5011.87 nM T20251 CXSB48 145986302 IC50 = 11300 nM T20251 C7J6XS 145986357 IC50 = 19952.62 nM T20251 CI9OL2 145986409 IC50 = 8000 nM T20251 C2UZ1G 145986549 IC50 = 15800 nM T20251 C9V3MF 145986593 IC50 = 12000 nM T20251 CPN29R 145986920 IC50 = 10000 nM T20251 C5R6BS 145987142 IC50 = 4600 nM T20251 CG1PV7 145987277 IC50 = 6309.57 nM T20251 CHOY46 145987281 Ki > 10000 nM T20251 C02VTZ 145987482 IC50 = 260 nM T20251 CI0PA9 145987771 IC50 = 16660 nM T20251 CZY0X1 145987861 IC50 = 2500 nM T20251 C8Q2EG 145988110 IC50 > 100000 nM T20251 CY1OF2 145988177 IC50 = 5100 nM T20251 COCV25 145988531 IC50 > 50000 nM T20251 C49EDV 145988588 IC50 = 8305 nM T20251 CUAY25 145988620 IC50 = 300 nM T20251 CGJI91 145988834 IC50 = 3800 nM T20251 CF42MQ 145988924 IC50 = 7600 nM T20251 CY3MR0 145989049 IC50 = 600 nM T20251 CEWA58 145989127 IC50 = 8000 nM T20251 CWYP01 145989394 IC50 = 950 nM T20251 CG9KC4 145989896 IC50 = 260 nM T20251 CTOL60 145990433 IC50 = 8635 nM T20251 C7GK3H 145990715 IC50 > 40000 nM T20251 CSZ4M5 145990737 IC50 > 40000 nM T20251 CMJ46R 145990794 IC50 = 7520 nM T20251 CU0K2Y 145990810 IC50 > 10000 nM T20251 CCI37B 145990833 IC50 = 1300 nM T20251 CMOY14 145991173 IC50 = 28200 nM T20251 CH5KI1 145991195 IC50 = 4600 nM T20251 C9WU5F 145991707 IC50 = 8700 nM T20251 C94VFQ 145991807 IC50 = 1340 nM T20251 C9YWM0 145991838 IC50 = 3400 nM T20251 CO49YW 145991861 IC50 = 1500 nM T20251 CR6MJ3 145992332 IC50 = 8000 nM T20251 C5LF2I 145992475 IC50 > 30000 nM T20251 C9PS8N 145993117 IC50 = 6210 nM T20251 C91EUQ 145993184 IC50 = 12100 nM T20251 CYV43P 145993203 IC50 = 210 nM T20251 C0Z6YX 145993493 IC50 = 2630 nM T20251 CE9QH0 145993537 IC50 = 16000 nM T20251 CW4O5A 145993860 IC50 > 40000 nM T20251 CN7EF3 145996526 IC50 > 40000 nM T20251 CHJ79V 145997874 IC50 > 30000 nM T20251 C3XF1S 145998078 IC50 = 30 nM T20251 CQR6C0 145998079 IC50 = 30 nM T20251 C0XEI1 145999051 IC50 > 1000 nM T20251 C6ME3G 145999062 IC50 > 1000 nM T20251 CF8Z2A 145999065 IC50 > 1000 nM T20251 CG1UY7 145999069 IC50 > 1000 nM T20251 C2KI5O 145999070 IC50 > 1000 nM T20251 CGE6S8 145999072 IC50 > 1000 nM T20251 C9XP0T 145999073 IC50 > 1000 nM T20251 CSM74D 145999085 IC50 > 1000 nM T20251 C6TK4I 145999086 IC50 > 1000 nM T20251 C9N6TA 145999163 IC50 > 1000 nM T20251 CZH5T4 145999312 IC50 > 1000 nM T20251 C4PIK7 145999315 IC50 > 1000 nM T20251 C7K0GD 145999319 IC50 > 1000 nM T20251 CY78CJ 145999744 IC50 > 1000 nM T20251 CSJ8R5 145999926 IC50 > 1000 nM T20251 CP89RK 145999927 IC50 > 1000 nM T20251 CXM20T 145999998 IC50 > 1000 nM T20251 CIL13H 145999999 IC50 > 1000 nM T20251 CW4K1Z 146000086 IC50 > 1000 nM T20251 C12WMX 146000087 IC50 > 1000 nM T20251 CAK72D 146000156 IC50 > 1000 nM T20251 C4T8EB 146000260 IC50 > 1000 nM T20251 C1ALS9 146000261 IC50 > 1000 nM T20251 CWTJ89 146000454 IC50 > 1000 nM T20251 CJ53IP 146000455 IC50 > 1000 nM T20251 CCL2Y6 146000550 IC50 > 1000 nM T20251 CR1P2S 146000752 IC50 > 1000 nM T20251 CM84OD 146001043 IC50 > 1000 nM T20251 C4HL7W 146001118 IC50 > 1000 nM T20251 C80YAQ 146001119 IC50 > 1000 nM T20251 CX8IG6 146001227 IC50 > 1000 nM T20251 C7QRP1 146001228 IC50 > 1000 nM T20251 CTYG98 146001229 IC50 > 1000 nM T20251 C2RJ1U 146176418 IC50 = 830 nM T20251 C8Z9OM 146205579 IC50 > 40000 nM T20251 CDYH19 146301731 IC50 > 30000 nM T20251 C7XPS6 146304252 IC50 > 30000 nM T20251 CFR58K 146304329 IC50 > 30000 nM T20251 C1TAC4 146499656 IC50 > 40000 nM T20251 C8P3GC 146499745 IC50 > 40000 nM T20251 C6JBU1 146538921 IC50 > 40000 nM T20251 CXG41R 146538922 IC50 > 40000 nM T20251 CSBC71 146680900 IC50 = 2400 nM T20251 C9YJZ5 147180858 IC50 = 979 nM T20251 C87WVL 147388287 IC50 = 6900 nM T20251 CB3N4D 151194558 IC50 = 180 nM T20251 C9L7IH 151773717 IC50 = 2700 nM T20251 CF4L1I 152092486 IC50 = 1530 nM T20251 CHD2X0 153404509 IC50 = 112100 nM T20251 C5LXC4 153605593 IC50 > 30000 nM T20251 CH61KN 153635907 IC50 = 160 nM T20251 C80USW 153635929 IC50 = 1520 nM T20251 CY2D5Z 153635933 IC50 = 1470 nM T20251 C2Z1JC 153635944 IC50 = 330 nM T20251 CC9LJ8 153635955 IC50 = 650 nM T20251 CV4LT9 153635960 IC50 = 1900 nM T20251 C9A5HO 153635975 IC50 = 410 nM T20251 C1SPV6 154726271 IC50 > 30000 nM T20251 CZE1S5 155126870 IC50 > 33000 nM T20251 CI6EB5 155126882 IC50 > 33000 nM T20251 CY1ZH2 155510358 IC50 = 13070 nM T20251 C2X3QO 155510360 IC50 > 30000 nM T20251 C9UF6S 155510524 IC50 = 1200 nM T20251 CYGN68 155510554 IC50 > 20000 nM T20251 CF2CU8 155510758 IC50 = 19000 nM T20251 CRD8I0 155510888 IC50 = 9410 nM T20251 C26NCB 155511048 IC50 = 4000 nM T20251 C7VS5G 155511937 IC50 = 18700 nM T20251 CXFK79 155512104 IC50 = 28200 nM T20251 CXW4J6 155512369 IC50 > 33000 nM T20251 CR1Z8A 155512529 IC50 = 2600 nM T20251 C8B0WD 155512870 IC50 > 50000 nM T20251 CVCK17 155513135 IC50 > 30000 nM T20251 C7L4TB 155513385 IC50 > 50118.72 nM T20251 CG73TZ 155513551 IC50 > 33000 nM T20251 CZEO50 155513953 IC50 = 25118.86 nM T20251 C2HPU4 155514097 IC50 = 678 nM T20251 C6M9EW 155514111 IC50 > 30000 nM T20251 CO09EN 155514507 IC50 = 4400 nM T20251 CD53LC 155514863 IC50 > 25000 nM T20251 C4JX1E 155514986 IC50 > 50118.72 nM T20251 C19KDA 155515076 IC50 = 2500 nM T20251 C86NAI 155515209 IC50 > 30000 nM T20251 C1DVH0 155515264 Ki = 1080 nM T20251 CPZ1J2 155515757 IC50 = 6400 nM T20251 CW4IZ2 155515867 IC50 > 30000 nM T20251 CCV0U2 155515900 IC50 = 5200 nM T20251 CDP7E5 155516065 IC50 > 31622.78 nM T20251 CHK09I 155516513 IC50 = 32300 nM T20251 C1OJ2X 155516584 IC50 = 8000 nM T20251 CVP8Q5 155516616 IC50 = 31120 nM T20251 CRW92X 155516645 IC50 > 30000 nM T20251 CH8YG1 155516670 Ki = 1020 nM T20251 CP1L3J 155516697 IC50 = 7100 nM T20251 C3PLC9 155516907 IC50 = 4000 nM T20251 CA3K9P 155517032 IC50 > 25000 nM T20251 C2X8HA 155517088 IC50 > 30000 nM T20251 CD9C4L 155517220 IC50 = 380 nM T20251 CY5UE9 155517299 Ki > 30000 nM T20251 CZ0RI7 155517469 IC50 = 17000 nM T20251 CYX2T8 155517511 IC50 = 26100 nM T20251 CU35GB 155517528 IC50 = 3 nM T20251 C01JPW 155517641 IC50 = 40477 nM T20251 CC2A9K 155517811 IC50 = 300 nM T20251 CXTR57 155518069 IC50 = 25900 nM T20251 CL1K2F 155518339 IC50 = 28800 nM T20251 C3XW1B 155518561 Ki = 14300 nM T20251 CRD79Z 155518589 IC50 > 25000 nM T20251 CY49NZ 155518625 IC50 > 20 nM T20251 CGCO97 155518865 IC50 = 16630 nM T20251 CVS35D 155518925 IC50 = 19000 nM T20251 CVH0P8 155519454 IC50 = 7943.28 nM T20251 CY1EN6 155519472 IC50 = 5300 nM T20251 C5KZG7 155519527 IC50 = 18000 nM T20251 C26VPM 155520046 IC50 > 10000 nM T20251 C1PJC7 155520619 IC50 > 33000 nM T20251 CKD52G 155520766 IC50 = 6060 nM T20251 CM0IC7 155521232 IC50 = 7943.28 nM T20251 C76JKY 155521282 Ki > 30000 nM T20251 CY2CK4 155521688 IC50 = 7500 nM T20251 C1M6KY 155521903 IC50 = 400 nM T20251 CQ06BH 155521919 IC50 = 38000 nM T20251 CZ8FN1 155522016 IC50 = 17270 nM T20251 CX41RI 155522177 IC50 = 21100 nM T20251 CGQ1X0 155522363 IC50 > 10000 nM T20251 C0ZXV4 155522886 IC50 > 25000 nM T20251 CAL9M0 155523067 IC50 > 50118.72 nM T20251 CAGO28 155523111 IC50 = 2110 nM T20251 CM1BV9 155523387 Ki > 60000 nM T20251 CH06BN 155523388 Ki = 820 nM T20251 CES5L2 155523448 IC50 > 10000 nM T20251 C37RVF 155523599 IC50 = 1500 nM T20251 C2LO4Y 155523731 IC50 > 25000 nM T20251 C15BIV 155523740 IC50 = 4200 nM T20251 C38OCA 155524170 IC50 = 2920 nM T20251 CVA8H7 155524476 IC50 > 30000 nM T20251 CLMK45 155524544 IC50 > 40000 nM T20251 C2EHI7 155524928 IC50 = 15848.93 nM T20251 CG71WI 155525128 IC50 > 25000 nM T20251 C94NTW 155525132 Ki = 9200 nM T20251 CMY98L 155525177 IC50 = 5600 nM T20251 C7E3UM 155525341 IC50 > 40000 nM T20251 CY7EM6 155525492 IC50 = 5 nM T20251 CZW45D 155525803 IC50 > 63095.73 nM T20251 C24PLM 155525923 IC50 = 553 nM T20251 CX59UT 155526046 IC50 = 1.1 nM T20251 CSI0N2 155526143 IC50 > 10000 nM T20251 C3W1DA 155526172 IC50 > 30000 nM T20251 CIR3K1 155526251 IC50 > 50118.72 nM T20251 CS05UF 155526423 IC50 > 10000 nM T20251 C17HOP 155526864 IC50 = 35500 nM T20251 CQ4XA9 155527433 IC50 > 20000 nM T20251 CL8Z3K 155527451 IC50 > 50118.72 nM T20251 C04OAY 155527550 IC50 = 50100 nM T20251 CT4B0F 155527719 Ki = 20050 nM T20251 C0DZ9X 155527985 IC50 = 7943.28 nM T20251 C05QTC 155528035 IC50 > 25000 nM T20251 CS0ER5 155528109 IC50 = 6100 nM T20251 CT1JB7 155528212 Ki = 3750 nM T20251 CHR60D 155528366 Ki = 10700 nM T20251 CN7I6O 155528434 Ki = 10750 nM T20251 CRGO31 155528777 IC50 = 17100 nM T20251 C5H9NQ 155529107 IC50 > 10000 nM T20251 C5QA2B 155529241 IC50 > 25000 nM T20251 C9L6OC 155529247 IC50 > 30000 nM T20251 C9U8FN 155529326 Ki > 30000 nM T20251 CW5TM8 155529670 IC50 > 31622.78 nM T20251 C8UM7E 155530060 IC50 > 10000 nM T20251 CFRQ41 155530069 IC50 = 32850 nM T20251 C4F7WU 155530183 IC50 = 8780 nM T20251 CBOJ48 155530271 IC50 > 50118.72 nM T20251 CQ6F7O 155530369 IC50 > 25000 nM T20251 C2WPD6 155530588 IC50 = 11000 nM T20251 C4L7ZO 155530653 Ki = 4100 nM T20251 CYH2Z6 155530878 IC50 = 14000 nM T20251 CCGZ20 155530937 IC50 > 32000 nM T20251 C5N7PS 155530991 IC50 = 2360 nM T20251 C86HGK 155531857 IC50 = 22000 nM T20251 CY59IV 155531989 IC50 = 1.4 nM T20251 CW14TB 155532044 IC50 = 1480 nM T20251 CQU09F 155532106 IC50 = 10000 nM T20251 CFL61W 155532250 IC50 > 10000 nM T20251 CZF0X4 155532360 IC50 > 10000 nM T20251 C7UBH8 155532385 Ki = 20230 nM T20251 CWEZ83 155532537 IC50 > 10000 nM T20251 C8IP7E 155532982 IC50 > 20000 nM T20251 CFR56S 155533031 IC50 > 50118.72 nM T20251 C5TFA7 155533222 IC50 > 10000 nM T20251 CAT9V1 155533370 IC50 > 30000 nM T20251 C6R8JM 155533521 IC50 > 50118.72 nM T20251 CZ3DW6 155533821 IC50 > 30000 nM T20251 CF2MD7 155533927 Ki = 24800 nM T20251 CGH63O 155534464 IC50 = 5400 nM T20251 CL7U8D 155534608 IC50 = 3 nM T20251 C82LDF 155534740 IC50 > 50118.72 nM T20251 C63HSA 155534748 IC50 > 30000 nM T20251 CVBC47 155535120 IC50 = 12000 nM T20251 C71YMQ 155535169 IC50 < 100 nM T20251 CNA92P 155535177 IC50 = 30000 nM T20251 CX7PM4 155535638 IC50 > 12589.25 nM T20251 CC5HJ6 155535796 IC50 = 18900 nM T20251 CHOC87 155535920 IC50 = 40000 nM T20251 C9JD7A 155535968 IC50 = 39810.72 nM T20251 C3F8NR 155536006 IC50 > 31622.78 nM T20251 C0BH6W 155536009 IC50 > 25000 nM T20251 CN07PE 155536057 IC50 > 30000 nM T20251 CDL9R5 155536374 IC50 = 5248.07 nM T20251 C52GJS 155536419 IC50 = 1500 nM T20251 CRI0X6 155536978 IC50 = 3200 nM T20251 CG6P2Z 155537026 IC50 = 80000 nM T20251 CY32TQ 155537053 IC50 = 8100 nM T20251 C8YO9Q 155537362 IC50 = 4 nM T20251 CY3S0M 155537382 IC50 = 14000 nM T20251 CL53AK 155537567 IC50 = 21700 nM T20251 CM3PB2 155537682 IC50 > 25000 nM T20251 CA0T9E 155537745 IC50 = 8450 nM T20251 CG8I5F 155538033 IC50 > 33000 nM T20251 C2APW9 155538169 IC50 = 32000 nM T20251 C6KX1G 155538348 IC50 = 6300 nM T20251 C4OEL6 155538351 IC50 = 5011.87 nM T20251 CUS3I9 155538644 IC50 > 25000 nM T20251 C8QX7D 155538795 Ki = 1200 nM T20251 CKNZ09 155539203 IC50 = 2900 nM T20251 CF6E1H 155539416 IC50 = 4740 nM T20251 CXV14T 155539760 IC50 = 2100 nM T20251 CCG68S 155539794 IC50 > 30000 nM T20251 C5Y4UG 155540068 IC50 = 2500 nM T20251 CK1G0I 155540170 IC50 = 4100 nM T20251 CD6J8H 155540340 IC50 = 2700 nM T20251 CDQF20 155540443 IC50 > 30000 nM T20251 CW2V3F 155540455 IC50 = 3000 nM T20251 CSMI71 155540479 Ki = 8200 nM T20251 CP2NY0 155540484 IC50 > 100000 nM T20251 C7LIO1 155540498 IC50 = 590 nM T20251 CFW15C 155540816 IC50 = 8540 nM T20251 C8WRH2 155540919 IC50 = 6400 nM T20251 CH6ND7 155541175 IC50 = 356180 nM T20251 C2IJL1 155541368 IC50 > 30000 nM T20251 CWQ7F0 155541490 IC50 = 5 nM T20251 CP2K9D 155541549 IC50 = 4400 nM T20251 C9SIN5 155541564 IC50 = 22000 nM T20251 C13HGT 155541849 IC50 = 2100 nM T20251 CQI12H 155541951 Ki = 2940 nM T20251 CL18DI 155542104 IC50 = 2200 nM T20251 C8PS6H 155542274 IC50 = 67800 nM T20251 C5T9KE 155542416 IC50 > 30000 nM T20251 CGKM58 155542422 IC50 = 17600 nM T20251 C2ZNB4 155542480 IC50 = 3900 nM T20251 CIPG54 155542639 IC50 = 3600 nM T20251 CWO01S 155542792 IC50 = 1700 nM T20251 CY8PB1 155542894 IC50 = 4000 nM T20251 CVNR95 155542898 IC50 > 30000 nM T20251 CDZ78J 155542932 IC50 = 6310 nM T20251 CU6H9N 155543153 IC50 > 10000 nM T20251 CKIJ48 155543371 IC50 = 360 nM T20251 C1FG3H 155543475 IC50 = 4500 nM T20251 CG7D9R 155543873 IC50 = 3300 nM T20251 CL9Z6H 155543895 IC50 = 7560 nM T20251 CF1AJ2 155544000 IC50 = 25118.86 nM T20251 CST86Y 155544326 Ki = 6540 nM T20251 CD9KW4 155544699 Ki = 18980 nM T20251 C8WGH1 155544876 IC50 = 12589.25 nM T20251 C7SQX2 155544997 IC50 = 1100 nM T20251 CURJ73 155545015 IC50 = 11000 nM T20251 C4I9LA 155545020 IC50 = 17900 nM T20251 CND38C 155545031 IC50 > 100000 nM T20251 CPB87M 155545130 IC50 = 1.7 nM T20251 C9H1RS 155545131 IC50 = 3600 nM T20251 CK4OU8 155545400 Ki = 9800 nM T20251 C9BVD8 155545737 IC50 > 50000 nM T20251 C8YG3O 155545771 IC50 > 10000 nM T20251 C2E5BY 155545899 IC50 > 30000 nM T20251 CB62FS 155546028 IC50 = 5400 nM T20251 CUI35S 155546230 IC50 = 13200 nM T20251 C6KXY5 155546286 IC50 = 2300 nM T20251 CPK82D 155546294 IC50 = 13000 nM T20251 CQSI68 155546312 IC50 > 10000 nM T20251 CD2PX1 155546796 IC50 = 9900 nM T20251 CI92YC 155546800 Ki = 12120 nM T20251 C7LZ3W 155546850 IC50 = 39810.72 nM T20251 C0VY9U 155547183 Ki = 5900 nM T20251 CH94MI 155547266 IC50 = 5500 nM T20251 CRN8Z6 155547317 IC50 > 31622.78 nM T20251 CQ6D2C 155547369 IC50 > 40000 nM T20251 CC83QJ 155547453 IC50 > 10 nM T20251 CU2QO9 155547462 IC50 = 8900 nM T20251 CQ62MW 155547536 IC50 = 450 nM T20251 CZ30SI 155547634 IC50 = 6309.57 nM T20251 CY6F3D 155547951 IC50 = 1600 nM T20251 CK3B4X 155548125 IC50 = 5900 nM T20251 CG8FO4 155548512 IC50 = 1100 nM T20251 CFD4W6 155548620 IC50 > 10000 nM T20251 C14SPW 155548636 IC50 = 8950 nM T20251 CRY3A2 155548898 IC50 > 30000 nM T20251 CNX8L6 155549162 Ki = 4100 nM T20251 CTQ9Y4 155549436 IC50 > 10000 nM T20251 CJD38X 155549583 IC50 = 10000 nM T20251 C0DHX7 155550192 IC50 = 1071.52 nM T20251 C8JI1D 155550286 IC50 = 1200 nM T20251 CAJ57R 155550406 IC50 = 2000 nM T20251 CEDN41 155550408 IC50 = 3 nM T20251 CR8DO6 155550599 IC50 = 830 nM T20251 C29BAV 155550731 IC50 = 1750 nM T20251 CWC8X9 155550748 IC50 > 30000 nM T20251 CHDG36 155550819 IC50 > 25000 nM T20251 CA5G2T 155551013 IC50 = 15300 nM T20251 CN9LP5 155551221 IC50 = 15000 nM T20251 CB73CQ 155551312 IC50 = 4 nM T20251 CZ7K0T 155551653 IC50 > 10000 nM T20251 C5LTO0 155551695 IC50 = 620 nM T20251 CK5F8L 155551725 IC50 > 10000 nM T20251 C5T3VG 155551984 IC50 = 13000 nM T20251 CJL9K4 155552042 IC50 = 1900 nM T20251 C26SHF 155552468 IC50 > 10000 nM T20251 CK52WB 155552587 IC50 = 1260 nM T20251 CGV1M3 155552611 IC50 = 3500 nM T20251 C1DV5G 155552667 IC50 = 21100 nM T20251 CX6QO1 155552713 IC50 = 670 nM T20251 CEN80B 155552714 IC50 = 1600 nM T20251 C2ZNL8 155552880 IC50 = 4300 nM T20251 C2QPM5 155553335 IC50 = 500 nM T20251 CN1B6E 155553350 IC50 = 1408 nM T20251 CUH7R2 155553391 IC50 > 10000 nM T20251 CORH39 155553574 IC50 > 20000 nM T20251 CT9S6V 155553775 IC50 > 10000 nM T20251 C09TOV 155553799 IC50 = 3600 nM T20251 CH18PL 155553803 IC50 = 19700 nM T20251 C7JCS2 155553955 IC50 > 25000 nM T20251 CRI95M 155554023 IC50 > 50000 nM T20251 CHP3R7 155554099 IC50 = 2100 nM T20251 C0I4KF 155555078 IC50 = 18000 nM T20251 CF78YP 155555080 IC50 > 30000 nM T20251 CGJO65 155555092 IC50 = 10600 nM T20251 CS8C4B 155555411 IC50 = 2800 nM T20251 C7TAB2 155555536 IC50 = 3100 nM T20251 C8Q2FG 155555556 IC50 > 30000 nM T20251 C76IMR 155555589 IC50 = 3500 nM T20251 C09FGY 155555863 IC50 > 25000 nM T20251 COK95C 155555928 IC50 > 12589.25 nM T20251 CRA05Z 155555980 IC50 > 12589.25 nM T20251 CFRD75 155555996 Ki > 40000 nM T20251 CIK75H 155556042 IC50 > 25000 nM T20251 C3TZ1X 155556063 IC50 = 9600 nM T20251 C8PI6V 155556175 Ki = 3560 nM T20251 CL8K4E 155556216 IC50 > 50000 nM T20251 CG80ZH 155556340 IC50 = 13300 nM T20251 C3WT2Q 155556441 IC50 > 30000 nM T20251 C7AZ5J 155556578 IC50 > 50118.72 nM T20251 CIY5U0 155556737 IC50 = 19952.62 nM T20251 C4AG5W 155557133 IC50 > 10000 nM T20251 CHVI34 155557396 IC50 = 2000 nM T20251 CK52DB 155557515 IC50 = 1400 nM T20251 CEX1O2 155557657 IC50 = 2350 nM T20251 C0T6WM 155558045 Ki > 30000 nM T20251 C2A1ZD 155558144 IC50 > 10000 nM T20251 CXD56L 155558183 IC50 > 10000 nM T20251 CR41JN 155558349 Ki = 5700 nM T20251 C92NTS 155558433 IC50 = 2500 nM T20251 CP31BL 155558617 IC50 > 1000 nM T20251 C4HPK2 155558743 IC50 > 25000 nM T20251 C9D1UW 155558867 IC50 = 7840 nM T20251 C4D1AF 155559052 IC50 = 18200 nM T20251 CJ82WQ 155559138 IC50 > 100000 nM T20251 CM0UH7 155559265 IC50 > 20 nM T20251 CKZT21 155559364 IC50 > 33000 nM T20251 C2AGR5 155559542 IC50 = 240 nM T20251 CTI7O1 155559782 IC50 = 10000 nM T20251 CKT84D 155559905 IC50 = 5200 nM T20251 CEF9N6 155560028 IC50 < 10000 nM T20251 C1U4ZL 155560181 IC50 = 280 nM T20251 CF4LM6 155560880 IC50 > 25000 nM T20251 CW3RA2 155561008 IC50 = 2500 nM T20251 CZ4BY2 155561096 Ki > 25000 nM T20251 CLO3B1 155561152 IC50 = 12000 nM T20251 CM7ZG9 155561160 IC50 > 25000 nM T20251 C9UYA8 155561280 IC50 = 5100 nM T20251 COSE65 155561444 IC50 = 10000 nM T20251 CM9L3Z 155561503 IC50 > 25000 nM T20251 C9HIU5 155561551 IC50 > 25000 nM T20251 CH9UY6 155562079 IC50 = 10000 nM T20251 C6T2RV 155562253 IC50 < 10000 nM T20251 CP52DQ 155562348 IC50 = 760 nM T20251 CS3T7F 155562863 IC50 = 2400 nM T20251 CWM03V 155563050 IC50 > 30000 nM T20251 CM23AF 155563334 IC50 > 10000 nM T20251 C85CNT 155563518 IC50 = 600 nM T20251 CAN0G3 155563660 IC50 = 1183 nM T20251 CG9QR6 155563968 IC50 = 680 nM T20251 CWOE21 155564042 IC50 > 30000 nM T20251 CFT46O 155564074 IC50 = 15000 nM T20251 CZ6TP2 155564129 IC50 = 300 nM T20251 CU7O1C 155564384 Ki = 18100 nM T20251 CZR6W0 155564401 IC50 = 1700 nM T20251 CMK03D 155564568 IC50 > 25000 nM T20251 CC5FE7 155564581 IC50 > 30000 nM T20251 CB7SJ5 155564720 IC50 = 570 nM T20251 CMR8A9 155565213 IC50 > 10000 nM T20251 CWK95R 155565459 IC50 = 17000 nM T20251 CEO89S 155565478 IC50 = 2600 nM T20251 CL63KT 155565570 IC50 = 904350 nM T20251 CJL8Y5 155565696 Ki > 30000 nM T20251 C43CBF 155566090 IC50 = 6 nM T20251 CX52IW 155566155 IC50 = 7830 nM T20251 C7WTF8 155566556 IC50 = 1700 nM T20251 C26IRL 155566625 IC50 = 1500 nM T20251 CTVY40 155566771 IC50 = 4500 nM T20251 CC2Q9P 155566780 IC50 = 109010 nM T20251 CUIS06 155566980 IC50 = 5800 nM T20251 CXKI62 155567017 IC50 = 2300 nM T20251 C8HR4Q 155567029 IC50 = 2030 nM T20251 C5YX9V 155567261 IC50 = 20380 nM T20251 C37BGO 155567311 IC50 > 30000 nM T20251 C9KQW3 155567372 IC50 = 1900 nM T20251 C08ZCY 155567532 IC50 > 30000 nM T20251 C7KPT9 155567536 IC50 = 3100 nM T20251 CU34OH 155567589 IC50 > 10000 nM T20251 C16AQH 155567592 IC50 > 30000 nM T20251 CB19FR 155567818 IC50 > 40000 nM T20251 CD5FO3 155567866 IC50 > 50118.72 nM T20251 CK9N0Z 155567885 Ki > 10000 nM T20251 CS9GW7 155568268 IC50 = 11000 nM T20251 C9ZR8N 155568412 IC50 = 25100 nM T20251 CR5HK7 155568706 IC50 = 9400 nM T20251 C8INK5 155568740 IC50 = 11000 nM T20251 CUT84A 155568798 IC50 = 1000 nM T20251 C1S8ZB 155568922 IC50 = 2300 nM T20251 CSC8Q5 155569142 IC50 = 9500 nM T20251 CBJ5F8 155569464 IC50 = 2200 nM T20251 CP9TR0 10324985 Ki > 10000 nM T20251 CB0I4L 24884859 IC50 = 8111.11 nM T20251 C7Y0EQ 24885255 IC50 = 9500 nM T20251 CYV2S9 24885661 IC50 = 750 nM T20251 C5Z2KD 24886136 IC50 = 571.43 nM T20251 CS5N4V 24886137 IC50 = 296.7 nM T20251 CP2O0E 24886138 IC50 = 2555.56 nM T20251 CZO3R2 24886366 IC50 = 7714.29 nM T20251 C90ROZ 24886368 IC50 = 1109.59 nM T20251 C7BYA1 44254046 IC50 = 2000 nM T20251 C65JLI 44254219 IC50 = 1166.67 nM T20251 D00AWM 9826520 IC50 = 1170 nM T20251 D00CCV 11669239 Ki = 2200 nM T20251 D00FAY 13007806 IC50 = 1500 nM T20251 D00NCL 46836562 IC50 = 28000 nM T20251 D00TGC 56951318 Ki > 15000 nM T20251 D00UIN 11739248 IC50 = 1000 nM T20251 D00WKK 11710246 IC50 > 60000 nM T20251 D01ABR 44414723 IC50 = 5840 nM T20251 D01BWV 9802572 IC50 = 150 nM T20251 D01FFX 24691160 Ki = 3800 nM T20251 D01GPC 53235534 IC50 = 19000 nM T20251 D01IWD 159502 IC50 = 5888.44 nM T20251 D01JYY 11323940 Ki = 7000 nM T20251 D01MCD 25059294 IC50 = 120 nM T20251 D01PIU 44297094 IC50 = 3467368.5 nM T20251 D01PYU 9821248 Ki = 530 nM T20251 D02BPT 942 IC50 = 245470.89 nM T20251 D02DCM 44230874 IC50 = 9000 nM T20251 D02EIB 25129433 IC50 = 643 nM T20251 D02FQG 54579974 IC50 = 8240 nM T20251 D02NMN 23634102 IC50 = 31000 nM T20251 D02QJW 2798 IC50 = 12.59 nM T20251 D02TPY 25025860 IC50 = 1200 nM T20251 D02TSN 46244454 IC50 = 50000 nM T20251 D02WWM 175064 IC50 = 2.188 nM T20251 D03BQV 3033806 IC50 > 10000 nM T20251 D03NRJ 10871642 Ki = 2500 nM T20251 D03PIP 11568942 Ki = 2400 nM T20251 D03PSY 44542667 IC50 = 10 nM T20251 D03RBD 49765077 IC50 = 0.26 nM T20251 D03WAE 1301094 Ki = 4.8 nM T20251 D03XKL 11641429 Ki = 300 nM T20251 D04ALU 3076 IC50 = 17378.01 nM T20251 D04SAO 9799518 IC50 > 100000 nM T20251 D04TPA 72163809 IC50 = 21000 nM T20251 D04TWX 9794475 Ki > 4000 nM T20251 D05KUM 135446209 IC50 = 12589.25 nM T20251 D05LKO 44414722 IC50 = 22900 nM T20251 D05UZY 11539096 IC50 = 1600 nM T20251 D05VAB 9886249 IC50 = 100 nM T20251 D05VQJ 25147749 IC50 = 13240 nM T20251 D05XPV 54759259 IC50 > 25000 nM T20251 D05ZUX 44207909 IC50 = 20000 nM T20251 D06BMZ 46885513 IC50 > 65000 nM T20251 D06EMC 11392888 IC50 = 20000 nM T20251 D06HOI 44249821 IC50 > 80000 nM T20251 D06LJL 9916282 IC50 > 10000 nM T20251 D06MBD 11176403 IC50 = 8500 nM T20251 D06NXC 24996886 IC50 = 1460 nM T20251 D06NXK 46890563 Ki = 10000 nM T20251 D06QIQ 44592241 Ki = 3500 nM T20251 D07ADX 54764565 IC50 = 21000 nM T20251 D07ETF 9838960 Ki = 9599.99 nM T20251 D07GBV 10091189 Ki = 80 nM T20251 D07LFR 44231007 IC50 = 11000 nM T20251 D07SGS 44292136 IC50 = 130 nM T20251 D08CZT 9882067 Ki = 5700 nM T20251 D08EKQ 46890532 IC50 = 4950 nM T20251 D08JCU 44439386 Ki = 3900 nM T20251 D08NQA 57523213 IC50 = 12200 nM T20251 D08QBS 44178080 IC50 = 9500 nM T20251 D08RQW 49871766 Ki > 8000 nM T20251 D08TBU 15723 IC50 > 100000 nM T20251 D08ZIS 13007805 IC50 = 1600 nM T20251 D09BWE 11473281 IC50 > 30000 nM T20251 D09FGL 9910393 IC50 > 30000 nM T20251 D09FIC 46890395 IC50 = 10700 nM T20251 D09GZH 667538 IC50 = 810 nM T20251 D09HFT 44439376 Ki > 9000 nM T20251 D09KEB 11493841 IC50 = 3162.28 nM T20251 D09PTP 57325421 IC50 > 10000 nM T20251 D0A0GU 44247568 IC50 > 10000 nM T20251 D0A2BE 2780 IC50 = 602.56 nM T20251 D0A5KP 11588169 IC50 = 36000 nM T20251 D0A7GW 45487772 Ki = 12700 nM T20251 D0AT5N 56835134 IC50 = 16000 nM T20251 D0BD6A 10278617 IC50 > 30000 nM T20251 D0BW0V 44589528 IC50 = 1000 nM T20251 D0C2GE 67161540 IC50 = 3367 nM T20251 D0C2NK 4541 IC50 = 2290.87 nM T20251 D0C6BP 11567667 Ki = 8000 nM T20251 D0CM6T 11314340 IC50 = 13400 nM T20251 D0D6GI 46888441 IC50 > 10000 nM T20251 D0D8JU 46885546 IC50 > 60000 nM T20251 D0DA1E 23642319 Ki > 10000 nM T20251 D0DM6F 11761968 IC50 = 7000 nM T20251 D0E3DM 44592118 Ki = 15700 nM T20251 D0E7VO 59627005 IC50 > 32000 nM T20251 D0EG5G 46888467 IC50 > 10000 nM T20251 D0F9AM 86277846 Ki = 4.2 nM T20251 D0FF6S 16038374 IC50 > 30000 nM T20251 D0FJ1I 46891225 IC50 = 380 nM T20251 D0FL1D 9842124 Ki = 290 nM T20251 D0G4SU 65825 IC50 = 2500 nM T20251 D0G7LE 10991121 Ki = 1800 nM T20251 D0G8UA 46890321 IC50 > 10000 nM T20251 D0GG2J 46890492 IC50 = 760 nM T20251 D0H3GI 25129090 IC50 = 462 nM T20251 D0H8XV 12963076 IC50 = 900 nM T20251 D0I2UC 44230733 IC50 = 7000 nM T20251 D0J2YB 23631116 IC50 = 1600 nM T20251 D0JD4C 9853498 IC50 = 49900 nM T20251 D0K7RO 11646379 IC50 = 27500 nM T20251 D0L1UK 3064778 Ki = 7943.28 nM T20251 D0L9YP 44254503 IC50 = 11589 nM T20251 D0LM5H 11466357 EC50 = 8000 nM T20251 D0M1BJ 5282279 IC50 = 1500 nM T20251 D0N2DN 25129089 IC50 = 680 nM T20251 D0N2KU 44517677 IC50 > 20000 nM T20251 D0N6OL 11452268 IC50 = 10000 nM T20251 D0ND5D 10493741 Ki = 7000 nM T20251 D0O8AR 16097523 IC50 = 5200 nM T20251 D0OQ5H 46891330 IC50 = 40 nM T20251 D0OR6O 91623362 IC50 > 100000 nM T20251 D0P0QI 9816778 IC50 > 33000 nM T20251 D0P2HR 3510 IC50 = 3730 nM T20251 D0P6JS 11675054 IC50 = 16000 nM T20251 D0P7VQ 9929425 IC50 = 1000 nM T20251 D0P8PH 656732 IC50 > 32000 nM T20251 D0PC5A 44243144 IC50 = 30800 nM T20251 D0PC5N 71455 Ki > 150000 nM T20251 D0PF9Q 11472798 IC50 > 30000 nM T20251 D0Q8LS 11427736 IC50 = 2000 nM T20251 D0QG6A 9980734 IC50 = 43651.58 nM T20251 D0R0TW 11964036 IC50 > 20000 nM T20251 D0R3XC 11524350 Ki > 10000 nM T20251 D0R5OF 46885515 IC50 > 30000 nM T20251 D0RC9T 9795587 IC50 = 4897.79 nM T20251 D0S1XC 25224941 IC50 = 4400 nM T20251 D0S9AY 44592244 Ki = 8500 nM T20251 D0S9CI 11989776 Ki > 9000 nM T20251 D0SN6R 44592197 Ki > 5500 nM T20251 D0T4QX 11646823 IC50 = 1000 nM T20251 D0T9VC 56840673 IC50 > 10000 nM T20251 D0TO6S 2396 IC50 = 1000 nM T20251 D0U7OD 16043230 IC50 = 6950 nM T20251 D0UG5M 9956146 Ki = 8820 nM T20251 D0V0YM 24871527 IC50 = 1000 nM T20251 D0V3ZG 25192022 IC50 > 3000 nM T20251 D0V8DH 53380803 IC50 = 580 nM T20251 D0V8KA 42645487 IC50 = 33000 nM T20251 D0W2FU 53347902 IC50 > 30000 nM T20251 D0W3XD 16049828 Ki > 8000 nM T20251 D0W7WV 11039077 Ki = 61400 nM T20251 D0W8CA 46846313 IC50 < 2800 nM T20251 D0X7HD 11184481 IC50 = 40000 nM T20251 D0X8GC 45487773 Ki > 10000 nM T20251 D0XF5P 44592119 Ki = 16400 nM T20251 D0Y3OO 11327430 IC50 = 14000 nM T20251 D0Y4BL 11676971 IC50 > 10000 nM T20251 D0Y8AB 46885586 IC50 > 60000 nM T20251 D0Z7TM 22273644 IC50 = 6600 nM T20251 D0Z8PT 54758482 IC50 = 5000 nM T20251 D0ZC3Q 44230732 IC50 = 9000 nM T76059 D06OMK 445643 Ki = 0.4 nM T76059 D0G7UX 5284373 Ki = 20 nM T76059 D02VJY 3037617 IC50 = 17 nM T76059 D04PGB 445501 Ki = 0.01 nM T76059 D06GSE 9906804 Ki = 1 nM T76059 CA9GD5 3504 Ki = 7.5 nM T76059 CO43LW 444590 IC50 = 1.8 nM T76059 C5PE3Q 445644 Ki = 10 nM T76059 CU90XH 654676 Ki > 30000 nM T76059 COQ2J6 3154008 Ki > 50000 nM T76059 CR81OM 3154010 Ki = 33000 nM T76059 CW0TS4 3219611 Ki > 50000 nM T76059 CB9XT6 3219624 Ki > 50000 nM T76059 C14GPZ 3221232 Ki > 50000 nM T76059 C57KPB 3817957 Ki = 33000 nM T76059 CKE6R9 3827638 IC50 = 2600 nM T76059 CK18XS 4320284 Ki = 2500 nM T76059 CEX07C 4919428 Ki = 30000 nM T76059 CZ71ST 4921127 Ki = 37000 nM T76059 C2HUW7 5282071 EC50 = 1.6 nM T76059 CBMA23 5289261 Ki = 3.5 nM T76059 CTVP96 9798935 Ki = 2 nM T76059 C9M6IN 9798937 Ki = 820 nM T76059 CB92GZ 9801420 Ki = 8.9 nM T76059 CO7BG6 9806733 Ki = 54 nM T76059 C1PNB2 9809312 Ki = 19 nM T76059 CZ7GL8 9809998 IC50 = 9.6 nM T76059 CRD1T0 9811664 IC50 > 100000 nM T76059 C6NUY1 9817974 Ki = 8000 nM T76059 CTW24K 9819275 Ki = 20000 nM T76059 CYC61Z 9819945 Ki = 6000 nM T76059 C9IS6O 9820942 Ki = 130 nM T76059 C1XZ6E 9824296 Ki = 52 nM T76059 CX8W7L 9827812 IC50 = 16000 nM T76059 CW65IP 9841778 Ki = 1482 nM T76059 CK1VQ4 9845338 Ki = 6 nM T76059 CAU04E 9847345 Ki = 86 nM T76059 C8FAH3 9847925 Ki = 870 nM T76059 C12GZJ 9865798 Ki = 470 nM T76059 CS7LG9 9866557 Ki = 34 nM T76059 C2C1OB 9870251 IC50 = 200 nM T76059 C0EXC1 9870370 Ki = 105 nM T76059 C7JUR0 9871036 Ki = 3 nM T76059 C2NUK6 9873530 Ki = 0.3 nM T76059 C5VPL6 9883775 Ki = 35000 nM T76059 C6O4DI 9885558 IC50 = 4400 nM T76059 CS6F8D 9885875 Ki = 250 nM T76059 CZN2C1 9885966 Ki = 131 nM T76059 CAJ08L 9891805 Ki = 5 nM T76059 CV1PE8 9895267 Ki = 20 nM T76059 CFO6C1 9903902 Ki = 1300 nM T76059 CCJ0D9 9906857 Ki = 42 nM T76059 CSR87K 9908335 Ki = 72 nM T76059 C58ZLO 9909789 Ki = 504 nM T76059 CX09OR 9928246 Ki = 742 nM T76059 CNF68M 9934108 Ki = 25 nM T76059 C3V6MH 9936215 Ki = 50 nM T76059 CV4D7Y 9936936 Ki = 332 nM T76059 C37WXC 9938653 Ki = 1 nM T76059 CN4Z9I 9955490 Ki = 7 nM T76059 CZ37BG 9960384 Ki = 1 nM T76059 CH89YV 9962928 Ki = 1 nM T76059 CB26MR 9962976 Ki = 1 nM T76059 C3R1PD 9981138 Ki = 280 nM T76059 CX4T5W 10056711 Ki = 1.5 nM T76059 C3YFU6 10079556 Ki = 6 nM T76059 C67NVY 10102537 Ki = 9 nM T76059 CRYA61 10112806 Ki = 360 nM T76059 CTLA57 10114768 Ki = 123 nM T76059 C0H6TX 10118511 Ki = 591 nM T76059 C7Y9UG 10138683 Ki = 420 nM T76059 C08VEM 10140711 Ki = 590 nM T76059 C03BSX 10155516 Ki = 12.2 nM T76059 C4CE6L 10161454 Ki = 104 nM T76059 C52TDP 10161566 Ki = 210 nM T76059 CIQH49 10161855 Ki = 150 nM T76059 C5PGQ8 10177566 Ki = 8.7 nM T76059 CV4IK3 10183195 Ki = 360 nM T76059 C0Y4IK 10183484 Ki = 82 nM T76059 CQN3P4 10198461 Ki > 10000 nM T76059 C8R5DX 10229698 Ki = 88 nM T76059 C7B0JO 10229811 Ki = 92 nM T76059 CS9HP2 10234693 Ki = 1 nM T76059 C57GIZ 10259637 IC50 = 0.77 nM T76059 C8DLF4 10260436 Ki = 38 nM T76059 C4RW1L 10260525 Ki = 7 nM T76059 C7GJ6Y 10276095 Ki = 84 nM T76059 C6GVC7 10301493 Ki = 640 nM T76059 CU7D3Z 10303855 Ki = 156 nM T76059 C2YUE4 10317191 Ki = 550 nM T76059 CSN72K 10371065 IC50 = 114 nM T76059 C4XD1F 10396050 Ki = 1 nM T76059 C1HOM8 10396073 IC50 = 2.9 nM T76059 CI4FP1 10396108 Ki = 10 nM T76059 C4O6QS 10463260 IC50 = 0.6 nM T76059 CZ0S3I 10463451 Ki = 29 nM T76059 CJ0LZ4 10474617 Ki = 11 nM T76059 CDFQ06 10486039 Ki = 3 nM T76059 CF3GI4 10508532 Ki = 900 nM T76059 CSIR58 10555604 IC50 = 40 nM T76059 CLOT05 10571272 IC50 = 116700 nM T76059 C6WJG4 10574954 Ki = 350 nM T76059 C0P3TN 10587060 Ki = 83000 nM T76059 C7F9PD 10618401 Ki = 570 nM T76059 CWDG54 10619661 Ki = 14000 nM T76059 C3IAZ8 10623440 Ki = 390 nM T76059 CR4IY5 10626978 IC50 = 1530 nM T76059 CC5DF2 10640341 Ki = 790 nM T76059 CL4C8T 10664741 IC50 = 21600 nM T76059 CE8TZ1 10668143 Ki = 370 nM T76059 CH9AV3 10685294 IC50 = 124100 nM T76059 C35GOE 10687366 IC50 > 200000 nM T76059 C1G6BY 10689335 Ki = 6500 nM T76059 CSO83D 10714474 Ki = 150 nM T76059 C12HRN 10715720 IC50 = 22300 nM T76059 CEVL01 10732772 IC50 = 3100 nM T76059 CF2A9U 10734201 Ki = 7200 nM T76059 C8TG7O 10741010 Ki = 220 nM T76059 CSYB76 10756782 Ki = 67000 nM T76059 C1K6HQ 10758826 Ki = 24000 nM T76059 CZ2OR8 10790307 Ki = 200 nM T76059 C63LIX 10834562 IC50 = 68200 nM T76059 C9TQ7U 11105029 EC50 = 21.1 nM T76059 C5NB9Z 11129344 IC50 = 17100 nM T76059 CO2RJ8 11181229 Ki = 137000 nM T76059 CZ29YS 11742535 Ki = 120 nM T76059 C0RHG3 11792025 Ki = 8400 nM T76059 CA1JR7 11800691 IC50 > 200000 nM T76059 CGR93V 11851094 Ki = 34 nM T76059 CR2BC8 11851095 Ki = 34 nM T76059 C58HTG 15380464 Ki = 725 nM T76059 C9VHU1 15380465 Ki = 130 nM T76059 C5WJK3 15380466 Ki = 30 nM T76059 CBG7J0 15380467 Ki = 60 nM T76059 C6UX1B 15380469 Ki = 12 nM T76059 C1O3HC 15380471 Ki = 20 nM T76059 CJ27ZQ 15380472 Ki = 103 nM T76059 CZI61J 15380473 Ki = 760 nM T76059 CGDE51 15380474 Ki = 210 nM T76059 CY4E8J 15380475 Ki = 32 nM T76059 C8IK5U 15380476 Ki = 24 nM T76059 CO0MS8 15516000 Ki = 110 nM T76059 C0S5YD 15545973 IC50 = 15 nM T76059 C7WJF0 15546641 EC50 = 9.2 nM T76059 C94PQN 16394002 Ki = 1500 nM T76059 CDK6Q3 16485668 Ki = 7600 nM T76059 CG12OR 20707827 Ki = 3 nM T76059 C6K9WT 20725894 Ki = 0.5 nM T76059 CW2F6L 21027754 Ki = 450 nM T76059 C0S5GA 21027755 Ki = 250 nM T76059 C9Y0RT 21027758 Ki = 18 nM T76059 CGA08F 21027759 Ki = 82 nM T76059 CH8C9X 21258251 Ki = 170 nM T76059 CFJ0N7 21258256 Ki = 13 nM T76059 COI19B 21363697 Ki = 143 nM T76059 C3C9LX 21363707 Ki = 54 nM T76059 CYT86D 21363714 Ki = 217 nM T76059 CEA2K3 22064769 Ki > 10000 nM T76059 CY4R0O 23555949 Ki = 42 nM T76059 CHG49U 24860365 Ki = 69 nM T76059 CH8EQ3 24860366 Ki = 85 nM T76059 C3C1RK 24860367 Ki = 126 nM T76059 CVU23R 24860368 Ki = 152 nM T76059 CWB04A 24860369 Ki = 171 nM T76059 C2JL4P 24860370 Ki = 201 nM T76059 CR0OU1 24860371 Ki = 225 nM T76059 CQ6K8G 24860372 Ki = 46 nM T76059 CTB24N 24860373 Ki = 60 nM T76059 CCXP98 24860374 Ki = 71 nM T76059 CKY5C1 24860375 Ki = 72 nM T76059 C83GJK 24860376 Ki = 100 nM T76059 C6SD1K 24860377 Ki = 110 nM T76059 C2LK7D 24860378 Ki = 123 nM T76059 C87AXJ 24860379 Ki = 131 nM T76059 CM3F2Y 24860380 Ki = 238 nM T76059 C0D4FK 24860381 Ki = 282 nM T76059 CQZ9I6 24860382 Ki = 583 nM T76059 CRZ43B 24860383 Ki = 586 nM T76059 CZ85UH 24860384 Ki = 1000 nM T76059 CK29UW 24860385 Ki = 153 nM T76059 C7I6EL 24860386 Ki = 20800 nM T76059 C61YFI 24860387 Ki = 208 nM T76059 CQIG36 24860388 Ki = 3100 nM T76059 C1V8WX 24860389 Ki = 91 nM T76059 CH3P2O 24860390 Ki = 31700 nM T76059 C5U9FE 24860391 Ki = 107 nM T76059 C63IOV 24860392 Ki = 110 nM T76059 C6IXT3 24860393 Ki = 114 nM T76059 CBKW67 24860394 Ki = 279 nM T76059 CJ73FA 24860395 Ki = 2300 nM T76059 C09HAI 24860396 Ki = 244 nM T76059 C6PFH1 24860397 Ki = 266 nM T76059 C5JY0D 24860398 Ki = 288 nM T76059 C84WFH 24860402 Ki = 183 nM T76059 CNLZ96 24860403 Ki = 236 nM T76059 CTLC58 35027274 IC50 = 100 nM T76059 CBX15K 42897553 Ki = 4700 nM T76059 CV1SX2 44265409 EC50 = 12 nM T76059 CBX13N 44269758 IC50 = 1.5 nM T76059 C6OUP3 44269765 IC50 = 19 nM T76059 CR9J7V 44269773 IC50 = 65 nM T76059 C2YM7N 44269774 IC50 = 126 nM T76059 C1Y8AV 44269775 IC50 = 94 nM T76059 CI27YN 44269786 IC50 = 273 nM T76059 CG5H3K 44269787 IC50 = 5.8 nM T76059 CM9EC2 44269801 IC50 = 133 nM T76059 CXYL79 44269804 IC50 = 590 nM T76059 C3RF5Y 44269806 IC50 = 4.4 nM T76059 CO5N4A 44269817 IC50 = 12 nM T76059 CUKA34 44269842 IC50 = 150 nM T76059 CDX04K 44269845 IC50 = 187 nM T76059 C0KXL4 44269846 IC50 = 43 nM T76059 C96LNO 44269847 IC50 = 3.8 nM T76059 CKEL40 44269849 IC50 = 19 nM T76059 CU5LH8 44269870 IC50 = 66 nM T76059 C6SN3J 44279552 IC50 > 1000 nM T76059 C18XMQ 44279663 IC50 > 1000 nM T76059 CBS95E 44279849 IC50 = 14 nM T76059 C1RAK8 44280039 Ki = 3.7 nM T76059 C69FGM 44280289 IC50 = 2.1 nM T76059 CYNR42 44280488 Ki > 10000 nM T76059 CYV0B7 44280537 Ki = 3100 nM T76059 CA29IB 44280566 Ki = 5200 nM T76059 C0ZX7Y 44280567 Ki = 6000 nM T76059 CFT18Q 44280568 Ki = 4400 nM T76059 CI47SZ 44280581 Ki = 7200 nM T76059 CUVJ79 44280582 Ki = 47000 nM T76059 C24LTB 44280606 Ki = 18000 nM T76059 C0WL4I 44280742 Ki = 420 nM T76059 C7WQH2 44280751 Ki = 480 nM T76059 CL8FN0 44280766 Ki = 320 nM T76059 CWHU46 44280776 Ki = 8000 nM T76059 C67YOK 44280790 Ki = 4400 nM T76059 CSKB97 44280791 Ki = 1400 nM T76059 CP6N8F 44280797 Ki = 3800 nM T76059 C0K8IC 44280799 Ki = 1300 nM T76059 C8VZY0 44280800 Ki = 12 nM T76059 CILS94 44280811 Ki = 86 nM T76059 C5G8JO 44280833 Ki = 32 nM T76059 C6C2KX 44280834 Ki = 2100 nM T76059 C6A0WV 44280845 Ki = 260 nM T76059 C8I9HQ 44280846 Ki = 2700 nM T76059 C7GN1W 44280850 Ki = 1500 nM T76059 CN2PS9 44280851 Ki = 850 nM T76059 C48DQA 44280852 Ki = 22 nM T76059 CN45YP 44280871 Ki = 1300 nM T76059 C0H6RY 44280888 Ki = 1000 nM T76059 C9N1YQ 44280917 Ki = 2300 nM T76059 CB1OE4 44280918 Ki = 47 nM T76059 C6UO7I 44280919 Ki = 740 nM T76059 CN9I3W 44280941 Ki = 1200 nM T76059 CK27HI 44280958 Ki > 50000 nM T76059 CFW93J 44280959 Ki > 50000 nM T76059 C56KBA 44281035 Ki = 400 nM T76059 CV1B3D 44281045 Ki = 120 nM T76059 C54BJK 44281046 Ki = 220 nM T76059 CS26ZL 44281058 Ki = 470 nM T76059 C7BIA5 44281072 Ki = 92 nM T76059 C43DEQ 44281082 Ki = 180 nM T76059 CCG2H5 44281092 Ki = 1200 nM T76059 CM96EN 44281103 Ki = 720 nM T76059 CXTP68 44281114 Ki > 50000 nM T76059 CO0VR5 44281130 Ki = 1300 nM T76059 CADL82 44281131 Ki = 22000 nM T76059 CKUR12 44281153 Ki > 50000 nM T76059 CLOF28 44281158 Ki = 820 nM T76059 C3OF7W 44281160 Ki = 9500 nM T76059 C6M8JF 44281206 Ki > 50000 nM T76059 CHG02K 44281207 Ki > 50000 nM T76059 C8UI7Y 44281208 Ki = 1100 nM T76059 CT69UY 44281209 Ki = 2400 nM T76059 CANW36 44281215 Ki = 32000 nM T76059 CJET58 44281216 Ki = 42000 nM T76059 COY8M2 44281230 Ki = 22000 nM T76059 CCJ91K 44281233 Ki = 2800 nM T76059 C5OJQ2 44281249 Ki > 50000 nM T76059 CJL61F 44281259 Ki > 50000 nM T76059 CWO5Q9 44281260 Ki > 50000 nM T76059 CDB38P 44281261 Ki = 24000 nM T76059 C1D9BI 44281262 Ki = 6300 nM T76059 CD2QG9 44281272 Ki = 5400 nM T76059 CV7TY3 44281280 Ki > 33000 nM T76059 C61NZB 44281286 Ki = 3900 nM T76059 CD7UC9 44281293 Ki > 50000 nM T76059 CO5E0F 44281298 Ki = 1300 nM T76059 COX6I8 44281299 Ki = 11000 nM T76059 CM7OB4 44281311 Ki = 13000 nM T76059 C65VBK 44281361 Ki = 640 nM T76059 C7WFB3 44281383 Ki = 1600 nM T76059 CPL10S 44281410 Ki = 1600 nM T76059 CP2RU7 44281411 Ki = 110 nM T76059 CHA8T5 44281412 Ki = 2200 nM T76059 C0WNT3 44281413 Ki = 13000 nM T76059 CZQC70 44281458 Ki > 50000 nM T76059 CP2K6S 44281459 Ki = 1400 nM T76059 CY36QT 44281487 Ki = 4200 nM T76059 CO57JP 44281695 Ki = 39000 nM T76059 CRG59M 44281696 Ki > 50000 nM T76059 C4RGM1 44287122 Ki = 207 nM T76059 CS3O2T 44294553 IC50 = 3.3 nM T76059 CFHW79 44294716 IC50 = 13 nM T76059 C8CM5N 44294717 IC50 = 5.6 nM T76059 C48QMD 44294726 IC50 = 2.4 nM T76059 CK3OQ4 44294727 IC50 = 2 nM T76059 CQ4G9T 44294866 IC50 = 470 nM T76059 C7V1GU 44294867 IC50 = 50 nM T76059 C0K7FS 44294868 IC50 = 180 nM T76059 C8DZ7M 44294869 IC50 = 500 nM T76059 CT36GW 44294871 IC50 = 9.4 nM T76059 CV65SR 44294876 IC50 = 46 nM T76059 CO0TL9 44294886 IC50 = 16 nM T76059 CSW9I5 44294887 IC50 = 3.2 nM T76059 CT7PM2 44294894 IC50 = 4 nM T76059 CN6AB9 44294895 IC50 = 170 nM T76059 CR0YF6 44294896 IC50 = 19 nM T76059 C8KJL3 44294897 IC50 = 71 nM T76059 CBZ7G2 44294938 IC50 = 180 nM T76059 CSBI84 44294939 IC50 = 570 nM T76059 CYL6X0 44294966 IC50 = 48 nM T76059 C3WK8M 44294990 IC50 = 0.4 nM T76059 CF8R6K 44295208 IC50 = 68 nM T76059 C1C9TW 44295523 Ki = 8.3 nM T76059 CU2A6K 44306123 EC50 = 18 nM T76059 C7WNM2 44306124 EC50 = 12 nM T76059 C86EOZ 44306135 EC50 = 13.6 nM T76059 C8T5NI 44306145 EC50 = 32 nM T76059 CF75NO 44306146 EC50 = 5.3 nM T76059 CUH17I 44306155 EC50 = 9 nM T76059 C6OQ4D 44306156 EC50 = 45 nM T76059 CN58YR 44306157 EC50 = 7.5 nM T76059 C8N7QZ 44306253 EC50 = 45 nM T76059 CD8O6N 44306280 EC50 = 7.5 nM T76059 C68IRQ 44306324 EC50 = 11.25 nM T76059 C46AQD 44309746 IC50 = 1.6 nM T76059 C72NFI 44309747 IC50 = 3.6 nM T76059 CTI60L 44309800 IC50 = 10 nM T76059 CMC52Q 44309855 IC50 = 74.8 nM T76059 COH7M3 44309856 IC50 = 5.1 nM T76059 C24URG 44309955 IC50 = 0.8 nM T76059 C1CD5Q 44309983 IC50 = 2.8 nM T76059 CZN4T6 44309984 IC50 = 0.7 nM T76059 C2C9GA 44312111 EC50 = 30 nM T76059 CW5ZR8 44312113 EC50 = 22 nM T76059 CO56DC 44312417 EC50 = 20.5 nM T76059 CER3Y9 44312559 EC50 = 7.4 nM T76059 CQ5H2I 44312595 EC50 = 12 nM T76059 CKO38Y 44337706 IC50 = 64 nM T76059 C4QJC3 44337851 IC50 = 26 nM T76059 CM38LX 44337859 IC50 = 12 nM T76059 CF4VZ3 44337877 IC50 = 8.2 nM T76059 C6V5LW 44337938 IC50 = 5.5 nM T76059 CP0U7C 44338501 IC50 = 200 nM T76059 C64ZIF 44340105 Ki = 175 nM T76059 C3FV8H 44340118 Ki = 190 nM T76059 CIS1X4 44340142 Ki = 5 nM T76059 CFR52J 44340151 Ki = 340 nM T76059 CU3O2I 44340152 Ki = 190 nM T76059 CLFQ54 44340165 Ki = 25 nM T76059 CK1A4T 44340166 Ki = 5 nM T76059 C5KSH2 44340326 Ki > 5000 nM T76059 C4D5TV 44340429 Ki = 6000 nM T76059 CKP76I 44340465 Ki = 400 nM T76059 C4KI2O 44340482 Ki = 130 nM T76059 CHV95O 44350652 Ki = 8100 nM T76059 CKQU96 44350663 Ki = 8300 nM T76059 C24PEN 44350671 Ki = 1500 nM T76059 CND94Q 44350709 Ki > 50000 nM T76059 C0YXR3 44350766 Ki = 1200 nM T76059 CZ6D5G 44350783 Ki = 10000 nM T76059 CJ6HO2 44360860 IC50 = 3.4 nM T76059 C0F3WL 44365027 Ki = 195 nM T76059 CXGI06 44365035 Ki = 12 nM T76059 CCA08O 44365058 Ki = 170 nM T76059 CVT27W 44365059 Ki = 120 nM T76059 CF97ST 44365150 Ki = 3 nM T76059 CNFK71 44365151 Ki = 95 nM T76059 CG96PA 44365152 Ki = 9 nM T76059 C2MQ1T 44365238 Ki = 70 nM T76059 C4RD0I 44365240 Ki = 116 nM T76059 CZ1QB9 44365271 Ki = 17 nM T76059 C50CGS 44365344 Ki = 78 nM T76059 C47LAT 44365384 Ki > 10000 nM T76059 C6FI7B 44365447 Ki = 107 nM T76059 CK0YA4 44365450 Ki = 194 nM T76059 CI59UY 44365487 Ki = 40 nM T76059 CSH76C 44365490 Ki = 17 nM T76059 CLBE84 44365587 Ki = 15 nM T76059 C5FR3M 44368603 Ki = 32 nM T76059 CRTX63 44368604 IC50 = 410 nM T76059 C0HB4I 44368605 Ki = 482 nM T76059 CJZ6I1 44368744 Ki = 1300 nM T76059 CAR35L 44383333 EC50 = 34.3 nM T76059 CZ50YE 44383482 EC50 = 23 nM T76059 C1FED5 44383746 EC50 = 12 nM T76059 CB1P6R 44383908 EC50 = 11.8 nM T76059 C8R5WF 44383962 EC50 = 6.1 nM T76059 C6T4NQ 44384095 EC50 = 5.7 nM T76059 C79TFY 44384115 EC50 = 2.7 nM T76059 CE0X3V 44384116 EC50 = 6.6 nM T76059 CVM90W 44384124 EC50 = 9.2 nM T76059 CV19BZ 44384125 EC50 = 7 nM T76059 CSG64P 44384126 EC50 = 14.9 nM T76059 C65GRN 44384267 EC50 = 3.4 nM T76059 C02QJT 44385122 EC50 = 10.3 nM T76059 CQH7N8 44385184 EC50 = 15.6 nM T76059 C0TJ7O 44385185 EC50 = 4.6 nM T76059 CXA4S0 44387197 Ki = 250 nM T76059 CP96AN 44407027 Ki = 330 nM T76059 CKR3O4 44407127 Ki = 7000 nM T76059 C78BIN 44407142 Ki = 2700 nM T76059 CMUE21 44407218 Ki = 357 nM T76059 CZD8Y4 44407219 Ki = 772 nM T76059 CMY5V3 44461925 Ki = 210 nM T76059 C7YWU8 44461941 Ki = 2.8 nM T76059 CQA89Y 44461954 Ki = 112 nM T76059 C9JN0R 44461955 Ki = 258 nM T76059 CG51ZB 44461956 Ki = 68 nM T76059 CN68YV 44461964 Ki = 81 nM T76059 C7SZ3Q 50994120 IC50 > 30000 nM T76059 CX6PV4 50994121 IC50 = 2800 nM T76059 CY5FL8 50994123 IC50 > 30000 nM T76059 CNZ46O 50994197 IC50 = 4200 nM T76059 CGQF17 50994198 IC50 = 120 nM T76059 CBIR56 50994199 IC50 = 150 nM T76059 C4T1YW 50994200 IC50 = 70 nM T76059 CU51AK 50994201 IC50 = 320 nM T76059 CD3X0R 50994202 IC50 = 260 nM T76059 CID87X 51049455 Ki = 4.5 nM T76059 C2V6RJ 56962328 IC50 = 130 nM T76059 CJ46RD 56962330 IC50 = 343 nM T76059 C1BUW4 57521458 IC50 = 510 nM T76059 CGU89M 57521460 IC50 = 2450 nM T76059 CKP31Q 57521461 IC50 = 100 nM T76059 C7D3PN 57521557 IC50 = 1050 nM T76059 CO6T0F 57521558 IC50 = 150 nM T76059 C2RVN0 57521777 IC50 = 60 nM T76059 C8PY2R 57521778 IC50 = 50 nM T76059 C0HOD9 57521879 IC50 = 50 nM T76059 CS7B2A 57521880 IC50 = 60 nM T76059 CGP03D 57521881 IC50 = 1800 nM T76059 C9V4QB 57521882 IC50 = 1200 nM T76059 C4C7LK 57522005 IC50 = 1100 nM T76059 C8YI0U 57522006 IC50 = 10100 nM T76059 C0KC6J 57522007 IC50 = 4600 nM T76059 CH89PN 57522008 IC50 = 3800 nM T76059 CG6TK3 57522120 IC50 = 1900 nM T76059 CWQ8J7 57522121 IC50 = 1900 nM T76059 CTCH51 57522237 IC50 = 1090 nM T76059 C8R2IJ 57522238 IC50 = 320 nM T76059 C1PBX3 57522239 IC50 = 800 nM T76059 CU5NP7 57522240 IC50 = 6100 nM T76059 C0P3TI 57522347 IC50 = 7600 nM T76059 C6WY9D 57522348 IC50 = 600 nM T76059 CM7ZV1 57522349 IC50 = 1000 nM T76059 C6FQ4X 57522350 IC50 = 5100 nM T76059 CHVK79 57522455 IC50 = 2400 nM T76059 C73XQS 57522456 IC50 = 4500 nM T76059 C4OJX2 57522457 IC50 = 670 nM T76059 CGIX69 57522458 IC50 = 230 nM T76059 CG2SO6 57522567 IC50 = 1180 nM T76059 CR9C3F 57522569 IC50 = 1500 nM T76059 C8SP3L 57522570 IC50 = 2570 nM T76059 CQ3I7G 57522682 IC50 = 1200 nM T76059 C5QM2O 57522683 IC50 = 21 nM T76059 CE7G2U 57522684 IC50 = 660 nM T76059 CA4R9I 57522685 IC50 = 750 nM T76059 C3EP9M 57522800 IC50 > 100000 nM T76059 C46EIF 57522801 IC50 = 200 nM T76059 CC85GJ 57522802 IC50 > 50000 nM T76059 CCUW31 57522803 IC50 > 50000 nM T76059 CV58SP 57522927 IC50 = 800 nM T76059 CT58KB 57522928 IC50 = 115 nM T76059 C95OGY 57522929 IC50 > 50000 nM T76059 CZI07G 57522930 IC50 = 3 nM T76059 C8B9HE 57522931 IC50 = 450 nM T76059 C7Y9SK 57523063 IC50 = 550 nM T76059 C4S5KW 57523064 IC50 = 1290 nM T76059 CT4NB0 57523068 IC50 > 100000 nM T76059 C0NUH8 57523069 IC50 = 1400 nM T76059 C2YN0S 57523070 IC50 = 870 nM T76059 CG5AB2 57783590 IC50 = 6.8 nM T76059 C2DIM5 70684253 IC50 = 3380 nM T76059 CYQH64 70684260 IC50 = 470 nM T76059 CG5D2W 70688508 IC50 = 2200 nM T76059 CWDU09 70688522 IC50 = 570 nM T76059 C14GSV 70690624 EC50 = 5 nM T76059 CWY7C0 70692710 IC50 = 310 nM T76059 CF34ES 70694690 Ki = 0.7 nM T76059 C5MK3W 70694725 IC50 = 8100 nM T76059 CD65LN 70694726 IC50 = 9100 nM T76059 CEZG14 70694756 IC50 = 2780 nM T76059 CU9RN3 70694757 IC50 = 60 nM T76059 CRWB36 71718375 Ki = 2800 nM T76059 C61TIG 71718376 Ki = 870 nM T76059 CR9FQ3 71718981 Ki = 500 nM T76059 CK36QR 71720180 Ki = 2100 nM T76059 CUT2Y6 71720824 Ki = 27700 nM T76059 C0H2QE 73345516 Ki = 50 nM T76059 C5EMH2 86277875 Ki = 90 nM T76059 CXF34A 89939931 Ki = 8.8 nM T76059 C29TEF 101167236 Ki = 4000 nM T76059 CCH84L 117967740 Ki = 23400 nM T76059 CXP8S2 117967763 Ki = 2000 nM T76059 CEY28F 117967783 Ki = 12400 nM T76059 C46GRQ 117967787 Ki = 3800 nM T76059 C2A8EM 117967798 Ki = 12100 nM T76059 CVP4Q3 117967801 Ki = 120000 nM T76059 CWTL26 117967814 Ki = 1000 nM T76059 C5GF3N 117967822 Ki = 51900 nM T76059 CJ26YR 117967829 Ki = 30700 nM T76059 C2AF1T 117967843 Ki = 3200 nM T76059 CRCH91 117967851 Ki = 26900 nM T76059 CT3DQ5 117967872 Ki = 71100 nM T76059 C7NTU4 117967885 Ki = 50300 nM T76059 CYS70L 117967909 Ki = 101000 nM T76059 CU86WK 117967913 Ki = 6000 nM T76059 CFA74P 117967937 Ki = 10900 nM T76059 C08BKM 117967939 Ki = 11500 nM T76059 CHN52K 117967946 Ki = 5600 nM T76059 C1ZYL4 117967947 Ki = 1200 nM T76059 CA6ZJ7 117967955 Ki = 317000 nM T76059 C2QZ3D 117967964 Ki = 6600 nM T76059 C07HJM 117967978 Ki = 22500 nM T76059 CSD64M 117968002 Ki = 6600 nM T76059 CTI1X7 117968005 Ki = 6800 nM T76059 CXP8N7 117968006 Ki = 4300 nM T76059 C4LAX1 117968012 Ki = 8700 nM T76059 C58LQV 117968031 Ki = 30100 nM T76059 CF1GO9 117968050 Ki > 300000 nM T76059 CXLE07 117968053 Ki = 7500 nM T76059 CXWU20 117968117 Ki = 46900 nM T76059 CZQB61 117968118 Ki = 12800 nM T76059 CG65FE 117968136 Ki = 25100 nM T76059 C5O7SB 117968142 Ki = 39700 nM T76059 C5EU1T 117968149 Ki = 49200 nM T76059 CEXT51 117975049 Ki = 3000 nM T76059 CELN63 118233557 IC50 = 14.3 nM T76059 CJ84MI 118233582 IC50 = 9.52 nM T76059 CBP3S9 118233586 IC50 = 13.39 nM T76059 CUW1S0 118233596 IC50 = 12.61 nM T76059 CNP23H 122192627 Ki = 600 nM T76059 CEMN03 122192628 Ki = 1200 nM T76059 C5ZF3W 122192629 Ki = 300 nM T76059 CG2U4V 122693787 IC50 = 11.19 nM T76059 CPJ47S 122693793 IC50 = 12.48 nM T76059 C4YI9N 122693794 IC50 = 824 nM T76059 CC0L6K 127024999 Ki = 22300 nM T76059 C0SKD7 127053468 Ki = 4200 nM T76059 CHSY35 137631778 Ki = 7 nM T76059 CQ9F8R 137632505 IC50 = 10.99 nM T76059 C86IDH 137633267 Ki = 11.8 nM T76059 CWM7H1 137634012 Ki = 49 nM T76059 CGWE89 137639136 Ki = 249 nM T76059 C35SVI 137639141 Ki = 7 nM T76059 CAI70F 137640680 Ki = 21.1 nM T76059 CAM69O 137642452 Ki = 49 nM T76059 COK87T 137642715 IC50 = 19.2 nM T76059 C1P6LO 137642835 Ki = 0.45 nM T76059 CKL06A 137645398 IC50 = 23.6 nM T76059 C8DKV2 137649029 Ki = 7 nM T76059 C4IRT9 137649504 Ki = 49 nM T76059 C0EQ5V 137649552 Ki = 18.8 nM T76059 C9N2BM 137649843 IC50 = 27 nM T76059 CXSK64 137650264 Ki = 49 nM T76059 C93ENA 137650602 IC50 = 22.1 nM T76059 C7LYA9 137652507 Ki = 49 nM T76059 CC3LT2 137652724 IC50 = 19.1 nM T76059 CRLW34 137656432 IC50 = 12.59 nM T76059 CQR9J3 137657364 Ki = 143 nM T76059 CM05LU 137658940 Ki = 7 nM T76059 CHK6O9 137660768 Ki = 7 nM T76059 C8DI6S 137661451 IC50 = 22.6 nM T76059 CMA0I1 145980548 Ki = 5 nM T76059 C24MVU 145981935 Ki = 7 nM T76059 C6Z4QJ 145982171 IC50 = 53.6 nM T76059 CIRN21 145988906 Ki = 1 nM T76059 CP16HY 145989176 IC50 = 800 nM T76059 C61QME 155547348 Ki = 210 nM T76059 CGA13H 44287121 Ki = 400 nM T76059 D06ZWX 6197 Ki = 3400 nM T00663 D02NNV 3038525 IC50 > 5000 nM T00663 D02ZQS 16095342 IC50 > 10000 nM T00663 D03LWG 53235510 IC50 > 10000 nM T00663 D07EHV 44814409 IC50 > 10000 nM T00663 D0A6VD 25073775 IC50 = 160 nM T00663 D0HY9S 73386890 IC50 = 242 nM T00663 D0X4MN 11597537 IC50 = 6 nM T00663 D03BNU 59604787 IC50 > 10000 nM T00663 D05SJB 10040667 IC50 = 32 nM T00663 D08DNZ 45102739 IC50 = 11 nM T00663 D0PG5N 25123232 IC50 = 7750 nM T00663 D0UY9Y 46869000 IC50 = 800 nM T00663 D0W7MG 11647397 IC50 = 210 nM T00663 D0W8BL 46868926 IC50 = 9 nM T00663 D0ZU8L 57340689 IC50 = 9 nM T00663 D0F8DL 176155 Ki = 90 nM T00663 D0T3ME 156422 IC50 = 1400 nM T00663 C9W4UM 290221 IC50 = 1500 nM T00663 C5DB6Y 447872 IC50 = 1.6 nM T00663 C3V0TX 447873 IC50 = 1.6 nM T00663 C9VW8M 449054 IC50 > 16000 nM T00663 CKG76T 579429 IC50 = 3162.28 nM T00663 C0EQ6J 622378 IC50 > 15848.93 nM T00663 C2Y0RL 626628 IC50 > 15848.93 nM T00663 CQ9PB5 684674 IC50 > 15848.93 nM T00663 CR93CZ 746075 IC50 = 1830 nM T00663 CK89TF 766948 IC50 = 398.11 nM T00663 CWO49I 826287 IC50 > 15848.93 nM T00663 CVY4C5 847353 IC50 > 15848.93 nM T00663 CKS84B 897877 IC50 = 1000 nM T00663 CG2BU0 921636 Ki > 10000 nM T00663 C3PBJ1 942437 IC50 = 31800 nM T00663 C6K8WV 979869 IC50 = 1100 nM T00663 C4XP1N 1100747 IC50 = 3162.28 nM T00663 C8HP2S 1208196 IC50 = 2430 nM T00663 CG0IU6 1228584 IC50 = 1900 nM T00663 CRGB47 1228713 IC50 = 620 nM T00663 CV9D8Y 1228716 IC50 = 350 nM T00663 C67OWG 1228882 IC50 = 590 nM T00663 C5F4WM 1473242 Ki > 4000 nM T00663 C0VQG3 1483690 Ki = 13000 nM T00663 C2EX5Q 1641795 IC50 = 6570 nM T00663 CLBQ01 1737773 IC50 = 750 nM T00663 C5VE3K 2231029 IC50 = 1700 nM T00663 CF8Z5H 2766666 Ki = 5200 nM T00663 CQN85O 2766806 Ki = 9900 nM T00663 C8UC4F 2766824 Ki = 5000 nM T00663 C7IF4L 2766825 Ki = 6700 nM T00663 CZHL80 2808202 IC50 = 2200 nM T00663 CW6P5E 2823737 IC50 > 15848.93 nM T00663 C3KEG9 2823738 IC50 = 10000 nM T00663 C8WSF5 3659633 IC50 = 559 nM T00663 CR0DJ8 4078145 IC50 = 40 nM T00663 C69GSP 4079571 IC50 = 2700 nM T00663 CW26HV 5337145 IC50 = 14190 nM T00663 CSFQ07 9549178 IC50 = 3 nM T00663 CN8K3H 9814292 IC50 = 950 nM T00663 C7Q6PF 9818586 Ki = 720 nM T00663 C71GHF 9826147 IC50 > 10000 nM T00663 CW8V0K 9864418 IC50 > 16000 nM T00663 COR3S2 9892736 IC50 = 150 nM T00663 CX5G3A 9928616 IC50 = 30 nM T00663 CN0AJ9 9934347 IC50 = 12 nM T00663 C0V7UW 9958506 IC50 = 30 nM T00663 CO4B8A 9982333 IC50 > 10000 nM T00663 C37GXK 9983303 IC50 > 16000 nM T00663 C93OCY 10021870 IC50 = 175 nM T00663 C4PRY1 10066845 IC50 = 18 nM T00663 C2C1BP 10089048 IC50 > 16000 nM T00663 CLA50K 10091293 IC50 = 33 nM T00663 CPN3T4 10092520 IC50 = 32 nM T00663 CBJU36 10093433 IC50 = 26 nM T00663 CF1P3X 10094511 IC50 = 28500 nM T00663 C9NO1X 10149689 IC50 = 202 nM T00663 CYE4T2 10151272 IC50 = 21 nM T00663 CN0QK4 10152189 IC50 = 3.4 nM T00663 C69DHW 10158652 IC50 < 16000 nM T00663 CR47IV 10172440 IC50 = 32 nM T00663 CQU9K5 10200651 Ki > 4000 nM T00663 C7QHS0 10215642 IC50 = 5.3 nM T00663 C9PFR4 10225532 IC50 = 61.2 nM T00663 C1I0SL 10247954 IC50 = 7 nM T00663 C9NJ1X 10269964 IC50 = 70 nM T00663 C7SFI1 10296883 IC50 > 10000 nM T00663 CB59MP 10310219 IC50 = 1.9 nM T00663 CFL5O8 10364826 IC50 = 15 nM T00663 C72AVO 10372770 IC50 = 500 nM T00663 C2G3YH 10384284 IC50 = 652 nM T00663 CJE04Q 10384407 IC50 = 108 nM T00663 CFD01W 10452031 IC50 = 17 nM T00663 CB0E2X 10472936 IC50 = 20 nM T00663 CT92AO 10475988 IC50 = 528 nM T00663 CRBL32 10477561 IC50 = 693 nM T00663 CRX6F0 10479082 IC50 > 16000 nM T00663 CB47LY 10847715 IC50 > 15848.93 nM T00663 CIB8M9 11353316 IC50 = 10000 nM T00663 C0APW4 11422034 IC50 = 70 nM T00663 CMI8G3 11478147 IC50 = 13000 nM T00663 CJ9OH7 11538129 IC50 = 410 nM T00663 CTG83F 11539329 Ki = 72 nM T00663 CACS26 11561968 Ki > 4000 nM T00663 CO9KP5 11583459 IC50 > 10000 nM T00663 CMIL86 11590363 Ki = 61 nM T00663 C5B3XJ 11620410 IC50 > 40000 nM T00663 CHB3F2 11626055 IC50 = 572 nM T00663 CGX96V 11626927 IC50 < 15848.93 nM T00663 C9T6SC 11640926 Ki = 18 nM T00663 C9VP4Y 11655237 IC50 = 82 nM T00663 CJ9KN7 11683817 IC50 > 10000 nM T00663 CU0E8O 11690457 Ki > 4000 nM T00663 CB0AP2 11705863 Ki > 4000 nM T00663 CVX17E 11740117 IC50 = 32 nM T00663 CS36BH 11843159 IC50 > 5000 nM T00663 CBC08P 11846124 IC50 = 60 nM T00663 CD60CH 11846125 IC50 = 37 nM T00663 CAZS08 11848309 IC50 > 10000 nM T00663 C43IVN 11848567 IC50 > 10000 nM T00663 C9LAY8 11848825 IC50 > 10000 nM T00663 CC09DE 11955790 IC50 = 59 nM T00663 CIQ7M6 14198571 IC50 > 15848.93 nM T00663 CH19QA 15680125 IC50 > 15848.93 nM T00663 CBF4X2 15991561 IC50 = 3162.28 nM T00663 C8TW5P 16007071 IC50 = 2.5 nM T00663 CFPW41 16007116 IC50 = 120 nM T00663 C9TU1O 16046126 IC50 > 1000 nM T00663 CKR57M 16086104 IC50 > 5000 nM T00663 C16NRY 16086114 IC50 = 145 nM T00663 C7Z4LV 16095343 IC50 > 10000 nM T00663 CQG45C 16109001 IC50 = 40000 nM T00663 CK1SZ0 16115350 IC50 > 10000 nM T00663 CZL8G5 16115351 IC50 = 540 nM T00663 CRO0D5 16115352 IC50 = 3500 nM T00663 C0C5AZ 16129582 IC50 = 57 nM T00663 CU56EW 16664858 IC50 = 251.19 nM T00663 C0PS7U 16750106 IC50 = 150 nM T00663 C5IYQ1 17027307 IC50 = 810 nM T00663 CL9BQ6 17748275 IC50 = 40000 nM T00663 C4SPG1 19007057 Ki > 4000 nM T00663 CC1E7R 21078798 Ki > 4000 nM T00663 C95ORH 22261071 IC50 = 52 nM T00663 CE7K3W 23532567 IC50 > 10000 nM T00663 CR3M1N 23644582 Ki > 4000 nM T00663 CVOT06 24535122 IC50 = 6900 nM T00663 CV9U8E 24745781 IC50 > 10000 nM T00663 C9FJZ6 24779711 IC50 = 120 nM T00663 CIN29Y 24801862 IC50 = 3 nM T00663 CZ12SD 24801863 IC50 = 270 nM T00663 C16DKC 24810995 IC50 > 300 nM T00663 CC8Y1U 24810996 IC50 = 360 nM T00663 CH21WG 24810997 IC50 = 96 nM T00663 CQ1D8M 24810999 IC50 = 360 nM T00663 CNI4W8 24811099 IC50 = 680 nM T00663 C0MXK3 24811100 IC50 = 260 nM T00663 CFZN51 24811101 IC50 = 110 nM T00663 CRF71M 24811102 IC50 = 50 nM T00663 CB8A2T 24811103 IC50 > 10000 nM T00663 CJ7M8K 24823663 IC50 = 114 nM T00663 CX0S9L 24854902 IC50 = 9487 nM T00663 C1SVT2 24854903 IC50 > 10000 nM T00663 C61KPI 24856363 IC50 > 16000 nM T00663 C4OWF8 24875373 IC50 = 85 nM T00663 CY8L7E 24896769 IC50 > 10000 nM T00663 C8DG1Y 24941253 IC50 = 6626 nM T00663 C6CVK4 24959046 IC50 > 100000 nM T00663 CU7I2E 24963046 IC50 = 788 nM T00663 CS3Q8B 24995659 Ki > 4000 nM T00663 CD0TB3 25024184 IC50 = 129 nM T00663 C6NU1D 25071599 IC50 = 325 nM T00663 CXD9K3 25071600 IC50 = 61 nM T00663 CYJ8F1 25074077 IC50 = 1000 nM T00663 C4OA5D 25113170 IC50 = 100 nM T00663 CF7C5B 25129829 IC50 > 10000 nM T00663 CXNM84 25129830 IC50 > 10000 nM T00663 CY2S1P 25129831 IC50 > 10000 nM T00663 CCK8D2 25154767 IC50 > 20000 nM T00663 C9ZKH4 25174103 IC50 = 9 nM T00663 CPY2C9 25203945 IC50 = 398.11 nM T00663 CEFT59 25210489 IC50 = 330 nM T00663 CXE16F 25218564 IC50 = 5011 nM T00663 C3RH2Q 25218565 IC50 = 6310 nM T00663 CMF51N 25222038 IC50 = 148 nM T00663 C15DIA 25222587 IC50 = 79 nM T00663 C7BAN0 25262260 IC50 > 20000 nM T00663 CV7AG6 25660569 IC50 = 1500 nM T00663 C5GZ8L 26704995 IC50 = 3900 nM T00663 CRY5L4 42537838 IC50 = 1200 nM T00663 CWS37O 42618140 IC50 > 25118.86 nM T00663 C2JV3O 42618143 IC50 > 25118.86 nM T00663 CG01BO 42618144 IC50 > 25118.86 nM T00663 CI5AE0 43623574 IC50 = 17200 nM T00663 C0HB4C 44129168 IC50 = 16800 nM T00663 CX16AN 44138038 Ki = 16 nM T00663 CO42DC 44138048 IC50 = 316.23 nM T00663 CL65QV 44138049 IC50 = 125.89 nM T00663 CR7TY6 44197572 IC50 > 20000 nM T00663 C1G2ZQ 44198874 IC50 > 20000 nM T00663 C75TAQ 44200209 IC50 = 83 nM T00663 C7W4AX 44200211 IC50 = 320 nM T00663 C16HSY 44200344 IC50 = 68 nM T00663 CBY7T8 44200468 IC50 = 510 nM T00663 C8KNA3 44219632 Ki > 4000 nM T00663 C0VIX4 44219633 Ki > 4000 nM T00663 CPT6F0 44224261 IC50 = 160 nM T00663 CMRG01 44236943 IC50 = 9900 nM T00663 C0HM6Z 44236944 IC50 = 900 nM T00663 CRT04D 44236945 IC50 = 2200 nM T00663 C46EDI 44236946 IC50 = 540 nM T00663 C37IRD 44236947 IC50 = 960 nM T00663 CGSA21 44236948 IC50 = 250 nM T00663 CGO6L3 44236949 IC50 = 1100 nM T00663 CYV31G 44236950 IC50 = 1400 nM T00663 C2D4LE 44236951 IC50 = 1000 nM T00663 C6IGK2 44236952 IC50 > 20000 nM T00663 CFU45N 44236953 IC50 > 20000 nM T00663 C07YUQ 44236954 IC50 = 200 nM T00663 C8HPQ7 44236955 IC50 = 290 nM T00663 CG8KU3 44236956 IC50 > 20000 nM T00663 CLK0U1 44236957 IC50 > 20000 nM T00663 C9L3XK 44236958 IC50 > 20000 nM T00663 CRJ9F0 44236959 IC50 > 20000 nM T00663 CBXL42 44236960 IC50 = 310 nM T00663 C9HR2S 44236961 IC50 = 1800 nM T00663 C1CD6L 44236962 IC50 = 2300 nM T00663 C34TLE 44236963 IC50 = 5000 nM T00663 CW3PO4 44236964 IC50 = 8900 nM T00663 CC93MW 44236965 IC50 = 5800 nM T00663 C1XQG3 44236966 IC50 = 2000 nM T00663 C82AFZ 44236967 IC50 = 2000 nM T00663 CTH0D7 44236968 IC50 = 6400 nM T00663 COF30J 44236969 IC50 > 20000 nM T00663 C6J0UF 44236970 IC50 > 20000 nM T00663 CP81MF 44236971 IC50 = 60 nM T00663 CTHS64 44236972 IC50 = 80 nM T00663 CNL6H4 44236973 IC50 = 410 nM T00663 C87WNK 44236974 IC50 = 210 nM T00663 CJ9VI7 44236975 IC50 = 530 nM T00663 C0FT5H 44236976 IC50 = 350 nM T00663 C1HX8I 44236977 IC50 = 1000 nM T00663 CET82Q 44236978 IC50 = 110 nM T00663 C59YJV 44236979 IC50 = 4800 nM T00663 CSI8C1 44236980 IC50 = 620 nM T00663 CF2YU6 44236981 IC50 = 11000 nM T00663 C19NBZ 44236982 IC50 > 20000 nM T00663 CH56RI 44404432 IC50 = 270 nM T00663 CUW89Z 44404434 IC50 = 10.9 nM T00663 CW8F3T 44404438 IC50 = 233 nM T00663 C9AJ1Y 44404441 IC50 = 3 nM T00663 C2RXS6 44404444 IC50 = 130 nM T00663 C2MT9X 44404797 IC50 = 3.3 nM T00663 CAC7Q5 44404813 IC50 = 1.259 nM T00663 C7F6KQ 44408641 IC50 = 8 nM T00663 C27KEP 44408669 IC50 = 44 nM T00663 CFY5E9 44408670 IC50 = 6 nM T00663 CI76KB 44408825 IC50 = 9 nM T00663 C3I1VN 44408826 IC50 = 207 nM T00663 CBC3X6 44408908 IC50 = 5 nM T00663 CY8LJ5 44408909 IC50 = 10 nM T00663 C3O7GC 44408936 IC50 = 15 nM T00663 CCW09A 44408944 IC50 = 3 nM T00663 C5YUK6 44431823 IC50 = 630.96 nM T00663 CO91FC 44431824 IC50 = 1000 nM T00663 CI95TS 44431825 IC50 > 15848.93 nM T00663 CJN16A 44431826 IC50 > 15848.93 nM T00663 CU75OI 44431827 IC50 > 15848.93 nM T00663 C2P8TK 44431828 IC50 > 15848.93 nM T00663 C2C4SX 44431829 IC50 = 2511.89 nM T00663 C9Y1ID 44431830 IC50 = 3162.28 nM T00663 CU20ER 44431831 IC50 = 251.19 nM T00663 CL87AX 44431832 IC50 = 1000 nM T00663 CA61VJ 44431833 IC50 = 501.19 nM T00663 C1KW0V 44431834 IC50 = 1584.89 nM T00663 CAX8F5 44440161 IC50 = 412 nM T00663 CM2E3N 44440217 IC50 = 708 nM T00663 C6RD3G 44440219 IC50 = 582 nM T00663 CIAJ70 44440220 IC50 = 5000 nM T00663 C52CDB 44440221 IC50 = 32 nM T00663 CFZS24 44440223 IC50 = 107 nM T00663 CSA87R 44440224 IC50 = 31 nM T00663 CH76CV 44440225 IC50 = 14 nM T00663 CKSO82 44440228 IC50 = 179 nM T00663 C8HWI1 44440229 IC50 = 120 nM T00663 CVD97U 44440230 IC50 = 48 nM T00663 C9AV4C 44440236 IC50 = 5 nM T00663 C60YEU 44444010 IC50 = 1000 nM T00663 C1HEB4 44444011 IC50 > 20000 nM T00663 CKB97N 44444012 IC50 = 3600 nM T00663 CE02WM 44444013 IC50 = 1300 nM T00663 C7GFW0 44444014 IC50 = 510 nM T00663 CZ73CR 44444016 IC50 = 1600 nM T00663 C7FTV8 44444018 IC50 = 530 nM T00663 C52NJF 44444019 IC50 = 930 nM T00663 CY0G7R 44444021 IC50 = 210 nM T00663 C5I8ND 44444024 IC50 = 440 nM T00663 CA7N3G 44444025 IC50 = 480 nM T00663 C0JGC3 44444026 IC50 = 3600 nM T00663 CER95H 44444027 IC50 = 760 nM T00663 C16XZW 44444028 IC50 = 15000 nM T00663 CA8Q2M 44444029 IC50 = 6500 nM T00663 CL4B1D 44444030 IC50 = 140 nM T00663 CAX59T 44444031 IC50 = 490 nM T00663 C0CIN7 44444033 IC50 > 20000 nM T00663 CY20IT 44444034 IC50 = 5200 nM T00663 CKD8E0 44444036 IC50 = 5000 nM T00663 CD8BK3 44444037 IC50 = 250 nM T00663 CDZO02 44444038 IC50 = 200 nM T00663 C7H3AL 44444039 IC50 = 240 nM T00663 CXK91I 44444991 IC50 = 7 nM T00663 CCP02M 44444992 IC50 = 3 nM T00663 CU80BP 44517743 IC50 > 10000 nM T00663 CKV96M 44571730 IC50 > 20000 nM T00663 C7Q1VU 44580077 IC50 > 16000 nM T00663 CL90SE 44580358 IC50 > 16000 nM T00663 CK1VE7 44580420 IC50 > 16000 nM T00663 CH2R7X 44580449 IC50 > 16000 nM T00663 C1VH0C 44580532 IC50 > 16000 nM T00663 CXC52J 44580649 IC50 > 16000 nM T00663 CE32BQ 44580689 IC50 > 16000 nM T00663 C8Z5AX 44580778 IC50 > 16000 nM T00663 C5Z3LI 44591740 IC50 = 16 nM T00663 CZ8XI5 44627578 Ki = 130 nM T00663 CKM3N2 44627579 IC50 = 297 nM T00663 CN30CM 44627580 IC50 = 365 nM T00663 C7NU3G 44627581 IC50 = 7 nM T00663 CDF41Q 44627582 IC50 = 4 nM T00663 CKI17J 44627583 IC50 = 390 nM T00663 C7EK0M 44627681 IC50 = 79 nM T00663 C8RVP9 44627682 IC50 = 140 nM T00663 C6E2LI 44627683 IC50 = 85 nM T00663 C21IGV 44627684 IC50 = 133 nM T00663 CG6UW5 44634494 IC50 = 13760 nM T00663 CJ0LU4 45104966 IC50 = 263 nM T00663 CJ32SA 45203151 IC50 = 1100 nM T00663 C2JVA4 45270368 IC50 = 250 nM T00663 CA4XQ3 45375859 IC50 = 5456 nM T00663 C46MWH 45488127 IC50 = 3950 nM T00663 C3P8YT 45488146 IC50 = 31800 nM T00663 CW2G7D 46868853 IC50 = 7 nM T00663 CR57OZ 46868855 IC50 = 324 nM T00663 CI8YE5 46868856 IC50 = 12 nM T00663 C94EPL 46868925 IC50 = 5 nM T00663 C0GU4D 46868930 IC50 = 160 nM T00663 C9ULP0 46869071 IC50 = 5300 nM T00663 CU52JS 46869075 IC50 = 3600 nM T00663 CFQT10 46869147 IC50 = 42500 nM T00663 CEK2I5 46869149 IC50 = 820 nM T00663 C2XQ4K 46869223 IC50 = 9400 nM T00663 C8U1AH 46869285 IC50 = 6 nM T00663 CKTD23 46869290 IC50 = 183 nM T00663 CV57OI 46869490 IC50 = 9 nM T00663 C9XHK0 46869491 IC50 = 14 nM T00663 C47JSD 46869493 IC50 = 14 nM T00663 C65NDB 46869609 IC50 = 31500 nM T00663 CP2A4Y 46869611 IC50 = 550 nM T00663 CQ0AU8 46869671 IC50 = 45600 nM T00663 C4RS7M 46869672 IC50 = 465 nM T00663 C1VZM6 46869673 IC50 = 5 nM T00663 CYI69K 46869674 IC50 = 25 nM T00663 C2PC6T 46869677 IC50 = 1500 nM T00663 CSL2N6 46869740 IC50 = 5900 nM T00663 C6V9CD 46869741 IC50 = 25 nM T00663 CZCQ05 46869742 IC50 = 1600 nM T00663 C09GAW 46869745 IC50 = 143 nM T00663 CVBG98 46869815 IC50 = 594 nM T00663 CU2D5N 46869816 IC50 = 18 nM T00663 C8WH7Q 46869817 IC50 = 80 nM T00663 CFOX43 46869876 IC50 = 197 nM T00663 CE0CY1 46869877 IC50 = 560 nM T00663 C2DW6T 46869878 IC50 = 33 nM T00663 C19DQG 46869879 IC50 = 34 nM T00663 CR1OH0 46869880 IC50 = 6 nM T00663 C8SFI1 46869881 IC50 = 9 nM T00663 CD1YH9 46869882 IC50 = 28 nM T00663 CQIC19 46879806 IC50 > 20000 nM T00663 C6WD4Q 46881329 IC50 = 6309.57 nM T00663 C6GQH3 46881341 IC50 = 12589.25 nM T00663 CEK6A9 46881342 IC50 = 3981.07 nM T00663 C84TWY 46881343 IC50 > 15848.93 nM T00663 C1DFI0 46881344 IC50 = 5011.87 nM T00663 CW32UX 46881345 IC50 > 15848.93 nM T00663 C8CE7P 46881351 IC50 = 10000 nM T00663 C7AE4V 46881352 IC50 = 1000 nM T00663 CP7UE5 46881353 IC50 > 15848.93 nM T00663 C32XZI 46881354 IC50 = 15848.93 nM T00663 CSQ8O9 46881355 IC50 = 6309.57 nM T00663 CO0SC4 46881358 IC50 = 1995.26 nM T00663 C4DXW0 46881359 IC50 = 630.96 nM T00663 CK67BQ 46881360 IC50 > 15848.93 nM T00663 CV4O5T 46881361 IC50 > 15848.93 nM T00663 CRD8S3 46884198 IC50 = 10.9 nM T00663 CRKV43 46884199 Ki = 5 nM T00663 CA2Y8J 46901260 IC50 > 20000 nM T00663 CQR9K1 46933384 IC50 > 100000 nM T00663 CHSF07 49806372 IC50 > 1000 nM T00663 CS18HZ 49839481 IC50 = 77 nM T00663 C83VHI 49864785 IC50 = 90000 nM T00663 C2UTK6 49864850 IC50 > 100000 nM T00663 CAE53W 49865153 IC50 = 78000 nM T00663 CDR47S 49867175 IC50 = 25 nM T00663 CH4FY5 50941455 IC50 = 24 nM T00663 CBR71Y 50941538 IC50 = 16 nM T00663 C4BN7W 50941539 IC50 = 29 nM T00663 C1HI2W 51346940 IC50 = 40 nM T00663 C5GPU9 51346941 IC50 = 90 nM T00663 CM24LF 52938983 IC50 > 20000 nM T00663 CA7HQ9 52941011 IC50 = 700 nM T00663 CA6BH5 52941226 IC50 = 5400 nM T00663 CMXC68 52941286 IC50 = 1500 nM T00663 C0DSA8 52941649 IC50 = 17000 nM T00663 C4O3RZ 52942227 IC50 > 50000 nM T00663 C3BKR7 52942436 IC50 = 6500 nM T00663 C8R9SA 52942482 IC50 = 37000 nM T00663 CAC3J5 52942507 IC50 = 1600 nM T00663 CTPH98 52942532 IC50 > 50000 nM T00663 CHP7M6 52943427 IC50 > 50000 nM T00663 CS8VA0 52943431 IC50 = 4400 nM T00663 CJU79I 52943626 IC50 = 900 nM T00663 C07JYV 52944873 IC50 = 2100 nM T00663 CB1UJ7 52944909 IC50 = 1600 nM T00663 CD2WZ5 52944914 IC50 = 1600 nM T00663 CY9B7D 52944962 IC50 > 50000 nM T00663 C1Z7KR 52946059 IC50 = 9000 nM T00663 CCMX82 52946092 IC50 = 27000 nM T00663 CPIK13 52946145 IC50 = 12600 nM T00663 C67TBV 52946152 IC50 = 1400 nM T00663 C6OH8X 52946172 IC50 > 50000 nM T00663 CC6Z1J 52947386 IC50 = 3800 nM T00663 CC5P4R 52947399 IC50 > 50000 nM T00663 C9O7FN 52947421 IC50 > 50000 nM T00663 C72TPI 52947422 IC50 > 50000 nM T00663 C3R4FI 52948519 IC50 = 920 nM T00663 CLU92X 52948565 IC50 = 31000 nM T00663 CDXL70 52948593 IC50 = 470 nM T00663 CO3EL9 52948602 IC50 > 50000 nM T00663 C3WHA1 52949737 IC50 > 50000 nM T00663 CMT75N 52949817 IC50 = 610 nM T00663 CBAD62 52949818 IC50 = 610 nM T00663 CSOB70 52950113 IC50 = 690 nM T00663 CW2KE5 53317337 IC50 = 38800 nM T00663 CJQN83 53317338 IC50 = 3020 nM T00663 CJ2P3V 53317339 IC50 = 504 nM T00663 C9E3FV 53317340 IC50 = 226 nM T00663 CBTX53 53317412 IC50 = 16000 nM T00663 COCN94 53317413 IC50 = 40 nM T00663 CHC29T 53317414 IC50 = 210 nM T00663 C82LCE 53317415 IC50 = 590 nM T00663 CR0DJ1 53317416 IC50 = 92 nM T00663 C28JAP 53317417 IC50 = 36 nM T00663 C8Q0OR 53318506 IC50 = 62 nM T00663 CP7T3N 53318709 IC50 = 54 nM T00663 CKD47I 53319944 IC50 = 99 nM T00663 CP7BR1 53319945 IC50 = 1020 nM T00663 C3TAC2 53320021 IC50 = 3900 nM T00663 COPI53 53321333 IC50 = 410 nM T00663 C0GLS5 53321334 IC50 = 120 nM T00663 C2V0QU 53321577 IC50 = 250 nM T00663 CG8KC9 53322569 IC50 = 9110 nM T00663 C3SA1K 53322570 IC50 = 310 nM T00663 COG9J2 53322644 IC50 = 130 nM T00663 CUR1A6 53322645 IC50 = 70 nM T00663 C25OEY 53322984 IC50 = 125 nM T00663 CK8Y5F 53323911 IC50 = 162 nM T00663 C9SHJ0 53323985 IC50 = 85 nM T00663 C49MDG 53323986 IC50 = 70 nM T00663 C3AVG0 53323987 IC50 = 430 nM T00663 C18SCR 53323988 IC50 = 14 nM T00663 C38RXW 53323989 IC50 = 22 nM T00663 CXWB94 53325188 IC50 = 110 nM T00663 C8VPW5 53325283 IC50 = 54 nM T00663 CA3X2Q 53325284 IC50 = 130 nM T00663 CIG7X9 53325285 IC50 = 94 nM T00663 C4A8JK 53325286 IC50 = 100 nM T00663 CI1RT4 53325287 IC50 = 280 nM T00663 CNT50E 53325288 IC50 = 24 nM T00663 CR91NJ 53325555 IC50 = 700 nM T00663 CBW0G7 53326484 IC50 = 9620 nM T00663 CV7I4O 53326555 IC50 = 32 nM T00663 C27IBZ 53326556 IC50 = 61 nM T00663 C5UK3J 53326557 IC50 = 950 nM T00663 CVJ6K9 53326558 IC50 = 160 nM T00663 C8NA4L 53384644 IC50 > 30000 nM T00663 CD0ZI6 53469858 IC50 = 245 nM T00663 CCG3H2 54580285 IC50 = 10 nM T00663 CJDM48 54580615 IC50 = 600 nM T00663 CPRC42 54580619 IC50 = 160 nM T00663 C56ARZ 54580647 IC50 = 7 nM T00663 CB4TJ8 54581287 IC50 = 50 nM T00663 C5U6YP 54581288 IC50 = 700 nM T00663 CNU9G4 54581289 IC50 = 4400 nM T00663 C39VAB 54581290 IC50 = 210 nM T00663 CT3JS6 54581291 IC50 = 7 nM T00663 CM7H3P 54581292 IC50 = 9 nM T00663 CEP18Y 54581359 IC50 > 50000 nM T00663 C6JPE1 54581360 IC50 = 52.2 nM T00663 CD2YU5 54581361 IC50 = 4480 nM T00663 C49RNQ 54581362 IC50 = 1230 nM T00663 CA8U3P 54581363 IC50 > 50000 nM T00663 C2ZN7A 54581623 IC50 = 1450 nM T00663 CH6VE9 54581624 IC50 = 160 nM T00663 CD4Z6Y 54581656 IC50 = 1330 nM T00663 C5V6OY 54582175 IC50 > 30000 nM T00663 C6B2UL 54582304 IC50 = 63 nM T00663 C1FR4Q 54582305 IC50 = 20 nM T00663 CP4HV1 54582306 IC50 = 10 nM T00663 CFG68S 54582307 IC50 = 4 nM T00663 C52OMN 54582618 IC50 = 340 nM T00663 C26UOY 54582645 IC50 = 240 nM T00663 C1OM6E 54583278 IC50 = 20 nM T00663 CNE41S 54583279 IC50 = 90 nM T00663 C6XC0E 54583280 IC50 = 30 nM T00663 CMCL04 54583281 IC50 = 60 nM T00663 CTQ70F 54583282 IC50 = 50 nM T00663 CCO5I2 54583368 IC50 = 12600 nM T00663 CECO89 54583369 IC50 = 1910 nM T00663 CFV81A 54583573 IC50 = 70 nM T00663 C0K8HF 54583574 IC50 = 200 nM T00663 CS83TL 54583576 IC50 = 320 nM T00663 CF72GE 54583602 IC50 = 390 nM T00663 C68FYO 54583603 IC50 = 1400 nM T00663 CM1TU0 54584242 IC50 = 70 nM T00663 CP6K3I 54584243 IC50 = 60 nM T00663 CR4E7O 54584244 IC50 = 80 nM T00663 CRKI30 54584315 IC50 = 945 nM T00663 C3P2HM 54584316 IC50 = 30400 nM T00663 CL69AG 54584317 IC50 = 364 nM T00663 CBA65Z 54584562 IC50 = 730 nM T00663 C2DRY7 54584563 IC50 = 130 nM T00663 C7GR5M 54584564 IC50 = 160 nM T00663 CC3BE2 54584594 IC50 = 650 nM T00663 CEJ0M6 54584595 IC50 = 340 nM T00663 C3EP6K 54584596 IC50 = 110 nM T00663 CD4WJ7 54584597 IC50 = 400 nM T00663 CT16HO 54585212 IC50 = 30 nM T00663 CNB2M9 54585213 IC50 = 90 nM T00663 CC8YN2 54585285 IC50 = 14800 nM T00663 CGA8X9 54585286 IC50 > 50000 nM T00663 CV69FU 54585287 IC50 > 50000 nM T00663 CR1X8Y 54585288 IC50 = 1030 nM T00663 CTY84H 54585289 IC50 > 50000 nM T00663 CWE79L 54585290 IC50 = 4810 nM T00663 C0FAG2 54585291 IC50 = 2460 nM T00663 CNLU49 54585292 IC50 = 4130 nM T00663 CPZ20X 54585507 IC50 = 100 nM T00663 CNUP53 54586040 IC50 = 880 nM T00663 C30VTY 54586163 IC50 = 170 nM T00663 CQNZ54 54586164 IC50 = 190 nM T00663 CUD8J0 54586233 IC50 = 49100 nM T00663 CT78AW 54586474 IC50 = 860 nM T00663 CGW36K 54586475 IC50 = 160 nM T00663 CE0C3W 54586476 IC50 = 200 nM T00663 C8IO1D 54586477 IC50 = 480 nM T00663 CWX92H 54586479 IC50 = 170 nM T00663 C40EQC 54586508 IC50 = 390 nM T00663 C6BX0V 54587174 IC50 = 730 nM T00663 CI49LN 54587175 IC50 > 20000 nM T00663 CI8ZH6 54587176 IC50 = 50 nM T00663 C1V8HM 54587177 IC50 = 60 nM T00663 CO1JB2 54587178 IC50 = 20 nM T00663 C3JAW8 54587179 IC50 = 30 nM T00663 CA5N6I 54587258 IC50 = 27400 nM T00663 CKX15Q 54587259 IC50 = 18300 nM T00663 CKQS27 54587260 IC50 = 14900 nM T00663 C57LBW 54587261 IC50 = 2670 nM T00663 CMH8N5 54587504 IC50 = 630 nM T00663 C8UC1Z 54587510 IC50 = 750 nM T00663 CL75DP 54587542 IC50 = 150 nM T00663 C0I4FV 54764508 IC50 = 37 nM T00663 C18TKF 54764593 IC50 = 7 nM T00663 CG78UW 56658171 IC50 = 11 nM T00663 C7LDZ3 56658303 IC50 = 280 nM T00663 C0MW6D 56658304 IC50 = 8 nM T00663 CK18JP 56661802 IC50 = 41 nM T00663 CE1O3B 56661803 IC50 = 14 nM T00663 CSJ6A9 56665092 IC50 = 3 nM T00663 C7HA6J 56665093 IC50 = 8 nM T00663 CS5HP6 56665245 IC50 = 30 nM T00663 C4SO3M 56665246 IC50 = 6 nM T00663 CE2PY0 56665247 IC50 = 6 nM T00663 C9AW1E 56668539 IC50 = 15 nM T00663 C0MR6D 56668696 IC50 = 7 nM T00663 CXF3R9 56668697 IC50 = 19 nM T00663 CU3I2J 56672173 IC50 = 71 nM T00663 CJ9I6K 56672174 IC50 = 2 nM T00663 CD5NZ4 56672175 IC50 = 6 nM T00663 CRAK61 56675421 IC50 = 8 nM T00663 CG3ZU0 56678888 IC50 = 52 nM T00663 CAP1M2 56682209 IC50 = 24 nM T00663 C9DO8G 56682210 IC50 = 2 nM T00663 CTO6N5 56834943 IC50 = 24 nM T00663 C97SLT 57340680 IC50 = 704 nM T00663 C0UDN5 57340685 IC50 = 130 nM T00663 CDP45J 57390517 IC50 = 140 nM T00663 C28LIB 57390518 IC50 = 130 nM T00663 C8DZ1N 57390519 IC50 = 12 nM T00663 C7K4LJ 57390520 IC50 = 240 nM T00663 C32DFY 57390767 IC50 = 140 nM T00663 CKUX48 57390768 IC50 = 200 nM T00663 C32FUN 57390769 IC50 = 72 nM T00663 C6P0YR 57390770 IC50 = 17 nM T00663 CH4X7D 57390771 IC50 = 160 nM T00663 CG51FX 57392289 IC50 = 31 nM T00663 C9EJN6 57392581 IC50 = 380 nM T00663 CP1D7N 57392582 IC50 = 320 nM T00663 CX0F1Z 57392583 IC50 = 78 nM T00663 C2IZ3W 57392739 IC50 = 7 nM T00663 C9P1SC 57393560 IC50 = 16 nM T00663 CVH4X0 57394043 IC50 = 17 nM T00663 CN3MB5 57394305 IC50 = 100 nM T00663 CLOD68 57394306 IC50 = 34 nM T00663 C1EYU6 57394468 IC50 = 32 nM T00663 CV9W8C 57395293 IC50 = 24 nM T00663 CQ2A1B 57395802 IC50 = 63 nM T00663 C15YOZ 57396060 IC50 = 48 nM T00663 CL4BN7 57396061 IC50 = 110 nM T00663 CW7XA9 57397040 IC50 = 13 nM T00663 C18MFO 57397857 IC50 = 35 nM T00663 C7KJ2W 57397858 IC50 = 2200 nM T00663 CB7DO2 57397859 IC50 = 49 nM T00663 CDI28Y 57397860 IC50 = 60 nM T00663 CKG0P1 57397861 IC50 = 170 nM T00663 C9A7RL 57397862 IC50 = 140 nM T00663 CH1QI7 57399519 IC50 = 27 nM T00663 CA0SR3 57399520 IC50 = 200 nM T00663 C8IFD4 57399521 IC50 = 48 nM T00663 CT5S8H 57400156 IC50 = 100 nM T00663 C2DG7X 57401275 IC50 = 45 nM T00663 C8FQH3 57402785 IC50 > 1000 nM T00663 C1HD8L 57402972 IC50 = 520 nM T00663 C8ZQ3A 57403022 IC50 = 70 nM T00663 CKIX12 57403023 IC50 = 15 nM T00663 C4VKU7 57403024 IC50 = 70 nM T00663 CZ5L4E 57403025 IC50 = 3500 nM T00663 CNP8C3 57403026 IC50 = 990 nM T00663 CDXK85 57403027 IC50 = 80 nM T00663 CH0NB1 57403028 IC50 = 2200 nM T00663 CJY46H 57403029 IC50 = 30 nM T00663 CI1A8M 57404048 IC50 = 7738 nM T00663 C6UAN1 57467725 IC50 = 2199 nM T00663 C7I4QD 57519510 IC50 = 159 nM T00663 CO57NK 58155042 IC50 = 680 nM T00663 CT3EW2 59292007 IC50 = 560 nM T00663 COH62U 60097413 IC50 > 3300 nM T00663 C06UMH 66958119 IC50 = 326 nM T00663 CV63UL 67240318 IC50 > 10000 nM T00663 C69OHY 68560854 IC50 > 20000 nM T00663 C25MEI 68561431 IC50 > 20000 nM T00663 CCD89X 68563058 IC50 > 20000 nM T00663 C0XCY9 68565200 IC50 > 20000 nM T00663 CW6BH7 68566254 IC50 > 20000 nM T00663 CQRP72 68567556 IC50 > 20000 nM T00663 C48EIQ 68568011 IC50 > 20000 nM T00663 CAWC35 68621678 IC50 > 1000 nM T00663 C3GTU1 69762142 IC50 > 10000 nM T00663 CQ8HE2 70690944 IC50 > 30000 nM T00663 C13FWG 70695135 IC50 > 30000 nM T00663 C0VZB2 70697173 IC50 > 30000 nM T00663 C2LU7I 70702008 IC50 = 7 nM T00663 CMPK41 70702010 IC50 = 117 nM T00663 CKT98U 71584212 IC50 = 1090 nM T00663 CI3MH6 71602620 IC50 > 20000 nM T00663 CCD0W3 71602669 IC50 = 24 nM T00663 C3D1CA 71602671 IC50 = 33 nM T00663 CG1DR3 71602672 IC50 = 12 nM T00663 CQ9A6D 71602719 IC50 = 46 nM T00663 CDU4I0 71602720 IC50 = 59 nM T00663 CP01YB 71602721 IC50 = 32 nM T00663 CX60NJ 71602722 IC50 = 38 nM T00663 CHU36E 71602723 IC50 = 54 nM T00663 C7MGB8 71602768 IC50 = 77 nM T00663 CZ8US1 71602769 IC50 = 43 nM T00663 C2GM5W 71602770 IC50 = 22 nM T00663 C9UY4L 71602771 IC50 = 15 nM T00663 C6O2KE 71602772 IC50 = 120 nM T00663 CA2J9W 71602817 IC50 = 250 nM T00663 CS4K2F 71602818 IC50 = 35 nM T00663 CY8H5Z 71602819 IC50 = 1400 nM T00663 C60VBS 71602820 IC50 = 63 nM T00663 CI09ER 71602821 IC50 = 50 nM T00663 C2KW8Y 71602864 IC50 = 640 nM T00663 CEX14A 71602865 IC50 = 640 nM T00663 CEF41S 71602866 IC50 = 110 nM T00663 CAM32B 71602867 IC50 = 120 nM T00663 CDH23B 71602868 IC50 = 80 nM T00663 CVUG79 71602911 IC50 = 170 nM T00663 C8AM1K 71655603 IC50 > 20000 nM T00663 C7OQC1 71720177 IC50 = 1860 nM T00663 CD3JF9 71745086 IC50 = 40 nM T00663 CZ4BX1 72547959 IC50 = 364 nM T00663 C8THP4 72946274 IC50 = 26 nM T00663 CYZP14 72946275 IC50 > 20000 nM T00663 C8T2WZ 72946276 IC50 = 70 nM T00663 C5N9JK 72946277 IC50 = 32 nM T00663 C3TM0X 72946450 IC50 = 126 nM T00663 CP8ZR3 72946451 IC50 = 523 nM T00663 C1IKA3 72946452 IC50 = 366 nM T00663 CWG15I 72946453 IC50 = 27 nM T00663 C2I8CL 72946454 IC50 = 134 nM T00663 CV5P7N 72946655 IC50 = 216 nM T00663 C98FIU 72946656 IC50 = 1 nM T00663 CJA75F 72946661 IC50 = 435 nM T00663 C0QL7V 72946851 IC50 = 19 nM T00663 C8GI2A 72946852 IC50 = 74 nM T00663 C1NKW5 72946853 IC50 = 52 nM T00663 C78GOJ 72946854 IC50 = 16 nM T00663 CO61VP 72946855 IC50 = 187 nM T00663 CG4YH2 72946856 IC50 = 24 nM T00663 C0HQ6V 72947058 IC50 = 587 nM T00663 C8J3WG 76328237 IC50 = 7 nM T00663 CJ2T9E 76332983 IC50 > 10000 nM T00663 CLTG58 78350466 IC50 = 1600 nM T00663 C54KDR 86763302 IC50 = 1895 nM T00663 C4HKT5 87057579 IC50 = 98 nM T00663 CQ2OB9 90292687 IC50 > 10000 nM T00663 CHI39S 90292823 IC50 > 10000 nM T00663 C5C9PB 90667115 IC50 = 218 nM T00663 CI4RH8 90667116 IC50 = 371 nM T00663 C4H0ZN 90667117 IC50 = 414 nM T00663 CTB63D 90667118 IC50 = 727 nM T00663 C5TPF3 90667119 IC50 = 173 nM T00663 C0INK4 90667120 IC50 = 3100 nM T00663 C80FXC 90667121 IC50 = 160 nM T00663 C98QUS 90667122 IC50 > 20000 nM T00663 C4YS9Z 90667123 IC50 = 12000 nM T00663 C4A3FO 90667124 IC50 > 20000 nM T00663 CG6C4H 90667125 IC50 = 132 nM T00663 CQIP37 90667126 IC50 = 374 nM T00663 C0HL7F 90667127 IC50 = 325 nM T00663 C6FRO8 90667128 IC50 = 218 nM T00663 CE0ID8 90667129 IC50 = 371 nM T00663 CZ45HF 90667130 IC50 = 680 nM T00663 CSJ4C2 90667131 IC50 = 326 nM T00663 CJU4V7 90667132 IC50 = 414 nM T00663 CBZ73T 90667133 IC50 = 727 nM T00663 CW3UI2 90667134 IC50 = 173 nM T00663 C0M3VU 90667135 IC50 = 0.28 nM T00663 CH7G1F 90667136 IC50 = 0.42 nM T00663 C7P8TV 90667137 IC50 = 0.78 nM T00663 CE05TI 90667138 IC50 = 0.3 nM T00663 CH4DI3 90667139 IC50 = 0.28 nM T00663 C1U9DY 90667140 IC50 = 0.31 nM T00663 C9JQE0 90667141 IC50 = 0.25 nM T00663 CIV0J1 90667142 IC50 = 1.2 nM T00663 C1C7PW 90667143 IC50 = 0.77 nM T00663 CLF96U 90667144 IC50 = 2.5 nM T00663 C49JZU 90667145 IC50 = 0.16 nM T00663 CE5M7Q 90667146 IC50 = 1800 nM T00663 C7V8BN 91754589 IC50 = 11 nM T00663 CQ2G3S 91754590 IC50 = 15 nM T00663 CJQ5N6 91936970 IC50 = 2100 nM T00663 C2GNI5 101891709 IC50 < 1 nM T00663 C6ZFW9 101913690 IC50 = 18 nM T00663 C9VSP7 101913691 IC50 = 26 nM T00663 C5DLO7 118143962 IC50 = 38 nM T00663 CK7O6G 118144051 IC50 = 230 nM T00663 CQ29IK 118144281 IC50 = 133 nM T00663 CZG4U9 118144359 IC50 = 62 nM T00663 C61FOL 118144367 IC50 = 114 nM T00663 CE7QM9 118144380 IC50 = 169 nM T00663 C8GU6M 118146727 IC50 = 141 nM T00663 CY82JT 118146747 IC50 = 37 nM T00663 CIDU81 118146748 IC50 = 130 nM T00663 C1OIF0 118146749 IC50 > 10000 nM T00663 C8TLS2 118146764 IC50 = 238 nM T00663 C32HVY 118146772 IC50 = 860 nM T00663 CULV52 118146793 IC50 = 71 nM T00663 CB2WI6 118146794 IC50 = 5184 nM T00663 CQFE90 118146797 IC50 = 3063 nM T00663 CA7H9O 118146798 IC50 = 4588 nM T00663 C1MI6J 118146804 IC50 = 23 nM T00663 CERD34 118146805 IC50 = 34 nM T00663 C48AZY 118146813 IC50 = 100 nM T00663 CKT2Q3 118146814 IC50 = 162 nM T00663 CJ4Z3K 118146817 IC50 = 2166 nM T00663 C7Q6RW 118146819 IC50 = 162 nM T00663 CH0I3M 118146826 IC50 = 162 nM T00663 CT29IZ 118146828 IC50 = 203 nM T00663 CHWP46 118146849 IC50 = 313 nM T00663 C4P9AK 118146855 IC50 = 80 nM T00663 CT8K0N 118146868 IC50 = 3300 nM T00663 CET9N4 118146870 IC50 = 31 nM T00663 C4PBE7 118146871 IC50 = 54 nM T00663 C6LEU5 118146872 IC50 = 28 nM T00663 CX08HF 118146873 IC50 = 594 nM T00663 CD8L5Y 118146874 IC50 = 116 nM T00663 CNI34V 118146882 IC50 = 23 nM T00663 C8K0GC 118146884 IC50 = 311 nM T00663 CQW3L7 118146891 IC50 = 201 nM T00663 C4O6MA 118146892 IC50 = 58 nM T00663 CZ35XB 118146932 IC50 = 141 nM T00663 C7NDK6 118146979 IC50 = 21 nM T00663 C56EHT 118146984 IC50 = 139 nM T00663 C3R5DA 118720654 IC50 = 115 nM T00663 C0KM6L 118720655 IC50 = 596 nM T00663 C3FY2J 118720656 IC50 = 1829 nM T00663 CGFD93 118720657 IC50 = 137 nM T00663 C8L9SK 118720658 IC50 = 34 nM T00663 C81HTM 118720659 IC50 = 29 nM T00663 CJ2NI1 118721229 IC50 = 350 nM T00663 CC05EY 118721230 IC50 = 710 nM T00663 C7HJ8Y 118721231 IC50 = 32 nM T00663 C5XMF8 118721232 IC50 = 12 nM T00663 CZY01I 118721233 IC50 = 5.5 nM T00663 C2USQ7 118721234 IC50 = 14 nM T00663 CDS2U3 118721235 IC50 = 31 nM T00663 C0H9OV 118721236 IC50 = 1.9 nM T00663 C83KJY 118721237 IC50 = 1.9 nM T00663 C13QEP 118721238 IC50 = 20 nM T00663 CVC3B0 118721239 IC50 = 7 nM T00663 C2F6MN 118721240 IC50 = 2200 nM T00663 C36PRN 118721241 IC50 = 1200 nM T00663 CY0J8A 118721242 IC50 = 400 nM T00663 CJLX62 118721243 IC50 = 540 nM T00663 C14BFC 118721244 IC50 = 2500 nM T00663 C6ETU2 118721245 IC50 = 400 nM T00663 CC4OF9 118725553 IC50 = 40 nM T00663 CR9ML7 118725554 IC50 = 12 nM T00663 CZ82KA 118725885 IC50 = 4220 nM T00663 CSV5K7 118725886 IC50 = 199 nM T00663 C9XV2B 118725887 IC50 = 1186 nM T00663 C6KCQ9 118725888 IC50 = 266 nM T00663 C6LCD8 118725889 IC50 = 255 nM T00663 CI96GZ 118725890 IC50 = 91 nM T00663 CL3KT6 118725891 IC50 = 269 nM T00663 C2JNF8 118725892 IC50 = 55 nM T00663 CU9KV7 118725893 IC50 = 33 nM T00663 C51HGX 118725894 IC50 = 82 nM T00663 C3HP6G 118725895 IC50 = 47 nM T00663 CR4K1M 118725896 IC50 = 45 nM T00663 C95CUL 118725897 IC50 = 133 nM T00663 CN27BI 118725898 IC50 = 25 nM T00663 CH1VK2 118725899 IC50 = 35 nM T00663 C5IM2Q 118725900 IC50 = 226 nM T00663 CP7DK8 118725901 IC50 = 79 nM T00663 CL8W3Q 118725902 IC50 = 180 nM T00663 CNL1Z4 118725903 IC50 = 2010 nM T00663 C5S2OE 118725904 IC50 = 2633 nM T00663 CL0CJ2 118725905 IC50 = 678 nM T00663 C4UTF5 118725906 IC50 = 2167 nM T00663 C4PQ8K 118725907 IC50 = 1216 nM T00663 CE7ZH9 118725908 IC50 = 170 nM T00663 CM7IQ3 118725909 IC50 = 1528 nM T00663 C3WF5U 118725910 IC50 = 79 nM T00663 CGR19E 118725911 IC50 = 12 nM T00663 CZ8RX6 118725912 IC50 = 61 nM T00663 CU9RB6 118725913 IC50 = 54 nM T00663 CBO8S2 118725914 IC50 = 213 nM T00663 C5CMS9 118725915 IC50 = 17 nM T00663 CEJ7T0 118725916 IC50 = 80 nM T00663 CHT6K9 118728811 Ki > 4000 nM T00663 CUA3Y2 118728812 Ki > 4000 nM T00663 CDQ78G 118728813 Ki > 4000 nM T00663 CZ6XL7 118728814 Ki > 4000 nM T00663 CMO67K 118728815 Ki > 4000 nM T00663 CR2M0Q 118728816 Ki > 4000 nM T00663 C62SCL 118728817 Ki > 4000 nM T00663 CSB30C 118728819 Ki > 4000 nM T00663 CV7XU8 118728820 Ki > 4000 nM T00663 C3J1EX 118728821 Ki > 4000 nM T00663 CIWB78 118728822 Ki > 4000 nM T00663 CP18SE 118728823 Ki > 4000 nM T00663 CM42CA 118728824 Ki > 4000 nM T00663 C9Q7CL 118728825 Ki > 4000 nM T00663 CCR3S0 118728826 Ki > 4000 nM T00663 CH3ZB0 118732094 IC50 > 10000 nM T00663 C0K5LC 118732096 IC50 > 10000 nM T00663 C4HM7F 118732099 IC50 > 10000 nM T00663 C2R9JZ 118732102 IC50 > 10000 nM T00663 C4IQ7C 118732107 IC50 > 10000 nM T00663 CSLU37 118732108 IC50 > 10000 nM T00663 CYRJ23 118732109 IC50 > 10000 nM T00663 CQCX41 118737057 IC50 > 10000 nM T00663 CI6R3E 122178086 IC50 > 10000 nM T00663 CFD0W1 122178087 IC50 > 10000 nM T00663 CRUE70 122178088 IC50 = 532 nM T00663 CMG2E7 122178091 IC50 = 81 nM T00663 CQ0F5Z 122178092 IC50 = 204 nM T00663 C4X7SD 122192466 IC50 > 10000 nM T00663 C0FM1R 130196825 IC50 = 416 nM T00663 C6OXE3 132134663 IC50 >= 1000 nM T00663 CEX92Y 135417092 IC50 = 9760 nM T00663 CRPC85 135432695 IC50 = 8890 nM T00663 CMXR51 135446691 IC50 = 4240 nM T00663 CI1JQ3 135449325 Ki = 550 nM T00663 C8GZ2B 135449326 Ki > 4000 nM T00663 C1JGA6 135454192 IC50 = 2370 nM T00663 CO6I2L 135523935 Ki > 4000 nM T00663 C1Q2AL 135523936 Ki > 4000 nM T00663 C2PQT5 135523937 Ki > 4000 nM T00663 CP2B4U 135523938 Ki > 4000 nM T00663 C0GMF7 135523939 Ki = 840 nM T00663 CSI4D2 135523940 Ki > 4000 nM T00663 COM67B 135523941 Ki = 3100 nM T00663 CX56SF 135523946 Ki = 2800 nM T00663 CWU14F 135523947 Ki = 3300 nM T00663 CX5LG4 135523948 Ki = 3900 nM T00663 CNY53K 135523949 Ki > 4000 nM T00663 C1HUP6 135523950 Ki = 2700 nM T00663 CA7HF8 135523951 Ki = 3000 nM T00663 CT08OB 135523952 Ki = 3400 nM T00663 C28SDI 135523953 Ki > 4000 nM T00663 CJ08EW 135523954 Ki = 1800 nM T00663 CZ87OT 135523955 Ki = 2700 nM T00663 C5Q0GA 135523957 Ki = 790 nM T00663 CF2G9Y 135523958 Ki > 4000 nM T00663 CGHE70 135523959 Ki = 2900 nM T00663 CWZ6R0 135523960 Ki > 4000 nM T00663 CIHM29 135523961 Ki > 4000 nM T00663 CHW83U 135523962 Ki = 3200 nM T00663 CD1G6A 135523963 Ki = 2500 nM T00663 CA41BZ 135523964 Ki = 3100 nM T00663 C4JCM5 135523965 Ki = 2800 nM T00663 C5EYW9 135533810 IC50 = 7650 nM T00663 CPV59N 135685787 Ki > 4000 nM T00663 CM3UC9 135883136 IC50 = 250 nM T00663 CM2UH4 135894362 IC50 > 1000 nM T00663 CY19DW 135894364 IC50 > 1000 nM T00663 CF1PS8 135934877 Ki > 4000 nM T00663 CTRL59 135976660 Ki = 2500 nM T00663 CQ84IZ 136180335 Ki > 4000 nM T00663 CM17FU 136198654 IC50 > 10000 nM T00663 C15HQK 136218656 IC50 > 1000 nM T00663 CZ06UK 136218660 IC50 > 1000 nM T00663 CML48X 136218661 IC50 > 1000 nM T00663 COB69I 136218662 IC50 > 1000 nM T00663 CSL6Q8 136218663 IC50 > 1000 nM T00663 CTFJ83 136226213 IC50 > 1000 nM T00663 C5EV8A 136240902 IC50 > 1000 nM T00663 CX9LB5 136240903 IC50 > 1000 nM T00663 CMC58H 136240944 IC50 > 1000 nM T00663 C60PRZ 136241012 IC50 > 1000 nM T00663 C1Q9YN 136252259 IC50 > 1000 nM T00663 CH9O7Z 137631713 IC50 = 17 nM T00663 C4V1EU 137636264 IC50 = 8 nM T00663 C1G6KJ 137637551 IC50 = 0.6 nM T00663 CLGH04 137638967 IC50 = 3 nM T00663 CNE0Z1 137639840 IC50 = 2 nM T00663 CS3RQ4 137639936 IC50 = 4 nM T00663 CT38UG 137641182 IC50 = 24 nM T00663 CYL1R5 137643579 IC50 = 2 nM T00663 CW3IE6 137645681 IC50 = 27 nM T00663 CAY2W4 137646016 IC50 = 2 nM T00663 CGNM85 137646697 IC50 = 3 nM T00663 C5UE8A 137649558 IC50 = 175 nM T00663 CN13EH 137650943 IC50 = 0.3 nM T00663 CLN2M3 137652755 IC50 = 23 nM T00663 C8MH2Z 137654276 IC50 = 3 nM T00663 CMJF60 137655822 IC50 = 2 nM T00663 CPY1U3 137656311 IC50 = 25 nM T00663 CBI64H 137657498 IC50 = 30 nM T00663 CZFJ89 137660093 IC50 = 253 nM T00663 CA3XC2 137660956 IC50 = 200 nM T00663 CS32IR 137661932 IC50 = 10 nM T00663 CZ9BN4 138320062 IC50 = 0.107 nM T00663 C6VB3O 145925651 IC50 >= 5000 nM T00663 C2MD1Q 155513187 IC50 > 10000 nM T00663 CFV10S 155529132 IC50 = 90 nM T00663 C2CG1A 155537016 IC50 > 10000 nM T00663 D00HVA 11624601 Ki = 52 nM T00663 D02PVB 8515 IC50 = 90 nM T00663 D06PJW 25182616 IC50 = 2000 nM T00663 D0D6MH 11617559 IC50 > 16000 nM T00663 D0E3KD 447874 IC50 = 590 nM T00663 D0H2PE 10236389 IC50 = 48 nM T00663 D0J3LR 11634725 Ki = 1400 nM T00663 D0L0HG 766949 IC50 = 199.53 nM T00663 D0OZ2S 11785878 IC50 = 7300 nM T00663 D0Q3NG 11715520 Ki = 520 nM T00663 D0R3MO 46864283 IC50 > 20000 nM T00663 D0S7IE 11658882 Ki = 3300 nM T00663 D0VJ2S 57340686 IC50 = 338 nM T31186 CBHX59 5494430 IC50 > 400000 nM T31186 CGZJ49 6911989 IC50 = 43500 nM T31186 CF2Z8H 73345264 IC50 = 85000 nM T31186 C6PHF8 73345266 IC50 = 4000 nM T31186 CY07SN 73348296 IC50 = 70000 nM T31186 COC3D9 87278522 IC50 = 27000 nM T31186 CBF2I4 87278547 IC50 = 15500 nM T31186 CPHV38 87278548 IC50 = 34000 nM T31186 CK10ZE 87278578 IC50 = 45000 nM T31186 CD9M2Z 87278583 IC50 = 43500 nM T31186 CP02TE 88568566 IC50 = 25000 nM T31186 C40SKD 88568567 IC50 = 32000 nM T31186 C2SPB4 88568595 IC50 = 21500 nM T31186 C4PFH0 88568626 IC50 = 18500 nM T31186 CWUR45 88568650 IC50 = 14000 nM T31186 CVP2B8 88568651 IC50 = 28000 nM T31186 CMI83B 88568652 IC50 = 11500 nM T31186 C51NPU 90644210 IC50 = 10500 nM T31186 C8WJT2 90644211 IC50 = 10500 nM T31186 C6D0LB 90644212 IC50 = 15500 nM T31186 C76GAJ 90644213 IC50 = 30000 nM T31186 CPZ41A 90644214 IC50 = 30500 nM T31186 C9QD4R 90644215 IC50 = 32500 nM T31186 CTXP81 90644216 IC50 = 49000 nM T31186 CP3FR5 90644217 IC50 = 49000 nM T31186 CXE82I 90644218 IC50 = 16500 nM T31186 CJXI38 90644219 IC50 = 51500 nM T31186 C2VZ6T 90644220 IC50 = 55500 nM T31186 C68DLC 90644221 IC50 = 39000 nM T31186 C90QLM 90644222 IC50 = 40500 nM T31186 CMG67U 90644223 IC50 = 48500 nM T31186 C9NB5J 118719257 IC50 > 400000 nM T31186 CTZ6U9 135450598 Ki = 28 nM T31186 C9Y0KB 135501934 IC50 > 400000 nM T31186 C8DGU1 135566702 IC50 = 95 nM T31186 C48ETA 135874011 IC50 = 41 nM T31186 COAK56 135924252 IC50 = 59 nM T31186 CAN6D4 135924253 IC50 = 6580 nM T31186 CFO84Y 136086421 IC50 > 400000 nM T31186 CM8GR9 136138688 IC50 = 15500 nM T31186 CUM1R3 136138689 IC50 = 56800 nM T31186 CG4L1M 136138690 IC50 = 54500 nM T31186 CCOP90 136138691 IC50 = 10000 nM T31186 C4XN9U 136138692 IC50 = 49300 nM T31186 C5YLP4 136138694 IC50 = 5350 nM T31186 CJ73VB 136138696 IC50 = 43000 nM T31186 CGPX35 136138698 IC50 = 1590 nM T31186 CWB34M 136138700 IC50 = 125 nM T31186 CV0EY9 136138703 IC50 = 2570 nM T31186 CG3WL4 136138705 IC50 = 56 nM T31186 C9Z2WY 136138707 IC50 = 85400 nM T31186 CNL69S 136138709 IC50 = 117 nM T31186 CF5B3P 136138716 IC50 = 3600 nM T31186 CBP2Y7 136138717 IC50 = 51 nM T31186 CMN04A 136138724 IC50 = 300000 nM T31186 C2VM5F 136138725 IC50 = 1350 nM T31186 CJ9M4A 136138730 IC50 = 160 nM T31186 C7X9VW 136138737 IC50 = 16 nM T31186 CEOA02 136138748 IC50 = 3140 nM T31186 CG17QK 136168052 IC50 = 14000 nM T31186 C0G8TQ 136219232 IC50 > 400000 nM T31186 CL36PF 136239280 IC50 > 400000 nM T31186 CRD1X8 136239419 IC50 > 400000 nM T31186 CEQ20H 136244199 IC50 > 400000 nM T31186 CJQ7O0 136244535 IC50 = 400000 nM T31186 C6W2FB 136244622 IC50 = 400000 nM T31186 CI5P4A 137007090 IC50 = 200000 nM T31186 CUY95S 137007091 IC50 = 130000 nM T31186 CRBD48 137169130 IC50 = 45000 nM T31186 CP5Z9C 137169131 IC50 = 55000 nM T31186 CK7R3T 137169132 IC50 > 400000 nM T31186 C19BNM 137169134 IC50 > 400000 nM T31186 CQ67ME 137169136 IC50 > 400000 nM T31186 CIK56Z 137169159 IC50 = 5000 nM T31186 C5NAP7 137169160 IC50 = 220000 nM T31186 CLT5O9 137169161 IC50 > 400000 nM T31186 C7DQC8 137169162 IC50 > 400000 nM T31186 COB83M 137169163 IC50 = 50000 nM T31186 C9HFC1 137169164 IC50 = 100000 nM T31186 C7S6FE 137169165 IC50 = 220000 nM T31186 C7D5EQ 137169166 IC50 > 400000 nM T31186 CMAZ31 137169167 IC50 = 180000 nM T31186 C8ID1Y 145975543 Ki = 382000 nM T38996 D01XBA 5035 IC50 = 4300 nM T38996 D03JRG 46937439 IC50 = 1500 nM T38996 D0CI4A 25105704 IC50 = 21 nM T38996 D0OX9E 50902705 IC50 = 200 nM T38996 CQ0IC4 63062 IC50 = 4800 nM T38996 CW21VY 16739265 IC50 = 1 nM T38996 C17GSK 21428808 IC50 = 14000 nM T38996 C3IHB0 21428850 IC50 = 6.3 nM T38996 C9QY5H 21428857 IC50 = 22 nM T38996 CVC98H 21428895 IC50 = 4 nM T38996 C23HQA 21428932 IC50 = 5590 nM T38996 C40CFO 21428968 IC50 = 10000 nM T38996 CK90LC 21428971 IC50 = 1000 nM T38996 C8IXU1 21429000 IC50 = 10 nM T38996 CT0C3Z 25105692 IC50 = 14 nM T38996 CA7XR1 25105696 IC50 = 6000 nM T38996 C0MHU9 25105697 IC50 = 3200 nM T38996 CRG7X8 25105698 IC50 = 17 nM T38996 C54TAV 25105699 IC50 = 19 nM T38996 CIPH75 25105700 IC50 = 85 nM T38996 C9H5WS 25105701 IC50 = 32 nM T38996 CMJ14L 25105702 IC50 = 79 nM T38996 C7EW5O 25105703 IC50 = 51 nM T38996 C9J7ZI 25105705 IC50 = 20 nM T38996 CMW3Y1 25105706 IC50 = 35 nM T38996 C5MZX7 25105707 IC50 = 300 nM T38996 C2ZF1U 25105708 IC50 = 380 nM T38996 C68JBL 25105709 IC50 = 37 nM T38996 CF6P7E 25105710 IC50 = 8.9 nM T38996 C30IGQ 25105711 IC50 = 48 nM T38996 C19VQY 25105712 IC50 = 870 nM T38996 C9TX2Y 25105713 IC50 = 11 nM T38996 C48BVE 25105714 IC50 > 20000 nM T38996 C3WPU2 25105715 IC50 = 1000 nM T38996 C8XHA1 25105716 IC50 = 3400 nM T38996 CH2A5B 44138051 IC50 = 25 nM T38996 CO0V5A 44438309 IC50 = 8 nM T38996 CXB2R1 44573118 IC50 = 6.4 nM T38996 CT6FP3 44573119 IC50 = 8 nM T38996 COD46G 44573120 IC50 = 3 nM T38996 C65LXN 44573121 IC50 = 3.5 nM T38996 CD6G3I 44573130 IC50 = 4 nM T38996 C40TOA 44573131 IC50 = 3.7 nM T38996 CRC8G1 44573132 IC50 = 2 nM T38996 C8N3CM 44573176 IC50 = 5.5 nM T38996 C0D4GS 44573191 IC50 = 12 nM T38996 CSZ0W7 44573597 IC50 = 40 nM T38996 CFQA45 44573598 IC50 = 70 nM T38996 C8Q5RD 44573599 IC50 = 110 nM T38996 CC09AZ 44573641 IC50 = 120 nM T38996 C39HWT 44573687 IC50 = 4 nM T38996 CT18AS 44573688 IC50 = 18 nM T38996 CWI75L 44573689 IC50 = 12 nM T38996 C14ZEX 44573690 IC50 = 3 nM T38996 C8A4LR 44573727 IC50 = 7 nM T38996 CBM42C 44573728 IC50 = 4 nM T38996 CBCX36 44573767 IC50 = 43 nM T38996 C5BDG2 44573768 IC50 = 130 nM T38996 CQ9X2N 44573769 IC50 = 38 nM T38996 CQ62KR 44573770 IC50 = 66 nM T38996 CB2G5X 44573806 IC50 = 100 nM T38996 C1GM3U 44573807 IC50 = 11 nM T38996 CZO1C6 44573808 IC50 = 7.4 nM T38996 CEX9F5 44573809 IC50 = 10 nM T38996 CP63HT 44591888 IC50 > 20000 nM T38996 CK8GV2 44591889 IC50 = 1900 nM T38996 CHVO21 44591890 IC50 = 2100 nM T38996 CP5VO4 44591891 IC50 = 2600 nM T38996 C09BTI 44591892 IC50 = 150 nM T38996 C9E5ZV 44591930 IC50 = 150 nM T38996 CCX35M 44591931 IC50 = 4250 nM T38996 CDY58B 44591932 IC50 = 5900 nM T38996 CBHW79 44591933 IC50 > 20000 nM T38996 CFOX18 44591934 IC50 = 3400 nM T38996 C0J3UF 46938432 IC50 = 210 nM T38996 C8LAD0 46938434 IC50 = 250 nM T38996 CMB63C 46938535 IC50 = 390 nM T38996 C3GPY4 46938537 IC50 = 290 nM T38996 CNSZ76 46938539 IC50 = 335 nM T38996 CRN3Z8 46938541 IC50 = 2660 nM T38996 CYO78K 46938928 IC50 = 10 nM T38996 CB06NU 46939226 IC50 = 2500 nM T38996 CP04XW 46939227 IC50 = 11800 nM T38996 C4B2SF 46939228 IC50 = 1200 nM T38996 CV8DS2 46939229 IC50 = 870 nM T38996 CX3QE6 46939321 IC50 = 3470 nM T38996 C2K4TB 46939322 IC50 = 2800 nM T38996 CR7L9X 46939323 IC50 = 2060 nM T38996 CQI17K 46939324 IC50 = 5780 nM T38996 CJ7VN8 46939407 IC50 = 1700 nM T38996 C2ZW8V 46939408 IC50 = 2000 nM T38996 CO5X0P 46939409 IC50 = 2270 nM T38996 CY05QU 46939410 IC50 = 3500 nM T38996 C1PZM4 46939489 IC50 = 5900 nM T38996 CX49SE 46939490 IC50 = 2700 nM T38996 C14XNH 49850293 IC50 = 16 nM T38996 CF31UA 50902617 IC50 = 1700 nM T38996 C58APV 50902621 IC50 = 320 nM T38996 CPUG80 50902623 IC50 = 5500 nM T38996 C3RNG4 50902707 IC50 = 6400 nM T38996 CH38VC 50902709 IC50 > 20000 nM T38996 CRC6V8 50902786 IC50 = 12000 nM T38996 C16FQK 50902788 IC50 = 320 nM T38996 CKE14R 50902876 IC50 = 1350 nM T38996 CAJ3L1 50902978 IC50 = 1 nM T38996 C47VGW 53393916 IC50 = 20000 nM T38996 C26TVP 56593045 IC50 = 86 nM T38996 CB27OD 56593054 IC50 = 6 nM T38996 C2XP8D 56593056 IC50 = 1540 nM T38996 C3ZYA2 56593082 IC50 = 20 nM T38996 C7ENU3 56846622 IC50 = 1400 nM T38996 C1CBU4 56846623 IC50 = 760 nM T38996 CEZA46 56846640 IC50 = 75 nM T38996 C47LNP 68182778 IC50 = 250 nM T38996 CBME89 68182839 IC50 = 820 nM T38996 C6AHP7 68183060 IC50 = 16 nM T38996 COXN56 68188986 IC50 = 25 nM T38996 CUBM27 71716675 IC50 = 2 nM T38996 CWB3V1 71718136 IC50 = 6 nM T38996 CRG3Z8 73099418 IC50 > 30000 nM T38996 CV9UO7 118722101 IC50 = 315 nM T38996 C1ZJ5C 118722102 IC50 = 290 nM T38996 C9OSG5 118722103 IC50 = 120 nM T38996 CUSE27 118722104 IC50 = 18 nM T38996 C84TOB 118722105 IC50 = 6 nM T38996 CYM54A 118722106 IC50 = 17 nM T38996 C8CDM2 118722107 IC50 = 636 nM T38996 CCEL04 118722108 IC50 = 115 nM T38996 CI5MY4 118722109 IC50 = 21 nM T38996 CPF97C 118722110 IC50 = 244 nM T38996 C09UXY 118722111 IC50 = 870 nM T38996 CD73JQ 118722112 IC50 = 468 nM T38996 COU89E 118722113 IC50 = 230 nM T38996 CRB6F1 118722114 IC50 = 72 nM T38996 CMRF75 118722115 IC50 = 820 nM T38996 CBF47Z 118722116 IC50 = 115 nM T38996 C92QNG 155537801 IC50 = 21 nM T38996 CVU9P7 155540036 IC50 = 1200 nM T38996 D07JMN 94459 IC50 = 3600 nM T38996 D07RPV 65490 IC50 = 21 nM T38996 D0IV2E 5280592 IC50 > 1000 nM T38996 D0T3HK 70517 IC50 = 3600 nM T43920 D0C2II 4100 IC50 = 20 nM T43920 D0E1SW 1986 Ki = 0.8 nM T43920 CG2Q9U 66824 Ki = 0.3 nM T43920 CJR96B 72879 IC50 = 1000000 nM T43920 C04JEX 73702 IC50 = 1000000 nM T43920 CCK5Y6 133125 IC50 = 550 nM T43920 C8KN4F 133683 IC50 = 20 nM T43920 C2GA7W 195627 IC50 = 730 nM T43920 CZL4G0 232992 Ki = 584 nM T43920 CPA95I 232993 Ki = 146 nM T43920 CD23RS 641380 IC50 = 550 nM T43920 CM5FP2 3769607 IC50 = 20 nM T43920 C83URK 4343109 IC50 = 20 nM T43920 CH62SB 5325614 IC50 = 480 nM T43920 C18GCW 13754314 Ki = 258 nM T43920 C4JD1S 13755238 Ki = 44 nM T43920 CA8D6Y 13755239 Ki = 107 nM T43920 CX4V9O 13904667 IC50 = 20 nM T43920 C28TEH 13904668 IC50 = 18 nM T43920 C7Q1BO 13904669 IC50 = 14 nM T43920 CE51MD 13904671 IC50 = 50 nM T43920 CXK68I 13904672 IC50 = 50 nM T43920 C7YX0N 15665951 IC50 = 370 nM T43920 C6DU3A 15665952 IC50 = 390 nM T43920 CK8BI3 15665953 IC50 = 520 nM T43920 C0ASB7 15665954 IC50 = 910 nM T43920 CL35KY 15665955 IC50 = 440 nM T43920 CW6LI5 15665958 IC50 = 450 nM T43920 CK72NU 15665961 IC50 = 310 nM T43920 CVSL38 15665962 IC50 = 940 nM T43920 CRXL21 15665963 IC50 = 230 nM T43920 C89TJU 15665964 IC50 = 910 nM T43920 C3NZO2 15665965 IC50 = 520 nM T43920 C2QL3W 15665966 IC50 = 520 nM T43920 CN7J6P 44343745 IC50 = 84 nM T43920 C6KUJ0 44343753 IC50 = 770 nM T43920 C5EIQ0 59552403 Ki = 0.2 nM T43920 CQN51D 118724498 IC50 = 441720 nM T43920 C8F9DB 135898802 IC50 = 37 nM T43920 CR17HF 155510806 Ki = 0.2 nM T43920 C2H9WX 155554455 Ki = 0.2 nM T43920 D06LVE 22784 Ki = 0.2 nM T43920 D09QHC 7370 IC50 = 2000 nM T97587 CTA32V 9831270 IC50 = 49 nM T97587 C7J3ZW 9847562 IC50 = 1.4 nM T97587 CV9X1Q 9871831 IC50 = 3.7 nM T97587 CSY94G 9893920 IC50 = 0.87 nM T97587 C5BXR9 9960341 IC50 = 1.6 nM T97587 C8J2IQ 9961835 IC50 = 0.2 nM T97587 C8AJ2G 9985610 IC50 = 0.64 nM T97587 C3VX4B 10175373 IC50 = 99 nM T97587 C1BK6W 10348108 IC50 = 20 nM T97587 CS12LU 10369544 IC50 = 0.5 nM T97587 C4D8CL 10415520 IC50 = 0.7 nM T97587 C4TGS8 15984101 IC50 = 0.51 nM T97587 CNG3Y6 20828691 IC50 = 0.07 nM T97587 C5XI2B 23647822 IC50 = 9.2 nM T97587 CV87US 23647823 IC50 = 106 nM T97587 C4NZC8 23647824 IC50 = 769 nM T97587 C7K6VJ 23647825 IC50 = 49 nM T97587 CTV02H 23647826 IC50 = 282 nM T97587 CD36OZ 23647827 IC50 = 216 nM T97587 CB54AV 23647828 IC50 = 15 nM T97587 CIN2D4 23647829 IC50 = 8.4 nM T97587 CDC59X 23647830 IC50 = 13 nM T97587 C23IKQ 23647831 IC50 = 1.3 nM T97587 CT19JC 23647832 IC50 = 1.3 nM T97587 C7RB6T 23647833 IC50 = 9.8 nM T97587 CUYM23 23647834 IC50 = 1.7 nM T97587 C0HD6M 23647835 IC50 = 95 nM T97587 CUP79Y 24875357 IC50 = 237 nM T97587 CG17MD 25147778 IC50 = 1.6 nM T97587 CS98GW 25242385 IC50 = 2.8 nM T97587 C78USC 44157321 IC50 = 0.09 nM T97587 C86VTZ 44157395 IC50 = 0.1 nM T97587 CF01CW 44157473 IC50 = 0.1 nM T97587 C5QDR9 44157717 IC50 = 0.2 nM T97587 CJ1GX4 44157718 IC50 = 0.3 nM T97587 CPI0L1 44270826 IC50 = 550 nM T97587 C2ITA9 44270830 IC50 = 330 nM T97587 CAYN82 44270836 IC50 = 160 nM T97587 CTU6S9 44270842 IC50 = 44 nM T97587 C9ONK1 44271028 IC50 = 35 nM T97587 CXM20K 44271069 IC50 = 0.1 nM T97587 CMX53A 44271083 IC50 = 2.7 nM T97587 CAU67L 44271148 IC50 = 3.9 nM T97587 CU2DL4 44271164 IC50 = 1.8 nM T97587 CR94DM 44271244 IC50 = 19 nM T97587 CR06WP 44271256 IC50 = 112 nM T97587 CKP31U 44271273 IC50 = 5 nM T97587 C0W9BH 44446215 IC50 = 123 nM T97587 CE29ZY 44446216 IC50 = 135 nM T97587 CT9G8Q 44446217 IC50 = 170 nM T97587 CS36EO 44446218 IC50 = 152 nM T97587 C02NZQ 44446219 IC50 = 353 nM T97587 C2S7QF 44446220 IC50 = 327 nM T97587 CV4L9G 44446221 IC50 = 450 nM T97587 CQXG81 44446222 IC50 = 143 nM T97587 CC8HU7 44446223 IC50 = 239 nM T97587 CV49GF 44446224 IC50 = 75 nM T97587 CP0TH8 44446225 IC50 = 179 nM T97587 CDM45Z 44446226 IC50 = 235 nM T97587 C1WRY6 44446227 IC50 = 222 nM T97587 CX6T3Z 44446228 IC50 = 130 nM T97587 CL9DG6 44446229 IC50 = 76 nM T97587 CWTX92 44446230 IC50 = 69 nM T97587 CD0QV3 44446231 IC50 = 67 nM T97587 COXP59 44446232 IC50 = 101 nM T97587 C8T6CM 44446233 IC50 = 19 nM T97587 C08SHV 44446234 IC50 = 67 nM T97587 C56TUJ 44446236 IC50 = 124 nM T97587 C1G6AZ 44446238 IC50 = 80 nM T97587 C7USF6 44446240 IC50 = 200 nM T97587 C7IU9H 44446241 IC50 = 196 nM T97587 C7R4QZ 44446243 IC50 = 28 nM T97587 C79HBR 44446248 IC50 = 1122 nM T97587 CG83CS 44446251 IC50 = 6807 nM T97587 C9UZ0X 44446256 IC50 = 4318 nM T97587 CF5DT9 44446259 IC50 = 510 nM T97587 C5ZQ3C 44446261 IC50 = 42 nM T97587 C9IS1C 44455093 IC50 = 285 nM T97587 CB51GK 44455095 IC50 = 2535 nM T97587 CX23CH 44455169 IC50 = 2100 nM T97587 CB9T2Z 44571247 IC50 = 831 nM T97587 C1R5VH 44571248 IC50 = 198 nM T97587 CBK28E 44571249 IC50 = 164 nM T97587 COG41E 44571293 IC50 = 50 nM T97587 CS80NQ 44571294 IC50 = 19 nM T97587 CP6M5Y 44571295 IC50 = 19 nM T97587 CB26YW 44587963 IC50 = 7.5 nM T97587 CVTM09 44587964 IC50 = 4.8 nM T97587 CG2RX4 44587965 IC50 = 12 nM T97587 C52MPU 44588004 IC50 = 2.8 nM T97587 C05GKL 44588445 IC50 = 2.9 nM T97587 CT81MC 44588480 IC50 = 2.2 nM T97587 C3KSC4 44588481 IC50 = 44 nM T97587 C0JS4X 44588482 IC50 = 1.9 nM T97587 CDPT75 44588524 IC50 = 630 nM T97587 CUCZ38 44588525 IC50 = 3.5 nM T97587 C05LYK 44588526 IC50 = 688 nM T97587 CT8PH7 45485800 IC50 = 0.34 nM T97587 CHP37W 45485803 IC50 = 0.16 nM T97587 CLFJ36 45485807 IC50 = 0.11 nM T97587 CTR5Z7 46229904 IC50 = 0.22 nM T97587 C3XAQ6 46229905 IC50 = 0.81 nM T97587 CSP19C 46229906 IC50 = 0.55 nM T97587 C40XVP 46229907 IC50 = 0.08 nM T97587 CI2O9L 46229908 IC50 = 0.25 nM T97587 C7F0MK 46229909 IC50 = 0.35 nM T97587 CO4D9I 46229910 IC50 = 0.08 nM T97587 CVL02P 46229911 IC50 = 0.42 nM T97587 CG7V9S 46229912 IC50 = 0.25 nM T97587 C0ML2V 46229913 IC50 = 0.13 nM T97587 C42KWF 46229914 IC50 = 0.13 nM T97587 CTK82C 46229915 IC50 = 0.11 nM T97587 CM43CI 46229916 IC50 = 0.13 nM T97587 CE4Q9R 46229917 IC50 = 0.16 nM T97587 C93TOU 46229918 IC50 = 0.14 nM T97587 CJX9A5 46229919 IC50 = 0.16 nM T97587 C93JUZ 49865755 IC50 = 2700 nM T97587 CQEB67 49865756 IC50 = 8300 nM T97587 CAO82G 49865757 IC50 = 9500 nM T97587 C5CPE8 49865758 IC50 = 6300 nM T97587 CZ4SH8 49865759 IC50 = 100 nM T97587 CYG30P 49865760 IC50 = 9000 nM T97587 CT5DJ6 49865761 IC50 = 6300 nM T97587 CX8C0E 49865762 IC50 = 7900 nM T97587 CI4Q6S 49865763 IC50 = 8700 nM T97587 CVP7M6 49865764 IC50 = 500 nM T97587 COSD80 49865765 IC50 = 1400 nM T97587 CB2RH6 49865766 IC50 = 1200 nM T97587 C7QNM0 49865842 IC50 = 2100 nM T97587 CT8H9I 49865843 IC50 = 1500 nM T97587 CL0O3V 49865844 IC50 = 1100 nM T97587 CMVB16 49865845 IC50 = 4400 nM T97587 CV3XC8 49865895 IC50 = 1500 nM T97587 CHI31D 49865896 IC50 = 6600 nM T97587 C5MK9C 49865897 IC50 = 1200 nM T97587 C4CR0M 49865898 IC50 = 300 nM T97587 CE2H9O 49865899 IC50 = 600 nM T97587 C1MJI2 49865946 IC50 = 700 nM T97587 C7QIX2 49865947 IC50 = 600 nM T97587 CZE86G 49865948 IC50 = 3000 nM T97587 C7TUL0 49865949 IC50 = 600 nM T97587 CP74MO 49865950 IC50 = 700 nM T97587 C8D7SR 49865996 IC50 = 2800 nM T97587 C6ZFN2 49865997 IC50 = 600 nM T97587 C3HNC7 49865998 IC50 = 1500 nM T97587 CPO1L3 49865999 IC50 = 900 nM T97587 CEK6Z9 49866051 IC50 = 200 nM T97587 C0G5SY 49866052 IC50 = 1500 nM T97587 CUW64X 49866053 IC50 = 500 nM T97587 C41GCZ 49866107 IC50 = 700 nM T97587 C4C7EB 49866108 IC50 = 400 nM T97587 C1NB5E 49866109 IC50 = 1000 nM T97587 C87SXF 49866110 IC50 = 2600 nM T97587 CK5ZC9 49866111 IC50 = 3400 nM T26463 D02ILH 341 Ki = 830 nM T26463 D05RQB 457964 EC50 = 2000 nM T26463 CZP5J2 3415 IC50 > 20000 nM T26463 C4DTF0 6665 IC50 > 500000 nM T26463 CLO15X 67277 IC50 = 32000 nM T26463 CQ87XE 72187 IC50 = 13400 nM T26463 CMR72P 127307 Ki = 14400 nM T26463 CQ1XM2 149664 Ki = 1400 nM T26463 C7Y0CH 238747 IC50 = 28000 nM T26463 C6NE8Z 389513 Ki = 1000 nM T26463 CO6A2E 451388 IC50 = 1000 nM T26463 C9L0ZN 481497 IC50 > 100000 nM T26463 CF2YG0 481498 IC50 = 63000 nM T26463 C9I6LT 481500 IC50 = 18000 nM T26463 CY24WL 481501 IC50 > 100000 nM T26463 C9U7BA 481504 IC50 = 93000 nM T26463 CU3P0Y 484047 IC50 > 40000 nM T26463 CL4X0H 491953 IC50 > 50000 nM T26463 CP8ZJ7 491954 IC50 = 26000 nM T26463 C61SXL 492406 IC50 > 40000 nM T26463 CXD5F2 496192 IC50 = 85000 nM T26463 CM6J2G 496196 Ki = 5000 nM T26463 CDW6L4 497307 IC50 = 480 nM T26463 CZJP19 497308 IC50 > 100000 nM T26463 CX9ZP0 497310 IC50 = 800 nM T26463 C74SZP 497311 IC50 = 15 nM T26463 CZ1A8T 503580 IC50 > 40000 nM T26463 C8UMS5 3005246 Ki = 36000 nM T26463 C3E1ZI 3012981 IC50 > 100000 nM T26463 C1FXQ4 5466207 Ki = 2600 nM T26463 C8F1DN 6482394 IC50 > 40000 nM T26463 C6OF2J 6914644 IC50 > 100000 nM T26463 CQP57I 9802791 IC50 > 500000 nM T26463 CF5TC2 9805202 IC50 = 5000 nM T26463 CHT36N 9828287 IC50 = 3000 nM T26463 C47XQV 9938296 IC50 = 5000 nM T26463 CA9Q4Z 10078740 IC50 = 1900 nM T26463 C1JN2O 10120254 IC50 > 10000 nM T26463 C7SO4T 10144617 IC50 > 10000 nM T26463 C3B2KX 10185481 IC50 > 10000 nM T26463 CB5O0Q 10185854 IC50 > 50000 nM T26463 CDQ6H2 10209030 IC50 > 10000 nM T26463 C58FZS 10230222 IC50 > 10000 nM T26463 C5AXK6 10230544 IC50 > 10000 nM T26463 CZ48MN 10385259 IC50 = 66000 nM T26463 C5O4HY 10647065 Ki = 7840 nM T26463 CNKU56 10893485 IC50 > 50000 nM T26463 CG2KN4 10918740 Ki = 156000 nM T26463 CB98DN 11014401 IC50 = 4300 nM T26463 CIYW64 11686018 IC50 > 10000 nM T26463 C7Z5LI 11764703 Ki = 548000 nM T26463 CUB20Q 15949381 IC50 > 10000 nM T26463 CEL84W 15956783 IC50 > 10000 nM T26463 COP0D7 15956784 IC50 > 10000 nM T26463 C51OVS 15956785 IC50 > 10000 nM T26463 CIU52S 21589997 IC50 > 12500 nM T26463 C0L2TF 23725128 IC50 > 100000 nM T26463 C1P2KY 24771829 EC50 = 350000 nM T26463 CO25RL 25000921 IC50 > 100000 nM T26463 CG9S8U 44396484 IC50 = 8000 nM T26463 CSQ5K2 44396511 Ki = 3750 nM T26463 CC2AE1 44396529 IC50 > 500000 nM T26463 C0GDR1 44396563 IC50 > 500000 nM T26463 CK8ZW1 44396581 IC50 > 500000 nM T26463 CE04QD 44396595 IC50 > 500000 nM T26463 CZ6DX1 44412144 IC50 = 1900 nM T26463 CGM62X 44412145 IC50 = 3300 nM T26463 CZ18LU 44412189 IC50 = 8900 nM T26463 C3MSG6 44412212 IC50 = 7900 nM T26463 C3JG6P 44412241 IC50 = 2300 nM T26463 C2U6NS 44412250 IC50 = 3500 nM T26463 C1WGS5 44412370 IC50 = 25000 nM T26463 CX1GZ9 44412378 IC50 = 19900 nM T26463 C1XN2M 44412379 IC50 = 19700 nM T26463 C7ZKR6 44412431 IC50 = 6900 nM T26463 CD72OK 44412489 IC50 = 21000 nM T26463 C5V2QB 44412490 IC50 = 3700 nM T26463 C6V1JG 44604808 IC50 > 20000 nM T26463 CQ1N2M 44605023 IC50 > 20000 nM T26463 CNK9D2 44607341 IC50 > 20000 nM T26463 CCQS46 46830304 IC50 > 20000 nM T26463 CVAT67 53317946 IC50 > 500000 nM T26463 CT7D5O 53320320 IC50 > 100000 nM T26463 CK6RI2 53324652 IC50 > 100000 nM T26463 CY32HG 54677477 IC50 > 10000 nM T26463 C0ZG2V 54709839 IC50 > 200000 nM T26463 CLT3Q8 54716246 IC50 > 10000 nM T26463 CU9M3O 56832906 IC50 > 200000 nM T26463 CDS0C6 66825540 IC50 > 500000 nM T26463 CH1S3G 71548918 IC50 > 25000 nM T26463 CFG02R 73669532 IC50 > 500000 nM T26463 C9DY6C 76318645 IC50 = 45000 nM T26463 CQ29OX 76325888 IC50 > 500000 nM T26463 CSJ2W1 86302310 EC50 = 80000 nM T26463 C6ZY2A 90654414 EC50 > 500000 nM T26463 CXN6B4 90654415 EC50 > 500000 nM T26463 CSH13R 90654416 EC50 > 500000 nM T26463 C0PC8E 90654417 EC50 = 250000 nM T26463 CR2OE7 90654418 EC50 > 500000 nM T26463 CRP0L2 90654419 EC50 = 70000 nM T26463 C1Y5EA 90654420 EC50 = 410000 nM T26463 CW1B9O 90654421 EC50 > 500000 nM T26463 CU4G2C 117940941 IC50 = 20200 nM T26463 CT6M7E 135435051 IC50 = 46000 nM T26463 CW0CR6 135435052 Ki = 44000 nM T26463 CD38IL 135435084 Ki = 7500 nM T26463 CD5QA6 135435086 Ki = 1760000 nM T26463 C63ONQ 135435181 IC50 > 50000 nM T26463 CZ4GP6 135446244 IC50 > 10000 nM T26463 CUBV31 135485600 IC50 = 2500 nM T26463 CZH2Y8 135537671 Ki = 2300 nM T26463 C1EDK4 136030640 IC50 > 100000 nM T26463 C2H5PQ 136215370 Ki = 1 nM T26463 C8BJ0A 134007 EC50 = 4000 nM T26463 C0UQH8 516384 EC50 = 8000 nM T26463 C91IWY 516389 EC50 = 3000 nM T26463 CID8Z7 516390 EC50 = 5000 nM T26463 CLU03S 516391 EC50 = 3000 nM T26463 C5P8LV 516396 EC50 = 4000 nM T26463 CT01UL 516397 EC50 = 1000 nM T26463 CP5BZ4 5271338 EC50 = 7000 nM T26463 D02DLW 5997 IC50 > 500000 nM T99089 D05ROI 44462760 IC50 = 0.4 nM T99089 D07POC 176870 IC50 = 60 nM T99089 D09GDD 11167602 IC50 = 1.5 nM T99089 D09XZB 123631 IC50 = 2000 nM T99089 D0AZ3C 5291 IC50 > 100000 nM T99089 D0J9ZR 4477 IC50 > 100000 nM T99089 D0K8KX 5280343 IC50 = 7589 nM T99089 D0TK7R 50922675 IC50 = 0.3 nM T99089 D0W5HK 216239 IC50 = 1 nM T99089 D0Y9EW 42611257 IC50 = 4 nM T99089 D02UFQ 11620908 IC50 > 10000 nM T99089 D03AND 11656518 IC50 = 20 nM T99089 D03LWG 53235510 IC50 = 4142 nM T99089 D04AHQ 71721540 IC50 = 1.5 nM T99089 D04MXN 56846693 IC50 = 82 nM T99089 D0E3TC 44259 IC50 = 4.5 nM T99089 D0F5JZ 24180719 Ki = 2.6 nM T99089 D0K0YC 9826528 IC50 = 6 nM T99089 D0M5XN 89670174 IC50 = 23 nM T99089 D0O2FN 16222096 IC50 = 1.8 nM T99089 D0T4QA 90456533 IC50 = 0.4 nM T99089 D0Z2FD 56931136 IC50 = 6 nM T99089 D04SWX 56924694 IC50 = 270 nM T99089 D0B7VP 46198319 IC50 = 26 nM T99089 D0T3ME 156422 IC50 = 83.4 nM T99089 CB37VR 5034 IC50 = 29.6 nM T99089 C63WLY 89644 IC50 > 10 ug.mL-1 T99089 C5JE2Z 104860 IC50 = 6.7 ug.mL-1 T99089 CI1NA5 159926 IC50 = 6.4 ug.mL-1 T99089 CYBA43 177458 IC50 > 10 ug.mL-1 T99089 C9VW8M 449054 IC50 > 16000 nM T99089 COI61Y 660701 IC50 > 100000 nM T99089 CG1YH4 690397 IC50 = 830 nM T99089 C41EFM 691845 IC50 = 670 nM T99089 C9IL3X 697391 IC50 = 6100 nM T99089 CKX97G 698872 IC50 = 730 nM T99089 CRB31Z 741849 IC50 = 2100 nM T99089 CH9O0J 751729 IC50 > 100000 nM T99089 C82CGY 777751 IC50 > 100000 nM T99089 C4D2FR 817983 IC50 = 30110 nM T99089 C2SW3J 838432 IC50 = 740 nM T99089 C62VFD 903392 IC50 = 2010 nM T99089 C3ZTU4 985658 IC50 = 11080 nM T99089 CP9L1G 1006450 IC50 = 2230 nM T99089 CRP32Q 1006453 IC50 = 3450 nM T99089 CJF53S 1016049 IC50 = 1020 nM T99089 CF80DN 1032682 IC50 > 100000 nM T99089 CD12EO 1040090 IC50 > 100000 nM T99089 C26TIY 1088625 IC50 > 100000 nM T99089 CGP84Q 1102777 IC50 = 470 nM T99089 C6X1YI 1124092 IC50 = 4010 nM T99089 CMS5J7 1207521 IC50 = 1800 nM T99089 C01WYP 1220545 IC50 = 1160 nM T99089 CJ7M4N 1236338 IC50 > 100000 nM T99089 COH8I7 1496173 IC50 = 630 nM T99089 CG3F6Y 1684063 IC50 = 2160 nM T99089 CKR8H5 1684186 IC50 = 770 nM T99089 CEPI38 1737233 IC50 = 1540 nM T99089 CPI69L 1740003 IC50 = 4110 nM T99089 C17WVD 1771530 IC50 = 2490 nM T99089 CD76PH 1774314 IC50 = 4020 nM T99089 CKG4R9 1774320 IC50 = 3240 nM T99089 CU0O5C 1776533 IC50 = 4750 nM T99089 CLOW51 1776608 IC50 = 1600 nM T99089 CN6O3E 1793969 IC50 = 1650 nM T99089 CS2JL0 1814300 IC50 = 310 nM T99089 C3B5PI 1814302 IC50 = 970 nM T99089 CCI76Z 1814304 IC50 = 820 nM T99089 CN3G5B 1814306 IC50 = 440 nM T99089 CG02RT 1814308 IC50 = 1140 nM T99089 CC54MB 1814310 IC50 = 500 nM T99089 C27FVB 2133813 IC50 = 570 nM T99089 CZ6EV4 2133817 IC50 = 100 nM T99089 C5GYO1 2730801 IC50 = 320 nM T99089 CZE13I 2816786 IC50 = 400 nM T99089 CJ5UL8 2855606 IC50 > 100000 nM T99089 CMG0F6 2961623 IC50 = 400 nM T99089 CB4QI1 2966018 IC50 = 3000 nM T99089 CHC5I0 2971839 IC50 = 1800 nM T99089 CFY1D0 2974957 IC50 = 17 nM T99089 CW3DC7 2977311 IC50 = 800 nM T99089 C4RH3J 3106064 IC50 = 1720 nM T99089 C1GTF0 3143674 IC50 > 100000 nM T99089 C2HUN0 3235666 IC50 > 100000 nM T99089 C2H0KF 3718048 IC50 = 380 nM T99089 C73RZL 3937063 IC50 = 900 nM T99089 C4FDE6 4647084 IC50 > 100000 nM T99089 CDQ3M7 5359485 IC50 = 1.6 ug.mL-1 T99089 C54BYP 5360741 IC50 = 4.8 ug.mL-1 T99089 CTFA62 5521855 IC50 = 37480 nM T99089 C6J1DO 5716697 IC50 = 900 nM T99089 CE0SB4 5753911 IC50 > 50000 nM T99089 CXZ30D 5753913 IC50 = 11360 nM T99089 CFO1B9 5753916 IC50 = 4600 nM T99089 CM87HL 5753919 IC50 = 57890 nM T99089 CK08PH 5753938 IC50 = 10910 nM T99089 CFSD40 6510636 IC50 = 17360 nM T99089 C6KN7F 6877485 IC50 > 100000 nM T99089 C9U7GE 7718544 IC50 = 340 nM T99089 CSX8V7 7897116 IC50 = 400 nM T99089 C5GE7T 9917045 IC50 = 7200 nM T99089 C5E7HJ 10217017 IC50 = 2 nM T99089 C7S9KW 10222594 IC50 = 40 nM T99089 CXC91Z 11167118 IC50 = 280 nM T99089 CC6VK1 11236275 IC50 = 310 nM T99089 CM30TC 11387552 EC50 = 100 nM T99089 C0Z9YQ 11433057 EC50 = 100 nM T99089 CZ73AJ 11476663 IC50 = 1 nM T99089 CD6QW4 11494370 IC50 = 20000 nM T99089 CU30IV 11501142 IC50 = 10000 nM T99089 CFMS75 11501578 IC50 = 27000 nM T99089 CWZS50 11501869 IC50 = 37000 nM T99089 CB6ME8 11503895 IC50 = 47 nM T99089 C7Q5JI 11516491 IC50 = 3 nM T99089 CUDR26 11518018 IC50 = 12 nM T99089 C8AY3B 11518031 IC50 = 0.46 nM T99089 C6D9OT 11522875 IC50 = 8000 nM T99089 C3LGD4 11523321 IC50 = 3.46 nM T99089 CXP87N 11523639 IC50 = 950 nM T99089 CL7X4Q 11530963 IC50 = 40000 nM T99089 CX4D8Z 11532611 IC50 = 16 nM T99089 CCU2B0 11544514 IC50 = 45000 nM T99089 CJ23SH 11545064 IC50 = 5200 nM T99089 C6I9YN 11545261 IC50 = 0.33 nM T99089 CP3JY9 11546962 IC50 = 8300 nM T99089 C7H9FD 11551727 IC50 = 26000 nM T99089 C60ORJ 11552560 IC50 = 4500 nM T99089 CCQ4L1 11552561 IC50 = 34000 nM T99089 C0OHL1 11561411 IC50 = 1240 nM T99089 CAXP50 11566757 IC50 = 0.87 nM T99089 C4NS5D 11573300 IC50 > 100000 nM T99089 COFT94 11573823 IC50 = 65000 nM T99089 CX2B3N 11574129 IC50 = 3000 nM T99089 C34QRP 11574273 IC50 = 790 nM T99089 CPLH36 11574625 IC50 = 2300 nM T99089 C03WNJ 11574718 IC50 = 26000 nM T99089 CE30QF 11574855 IC50 = 7 nM T99089 C4O0VX 11580569 IC50 = 14000 nM T99089 C1HCK9 11581360 IC50 = 8800 nM T99089 CX4W5I 11583265 IC50 > 100000 nM T99089 CEM6P4 11583341 IC50 = 24 nM T99089 CKWN65 11588629 IC50 = 1300 nM T99089 C40YLN 11590139 IC50 = 39000 nM T99089 CK63UF 11595532 IC50 = 4000 nM T99089 C28FJS 11597486 IC50 = 61 nM T99089 CZGU14 11601866 IC50 = 1.4 nM T99089 CQ9DC4 11602668 IC50 = 33000 nM T99089 CTB45J 11603925 IC50 = 14000 nM T99089 C8YIS9 11604883 IC50 = 333 nM T99089 CZD5J8 11605467 IC50 = 497 nM T99089 C8A2LO 11610758 IC50 = 1.2 nM T99089 CP62YV 11616462 IC50 = 0.02 nM T99089 CBWP68 11624720 IC50 = 3000 nM T99089 C0OGU9 11624721 IC50 = 9800 nM T99089 CS17RF 11624965 IC50 = 0.22 nM T99089 CSM62L 11626920 IC50 = 27 nM T99089 C9K7QI 11632277 IC50 = 38000 nM T99089 CH7YA4 11633452 IC50 > 100000 nM T99089 CU98ZH 11633786 IC50 = 15 nM T99089 CS2K5N 11634109 IC50 = 192 nM T99089 C34HID 11634929 IC50 = 135 nM T99089 CMSA04 11639637 IC50 = 0.34 nM T99089 C4RX1P 11639649 IC50 = 5200 nM T99089 C6L4EZ 11645222 IC50 = 33000 nM T99089 C8Y6CU 11653652 IC50 = 0.03 nM T99089 C24KYX 11659444 IC50 = 77 nM T99089 C3PT8Y 11660026 IC50 = 74000 nM T99089 C8J7IA 11660270 IC50 = 0.39 nM T99089 C40LAT 11660528 IC50 = 3800 nM T99089 CAW41S 11667128 IC50 = 2.4 nM T99089 CT29KC 11667144 IC50 = 4000 nM T99089 CULF07 11676720 IC50 = 16 nM T99089 C4Q2OK 11681939 IC50 > 100000 nM T99089 CK42CI 11682654 IC50 = 3500 nM T99089 C8JW5Z 11696578 IC50 = 1120 nM T99089 C4WM6K 11697289 IC50 = 26 nM T99089 C6LQ9H 11702547 IC50 = 4200 nM T99089 CZ4E6K 11703339 IC50 = 12 nM T99089 C86TWZ 11704203 IC50 = 37000 nM T99089 CE30QZ 11704625 IC50 = 14 nM T99089 CQ2P3D 11704845 IC50 = 45 nM T99089 CAL4G1 11705461 IC50 = 90 nM T99089 CI0CM8 11709835 IC50 = 1400 nM T99089 CW5H0K 11710340 IC50 = 3000 nM T99089 CVR15H 11710382 IC50 = 26000 nM T99089 CGI1D9 11717001 Ki = 0.13 nM T99089 C1DF0R 11717449 IC50 = 490 nM T99089 C8O1MN 11719900 IC50 = 45 nM T99089 C5YXA3 11720025 IC50 > 100000 nM T99089 C2EX5W 11737996 IC50 = 900 nM T99089 C8MOK3 11750699 IC50 = 25 nM T99089 C39TYN 11841124 IC50 > 100000 nM T99089 CHAD78 11841127 IC50 > 100000 nM T99089 CA2LF8 11947957 IC50 = 236.7 nM T99089 CDGF78 15282555 IC50 = 2700 nM T99089 C7LB4I 15949613 IC50 = 900 nM T99089 CS3EB6 16044861 IC50 = 1.4 nM T99089 C0Z6VU 16045086 IC50 = 1 nM T99089 CA1T2U 16045087 IC50 = 16 nM T99089 C04TRQ 16045682 IC50 = 3 nM T99089 C35ILP 16045759 IC50 = 52 nM T99089 CQ4O0Y 16045761 IC50 = 3 nM T99089 C1VS7Q 16045839 IC50 = 1.1 nM T99089 CCFT24 16046014 IC50 = 1.4 nM T99089 CE43QM 16064288 IC50 = 130 nM T99089 CELY15 16064449 IC50 = 780 nM T99089 C8UOX0 16064748 IC50 = 480 nM T99089 CFKE48 16064750 IC50 = 120 nM T99089 CC7QD3 16064891 IC50 = 210 nM T99089 CLG6R7 16064892 IC50 = 42 nM T99089 C0C2QW 16064893 IC50 = 620 nM T99089 CM3A7W 16066694 IC50 = 19 nM T99089 CVE6C8 16086088 IC50 = 27 nM T99089 CU5Y7N 16101466 IC50 = 199 nM T99089 C5VPH9 16129448 IC50 > 10000 nM T99089 CZ08YH 16214904 IC50 = 53 nM T99089 CFN5D6 16223710 IC50 = 5.1 nM T99089 CB65EI 16223711 IC50 = 45 nM T99089 C8EF0N 16223900 IC50 = 49 nM T99089 C45HCU 16223901 IC50 = 93 nM T99089 CVIU65 16223902 IC50 = 1550 nM T99089 C1L8UO 16224102 IC50 = 933 nM T99089 CK5TJ0 16678105 IC50 = 17.4 nM T99089 C0EV8X 19355820 IC50 > 1000 nM T99089 C6AV4G 21023795 IC50 = 14 nM T99089 C4AK5J 21037180 IC50 = 25 nM T99089 C9YR7W 21037208 IC50 = 68 nM T99089 C8ID6R 21037243 EC50 > 10000 nM T99089 C2V1EQ 21037245 EC50 > 10000 nM T99089 CZ23BW 21037364 IC50 = 140 nM T99089 CJ4E1M 22040403 IC50 = 2700 nM T99089 C8VJ3A 22040410 IC50 = 1300 nM T99089 CHFO54 22040436 EC50 = 7000 nM T99089 CJ3UH0 22040625 IC50 = 11 nM T99089 C02DQZ 22040627 IC50 = 11 nM T99089 CCA1D7 22040647 IC50 = 39 nM T99089 C4RP8N 22040656 IC50 = 63 nM T99089 C9A4LW 22040760 IC50 = 13 nM T99089 CI3V6C 22040802 IC50 = 130 nM T99089 C9WU0J 22040805 IC50 = 2400 nM T99089 CDN61H 22040847 IC50 = 39 nM T99089 C3SX8H 22040857 IC50 = 9000 nM T99089 C6NM3T 22040925 IC50 = 140 nM T99089 CC84UT 22040937 IC50 = 1900 nM T99089 CZM5W1 22040941 IC50 = 8 nM T99089 C6FMB5 22040978 IC50 = 500 nM T99089 CRJ4H3 22041111 IC50 = 7700 nM T99089 CO37NP 22041112 IC50 = 4400 nM T99089 C4UMZ2 22041119 IC50 = 300 nM T99089 CI5KM3 22041171 IC50 = 88 nM T99089 C51FDU 22041175 IC50 = 26 nM T99089 CR3G0K 22041260 EC50 = 3200 nM T99089 C69BSO 22041261 IC50 = 28 nM T99089 CGX61W 22041319 IC50 = 45 nM T99089 CDM83W 22057968 IC50 = 2 nM T99089 CQJ59G 22185379 IC50 = 8 nM T99089 CFMT70 22185475 IC50 = 6 nM T99089 C0X7MW 22185489 IC50 = 13 nM T99089 CL5D8X 22256705 IC50 = 33 nM T99089 CXS28L 22918445 IC50 = 338 nM T99089 C7HUS0 23585267 IC50 = 32 nM T99089 CHQ23N 23585318 IC50 = 26 nM T99089 COSI68 23585320 IC50 = 20 nM T99089 CR2AN0 24180721 IC50 > 100000 nM T99089 CC6JO7 24737670 IC50 = 19 nM T99089 CZ8BQ6 24737709 IC50 = 110 nM T99089 C4GUC1 24738493 IC50 = 316 nM T99089 CLH3G9 24738495 IC50 = 718 nM T99089 CCO8T6 24738496 IC50 = 407 nM T99089 CHU49V 24757938 IC50 = 40 nM T99089 C7YG1N 24759534 IC50 = 550 nM T99089 CCPS81 24764502 IC50 > 35000 nM T99089 CC13WT 24768568 IC50 = 99 nM T99089 CCP2M3 24822704 IC50 = 32 nM T99089 CA4D9N 24829351 IC50 = 6 nM T99089 CCS58O 24863072 IC50 = 70 nM T99089 C6R4ZU 24863189 IC50 = 310 nM T99089 C6C2GX 24863500 IC50 = 110 nM T99089 CYVB83 24863584 IC50 = 18 nM T99089 CQ15ML 24863670 IC50 = 21 nM T99089 C4XZ3N 24863671 IC50 = 270 nM T99089 CU53DP 24878669 IC50 = 1400 nM T99089 C6Q4FC 24878670 IC50 = 92000 nM T99089 CUIS63 24878671 IC50 = 650 nM T99089 CGKA14 24878672 IC50 = 2500 nM T99089 C0P4HO 24879140 IC50 = 2900 nM T99089 CBUG02 24879141 IC50 = 1160 nM T99089 CSJ7T8 24879142 IC50 = 16000 nM T99089 CBL6M7 24879143 IC50 = 14000 nM T99089 CE74NO 24879204 IC50 = 12000 nM T99089 C48MIN 24879205 IC50 = 1200 nM T99089 CG5VC1 24879206 IC50 = 45000 nM T99089 CY18ZW 24879207 IC50 = 18000 nM T99089 C1XL8V 24879208 IC50 = 10000 nM T99089 C9SM2H 24879209 IC50 = 3800 nM T99089 CTPU27 24879260 IC50 = 76000 nM T99089 CBQN65 24879261 IC50 = 70000 nM T99089 CZ8CR2 24879262 IC50 = 45000 nM T99089 CD1QW9 24879263 IC50 = 36000 nM T99089 C8UPO4 24879264 IC50 = 5500 nM T99089 CDCN49 24879265 IC50 = 410 nM T99089 CYTM29 24879326 IC50 = 26000 nM T99089 C2F6KO 24879328 IC50 = 560 nM T99089 C6S2JM 24879329 IC50 > 100000 nM T99089 C1BJT3 24879330 IC50 = 22000 nM T99089 CK83CA 24879331 IC50 = 16000 nM T99089 C1CP0D 24879390 IC50 = 4700 nM T99089 CJZB61 24879392 IC50 = 19000 nM T99089 C8L0FE 24879393 IC50 = 31000 nM T99089 CT12IR 24879394 IC50 = 16000 nM T99089 C3T4CF 24879395 IC50 = 9800 nM T99089 CH4F5C 24879396 IC50 = 7400 nM T99089 C6TRZ7 24879462 IC50 = 44000 nM T99089 CKJ12G 24879463 IC50 = 1500 nM T99089 CGL5B4 24879464 IC50 = 29000 nM T99089 C4YA3G 24879465 IC50 = 29000 nM T99089 C96NEC 24879466 IC50 = 18000 nM T99089 CTZD56 24879467 IC50 = 22000 nM T99089 CAX20R 24879527 IC50 = 10000 nM T99089 CW8HQ4 24879528 IC50 = 56000 nM T99089 CBT3Y5 24879529 IC50 = 13000 nM T99089 C0ZBE3 24879530 IC50 = 19000 nM T99089 C7SQE5 24879531 IC50 = 34000 nM T99089 CV8Z3B 24879532 IC50 = 11000 nM T99089 C13QYB 24884503 IC50 = 24 nM T99089 C5E1YD 24891645 IC50 = 77 nM T99089 C2T9IQ 24891646 IC50 = 38 nM T99089 C4B7ND 24891647 IC50 = 57 nM T99089 C7Y8KZ 24891698 IC50 = 26.92 nM T99089 C6HE2Y 24891699 IC50 = 32 nM T99089 CK1R3B 24891700 IC50 = 51 nM T99089 CCY7G3 24891701 IC50 = 190 nM T99089 CJH19T 24894883 IC50 = 50000 nM T99089 CB5TP8 24894992 IC50 = 38000 nM T99089 CN13JF 24899915 IC50 = 0.74 ug.mL-1 T99089 CBWR97 24899916 IC50 = 1.5 ug.mL-1 T99089 C9F2JD 24899917 IC50 > 10 ug.mL-1 T99089 C64MTI 24900160 IC50 = 7.4 ug.mL-1 T99089 CO2I6Q 24900161 IC50 = 9 ug.mL-1 T99089 CQL3U0 24963235 IC50 = 1700 nM T99089 C26IGP 24963239 IC50 = 28 nM T99089 CJZE02 24963588 IC50 = 17 nM T99089 CAL45P 24963945 IC50 = 260 nM T99089 C1E7SQ 24964302 IC50 = 5 nM T99089 CA0QG4 24964658 IC50 = 6.5 nM T99089 C2U9TM 24965013 IC50 = 156 nM T99089 C09IXV 24965362 IC50 = 9 nM T99089 CR8N5G 24965367 IC50 = 1400 nM T99089 CTY2A7 24965371 IC50 = 41.5 nM T99089 C12PMT 24966065 IC50 = 18 nM T99089 CKRV37 24966066 IC50 = 15.4 nM T99089 C9YN2Q 24967131 IC50 = 42 nM T99089 COD0C3 24967871 IC50 = 216 nM T99089 CJ7ZD9 24968217 IC50 = 1500 nM T99089 C7HJU9 24968561 IC50 = 6.7 nM T99089 CT7S6C 24969040 IC50 = 360 nM T99089 CFDW17 24969041 IC50 > 10000 nM T99089 CD5HQ0 24969301 IC50 = 1540 nM T99089 C9NA3Z 24969303 IC50 > 10000 nM T99089 C9TQ4B 24969304 IC50 > 10000 nM T99089 C92TKX 24969393 IC50 = 1570 nM T99089 C78KAJ 24969394 IC50 > 10000 nM T99089 C97NFP 24969396 IC50 > 10000 nM T99089 C9FS1C 24969397 IC50 = 360 nM T99089 C85RQC 24969401 IC50 = 4270 nM T99089 CC23PA 24969484 IC50 > 10000 nM T99089 CDBL83 24969487 IC50 > 10000 nM T99089 CO4A0P 24969567 IC50 = 1030 nM T99089 CTJP28 24969568 IC50 > 10000 nM T99089 CL9UY3 24969569 IC50 > 10000 nM T99089 C0VK5E 24969668 IC50 = 500 nM T99089 CB9C5O 24969749 IC50 = 540 nM T99089 CW26KA 24969750 IC50 = 3600 nM T99089 C4AXL1 24969752 IC50 > 10000 nM T99089 CG6B9I 24969834 IC50 > 10000 nM T99089 C2M4FP 24969839 IC50 = 240 nM T99089 CB89UG 24969923 IC50 = 5880 nM T99089 C3K2VT 24970000 IC50 = 6340 nM T99089 CX8MC1 24970159 IC50 > 10000 nM T99089 CB0XA4 24970161 IC50 > 10000 nM T99089 CL7A6B 24970246 IC50 > 10000 nM T99089 C4G9WP 24986335 IC50 = 89 nM T99089 CDF57P 24995525 IC50 = 2.5 nM T99089 C9QO8R 25023945 IC50 = 57710 nM T99089 C4Y3FG 25023946 IC50 = 3750 nM T99089 CA61PS 25066845 IC50 = 22 nM T99089 CR46MG 25066846 IC50 = 2 nM T99089 C9Z3LB 25093294 IC50 = 86000 nM T99089 CM0E1C 25093324 IC50 = 68 nM T99089 CM4R0H 25093325 IC50 = 4.4 nM T99089 C5JX6H 25093326 IC50 = 1.5 nM T99089 C1DGE0 25093327 IC50 = 94 nM T99089 C9UW5V 25093328 IC50 = 70 nM T99089 C96EVA 25118036 IC50 = 51 nM T99089 CTV54O 25123227 IC50 > 10000 nM T99089 CG3XC9 25124150 IC50 = 80 nM T99089 CO2IR5 25124816 IC50 > 2000 nM T99089 C1IYN7 25127854 IC50 > 1000 nM T99089 CKD14B 25127856 IC50 = 290 nM T99089 CJBX60 25128180 IC50 > 1000 nM T99089 CC5SD9 25128181 IC50 > 1000 nM T99089 C9PL5S 25137959 IC50 > 25000 nM T99089 CVJ0S5 25137960 IC50 = 14 nM T99089 CJL80R 25161176 IC50 = 70 nM T99089 C85KCS 25178328 IC50 = 8000 nM T99089 CIG4H0 25178539 IC50 = 1200 nM T99089 C4GI6J 25178540 IC50 = 8400 nM T99089 CB6QT3 25195001 IC50 = 7 nM T99089 CYK1V8 25206185 IC50 = 5.6 nM T99089 C6FGQ1 25206346 IC50 = 47 nM T99089 C8ZBN0 25206349 IC50 = 15 nM T99089 CRO09K 25211064 IC50 = 8800 nM T99089 C41TLH 42603880 IC50 = 82000 nM T99089 CDM2N3 42606902 IC50 = 5940 nM T99089 CWS37O 42618140 IC50 > 10000 nM T99089 C2JV3O 42618143 IC50 > 10000 nM T99089 CG01BO 42618144 IC50 > 10000 nM T99089 CLD0M5 42625161 IC50 = 40 nM T99089 CS1CB9 42625162 IC50 = 85 nM T99089 CRUS43 42625163 IC50 > 100000 nM T99089 C27GYX 42625164 IC50 = 15900 nM T99089 CJ9EQ2 42625165 IC50 = 17200 nM T99089 CL8R1T 42625166 IC50 = 14000 nM T99089 C41PMY 42625241 IC50 = 28 nM T99089 CZPU80 42625242 IC50 > 100000 nM T99089 CDT39F 42625243 IC50 > 100000 nM T99089 CV5X0D 42625244 IC50 = 16700 nM T99089 C7HYW8 42625245 IC50 = 10000 nM T99089 CPV58O 42625246 IC50 > 100000 nM T99089 C3M2OV 42625324 IC50 = 10000 nM T99089 CC95QE 42625325 IC50 = 850 nM T99089 CV6CR3 42625326 IC50 > 100000 nM T99089 CK4Y8O 42625327 IC50 > 100000 nM T99089 CRP62O 42625328 IC50 > 100000 nM T99089 CIRG39 42625329 IC50 = 12200 nM T99089 CIR6N1 42625412 IC50 = 10000 nM T99089 C21YCQ 42625413 IC50 = 32500 nM T99089 CA1Y7G 42625505 IC50 = 23 nM T99089 CIGZ52 42626129 IC50 > 100000 nM T99089 CE6X4U 42626130 IC50 > 100000 nM T99089 C0IYC6 42626192 IC50 = 100 nM T99089 CMV35J 42626193 IC50 = 14 nM T99089 CN7A2L 42626194 IC50 > 100000 nM T99089 C98ZKU 42626195 IC50 > 100000 nM T99089 CP06XJ 42626196 IC50 = 21 nM T99089 C3GA4B 42626197 IC50 = 12 nM T99089 CWRD96 42626265 IC50 = 27 nM T99089 CLZ5T1 42626266 IC50 = 52 nM T99089 C4NW1Z 42626267 IC50 = 2840 nM T99089 CV3KQ7 42626268 IC50 = 600 nM T99089 C62UVE 42626269 IC50 = 860 nM T99089 CUA5H1 42626270 IC50 = 22 nM T99089 CEZW83 42626338 IC50 = 163 nM T99089 CQ9UV2 42626339 IC50 = 60 nM T99089 C5QG1C 42626340 IC50 = 46 nM T99089 CZ0CB6 42626341 IC50 = 61 nM T99089 CP2US6 42626342 IC50 = 305 nM T99089 CE2G9C 42626343 IC50 = 29 nM T99089 C4CX1E 42628843 IC50 = 5 nM T99089 CU9E4P 42629114 IC50 > 10000 nM T99089 CJ5U1X 42639664 IC50 = 6.5 ug.mL-1 T99089 CJT32G 42641056 IC50 = 600 nM T99089 CH8JQ9 42647197 IC50 = 464 nM T99089 CZP1I5 44131523 IC50 = 5 nM T99089 CRW8G5 44131524 IC50 = 4890 nM T99089 CYL5C1 44131526 IC50 = 168 nM T99089 CRN89T 44131527 IC50 = 187 nM T99089 CS15GI 44131710 IC50 = 4 nM T99089 C4LV1X 44131711 IC50 = 6 nM T99089 COH4S6 44131713 IC50 = 30 nM T99089 C7CJ9L 44132041 IC50 = 273 nM T99089 CLC25G 44132209 IC50 = 650 nM T99089 CZN36J 44132210 IC50 = 1080 nM T99089 CVEL46 44132212 IC50 = 222 nM T99089 CJ2U8W 44132374 IC50 = 43 nM T99089 CVC68Z 44132375 IC50 = 7 nM T99089 CN8D9W 44132531 IC50 = 134 nM T99089 CRAF54 44132532 IC50 = 280 nM T99089 CW8J5B 44132533 IC50 = 75 nM T99089 C1C0EF 44132534 IC50 = 640 nM T99089 C81MAW 44132690 IC50 = 7 nM T99089 C60THF 44132691 IC50 = 220 nM T99089 CKH43U 44132693 IC50 = 1700 nM T99089 CQB12C 44132694 IC50 = 8200 nM T99089 C7CH1O 44132849 IC50 = 600 nM T99089 CMIJ65 44132851 IC50 = 20 nM T99089 CF8IC2 44132852 IC50 = 101 nM T99089 C42STZ 44132853 IC50 = 15 nM T99089 C59VWU 44133012 IC50 = 2 nM T99089 CMG6E1 44133013 IC50 = 6 nM T99089 CL41OB 44133016 IC50 = 16000 nM T99089 C24APO 44133177 IC50 = 320 nM T99089 CW67CZ 44133180 IC50 = 3 nM T99089 C7OF9J 44133181 IC50 = 2 nM T99089 CIL5W6 44133361 IC50 = 750 nM T99089 CJK24I 44133362 IC50 = 3800 nM T99089 CVO95C 44133363 IC50 = 107 nM T99089 CM92WZ 44133364 IC50 = 246 nM T99089 C8TDB9 44133365 IC50 = 76 nM T99089 C1X4ZY 44133544 IC50 = 21 nM T99089 CZ20KG 44133545 IC50 = 390 nM T99089 CQ9M1C 44133546 IC50 = 133 nM T99089 CW8QC6 44133547 IC50 = 4200 nM T99089 CH9U7K 44133548 IC50 = 71 nM T99089 CZ0DA5 44133720 IC50 = 870 nM T99089 CMO9J8 44133721 IC50 = 7 nM T99089 CLSG50 44133722 IC50 = 21 nM T99089 CT6L2M 44133724 IC50 = 176 nM T99089 C94MCL 44133726 IC50 = 84 nM T99089 C4NDM9 44133727 IC50 = 108 nM T99089 CCSZ12 44133728 IC50 = 634 nM T99089 CV35ZJ 44133905 IC50 = 10 nM T99089 C97QTV 44133906 IC50 = 96 nM T99089 C3G4NP 44133907 IC50 = 10000 nM T99089 CI7OR1 44133908 IC50 = 8 nM T99089 CR2G0E 44133909 IC50 = 8 nM T99089 C4NP8V 44133910 IC50 = 105 nM T99089 CY1I5F 44133911 IC50 = 580 nM T99089 CTQ1A5 44133913 IC50 = 48 nM T99089 CZV39F 44133914 IC50 = 4 nM T99089 C5F6PH 44134083 IC50 = 80 nM T99089 C9WFA4 44134086 IC50 = 4 nM T99089 C7UIJ2 44134087 IC50 = 5 nM T99089 C8M2WR 44134089 IC50 = 3 nM T99089 CL0O7M 44134090 IC50 = 34 nM T99089 C4QOM5 44134091 IC50 = 306 nM T99089 CO42DC 44138048 IC50 > 10000 nM T99089 CL65QV 44138049 IC50 > 10000 nM T99089 CC9W0L 44185009 IC50 = 56 nM T99089 C1M8UL 44185010 IC50 = 22 nM T99089 CWT0K9 44185011 IC50 = 47 nM T99089 C2Q8MJ 44185012 IC50 = 37 nM T99089 CM4R5H 44185013 IC50 = 12 nM T99089 CAM26B 44185065 IC50 = 16 nM T99089 CW76EU 44185067 IC50 = 6 nM T99089 C2H5XO 44185068 IC50 = 37 nM T99089 CFTR94 44185069 IC50 = 220 nM T99089 C64GVD 44185123 IC50 = 1 nM T99089 CD04VP 44185124 IC50 = 25 nM T99089 C0YWR1 44185125 IC50 = 8 nM T99089 CVC9N0 44185126 IC50 = 106 nM T99089 CS5OR8 44185840 IC50 = 346 nM T99089 C3OZ0X 44185841 IC50 = 23 nM T99089 CRUD71 44185842 IC50 = 1060 nM T99089 C5GRD7 44185843 IC50 = 10 nM T99089 CJ15VW 44185844 IC50 = 3140 nM T99089 CVM46R 44185900 IC50 > 10000 nM T99089 C84DOE 44185901 IC50 = 5200 nM T99089 C12VEW 44185902 IC50 = 90 nM T99089 C3ZAK0 44185961 IC50 = 430 nM T99089 CL74HV 44186294 IC50 = 59000 nM T99089 CTB03L 44186295 IC50 = 559 nM T99089 CV6NG7 44186296 IC50 = 10000 nM T99089 C81UIO 44186297 IC50 = 6500 nM T99089 C9Q4XW 44186359 IC50 = 1330 nM T99089 CUTO28 44186360 IC50 = 1 nM T99089 CZEN24 44186361 IC50 = 12 nM T99089 C3PG7E 44186362 IC50 = 7 nM T99089 CVA0Z8 44186363 IC50 = 37 nM T99089 CY40HO 44186413 IC50 = 638 nM T99089 CEFN41 44186414 IC50 = 17 nM T99089 C3W8HZ 44186415 IC50 = 24 nM T99089 CS5OR3 44186416 IC50 = 167 nM T99089 CB5U6Q 44186417 IC50 > 100000 nM T99089 CSV05I 44186463 IC50 = 79 nM T99089 C7RQ3H 44186464 IC50 = 4600 nM T99089 CCFQ29 44187005 IC50 = 0.16 nM T99089 C6L0DV 44199408 IC50 = 38 nM T99089 CKJ29G 44199417 IC50 = 61 nM T99089 CN0D5T 44199425 IC50 = 17 nM T99089 C1X2HU 44199429 IC50 = 917 nM T99089 CMT07V 44207795 IC50 = 0.8 nM T99089 C6FKU5 44207796 IC50 = 1.6 nM T99089 CPHJ03 44207797 IC50 = 0.6 nM T99089 CPM2Y8 44217243 IC50 = 110 nM T99089 C0J7XH 44223152 IC50 = 14 nM T99089 CXNB60 44223174 IC50 = 2.2 nM T99089 CX7YO1 44223205 IC50 = 8.2 nM T99089 CD91HX 44223206 IC50 = 4.8 nM T99089 C5N4AB 44223207 IC50 = 1.8 nM T99089 CHA12Y 44223280 IC50 = 6.3 nM T99089 C9LHU2 44223282 IC50 = 19 nM T99089 C4CTE2 44223283 IC50 = 87 nM T99089 C6A7VR 44223334 IC50 = 6.2 nM T99089 C2Z8JX 44223468 IC50 = 7.5 nM T99089 CH0I7B 44223469 IC50 = 2.3 nM T99089 C42DBL 44223470 IC50 = 13 nM T99089 CF6U5Q 44223471 IC50 = 1.7 nM T99089 C1ZS2O 44223472 IC50 = 1.3 nM T99089 CDL87A 44223473 IC50 = 2.4 nM T99089 CG4EH1 44223627 IC50 = 32 nM T99089 CG74KN 44223631 IC50 = 2.4 nM T99089 C0XR3Z 44223650 IC50 = 4 nM T99089 CI8ZU0 44223675 IC50 = 1.1 nM T99089 CQ1N4G 44223692 IC50 = 12 nM T99089 CWCB51 44223693 IC50 = 2.7 nM T99089 CV6ZU8 44223890 IC50 = 9.2 nM T99089 CJ5Q7A 44223895 IC50 = 5.8 nM T99089 C8KT6W 44223912 IC50 = 3.4 nM T99089 C8KUI4 44223914 IC50 = 210 nM T99089 CM2T9S 44223915 IC50 = 88 nM T99089 CR7K2T 44223999 Ki = 1 nM T99089 CC38RW 44225585 IC50 = 87 nM T99089 CPRT47 44225586 IC50 = 1 nM T99089 CPH82M 44225587 IC50 = 4 nM T99089 C5SPW7 44225811 IC50 = 54.1 nM T99089 CF9OE0 44225812 IC50 < 2 nM T99089 CIP43R 44225813 IC50 = 0.4 nM T99089 C4JBC2 44225814 IC50 = 0.3 nM T99089 CR6SM1 44226026 IC50 = 8.5 nM T99089 CCT62X 44226027 IC50 = 43.5 nM T99089 CD29GR 44226028 IC50 = 0.5 nM T99089 C0UTL8 44226029 IC50 = 70.8 nM T99089 C89SFK 44226241 IC50 = 17 nM T99089 C7MB0L 44226447 IC50 = 0.9 nM T99089 CJUX24 44226448 IC50 = 9.7 nM T99089 CVT2A7 44226449 IC50 < 0.32 nM T99089 CA0C6B 44226657 IC50 = 3 nM T99089 CXM4N6 44227053 IC50 = 2 nM T99089 C8RDU2 44227055 IC50 = 0.4 nM T99089 C1CBY7 44227056 IC50 = 4.4 nM T99089 CF2BJ7 44227270 IC50 = 17 nM T99089 CJK49R 44227271 IC50 = 0.7 nM T99089 C2GHR8 44227272 IC50 = 4.4 nM T99089 CHX90P 44227273 IC50 = 45 nM T99089 CXD0P8 44227274 IC50 = 0.4 nM T99089 CC21ZI 44227474 IC50 > 1000 nM T99089 CI4CB1 44227477 IC50 > 1000 nM T99089 CZ37UW 44227694 IC50 = 46.6 nM T99089 CEL61X 44229839 IC50 > 10000 nM T99089 CY6C2X 44230849 IC50 = 1.6 nM T99089 CV7Q1M 44230852 IC50 = 40 nM T99089 CEW5F9 44230853 IC50 = 3.2 nM T99089 CK7LA1 44230854 IC50 = 1125 nM T99089 C7HC6Z 44230986 IC50 = 107 nM T99089 C4VL2B 44230987 IC50 = 167 nM T99089 CD5VW9 44230988 IC50 = 2.2 nM T99089 CJN28A 44230989 IC50 = 137 nM T99089 CR5C7A 44230990 IC50 = 4.4 nM T99089 C2Y8CF 44231119 IC50 = 1.5 nM T99089 CE5J4A 44231120 IC50 = 49 nM T99089 C0YE3K 44231121 IC50 = 2.2 nM T99089 C3T0VZ 44231122 IC50 = 1.1 nM T99089 C47HYD 44231123 IC50 = 86 nM T99089 CQW47T 44231243 IC50 = 1.4 nM T99089 C23DUC 44231244 IC50 = 1 nM T99089 CUJD31 44231246 IC50 = 8 nM T99089 C4ZV1S 44231247 IC50 = 0.76 nM T99089 C9GK4E 44231363 IC50 = 27 nM T99089 CC6B2Z 44231366 IC50 = 948 nM T99089 CDKW96 44231489 IC50 = 1560 nM T99089 C18YHD 44231490 IC50 = 60 nM T99089 CAKX67 44231491 IC50 = 59 nM T99089 CJW38K 44231605 IC50 = 31 nM T99089 CL2Q8X 44231720 IC50 = 1.4 nM T99089 C1JVN2 44231722 IC50 = 298 nM T99089 C41EIK 44231723 IC50 = 1.2 nM T99089 C2JU5V 44242890 IC50 = 93 nM T99089 CMO40X 44243006 IC50 = 2229 nM T99089 CDUE95 44243085 IC50 = 480 nM T99089 CI4DL6 44243129 IC50 = 121 nM T99089 CBG0P4 44243179 IC50 = 293 nM T99089 C8JVN0 44243219 IC50 = 52 nM T99089 CR30HI 44243260 IC50 = 165 nM T99089 C3EW0M 44243435 IC50 = 340 nM T99089 CT91HE 44243438 IC50 = 332 nM T99089 CTUV41 44243472 IC50 = 155 nM T99089 CA7NS4 44406429 IC50 = 13 nM T99089 CN3PH6 44406460 IC50 = 6 nM T99089 C43KQJ 44406537 IC50 = 12 nM T99089 CU09CR 44406595 IC50 = 1585 nM T99089 CC8Q4N 44406731 IC50 = 49600 nM T99089 C6B7KF 44406750 IC50 = 14000 nM T99089 CA5Q0P 44442388 IC50 = 34 nM T99089 C65YCN 44442389 IC50 = 138 nM T99089 CW02SD 44442390 IC50 = 175 nM T99089 C73GEP 44442391 IC50 = 6830 nM T99089 CX56BF 44442392 IC50 = 221 nM T99089 C6L3GV 44442393 IC50 = 1030 nM T99089 CX3J2I 44442394 IC50 = 397 nM T99089 C5QJ0P 44442395 IC50 = 634 nM T99089 CC3Z7Q 44442396 IC50 = 5 nM T99089 CLR10Z 44442397 IC50 = 110 nM T99089 C9UOK1 44442398 IC50 = 100 nM T99089 CE9T6W 44442399 IC50 = 153 nM T99089 CM6K2R 44442400 IC50 = 594 nM T99089 CW8JC5 44442401 IC50 = 349 nM T99089 CD1TY7 44442402 IC50 = 100 nM T99089 C4POG9 44442403 IC50 = 104 nM T99089 C0XHW1 44442404 IC50 = 112 nM T99089 CBSM51 44442405 IC50 = 156 nM T99089 CNT36H 44442406 IC50 = 142 nM T99089 CRA0Q8 44442407 IC50 = 165 nM T99089 C7YZ3M 44442408 IC50 = 101 nM T99089 CY9G0Q 44442409 IC50 = 146 nM T99089 C6XAR9 44442410 IC50 = 39 nM T99089 CJU4F6 44442411 IC50 = 64 nM T99089 CO0N1A 44442412 IC50 = 232 nM T99089 CIR9A7 44442413 IC50 = 192 nM T99089 CBQ51S 44442414 IC50 = 2560 nM T99089 CHP41T 44442415 IC50 = 191 nM T99089 CI26UX 44442416 IC50 = 154 nM T99089 C2W1RN 44442417 IC50 = 122 nM T99089 C4A9FD 44442418 IC50 = 69 nM T99089 CKC3J0 44442419 IC50 = 40 nM T99089 C10MKH 44448311 IC50 = 274 nM T99089 C1QN4V 44448333 IC50 = 141 nM T99089 CLQF97 44448334 IC50 = 469 nM T99089 C73THQ 44448354 IC50 = 16 nM T99089 C8XOE9 44448666 IC50 = 10 nM T99089 CEOA67 44448669 IC50 = 83 nM T99089 C0DPU3 44448725 IC50 = 18 nM T99089 CFQN07 44448726 IC50 = 85 nM T99089 CR85LO 44448746 IC50 = 40 nM T99089 C5Y2JR 44448747 IC50 = 3 nM T99089 CA76JX 44448748 IC50 = 4 nM T99089 C7N2AQ 44473101 IC50 = 34 nM T99089 C4MG3F 44473102 IC50 = 56 nM T99089 CA85NJ 44473103 IC50 = 44 nM T99089 C6Q7NU 44479258 IC50 = 2120 nM T99089 C29ZDL 44479262 IC50 = 23740 nM T99089 C0Y5OQ 44479517 IC50 = 2740 nM T99089 C3VRO9 44557921 IC50 > 10000 nM T99089 CVLW62 44569182 IC50 > 100000 nM T99089 CFQ6C8 44569219 IC50 > 100000 nM T99089 C1QLZ3 44571660 IC50 = 5 nM T99089 CDW02V 44571710 IC50 = 10500 nM T99089 C1L7TV 44571711 IC50 = 1 nM T99089 CT4DF8 44571712 IC50 = 21100 nM T99089 CJ69GM 44571753 IC50 = 580 nM T99089 CY0I9Q 44571754 IC50 = 1200 nM T99089 C4EHC9 44571755 IC50 = 625 nM T99089 CI8V0L 44571800 IC50 = 322 nM T99089 C7S0LB 44571801 IC50 = 16 nM T99089 CVJU90 44571802 IC50 = 15 nM T99089 C85RJP 44571803 IC50 = 16 nM T99089 CWFB42 44571820 IC50 = 320 nM T99089 CTRD67 44571867 IC50 = 15 nM T99089 CWN95Q 44571868 IC50 = 28 nM T99089 CQ09OS 44571869 IC50 = 237 nM T99089 C7M0ET 44571870 IC50 = 11 nM T99089 CTM2J1 44571913 IC50 = 30 nM T99089 C58MVO 44571914 IC50 = 115 nM T99089 CX5GH1 44571915 IC50 = 9 nM T99089 C21DSM 44571916 IC50 = 14 nM T99089 CWP80I 44571963 IC50 = 48 nM T99089 CGIH39 44571964 IC50 = 116 nM T99089 CCM0D8 44571965 IC50 = 38 nM T99089 C0M7TJ 44571966 IC50 = 79 nM T99089 CV17DO 44572009 IC50 = 48 nM T99089 C03AOY 44572010 IC50 = 205 nM T99089 CLG7X2 44572011 IC50 = 16 nM T99089 C9IPZ6 44572058 IC50 = 35 nM T99089 C42XRK 44572059 IC50 = 17 nM T99089 CDRK26 44572109 IC50 = 76 nM T99089 CP04MY 44583650 IC50 = 7 nM T99089 CM2RZ1 44586991 IC50 = 0.57 nM T99089 CFHM64 44587046 IC50 = 3.91 nM T99089 CW9KM4 44587047 IC50 = 0.04 nM T99089 C1MH9X 44587048 IC50 = 0.09 nM T99089 CFL31E 44587049 IC50 = 1.16 nM T99089 CMKX28 44587190 IC50 = 0.05 nM T99089 CY4V5F 44587191 IC50 = 0.56 nM T99089 C8KCO7 44587210 IC50 = 4.02 nM T99089 CTH20X 44587211 IC50 = 0.47 nM T99089 CU8E5Z 44587234 IC50 = 0.85 nM T99089 CXQ8E3 44587235 IC50 = 0.23 nM T99089 C9O4LW 44587236 IC50 = 969.6 nM T99089 C5FW7T 44587271 IC50 = 433.8 nM T99089 C3MO4A 44587272 IC50 = 68.4 nM T99089 CR3VE4 44587273 IC50 = 4.1 nM T99089 CI1K9L 44587274 IC50 = 2.1 nM T99089 CRZ43D 44587295 IC50 = 2.9 nM T99089 CY09FE 44587296 IC50 = 3.1 nM T99089 CWU29I 44587510 IC50 = 331 nM T99089 CNU73X 44587528 IC50 = 41.7 nM T99089 C8O3ES 44587529 IC50 = 170 nM T99089 C58DLS 44587530 IC50 = 110 nM T99089 C5QXC0 44587531 IC50 = 5.3 nM T99089 C5R2EI 44587550 IC50 = 25.7 nM T99089 CQN15G 44587551 IC50 = 10.5 nM T99089 C7OI4S 44587552 IC50 = 3.9 nM T99089 CM0UX7 44587582 IC50 = 5.4 nM T99089 CCS62T 44587583 IC50 = 2.1 nM T99089 CB4O9Z 44587584 IC50 = 79.4 nM T99089 C3Y5AW 44589519 IC50 = 7 nM T99089 C09EWJ 44590206 IC50 = 31 nM T99089 C3LZ6B 44593434 IC50 = 49 nM T99089 C7BX3O 44602984 IC50 = 80 nM T99089 C86VZL 44602985 IC50 = 67 nM T99089 C8KI5C 44603044 IC50 = 24000 nM T99089 C4M2KB 44654329 IC50 = 190 nM T99089 CGX7Q4 45267129 IC50 = 1450 nM T99089 C4GRT3 45267957 IC50 > 10000 nM T99089 C65XTQ 45267989 IC50 > 10000 nM T99089 C0DN8Q 45268879 IC50 = 7070 nM T99089 C3VI6H 45268883 IC50 = 170 nM T99089 CF17WS 45269730 IC50 = 160 nM T99089 CCZ72A 45271358 IC50 > 10000 nM T99089 C17RYH 45271371 IC50 = 410 nM T99089 C8L9ZU 45273140 IC50 = 270 nM T99089 CWI2D1 45375869 IC50 = 30 nM T99089 C2D6QS 45486182 IC50 < 2 nM T99089 C82YQR 45486184 IC50 = 9.1 nM T99089 CLMF90 45486187 IC50 = 3.8 nM T99089 C76ENX 45486190 IC50 < 0.3 nM T99089 CE1MZ4 45486203 IC50 = 302 nM T99089 CR6E9Y 45486205 IC50 = 22.8 nM T99089 C28GPA 45486206 IC50 = 39.4 nM T99089 CO81AX 45486208 IC50 = 151 nM T99089 C4V1FW 45486210 IC50 = 2.1 nM T99089 CPO7F8 45486211 IC50 = 4.9 nM T99089 C6EX1G 45486212 IC50 = 8.4 nM T99089 CDK4T2 45486218 IC50 = 57.9 nM T99089 COI1M7 45486219 IC50 = 36 nM T99089 CVJ34H 45486222 IC50 > 1000 nM T99089 CEQ4O7 45486223 IC50 = 6.4 nM T99089 CVK3E8 45486224 IC50 = 67 nM T99089 CB6L4I 45486225 IC50 = 6.7 nM T99089 CQ8J5U 45486226 IC50 = 75.9 nM T99089 C4UF0V 45503363 IC50 = 140 nM T99089 CYQ8B2 45503364 IC50 = 190 nM T99089 C32HLA 45503367 IC50 = 140 nM T99089 C2KZ8V 46196674 IC50 = 27 nM T99089 CV4GE7 46196675 IC50 = 70 nM T99089 CI84VY 46196676 IC50 = 75 nM T99089 CT1P2W 46196677 IC50 = 40 nM T99089 CG2AU5 46196996 IC50 = 62 nM T99089 C38BVC 46196997 IC50 = 122 nM T99089 CCL6H2 46196998 IC50 = 52 nM T99089 CF3GQ1 46196999 IC50 = 76 nM T99089 CO9ML6 46197110 IC50 = 70 nM T99089 CW3ZC7 46197111 IC50 = 2200 nM T99089 CXYD95 46197658 IC50 = 83 nM T99089 C61LOS 46197659 IC50 = 1190 nM T99089 C2U6BA 46197660 IC50 = 147 nM T99089 CRU91A 46197661 IC50 = 210 nM T99089 C1UN6H 46197662 IC50 = 104 nM T99089 C15SIF 46197769 IC50 = 28000 nM T99089 CV7B0P 46197770 IC50 = 124 nM T99089 C2C6OJ 46197771 IC50 = 140 nM T99089 CJB83Y 46197772 IC50 = 70000 nM T99089 CL5Q6E 46197773 IC50 = 620 nM T99089 CD1B2I 46197872 IC50 = 42 nM T99089 CCOB85 46197873 IC50 = 142 nM T99089 C5WPQ2 46197874 IC50 = 7800 nM T99089 COSG68 46197875 IC50 = 170 nM T99089 CC1OD0 46197876 IC50 = 84 nM T99089 C7S9KB 46197980 IC50 = 176 nM T99089 C4D1FE 46197981 IC50 = 143 nM T99089 CH5ZX1 46197982 IC50 = 164 nM T99089 CKD01G 46197983 IC50 = 830 nM T99089 C6Y7NW 46197984 IC50 = 90 nM T99089 CIJ2C6 46198095 IC50 = 2900 nM T99089 C3OJS6 46198096 IC50 = 130 nM T99089 CM37LV 46198097 IC50 = 54 nM T99089 C32EMV 46198098 IC50 = 36 nM T99089 C6FK0L 46198099 IC50 = 190 nM T99089 CS8P1X 46198205 IC50 = 240 nM T99089 C6OQH7 46198206 IC50 = 11 nM T99089 C2XF3D 46198207 IC50 = 510 nM T99089 COX8S7 46198208 IC50 = 14 nM T99089 C5CP2F 46198209 IC50 = 35 nM T99089 CQ1D4O 46198316 IC50 = 251 nM T99089 CGU80Q 46198317 IC50 = 100 nM T99089 CM58LS 46198318 IC50 = 383 nM T99089 CL7UY0 46198320 IC50 = 197 nM T99089 CBO87C 46198375 IC50 < 0.32 nM T99089 CUA97D 46209401 IC50 = 2 nM T99089 CMBJ68 46222580 IC50 = 26 nM T99089 C1GO2Y 46222581 IC50 = 360 nM T99089 CR2G0M 46228457 IC50 = 26 nM T99089 CRQ0V5 46228458 IC50 = 195 nM T99089 CIV52B 46228459 IC50 = 740 nM T99089 CCF60G 46228460 IC50 = 128 nM T99089 C2P9QO 46228508 IC50 = 89 nM T99089 CH8M7J 46228509 IC50 = 123 nM T99089 C2Q5RG 46228510 IC50 = 400 nM T99089 CUY82H 46228511 IC50 = 21300 nM T99089 CZ76CV 46228524 IC50 = 17800 nM T99089 CCF84Y 46228525 IC50 = 730 nM T99089 CW96RT 46228526 IC50 = 690 nM T99089 CCO78J 46228527 IC50 = 620 nM T99089 CQKD47 46228552 IC50 = 87000 nM T99089 C82CNS 46228553 IC50 = 94000 nM T99089 CXV41S 46228554 IC50 = 68000 nM T99089 C59GQX 46228555 IC50 = 42000 nM T99089 CJ1V9Y 46228556 IC50 = 14 nM T99089 C8J4GN 46228587 IC50 > 10000 nM T99089 CZR4K2 46228588 IC50 = 79000 nM T99089 CXE9G2 46228589 IC50 = 49 nM T99089 CK07MJ 46228590 IC50 = 6700 nM T99089 C9TW1K 46228617 IC50 = 15000 nM T99089 CJ0M5L 46228618 IC50 = 71 nM T99089 CZ7AI8 46228619 IC50 = 23 nM T99089 CG10QD 46228620 IC50 = 6480 nM T99089 CGE71D 46228640 IC50 = 17 nM T99089 C1BZ8D 46228641 IC50 = 40 nM T99089 C4IJ0T 46228642 IC50 = 57 nM T99089 CHS4I6 46228643 IC50 > 10000 nM T99089 CRX8M3 46228664 IC50 = 115 nM T99089 C94GNC 46228665 IC50 = 15400 nM T99089 CK9HB1 46228666 IC50 = 920 nM T99089 CN1SB2 46228667 IC50 > 100000 nM T99089 C6RNZ2 46228694 IC50 > 100000 nM T99089 CYJG41 46228695 IC50 = 22000 nM T99089 C9J3EO 46228696 IC50 > 100000 nM T99089 CLJ4Z0 46228697 IC50 = 93000 nM T99089 C1KG2A 46228728 IC50 = 1000 nM T99089 CVI1J2 46228729 IC50 = 79000 nM T99089 CKX81Z 46228730 IC50 = 92000 nM T99089 C7NFH5 46228731 IC50 > 100000 nM T99089 C8XB1I 46228766 IC50 = 38000 nM T99089 C3YT8B 46228767 IC50 = 13700 nM T99089 CPA46C 46228768 IC50 = 87 nM T99089 CH0ES4 46228769 IC50 = 48 nM T99089 C2B5ES 46228792 IC50 = 15 nM T99089 C0NP5I 46228793 IC50 = 23 nM T99089 C9NRH2 46228794 IC50 = 6800 nM T99089 COW38I 46228795 IC50 = 90 nM T99089 CR0EO8 46228796 IC50 = 4700 nM T99089 C1Z4XW 46228797 IC50 = 8000 nM T99089 CA4M3D 46228798 IC50 = 187 nM T99089 C8CX5F 46228818 IC50 > 100000 nM T99089 C9EMG4 46228819 IC50 = 57000 nM T99089 CCG2J8 46228820 IC50 > 100000 nM T99089 C8ZO7J 46228821 IC50 = 11300 nM T99089 C6E5PY 46228822 IC50 = 356 nM T99089 C07ZPY 46228823 IC50 = 590 nM T99089 COW7Q6 46228824 IC50 = 500 nM T99089 C6L0JY 46228825 IC50 > 10000 nM T99089 CLS64M 46228853 IC50 > 100000 nM T99089 CH82DK 46228854 IC50 = 1660 nM T99089 CH65DP 46228855 IC50 = 850 nM T99089 CJ85WB 46228856 IC50 = 124 nM T99089 CE60UA 46228857 IC50 > 100000 nM T99089 CC0AT1 46228858 IC50 > 10000 nM T99089 CAE8F0 46228859 IC50 > 10000 nM T99089 C5QU9B 46228860 IC50 = 240 nM T99089 CJZA13 46228900 IC50 = 15900 nM T99089 C8KNZ9 46228901 IC50 = 1560 nM T99089 CPY3I0 46228902 IC50 = 14000 nM T99089 CQ8V3N 46228903 IC50 = 25200 nM T99089 C3EBU0 46228904 IC50 > 100000 nM T99089 C68LVX 46228905 IC50 = 770 nM T99089 C5JZF2 46228906 IC50 = 33 nM T99089 CX0J3H 46228907 IC50 = 340 nM T99089 CZM90S 46228908 IC50 = 64 nM T99089 CJ9EI6 46228945 IC50 = 21100 nM T99089 C4F7IE 46228946 IC50 > 100000 nM T99089 C6N2SC 46228947 IC50 = 2750 nM T99089 C48RIK 46228948 IC50 = 1120 nM T99089 CI9WF8 46228949 IC50 = 33 nM T99089 CYP51A 46228950 IC50 = 6900 nM T99089 C3T8AM 46228951 IC50 = 7 nM T99089 CIM53K 46847263 IC50 = 1.7 nM T99089 C7H4YM 46865419 IC50 = 80 nM T99089 C4MKC5 46870033 IC50 = 17 nM T99089 CJMO86 46879449 IC50 = 0.51 nM T99089 C4KQ3H 46879450 IC50 = 0.5 nM T99089 CNH1L4 46879451 IC50 = 12 nM T99089 C8FC5Y 46879452 IC50 = 0.44 nM T99089 C6Z1XG 46879458 IC50 = 42 nM T99089 CIY3O5 46879459 IC50 = 98 nM T99089 C75CRZ 46879460 IC50 = 18 nM T99089 CT6QA4 46879461 IC50 = 30 nM T99089 CV03IY 46879517 IC50 = 8.7 nM T99089 CSO84N 46879518 IC50 = 8.2 nM T99089 CF1BT0 46879519 IC50 = 21 nM T99089 CBRS82 46879520 IC50 = 1 nM T99089 CK7LQ4 46879877 IC50 = 552 nM T99089 C79IHJ 46879959 IC50 = 842 nM T99089 C9XLF4 46879960 IC50 = 308 nM T99089 CQ25VN 46879961 IC50 > 10000 nM T99089 CZ6D2P 46880014 IC50 = 2 nM T99089 C09EYD 46880015 IC50 = 1.5 nM T99089 CMO47N 46880016 IC50 = 57 nM T99089 C2WA7P 46880017 IC50 = 139 nM T99089 CXTC97 46880018 IC50 = 34 nM T99089 C2DUH7 46880019 IC50 = 40 nM T99089 CGQ93K 46880020 IC50 = 318 nM T99089 CSD1Q7 46880021 IC50 = 41 nM T99089 C0G1KP 46880074 IC50 = 1 nM T99089 CB14IR 46880075 IC50 = 0.49 nM T99089 C5WD3A 46880076 IC50 < 0.32 nM T99089 C0F9VH 46880077 IC50 = 26 nM T99089 C6NGU8 46880078 IC50 = 117 nM T99089 CQT06S 46880079 IC50 = 44 nM T99089 CZYQ96 46880102 IC50 < 0.32 nM T99089 CI72BX 46880103 IC50 < 0.32 nM T99089 C7SK8G 46880104 IC50 < 0.32 nM T99089 CAFD60 46880105 IC50 = 20 nM T99089 COA93M 46880106 IC50 = 38 nM T99089 CF24RO 46880107 IC50 = 113 nM T99089 CJOM49 46880136 IC50 = 0.38 nM T99089 C7ZMV0 46880137 IC50 < 0.32 nM T99089 CQY7E2 46880138 IC50 < 0.32 nM T99089 C4V3UA 46880139 IC50 = 112 nM T99089 CHZL13 46880140 IC50 = 44 nM T99089 CL0W5N 46880141 IC50 = 941 nM T99089 CWL70U 46880217 IC50 < 0.32 nM T99089 C9AZE3 46880218 IC50 < 0.32 nM T99089 C4MT6A 46880225 IC50 = 84 nM T99089 CKXA51 46880226 IC50 = 393 nM T99089 C5YQC6 46880227 IC50 = 326 nM T99089 C0V6PO 46880228 IC50 = 362 nM T99089 C38CFM 46880229 IC50 = 219 nM T99089 C0NT9Z 46883533 IC50 > 10000 nM T99089 C1G4BN 46883535 IC50 > 10000 nM T99089 C12VIL 46883538 IC50 > 10000 nM T99089 CV28UF 46883539 IC50 = 100 nM T99089 CS4VH0 46883569 IC50 > 10000 nM T99089 C6M5GU 46883570 IC50 = 6200 nM T99089 CC1I3F 46883571 IC50 > 10000 nM T99089 C16TPN 46883708 IC50 = 1100 nM T99089 C3AVB1 46883709 IC50 = 4000 nM T99089 CZ8XB2 46883710 IC50 = 660 nM T99089 CMR2G9 46883711 IC50 = 60 nM T99089 CL0ZT3 46883714 IC50 = 25 nM T99089 CQ4X5O 46883715 IC50 = 40 nM T99089 C9EL2F 46883716 IC50 = 53 nM T99089 CG0VM7 46883717 IC50 = 160 nM T99089 C1N6OV 46883718 IC50 = 130 nM T99089 CZB28E 46883719 IC50 = 68 nM T99089 C4PS8I 46883720 IC50 = 110 nM T99089 CEH9Q2 46883721 IC50 = 110 nM T99089 C5PD6F 46883722 IC50 = 66 nM T99089 CPF9D2 46883723 IC50 = 66 nM T99089 CV42XD 46885361 IC50 > 10000 nM T99089 C9TME7 46885362 IC50 = 540 nM T99089 C0P7GZ 46885363 IC50 = 1110 nM T99089 CQ0ZK1 46885411 IC50 > 10000 nM T99089 C9XB7U 46885412 IC50 > 10000 nM T99089 CGYW52 46885477 IC50 > 10000 nM T99089 COJA32 46892971 IC50 = 1200 nM T99089 C7E9SF 46899944 IC50 = 17 nM T99089 C5T4OX 46899945 IC50 = 64 nM T99089 C4UG0X 46899948 IC50 = 258 nM T99089 CC0A1B 46900109 IC50 = 59 nM T99089 CPCD05 46900110 IC50 = 141 nM T99089 CJ5L9R 46900111 IC50 = 405 nM T99089 C20YBF 46900112 IC50 = 69 nM T99089 CVS9U2 46900113 IC50 = 42 nM T99089 CCBO60 46900264 IC50 = 17 nM T99089 C16LWK 46900265 IC50 = 25 nM T99089 C1I6HG 46900266 IC50 = 730 nM T99089 CP45QN 46900267 IC50 = 1670 nM T99089 CAOI74 46900268 IC50 = 1370 nM T99089 CFNK12 46900424 IC50 = 55 nM T99089 CK7T2S 46900425 IC50 = 58 nM T99089 C10CRA 46900426 IC50 = 87 nM T99089 C0Z9PF 46900427 IC50 = 69 nM T99089 CCV9L5 46900428 IC50 = 51 nM T99089 CQR3A5 46901756 IC50 = 5 nM T99089 CZ7M4V 46919120 IC50 = 180.1 nM T99089 C5WBZ7 46919121 IC50 < 1 nM T99089 CNL40R 46919122 IC50 = 413.9 nM T99089 CWGT04 46919517 IC50 = 9.1 nM T99089 CP59KI 46919518 IC50 = 15 nM T99089 C9E4YG 46919605 IC50 = 2 nM T99089 C9Z2QG 46919606 IC50 = 3 nM T99089 C9O0AN 46927521 EC50 = 9 nM T99089 C1L2PQ 46927522 EC50 = 4 nM T99089 C6OJA1 46927597 EC50 = 7 nM T99089 C9PAT7 46927672 IC50 = 3.8 nM T99089 CSOG58 46937280 IC50 = 240 nM T99089 C02IJE 46937281 IC50 = 230 nM T99089 C7LK1C 46945257 IC50 = 19500 nM T99089 CHX76J 49784892 IC50 > 1000 nM T99089 CA1H8S 49784893 IC50 > 1000 nM T99089 CTZG05 49784988 IC50 > 1000 nM T99089 CG2IO7 49785079 IC50 > 1000 nM T99089 CZI34V 49785167 IC50 > 1000 nM T99089 CJK65T 49785253 IC50 > 1000 nM T99089 C3NV0J 49785827 IC50 > 1000 nM T99089 C1AR4G 49785829 IC50 > 1000 nM T99089 CR9WA4 49836427 IC50 = 0.51 nM T99089 CX1ZO4 49836539 IC50 = 0.23 nM T99089 C7F8JO 49836540 IC50 < 0.1 nM T99089 C0X2FY 49836541 IC50 < 0.32 nM T99089 C82UYD 49836542 IC50 = 1.4 nM T99089 CL1CV3 49836646 IC50 = 7.3 nM T99089 C9V1JH 49836647 IC50 = 1.9 nM T99089 C1G8OB 49836648 IC50 = 2 nM T99089 CU3KH0 49836649 IC50 = 1 nM T99089 CWTL58 49836748 IC50 = 0.61 nM T99089 CJX81B 49836749 IC50 = 0.38 nM T99089 CDXE39 49836750 IC50 = 9.6 nM T99089 COYU08 49836854 IC50 = 0.35 nM T99089 C2RO1T 49836856 IC50 = 61 nM T99089 CFX3P6 49836857 IC50 = 0.5 nM T99089 C5R6HU 49836964 IC50 < 0.32 nM T99089 CXW48M 49836965 IC50 < 0.1 nM T99089 CO3K1E 49836966 IC50 = 0.11 nM T99089 C1AZW5 49836968 IC50 = 0.71 nM T99089 CTC01J 49837087 IC50 = 0.41 nM T99089 CD1XZ0 49837088 IC50 = 10 nM T99089 CGO4Q1 49837089 IC50 = 1.2 nM T99089 CUM13L 49837090 IC50 = 0.52 nM T99089 C5H0XP 49837198 IC50 = 0.77 nM T99089 CGO6B2 49837300 IC50 < 0.32 nM T99089 CTH0Z6 49837301 IC50 < 0.32 nM T99089 CNA43S 49837401 IC50 < 0.32 nM T99089 CSI9D6 49837402 IC50 < 0.32 nM T99089 CN89TG 49840317 IC50 > 15000 nM T99089 CY48DE 49849970 IC50 = 1.4 nM T99089 CUS56N 49863686 IC50 > 100000 nM T99089 CIU7C1 49863687 IC50 > 100000 nM T99089 CHL4D9 49863710 IC50 > 100000 nM T99089 CUCO48 49863711 IC50 = 92.3 nM T99089 CCPS95 49863903 IC50 = 54 nM T99089 CZIR49 49863968 IC50 = 6600 nM T99089 CMJ70C 50912930 IC50 = 0.54 nM T99089 CS7J8G 50937465 IC50 = 2.9 nM T99089 C36LQJ 50940491 IC50 = 4 nM T99089 C2Q0GE 50990922 IC50 = 3 nM T99089 CT7UB5 50990960 IC50 = 7 nM T99089 C61DVY 50990961 IC50 = 2.7 nM T99089 CV3UP9 50992247 IC50 = 2.1 nM T99089 CSW27B 50994972 IC50 = 374 nM T99089 CYNX05 50994975 IC50 = 129 nM T99089 C4XV7W 50994976 IC50 = 174 nM T99089 CE73LF 50994977 IC50 = 190 nM T99089 C53WVZ 50995007 IC50 = 83.18 nM T99089 C8OWU5 50995160 IC50 = 367 nM T99089 CZ4B5Q 50995530 IC50 = 0.9 nM T99089 CMR62F 50995532 IC50 = 1.096 nM T99089 CD7KN6 50995705 EC50 = 2.6 nM T99089 CRJL51 50995706 IC50 = 5.6 nM T99089 CRB3V5 50995710 IC50 = 3.2 nM T99089 C59ESV 50996310 IC50 = 1.8 nM T99089 CL7FA8 50997340 IC50 = 36 nM T99089 C63VKR 50997526 IC50 = 141.25 nM T99089 CWN50H 50997675 IC50 = 43 nM T99089 CLIK35 50997676 IC50 = 247 nM T99089 CBQU14 50997677 IC50 = 299 nM T99089 COC1I5 50997678 IC50 = 228 nM T99089 CTMF09 50997679 IC50 = 128 nM T99089 CWN54R 51003389 IC50 = 4.2 nM T99089 C5OUV8 51003390 IC50 = 240 nM T99089 C5X9OM 51354603 IC50 = 61 nM T99089 C4DSG2 51354885 IC50 = 8 nM T99089 CQ85FC 51354886 IC50 = 3.3 nM T99089 C7MOQ0 51354887 IC50 = 2.9 nM T99089 C5KVT1 51355181 IC50 = 5 nM T99089 CS5F4Z 51355182 IC50 = 6 nM T99089 C4NFL7 51355183 IC50 = 4 nM T99089 C4W6PY 51355459 IC50 = 5 nM T99089 C95FWU 51355461 IC50 = 2.2 nM T99089 C4J3RE 51355733 IC50 = 7 nM T99089 C7LO2Y 52932687 IC50 = 630 nM T99089 C6DKQ4 52932689 IC50 = 100 nM T99089 C87LMF 52932691 IC50 = 32000 nM T99089 CNW01S 52932692 IC50 = 1300 nM T99089 C7XI4R 52932914 IC50 = 160 nM T99089 C8FBT0 52932915 IC50 = 800 nM T99089 CBVW62 52932917 IC50 = 2500 nM T99089 C7XVM5 52933152 IC50 = 1000 nM T99089 C1L6UP 52933587 IC50 = 40 nM T99089 CG04VW 52933647 IC50 = 79 nM T99089 C4L8GI 52934106 IC50 = 50 nM T99089 C9UYP8 52934570 IC50 = 130 nM T99089 CE8L9U 52934573 IC50 = 1000 nM T99089 CL16MA 52934795 IC50 = 400 nM T99089 C91KNR 52934796 IC50 = 250 nM T99089 CQ2ET7 52935028 IC50 = 10000 nM T99089 CJ1E7O 52935890 IC50 = 79 nM T99089 CD1XK2 52936114 IC50 = 1000 nM T99089 CK12ZP 52936117 IC50 = 4000 nM T99089 C4DLK1 52941323 IC50 = 4400 nM T99089 C02RNH 52941410 IC50 = 730 nM T99089 CKWC23 52942546 IC50 = 1330 nM T99089 CVE49F 52943666 IC50 > 10000 nM T99089 CI4Z7O 52943694 IC50 = 1710 nM T99089 C43TJA 52944042 IC50 = 970 nM T99089 C9MV6T 52945093 IC50 > 10000 nM T99089 CD9G0Y 52945288 IC50 = 1200 nM T99089 CG0BA4 52946221 IC50 = 740 nM T99089 CN8X0H 52947491 IC50 = 840 nM T99089 CDV8T6 52948574 IC50 = 3700 nM T99089 CWY5V9 52948575 IC50 = 1840 nM T99089 CUZ65L 52948582 IC50 > 10000 nM T99089 C4Q9IX 52948946 IC50 = 1600 nM T99089 CQ6IB5 52949635 IC50 = 1.2 nM T99089 CPM59C 52950212 IC50 = 1.4 nM T99089 C1SKV3 53249125 EC50 = 2100 nM T99089 CFRH86 53302367 IC50 = 1.6 nM T99089 CEZ7P6 53313343 IC50 = 1.6 nM T99089 CNKP63 53316555 IC50 = 1400 nM T99089 CN3Y4C 53316581 IC50 = 5 nM T99089 CDX1O6 53316582 IC50 = 2 nM T99089 C65DAZ 53316583 IC50 < 2 nM T99089 C3LTA4 53317522 IC50 = 93 nM T99089 C87OAQ 53317986 IC50 = 0.8 nM T99089 CE1V5K 53319219 IC50 = 3 nM T99089 CM0N2P 53319337 IC50 = 5.2 nM T99089 C7XI0Q 53319338 IC50 = 179 nM T99089 C1L8WR 53319339 IC50 = 2.4 nM T99089 CFN2J5 53320305 IC50 = 5800 nM T99089 CIOP36 53320502 IC50 = 1200 nM T99089 CC2IW7 53320600 IC50 = 4.3 nM T99089 CN1TI4 53320630 IC50 = 38 nM T99089 CZN0B8 53320631 IC50 = 0.3 nM T99089 CMQI43 53321817 IC50 = 570 nM T99089 CW7B3H 53321844 IC50 = 1500 nM T99089 C92UFO 53321929 IC50 = 5 nM T99089 CY0V2M 53323287 IC50 = 14 nM T99089 C4HKE1 53323288 IC50 = 5.7 nM T99089 CA4T3Y 53323289 IC50 = 2.7 nM T99089 CNW02P 53323290 IC50 = 0.8 nM T99089 CP41WD 53324073 IC50 = 4 nM T99089 CJ4G3Y 53324074 IC50 = 2 nM T99089 C62GPL 53324318 IC50 = 8200 nM T99089 CL4G1V 53324616 IC50 = 30 nM T99089 CNO54Z 53324617 IC50 = 2.3 nM T99089 CFP84X 53324920 IC50 = 3.2 nM T99089 CBY49I 53325802 IC50 = 32 nM T99089 CD9O2F 53325830 IC50 < 2 nM T99089 C1EXW0 53325922 IC50 = 2 nM T99089 C2JB0Z 53325923 IC50 = 1.6 nM T99089 CCK30V 53379548 IC50 = 2490 nM T99089 C48TNF 53379553 IC50 = 59110 nM T99089 CCTS15 53380119 IC50 = 9070 nM T99089 CGVD50 53380120 IC50 = 13540 nM T99089 C5S1UJ 53380121 IC50 = 3760 nM T99089 CHK92L 53380218 IC50 = 22650 nM T99089 CF7U6Q 53380219 IC50 = 45090 nM T99089 CD19RY 53380221 IC50 = 28510 nM T99089 C4SWC9 53380318 IC50 = 21990 nM T99089 CZ3OU5 53380319 IC50 = 20500 nM T99089 CF9JU3 53380320 IC50 = 91550 nM T99089 CK21TC 53380322 IC50 = 1620 nM T99089 CC1D5H 53380323 IC50 = 2810 nM T99089 C4GB3K 53380324 IC50 = 8890 nM T99089 CVG90B 53389651 IC50 > 10000 nM T99089 C3HMP1 53484099 IC50 = 8.6 nM T99089 CTGC73 54580078 IC50 = 3800 nM T99089 CL5Q6F 54580136 IC50 = 8 nM T99089 CQOT43 54580519 IC50 = 7 nM T99089 C89YCL 54580728 EC50 = 1000 nM T99089 CA9I0J 54580729 EC50 = 3700 nM T99089 CCJ4O1 54580890 IC50 = 3 nM T99089 C95MIN 54580891 IC50 = 4 nM T99089 CEL5N4 54580892 IC50 = 4 nM T99089 C9GWT2 54581065 IC50 = 660 nM T99089 CNQ0K4 54581121 IC50 = 410 nM T99089 C3S5AM 54581683 IC50 > 1000 nM T99089 CT8XP5 54581685 IC50 > 1000 nM T99089 C4X6DP 54581730 EC50 = 10000 nM T99089 C2KHN1 54581731 EC50 = 2900 nM T99089 CUDL04 54581778 IC50 = 37 nM T99089 CMZH76 54581779 IC50 = 3 nM T99089 CGL63B 54581944 IC50 = 5 nM T99089 C8MG6Q 54581945 IC50 = 670 nM T99089 CWQ62A 54582154 IC50 = 37.9 nM T99089 C7E8XC 54582155 IC50 = 8.1 nM T99089 CYJ3V4 54582156 IC50 = 10.7 nM T99089 C1V9TZ 54582157 IC50 = 350 nM T99089 CS87QB 54582674 IC50 = 647 nM T99089 CKV3C4 54582675 IC50 = 861 nM T99089 CS0PL6 54582676 IC50 = 0.66 nM T99089 CO87VE 54582742 IC50 = 8 nM T99089 CL7P3T 54582868 IC50 = 180 nM T99089 CAWE03 54582869 IC50 = 6 nM T99089 CBTW13 54583042 IC50 = 130 nM T99089 CO6B0E 54583043 IC50 = 7.9 nM T99089 CZRH05 54583044 IC50 = 2400 nM T99089 C6HCS1 54583107 IC50 = 970 nM T99089 CD4I8V 54583108 IC50 = 920 nM T99089 CDJ6G8 54583634 IC50 = 468 nM T99089 C4ZR2K 54583635 IC50 > 1000 nM T99089 C8ZRQ6 54583636 IC50 = 8 nM T99089 C2LUN7 54583637 IC50 = 0.57 nM T99089 CYU57L 54583878 IC50 = 799 nM T99089 C6K2HE 54584047 IC50 > 10000 nM T99089 CH9XG2 54584103 IC50 = 8 nM T99089 CV3E2I 54584104 IC50 = 600 nM T99089 CASX62 54584105 IC50 = 140 nM T99089 CSTH09 54584106 IC50 = 2000 nM T99089 C9ZC3U 54584611 IC50 > 1000 nM T99089 CK2Q9W 54584612 IC50 = 3.8 nM T99089 CD4B5P 54584613 IC50 = 3.2 nM T99089 CP7U4T 54584640 EC50 = 1000 nM T99089 CKFC13 54584711 IC50 = 3 nM T99089 CU8NQ4 54584712 IC50 = 21 nM T99089 C1O4MD 54584830 IC50 = 7 nM T99089 CD73TV 54584831 IC50 = 10 nM T99089 CE5B2W 54584832 IC50 = 4 nM T99089 C1XJW8 54584998 IC50 > 10000 nM T99089 CJ58MO 54584999 IC50 > 10000 nM T99089 C92ZHV 54585000 IC50 > 10000 nM T99089 C6Q8OC 54585001 IC50 = 110 nM T99089 C87OYZ 54585557 IC50 = 1540 nM T99089 C3BGY8 54585558 IC50 = 72.5 nM T99089 C0OY2N 54585559 IC50 = 4.6 nM T99089 CBUK26 54585560 IC50 = 1.25 nM T99089 C1D2OF 54585666 IC50 = 3 nM T99089 CLA1K6 54585957 IC50 > 10000 nM T99089 C3PGE2 54585958 IC50 = 25.7 nM T99089 CV7HJ8 54585959 IC50 = 2000 nM T99089 C2J4AW 54586018 IC50 = 450 nM T99089 CE18QV 54586536 IC50 = 23 nM T99089 C9LYS4 54586537 IC50 = 788 nM T99089 CZ9VQ3 54586538 IC50 = 3.7 nM T99089 CU0WR1 54586539 IC50 = 607 nM T99089 C5ITJ1 54586540 IC50 = 4.9 nM T99089 C7QWJ6 54586541 IC50 = 5 nM T99089 CFE96Y 54586652 IC50 = 3 nM T99089 CKI74Z 54586653 IC50 = 3 nM T99089 CJI6G8 54586767 IC50 = 5 nM T99089 CM31XW 54586768 IC50 = 5 nM T99089 CA4WF9 54586933 IC50 = 83 nM T99089 C0P7RF 54587401 IC50 = 13 nM T99089 CTB8J1 54587402 IC50 = 3 nM T99089 C6JVP8 54587568 IC50 > 1000 nM T99089 CQK04T 54587569 IC50 = 55 nM T99089 CRB13M 54587570 IC50 = 328 nM T99089 CS21RZ 54587660 IC50 = 7 nM T99089 CNB28I 54675261 IC50 = 32 nM T99089 CU9NY2 54675336 IC50 = 1.3 nM T99089 C6SW5P 54675374 IC50 = 0.2 nM T99089 CO6EN5 54675413 IC50 = 10 nM T99089 C6KE7Z 54675418 IC50 = 40 nM T99089 CLZ53I 54675419 IC50 = 6.3 nM T99089 C9SXQ0 54675442 IC50 = 8 nM T99089 C10VXC 54675444 IC50 = 79 nM T99089 CG35NE 54675446 IC50 = 16 nM T99089 CV6X5K 54675470 IC50 = 32 nM T99089 C4OZC7 54675473 IC50 = 1.3 nM T99089 C3YZ9F 54675501 IC50 = 0.6 nM T99089 C9YKJ7 54764764 IC50 = 8 nM T99089 CKV76W 54764765 IC50 = 10 nM T99089 CYFP20 54764766 IC50 = 6 nM T99089 CETW26 54764767 IC50 = 17 nM T99089 CEJR67 54764768 IC50 = 8 nM T99089 CY0TN4 56658293 IC50 = 2600 nM T99089 C6BE9H 56658294 IC50 = 530 nM T99089 CCY5N4 56658295 IC50 = 38 nM T99089 CP1W9R 56658296 IC50 = 18 nM T99089 CU36FV 56658297 IC50 = 29 nM T99089 C04BHC 56658298 IC50 = 38 nM T99089 CN8XD6 56658305 IC50 = 36 nM T99089 CLE4Y5 56658307 IC50 = 173 nM T99089 C4MJ5O 56658311 IC50 = 12 nM T99089 C7NP3M 56658312 IC50 = 1.8 nM T99089 CN4J9K 56658587 IC50 = 82 nM T99089 CH7Q4P 56659673 EC50 = 10 nM T99089 CN4U5R 56659674 EC50 = 8 nM T99089 C7I9AJ 56659836 EC50 = 7 nM T99089 CP2KY0 56661794 IC50 = 110 nM T99089 CN01KB 56661795 IC50 = 17 nM T99089 CJTU92 56661796 IC50 = 18 nM T99089 CBI7G3 56661797 IC50 = 19 nM T99089 CX62TD 56661798 IC50 = 200 nM T99089 CXE20W 56661799 IC50 = 400 nM T99089 CZ5XD1 56661804 IC50 = 80 nM T99089 C5XU3W 56661805 IC50 = 59 nM T99089 C6N0EJ 56661815 IC50 = 5.3 nM T99089 C91EDC 56661816 IC50 = 16 nM T99089 CG01XH 56662039 IC50 = 118 nM T99089 CFG9E7 56662196 IC50 = 113 nM T99089 C6RL1P 56663136 EC50 = 24 nM T99089 CBR9N7 56663302 IC50 = 9 nM T99089 CU0AC8 56663303 EC50 = 580 nM T99089 C2YO4N 56665241 IC50 = 61 nM T99089 C1DJ0Y 56665242 IC50 = 76 nM T99089 CE13AF 56665248 IC50 = 113 nM T99089 CJ85KT 56665256 IC50 = 4.2 nM T99089 C6VLY7 56665257 IC50 = 6.9 nM T99089 C4FD9N 56665258 IC50 = 0.5 nM T99089 C4RH8B 56665517 IC50 = 696 nM T99089 CKO56E 56668698 IC50 = 62 nM T99089 CJS5R1 56668699 IC50 = 100 nM T99089 CP0H1C 56668709 IC50 = 320 nM T99089 C7VMK6 56668710 IC50 = 0.2 nM T99089 C3C5MB 56668951 IC50 = 179 nM T99089 CH7G4I 56670002 IC50 = 1358 nM T99089 CQ1RX6 56670003 EC50 = 10 nM T99089 C8JY6A 56670156 EC50 = 52 nM T99089 CHFG31 56672169 IC50 = 150 nM T99089 CY8P0Z 56672170 IC50 = 29 nM T99089 CO65KN 56672171 IC50 = 120 nM T99089 CH37GX 56672177 IC50 = 96 nM T99089 C3BTJ1 56672436 IC50 = 290 nM T99089 CZXV87 56673516 EC50 = 11 nM T99089 C7YKI3 56673668 IC50 = 12 nM T99089 CC7T2A 56674921 IC50 = 190 nM T99089 CNF2C9 56675551 IC50 = 8.3 nM T99089 CA4RH3 56675552 IC50 = 170 nM T99089 CFU28L 56675553 IC50 = 25 nM T99089 C2JA0L 56675554 IC50 = 4.5 nM T99089 CGKN93 56675555 IC50 = 190 nM T99089 CRL0J4 56675556 IC50 = 40 nM T99089 CCAN48 56675557 IC50 = 140 nM T99089 CI17LQ 56675558 IC50 = 99 nM T99089 C31OWJ 56675570 IC50 = 46 nM T99089 C4CVI6 56675571 IC50 = 0.7 nM T99089 C4IR8B 56675821 IC50 = 1850 nM T99089 CO0U8T 56675936 IC50 = 229 nM T99089 CWB68U 56676987 IC50 = 5 nM T99089 CQK28C 56678886 IC50 = 110 nM T99089 C4ZX6A 56678887 IC50 = 13 nM T99089 C4FK3H 56678889 IC50 = 86 nM T99089 CJ47GL 56678899 IC50 = 1 nM T99089 CZ48XY 56679129 IC50 = 1664 nM T99089 C9NC2S 56680317 EC50 = 99 nM T99089 C8X0SE 56680318 IC50 = 1970 nM T99089 CM2H0R 56682202 IC50 = 1.4 nM T99089 C8SXR2 56682203 IC50 = 19 nM T99089 C64BDP 56682204 IC50 = 63 nM T99089 C5IQR3 56682205 IC50 = 33 nM T99089 CT1J5E 56682215 IC50 = 3.5 nM T99089 CQIS53 56682425 IC50 = 333 nM T99089 CH89ZU 56682426 IC50 = 10000 nM T99089 C19PCK 56683489 EC50 = 21 nM T99089 CV6GM9 56695913 IC50 = 1840 nM T99089 C1L5QU 56834881 IC50 = 58 nM T99089 CGEV72 56834882 IC50 = 2 nM T99089 C87YOZ 56929808 EC50 = 230 nM T99089 CGQ94I 56950740 IC50 > 100000 nM T99089 CN1XL0 56950741 IC50 > 100000 nM T99089 C3ER0V 56950742 IC50 = 64000 nM T99089 CEZ14X 56950743 IC50 > 100000 nM T99089 CTL49B 56950878 IC50 > 100000 nM T99089 CM5HO1 56950881 IC50 = 900 nM T99089 C9CLJ0 56950882 IC50 = 800 nM T99089 CG0VC7 56950883 IC50 = 860 nM T99089 CE1GO5 56950884 IC50 = 1400 nM T99089 CLQ4Z9 56950885 IC50 = 890 nM T99089 C40BPN 56951005 IC50 = 1700 nM T99089 CL9XP2 56951006 IC50 = 1500 nM T99089 CKV5O2 56951007 IC50 = 2500 nM T99089 C97QIR 56951008 IC50 = 2700 nM T99089 C61LYC 56951317 IC50 = 0.6 nM T99089 CB5V2D 56953628 IC50 = 101 nM T99089 C1A9IE 56953629 IC50 = 336 nM T99089 C48UTY 56953737 IC50 > 15000 nM T99089 CSPK46 56953738 IC50 = 355 nM T99089 C1ITV4 56953739 IC50 = 134 nM T99089 CO38GU 56953869 IC50 = 956 nM T99089 CS12TI 56953870 IC50 = 1134 nM T99089 CA2K6G 56953871 IC50 > 15000 nM T99089 CGBF17 56953872 IC50 = 649 nM T99089 C1ZQG0 56953873 IC50 = 324 nM T99089 CB83NX 56953992 IC50 = 645 nM T99089 CN7P1B 56953993 IC50 = 339 nM T99089 CI47JS 56953994 IC50 = 174 nM T99089 CIQJ93 56953995 IC50 = 308 nM T99089 C8DVS5 56953996 IC50 = 276 nM T99089 CL6W0K 56954119 IC50 = 109 nM T99089 CC31UP 56954120 IC50 = 183 nM T99089 C3BW5T 56954121 IC50 = 142 nM T99089 CKIC60 56954122 IC50 = 469 nM T99089 CN2L0O 56954123 IC50 = 84 nM T99089 CNH3A5 56954221 IC50 = 505 nM T99089 CE4YV5 56954222 IC50 = 681 nM T99089 CT95JA 56954223 IC50 > 1667 nM T99089 C73ZPH 56954224 IC50 = 21 nM T99089 C2ONU1 56954225 IC50 = 62 nM T99089 CL1IA3 56954309 IC50 = 1131 nM T99089 CNQ2G0 56955962 IC50 = 7 nM T99089 C7SJC2 56956247 IC50 = 3.02 nM T99089 C1FY0P 56965341 IC50 = 1 nM T99089 C01OBF 57342892 IC50 = 3400 nM T99089 CIWA26 57343054 IC50 = 9.5 nM T99089 CEOI16 57343055 IC50 = 0.1096 nM T99089 C4G7QD 57343225 IC50 = 0.18 nM T99089 C5DXS3 57343766 IC50 = 17 nM T99089 C32MLB 57343972 IC50 = 19 nM T99089 C8Q9ML 57344791 IC50 = 45 nM T99089 C89XBT 57344794 IC50 = 1 nM T99089 CT6H9M 57344795 IC50 = 9 nM T99089 C2WFQ3 57344993 IC50 = 18 nM T99089 CH71KO 57345095 IC50 = 41 nM T99089 C5YB9H 57345097 IC50 = 62 nM T99089 C3FY9A 57345328 IC50 = 1 nM T99089 CW9X3F 57386061 IC50 = 43 nM T99089 C8FS6P 57390778 IC50 = 15400 nM T99089 C13LDJ 57390779 IC50 = 2450 nM T99089 C3F0BW 57390780 IC50 = 38 nM T99089 CHY5D4 57390781 IC50 = 3 nM T99089 CC6ZD0 57390813 IC50 = 4 nM T99089 CB7KU9 57390814 IC50 = 1600 nM T99089 C82VXN 57391632 IC50 = 1780 nM T99089 CHI6C9 57392569 IC50 = 660 nM T99089 C4TXW2 57392593 IC50 = 3 nM T99089 CM8CB4 57392634 IC50 = 1210 nM T99089 CCP74G 57392635 IC50 = 212 nM T99089 CX2A5Y 57392636 IC50 = 1330 nM T99089 C7QGI8 57393255 IC50 = 290 nM T99089 CO0C5I 57394104 IC50 = 25000 nM T99089 CKVG97 57394105 IC50 = 26 nM T99089 CD2P1K 57394289 IC50 = 70 nM T99089 CDBV60 57394290 IC50 = 1 nM T99089 C1DAU4 57394291 IC50 = 390 nM T99089 CA75YZ 57394913 IC50 = 33.9 nM T99089 C8ZTY5 57394914 IC50 = 45.7 nM T99089 C0IJ9K 57394998 IC50 = 349 nM T99089 CKDR51 57395014 IC50 = 6.3 nM T99089 C13PQB 57395380 IC50 = 33 nM T99089 CO4WY9 57396045 IC50 = 180 nM T99089 C7EOQ2 57396104 IC50 = 67 nM T99089 CB1C3G 57396105 IC50 = 112 nM T99089 CE1VH5 57396728 IC50 = 1680 nM T99089 CO4QP1 57397207 IC50 = 2 nM T99089 CT4MN6 57397844 IC50 = 5300 nM T99089 C4J6UZ 57397845 IC50 = 45 nM T99089 C2JWM3 57397846 IC50 = 640 nM T99089 C8EM4N 57397875 IC50 = 28 nM T99089 CB47HC 57397876 IC50 = 40 nM T99089 CAN16F 57397919 IC50 = 14500 nM T99089 CZ1F9G 57397920 IC50 = 724 nM T99089 CT7D3Y 57398497 IC50 = 117 nM T99089 CN28HT 57398498 IC50 = 35 nM T99089 CM0C2E 57398516 IC50 = 35 nM T99089 C0BGR6 57399335 IC50 = 3 nM T99089 CS10GU 57399339 IC50 = 8600 nM T99089 CC04QG 57399505 IC50 = 2200 nM T99089 CVX1I4 57399506 IC50 = 600 nM T99089 C7DJ9Q 57399527 IC50 = 17 nM T99089 CPS08J 57399528 IC50 = 5 nM T99089 CVKR29 57399561 IC50 = 1540 nM T99089 C25ULW 57399562 IC50 = 5 nM T99089 CP0AL9 57399563 IC50 = 4 nM T99089 C1G6VF 57400171 IC50 = 18 nM T99089 CU4E6C 57400186 IC50 = 297 nM T99089 C7TAI9 57400292 IC50 = 1230 nM T99089 CJ7Y2K 57400603 IC50 = 2.2 nM T99089 CO63XJ 57401264 IC50 = 1300 nM T99089 C7BSY8 57401314 IC50 = 507 nM T99089 C3QEI9 57401315 IC50 = 275 nM T99089 C1IJV5 57401316 IC50 = 50 nM T99089 COZ7Q8 57401317 IC50 = 1120 nM T99089 C5UOF8 57401958 IC50 = 296 nM T99089 C0C6PE 57401959 IC50 = 293 nM T99089 CNVO29 57402060 IC50 = 3900 nM T99089 CX5O1I 57402078 IC50 = 1370 nM T99089 C6N8AU 57402861 IC50 = 1300 nM T99089 CL7MW8 57403007 IC50 = 150 nM T99089 CQH79M 57403036 IC50 = 4730 nM T99089 CA4L2E 57403037 IC50 = 14 nM T99089 CRJ9Q6 57403038 IC50 = 1 nM T99089 C2GYT1 57403706 IC50 > 10000 nM T99089 CB45FY 57403707 IC50 = 3470 nM T99089 C3R0XQ 57403708 IC50 = 3770 nM T99089 COQ75N 57403736 IC50 = 19 nM T99089 CA47JG 57433668 IC50 = 23 nM T99089 CE59QS 57505507 IC50 > 1000 nM T99089 C8P6RD 57505528 IC50 = 290 nM T99089 C4T7PW 57523998 IC50 = 31 nM T99089 C1Q7LS 57523999 IC50 = 195 nM T99089 CPS79I 57524088 IC50 = 54 nM T99089 C0CJ8Z 57524184 IC50 = 42 nM T99089 C8ICV2 57524400 IC50 = 58 nM T99089 CL72NQ 57524403 IC50 = 13 nM T99089 CAU0K1 57524478 IC50 = 53 nM T99089 C5FYG0 57568454 IC50 = 9 nM T99089 CN41VS 57568471 IC50 = 0.4 nM T99089 C5W4AZ 57568472 IC50 = 20 nM T99089 CE34TF 57568477 IC50 = 4 nM T99089 C6WMQ8 57568487 EC50 = 100 nM T99089 CW9L6C 57568544 IC50 = 1 nM T99089 CV1UP2 57568562 EC50 = 100 nM T99089 CK3NU1 57568594 IC50 < 0.4 nM T99089 CSA80G 57568606 IC50 = 10 nM T99089 CMR7A9 57568636 IC50 = 4 nM T99089 C6L9JH 57568638 EC50 = 400 nM T99089 C9AS4Q 57568659 IC50 < 0.4 nM T99089 CRF8M0 57708566 IC50 = 650 nM T99089 C4CJG6 57856282 IC50 = 6.5 nM T99089 CO1SN5 57989641 IC50 = 0.3 nM T99089 CJSR42 57989722 IC50 = 7 nM T99089 C61YOS 57989790 IC50 = 51 nM T99089 CHS76K 57989798 IC50 = 536 nM T99089 C9TN8I 57989818 IC50 = 28 nM T99089 C0FW7J 57989820 IC50 = 39.81 nM T99089 CR5IO7 57989894 IC50 = 1 nM T99089 CY5AF4 57989971 IC50 = 13 nM T99089 C1OV8I 57990029 IC50 = 10.96 nM T99089 CUPG23 57990033 IC50 = 28 nM T99089 C6BPR2 58985201 IC50 > 30000 nM T99089 CXT56U 59454465 IC50 = 170 nM T99089 CZ24KM 59454479 IC50 = 12 nM T99089 C5GV2P 59454483 IC50 = 13 nM T99089 C7N3LA 59454484 IC50 = 25 nM T99089 CCH48T 59454492 IC50 = 290 nM T99089 C8DT3V 59454506 IC50 = 18 nM T99089 C2BGR6 59506918 IC50 = 91 nM T99089 C0KZ6L 59507002 IC50 = 150 nM T99089 C6EJ9G 59507062 IC50 = 51 nM T99089 CHQK85 59507068 IC50 = 73 nM T99089 C8W5HT 59548263 IC50 > 1000 nM T99089 CVF1B2 59548283 IC50 > 1000 nM T99089 CC8UV3 59548383 IC50 > 1000 nM T99089 CD4ET2 59548402 IC50 > 1000 nM T99089 CES59T 59548403 IC50 > 1000 nM T99089 CBT21W 59548454 IC50 > 1000 nM T99089 CX8C2U 59548480 IC50 > 1000 nM T99089 CXJ63M 59603829 IC50 = 1500 nM T99089 CQEU96 59603842 IC50 = 19 nM T99089 CLH49Z 59790029 IC50 = 3 nM T99089 CW2GE7 59790182 EC50 = 100 nM T99089 C67DXJ 59823451 IC50 = 21.4 nM T99089 CN45KF 59823454 IC50 = 30.9 nM T99089 CZ2N7J 59823457 IC50 > 10000 nM T99089 CL4M6J 59823458 IC50 = 16.6 nM T99089 C8T6GZ 59823460 IC50 = 13.8 nM T99089 C27JOC 59823461 IC50 = 20.9 nM T99089 CGT41K 59823462 IC50 = 25.1 nM T99089 C5SC3K 59823463 IC50 = 19.5 nM T99089 C0K7JN 59823464 IC50 = 692 nM T99089 CNH9C6 59823465 IC50 = 9.6 nM T99089 C9QRX3 60098131 IC50 = 90 nM T99089 C9W0PE 60150671 IC50 = 570 nM T99089 C9NAL6 60152613 IC50 = 0.4 nM T99089 C5KD3Z 60154714 IC50 > 1000 nM T99089 CN0D8O 60154913 IC50 = 120 nM T99089 C9E6ZO 60154914 IC50 = 190 nM T99089 CS0L4D 60154996 IC50 > 1000 nM T99089 C59MPL 60154998 IC50 = 1600 nM T99089 CCO8H2 60154999 IC50 = 720 nM T99089 C1Z8VW 60155000 IC50 = 3600 nM T99089 C40TDP 60155001 IC50 = 520 nM T99089 C1UI3P 60155086 IC50 > 1000 nM T99089 C0DM1I 60165270 IC50 = 12 nM T99089 C46RPN 60196912 IC50 = 19 nM T99089 C52PMH 60196913 IC50 = 62 nM T99089 CTB23Y 60196914 IC50 = 2 nM T99089 C2Y9QK 60196916 IC50 = 8 nM T99089 CL90JM 60196917 IC50 = 814 nM T99089 C7FL4M 60197009 IC50 = 733 nM T99089 CD9ST6 60197011 IC50 = 18 nM T99089 C0Y2GI 60197014 IC50 = 17 nM T99089 C46JDT 60197113 IC50 = 11 nM T99089 CU69TF 60197114 IC50 = 100 nM T99089 CVB04X 60197118 IC50 = 44 nM T99089 C8IYB5 60197208 IC50 = 33 nM T99089 C8QY3Z 60197213 IC50 = 0.2 nM T99089 CF72YM 60197214 IC50 = 0.3 nM T99089 C5AUZ3 60197314 IC50 = 0.2 nM T99089 C8X4BC 60197315 IC50 = 0.2 nM T99089 CJBW03 60197316 IC50 = 0.3 nM T99089 C37IKA 60197416 IC50 = 3 nM T99089 CX2N4J 60197515 IC50 = 851 nM T99089 CP2YO9 60197609 IC50 = 603 nM T99089 CO32KC 60197610 IC50 = 110 nM T99089 CU93PB 66554192 IC50 = 300 nM T99089 CZ7Y1D 66563698 IC50 = 180 nM T99089 CCX0O1 66868153 IC50 = 239 nM T99089 C5TKV7 67053220 IC50 = 13 nM T99089 CU5IJ8 67053231 IC50 = 13 nM T99089 C34TLO 67155626 IC50 = 8.2 nM T99089 CV63UL 67240318 IC50 > 10000 nM T99089 CZJS42 67970606 IC50 = 7 nM T99089 CI9XT5 67970652 IC50 = 67 nM T99089 CGY3O4 67970808 IC50 = 8.2 nM T99089 C09NPT 67970942 IC50 = 149 nM T99089 C0V1YT 67971007 IC50 = 131 nM T99089 CTN06A 67971055 IC50 = 83 nM T99089 C2KVA0 67971197 IC50 = 19 nM T99089 C1ACK8 67971360 IC50 = 11 nM T99089 CWX29O 67991931 IC50 = 16 nM T99089 CX08WF 67995742 IC50 = 63 nM T99089 CH86NY 67995748 IC50 = 40 nM T99089 CE1C9K 67995854 IC50 = 50 nM T99089 C76ZXO 67995947 IC50 = 13 nM T99089 CHI27U 67995956 IC50 = 1 nM T99089 CQM36K 67996004 IC50 = 5 nM T99089 C1CWR6 67996103 IC50 = 79 nM T99089 C4SY7A 67996169 IC50 = 0.5 nM T99089 CJ0M7V 67996291 IC50 = 1 nM T99089 C02XNI 67996483 IC50 = 6 nM T99089 CQXI95 67996588 IC50 = 4 nM T99089 CW17YX 68281294 IC50 > 5000 nM T99089 CU57RD 68304261 IC50 = 250 nM T99089 CD9YL6 68304991 IC50 = 20 nM T99089 C24NDT 68305023 IC50 = 200 nM T99089 CT6D9Q 68305115 IC50 = 13 nM T99089 C0CEX5 68305269 IC50 = 2000 nM T99089 CYAS06 68305303 IC50 = 500 nM T99089 C3JE5H 68356029 IC50 = 371 nM T99089 CGM78B 68472574 IC50 = 2 nM T99089 CB8O4N 68475743 IC50 = 9.5 nM T99089 C5QZW4 68486699 IC50 = 36 nM T99089 CY0DU7 68489225 IC50 = 150 nM T99089 C68QHU 68490094 IC50 = 40 nM T99089 C4XJ6F 68513796 IC50 = 254 nM T99089 CAIO65 68796885 IC50 = 10 nM T99089 C5DGR9 69036886 IC50 = 2035 nM T99089 C4BT3M 69037249 IC50 = 1.2 nM T99089 C07ETL 69934912 IC50 = 6300 nM T99089 CL56IP 70648329 IC50 = 4 nM T99089 C90UOE 70648331 IC50 = 6 nM T99089 CM8VW3 70648666 IC50 = 6 nM T99089 C0FW2K 70648683 IC50 = 0.5 nM T99089 CE61CB 70648685 IC50 = 1 nM T99089 CO9VX3 70649090 IC50 = 8 nM T99089 C1WF5Y 70649102 IC50 = 32 nM T99089 CX1FS0 70649109 IC50 = 1 nM T99089 CQE6V9 70649110 IC50 = 1 nM T99089 CI7L1V 70649115 IC50 = 4 nM T99089 CD3FH7 70649129 IC50 = 6 nM T99089 C0L3KI 70649136 IC50 = 1 nM T99089 CQJ04E 70649137 IC50 = 1000 nM T99089 CRPZ67 70649546 IC50 = 0.6 nM T99089 CIP0R1 70681402 IC50 = 140 nM T99089 CR6QD9 70681403 IC50 > 10000 nM T99089 CU2R4E 70681940 IC50 = 7480 nM T99089 CCR80K 70683505 IC50 > 10000 nM T99089 CD7P4Z 70683506 IC50 > 10000 nM T99089 C6VYT3 70683507 IC50 = 10 nM T99089 C7WJV3 70683520 IC50 = 6 nM T99089 C4H1YN 70683521 IC50 = 0.5 nM T99089 C73WHU 70683665 IC50 = 407 nM T99089 C9THU7 70683668 IC50 = 80 nM T99089 C3ZY9V 70685605 IC50 = 128 nM T99089 CFMJ68 70685606 IC50 = 9 nM T99089 CMY8U3 70687757 IC50 = 72 nM T99089 CIL45P 70687767 IC50 = 15 nM T99089 C63NKC 70687931 IC50 > 10000 nM T99089 C94LEG 70688667 IC50 = 2000 nM T99089 CK6YS5 70689807 IC50 = 239.88 nM T99089 CAI8P9 70691945 IC50 = 338.84 nM T99089 CI6X1V 70691959 IC50 = 0.4 nM T99089 C9DB2A 70694163 IC50 > 10000 nM T99089 CF0L1C 70696119 IC50 = 3606 nM T99089 CT0WC5 70696120 IC50 = 71 nM T99089 CN6MQ5 70696121 IC50 = 13 nM T99089 CN6WH1 70696122 IC50 = 8.7 nM T99089 C7U9QP 70696131 IC50 = 0.5 nM T99089 CD7E8J 70702306 IC50 = 192 nM T99089 CO41NU 71449525 IC50 = 80 nM T99089 C1CQ6R 71450431 IC50 = 23 nM T99089 CAZ3X8 71451311 IC50 = 3.5 nM T99089 CJ1QX0 71451319 IC50 = 52 nM T99089 CEBO91 71452977 IC50 > 10000 nM T99089 CF83BP 71453141 IC50 = 1.9 nM T99089 CR84JX 71453419 IC50 > 1000 nM T99089 CC0B7J 71456634 IC50 = 39 nM T99089 CZ0JA6 71456644 IC50 = 1.3 nM T99089 CJ95FM 71456645 IC50 = 1.2 nM T99089 C4JN5B 71456646 IC50 = 0.7 nM T99089 C7X4MD 71456750 IC50 = 810 nM T99089 CHC18F 71458487 IC50 = 6.8 nM T99089 CY1J6W 71458499 IC50 = 5.1 nM T99089 CHQZ25 71459584 IC50 > 10000 nM T99089 C5HF2X 71460335 IC50 = 1 nM T99089 C4V5GM 71460336 IC50 = 0.9 nM T99089 CVR7F1 71461211 IC50 = 22 nM T99089 CZ6M0W 71462036 IC50 = 3 nM T99089 C37IZM 71518995 IC50 > 10000 nM T99089 C68LCK 71518996 IC50 = 4170 nM T99089 CGF07H 71518997 IC50 = 7940 nM T99089 CTS9V7 71524844 IC50 = 580 nM T99089 C18WLF 71524885 IC50 > 10000 nM T99089 CMB61W 71524886 IC50 > 10000 nM T99089 C1UAL5 71524887 IC50 > 10000 nM T99089 C12CBZ 71524888 IC50 > 10000 nM T99089 C79KSW 71524889 IC50 > 10000 nM T99089 CV1O5J 71524932 IC50 > 10000 nM T99089 C38WUT 71524933 IC50 > 10000 nM T99089 C0BQK4 71524934 IC50 = 330 nM T99089 C5OV9C 71524935 IC50 = 9400 nM T99089 C1SU3J 71524936 IC50 > 10000 nM T99089 C0MEX7 71524978 IC50 = 14000 nM T99089 CQ1C4P 71524979 IC50 > 10000 nM T99089 C85MJU 71524980 IC50 > 10000 nM T99089 C2OS9F 71524981 IC50 > 10000 nM T99089 CZ8T5O 71524982 IC50 = 3600 nM T99089 CT90UG 71525021 IC50 = 9 nM T99089 C2BX7R 71525024 IC50 = 42 nM T99089 CU69TN 71525025 IC50 = 29 nM T99089 CBF84J 71525027 IC50 > 100000 nM T99089 CHQK51 71525066 IC50 > 100000 nM T99089 CT9CH6 71525067 IC50 > 10000 nM T99089 CP41CH 71525069 IC50 = 1100 nM T99089 CYL6J2 71525070 IC50 > 10000 nM T99089 CFW37Q 71525071 IC50 > 10000 nM T99089 CUX15V 71525104 IC50 = 190 nM T99089 CY6S9V 71570573 IC50 = 360 nM T99089 CK1MO3 71570722 IC50 = 3 nM T99089 CYVP02 71570866 IC50 = 36 nM T99089 CPGN04 71582940 IC50 = 28.84 nM T99089 C53GDJ 71582941 IC50 = 300 nM T99089 C27PFR 71582942 IC50 = 100 nM T99089 CWG78B 71583043 IC50 = 208.93 nM T99089 C4W1XT 71583044 IC50 = 67 nM T99089 C5IGH7 71583154 IC50 = 168 nM T99089 C6O4RB 71583157 IC50 = 45 nM T99089 CXWE43 71583159 IC50 = 45 nM T99089 C8YQ4F 71583160 IC50 = 25 nM T99089 C3F8MJ 71583269 IC50 = 257.04 nM T99089 CG17NA 71583271 IC50 = 230 nM T99089 C6DO5H 71583273 IC50 = 74 nM T99089 CQP5V0 71583274 IC50 = 4 nM T99089 C8THY0 71583275 IC50 = 5 nM T99089 C9IOY7 71583377 IC50 = 8 nM T99089 CWO26F 71583378 IC50 = 38.9 nM T99089 CUYC39 71583380 IC50 = 10 nM T99089 C9HQR0 71583494 IC50 = 25 nM T99089 CCJ37F 71583495 IC50 = 430 nM T99089 CLB5J6 71583602 IC50 = 20 nM T99089 C2PZ5G 71583603 IC50 = 573 nM T99089 CW20DX 71583604 IC50 = 25 nM T99089 CZ31PU 71583657 IC50 = 230 nM T99089 CN8ZD6 71584271 IC50 = 398.11 nM T99089 CNH8G5 71584401 IC50 = 263.03 nM T99089 C56ICO 71584402 IC50 = 131.83 nM T99089 CQ4ZV3 71584403 IC50 = 369 nM T99089 CBX50I 71584404 IC50 = 917 nM T99089 CEJ69H 71584405 IC50 = 601 nM T99089 C72PUL 71584406 IC50 = 2290.87 nM T99089 CEXG64 71584539 IC50 = 5370.32 nM T99089 C8KHE0 71584540 IC50 = 777 nM T99089 CFJ45Z 71584541 IC50 = 330 nM T99089 CI5VT4 71584542 IC50 = 350 nM T99089 C8IG3A 71584543 IC50 = 280 nM T99089 CKCO49 71584544 IC50 = 89 nM T99089 CGM5P4 71584661 IC50 = 52.48 nM T99089 CA0GI1 71584662 IC50 = 130 nM T99089 CY28UI 71627417 IC50 = 22 nM T99089 C0XEQ1 71682500 IC50 > 5000 nM T99089 CRK2G6 71718268 IC50 = 16 nM T99089 CU83YL 71730951 IC50 = 18 nM T99089 C1TD4L 71731206 IC50 = 7.9 nM T99089 C7F3ZM 71736390 IC50 = 8.4 nM T99089 C9EM5X 71736552 IC50 = 4.3 nM T99089 CKYO24 71736864 IC50 = 18 nM T99089 CA1JH2 71815073 IC50 = 190 nM T99089 C1E4RK 71818600 IC50 = 19 nM T99089 CX78NJ 71818601 IC50 = 18 nM T99089 C8WZ1R 71818732 IC50 = 14 nM T99089 C4B7ZW 71818733 IC50 = 9.5 nM T99089 C0QBF6 72375428 IC50 = 3.4 nM T99089 CL14JN 73330891 IC50 = 3.15 nM T99089 CXW8L5 73330892 IC50 = 2.78 nM T99089 CK9ST7 73330893 IC50 = 1.2 nM T99089 CINP24 73330894 IC50 = 19.1 nM T99089 CK3FN2 73331037 IC50 = 29.4 nM T99089 CX2I7B 73331038 IC50 = 1.03 nM T99089 CJC7V0 73331039 IC50 = 7.13 nM T99089 CMJY29 73331040 IC50 = 1.6 nM T99089 CB96JV 73331041 IC50 = 1.3 nM T99089 CKT5E7 73331182 IC50 = 2.17 nM T99089 CNO0C9 73331183 IC50 = 3.62 nM T99089 C7PI5W 73331184 IC50 = 1.5 nM T99089 C4CRH9 73331185 IC50 = 4.82 nM T99089 C0FYW2 73331186 IC50 = 8.07 nM T99089 C6XHO8 73331320 IC50 = 0.79 nM T99089 C6TA4H 73331323 IC50 = 2.51 nM T99089 CU60BO 73331324 IC50 = 2.71 nM T99089 CF3C1P 73331464 IC50 = 3.03 nM T99089 CEAF70 73425627 IC50 = 0.8 nM T99089 CD84TH 73425628 IC50 = 0.8 nM T99089 C2UGD3 73425629 IC50 = 0.1 nM T99089 C3QDX5 73425728 IC50 = 0.6 nM T99089 CC7GL1 73427048 IC50 = 70 nM T99089 CF2C5V 73427050 IC50 = 11 nM T99089 CJPU56 73427150 IC50 = 220 nM T99089 CX5K0Z 73427151 IC50 = 7 nM T99089 CQJ0R1 73427152 IC50 = 80 nM T99089 C1QFO2 73427153 IC50 = 7 nM T99089 CKI3Z2 73427155 IC50 = 7 nM T99089 C80SEC 73504974 IC50 = 187 nM T99089 CK1BY2 73504975 IC50 = 165 nM T99089 CE79YJ 73505176 IC50 = 1780 nM T99089 CC75WA 73505177 IC50 = 3260 nM T99089 C2LGB5 73505178 IC50 = 4060 nM T99089 CFG01S 73505179 IC50 = 942 nM T99089 C3KVB2 73505180 IC50 = 73 nM T99089 C0JF6O 75596779 IC50 = 157 nM T99089 C5BV3G 76310396 IC50 = 880 nM T99089 CX4H6I 86583042 IC50 = 8 nM T99089 CVR43W 86583044 IC50 > 1000 nM T99089 CA81UY 86583045 IC50 > 1000 nM T99089 CI2CG1 89670173 IC50 = 23 nM T99089 C1HW4B 89735655 IC50 = 1100 nM T99089 C7TJR3 89814000 IC50 = 27 nM T99089 C4WP7D 89827799 IC50 = 7.7 nM T99089 CZJ8N6 90116353 IC50 = 3.5 nM T99089 CB7R6C 90116945 IC50 = 4.2 nM T99089 CNR6C3 90120675 IC50 = 31 nM T99089 C6RZ7J 90408826 IC50 = 0.4 nM T99089 CW61DN 90488999 IC50 = 2.1 nM T99089 CY9FE6 90655275 IC50 = 551 nM T99089 C1CFP6 90655276 IC50 = 573 nM T99089 CI8XW3 90655277 IC50 = 110 nM T99089 CT28VM 90655278 IC50 = 240 nM T99089 C8N5TF 90655279 IC50 = 280 nM T99089 CPN1I6 90655280 IC50 = 670 nM T99089 CW1LJ4 90655281 IC50 = 410 nM T99089 CAC3D4 90655282 IC50 > 10000 nM T99089 CKO3Z1 90655283 IC50 = 290 nM T99089 C7S8KR 90655284 IC50 = 510 nM T99089 CY0T9O 90655285 IC50 = 340 nM T99089 CG9HX4 90655286 IC50 = 390 nM T99089 C7DT3G 90655287 IC50 = 230 nM T99089 C8RA1Y 90655288 IC50 = 37 nM T99089 C1B7TW 90655289 IC50 = 210 nM T99089 CVO26Z 90655290 IC50 = 300 nM T99089 CO5M8T 90655291 IC50 = 48 nM T99089 CXNB56 90655292 IC50 = 220 nM T99089 CW08SL 90655293 IC50 = 48 nM T99089 CC2P7K 90655294 IC50 = 360 nM T99089 CBX47C 90655295 IC50 = 290 nM T99089 CWD4O3 90655989 IC50 > 50000 nM T99089 CMH6T8 90664306 IC50 = 1.6 nM T99089 CND1X5 90670915 IC50 = 314 nM T99089 C92HCD 102531936 EC50 < 500 nM T99089 C4MBJ3 102531937 IC50 < 100 nM T99089 C4UTP7 102531938 IC50 < 100 nM T99089 CTGP06 117996541 IC50 = 416.87 nM T99089 CY3L2E 117996700 IC50 > 10000 nM T99089 CVP10Z 117996749 IC50 = 2900 nM T99089 CG7QL4 118705925 IC50 = 38.3 nM T99089 C4AHL2 118711367 IC50 > 10000 nM T99089 C5E6DW 118720154 IC50 = 12 nM T99089 C0XWT1 118720155 IC50 = 4.21 nM T99089 CKA6P4 118720156 IC50 = 13.5 nM T99089 C63KJT 118720157 IC50 = 10.8 nM T99089 C9UQA1 118720457 IC50 = 0.669 nM T99089 CRJ82K 118720458 IC50 = 2.56 nM T99089 CS45ZU 118720459 IC50 = 1.77 nM T99089 CQP9B3 118720460 IC50 = 7.44 nM T99089 C5OIW3 118720461 IC50 = 471 nM T99089 CWQC25 118720462 IC50 = 6430 nM T99089 C3KLI5 118723185 IC50 > 100000 nM T99089 CD1RU5 118725683 IC50 = 2470 nM T99089 C17SHY 118725687 IC50 = 40400 nM T99089 CZVH46 118725690 IC50 = 650 nM T99089 C6GQL2 118725758 IC50 = 531 nM T99089 C5QC8E 118730408 IC50 > 1000 nM T99089 C4TXF2 118730409 IC50 > 1000 nM T99089 CN2A9O 118730410 EC50 = 190 nM T99089 COF69K 118730411 IC50 = 8 nM T99089 CEJ1S6 118730412 IC50 = 66 nM T99089 CQ0T5Z 118730413 IC50 = 13 nM T99089 CF47CO 118730414 IC50 > 1000 nM T99089 CEJ67D 118730415 IC50 > 1000 nM T99089 C5SI6Q 118730416 IC50 > 1000 nM T99089 CR0H9D 118730417 IC50 > 1000 nM T99089 CGDW48 118730418 IC50 > 1000 nM T99089 C23KFD 118730419 IC50 > 1000 nM T99089 CJ9SA8 118730420 IC50 > 1000 nM T99089 C0HK5A 118730421 IC50 > 1000 nM T99089 C1Q0UN 118730422 IC50 > 1000 nM T99089 C1K0PE 118730423 IC50 > 1000 nM T99089 CQCX41 118737057 IC50 = 15 nM T99089 CESI90 118988423 IC50 = 54 nM T99089 C0UT7G 122177477 IC50 = 6.8 nM T99089 CSF49R 122177478 IC50 = 40 nM T99089 CDQ60H 122179517 IC50 = 149 nM T99089 CS07QW 122179518 IC50 = 177 nM T99089 C6HB9Q 122179519 IC50 = 68 nM T99089 CH6C3N 122179520 IC50 = 917 nM T99089 C4P2OM 122179521 IC50 = 593 nM T99089 CQ52KS 122179522 IC50 = 51 nM T99089 CBS2G4 122179523 IC50 = 48 nM T99089 CXN92S 122179524 IC50 = 4310 nM T99089 CQ48MD 122179525 IC50 = 533 nM T99089 CHC9Z8 122179526 IC50 = 17 nM T99089 CSFU53 122179527 IC50 = 122 nM T99089 CRH7W6 122179528 IC50 = 25 nM T99089 CKFP69 122179529 IC50 = 10 nM T99089 C9KF6J 122179530 IC50 = 16 nM T99089 CG3OM1 122179531 IC50 = 3 nM T99089 C29LPV 122179532 IC50 = 131 nM T99089 CO5TH2 122179533 IC50 = 107 nM T99089 CAPV50 122179534 IC50 = 21 nM T99089 CL4OW0 122179535 IC50 = 11 nM T99089 C08KEM 122179540 IC50 = 2500 nM T99089 CG0RP7 122179547 IC50 = 6200 nM T99089 C1A0SQ 122179548 IC50 = 5900 nM T99089 C5B6QT 122189918 IC50 = 668 nM T99089 COWC81 127025601 IC50 = 2.9 nM T99089 C1HGA4 127025889 IC50 = 2.1 nM T99089 CF61HD 127025890 IC50 = 74 nM T99089 CM74CE 127025891 IC50 = 34 nM T99089 CAPU43 127026035 IC50 > 30 nM T99089 CQVU25 127026051 IC50 = 17 nM T99089 CZVP92 127028061 IC50 = 67 nM T99089 CZ3G8X 127028062 IC50 = 854 nM T99089 C2KCN9 127028071 IC50 > 12500 nM T99089 CN32ML 127028362 IC50 = 2.9 nM T99089 C1K5UC 127028929 IC50 = 20 nM T99089 C6KM3T 127034964 IC50 = 2 nM T99089 CF5WH1 127039888 IC50 = 7820 nM T99089 CH09EC 127041357 IC50 > 12500 nM T99089 C0D7RE 127042274 IC50 > 12500 nM T99089 C6NZ1Q 127042619 IC50 > 12500 nM T99089 CS2AP8 127042622 IC50 = 2.7 nM T99089 CL40ZB 127042623 IC50 = 3.1 nM T99089 CJ45OF 127042624 IC50 = 45 nM T99089 C3NMP8 127042932 IC50 = 5010 nM T99089 CP9L4A 127042940 IC50 = 1.9 nM T99089 CJ1G3I 127045769 IC50 = 1 nM T99089 CKL75H 127045770 IC50 = 1 nM T99089 CN7Z1E 127045771 IC50 = 216 nM T99089 CHM08S 127045839 IC50 = 141 nM T99089 C8W9VK 127045991 IC50 = 177 nM T99089 C2S9ZM 127046079 IC50 = 57 nM T99089 CFP01I 127046080 IC50 = 44 nM T99089 C8LRC5 127046081 IC50 = 15 nM T99089 C1BLZ3 127046082 IC50 = 122 nM T99089 CGO7P6 127046232 IC50 = 420 nM T99089 C9P5OW 127046289 IC50 = 68 nM T99089 CM05VG 127046445 IC50 = 17 nM T99089 CJZ6X2 127046446 IC50 = 26 nM T99089 CNA7K2 127046457 IC50 = 13 nM T99089 CC2AP7 127046458 IC50 = 240 nM T99089 CJ8V6Q 127046459 IC50 = 453 nM T99089 CSX5M4 127046460 IC50 = 38 nM T99089 CN26AU 127046461 IC50 = 2031 nM T99089 CAG9K7 127046489 IC50 = 95 nM T99089 CA6WZ4 127046615 IC50 = 5 nM T99089 CR7V4J 127047050 IC50 = 3 nM T99089 C2UBH1 127047051 EC50 = 1510 nM T99089 C7U9GE 127047125 IC50 = 563 nM T99089 CKU72G 127047243 IC50 = 2 nM T99089 C7P9XY 127047244 IC50 = 26 nM T99089 CFBT16 127047245 IC50 = 356 nM T99089 CK5XG8 127047246 IC50 = 22 nM T99089 C6DP7Y 127047275 IC50 = 131 nM T99089 C3DVM9 127047276 IC50 = 1230 nM T99089 CXK40B 127047368 IC50 > 10000 nM T99089 CEND36 127047369 IC50 > 10000 nM T99089 C34NAH 127047506 IC50 = 785 nM T99089 C2GA5N 127047507 IC50 = 1512 nM T99089 C38WDB 127047508 IC50 = 3530 nM T99089 CLXZ13 127047509 IC50 = 1210 nM T99089 CHC2M7 127047632 IC50 = 110 nM T99089 C0U1FB 127047676 IC50 = 1000 nM T99089 C3YWV1 127047786 IC50 = 50 nM T99089 CLPC17 127047787 IC50 = 125 nM T99089 C81LVM 127047788 IC50 = 1030 nM T99089 C12AUN 127047893 IC50 = 111 nM T99089 CMBQ27 127047908 IC50 = 182 nM T99089 COTB30 127047909 IC50 = 434 nM T99089 CM81AR 127047922 IC50 = 4300 nM T99089 CRV7N4 127048021 IC50 = 27 nM T99089 C4JKZ1 127048022 EC50 = 8090 nM T99089 C67PQF 127048023 IC50 = 4 nM T99089 CC7IS1 127048327 IC50 = 1490 nM T99089 CK03IO 127048328 IC50 = 610 nM T99089 C2KYI6 127048329 IC50 = 230 nM T99089 C1JZ8I 127048676 IC50 = 720 nM T99089 CLN2V6 127048677 IC50 = 2540 nM T99089 CP6D8F 127048678 IC50 = 670 nM T99089 CBEM37 127049658 IC50 > 10000 nM T99089 CJG89B 127049660 IC50 = 840 nM T99089 C6OP7G 127049661 IC50 = 55 nM T99089 CP9T1K 127049662 IC50 = 420 nM T99089 CW0Y3A 127049663 IC50 = 60 nM T99089 CB2M4K 127049664 IC50 = 210 nM T99089 CSV6H4 127049665 IC50 = 1640 nM T99089 CT6W1K 127049960 IC50 > 10000 nM T99089 C1CFZ7 127049961 IC50 = 300 nM T99089 CGWP70 127049962 IC50 = 9870 nM T99089 C4KAX3 127049963 IC50 > 10000 nM T99089 CAQL02 127049964 IC50 > 10000 nM T99089 C0FU7Y 127049965 IC50 = 200 nM T99089 C0XS1L 127051137 IC50 = 1000 nM T99089 C0AJS1 127051166 IC50 > 10000 nM T99089 CQ1K5O 127051167 IC50 > 10000 nM T99089 CKC0Z6 127051168 IC50 > 10000 nM T99089 CA91BN 127051468 IC50 = 5920 nM T99089 CV3L6M 127052123 IC50 = 1200 nM T99089 CTV2I4 127052124 IC50 > 10000 nM T99089 CJ21BE 127052125 IC50 > 10000 nM T99089 CVB1C9 127052416 IC50 = 130 nM T99089 C74KCH 127052706 IC50 = 250 nM T99089 C0FM1R 130196825 IC50 = 8294 nM T99089 CM2J3B 131953483 IC50 > 1000 nM T99089 CBI35E 132275094 IC50 = 14 nM T99089 CU1H0W 132497402 IC50 = 77.2 nM T99089 CSZA35 134133678 IC50 = 10120 nM T99089 CXSB18 134133754 IC50 = 22010 nM T99089 CRH7A2 134135364 IC50 = 1760 nM T99089 C62GWK 134141404 IC50 = 2400 nM T99089 C4QT7E 134142822 IC50 > 50000 nM T99089 C7I5JQ 134144573 IC50 = 2560 nM T99089 CDMB08 134145603 IC50 > 50000 nM T99089 CVNG59 134145628 IC50 = 8930 nM T99089 CMY13K 134146982 IC50 = 24230 nM T99089 CUZ48A 134149722 IC50 = 680 nM T99089 CU4T3D 134149937 IC50 = 33490 nM T99089 CYL31R 134150731 IC50 = 280 nM T99089 C8OP5K 134151586 IC50 = 3270 nM T99089 CC3Y0N 134152150 IC50 = 1840 nM T99089 C9B6PV 134152705 IC50 = 370 nM T99089 C8WVZ0 134152967 IC50 = 2900 nM T99089 CPZ10X 134155617 IC50 = 17810 nM T99089 C29UML 134155621 IC50 = 1800 nM T99089 CMPS85 134155826 IC50 = 920 nM T99089 C2AN7T 134611886 IC50 > 100000 nM T99089 CX1FA8 135399664 IC50 < 2 nM T99089 CKY3I2 135401910 IC50 = 0.2 nM T99089 C2H0FA 135401911 IC50 < 2 nM T99089 C85QZP 135453073 IC50 = 18000 nM T99089 CHJU83 135466457 IC50 = 0.15 nM T99089 CQ7L2Y 135482542 IC50 = 29420 nM T99089 CMW1V4 135505774 IC50 = 16 nM T99089 C2GQW0 135508240 IC50 = 0.48 nM T99089 C8B5GZ 135513879 IC50 = 339 nM T99089 CEK31P 135566415 IC50 > 20000 nM T99089 C8P7BR 135688666 IC50 > 100000 nM T99089 CX4ZB3 135863110 IC50 > 10000 nM T99089 C30RIL 135895396 IC50 = 250 nM T99089 CC7J0Q 135923565 IC50 = 4900 nM T99089 CJL23B 135936239 IC50 = 130 nM T99089 C51AMW 135981332 IC50 = 720 nM T99089 CG9PJ7 135993841 IC50 = 655.2 nM T99089 CN47FL 136030704 IC50 = 35 nM T99089 CDYC36 136030724 IC50 = 16 nM T99089 CW7G2B 136042252 IC50 = 954 nM T99089 C5HUM3 136045809 IC50 = 18.4 nM T99089 CZU9M0 136073752 IC50 = 110 nM T99089 CG1R7B 136087060 IC50 > 10000 nM T99089 C8YZS6 136141580 IC50 = 47 nM T99089 C3COS8 136160805 IC50 = 0.5 nM T99089 CGKV52 136164074 IC50 = 1600 nM T99089 CZ7EX0 136183413 IC50 > 30000 nM T99089 CI6V9T 136192928 IC50 = 4 nM T99089 C4KSL5 136235605 IC50 = 8800 nM T99089 C4P5VI 137631729 IC50 > 10000 nM T99089 C4N0LW 137631825 IC50 > 1000 nM T99089 C7NFX9 137632089 IC50 = 24.1 nM T99089 C9OV8U 137632895 IC50 = 140 nM T99089 C4JIL5 137633313 IC50 = 46.1 nM T99089 C51IZU 137633597 IC50 = 25.1 nM T99089 CI1E8V 137634241 IC50 > 10000 nM T99089 CP8UG5 137634530 IC50 = 0.3 nM T99089 CN4BD6 137634880 IC50 = 21.4 nM T99089 C95VXH 137634988 IC50 = 39.1 nM T99089 C2FGN9 137635830 IC50 = 68.2 nM T99089 C8DTW2 137636634 IC50 = 135 nM T99089 C08MHJ 137636777 IC50 = 2.8 nM T99089 C0OWY3 137636794 IC50 > 10000 nM T99089 CV3A5G 137637973 IC50 = 60 nM T99089 COT76N 137638146 IC50 = 38.6 nM T99089 C3M5ET 137638260 IC50 = 8.4 nM T99089 C7TN8O 137639492 IC50 = 22.4 nM T99089 COBX17 137640041 IC50 = 441 nM T99089 CF5I3U 137640119 IC50 = 59.5 nM T99089 C0SJ2W 137640898 IC50 = 4.3 nM T99089 CA13KP 137642491 IC50 = 18.7 nM T99089 CDG2S9 137643098 IC50 = 152 nM T99089 CRI78Y 137643278 IC50 = 143 nM T99089 C9SOI8 137644117 IC50 > 2000 nM T99089 CHM1K2 137644157 IC50 = 88.6 nM T99089 C23ACF 137644903 IC50 > 2000 nM T99089 CQS67M 137644972 IC50 > 5000 nM T99089 CL8W4P 137647062 IC50 = 14.3 nM T99089 CIJK82 137647304 IC50 > 10000 nM T99089 C97LQG 137647372 IC50 = 169.2 nM T99089 C0KZ9Q 137647934 IC50 = 201 nM T99089 CGQ02E 137648059 IC50 = 10.5 nM T99089 CZ2B1S 137648159 IC50 = 30.8 nM T99089 CB7M8Z 137648383 IC50 = 21.6 nM T99089 CL9HT1 137648599 IC50 = 19.5 nM T99089 C8FV4X 137649404 IC50 = 35.8 nM T99089 CJMW91 137649638 IC50 > 1000 nM T99089 CNTC73 137649645 IC50 = 80.2 nM T99089 CF1H4X 137650051 IC50 > 10000 nM T99089 C1BUD8 137650370 IC50 = 145 nM T99089 CE7KF3 137650390 IC50 = 12.2 nM T99089 C3O6KY 137652367 IC50 = 29.1 nM T99089 CBVE69 137652761 IC50 = 388 nM T99089 CYMU46 137654572 IC50 = 178 nM T99089 CHSL51 137654792 IC50 = 43.1 nM T99089 CVCD38 137654923 IC50 = 18.3 nM T99089 CF8HI3 137655054 IC50 = 44.1 nM T99089 CF2PV0 137655959 IC50 = 901.8 nM T99089 C21RYV 137656620 IC50 = 237 nM T99089 CMPJ36 137656808 IC50 = 21.2 nM T99089 C6Y8BI 137656893 IC50 = 31.5 nM T99089 CHF87V 137657244 IC50 > 1000 nM T99089 CN7J2A 137657347 IC50 > 10000 nM T99089 CVQF35 137659532 IC50 = 251 nM T99089 C2VQL7 137660816 IC50 = 13.9 nM T99089 CZ4WT5 137661137 IC50 = 18.5 nM T99089 C1W3PN 137661841 IC50 > 1000 nM T99089 CA4V9R 137661906 IC50 = 260 nM T99089 C2JI6T 138393294 IC50 > 1000 nM T99089 C68OZS 138403232 IC50 = 420 nM T99089 CK90OA 138753620 IC50 = 272.3 nM T99089 COB9P2 141456067 IC50 = 3400 nM T99089 C6CN8H 142739455 IC50 = 316 nM T99089 C6VB3O 145925651 IC50 >= 5000 nM T99089 CB3Z1W 145949428 IC50 = 32 nM T99089 CT25FH 145950796 IC50 = 23.6 nM T99089 CHKS76 145952159 IC50 = 215.6 nM T99089 C1G0PH 145952494 IC50 = 407.2 nM T99089 C9WYS2 145954493 IC50 = 40.9 nM T99089 CF1T9Y 145954667 IC50 = 171.5 nM T99089 CX80ZF 145954847 IC50 = 85.2 nM T99089 CBR2Q7 145956253 IC50 = 476.3 nM T99089 C5VSC7 145956704 IC50 = 20 nM T99089 CZ3G0H 145959478 IC50 = 487.8 nM T99089 C7RQ8I 145960033 IC50 = 105.6 nM T99089 C7O0EG 145964682 EC50 = 240 nM T99089 CT49MR 145965412 IC50 = 6 nM T99089 C4NP2V 145965631 IC50 > 50000 nM T99089 C9H4TP 145966705 EC50 = 540 nM T99089 CR6O2S 145967668 IC50 = 5851 nM T99089 C49QZE 145967671 IC50 = 158 nM T99089 C0UZ6Q 145967831 IC50 = 1785 nM T99089 C2CHJ9 145967839 IC50 = 810 nM T99089 C5E8ZK 145968310 IC50 = 27 nM T99089 CTX9I2 145968517 IC50 = 69 nM T99089 C0Y1IT 145968532 IC50 = 973 nM T99089 CL0BO5 145968619 IC50 > 10000 nM T99089 CHAU61 145968737 IC50 = 21 nM T99089 CK1N7F 145968871 IC50 = 93 nM T99089 CBJ0F1 145968889 IC50 = 503 nM T99089 C0BG4F 145968971 IC50 = 442 nM T99089 CFC48X 145969905 IC50 = 791 nM T99089 C4D3BL 145970607 IC50 = 33 nM T99089 C8NK3O 145970839 IC50 = 17 nM T99089 CP6QH1 145971042 IC50 = 9866 nM T99089 C87WHG 145973554 IC50 = 0.3 nM T99089 CLN2D9 145973734 EC50 = 480 nM T99089 C76RQZ 145976309 IC50 = 0.9 nM T99089 CBR8K6 145976838 IC50 = 3900 nM T99089 C59VIT 145977243 IC50 > 50000 nM T99089 C93ZOX 145977611 IC50 = 5 nM T99089 CG9BL6 145979052 IC50 = 39300 nM T99089 C2I5WD 145979310 IC50 = 29.7 nM T99089 C0DOU5 145979395 IC50 = 510 nM T99089 CQ03XU 145980353 IC50 > 200000 nM T99089 C16ENO 145980866 IC50 = 223.87 nM T99089 CTC34W 145981191 IC50 = 21300 nM T99089 CI24XE 145981336 IC50 > 200000 nM T99089 CJPU41 145981957 IC50 = 1000 nM T99089 C6T4MU 145982183 IC50 = 19 nM T99089 CSWY46 145982727 IC50 = 73.9 nM T99089 CIYQ21 145982961 IC50 = 5.75 nM T99089 CBR08X 145983359 IC50 = 13 nM T99089 CE2X6V 145983518 IC50 = 44 nM T99089 C4QE7K 145983757 IC50 = 2600 nM T99089 CFRC51 145984297 IC50 = 73.8 nM T99089 CLV2K6 145984391 IC50 > 200000 nM T99089 C1DM4I 145984486 IC50 = 2900 nM T99089 COPW70 145984516 IC50 = 2700 nM T99089 C4ID8J 145984666 IC50 = 51 nM T99089 C06ECS 145984689 IC50 = 352 nM T99089 C05VIR 145984747 IC50 = 46 nM T99089 CGT8Z5 145984754 IC50 = 168 nM T99089 CW6ZJ2 145984860 IC50 = 87 nM T99089 CI1VH9 145985185 IC50 > 200000 nM T99089 CR91FS 145985335 IC50 = 24 nM T99089 CSQ34B 145985725 IC50 = 20.3 nM T99089 CQ5S2M 145985741 IC50 = 421 nM T99089 CL3HZ6 145986481 IC50 = 48900 nM T99089 C10TUA 145986573 IC50 = 280 nM T99089 CS78MW 145986924 IC50 = 156000 nM T99089 C1FE9Y 145987180 IC50 = 4.786 nM T99089 C96XWA 145987467 IC50 = 1.698 nM T99089 CK8S4V 145988419 IC50 = 48 nM T99089 CI7M2B 145988861 IC50 = 12.6 nM T99089 CNLH48 145988888 IC50 = 18700 nM T99089 CBC9Q6 145989837 IC50 = 61 nM T99089 CMQG17 145990430 IC50 = 1360 nM T99089 CB0AC5 145990447 IC50 = 5210 nM T99089 C2GWJ6 145990512 IC50 = 124000 nM T99089 C3WRL8 145990775 IC50 > 200000 nM T99089 CC1Z8Y 145991567 IC50 = 23100 nM T99089 CR76UY 145991825 IC50 = 35600 nM T99089 C6UNJ7 145992396 IC50 = 95900 nM T99089 CRT48W 145993502 IC50 = 5230 nM T99089 CF57DG 146020550 IC50 = 125.7 nM T99089 CCO93U 154634893 IC50 = 453 nM T99089 C5DMK6 154634900 IC50 > 1000 nM T99089 CVY7N6 154634909 IC50 = 795 nM T99089 C7YD9F 154634910 IC50 > 1000 nM T99089 CE4V9P 154634911 IC50 = 856 nM T99089 C9CQ3T 154634913 IC50 = 272 nM T99089 CEC1D3 154634916 IC50 > 1000 nM T99089 CGO62P 154634918 IC50 = 190 nM T99089 C41FIQ 154634920 IC50 = 39 nM T99089 C6XWC7 154634922 IC50 = 334 nM T99089 C2NKF8 155076930 IC50 = 13.4 nM T99089 CY1ZH2 155510358 IC50 = 158 nM T99089 CB0IE5 155511260 IC50 = 2600 nM T99089 C0O5DS 155511991 IC50 = 3.9 nM T99089 C73ZFN 155512053 IC50 = 390 nM T99089 CZ5S2M 155512875 IC50 = 3.5 nM T99089 C1LC2I 155513138 IC50 = 0.2 nM T99089 C2MD1Q 155513187 IC50 > 10000 nM T99089 C8DAU4 155513645 IC50 = 7.4 nM T99089 C60ASE 155514455 IC50 = 7 nM T99089 CI54TD 155514548 IC50 = 3740 nM T99089 C2BA1L 155514841 IC50 = 6320 nM T99089 CX2E0D 155514846 IC50 = 7410 nM T99089 CX8LF1 155515119 IC50 = 100 nM T99089 CX6SR0 155516442 IC50 = 940 nM T99089 C13KCF 155517164 IC50 = 83.1 nM T99089 C40CDF 155518050 IC50 = 9 nM T99089 CS31UH 155519078 IC50 = 5320 nM T99089 CMH01P 155519212 IC50 = 189 nM T99089 C3M6GZ 155519761 IC50 = 220 nM T99089 CEZ4O1 155520166 IC50 = 198 nM T99089 C2IC0U 155520258 IC50 = 320 nM T99089 CRNT47 155520316 IC50 = 87200 nM T99089 CU6Z5O 155520650 IC50 = 110 nM T99089 C8P6FS 155520920 IC50 > 300 nM T99089 CP4JL5 155521754 IC50 < 10000 nM T99089 CM3DB7 155523430 IC50 = 1290 nM T99089 CLB37N 155524340 IC50 = 919 nM T99089 CD2U5W 155524889 IC50 = 212 nM T99089 C6BAZ7 155525737 IC50 = 14 nM T99089 CYZ16N 155526190 IC50 > 1000 nM T99089 CZQ8D2 155526237 IC50 = 4170 nM T99089 C3QDI9 155526245 IC50 = 6.2 nM T99089 C46UIC 155526269 IC50 = 688 nM T99089 CH87DO 155527260 IC50 = 21 nM T99089 C6AGH4 155527315 IC50 > 1000 nM T99089 CH02ZE 155530305 IC50 = 45 nM T99089 CL0V4U 155530858 IC50 = 640 nM T99089 CLY07C 155530863 IC50 = 830 nM T99089 CC0WN1 155531780 IC50 = 342 nM T99089 CTMD13 155531884 IC50 = 30 nM T99089 CVQ24P 155532080 IC50 = 3210 nM T99089 CS69CA 155532132 IC50 = 1.9 nM T99089 CAB6E5 155532196 IC50 = 160 nM T99089 C6GT5Q 155533377 IC50 = 475 nM T99089 CI6B1M 155534397 IC50 = 2115 nM T99089 CKN58D 155534426 IC50 = 157 nM T99089 CH41LY 155534535 IC50 = 29 nM T99089 C0W8FZ 155534624 IC50 = 3690 nM T99089 CB9MT3 155535246 IC50 = 12.3 nM T99089 CF37GO 155535511 IC50 = 354 nM T99089 CC3ZU4 155536475 IC50 = 34.5 nM T99089 C8CK3X 155536944 IC50 = 38 nM T99089 CJ6SF9 155538658 IC50 = 303 nM T99089 C7PGF1 155539109 IC50 > 300 nM T99089 C5J8CV 155540640 IC50 = 26 nM T99089 C4R3QZ 155541552 IC50 = 2.3 nM T99089 CEJO32 155541565 IC50 = 43.7 nM T99089 C2AV3O 155541683 IC50 = 92 nM T99089 CX0J3Y 155543780 IC50 = 11.4 nM T99089 C8ZF4H 155544511 IC50 = 15700 nM T99089 C8T0MQ 155544690 IC50 = 3250 nM T99089 CY3H1I 155545239 IC50 = 348 nM T99089 C9L2CV 155546337 IC50 > 300 nM T99089 CQXE36 155547334 IC50 = 51.6 nM T99089 CB45ZE 155548916 IC50 = 34.1 nM T99089 CQF73Y 155549371 IC50 = 440 nM T99089 CHM75U 155549823 IC50 = 140 nM T99089 CG0IV2 155550125 IC50 > 300 nM T99089 C0IK8P 155550720 IC50 = 410 nM T99089 C0W7YS 155551457 IC50 > 300 nM T99089 CAH09B 155552200 IC50 = 300 nM T99089 CHE5F1 155553390 IC50 = 26800 nM T99089 C2T4PR 155553405 IC50 = 1.2 nM T99089 C30HXP 155554372 IC50 = 47 nM T99089 CD5V3C 155556809 IC50 = 13.4 nM T99089 C59PVM 155557441 IC50 > 1000 nM T99089 CP60UD 155557689 IC50 = 1700 nM T99089 CC7ES5 155557982 IC50 = 2.1 nM T99089 CBYQ06 155559698 IC50 = 237 nM T99089 CYC23K 155560669 IC50 = 700 nM T99089 C3ISX8 155560929 IC50 = 370 nM T99089 C8SP4L 155562403 IC50 > 300 nM T99089 CLU0T2 155562940 IC50 = 540 nM T99089 C81JZW 155563388 IC50 = 150 nM T99089 CQ1Y5C 155564359 IC50 = 251 nM T99089 CFOH01 155564397 IC50 = 488 nM T99089 CM47DW 155565162 IC50 > 300 nM T99089 C62CIM 155565320 IC50 = 9420 nM T99089 CSA97I 155565690 IC50 = 470.3 nM T99089 C9QAE3 155566144 IC50 = 436 nM T99089 CH3NO1 155566774 IC50 = 15.8 nM T99089 C69ICK 155567369 IC50 = 17 nM T99089 CC0DK2 155567575 IC50 = 41 nM T99089 C0E8CV 155568098 IC50 = 1050 nM T99089 C0V2MU 135398506 IC50 = 0.16 nM T99089 CR6MZ8 136030631 IC50 < 2 nM T99089 CQ5P6E 49837197 IC50 = 2.3 nM T99089 D00NWF 5730 IC50 = 230 nM T99089 D01DDB 11515006 IC50 = 7900 nM T99089 D02BXJ 46864270 IC50 = 26 nM T99089 D06QWO 14824655 IC50 > 10 ug.mL-1 T99089 D06WJA 9950176 IC50 = 10 nM T99089 D09ADW 53484100 IC50 = 0.7 nM T99089 D0A1CM 5281855 IC50 = 1760 nM T99089 D0C0ZC 11676786 IC50 < 1 nM T99089 D0D6MH 11617559 IC50 > 4800 nM T99089 D0G3SZ 6918469 IC50 = 3.3 ug.mL-1 T99089 D0GD8Y 3006531 IC50 = 250 nM T99089 D0OR5S 11631107 IC50 = 18000 nM T99089 D0OZ2S 11785878 IC50 = 540 nM T99089 D0T3PW 5281672 IC50 = 1562 nM T99089 D0Z5TQ 5924208 IC50 = 10.71 nM T23276 D0W5HK 216239 IC50 = 18.1 nM T23276 D02UFQ 11620908 IC50 > 10000 nM T23276 D05ADP 160355 IC50 = 34000 nM T23276 D0E3TC 44259 IC50 = 1310 nM T23276 D0L1GD 58282870 IC50 = 20 nM T23276 D0LF1U 5287969 IC50 = 16000 nM T23276 D0O6ZO 9952773 IC50 > 10000 nM T23276 D0Q4IX 71727581 IC50 = 1.2 nM T23276 D0X4MN 11597537 IC50 = 480 nM T23276 D0WS1V 448991 IC50 = 3300 nM T23276 D00PWQ 3820 IC50 = 20000 nM T23276 D00BPA 4592 IC50 = 25000 nM T23276 D04FHB 6918852 Ki > 50000 nM T23276 D0T3ME 156422 IC50 > 20000 nM T23276 C4MNG8 445840 IC50 > 10000 nM T23276 CVN83J 656950 IC50 > 10000 nM T23276 CDK3J0 5703619 IC50 = 1146 nM T23276 C5AL8S 6445230 EC50 = 0.55 nM T23276 CPQ13K 9933545 IC50 > 100000000 nM T23276 C0V7UW 9958506 IC50 > 11000 nM T23276 C2W3AV 9995236 IC50 > 100000 nM T23276 CV8TY1 9996476 IC50 > 10000 nM T23276 CUY0F8 10005715 IC50 > 10000 nM T23276 CF1D6Y 10075240 IC50 > 10000 nM T23276 CPS9U3 10319232 IC50 > 10000 nM T23276 CLX54H 11317348 IC50 > 10000 nM T23276 C0APW4 11422034 IC50 > 10000 nM T23276 CTG83F 11539329 Ki > 9200 nM T23276 CMIL86 11590363 Ki > 9200 nM T23276 C9T6SC 11640926 Ki > 9200 nM T23276 CJ9KN7 11683817 IC50 > 10000 nM T23276 CU0E8O 11690457 Ki > 2900 nM T23276 CB0AP2 11705863 Ki > 10000 nM T23276 CVC2S4 11722798 IC50 > 10000 nM T23276 CHR92S 11858109 IC50 > 100000 nM T23276 C7LB4I 15949613 IC50 > 10000 nM T23276 CZK8V6 16043304 IC50 = 400 nM T23276 C9TU1O 16046126 IC50 > 1000 nM T23276 CGC34R 16118737 IC50 > 100000 nM T23276 C9BI2Y 23060924 IC50 > 1100 nM T23276 C2NLE3 23060985 IC50 > 1100 nM T23276 CE7K3W 23532567 IC50 > 10000 nM T23276 CQNP54 24764449 IC50 = 100000 nM T23276 C4Z9CN 24769780 IC50 > 100000 nM T23276 CS3Q8B 24995659 IC50 > 2000 nM T23276 CTV54O 25123227 IC50 > 10000 nM T23276 C6FGQ1 25206346 IC50 > 10000 nM T23276 CU9E4P 42629114 IC50 > 10000 nM T23276 CEL61X 44229839 IC50 > 10000 nM T23276 CYE36B 44241613 IC50 > 40000 nM T23276 C6LG5T 44241614 IC50 > 40000 nM T23276 C7PRE3 44315929 IC50 = 90000 nM T23276 CUY8A3 44401410 IC50 = 300 nM T23276 C8L5ZH 44401437 IC50 > 1000 nM T23276 CIB5V1 44401506 IC50 = 750 nM T23276 C5C3BG 44401556 IC50 > 1000 nM T23276 CH0CT1 44451687 IC50 > 1100 nM T23276 C5MQX7 44451688 IC50 > 1100 nM T23276 C8K5LD 44451690 IC50 > 1100 nM T23276 C0HY3S 44451713 IC50 > 1100 nM T23276 C3VRO9 44557921 IC50 > 10000 nM T23276 C87FEM 45270051 IC50 > 40000 nM T23276 CU53FK 45273505 IC50 > 40000 nM T23276 CMB32E 46203864 IC50 = 980 nM T23276 CUA97D 46209401 IC50 > 10000 nM T23276 C60GAV 46929544 IC50 > 8000 nM T23276 CP34VL 46929748 IC50 > 1000 nM T23276 CJ2E9Q 46929857 IC50 > 25000 nM T23276 CB0S2P 49842666 IC50 > 100000 nM T23276 CAI20B 49842778 IC50 > 100000 nM T23276 CD2K4R 50908681 Ki > 1000000 nM T23276 COVJ29 50994971 IC50 = 4800 nM T23276 CEQN27 52936621 Ki > 2000 nM T23276 CD4H3S 53354074 Ki > 1000 nM T23276 C8NA4L 53384644 IC50 > 30000 nM T23276 CM8JX1 56604907 IC50 = 25000 nM T23276 CN96GA 57685722 IC50 = 207 nM T23276 CRZY38 57686268 IC50 = 25 nM T23276 CPVO76 57686351 IC50 = 43 nM T23276 CP2B1Q 57686448 IC50 = 41 nM T23276 CI19SK 57686585 IC50 = 135 nM T23276 C2ZUY5 58282827 IC50 = 7.9 nM T23276 C8MBE7 58282833 IC50 = 74 nM T23276 C1MR8Q 60097495 IC50 > 10000 nM T23276 CV63UL 67240318 IC50 > 10000 nM T23276 C1IEJ2 70789254 IC50 = 60000 nM T23276 C8T7ZP 70789255 IC50 = 37000 nM T23276 CEBO91 71452977 IC50 > 10000 nM T23276 CHQZ25 71459584 IC50 > 10000 nM T23276 CZ31PU 71583657 IC50 > 10000 nM T23276 CV4HO3 71726759 IC50 = 1070 nM T23276 C35NLY 71726760 IC50 = 150 nM T23276 C6NVW2 71726764 IC50 = 510 nM T23276 CIN10C 71727133 IC50 = 2.7 nM T23276 COI5S0 71727368 IC50 = 3.9 nM T23276 CV2CR0 71727369 IC50 = 13 nM T23276 C2XZW3 72708899 IC50 > 40000 nM T23276 CKN46T 72708901 IC50 > 40000 nM T23276 CJ2T9E 76332983 IC50 > 10000 nM T23276 C6ZSG5 84973107 IC50 = 20 nM T23276 C5VA2J 84973109 IC50 = 18 nM T23276 CP0WM3 86696674 IC50 = 7.9 nM T23276 C1O0BS 89794860 IC50 = 85 nM T23276 C54NBM 89795059 IC50 = 27 nM T23276 CYLX17 89795073 IC50 = 62 nM T23276 CO1UM8 89795095 IC50 = 9610 nM T23276 CPHT17 89795256 IC50 = 19 nM T23276 C6KBW4 89795275 IC50 = 26 nM T23276 CW5O1N 89795280 IC50 = 550 nM T23276 C15FCX 89795282 IC50 = 74 nM T23276 CN4VB6 89795308 IC50 = 3.8 nM T23276 CSK8C3 89807688 IC50 = 5 nM T23276 C6GME9 89807821 IC50 = 43 nM T23276 C0Y8ZK 91933875 IC50 > 1000 nM T23276 C2TSV7 122177851 IC50 = 65 nM T23276 CEK9S7 122177852 IC50 = 43 nM T23276 C40APN 122177853 IC50 = 20 nM T23276 CCN6F5 122177854 IC50 = 25 nM T23276 CE68SL 122177855 IC50 = 46 nM T23276 CSFJ19 122177913 IC50 = 57 nM T23276 C53NSH 122177914 IC50 = 76 nM T23276 CJD03F 122177915 IC50 = 87 nM T23276 CX8JI0 122177916 IC50 = 89 nM T23276 CJI3N8 122177917 IC50 = 95 nM T23276 CJHF98 122177918 IC50 = 23 nM T23276 CU15EY 122177919 IC50 = 32 nM T23276 CGDL13 122177920 IC50 = 89 nM T23276 CVE19K 122177921 IC50 = 23 nM T23276 CB1HF0 122177922 IC50 = 43 nM T23276 CER2Y0 122177923 IC50 = 21 nM T23276 COQ7U6 122177924 IC50 = 23 nM T23276 CV1A2F 122177925 IC50 = 24 nM T23276 CJ6RM1 122177926 IC50 = 35 nM T23276 CC13JY 122177927 IC50 = 47 nM T23276 CWM37L 123897305 IC50 = 3100 nM T23276 CQ1V6G 127045826 IC50 = 16.7 nM T23276 C6KL7C 127045928 IC50 = 74.2 nM T23276 CHK16Q 127045929 IC50 = 154 nM T23276 CF4XM2 127045932 IC50 = 78.7 nM T23276 CC9FG2 127045933 IC50 = 26.3 nM T23276 CBQ2N5 127046246 IC50 = 833 nM T23276 CLM41O 127046585 IC50 = 19.4 nM T23276 CO6Q4N 127047015 IC50 = 35.9 nM T23276 CTCR73 127047016 IC50 = 46.3 nM T23276 C6AVN3 127047018 IC50 = 29.2 nM T23276 CLG53I 127047019 IC50 = 72.4 nM T23276 CK49NV 127047027 IC50 = 53.4 nM T23276 C3WGY8 127047160 IC50 = 38.7 nM T23276 CZ3NX1 127047176 IC50 = 66.9 nM T23276 CG89KZ 127047589 IC50 = 55.5 nM T23276 CLO6T3 127047590 IC50 = 26.4 nM T23276 CY3J0C 127047591 IC50 = 29.3 nM T23276 CKQ9P4 127047724 IC50 = 22.2 nM T23276 CO6DK5 127047745 IC50 = 106 nM T23276 C0FM1R 130196825 IC50 = 13545 nM T23276 C7PS8C 135271570 IC50 = 6900 nM T23276 CG67XB 137210065 IC50 = 111 nM T23276 C0CV4B 137210066 IC50 = 32.3 nM T23276 C3FC1W 137631894 IC50 > 10000 nM T23276 C10BTW 137632556 IC50 > 10000 nM T23276 C2J9GO 137633617 IC50 > 10000 nM T23276 C7MD0H 137635615 IC50 = 790 nM T23276 CML76T 137635976 IC50 > 10000 nM T23276 CS9AW4 137636754 IC50 = 7600 nM T23276 C7R0MS 137638615 IC50 > 10000 nM T23276 CGR5B1 137642299 IC50 = 8700 nM T23276 C26HIT 137643417 IC50 > 10000 nM T23276 CDA2N6 137644922 IC50 = 278 nM T23276 CAT49C 137645403 IC50 > 10000 nM T23276 CUES49 137646218 IC50 > 10000 nM T23276 CS6J8X 137646633 IC50 > 10000 nM T23276 C9Z6NB 137646838 IC50 = 5200 nM T23276 C2HFR6 137648529 IC50 > 10000 nM T23276 CYR2I7 137649411 IC50 > 10000 nM T23276 C17GBS 137649678 IC50 > 10000 nM T23276 CEO70C 137650358 IC50 > 10000 nM T23276 C4NM0R 137650776 IC50 > 10000 nM T23276 CL3P8Q 137653011 IC50 = 7300 nM T23276 C5B9AM 137653362 IC50 = 8300 nM T23276 C8K0OY 137655533 IC50 > 10000 nM T23276 C83XOY 137657177 IC50 = 1620 nM T23276 CF7U5Y 137657487 IC50 > 10000 nM T23276 C3SD7B 137658277 IC50 > 10000 nM T23276 CVY3F0 137658568 IC50 > 10000 nM T23276 CJK81S 137659431 IC50 = 4700 nM T23276 CUS48N 137659983 IC50 > 10000 nM T23276 C6VB3O 145925651 IC50 >= 5000 nM T23276 C5TS1A 145964021 IC50 = 93 nM T23276 C8QAU0 145965069 IC50 = 952 nM T23276 CQJP12 145968722 IC50 = 45 nM T23276 CD7X3A 145969845 IC50 = 228 nM T23276 CG01BZ 145973754 IC50 = 34 nM T23276 C6X8PU 145975686 IC50 = 19 nM T23276 C28XFL 145977776 IC50 = 663 nM T23276 C2FA4R 145978301 IC50 = 17 nM T23276 CHIB04 146634736 IC50 = 21 nM T23276 C3MR9I 146634737 IC50 = 3.6 nM T23276 C6Q3UP 146634739 IC50 = 1.5 nM T23276 CX76AZ 146634741 IC50 = 4.1 nM T23276 C10WET 148308905 IC50 = 3.3 nM T23276 C86HPW 155518524 IC50 = 65000 nM T23276 D00HVA 11624601 Ki > 9200 nM T23276 D01MNK 25125014 IC50 = 3730 nM T23276 D02XHC 448912 IC50 = 18000 nM T23276 D04PEI 11467730 IC50 > 50000 nM T23276 D07OAT 456214 IC50 = 9000 nM T23276 D07OXC 11650194 IC50 > 100000 nM T23276 D08XVZ 24866313 IC50 = 4 nM T23276 D09RYV 9911652 IC50 > 100000000 nM T23276 D0OZ2S 11785878 IC50 > 100000 nM T23276 D0Q3NG 11715520 Ki > 9200 nM T23276 D0S7IE 11658882 Ki > 9200 nM T23276 D0UN9O 3385203 IC50 >= 10000 nM T23276 D0V0QJ 389898 IC50 = 82900 nM T23276 D0ZG4G 11493598 Ki = 310 nM T85616 D04JTD 219104 IC50 = 2110 nM T85616 CI7MW0 9852185 Ki = 3110 nM T85616 C5DL2O 15335087 IC50 = 510 nM T85616 C6W2MC 71487261 IC50 = 340 nM T85616 CB52OT 71487263 IC50 = 7310 nM T85616 CJC7Y6 71562811 IC50 = 170 nM T85616 CM1VW2 71562812 IC50 = 90 nM T85616 CG3U8R 71562814 IC50 = 240 nM T85616 C6VPK1 71562930 IC50 = 450 nM T85616 CU35ZW 71562931 IC50 = 540 nM T85616 CBM95V 136240922 IC50 = 290 nM T81503 D0Q0PR 54675769 IC50 = 154 nM T81503 CLQ19N 54695811 IC50 = 43 nM T81503 CJ4Q5C 54695812 IC50 = 137 nM T81503 CN2LR7 54695813 IC50 = 276 nM T81503 CWGP52 54697399 IC50 = 75 nM T81503 CWL92P 54708659 IC50 = 22 nM T81503 C0QL6P 54713406 IC50 = 891 nM T81503 C50NPL 54721832 IC50 = 131 nM T81503 C94HJN 54729434 IC50 > 10000 nM T81503 CNQI70 54729435 IC50 = 17 nM T81503 CK9Q2M 54729436 IC50 = 86 nM T81503 C6ECK7 54729437 IC50 = 219 nM T81503 CU04CO 54729438 IC50 = 140 nM T81503 C0T2FR 54729439 IC50 = 190 nM T81503 C9F2HC 54729448 IC50 > 10000 nM T81503 CG90ET 54729449 IC50 > 10000 nM T81503 CI78JU 54729450 IC50 = 20 nM T81503 C30HTF 54729451 IC50 = 116 nM T81503 CFWS93 54729452 IC50 = 110 nM T81503 CEA05G 54730369 IC50 = 34 nM T81503 CI1SU0 54730370 IC50 = 280 nM T81503 CIE25B 54730375 IC50 > 10000 nM T81503 C8ZM7I 54730379 IC50 = 41 nM T81503 C1E4WO 54730380 IC50 = 106 nM T81503 C73YWX 54730381 IC50 = 320 nM T81503 C6C1KM 54730382 IC50 = 598 nM T81503 CD2P1F 54732401 IC50 < 5 nM T81503 CMIN96 54732402 IC50 = 44 nM T81503 CR9TB4 54732403 IC50 = 460 nM T81503 CG92WX 54732408 IC50 > 10000 nM T81503 C4GHD2 54732409 IC50 = 19 nM T81503 CHGE48 54732410 IC50 = 120 nM T81503 D0C9BH 54706138 IC50 < 5 nM T33492 D04NDM 165580 IC50 = 21000000 nM T33492 D05JNI 8378 IC50 = 8000000 nM T33492 D07JZF 441306 IC50 = 8000000 nM T33492 D0GZ7B 5328779 IC50 > 333000 nM T33492 CI26AQ 1607 IC50 = 360 nM T33492 C5IF7O 2259 IC50 = 12 nM T33492 CW68ZS 61672 IC50 = 4000 nM T33492 CYTJ80 78402 IC50 > 10000 nM T33492 CH67EZ 91286 IC50 > 111000 nM T33492 C0O3TQ 126437 IC50 = 1230 nM T33492 CH6PG4 203854 IC50 > 10000 nM T33492 CZTD26 220436 IC50 > 111000 nM T33492 C80UDV 334474 IC50 > 111000 nM T33492 CS2B8E 397888 IC50 = 12000 nM T33492 CESM72 439530 IC50 = 18000000 nM T33492 C0KE3R 442614 IC50 > 100000 nM T33492 CX9UA1 443385 IC50 = 9100000 nM T33492 CX8VI4 561354 IC50 = 9170 nM T33492 C34CEH 676561 IC50 = 710 nM T33492 C2Z0SV 685482 IC50 > 333000 nM T33492 CAPG06 726820 IC50 > 333000 nM T33492 C9NYF1 728520 IC50 = 5280 nM T33492 CF32MI 766914 IC50 > 333000 nM T33492 CE10WO 776842 IC50 = 110 nM T33492 C18SJQ 885337 IC50 > 10000 nM T33492 C2P9DB 1005270 IC50 > 15000 nM T33492 C47QWD 1025279 IC50 = 1000 nM T33492 C13SDI 1115047 IC50 = 500 nM T33492 CSO84U 1188215 IC50 > 10000 nM T33492 CBG3X5 1236521 IC50 = 40000 nM T33492 C2REL7 1239884 IC50 > 333000 nM T33492 C0SKV6 1325590 IC50 > 10000 nM T33492 CIZ70U 1325673 IC50 > 10000 nM T33492 CLA9J7 1540149 IC50 = 34000 nM T33492 CU5PF6 1652110 IC50 > 333000 nM T33492 CRL05A 1771058 IC50 = 7700 nM T33492 CP31XF 2030903 IC50 = 4930 nM T33492 C8WS4M 2040507 IC50 > 10000 nM T33492 CQI6S5 2243892 IC50 = 111000 nM T33492 C80CJH 2441756 IC50 = 14130 nM T33492 CAT8Q3 3000500 IC50 = 8000000 nM T33492 CI34YK 3121217 IC50 = 5620 nM T33492 C4N0CE 5328793 IC50 > 333000 nM T33492 C48BJI 5336179 IC50 = 1080 nM T33492 C3YD4V 5351985 IC50 = 14000 nM T33492 CX30RB 5411062 IC50 > 333000 nM T33492 CO01XP 5478021 IC50 > 111000 nM T33492 C26DVM 6211778 IC50 > 333000 nM T33492 C5PT6B 6245483 IC50 > 111000 nM T33492 CO6J1X 6304702 IC50 = 12000 nM T33492 C2MZ9A 7083198 IC50 = 950 nM T33492 CL6Z8O 7454864 IC50 = 19000 nM T33492 C6XP2L 9139208 IC50 = 35480 nM T33492 CO5Q7F 10338255 IC50 = 22300 nM T33492 CRBZ37 10494779 IC50 > 111000 nM T33492 C0YD4S 10640393 IC50 > 111000 nM T33492 CG07YZ 10663416 IC50 > 111000 nM T33492 CIO2Y3 11220435 Ki = 3190 nM T33492 C5F6NY 11370831 IC50 = 55300 nM T33492 CBU10H 11520588 IC50 = 1000 nM T33492 CRS8D5 12525013 IC50 = 30000 nM T33492 CT91GZ 16098813 IC50 = 5800 nM T33492 CKZ5B8 16098830 IC50 = 1000 nM T33492 CV8TP1 16221202 IC50 = 17500 nM T33492 CJ32LD 16221204 IC50 = 31000 nM T33492 CFD49E 16221206 IC50 = 47000 nM T33492 C17EIS 16221208 IC50 = 14100 nM T33492 C1MRB8 16221210 IC50 = 33000 nM T33492 CT32AS 16221263 IC50 = 25000 nM T33492 C67THG 16221322 IC50 = 48000 nM T33492 CIW39K 16221324 IC50 = 14100 nM T33492 CO42ZD 16434867 IC50 = 50120 nM T33492 CE0Q5Z 17390511 IC50 = 44000 nM T33492 CX30ZC 17756086 IC50 = 37000 nM T33492 C4KUW5 18230892 IC50 = 79430 nM T33492 C2RSJ0 41587290 IC50 = 11220 nM T33492 C7UM4C 42630956 IC50 = 27000 nM T33492 CD97JI 42915055 IC50 = 44670 nM T33492 CZQN61 44574209 IC50 = 1800000 nM T33492 CF48PX 45353287 IC50 = 44670 nM T33492 C9VHP4 46229345 IC50 = 35000 nM T33492 C92NHR 46229346 IC50 = 5000 nM T33492 CCM26J 56837840 IC50 > 111000 nM T33492 CPA1M7 57521375 IC50 > 111000 nM T33492 C98GSX 57521376 IC50 > 111000 nM T33492 C6UIY2 57521377 IC50 > 111000 nM T33492 C3V0GK 57521378 IC50 > 111000 nM T33492 CX82UH 57521379 IC50 > 111000 nM T33492 C13AUV 57521485 IC50 > 111000 nM T33492 CRZ52K 57521486 IC50 > 111000 nM T33492 C0UT7F 57521488 IC50 > 111000 nM T33492 C7ID1U 57521489 IC50 > 111000 nM T33492 CQK0F8 57521585 IC50 > 111000 nM T33492 CM8VZ1 57521586 IC50 > 111000 nM T33492 C13XAL 57521587 IC50 > 111000 nM T33492 C9HV4M 57521588 IC50 > 111000 nM T33492 C3U9EO 57521589 IC50 > 111000 nM T33492 CN72YQ 57521691 IC50 > 111000 nM T33492 C3AXR7 57521692 IC50 > 111000 nM T33492 C4FIE9 57521693 IC50 > 111000 nM T33492 CR38GS 57521694 IC50 > 111000 nM T33492 C6CUL8 57521695 IC50 > 111000 nM T33492 CJ6Z3M 57521803 IC50 > 111000 nM T33492 CG5YJ9 57521804 IC50 > 111000 nM T33492 C5E6VB 57521805 IC50 > 111000 nM T33492 CB1E5V 57521806 IC50 > 111000 nM T33492 C1L0TI 57521807 IC50 > 111000 nM T33492 CP36UT 57521909 IC50 > 111000 nM T33492 C4HP8U 57521910 IC50 > 111000 nM T33492 CQV97O 57521911 IC50 > 111000 nM T33492 CYO01C 57521912 IC50 > 111000 nM T33492 C7VBQ4 57522032 IC50 > 111000 nM T33492 C8J3FI 57522033 IC50 > 111000 nM T33492 CB3L2W 57522034 IC50 > 111000 nM T33492 CTO5S8 57522035 IC50 > 111000 nM T33492 CTRX83 57522599 IC50 > 111000 nM T33492 CRP57E 57522600 IC50 > 111000 nM T33492 CQUG46 57522601 IC50 > 111000 nM T33492 CIJ19L 57522602 IC50 > 111000 nM T33492 C6DC1K 57522711 IC50 > 111000 nM T33492 CB9OC3 57522712 IC50 > 111000 nM T33492 CN7Q3O 57522716 IC50 > 111000 nM T33492 CP2LO3 57522717 IC50 > 111000 nM T33492 CUA7L4 57522821 IC50 > 111000 nM T33492 CW31RU 57522822 IC50 > 111000 nM T33492 CPOR59 57522823 IC50 > 111000 nM T33492 CJA90N 57522824 IC50 > 111000 nM T33492 CBSY92 57522825 IC50 > 111000 nM T33492 C0QLK6 57522826 IC50 > 111000 nM T33492 C3BI1S 57522959 IC50 > 111000 nM T33492 CNF76K 57522960 IC50 > 111000 nM T33492 CWL8R4 57522961 IC50 > 111000 nM T33492 CIL52C 57522962 IC50 > 111000 nM T33492 C09IFB 57522963 IC50 > 111000 nM T33492 CTP92I 57522964 IC50 > 111000 nM T33492 CQ97US 57523098 IC50 > 111000 nM T33492 CQ82LU 57523099 IC50 > 111000 nM T33492 C08FVX 57523100 IC50 > 111000 nM T33492 C5CQT0 57523101 IC50 > 111000 nM T33492 CAF3X4 57523102 IC50 > 111000 nM T33492 C6AZ0X 60148508 IC50 = 12000 nM T33492 CO4P2S 60148514 IC50 = 37000 nM T33492 CH95XR 60165808 IC50 = 18000 nM T33492 C1Q7GJ 60165957 IC50 > 111000 nM T33492 CQZ2N7 60165960 IC50 > 111000 nM T33492 CMW7P2 60165963 IC50 > 111000 nM T33492 CHW9Y7 60166112 IC50 > 111000 nM T33492 CNF46Y 66489030 IC50 = 26000 nM T33492 CB6A5C 70674149 IC50 > 10000 nM T33492 CXAT75 70690590 IC50 > 111000 nM T33492 CWU83Q 70696734 IC50 > 111000 nM T33492 C9M8FA 71449815 IC50 > 333000 nM T33492 CA71WP 71450009 IC50 = 37000 nM T33492 C5VT8U 71451618 IC50 = 11000 nM T33492 CHW4O9 71451620 IC50 = 15000 nM T33492 CX6JV8 71451621 IC50 = 46000 nM T33492 CYI5H3 71451622 IC50 = 20000 nM T33492 CJ68NX 71451623 IC50 = 69000 nM T33492 CP3FA6 71451624 IC50 = 74000 nM T33492 C9CUO8 71452527 IC50 = 1620 nM T33492 CAJ47F 71452528 IC50 = 260 nM T33492 CHD2O4 71453458 IC50 = 8500 nM T33492 CJ83PN 71453459 IC50 = 138000 nM T33492 C69BNH 71453460 IC50 = 13000 nM T33492 CXM5V1 71453461 IC50 > 333000 nM T33492 CI6O5J 71453649 IC50 > 111000 nM T33492 C51XKH 71454291 IC50 = 1540 nM T33492 C4TWY0 71455170 IC50 = 75000 nM T33492 C34SCA 71456960 IC50 = 6900 nM T33492 C7FPV4 71456961 IC50 = 34000 nM T33492 C4VO0K 71456962 IC50 > 333000 nM T33492 CZ3K8E 71457146 IC50 > 111000 nM T33492 CN4CR6 71458831 IC50 = 51000 nM T33492 CCLK82 71458832 IC50 = 111000 nM T33492 CX9SE4 71460811 IC50 > 111000 nM T33492 CRT0H9 71461477 IC50 = 940 nM T33492 C1H3AJ 71461478 IC50 = 1810 nM T33492 CHCX75 71461479 IC50 = 570 nM T33492 CIM47J 71462348 IC50 = 38000 nM T33492 C9D6YL 71462349 IC50 = 28000 nM T33492 CBHZ04 71462352 IC50 = 29000 nM T33492 C04MQY 71544698 IC50 > 111000 nM T33492 CXY45D 71544701 IC50 > 111000 nM T33492 C6SZ7F 71544702 IC50 > 111000 nM T33492 C3ARJ0 71544866 IC50 = 12000 nM T33492 CBOR04 71544868 IC50 > 111000 nM T33492 CG3VH5 71545025 IC50 = 5200 nM T33492 C7KLX0 71545027 IC50 = 6700 nM T33492 CZ7NG2 71546175 IC50 > 111000 nM T33492 CEM9V0 71546176 IC50 > 111000 nM T33492 CS7ZY0 71546177 IC50 > 111000 nM T33492 CKJ42V 71546178 IC50 > 111000 nM T33492 C9JI8X 71546179 IC50 > 111000 nM T33492 CA49VP 71546347 IC50 = 61000 nM T33492 C7R0VX 71546348 IC50 > 111000 nM T33492 C7NIU6 71546350 IC50 > 111000 nM T33492 CTA72F 71546351 IC50 > 111000 nM T33492 C3B2LW 71546514 IC50 > 111000 nM T33492 C4WZ3O 71546516 IC50 = 45000 nM T33492 CYL3F6 71546517 IC50 = 18000 nM T33492 CTI3N1 71546518 IC50 = 37000 nM T33492 CK0C3J 71546671 IC50 = 37000 nM T33492 CZ49YE 71546672 IC50 = 37000 nM T33492 CH46SD 71546675 IC50 = 37000 nM T33492 C1Z0GN 71546826 IC50 > 111000 nM T33492 CDA9V1 71546829 IC50 > 111000 nM T33492 C1VIY2 71546831 IC50 > 111000 nM T33492 C9Q4YR 71546833 IC50 > 111000 nM T33492 C3Y9MP 71546979 IC50 > 111000 nM T33492 C41YVT 71546981 IC50 > 111000 nM T33492 C28KSH 71546982 IC50 > 111000 nM T33492 C4MSG0 71546985 IC50 = 11000 nM T33492 C7U1WD 71546986 IC50 > 111000 nM T33492 C1O5HY 71547124 IC50 > 111000 nM T33492 C7VJN5 71547126 IC50 = 5000 nM T33492 C3GPU9 71547128 IC50 > 111000 nM T33492 CO38NF 71547129 IC50 > 111000 nM T33492 C9Q4DA 71547131 IC50 = 15000 nM T33492 CVS84W 71582100 IC50 = 3800 nM T33492 C94DIL 73334714 IC50 > 111000 nM T33492 CRZ62F 73355036 IC50 = 5000 nM T33492 CMU46W 76029213 IC50 > 111000 nM T33492 CA4F7D 76311078 IC50 > 111000 nM T33492 C40TDU 76311079 IC50 > 111000 nM T33492 CF08AN 76311080 IC50 > 111000 nM T33492 CT05OM 76311081 IC50 = 37000 nM T33492 C24IZB 76311082 IC50 = 12000 nM T33492 CC84YZ 76314698 IC50 = 37000 nM T33492 CTQW89 76314699 IC50 > 111000 nM T33492 CVN17S 76318268 IC50 > 111000 nM T33492 C32WVQ 76318269 IC50 > 111000 nM T33492 C9KN5G 76318270 IC50 = 37000 nM T33492 C9Y0MW 76321973 IC50 > 111000 nM T33492 CF24IO 76321974 IC50 > 111000 nM T33492 C8NP5E 76329155 IC50 > 111000 nM T33492 CE8A1M 76329156 IC50 = 37000 nM T33492 C8WB7V 76332814 IC50 > 111000 nM T33492 CL3QN6 76332815 IC50 = 37000 nM T33492 CJSL58 76332816 IC50 = 12000 nM T33492 C3D6MK 76336438 IC50 = 37000 nM T33492 CB6YU7 86291808 IC50 = 5500 nM T33492 C6JV2S 86765191 IC50 = 12000 nM T33492 CQU1J7 86765192 IC50 = 12000 nM T33492 C30VXB 86765193 IC50 > 111000 nM T33492 CK1Y4C 86765194 IC50 = 12000 nM T33492 CN64AH 86765195 IC50 = 1000 nM T33492 C9NV1H 86765208 IC50 > 111000 nM T33492 CT6YB9 90643550 IC50 > 111000 nM T33492 C3LS5W 90643551 IC50 > 111000 nM T33492 CDQG63 90643552 IC50 > 111000 nM T33492 CH25QC 90643553 IC50 = 37000 nM T33492 C8QC2J 110206286 IC50 = 790 nM T33492 C4WE5F 110207923 IC50 = 1530 nM T33492 CUVY69 118070452 IC50 = 37000 nM T33492 CG94AY 118070454 IC50 = 12000 nM T33492 CFQ3A4 118721722 IC50 = 390 nM T33492 C5M8NJ 118721723 IC50 = 150 nM T33492 CFP6G9 118721724 IC50 = 810 nM T33492 C3ZOW1 118721725 IC50 = 450 nM T33492 C9JEB8 118727325 IC50 > 10000 nM T33492 CVL96K 118728738 IC50 = 3700 nM T33492 CVWY39 118728739 IC50 = 1280 nM T33492 CC42ZN 118728740 IC50 = 1620 nM T33492 C8N0QE 118728741 IC50 = 220 nM T33492 CNH9E7 118728742 IC50 = 6030 nM T33492 C65CJL 118728743 IC50 = 3660 nM T33492 CK2C9Z 118728744 IC50 = 1300 nM T33492 CJ3C4L 118735563 IC50 > 111000 nM T33492 CBZF47 118735565 IC50 > 111000 nM T33492 CUN56B 118735568 IC50 > 111000 nM T33492 CQC6B9 118735570 IC50 = 12000 nM T33492 CYIM15 118735572 IC50 = 12000 nM T33492 C6GZL3 118735573 IC50 > 111000 nM T33492 CCA73K 118735574 IC50 > 111000 nM T33492 CTN0Y6 118735576 IC50 = 12000 nM T33492 CDC9A2 118735578 IC50 > 111000 nM T33492 CXB0R3 118735580 IC50 > 111000 nM T33492 CP1W7A 118735582 IC50 = 1000 nM T33492 C46INW 118735583 IC50 > 111000 nM T33492 CXJG20 118735584 IC50 > 111000 nM T33492 CGN27Z 118735585 IC50 = 37000 nM T33492 CFKO57 118735587 IC50 > 111000 nM T33492 CR7UK8 118735588 IC50 > 111000 nM T33492 CU0KP6 118735590 IC50 = 12000 nM T33492 CH30JX 121478365 IC50 = 38000 nM T33492 CT1RL3 122179149 IC50 > 111000 nM T33492 CM9AU7 122179162 IC50 > 111000 nM T33492 C98KOJ 122179163 IC50 = 63000 nM T33492 C7Q9FC 122179164 IC50 > 111000 nM T33492 CY2Q4V 122181724 IC50 = 1000 nM T33492 CK91CX 122181725 IC50 = 1000 nM T33492 CG3O5N 122483604 IC50 > 111000 nM T33492 C7BL9T 122484905 IC50 = 6200 nM T33492 C3FS6Y 122484906 IC50 = 6300 nM T33492 CS1DF2 127025946 IC50 = 1700 nM T33492 CG8BR2 127028127 IC50 = 2200 nM T33492 CLT35C 127043728 IC50 > 111000 nM T33492 CJA2I1 127044083 IC50 = 63000 nM T33492 CBFS34 127044239 IC50 > 111000 nM T33492 CE15TB 127044402 IC50 > 111000 nM T33492 CF64IU 127044403 IC50 > 111000 nM T33492 C12IUQ 127044404 IC50 = 90000 nM T33492 CBE49O 127044405 IC50 > 111000 nM T33492 CM19WU 127044406 IC50 = 19000 nM T33492 CU15SD 127044408 IC50 > 111000 nM T33492 C0X5YU 127044409 IC50 = 30000 nM T33492 C3XO0J 127044411 IC50 > 111000 nM T33492 COX07F 127044412 IC50 = 111000 nM T33492 C5OQ3T 127044413 IC50 > 111000 nM T33492 C38YZG 127044414 IC50 > 60000 nM T33492 C0SP4E 127044557 IC50 = 43000 nM T33492 CPEU65 127044559 IC50 > 111000 nM T33492 C1W8YR 127044560 IC50 > 111000 nM T33492 C4ZI7L 129751977 IC50 = 1010 nM T33492 C8TM2K 129881957 IC50 = 190 nM T33492 CP7E6T 129881996 IC50 = 160 nM T33492 C72SJL 129883811 IC50 = 4100 nM T33492 C0C7LT 129883861 IC50 = 1250 nM T33492 CYI8M7 129883900 IC50 = 1210 nM T33492 C6X7VK 129883904 IC50 = 610 nM T33492 CRK13E 129883976 IC50 = 1120 nM T33492 CVE65K 129884019 IC50 = 5900 nM T33492 C9L1GO 129896914 IC50 = 1000 nM T33492 C2BV6U 132577626 IC50 = 1390 nM T33492 C6JL5C 132577627 IC50 = 1920 nM T33492 C6DQL0 132577629 IC50 = 750 nM T33492 C94PEK 134132337 IC50 = 675 nM T33492 C1BN0D 134135136 IC50 = 4310 nM T33492 CU50NE 134138761 IC50 = 1230 nM T33492 C3AJ4Y 134140308 IC50 = 1200 nM T33492 C4W5YX 134140937 IC50 = 1370 nM T33492 CVH14W 134142079 IC50 = 1450 nM T33492 C9KZI1 134150902 IC50 = 1560 nM T33492 CE49RL 134156830 IC50 = 1090 nM T33492 C5DA0Z 135163962 IC50 = 12000 nM T33492 CC57MQ 135400994 IC50 = 18000 nM T33492 C7PO0L 135541470 IC50 > 111000 nM T33492 CS8HM5 135815232 IC50 = 11000 nM T33492 C1R7MT 135875770 IC50 = 111000 nM T33492 CVR0T7 136236290 IC50 = 48000 nM T33492 CTG7U8 136236291 IC50 = 39000 nM T33492 C5K9YU 136236292 IC50 = 35000 nM T33492 CLEM70 136236293 IC50 = 7100 nM T33492 C04RXQ 136236294 IC50 = 4100 nM T33492 CEBA65 136236295 IC50 = 220000 nM T33492 CN0VR1 136236296 IC50 = 12000 nM T33492 CF7M6P 136236297 IC50 = 2600 nM T33492 C8EZC7 136236298 IC50 = 111000 nM T33492 CR31TD 136236299 IC50 = 111000 nM T33492 CNIM68 136236300 IC50 = 32000 nM T33492 CQZ79S 137633472 IC50 > 111000 nM T33492 CEMW84 137634763 IC50 = 1000 nM T33492 CY83RB 137635101 IC50 > 111000 nM T33492 CY4BH7 137635982 IC50 = 12000 nM T33492 CP8I0N 137635992 IC50 > 111000 nM T33492 CC1X7N 137637372 IC50 = 33300 nM T33492 CSKE17 137638583 IC50 = 27500 nM T33492 C7K5XB 137638718 IC50 > 111000 nM T33492 CY0G2M 137639745 IC50 = 11900 nM T33492 CE93VQ 137639878 IC50 > 111000 nM T33492 C7KVT8 137640123 IC50 = 1000 nM T33492 CT5YB3 137641552 IC50 > 100000 nM T33492 C7EHL1 137643195 IC50 > 111000 nM T33492 CQ89WF 137644721 IC50 = 20200 nM T33492 C7LY3U 137645346 IC50 = 14000 nM T33492 CT8A6V 137645479 IC50 = 1000 nM T33492 CTD0Q1 137645708 IC50 = 12000 nM T33492 C83FEH 137646143 IC50 > 111000 nM T33492 CR72BP 137646560 IC50 = 12000 nM T33492 CW24CA 137650951 IC50 = 16000 nM T33492 C2MP3A 137650968 IC50 = 1000 nM T33492 C2RVW9 137651075 IC50 = 22200 nM T33492 C7SUD6 137652086 IC50 > 111000 nM T33492 C9X2IG 137652438 IC50 > 111000 nM T33492 CY25WR 137653301 IC50 > 111000 nM T33492 CDQ41E 137656446 IC50 > 111000 nM T33492 CZX8J7 137658040 IC50 > 100000 nM T33492 CZ01OK 137658578 IC50 = 1000 nM T33492 CHXA46 137659333 IC50 = 12000 nM T33492 CB9GY3 137660083 IC50 > 111000 nM T33492 C09XQR 137661166 IC50 > 111000 nM T33492 CM78PY 138454772 IC50 = 7000 nM T33492 C6KZP1 139593958 IC50 = 63 nM T33492 C81WPC 139593986 IC50 = 26 nM T33492 CDU5H3 145949386 IC50 = 13000 nM T33492 CRS2C9 145949970 IC50 = 15000 nM T33492 CDM0W7 145951675 IC50 = 48000 nM T33492 CN16JZ 145951972 IC50 = 16000 nM T33492 CO8TH1 145954631 IC50 = 20000 nM T33492 CF90QJ 145956398 IC50 = 40000 nM T33492 C8Q5BD 145960258 IC50 = 20000 nM T33492 CK83GM 145982803 IC50 = 160 nM T33492 C2WO8C 145982960 IC50 = 630 nM T33492 CS9L5D 145983163 IC50 = 64 nM T33492 CE2A0Q 145983563 IC50 = 3300 nM T33492 C61ZPL 145983762 IC50 = 980 nM T33492 CVQ4G0 145983767 IC50 = 3650 nM T33492 C5M2JX 145983887 IC50 = 230 nM T33492 C7Z4HY 145984004 IC50 = 81 nM T33492 C7SE0X 145984229 IC50 = 600 nM T33492 CT8P1S 145984246 IC50 = 340 nM T33492 CE0N3L 145984315 IC50 = 6730 nM T33492 C5IJN8 145984662 IC50 = 720 nM T33492 C0W3ZP 145985218 IC50 = 1590 nM T33492 CF8U0M 145985434 IC50 = 860 nM T33492 C95TOG 145985558 IC50 = 900 nM T33492 CZVU04 145985759 IC50 > 15000 nM T33492 CA2R9X 145985836 IC50 = 340 nM T33492 CUJ6W5 145985887 IC50 = 840 nM T33492 C7FIS3 145985899 IC50 = 1220 nM T33492 CPI14D 145985918 IC50 = 530 nM T33492 C9E1BP 145985980 IC50 = 25 nM T33492 CX4R2M 145986039 IC50 = 232 nM T33492 CSV38F 145986188 IC50 = 1020 nM T33492 C7JP2N 151276071 IC50 = 100 nM T33492 CN5B4U 155510460 IC50 = 710 nM T33492 CCP8V7 155511883 IC50 = 90 nM T33492 CV69GT 155511965 IC50 = 192 nM T33492 C3PQ4I 155514436 IC50 = 68 nM T33492 CGT9M7 155514788 IC50 = 35 nM T33492 CTFA82 155515608 IC50 = 110 nM T33492 CZ2AH9 155518351 IC50 = 158 nM T33492 CF5NE1 155519048 IC50 = 34100 nM T33492 C3BZS7 155522234 IC50 = 3500 nM T33492 C1XC9R 155525490 IC50 = 12100 nM T33492 C2C8QK 155527697 IC50 = 500 nM T33492 CK4F1S 155530696 IC50 = 5 nM T33492 C9JQ5R 155532411 IC50 = 190 nM T33492 CP7IM4 155537726 IC50 = 150 nM T33492 C0T8MV 155547340 IC50 = 457 nM T33492 CR06HT 155549764 IC50 = 3700 nM T33492 C3RC9M 155551925 IC50 = 1490 nM T33492 C0F9WC 155554203 IC50 = 2300 nM T33492 CD5NV9 155555272 IC50 = 172 nM T33492 CZU1M4 155562716 IC50 = 22 nM T33492 C4LXT8 155564630 IC50 = 570 nM T33492 C9B1AO 155566616 IC50 = 86 nM T33492 D01NTW 5328768 IC50 > 333000 nM T33492 D02BUW 2061 IC50 > 333000 nM T33492 D07SQW 72394 IC50 = 30000000 nM T33492 D09KUE 259210 IC50 = 1000 nM T33492 D0Q3GG 667601 IC50 = 12000 nM T72881 D00QET 5281040 IC50 < 5000 nM T72881 D05MCS 44473151 IC50 = 36000 nM T72881 CUF65V 2261273 IC50 = 1900 nM T72881 C79DVG 56589615 IC50 > 3000 nM T72881 CU86FL 58034959 IC50 = 35 nM T72881 CW19CN 122670086 IC50 = 7.8 nM T72881 CO81KV 122670103 IC50 = 0.66 nM T72881 C86VYP 122670110 IC50 = 0.28 nM T72881 CK2B0J 138857937 IC50 = 2.4 nM T72881 CU95NM 145983649 IC50 = 6190 nM T72881 C76ACJ 145985137 IC50 = 30 nM T72881 CM62SF 145985303 IC50 = 15860 nM T72881 CN8G1X 145993375 IC50 = 1800 nM T72881 CS27OA 150767852 IC50 = 16 nM T72881 C0O7RL 155513699 IC50 = 8.65 nM T72881 CU56QS 155514039 IC50 = 7.9 nM T72881 C03QFT 155514291 IC50 = 27.4 nM T72881 CV7H9X 155514523 IC50 = 158 nM T72881 CGE90A 155515058 IC50 = 0.758 nM T72881 CL9QK7 155515277 IC50 = 27.7 nM T72881 CVI2D6 155518247 IC50 = 11.5 nM T72881 C3LC2H 155523754 IC50 = 1.41 nM T72881 C7XH4U 155525620 IC50 = 15.5 nM T72881 CRY0J2 155530520 IC50 = 0.381 nM T72881 CYB6A8 155531199 IC50 = 24.3 nM T72881 CC62BH 155532184 IC50 = 31.8 nM T72881 C15UYV 155532743 IC50 = 3.71 nM T72881 C3IXY0 155538051 IC50 = 1.05 nM T72881 C7O4TV 155543878 IC50 = 0.36 nM T72881 C3LK0J 155544798 IC50 = 6.42 nM T72881 CI6UZ9 155546599 IC50 = 13 nM T72881 C5VU2K 155550738 IC50 = 0.28 nM T72881 C6WCU9 155552988 IC50 = 1.97 nM T72881 CHI4B5 155553658 IC50 = 14 nM T72881 CIAY61 155553929 IC50 = 5.26 nM T72881 CZH04D 155559637 IC50 = 7.09 nM T72881 CXE0N3 155560141 IC50 = 109 nM T72881 CWYM30 155560185 IC50 = 157 nM T72881 C6K3MC 155564144 IC50 = 4.74 nM T72881 CBWQ63 155564396 IC50 = 8.5 nM T72881 C5QYB7 155565891 IC50 = 0.63 nM T30081 D01XYJ 35370 Ki = 2900 nM T30081 D03TGJ 5282192 IC50 > 500000 nM T30081 D07XSN 6253 IC50 > 1000000 nM T30081 D0Z8EX 18283 Ki = 580000 nM T30081 D06CCR 50313 Ki = 140 nM T30081 D0TJ9S 445212 Ki = 16100 nM T30081 D0Z9LP 446727 Ki = 100 nM T30081 CP25DX 65049 IC50 > 1000000 nM T30081 CD85ZQ 65159 Ki = 445000 nM T30081 CO4UY8 72230 Ki = 425000 nM T30081 CO15BF 72327 Ki = 180 nM T30081 CRM8J6 162419 IC50 = 14000 nM T30081 CVZ48I 174316 Ki = 90 nM T30081 CVDG62 452392 IC50 = 44000 nM T30081 CPJ56E 452395 IC50 = 53000 nM T30081 C93KDB 459905 Ki = 210 nM T30081 C5FS1E 477012 Ki = 1040000 nM T30081 CI0S8N 477015 Ki = 970000 nM T30081 CUW3B2 491807 IC50 > 1000000 nM T30081 C8WS5I 491808 IC50 > 1000000 nM T30081 CYTV93 491811 IC50 > 1000000 nM T30081 C71RDP 497634 IC50 = 3100 nM T30081 CX2LN9 497636 IC50 = 1200 nM T30081 CLI98Q 497637 IC50 = 3300 nM T30081 CS78DH 504626 IC50 > 500000 nM T30081 CO93FT 506492 IC50 = 73000 nM T30081 CN4A5U 508215 Ki = 220000 nM T30081 CZCE20 508216 Ki = 110000 nM T30081 CO9RJ8 510135 Ki = 40000 nM T30081 CNX65O 514178 IC50 = 7800 nM T30081 C3LE1J 3000238 Ki = 1690000 nM T30081 CC8TV9 3000253 Ki = 1600000 nM T30081 CVO3D5 3000254 Ki = 54000 nM T30081 C04TFN 3000255 Ki = 1690000 nM T30081 CG1QZ5 3000256 Ki = 1275000 nM T30081 CZF20L 3006428 Ki = 32000 nM T30081 CW0B1Q 3006429 Ki = 4700 nM T30081 CB1UY3 3006430 Ki = 43500 nM T30081 CMY59Q 3006432 Ki = 280000 nM T30081 C3KGQ8 3007847 Ki = 2000 nM T30081 CETR09 3034569 Ki = 12000 nM T30081 CW15OC 6439190 Ki = 220 nM T30081 CA89BP 6476766 IC50 > 1000000 nM T30081 CJB97H 6476767 IC50 > 1000000 nM T30081 C59CWM 6477687 IC50 = 3000 nM T30081 CH7M6L 6477690 IC50 = 9800 nM T30081 C2OH8G 6477696 IC50 = 22000 nM T30081 C1BF5V 9837976 Ki = 420000 nM T30081 C5O8EM 9906078 Ki = 62900 nM T30081 CBM0K2 9971180 IC50 = 57000 nM T30081 CHNO31 10003208 IC50 = 2300 nM T30081 CQ26PR 10040442 IC50 = 30000 nM T30081 CZ1A0R 10097595 IC50 > 1000000 nM T30081 C3EF4R 10198687 Ki = 2900 nM T30081 CT9JP4 10269114 IC50 > 500000 nM T30081 CM2L4O 10406438 Ki = 85800 nM T30081 C2G4OQ 10978846 IC50 = 40000 nM T30081 C82JAI 11438492 Ki = 69800 nM T30081 C8HVL6 11825312 IC50 = 4600 nM T30081 CG5E1H 11827046 IC50 = 2 nM T30081 C2KNL5 14308783 Ki = 975000 nM T30081 C0PHT1 14606828 IC50 = 99000 nM T30081 C7W9FV 15227900 IC50 > 50000 nM T30081 C2Z9KL 15227901 IC50 = 50000 nM T30081 C6Q3KN 15227902 IC50 > 50000 nM T30081 CG1D2I 15227903 IC50 > 50000 nM T30081 CYQ94X 15227904 IC50 > 50000 nM T30081 C5KD4V 15227905 IC50 > 50000 nM T30081 CU8B2A 15227906 IC50 > 50000 nM T30081 CWX5O0 15227907 IC50 > 50000 nM T30081 CT0CV1 15227908 IC50 > 50000 nM T30081 C4MUA1 22489180 IC50 > 1000000 nM T30081 CM91RP 24750302 IC50 > 500000 nM T30081 C07PEZ 24750303 IC50 > 500000 nM T30081 CTO90W 24750304 IC50 > 500000 nM T30081 CW2HP5 24750413 IC50 > 500000 nM T30081 C6ZE3D 44269001 Ki = 2000 nM T30081 C0R2AF 44286728 IC50 = 25000 nM T30081 CH4E8O 44286741 IC50 > 50000 nM T30081 CXTL42 44286784 IC50 > 50000 nM T30081 C9TFB7 44286896 Ki = 4300 nM T30081 CU5C7P 44333373 IC50 = 33000 nM T30081 C6CBN2 44333378 IC50 = 28000 nM T30081 C0EU3K 44333390 IC50 = 3500 nM T30081 CGYW24 44333414 IC50 = 180000 nM T30081 C76KRP 44333420 IC50 = 23000 nM T30081 C09IHV 44333437 IC50 = 491000 nM T30081 CGK2H1 44333745 IC50 = 27000 nM T30081 C12KRO 44333760 IC50 = 4100 nM T30081 CB5C8I 44355754 IC50 = 11000 nM T30081 C4G8PD 44355755 IC50 = 28000 nM T30081 CVH87D 44355905 IC50 = 4600 nM T30081 CR6Y8V 44355914 IC50 = 20000 nM T30081 CP9QL3 44355988 IC50 = 17000 nM T30081 C6ZO2D 44356613 IC50 = 19000 nM T30081 C17QOA 44420577 IC50 > 500000 nM T30081 C9HVL3 44420578 IC50 > 500000 nM T30081 CHP3U9 44420579 IC50 > 500000 nM T30081 CIQ47X 44420582 IC50 > 500000 nM T30081 CQY8X5 44437450 IC50 > 1000000 nM T30081 C5H7LS 44437451 IC50 > 1000000 nM T30081 CD0AN5 44437452 IC50 > 500000 nM T30081 C4YH3T 44437453 IC50 > 1000000 nM T30081 C2QO0P 44437477 IC50 > 500000 nM T30081 C9OE0G 44437478 IC50 > 500000 nM T30081 CO0N8X 44437480 IC50 > 1000000 nM T30081 C4V2AD 44560487 IC50 = 13000 nM T30081 CPM1F3 44560491 IC50 = 405000 nM T30081 C2XN5Q 44560560 IC50 = 10000 nM T30081 C3BJE2 46197226 IC50 > 500000 nM T30081 C8WR4I 46197456 IC50 > 500000 nM T30081 C2Y0QN 46197457 IC50 > 500000 nM T30081 CPA6D7 46700799 IC50 = 366000 nM T30081 CWJY16 46874452 IC50 > 500000 nM T30081 C1PCR5 46884564 IC50 = 71000 nM T30081 C4NK8W 46884565 IC50 = 75000 nM T30081 C48RWL 46884566 IC50 >= 500000 nM T30081 CN9RI6 46884567 IC50 = 109000 nM T30081 C8DP0M 46885250 IC50 = 316000 nM T30081 CQWV32 46885301 IC50 = 318000 nM T30081 CG74UX 46885302 IC50 = 177000 nM T30081 C9V5IT 46888106 IC50 = 105000 nM T30081 CB6PI7 46888107 IC50 = 311000 nM T30081 CB3V5I 46888108 IC50 = 114000 nM T30081 C9DI3F 46888151 IC50 = 86000 nM T30081 C9MZK2 46888152 IC50 = 60000 nM T30081 CUR4G7 46913823 IC50 = 200 ug.mL-1 T30081 CSQL06 54768280 IC50 = 200 ug.mL-1 T30081 CB9DU0 54768281 IC50 = 200 ug.mL-1 T30081 CUN04G 54768283 IC50 = 200 ug.mL-1 T30081 C2P3CT 90663608 IC50 > 1000000 nM T30081 C7MA3K 135398592 IC50 = 115000 nM T30081 C6Z4QV 135425312 Ki = 25000 nM T30081 C63BVC 135433410 Ki = 2060 nM T30081 CV0HE2 135499520 IC50 > 500000 nM T30081 C4K1FL 136118006 IC50 > 500000 nM T30081 CQGF80 136118007 IC50 > 500000 nM T30081 CR37CF 136118008 IC50 > 500000 nM T30081 D01GLG 5789 IC50 = 26 nM T30081 D0C7YS 160155 Ki = 20000 nM T30081 D0G5VO 135415618 Ki = 50 nM T30081 D0I6UV 6477686 IC50 = 180 nM T30081 D0M4MA 6035 Ki = 5060 nM T30081 D0O7GD 452142 IC50 >= 500000 nM T55781 D03ZBT 11626560 IC50 > 100 nM T55781 D0C4RB 36314 IC50 = 4900 nM T55781 D0W5HK 216239 IC50 = 1370 nM T55781 D00DRL 44137946 IC50 = 24 nM T55781 D03LWG 53235510 IC50 > 10000 nM T55781 D05PZB 135398495 IC50 = 1 nM T55781 D06DMQ 59472121 Ki = 30 nM T55781 D0E3TC 44259 IC50 = 11.6 nM T55781 D0O6WV 24794418 IC50 = 14 nM T55781 D03BNU 59604787 IC50 > 10000 nM T55781 D03RHV 72793043 IC50 = 600 nM T55781 D08OEW 72792975 IC50 = 72 nM T55781 D0M9TR 72793042 IC50 = 1130 nM T55781 CGAN35 2856 IC50 = 11000 nM T55781 CWQ7U1 696836 IC50 = 2060 nM T55781 C1C5EJ 784137 IC50 > 30000 nM T55781 CACS26 11561968 Ki > 2000 nM T55781 CU0E8O 11690457 Ki > 2000 nM T55781 CF57GK 46215462 IC50 = 15 nM T55781 CG6KA7 50945534 IC50 > 30000 nM T55781 CJ98GR 50947631 IC50 = 2250 nM T55781 C1SA2T 52109814 IC50 = 3560 nM T55781 CV8U6Y 52110137 IC50 = 680 nM T55781 CXSE16 52111270 IC50 = 4170 nM T55781 C3RC8Q 52111275 IC50 = 1240 nM T55781 CSF0Q5 52111278 IC50 = 1080 nM T55781 CUPV64 52111292 IC50 = 2900 nM T55781 C3V5XE 53355503 IC50 = 2.9 nM T55781 CC62KV 54915268 IC50 = 3000 nM T55781 CBOD63 56835089 IC50 = 2440 nM T55781 CD6Y9Z 57395116 IC50 = 2340 nM T55781 C8W6IG 57395117 IC50 = 970 nM T55781 CG7S0D 57396882 IC50 = 6930 nM T55781 C1MR8Q 60097495 IC50 > 1000 nM T55781 C10AMI 66553589 IC50 > 10000 nM T55781 CV63UL 67240318 IC50 > 10000 nM T55781 CJLT43 67471113 IC50 = 56 nM T55781 CXR9Y0 68212353 IC50 = 120 nM T55781 CEH69L 68212361 IC50 = 25 nM T55781 C4V3DJ 68212395 IC50 = 56 nM T55781 CPZ8D7 68212421 IC50 = 140 nM T55781 CBUE63 68212479 IC50 = 1400 nM T55781 CR0B8N 68212480 IC50 = 1.8 nM T55781 CZJ83X 68212482 IC50 = 0.25 nM T55781 C1QXE9 68212489 IC50 = 62 nM T55781 C5H8DO 68212494 IC50 = 4500 nM T55781 C2WDO9 68212498 IC50 = 74 nM T55781 C7PT2D 68212505 IC50 = 0.76 nM T55781 CKPF54 68212509 IC50 = 0.15 nM T55781 C40GFP 68212528 IC50 = 7000 nM T55781 CJY4P6 68212724 IC50 = 18 nM T55781 C2ZCD6 68212733 IC50 = 10 nM T55781 C4ARE2 68212746 IC50 = 8.2 nM T55781 CTM2R4 68212750 IC50 = 530 nM T55781 C5MG7K 68212755 IC50 = 13 nM T55781 COV36W 68212757 IC50 = 5.8 nM T55781 C51DUT 68212759 IC50 = 13 nM T55781 CL95KS 68212760 IC50 = 200 nM T55781 CQD3H2 68212763 IC50 = 400 nM T55781 C6GU4S 68212779 IC50 = 2400 nM T55781 CG5VP7 68212780 IC50 = 860 nM T55781 CJR90K 68212791 IC50 = 10 nM T55781 CS5C0R 68212798 Ki = 0.33 nM T55781 C2B8DE 70681768 IC50 = 9600 nM T55781 CQAU72 70681769 IC50 = 170 nM T55781 CG80HU 70681780 Ki = 2 nM T55781 C8JYH4 70686029 IC50 = 2800 nM T55781 C7LVS2 70692345 IC50 = 14 nM T55781 CWP13X 70695379 IC50 = 2400 nM T55781 CM0D3O 70696465 IC50 = 28000 nM T55781 CTB5O3 70696471 IC50 = 64 nM T55781 C5Q3YE 70697396 IC50 = 2200 nM T55781 CH0B8N 70789756 IC50 = 4680 nM T55781 CA3O6K 71552696 IC50 = 126 nM T55781 C1NPL0 71552941 IC50 = 1920 nM T55781 CA4PS8 71552942 IC50 = 775 nM T55781 C4Q2HC 71721525 IC50 = 4.3 nM T55781 CQ3JN8 71819732 IC50 = 17 nM T55781 C9NVM8 72192165 IC50 = 5.2 nM T55781 C7A8XR 72547635 IC50 = 150 nM T55781 CUPN10 72547636 IC50 = 37 nM T55781 C5MI7D 72547637 IC50 = 11 nM T55781 CD93WQ 72547638 IC50 = 24 nM T55781 C49RTS 72547864 IC50 = 120 nM T55781 C45UFT 72547868 IC50 = 180 nM T55781 CM23ZS 72548104 IC50 = 47 nM T55781 CO7MN3 72548105 IC50 > 30000 nM T55781 CH05EK 72551069 IC50 = 23 nM T55781 C07THM 72551070 IC50 = 40 nM T55781 CVNK29 72551073 IC50 = 2.1 nM T55781 CO3UW2 72551074 IC50 = 9 nM T55781 CP09RS 72792559 IC50 > 30000 nM T55781 C3PTC7 72792560 IC50 = 12 nM T55781 C12IMZ 72792561 IC50 = 18 nM T55781 C2E0RN 72792562 IC50 = 1.1 nM T55781 CZXU21 72792563 IC50 = 1.7 nM T55781 CD7UM4 72792564 IC50 = 0.7 nM T55781 C38OCL 72792627 IC50 = 0.69 nM T55781 C39PHS 72792906 IC50 = 3.4 nM T55781 C6HYA4 72792907 IC50 = 0.69 nM T55781 C16ETP 72792908 IC50 = 1.3 nM T55781 CNSX89 72792909 IC50 = 0.81 nM T55781 C7HXN3 72792910 IC50 = 1250 nM T55781 CGP01I 72792971 IC50 = 1.8 nM T55781 CXNF57 72792972 IC50 = 4.5 nM T55781 CGDL83 72792973 IC50 = 18 nM T55781 CJGF34 72792974 IC50 = 34 nM T55781 C4N9TK 72792977 IC50 = 200 nM T55781 C5B9CI 72793044 IC50 > 30000 nM T55781 C86UHM 72793045 IC50 = 2700 nM T55781 C75QHA 72793046 IC50 = 540 nM T55781 C1MPN7 72793047 IC50 = 170 nM T55781 CRJ81Y 72793048 IC50 = 50 nM T55781 CL9EA5 72793105 IC50 = 19 nM T55781 CVT7A9 72793106 IC50 = 44 nM T55781 C39VXU 72793107 IC50 = 380 nM T55781 C43SNK 72793108 IC50 = 16500 nM T55781 C9XAE8 72793109 IC50 = 83 nM T55781 CZA34R 72793110 IC50 = 110 nM T55781 CU9R4X 72793111 IC50 = 14 nM T55781 CD2K0R 72793177 IC50 = 320 nM T55781 CP26TN 72793178 IC50 = 220 nM T55781 CKV95R 72793179 IC50 = 44 nM T55781 CH80BD 72793182 IC50 = 12600 nM T55781 CAJ65L 72793183 IC50 > 30000 nM T55781 CVR1I4 72793252 IC50 = 67 nM T55781 CJWB46 72793253 IC50 = 5900 nM T55781 CMIH15 72793254 IC50 = 2500 nM T55781 C30IXP 72793255 IC50 = 8.4 nM T55781 C6YFO5 72793256 IC50 = 4.1 nM T55781 CJG79M 72793257 IC50 = 13 nM T55781 CK6U5Z 72793332 IC50 = 8 nM T55781 CI6JX5 72793333 IC50 = 230 nM T55781 CA4ET8 72793334 IC50 = 15 nM T55781 C6JW5N 72793335 IC50 = 29 nM T55781 CROW51 72793336 IC50 = 39 nM T55781 C65KJA 72793337 IC50 = 14 nM T55781 C7IA8R 72793397 IC50 = 6.7 nM T55781 CD85ZE 72793399 IC50 = 6.3 nM T55781 CI4E7H 72793400 IC50 = 14 nM T55781 C02GET 72793401 IC50 = 590 nM T55781 C9WYE4 72793466 IC50 = 37 nM T55781 C37FKG 72793468 IC50 = 62 nM T55781 COU2I8 72793469 IC50 = 1000 nM T55781 C49MHY 72793532 IC50 = 110 nM T55781 C3K2BV 72793533 IC50 = 620 nM T55781 C5UH4O 72793534 IC50 = 170 nM T55781 C2Z6FI 72793535 IC50 = 9900 nM T55781 CLTB82 72793536 IC50 = 2400 nM T55781 CQ7KX1 72793601 IC50 = 18 nM T55781 CW0PY4 72793602 IC50 = 570 nM T55781 CKB3O6 72793603 IC50 = 950 nM T55781 CI9L8K 72793604 IC50 = 15200 nM T55781 CMD9F8 72793605 IC50 = 6.3 nM T55781 CE60AT 72793606 IC50 = 2.8 nM T55781 C75UBS 72793607 IC50 = 3.9 nM T55781 C51VIE 72793608 IC50 = 27 nM T55781 COL6Y5 72793609 IC50 = 7.3 nM T55781 CJ9C7M 72793610 IC50 = 86 nM T55781 CGCL01 72793611 IC50 = 59 nM T55781 CZ5QY9 72793612 IC50 > 30000 nM T55781 CJ87CG 73211763 IC50 = 1.7 nM T55781 C1V3NZ 73425588 IC50 = 0.74 nM T55781 CQ4ZH2 74538669 IC50 = 4.4 nM T55781 CG7VE4 76309971 IC50 = 140 nM T55781 C17BGH 76328134 IC50 = 160 nM T55781 CH8W7D 77461036 IC50 > 1000 nM T55781 CHIZ70 89495685 IC50 = 1.3 nM T55781 CS6IA4 89495748 IC50 = 1.6 nM T55781 CW1OS0 89495775 IC50 = 0.57 nM T55781 C61JAN 91966173 IC50 = 7840 nM T55781 CQVL13 91966182 IC50 = 3430 nM T55781 CL2DH6 118433464 IC50 = 3.2 nM T55781 C01OAD 118433470 IC50 = 4.9 nM T55781 C9ENZ0 118433703 IC50 = 5.2 nM T55781 CQU1R4 118443520 IC50 = 22 nM T55781 C8OSQ4 118443521 IC50 = 3.5 nM T55781 CAM76F 118443524 IC50 = 3.6 nM T55781 C3DEP2 118443546 IC50 = 4.3 nM T55781 CGO6B1 118443548 IC50 = 1068 nM T55781 CADG96 118443549 IC50 = 5.2 nM T55781 CM92EG 118443553 IC50 = 19 nM T55781 CVWR20 118443556 IC50 = 20 nM T55781 CC9FK0 118443560 IC50 = 2.6 nM T55781 CRZ68N 118443583 IC50 = 2.5 nM T55781 C9I5MC 118443585 IC50 = 4.9 nM T55781 CE42TF 118443586 IC50 = 72 nM T55781 C5YJT1 118443594 IC50 = 2 nM T55781 CL0YO5 118443595 Ki = 0.43 nM T55781 CG3K5V 118443597 IC50 = 3.5 nM T55781 C12WAU 118446433 IC50 = 78 nM T55781 CFBY13 118446434 IC50 = 3.5 nM T55781 CY6C1E 122179442 IC50 > 10000 nM T55781 C08KEM 122179540 IC50 = 5400 nM T55781 CG0RP7 122179547 IC50 = 4700 nM T55781 C1A0SQ 122179548 IC50 = 5100 nM T55781 C8KXV1 127025843 IC50 > 1000 nM T55781 CB5JD0 127043185 IC50 = 10200 nM T55781 CRC8Y3 127043566 IC50 > 30000 nM T55781 CV7L1K 127043900 IC50 = 1840 nM T55781 C34VIW 127045062 IC50 > 30000 nM T55781 CS9H0C 127045063 IC50 = 7270 nM T55781 C2QDF3 127045215 IC50 = 1720 nM T55781 C4KH2E 127045219 IC50 > 30000 nM T55781 CK36LR 127045379 IC50 > 30000 nM T55781 CWJ1H6 127045411 IC50 = 1140 nM T55781 C0Q7TL 127045560 IC50 = 2010 nM T55781 C9LP2C 127045567 IC50 > 30000 nM T55781 C8ERJ7 127045762 IC50 > 1000 nM T55781 C7JC5K 134132904 IC50 = 1.8 nM T55781 C5DSV1 134134351 IC50 = 54 nM T55781 CYB46P 134135659 IC50 = 150 nM T55781 CDH31O 134136945 EC50 = 34 nM T55781 C46XTD 134138113 IC50 = 86 nM T55781 CK75ZI 134138785 IC50 = 13 nM T55781 CCE1O4 134138988 IC50 = 3 nM T55781 C9V4CG 134140406 EC50 = 150 nM T55781 C5C4TS 134141052 IC50 = 94 nM T55781 CWI41J 134141468 EC50 = 490 nM T55781 CYM06R 134142159 IC50 = 160 nM T55781 CZB68J 134142873 EC50 = 210 nM T55781 CX03CP 134143856 IC50 = 140 nM T55781 C5C2TA 134144975 IC50 = 4 nM T55781 CE12IN 134145489 IC50 = 170 nM T55781 CM4U6L 134147181 IC50 = 9.6 nM T55781 CBES34 134147807 IC50 = 4.1 nM T55781 C60FLZ 134148014 EC50 = 150 nM T55781 CDUX09 134148124 IC50 = 65 nM T55781 CGIT02 134149104 IC50 = 4.1 nM T55781 C4CA2M 134149641 IC50 = 17 nM T55781 C36GLZ 134150279 EC50 = 160 nM T55781 CZ42MI 134150952 IC50 = 11 nM T55781 C39AMZ 134151100 EC50 = 72 nM T55781 C10BFN 134151512 IC50 = 30 nM T55781 C8M3RH 134152780 IC50 = 5 nM T55781 C5PV8R 134153049 IC50 = 3.9 nM T55781 C4M7XF 134153576 IC50 = 80 nM T55781 C4AR9L 134153778 EC50 = 690 nM T55781 C6GC3U 134154700 IC50 = 8.9 nM T55781 C20PJY 134156194 IC50 = 5.6 nM T55781 CHN5R6 134156911 IC50 = 16 nM T55781 C70ZRI 134157187 IC50 = 4.9 nM T55781 CXC69T 137321158 IC50 = 29 nM T55781 C25ERN 137631967 IC50 = 4.4 nM T55781 C06JRX 137637094 IC50 = 36.9 nM T55781 C7TG3J 137641313 IC50 = 7585.78 nM T55781 C1DK0P 137651391 IC50 = 7.1 nM T55781 CV5H3Z 137657932 IC50 = 30.9 nM T55781 CE84NX 144944001 IC50 = 24 nM T55781 C65YWX 145964882 IC50 = 2500 nM T55781 CHC3T0 145965031 IC50 > 10000 nM T55781 CP92ZF 145965329 IC50 = 640 nM T55781 C9HXI4 145966620 IC50 = 2300 nM T55781 CQE9M5 145966810 IC50 = 480 nM T55781 C1EH6C 145967078 IC50 = 8700 nM T55781 CWJ12M 145969155 IC50 = 92 nM T55781 CGW5S1 145969844 IC50 = 2000 nM T55781 CB8R3A 145970271 IC50 > 10000 nM T55781 C40VIL 145972979 IC50 = 6200 nM T55781 CQBY19 145974023 IC50 > 10000 nM T55781 C4X7CT 145977420 IC50 = 5400 nM T55781 CLA57T 145978300 IC50 = 8900 nM T55781 C6KDQ5 145979093 IC50 = 22 nM T55781 CV7QY8 145981517 IC50 = 3.1 nM T55781 CG0R3A 145984368 IC50 = 90 nM T55781 CV78XO 145985621 IC50 = 61 nM T55781 CX5MB2 145986730 IC50 = 13 nM T55781 C1V6RA 145988134 IC50 > 100000 nM T55781 CD98JK 145989189 IC50 = 13 nM T55781 CWH69B 145989428 IC50 = 2.2 nM T55781 CZCS58 145989494 IC50 = 1.2 nM T55781 C0PHA7 145990595 IC50 = 40 nM T55781 CN6T4K 145991513 IC50 = 9 nM T55781 CMBH76 145991936 IC50 = 1.3 nM T55781 C0SO4N 145993259 IC50 = 4.9 nM T55781 CI7F4G 145994227 IC50 = 4.1 nM T55781 CL4B2M 155512535 IC50 = 2630 nM T55781 C81YCJ 155513061 IC50 = 3120 nM T55781 CTSM92 155538441 IC50 = 25 nM T55781 CC5F3I 155562216 IC50 = 3950 nM T55781 C40IYS 155562258 IC50 = 4.2 nM T55781 D0N4LR 53469448 IC50 = 474 nM T55781 D0Q0YV 24944925 IC50 = 6456.54 nM T99455 D00STL 644241 IC50 = 12.7 nM T99455 D0AZ3C 5291 IC50 = 14 nM T99455 D0E6XR 3062316 EC50 = 0.04 nM T99455 D0H0EQ 24826799 EC50 = 0.05 nM T99455 D0OB0F 5328940 IC50 = 20 nM T99455 D0R0MW 5329102 EC50 > 1000 nM T99455 D02LJW 23635314 IC50 = 100 nM T99455 D02XNW 5494449 IC50 = 50.12 nM T99455 D06JHV 46848036 IC50 = 6.2 nM T99455 D0E3TC 44259 IC50 = 121.8 nM T99455 D0U3EP 445154 IC50 = 28000 nM T99455 D05HDJ 49782106 EC50 = 7150 nM T99455 D0EF5T 44129660 EC50 = 430 nM T99455 D0JY1I 42613483 IC50 = 2700 nM T99455 D0L7XM 42628828 EC50 = 40 nM T99455 D0OE4F 4369496 IC50 = 100 nM T99455 D0ZH4I 76071870 IC50 > 10000 nM T99455 D01EFO 9864718 IC50 = 398.11 nM T99455 C6SB2N 123596 EC50 = 90 nM T99455 CV5MS2 2475277 EC50 = 1300 nM T99455 CCPF82 5312285 EC50 = 720 nM T99455 CZR3M4 9799152 IC50 = 100000 nM T99455 CY3MK1 9807952 IC50 = 3.981 nM T99455 CI3O6X 9814609 IC50 = 61659.5 nM T99455 CX9DG5 9822042 IC50 = 199.53 nM T99455 CSH0A9 9847014 IC50 = 346.74 nM T99455 C3UQL7 9860872 IC50 = 33884.42 nM T99455 CC90FJ 9869737 IC50 = 512 nM T99455 CIZ13L 9943193 IC50 = 602.56 nM T99455 CUKH27 9943194 IC50 = 707.95 nM T99455 CU78NO 9947433 IC50 = 151.36 nM T99455 CYT7R9 9953676 IC50 = 794.33 nM T99455 CJ40GO 9965429 IC50 = 1513.56 nM T99455 CTE3K0 9982070 IC50 = 3162.28 nM T99455 CP23QA 10007129 IC50 = 10 nM T99455 CLI9A3 10029363 IC50 = 63.1 nM T99455 C0G5DK 10039959 IC50 = 7943.28 nM T99455 CT9F2H 10053560 IC50 = 5.012 nM T99455 C8EW6P 10095381 IC50 = 2187.76 nM T99455 C3P8WK 10110378 IC50 = 1000 nM T99455 C63CFD 10111108 IC50 = 1288.25 nM T99455 CL42XS 10136330 IC50 = 794.33 nM T99455 CUW34X 10157645 IC50 = 1905.46 nM T99455 COC30E 10181160 IC50 = 199.53 nM T99455 CN51JQ 10292737 IC50 = 446.68 nM T99455 CG2L4Z 10343860 IC50 = 602.56 nM T99455 CYW13A 10348904 IC50 = 10 nM T99455 C7TJ9U 10483163 IC50 = 7.079 nM T99455 CS0DE8 10493971 IC50 > 3000 nM T99455 C78FPR 10501266 IC50 = 371.54 nM T99455 CU6G5Y 10708835 IC50 = 1202.26 nM T99455 CO61VZ 11161166 IC50 = 24000 nM T99455 C94MLD 11165739 EC50 = 390 nM T99455 C2KT9E 11168002 IC50 = 4.074 nM T99455 C89EZO 11180525 IC50 = 16.98 nM T99455 C3FL9M 11199480 IC50 > 100000 nM T99455 CJTP13 11280103 IC50 = 3801.89 nM T99455 CPW2Y8 11326963 EC50 = 4470 nM T99455 C1DF5Z 11336923 EC50 = 330 nM T99455 CKY3E2 11338122 IC50 = 199.53 nM T99455 CH4O8K 11347791 EC50 = 1660 nM T99455 C4RLW0 11368874 IC50 = 26000 nM T99455 C3OCV2 11371778 IC50 = 1000 nM T99455 CHJV86 11381980 EC50 = 470 nM T99455 C14XYD 11385486 IC50 > 10000 nM T99455 C3O0WI 11438191 IC50 = 5128.61 nM T99455 C3EXM4 11440028 IC50 = 398.11 nM T99455 C2E0GS 11461932 EC50 = 1800 nM T99455 C7I6AG 11474111 IC50 = 501.19 nM T99455 C0YH2X 11478363 IC50 = 1.25 nM T99455 CMW72Q 11488124 IC50 = 724.44 nM T99455 C57TKI 11565665 IC50 = 18000 nM T99455 C43JZU 11604436 IC50 = 3800 nM T99455 CGU7N0 11604739 IC50 = 12900 nM T99455 CLJ81E 11630507 IC50 = 20000 nM T99455 C6SGF3 11644985 IC50 = 16000 nM T99455 CJK78Z 11652152 IC50 = 8000 nM T99455 CAJS96 11662893 IC50 = 14600 nM T99455 CH3S9K 11666294 IC50 = 20000 nM T99455 C95EPO 11666668 IC50 = 35000 nM T99455 CKAH36 11669784 IC50 = 9500 nM T99455 CJ89UZ 11687939 IC50 > 100000 nM T99455 C7RDH3 11709536 IC50 > 100000 nM T99455 CFJ4I7 11723151 IC50 = 3311.31 nM T99455 C7C2FM 11737638 IC50 = 1513.56 nM T99455 CVFS29 11751305 IC50 = 64.57 nM T99455 CPJ7C9 11774222 EC50 = 580 nM T99455 CUDO23 11994441 IC50 = 25.12 nM T99455 C02DIH 14347011 IC50 = 1819.7 nM T99455 CZB2V0 16750146 IC50 = 20.89 nM T99455 C6XC2W 23145852 IC50 = 10.96 nM T99455 CUVB29 23145858 IC50 = 3.981 nM T99455 CO0T3M 24825778 IC50 = 750 nM T99455 CIFO50 24897305 IC50 = 11000 nM T99455 CYXC26 24958918 IC50 = 10000 nM T99455 CVUK27 24958920 IC50 = 2500 nM T99455 C35LZO 24959284 IC50 = 2500 nM T99455 CIZQ04 24959285 IC50 = 15000 nM T99455 C47ING 24959648 IC50 = 10000 nM T99455 C4V9GI 24960018 IC50 = 500 nM T99455 CWLR85 24960379 IC50 = 10000 nM T99455 CHC6A5 25017304 IC50 = 1378 nM T99455 C38YMD 25017555 IC50 = 7083 nM T99455 CDHM05 25017557 IC50 = 739.5 nM T99455 CFU60Y 25235817 IC50 = 436 nM T99455 C8B6TY 42628503 EC50 < 500 nM T99455 C15OSL 42633116 EC50 = 250 nM T99455 CO1I2D 42633117 EC50 = 1200 nM T99455 CO7YL0 42633119 EC50 > 10000 nM T99455 CWF2S8 42633305 EC50 = 160 nM T99455 CKCO80 42633306 EC50 = 400 nM T99455 CCI8P7 42633666 EC50 = 1320 nM T99455 CSH3I9 42633667 EC50 = 2200 nM T99455 CPNK96 42633668 EC50 = 4340 nM T99455 CL04QK 42633670 EC50 > 10000 nM T99455 C7DA0B 42633859 EC50 = 9680 nM T99455 CLM7B9 42634040 EC50 = 490 nM T99455 C6DK1W 42634389 EC50 > 10000 nM T99455 C87GKI 42634390 EC50 = 918 nM T99455 CK15FQ 42634392 EC50 = 406 nM T99455 CCN5O4 42634553 EC50 = 1340 nM T99455 C2H1SJ 42634556 EC50 = 48 nM T99455 C1M8SR 42634557 EC50 = 1960 nM T99455 C48YFI 42634730 EC50 = 5600 nM T99455 C8L5RN 42635093 EC50 = 150 nM T99455 CQ9F8I 42635272 EC50 = 120 nM T99455 CG2P1M 42635644 EC50 = 1230 nM T99455 C4JRG0 42635811 EC50 = 140 nM T99455 CCOV80 42635815 EC50 = 100 nM T99455 C7K9YE 44194683 EC50 = 420 nM T99455 C9G6QE 44194684 EC50 = 340 nM T99455 CBP7D2 44194685 EC50 = 240 nM T99455 CBD90A 44194780 EC50 = 920 nM T99455 COK3J5 44194781 EC50 = 970 nM T99455 C7XOD2 44194782 EC50 = 1150 nM T99455 C4T0HN 44194783 EC50 = 1270 nM T99455 C63UIZ 44194784 EC50 = 1240 nM T99455 CMRX16 44273620 IC50 = 5754.4 nM T99455 CCH89M 44300026 IC50 = 1995.26 nM T99455 CH4ND7 44340691 IC50 = 9772.37 nM T99455 CK2CU3 44340703 IC50 = 17378.01 nM T99455 CY0XF5 44340726 IC50 = 67608.3 nM T99455 C2F7SL 44395745 IC50 = 10000 nM T99455 C0TED6 44395746 IC50 = 5011.87 nM T99455 CZR42M 44395763 IC50 = 575.44 nM T99455 CJ0Z5K 44395813 IC50 = 8912.51 nM T99455 CU9XQ0 44395880 IC50 = 10000 nM T99455 CYF8U6 44395904 IC50 = 1000 nM T99455 C5DR6W 44395926 IC50 = 10000 nM T99455 C4R8EB 44410932 IC50 = 23000 nM T99455 CI82UE 45270897 IC50 > 10000 nM T99455 C4UM6Y 45273507 IC50 > 10000 nM T99455 CR4A6B 46703970 EC50 > 10000 nM T99455 CH9AW2 46865999 IC50 = 500 nM T99455 C4FX6S 46866098 IC50 = 500 nM T99455 CK6UL0 46866099 IC50 = 200 nM T99455 C67UEP 46881960 IC50 = 8 nM T99455 C71XDW 49780994 EC50 = 330 nM T99455 CEAH78 49780998 EC50 = 5000 nM T99455 CHS50Y 49780999 EC50 = 2920 nM T99455 C9WOE2 49781000 EC50 = 480 nM T99455 CGV34K 49781215 EC50 = 90 nM T99455 C84ZOI 49781216 EC50 = 360 nM T99455 C4K9DH 49781217 EC50 = 810 nM T99455 C34JPY 49781218 EC50 = 400 nM T99455 C7YET3 49781219 EC50 = 290 nM T99455 C48NTZ 49781220 EC50 = 170 nM T99455 C7QON3 49781221 EC50 > 10000 nM T99455 CHUG72 49781431 EC50 > 10000 nM T99455 CQ43VM 49781432 EC50 > 10000 nM T99455 CDU34O 49781433 EC50 > 10000 nM T99455 CSE62H 49781434 EC50 > 10000 nM T99455 CL51PM 49781435 EC50 > 10000 nM T99455 CE1N9P 49781436 EC50 > 10000 nM T99455 CF4TU7 49781437 EC50 > 10000 nM T99455 CH4MI1 49781662 EC50 > 10000 nM T99455 CQOW70 49781663 EC50 > 10000 nM T99455 C46TMR 49781664 EC50 > 10000 nM T99455 CG2I3L 49781665 EC50 > 10000 nM T99455 COW0H6 49781667 EC50 > 10000 nM T99455 CBH02L 49781668 EC50 = 1440 nM T99455 C6-DEC-09 49781877 EC50 > 10000 nM T99455 CGI64U 49781878 EC50 = 6890 nM T99455 C38FVM 49781879 EC50 = 380 nM T99455 CVT73X 49781880 EC50 = 760 nM T99455 C7X9UG 49781881 EC50 = 300 nM T99455 C5I3OF 49781882 EC50 = 270 nM T99455 C1T6CN 49782104 EC50 = 400 nM T99455 C6WOK4 49782105 EC50 = 350 nM T99455 CKQC50 49782107 EC50 = 6890 nM T99455 CWHY47 49782108 EC50 = 690 nM T99455 CGC82O 49782109 EC50 = 2960 nM T99455 C80XEK 49782334 EC50 = 6920 nM T99455 C2BNW5 49782337 EC50 = 160 nM T99455 C1EA9K 49782338 EC50 = 1700 nM T99455 C2Y6QS 50938552 IC50 > 10000 nM T99455 CS3LT9 51030149 IC50 = 671 nM T99455 C1XRG0 51030150 IC50 = 507 nM T99455 C3PDJ8 51030250 IC50 = 774 nM T99455 CAQ4V6 51030532 IC50 = 480 nM T99455 CX47EM 51030534 IC50 = 1300 nM T99455 CSZ36G 51030713 IC50 = 177 nM T99455 CA6U5X 51030714 IC50 = 491 nM T99455 C9NYP4 51036677 IC50 > 10000 nM T99455 C4WRY3 51037112 IC50 > 10000 nM T99455 CNWO03 51037408 IC50 = 5 nM T99455 CLO1I6 51037410 IC50 = 6 nM T99455 CZ2H3T 51037608 IC50 = 19 nM T99455 CK8J5T 51037609 IC50 = 904 nM T99455 CYO9W0 51037823 IC50 = 458 nM T99455 CF7HX6 51037824 IC50 = 161 nM T99455 CMX3I7 51037825 IC50 = 19 nM T99455 CRI28Z 51037948 IC50 > 10000 nM T99455 C4XT7P 51038497 IC50 = 24 nM T99455 CKB79R 51038498 IC50 = 125 nM T99455 C75JSI 51038499 IC50 = 7 nM T99455 C6PG5F 51351510 IC50 = 20.1 nM T99455 CHAV48 52940594 IC50 = 2500 nM T99455 CAK80G 52940928 IC50 = 2500 nM T99455 C02ALP 52940992 IC50 > 20000 nM T99455 CSM30J 52941799 IC50 = 2500 nM T99455 CFY5K7 52941942 IC50 = 10000 nM T99455 CPU53W 52941997 IC50 = 2500 nM T99455 C1LN4J 52942048 IC50 = 500 nM T99455 C69VKZ 52942052 IC50 = 2500 nM T99455 C0QFI8 52942203 IC50 > 20000 nM T99455 C7D5FE 52942236 IC50 > 20000 nM T99455 C0S7OM 52943049 IC50 = 2500 nM T99455 CQZ98C 52943259 IC50 = 2500 nM T99455 CZ3X7O 52943392 IC50 > 20000 nM T99455 C9L3HD 52943395 IC50 = 20000 nM T99455 CCBA25 52944595 IC50 > 20000 nM T99455 C1XN6P 52944599 IC50 > 20000 nM T99455 C1H8GZ 52944627 IC50 > 20000 nM T99455 C90JQR 52945824 IC50 > 20000 nM T99455 CPVD21 52945847 IC50 > 20000 nM T99455 C62EXZ 52946812 IC50 = 10000 nM T99455 C3WI7B 52947902 IC50 = 2500 nM T99455 CK08IW 52948022 IC50 = 2500 nM T99455 CJ1XR3 52948871 EC50 > 10000 nM T99455 C4Q6XB 52949498 IC50 > 20000 nM T99455 CCXY64 54581006 IC50 = 5510 nM T99455 C36DEH 54582045 IC50 = 277 nM T99455 CPI87W 54583990 IC50 > 2000 nM T99455 CIE67G 54585892 IC50 = 3780 nM T99455 CAIO65 68796885 EC50 = 0.04 nM T99455 C91HPI 71300299 IC50 > 5000 nM T99455 CC98EU 71449991 IC50 = 2.67 nM T99455 CV21PC 71449992 IC50 = 5.96 nM T99455 CG59TB 71449993 IC50 = 0.45 nM T99455 C23ETA 71450038 IC50 = 1.66 nM T99455 C3B7IP 71450039 IC50 = 0.36 nM T99455 C0XL6Z 71451816 IC50 = 2.25 nM T99455 CQM05U 71451817 IC50 = 0.6 nM T99455 CVE9P2 71451818 IC50 = 0.52 nM T99455 C30FHU 71453635 IC50 = 0.54 nM T99455 CR7DI8 71453636 IC50 = 1.01 nM T99455 C8K6BL 71453637 IC50 = 19.1 nM T99455 C12IUO 71453638 IC50 = 0.52 nM T99455 CIEK84 71453639 IC50 = 0.72 nM T99455 C0FTX4 71453675 IC50 = 0.33 nM T99455 CK7V6O 71453676 IC50 = 0.42 nM T99455 CU42QX 71455363 IC50 = 0.52 nM T99455 C4X9GT 71455364 IC50 = 0.78 nM T99455 CVY26H 71455365 IC50 = 1.18 nM T99455 C3X1OP 71455406 IC50 = 0.52 nM T99455 COUR46 71455407 IC50 = 1.03 nM T99455 C8IV0R 71455408 IC50 = 1.01 nM T99455 CY2G7S 71457180 IC50 = 0.7 nM T99455 CXA9W8 71457181 IC50 = 0.98 nM T99455 CCT0X3 71459003 IC50 = 17.8 nM T99455 C01XBA 71459004 IC50 = 2.56 nM T99455 C0WF3X 71459043 IC50 = 1.94 nM T99455 CJ3PO5 71459044 IC50 = 15 nM T99455 CW0X4B 71460798 IC50 = 3.44 nM T99455 CE84WT 71460799 IC50 = 12.8 nM T99455 CG0F1R 71460800 IC50 = 1629 nM T99455 CZM79U 71460801 IC50 = 22.6 nM T99455 CWT1E8 71460802 IC50 = 0.69 nM T99455 CZ72YB 71460803 IC50 = 302 nM T99455 C8KL1P 71460845 IC50 = 1.42 nM T99455 C7XZ6K 71460846 IC50 = 66 nM T99455 CS08OH 71462551 IC50 = 0.45 nM T99455 CB45LP 71462552 IC50 = 0.41 nM T99455 C1IT5U 71550931 IC50 = 355 nM T99455 C5V8IC 71602940 IC50 = 4.73 nM T99455 C6SV9J 71602987 IC50 = 4125.31 nM T99455 CCQ25W 71602988 IC50 = 4.79 nM T99455 C6LKO2 71602989 IC50 = 3.21 nM T99455 C93MLS 71602992 IC50 = 34.77 nM T99455 CSP7K1 71603051 IC50 = 2754.9 nM T99455 CH7D8G 71603053 IC50 = 3.78 nM T99455 CHZ7U8 71603054 IC50 = 294.34 nM T99455 CWE69D 71603113 IC50 = 0.52 nM T99455 C4WT7O 71603114 IC50 = 2.34 nM T99455 CR08FQ 71603115 IC50 = 1.48 nM T99455 CE09DT 71603116 IC50 = 350.08 nM T99455 C4NM3G 71603117 IC50 = 1110.42 nM T99455 C62ZYM 71603170 IC50 = 63.31 nM T99455 CU8Z1W 71603171 IC50 = 6.34 nM T99455 CG80HO 73345816 IC50 = 199.53 nM T99455 CKA92Y 73348812 IC50 = 33189.45 nM T99455 CEUP75 73351906 IC50 = 50118.72 nM T99455 C7DSE2 73351907 IC50 = 10000 nM T99455 C8SUY0 73354884 IC50 = 398.11 nM T99455 CPJC10 73356444 IC50 = 1000 nM T99455 CCIS39 73356445 IC50 = 5370.32 nM T99455 C2PAK9 73438493 IC50 = 10 nM T99455 CHI51J 76070594 IC50 = 390 nM T99455 C8VAD5 76070929 IC50 > 10000 nM T99455 CB4V1R 76071142 IC50 = 380 nM T99455 CBAT06 76071144 IC50 = 89 nM T99455 C7SH1T 76071506 IC50 = 210 nM T99455 CS87EI 76071624 IC50 = 880 nM T99455 CGC0K4 76071869 IC50 > 10000 nM T99455 C9A8IG 79072608 IC50 = 255 nM T99455 CBP5K7 91183030 IC50 > 10000 nM T99455 CO07DQ 101879028 IC50 = 50 nM T99455 CG7YK9 101879029 IC50 = 17 nM T99455 CS8N1X 101879030 IC50 = 130 nM T99455 CUSN35 101879031 IC50 = 70 nM T99455 CY7BI2 118706214 IC50 > 10000 nM T99455 CDIA30 118722069 IC50 = 78600 nM T99455 C2SFD8 118722070 IC50 = 354000 nM T99455 C7CKE4 118722071 IC50 > 500000 nM T99455 C9ZW4S 118722072 IC50 = 385 nM T99455 CJPC58 118722073 IC50 > 500000 nM T99455 C53MDX 118722074 IC50 = 141000 nM T99455 CFC4T9 118722075 IC50 > 500000 nM T99455 CO9AY0 118722076 IC50 = 16100 nM T99455 C7YB8R 118722077 IC50 > 500000 nM T99455 CHD5Y4 118722078 IC50 = 6060 nM T99455 CIQ5K8 118722079 IC50 = 1440 nM T99455 C6CW9X 118722080 IC50 = 13500 nM T99455 C0M1KE 118722081 IC50 = 872 nM T99455 C5TD1S 118722083 IC50 = 277000 nM T99455 CF3YQ1 118722084 IC50 > 500000 nM T99455 CPR97Z 118722085 IC50 > 500000 nM T99455 CZ0I1M 118722086 IC50 = 91800 nM T99455 C2ACT5 118722089 IC50 > 500000 nM T99455 C5LBT6 118722090 IC50 = 563 nM T99455 CQ1S2N 118722091 IC50 = 266000 nM T99455 CQCX41 118737057 IC50 = 1 nM T99455 CUP4S1 122183740 IC50 = 14.2 nM T99455 CT12MC 122183741 IC50 = 15.9 nM T99455 CV3FM4 122183742 IC50 = 213.5 nM T99455 CVM71G 122183743 IC50 = 41.02 nM T99455 C48MKU 122183744 IC50 = 43.27 nM T99455 C2MK8C 122183745 IC50 = 46.2 nM T99455 CN3VR2 122183746 IC50 = 50.6 nM T99455 C43ELH 122183747 IC50 = 178 nM T99455 CG71PU 122183748 IC50 = 326 nM T99455 CUWG02 122183749 IC50 = 129.1 nM T99455 C6SQI8 122183750 IC50 = 26.58 nM T99455 C5X8JH 122183808 IC50 = 117.4 nM T99455 CG3ZX6 122183809 IC50 = 16.87 nM T99455 CM3NO8 122183810 IC50 = 175.3 nM T99455 C2P9NG 122186622 IC50 > 1000 nM T99455 CSVT14 122186623 IC50 = 300 nM T99455 C2V7EG 122189041 IC50 > 500000 nM T99455 C6MU0Y 122189043 IC50 = 66 nM T99455 C19CBJ 122189044 IC50 = 1156 nM T99455 CEQ5W9 122189045 IC50 = 45600 nM T99455 C5EX7F 122189047 IC50 = 276 nM T99455 C0JYX4 122189048 IC50 = 60670 nM T99455 C4UK5I 122189049 IC50 = 10220 nM T99455 CDT8R6 122189050 IC50 = 112 nM T99455 CR2Y7P 122189051 IC50 = 63300 nM T99455 C5OR0G 122189052 IC50 = 940 nM T99455 C82CRO 122189053 IC50 > 500000 nM T99455 CJ9HI8 122189054 IC50 = 19070 nM T99455 C9JI1S 122189056 IC50 > 500000 nM T99455 CYF0W2 122189057 IC50 = 143 nM T99455 C2YT3F 122189058 IC50 > 500000 nM T99455 CDY7N9 122189059 IC50 = 5050 nM T99455 C9Y5NU 122189060 IC50 = 89700 nM T99455 C54KBN 122189061 IC50 = 73 nM T99455 CR81XY 122189062 IC50 = 321 nM T99455 C4NK6A 122189064 IC50 = 444180 nM T99455 CO36WE 122189065 IC50 = 16 nM T99455 CL72TM 122189066 IC50 = 421 nM T99455 C6ZHF0 122189067 IC50 = 1837 nM T99455 CQ2SD8 122189068 IC50 > 500000 nM T99455 CDX9H3 122190820 IC50 = 2590 nM T99455 CSV74J 122190821 IC50 = 8530 nM T99455 C3ZQJ4 122190822 IC50 = 14550 nM T99455 C4AM5V 122190823 IC50 > 100000 nM T99455 CU3O4Q 122190824 IC50 = 9250 nM T99455 C4BL5S 122190825 IC50 = 11300 nM T99455 CZBP91 122190826 IC50 = 9240 nM T99455 C3PB0Z 122190828 IC50 = 4400 nM T99455 CT32LN 122190829 IC50 = 6200 nM T99455 C1EBW9 122190830 IC50 = 8960 nM T99455 CZ26FY 122190831 IC50 = 73910 nM T99455 C5Z2DL 122190832 IC50 = 35660 nM T99455 CW84RP 122190867 IC50 > 100000 nM T99455 CHU8E2 122190868 IC50 = 42170 nM T99455 CF2W4A 122190869 IC50 = 35040 nM T99455 CUP8H1 122190870 IC50 = 15320 nM T99455 CFR2Z0 122190871 IC50 = 51920 nM T99455 CV2N9D 122190872 IC50 > 100000 nM T99455 CL42TR 122190873 IC50 > 100000 nM T99455 C6QY7L 122196083 IC50 = 14 nM T99455 CP0WN2 122196084 IC50 = 86 nM T99455 CG48DP 122196085 IC50 = 49200 nM T99455 C0LWG4 122196086 IC50 = 3410 nM T99455 C0I6AZ 122196188 IC50 = 180 nM T99455 CJCH07 122196189 IC50 > 100000 nM T99455 CM0X4J 122196190 IC50 = 2760 nM T99455 CA8U7J 122196191 IC50 = 83520 nM T99455 C8LAJ2 122196192 IC50 > 100000 nM T99455 C47IXK 122196193 IC50 = 2370 nM T99455 C6BPW7 122196194 IC50 = 1890 nM T99455 CFE6L4 122196195 IC50 = 22760 nM T99455 CN4J5W 122196196 IC50 = 8560 nM T99455 CI9J5Z 122196197 IC50 = 75290 nM T99455 CU9V8Q 122196198 IC50 = 31 nM T99455 CL07SV 122196199 IC50 = 18 nM T99455 CWU4J7 122196200 IC50 = 56270 nM T99455 CRXT48 122196201 IC50 > 100000 nM T99455 CEQ32S 122196202 IC50 = 250 nM T99455 CS3U0R 122196203 IC50 > 100000 nM T99455 CQL0W7 122197565 IC50 > 10000 nM T99455 C6KM3T 127034964 EC50 = 1 nM T99455 C1BZ4L 127034965 EC50 = 3 nM T99455 C3IRJ0 127048197 IC50 > 10000 nM T99455 CZ07TW 127048198 IC50 > 10000 nM T99455 CS0H2C 127048199 IC50 > 10000 nM T99455 C1OE2F 127049532 IC50 = 580 nM T99455 C5P8TC 127049857 IC50 > 10000 nM T99455 CPQ35R 127049870 IC50 = 3880 nM T99455 CQO3X7 127049871 IC50 > 10000 nM T99455 C5H8LK 127051998 IC50 > 10000 nM T99455 CGT0B1 127052321 IC50 > 10000 nM T99455 C7NH6A 127052914 IC50 > 10000 nM T99455 CKB1Y6 127052915 IC50 > 10000 nM T99455 C6RPF1 130364436 IC50 > 10000 nM T99455 CSY34O 130364443 IC50 > 10000 nM T99455 CI9H2W 130364450 IC50 > 10000 nM T99455 CM4TO5 130364451 IC50 = 2100 nM T99455 CV4DH7 130364460 IC50 > 10000 nM T99455 CW91ZV 130364461 IC50 > 10000 nM T99455 CQIZ43 130364463 IC50 = 9900 nM T99455 C4IKC6 130364464 IC50 > 10000 nM T99455 C0X6JS 130364465 IC50 > 10000 nM T99455 C0ZGC1 130364467 IC50 > 10000 nM T99455 CO9C5Q 130364468 IC50 > 10000 nM T99455 CQW3P1 130364471 IC50 > 10000 nM T99455 CHWX05 130364473 IC50 = 8700 nM T99455 CLB65Y 130364478 IC50 = 4300 nM T99455 CUZG19 130364481 IC50 > 10000 nM T99455 C34OMJ 130364482 IC50 > 10000 nM T99455 C6TWR3 130364484 IC50 > 10000 nM T99455 C8SF5Q 130364488 IC50 = 547 nM T99455 CS5C4E 130364494 IC50 > 10000 nM T99455 CVQ32Y 130364503 IC50 > 10000 nM T99455 CV8B0Y 130364506 IC50 > 10000 nM T99455 CHX23J 130364524 IC50 = 10000 nM T99455 CHYL89 130364535 IC50 > 10000 nM T99455 CBI35E 132275094 IC50 = 942 nM T99455 CCG06O 134131688 IC50 = 122000 nM T99455 CFE03W 134131725 IC50 = 16200 nM T99455 CC3Y5M 134131924 IC50 = 320 nM T99455 C60IDE 134134575 IC50 = 220 nM T99455 C4TJD6 134135198 IC50 = 24 nM T99455 CUP01F 134135273 IC50 = 19 nM T99455 CKQV02 134135339 IC50 > 500000 nM T99455 CM3J8P 134137546 IC50 = 58000 nM T99455 C9QFX5 134139856 IC50 = 2280 nM T99455 C6Q9BT 134140130 IC50 = 15 nM T99455 CF0M3H 134140636 IC50 = 2580 nM T99455 C4AI2O 134141645 IC50 = 0.012 ug.mL-1 T99455 C0UT6Y 134141669 IC50 > 500000 nM T99455 CZA63L 134143363 IC50 = 1980 nM T99455 C3NS0E 134144264 IC50 = 19 nM T99455 CEU0N9 134144345 IC50 = 1440 nM T99455 C0R1TX 134144394 IC50 = 640 nM T99455 CF7KV6 134144611 IC50 = 1150 nM T99455 C18KJH 134145016 IC50 = 0.012 ug.mL-1 T99455 C35XCY 134145509 IC50 = 1690 nM T99455 C7W6PG 134147256 IC50 = 4520 nM T99455 C8AJ9S 134148237 IC50 = 2250 nM T99455 CJ7A2M 134148351 IC50 = 440 nM T99455 C8YCR0 134148385 IC50 = 19 nM T99455 CCL1G8 134148410 IC50 = 2650 nM T99455 C37NPG 134148847 IC50 = 385 nM T99455 CUL93K 134150012 IC50 > 500000 nM T99455 CI4EO5 134150056 IC50 > 500000 nM T99455 C1EY7B 134153245 IC50 = 890 nM T99455 CLC89D 134153463 IC50 = 0.012 ug.mL-1 T99455 CFTL08 134155527 IC50 = 560 nM T99455 CAOK49 134155843 IC50 > 500000 nM T99455 CX6Q8G 134157397 IC50 > 500000 nM T99455 CQR94G 134198433 IC50 > 10000 nM T99455 C46QAS 135441185 EC50 = 10 nM T99455 C0PVG7 135819982 EC50 = 360 nM T99455 C2PJK6 135820173 EC50 = 70 nM T99455 C53LFX 135820297 EC50 = 970 nM T99455 CP7KZ8 135820466 EC50 = 1800 nM T99455 CQK62L 135820498 EC50 = 560 nM T99455 C4PD2G 135820511 EC50 = 30 nM T99455 CDT7E4 136211077 IC50 > 100 nM T99455 C5VE4K 137636547 IC50 > 10000 nM T99455 CZ05TY 137637593 IC50 > 10000 nM T99455 C6PKY7 137645383 IC50 > 10000 nM T99455 CHR9E0 137651685 IC50 = 414 nM T99455 CY53VO 137651787 IC50 > 10000 nM T99455 CE8DW7 137658399 IC50 > 10000 nM T99455 CU61WM 137658936 IC50 > 10000 nM T99455 CY9N8Q 137662234 IC50 = 8100 nM T99455 C0PYR1 138454771 EC50 < 10 nM T99455 CO9P7G 145351804 IC50 > 1000 nM T99455 CBR08X 145983359 IC50 = 1107 nM T99455 CE2X6V 145983518 IC50 = 435 nM T99455 C4ID8J 145984666 IC50 = 211 nM T99455 CD49VM 155295006 IC50 > 10000 nM T99455 CA8IF5 155510457 IC50 = 10660 nM T99455 CSHC63 155510467 IC50 > 10000 nM T99455 CG09WO 155512858 IC50 > 10000 nM T99455 C6H8ZU 155513172 IC50 = 2220 nM T99455 COI8N1 155513641 IC50 = 3720 nM T99455 CZDH58 155514096 IC50 > 10000 nM T99455 CEB08Z 155514919 IC50 = 6280 nM T99455 C84GJO 155517474 IC50 > 10000 nM T99455 CHQ5X7 155518340 IC50 = 6230 nM T99455 CP1B5K 155518600 IC50 = 520 nM T99455 C63PZX 155518871 IC50 > 10000 nM T99455 CC1A2U 155518947 IC50 = 4280 nM T99455 C1U3HE 155522045 IC50 = 110 nM T99455 C8EZ6J 155523550 IC50 = 31610 nM T99455 CF72IY 155527080 IC50 = 17560 nM T99455 CITV17 155527171 IC50 = 5750 nM T99455 C8DF2W 155529116 IC50 = 2160 nM T99455 CNP8T7 155530083 IC50 = 237 nM T99455 CK10UA 155531677 IC50 = 3696 nM T99455 C54ARD 155532371 IC50 = 170 nM T99455 C4DT6V 155532665 IC50 = 2340 nM T99455 CWLZ25 155535008 IC50 > 10000 nM T99455 C8NA6L 155536370 IC50 = 437 nM T99455 CL9X4S 155540971 IC50 = 2450 nM T99455 C3Q9UA 155541932 IC50 > 10000 nM T99455 CI27QV 155546853 IC50 > 10000 nM T99455 CYP2O5 155547984 IC50 = 1452 nM T99455 CB85AE 155550823 IC50 = 380 nM T99455 CL8KR2 155552517 IC50 = 989.3 nM T99455 C1TA9J 155553503 IC50 > 10000 nM T99455 CJS68O 155553593 IC50 = 290 nM T99455 C8BAU3 155554243 IC50 > 10000 nM T99455 CCQF25 155555943 IC50 > 10000 nM T99455 C9QM2K 155559937 IC50 = 1500 nM T99455 CN9LE6 155560662 IC50 = 5850 nM T99455 CHLY93 155562871 IC50 = 5345 nM T99455 C60KLJ 155564326 IC50 = 4992 nM T99455 C4BS6J 155565938 IC50 = 5637 nM T99455 CINX89 155566065 IC50 = 5120 nM T99455 CVMG35 155566307 IC50 = 1350 nM T99455 C7Q4RY 155566792 IC50 = 1813 nM T99455 CP69SU 155567937 IC50 > 10000 nM T99455 C8VT6Z 155568644 IC50 = 1990 nM T99455 D00AII 5281727 IC50 = 10000 nM T99455 D03EHM 24905142 IC50 = 18 nM T99455 D03NPX 447077 IC50 = 2 nM T99455 D03PLP 11579996 IC50 = 8000 nM T99455 D05UJT 5311510 EC50 = 140 nM T99455 D05XGZ 11536458 IC50 = 42000 nM T99455 D08RZB 11153014 IC50 = 3 nM T99455 D0AW4W 11537051 IC50 = 6000 nM T99455 D0AZ0Y 11514345 IC50 = 20000 nM T99455 D0H4YH 11594901 IC50 = 10000 nM T99455 D0I3XZ 11601743 IC50 = 4200 nM T99455 D0N7AJ 11409972 IC50 = 580 nM T99455 D0O9NE 5388063 IC50 = 10000 nM T99455 D0PI0R 11609210 IC50 = 14000 nM T99455 D0QG6G 11493254 IC50 = 14000 nM T84631 D05EAM 4735 IC50 = 10400 nM T84631 D05PHH 3447 IC50 = 4610 nM T84631 D07UWV 92722 Ki = 53000 nM T84631 D07XHO 4413 IC50 = 21100 nM T84631 D0I0RJ 16231 IC50 > 50000 nM T84631 D0I5HF 10182969 Ki = 0.08 nM T84631 D0J0BU 10275777 Ki = 0.117 nM T84631 D0KG3R 9875401 Ki = 0.4 nM T84631 D0M7JT 216210 Ki > 1000 nM T84631 D00LOB 9866964 Ki = 3300 nM T84631 D01MUU 183797 Ki = 3680 nM T84631 D05TKW 16098914 IC50 = 1900 nM T84631 D07BRZ 9939865 Ki = 4.6 nM T84631 D07KWN 99514 Ki = 13385 nM T84631 D0I7MX 9871765 Ki = 22.5 nM T84631 D0ID3W 9911502 Ki = 4 nM T84631 D0PK7J 56599309 Ki = 206 nM T84631 D0X2NN 9826322 IC50 = 2.7 nM T84631 D02INZ 2387 IC50 = 4500 nM T84631 D02MHE 9806376 IC50 = 301 nM T84631 D02QTV 122267 IC50 = 16 nM T84631 D03QJN 9895762 Ki = 0.15 nM T84631 D0D5RH 11641515 Ki = 1.8 nM T84631 D0E2MJ 5496659 Ki = 0.4 nM T84631 D0J9UI 9807238 Ki = 1.3 nM T84631 D0K1PR 1747 Ki = 22000 nM T84631 D0N7WR 108040 Ki = 20400 nM T84631 D0S2JG 9913629 Ki = 1100 nM T84631 D0T4UL 11634458 IC50 = 0.57 nM T84631 CR8YG3 1308 Ki = 34 nM T84631 C71WRJ 1503 Ki = 8900 nM T84631 CY5B9C 1504 Ki = 2100 nM T84631 C2KE5Q 1508 Ki = 2700 nM T84631 C4S1PB 4300 Ki = 115000 nM T84631 CL1T7V 4301 Ki = 12000 nM T84631 C8D4SG 5107 Ki = 0.9 nM T84631 C2OG9Z 47978 IC50 = 100 nM T84631 CMG15V 122129 Ki = 7 nM T84631 CS5RN9 178051 Ki = 47973.34 nM T84631 CZP0Y1 204101 Ki = 0.19 nM T84631 CM32OH 402499 IC50 > 50000 nM T84631 C4Q9XJ 402501 IC50 > 50000 nM T84631 C3YP0R 444562 Ki = 26000 nM T84631 C3R5AJ 445480 Ki = 22 nM T84631 CRN1F6 445481 Ki = 18 nM T84631 C2Z0XW 445482 Ki = 0.7 nM T84631 CR4KE5 445844 Ki = 19000 nM T84631 CU6X2A 445847 Ki = 31000 nM T84631 CI64QU 446399 IC50 = 33 nM T84631 CHD15V 446604 Ki = 38018.94 nM T84631 C9GU2P 446605 Ki = 42657.95 nM T84631 C7IE4P 446606 Ki = 20989.4 nM T84631 C4M8WT 446979 Ki = 28 nM T84631 CS4OB0 446982 Ki = 25 nM T84631 C5E3YX 446984 Ki = 9 nM T84631 C17BWY 447193 Ki = 0.76 nM T84631 CM3T9E 447194 Ki = 0.059 nM T84631 CZC4U1 447359 Ki = 4 nM T84631 CNO6G5 447360 Ki = 1.1 nM T84631 C85OTU 447361 Ki = 3 nM T84631 C9QXV5 447362 Ki = 1 nM T84631 C5UX1L 447478 Ki = 990 nM T84631 CVND42 447482 Ki = 2400 nM T84631 C4OKV5 447486 Ki = 34000 nM T84631 CC9G5O 447490 Ki = 34000 nM T84631 CR2DX3 447496 Ki = 300 nM T84631 COYS31 447502 Ki = 6800 nM T84631 CVI28M 447508 Ki = 52 nM T84631 CS09BE 447510 Ki = 570 nM T84631 C87GLP 447540 Ki = 65000 nM T84631 C6FD5N 447889 Ki = 15135.61 nM T84631 CK9Q4X 448061 Ki = 13 nM T84631 C43LRO 448062 Ki = 1.6 nM T84631 COK45L 448065 Ki = 0.27 nM T84631 CFMI91 448548 Ki = 3000 nM T84631 CSL82K 449091 Ki = 26000 nM T84631 COK61H 639391 Ki = 0.66 nM T84631 C9D4IN 754821 IC50 > 50000 nM T84631 CB5C6X 1034712 IC50 = 4224 nM T84631 C1CNZ9 2756474 Ki = 680000 nM T84631 CER5L6 2796875 Ki = 11 nM T84631 CO4K7H 3037565 IC50 = 11418 nM T84631 C24VNC 3083488 Ki = 41020.41 nM T84631 C0K7TF 3123858 IC50 > 50000 nM T84631 C8KD9E 3162843 IC50 > 50000 nM T84631 CQ6N8P 3496895 Ki = 13 nM T84631 CT8JE1 4655928 Ki = 1400 nM T84631 CZEI30 5282448 IC50 = 11 nM T84631 C0KI2N 5287439 Ki = 0.1 nM T84631 CPZ6A3 5287506 Ki = 8000 nM T84631 C48TEQ 5287836 Ki = 13 nM T84631 CQ26VM 5289531 Ki = 15000 nM T84631 C1B9GP 5400404 IC50 > 50000 nM T84631 C0CV5L 5496928 IC50 = 270 nM T84631 CAW1P7 5497056 Ki = 0.9 nM T84631 C7SYK9 6102731 IC50 = 35 nM T84631 C5YL6I 6420136 Ki = 18 nM T84631 C2ZRF5 6540265 Ki = 3 nM T84631 C5XV7G 6540266 Ki = 0.07 nM T84631 CY1J7X 6540267 Ki = 89 nM T84631 CN57IY 6540268 Ki = 3 nM T84631 C8MS7Y 6852168 Ki = 6 nM T84631 CN2B6S 6852211 Ki = 10000 nM T84631 C49IOZ 6857707 Ki = 140000 nM T84631 CM8R6E 6914706 IC50 = 160 nM T84631 CNZA87 9112697 IC50 > 200000 nM T84631 CX34ZD 9549214 Ki = 0.14 nM T84631 CME7Y3 9549257 Ki = 90 nM T84631 CXY5Z7 9549258 Ki = 15 nM T84631 CYRC97 9549259 Ki = 47 nM T84631 CAE25N 9549260 Ki = 1 nM T84631 CK64FD 9794516 IC50 >= 10300 nM T84631 CJ52KF 9794796 IC50 = 90000 nM T84631 CVFE34 9800775 IC50 = 1190 nM T84631 C92QSE 9801235 IC50 > 100000 nM T84631 C2FHU7 9801905 IC50 = 640 nM T84631 C3CL2G 9803364 Ki = 11 nM T84631 C4VX9Y 9803558 Ki = 8 nM T84631 CTA52P 9803848 Ki > 15000 nM T84631 C8QGS1 9804434 Ki = 16 nM T84631 CDN8P2 9804727 Ki = 103000 nM T84631 C1FIN6 9804775 IC50 > 130 nM T84631 C4OTK6 9805415 Ki = 1.9 nM T84631 CAKN38 9805632 Ki = 3.8 nM T84631 C6JIT7 9806444 IC50 = 3300 nM T84631 CBKL18 9806644 IC50 = 13 nM T84631 CW3NK6 9806974 Ki = 9.5 nM T84631 CKP97L 9807142 Ki = 1.2 nM T84631 CX1C7P 9807257 Ki = 260 nM T84631 C6F3XK 9807686 Ki = 43 nM T84631 CS62VX 9808020 IC50 = 0.83 nM T84631 CAG59M 9808035 Ki = 47 nM T84631 CTS98Y 9808170 Ki = 4.9 nM T84631 CH9IE6 9808346 IC50 = 2.3 nM T84631 CZS3H5 9808724 Ki = 3400 nM T84631 C2AXV0 9809479 Ki = 1.1 nM T84631 C60AVD 9812184 Ki = 910 nM T84631 CLTO67 9821317 IC50 > 100000 nM T84631 C4KEZ2 9821506 Ki > 500 nM T84631 CNCV95 9823140 IC50 = 1708 nM T84631 CJ2G7A 9823668 IC50 = 21 nM T84631 CX6DA7 9823789 Ki = 1600 nM T84631 CD3AP6 9824122 Ki = 198 nM T84631 CZ64PW 9824925 Ki = 164 nM T84631 C1YZP2 9825165 Ki = 39 nM T84631 CTG89N 9825830 Ki = 5 nM T84631 CPB20R 9826345 Ki = 3 nM T84631 CKH36Z 9826433 IC50 = 12 nM T84631 CS1DL7 9826716 IC50 = 3.6 nM T84631 CYR35V 9827147 IC50 = 34 nM T84631 CB82VS 9827306 Ki = 5.7 nM T84631 CK5VW1 9827389 IC50 = 3.9 nM T84631 CA7W3I 9827682 IC50 = 13 nM T84631 C6J0KE 9827723 Ki = 600 nM T84631 CGN48U 9827867 IC50 = 6000 nM T84631 CEJ3D7 9827921 Ki = 38 nM T84631 CVP0C6 9828249 IC50 = 15 nM T84631 CGD13M 9828337 IC50 = 14 nM T84631 CB65VJ 9828393 Ki = 10 nM T84631 CE0HD3 9828470 Ki = 84800 nM T84631 CRH01E 9828697 Ki = 500 nM T84631 C9A5SY 9828818 Ki = 21978.6 nM T84631 COW7Q3 9829120 Ki = 1.3 nM T84631 CP2X5B 9829453 Ki = 28 nM T84631 C7BW5P 9829585 Ki < 0.1 nM T84631 C5RVZ4 9829804 Ki = 62 nM T84631 C8RV5E 9830070 Ki = 500 nM T84631 C4F8CN 9830285 IC50 = 1410 nM T84631 C4T5BQ 9830932 Ki = 360 nM T84631 CH38SL 9840270 Ki = 220 nM T84631 CVO5R3 9842851 IC50 = 1370 nM T84631 C53JFK 9844392 Ki = 19 nM T84631 CC4Y8V 9845104 Ki = 275 nM T84631 C6VAG8 9845526 IC50 = 84 nM T84631 C2TA1I 9845742 IC50 > 30000 nM T84631 CM8Y9G 9846259 IC50 = 10000 nM T84631 C8I4LS 9846496 Ki = 900 nM T84631 CM0OU9 9847373 IC50 > 2500 nM T84631 CU2H1W 9848037 IC50 = 120 nM T84631 C5Z2RH 9848091 IC50 = 104 nM T84631 CSQ8V7 9848265 IC50 = 7.3 nM T84631 CX25MR 9848465 Ki = 0.5 nM T84631 CW3EC6 9848592 Ki = 5300 nM T84631 CCL5G3 9848846 IC50 = 0.55 nM T84631 C80PNB 9849423 IC50 = 1.6 nM T84631 CS9HQ0 9850467 IC50 = 19.3 nM T84631 CH9L1I 9850515 Ki = 1.8 nM T84631 CEQ92L 9850889 IC50 = 1.6 nM T84631 CR7S2O 9851195 Ki = 1.1 nM T84631 CP8CY7 9859977 IC50 > 200000 nM T84631 CRTD24 9863579 Ki = 55000 nM T84631 CB86RC 9864323 Ki = 50 nM T84631 CF74PR 9864759 IC50 = 1120 nM T84631 C89JRZ 9868633 Ki = 8300 nM T84631 CQ5J9K 9868873 Ki = 0.1 nM T84631 CL6QS0 9868922 Ki = 2100 nM T84631 CDVE40 9869375 Ki = 0.78 nM T84631 C5A1LI 9870767 IC50 = 4.5 nM T84631 C38BTY 9870834 Ki = 0.75 nM T84631 CZ9LR2 9870910 Ki = 4500 nM T84631 C1AW6N 9870947 Ki = 20 nM T84631 CIL85V 9871029 IC50 = 38 nM T84631 C9UB6X 9871197 Ki = 3.5 nM T84631 CX51SZ 9871369 IC50 = 1.6 nM T84631 CHP0C8 9872347 Ki = 400 nM T84631 CIZ61P 9872423 Ki > 75400 nM T84631 C6ZB3K 9872552 IC50 = 18 nM T84631 CG0L6A 9873029 IC50 = 3.2 nM T84631 CAJ92Z 9873782 Ki = 22 nM T84631 C5LV1Z 9873979 IC50 = 6000 nM T84631 CPU3D1 9881263 IC50 > 200000 nM T84631 CS78YB 9882885 IC50 > 200000 nM T84631 C2F5NS 9884570 Ki = 1300 nM T84631 C83BSN 9885116 Ki = 4200 nM T84631 CQP0V2 9886960 Ki = 460 nM T84631 CJT9X7 9887558 Ki = 102 nM T84631 C6A4TL 9890540 Ki = 11 nM T84631 C17NPU 9890541 IC50 = 20.9 nM T84631 CC3R5Y 9890878 Ki = 0.18 nM T84631 CO4QD2 9891154 Ki = 3.4 nM T84631 C7E1IV 9891337 IC50 = 20.6 nM T84631 CT6W0R 9891759 Ki = 4400 nM T84631 CD13TH 9891795 IC50 > 10000 nM T84631 C80RWQ 9892098 Ki = 1.9 nM T84631 C1M2PU 9892103 IC50 = 3510 nM T84631 C8UV6Y 9892106 Ki = 0.33 nM T84631 C79RJF 9892295 IC50 = 750 nM T84631 C7I5RG 9892392 Ki = 16000 nM T84631 CG5VS0 9892818 IC50 = 29 nM T84631 C6QE7Y 9893007 IC50 > 11000 nM T84631 CKN8D4 9893040 Ki = 92 nM T84631 CXY68Z 9893122 IC50 = 337 nM T84631 CNJ0W1 9893177 IC50 = 1390 nM T84631 C4A6TQ 9893238 Ki = 3 nM T84631 C5IG2W 9893544 Ki = 0.32 nM T84631 C4DHN5 9894203 Ki = 1.5 nM T84631 CB4O8L 9894223 Ki = 2.7 nM T84631 C13KVD 9894553 Ki = 2000 nM T84631 CCSP64 9894606 Ki = 170 nM T84631 CKDP84 9895193 Ki = 1700 nM T84631 CZY9L0 9905436 IC50 = 174000 nM T84631 C0SP6Q 9906596 Ki = 120 nM T84631 C2HN7L 9907201 Ki = 42 nM T84631 C85SEZ 9908687 IC50 > 10000 nM T84631 CMC95R 9910164 Ki = 165 nM T84631 CAP0O8 9910540 Ki = 50 nM T84631 CD5LQ0 9910982 Ki > 15000 nM T84631 CAWD59 9911275 IC50 = 30 nM T84631 CS6QF5 9912191 Ki > 30000 nM T84631 C75QYP 9912650 IC50 = 5.8 nM T84631 CJ5Y8N 9912741 IC50 = 20 nM T84631 C0LKE7 9912771 Ki = 31 nM T84631 C8GJF3 9913055 IC50 = 39.6 nM T84631 CU94XJ 9913274 IC50 = 95 nM T84631 C4N0IJ 9913371 IC50 = 10 nM T84631 CUF7C2 9913912 IC50 = 9.9 nM T84631 C49HMD 9914510 Ki = 1.7 nM T84631 C1C3VT 9914538 IC50 = 11 nM T84631 CUVX26 9914911 Ki = 360 nM T84631 CC0D5H 9915041 Ki = 0.91 nM T84631 CPZ50Y 9915193 Ki = 0.29 nM T84631 CVND52 9915545 Ki > 10000 nM T84631 C2GWH3 9916339 Ki = 71 nM T84631 CX45DI 9916346 Ki = 1760 nM T84631 CH8QJ4 9916876 Ki = 0.014 nM T84631 CHG59Y 9916885 Ki = 330 nM T84631 C0Z3HS 9917367 IC50 = 39 nM T84631 CK2H1C 9917705 Ki = 0.52 nM T84631 CF9SD1 9917846 IC50 = 2 nM T84631 CFO1K9 9922130 Ki > 1000000 nM T84631 CLZ53G 9922131 Ki > 1000000 nM T84631 CAP64B 9929157 Ki = 9 nM T84631 C2TO4N 9931543 Ki = 2900 nM T84631 C9I2ES 9931785 IC50 = 1500 nM T84631 CY0TP3 9932394 IC50 = 20 nM T84631 CI8JS1 9933581 IC50 = 24 nM T84631 C7H6NL 9933675 IC50 = 8 nM T84631 C85LIU 9934003 Ki = 0.15 nM T84631 CS9Y5I 9934133 IC50 = 7200 nM T84631 C7V9BM 9934351 Ki = 4 nM T84631 CLT7P8 9934591 IC50 = 2 nM T84631 CSY16U 9934960 Ki = 11.5 nM T84631 C38QWF 9935364 Ki = 0.06 nM T84631 CG3B1P 9935390 Ki = 0.5 nM T84631 C1XT2Y 9935746 Ki = 2 nM T84631 CL2NV0 9935925 IC50 > 870 nM T84631 C5KS0R 9936020 IC50 = 6 nM T84631 CKLJ26 9936190 IC50 > 100000 nM T84631 C49DRC 9936691 IC50 = 376 nM T84631 CL0U1E 9936850 IC50 = 0.5 nM T84631 CDT2W8 9936861 Ki = 2.8 nM T84631 CG96QC 9936983 Ki = 3.9 nM T84631 COA4R0 9937032 Ki = 2.3 nM T84631 C07XOI 9937041 Ki = 29 nM T84631 CC9QH7 9937406 IC50 = 270 nM T84631 CK76DL 9937410 Ki = 10 nM T84631 C8F5CW 9937921 Ki = 0.15 nM T84631 C8LR4T 9938917 Ki = 1.7 nM T84631 CNE34O 9939021 IC50 = 1 nM T84631 CDT95S 9939426 Ki = 980 nM T84631 C1RHT8 9949886 Ki = 210 nM T84631 CD27EJ 9951054 IC50 = 66 nM T84631 CP06LN 9953722 Ki = 15 nM T84631 CD7ZO5 9954791 Ki = 3.9 nM T84631 C0R4GE 9954812 IC50 = 7.5 nM T84631 CX85LD 9954980 Ki = 0.43 nM T84631 CK9N1A 9955155 IC50 = 0.9 nM T84631 CP7A2W 9955292 Ki = 1200 nM T84631 CSI62L 9955475 IC50 = 851 nM T84631 C3EPC4 9955758 Ki > 22000 nM T84631 CV96ZD 9955999 Ki = 110 nM T84631 C58QTM 9956404 Ki = 1 nM T84631 CY5OI8 9956416 IC50 = 5000 nM T84631 C8Y4EG 9956632 Ki = 16 nM T84631 CW4SU3 9956768 Ki = 7500 nM T84631 CI84CP 9957386 Ki = 0.35 nM T84631 CN36AS 9957822 Ki = 0.63 nM T84631 C85CTV 9957994 IC50 = 646 nM T84631 CLM2E6 9958023 Ki = 150 nM T84631 CE39JM 9958168 Ki = 3900 nM T84631 CU2YV0 9958249 IC50 = 7.8 nM T84631 C76ZFQ 9958477 Ki = 1300 nM T84631 CRM6L7 9958614 IC50 = 11 nM T84631 CLW0D4 9959111 IC50 = 3 nM T84631 C2Y0QV 9959268 IC50 = 3.4 nM T84631 CEHA54 9959604 IC50 = 2.1 nM T84631 CX59ZG 9959715 Ki = 350 nM T84631 CBC2K3 9959749 IC50 = 0.8 nM T84631 C0C1FQ 9959919 Ki = 1.5 nM T84631 COMH01 9961613 Ki = 1.7 nM T84631 C0TV8Q 9962561 Ki >= 200000 nM T84631 CTMU52 9978512 IC50 = 200 nM T84631 C3BNE7 9979006 IC50 = 1015 nM T84631 C3S7IV 9979724 Ki = 262 nM T84631 CV81FG 9980363 IC50 = 500 nM T84631 C38MBH 9981197 Ki = 0.07 nM T84631 C4CH0E 9981449 Ki = 99000 nM T84631 CWGL23 9982191 Ki = 130 nM T84631 C6XM2Z 9982428 Ki = 0.041 nM T84631 CK6XE9 9982431 IC50 > 30000 nM T84631 CY3Z7I 9982644 IC50 = 170 nM T84631 C5SA7F 9983043 IC50 > 2500 nM T84631 C5UGC0 9983309 Ki = 0.046 nM T84631 CCP75S 9983704 Ki = 6.4 nM T84631 C59OAZ 9983994 IC50 = 5.3 nM T84631 CZ50EY 9984282 IC50 = 1.9 nM T84631 C0OA9T 9984718 Ki = 270 nM T84631 CIP45F 9984838 IC50 = 3.5 nM T84631 CZ6TD1 9985759 Ki = 21 nM T84631 CKP2Z7 9987204 Ki > 33700 nM T84631 CKIP10 9987251 IC50 = 79000 nM T84631 CEC95B 9997816 Ki = 400 nM T84631 CE75GM 10000477 IC50 = 640 nM T84631 CJ0Q2S 10002821 Ki = 6 nM T84631 CVQN23 10003356 Ki = 11 nM T84631 C56FZK 10003877 IC50 = 15000 nM T84631 C4KCS7 10004019 Ki = 3600 nM T84631 CU9QI6 10004529 Ki = 0.037 nM T84631 C9O5SJ 10004800 Ki = 0.77 nM T84631 CH5BV6 10005347 Ki = 29991.63 nM T84631 C8I7YZ 10006319 IC50 = 200 nM T84631 CZJ38W 10006399 IC50 > 25000 nM T84631 CR34FA 10007463 Ki = 0.14 nM T84631 CFQV59 10007890 Ki = 2.4 nM T84631 CGL95Q 10008517 Ki = 3890.45 nM T84631 C7Q8PK 10009640 Ki = 0.016 nM T84631 CB1SY8 10023491 IC50 = 1700 nM T84631 C8ME3O 10024183 Ki = 7 nM T84631 CBM0Q3 10026319 Ki = 0.048 nM T84631 CF1V4K 10027758 Ki = 3 nM T84631 CW5JH1 10028252 Ki = 0.9 nM T84631 C3SU6O 10028986 Ki = 0.4 nM T84631 CX4TI5 10029172 Ki = 340 nM T84631 C3E4DR 10029213 IC50 = 6700 nM T84631 C4PFW9 10029239 Ki = 0.55 nM T84631 CI2O5B 10029343 Ki = 1.1 nM T84631 CB4Y7M 10030046 IC50 = 24 nM T84631 CTO52N 10030167 Ki = 5 nM T84631 CDL3M7 10030847 Ki = 8 nM T84631 C5LQ4A 10032429 Ki = 1.7 nM T84631 CUG6R3 10037159 Ki = 27 nM T84631 CSX68Z 10043156 IC50 = 1100 nM T84631 CK4W6M 10047815 IC50 = 52000 nM T84631 C3DIK1 10048418 IC50 = 61 nM T84631 C9R8YW 10048823 Ki = 50.5 nM T84631 C8FKM2 10049151 IC50 = 39000 nM T84631 CILJ89 10050878 IC50 = 28 nM T84631 C80QYS 10051154 Ki = 92000 nM T84631 C08PUS 10051441 IC50 = 81 nM T84631 CVY28G 10051489 Ki = 4.2 nM T84631 C29DTM 10051582 Ki = 0.2 nM T84631 CU9I7D 10051599 Ki = 12 nM T84631 CHZL08 10051960 Ki = 3.4 nM T84631 C3QP6V 10052373 Ki = 54 nM T84631 CXL9H7 10052619 Ki = 51 nM T84631 COP2U4 10052951 Ki = 3 nM T84631 CFCT67 10053115 Ki = 0.5 nM T84631 CDE42G 10053298 Ki = 5500 nM T84631 CXZ2V3 10054210 Ki = 1.3 nM T84631 C1OI8R 10066101 Ki = 4600 nM T84631 C6F4SZ 10067786 Ki = 12 nM T84631 CBV7N2 10070407 IC50 = 4100 nM T84631 CW28HS 10071127 Ki = 11 nM T84631 CI2KG6 10072299 IC50 > 30000 nM T84631 CP65QI 10073006 Ki = 0.023 nM T84631 CV5F8U 10073425 Ki = 3.3 nM T84631 C7TU4O 10073666 Ki = 0.6 nM T84631 CB04YW 10073864 IC50 > 100000 nM T84631 CF4R2W 10074230 IC50 = 260 nM T84631 CF18ZA 10074434 Ki = 2.8 nM T84631 CUOC38 10074752 Ki = 4.7 nM T84631 CAT42M 10074892 Ki > 300000 nM T84631 C9ZCS2 10074922 IC50 = 1600 nM T84631 CF0R6D 10074927 IC50 > 25000 nM T84631 C2CUX3 10075442 Ki = 1.8 nM T84631 COL31T 10075735 Ki = 0.1 nM T84631 C46JXH 10076965 IC50 = 72 nM T84631 CD0VO9 10078364 IC50 = 27 nM T84631 CR0ZL7 10091675 IC50 = 1600 nM T84631 CP38MH 10091962 IC50 = 1500 nM T84631 CPY49G 10092707 IC50 = 11750 nM T84631 CZM79H 10093390 Ki > 15000 nM T84631 C4P3ZO 10093667 IC50 = 15000 nM T84631 C3TDM1 10094168 Ki = 5 nM T84631 C2VT9U 10094219 Ki = 0.5 nM T84631 CZH3W7 10094378 Ki = 160000 nM T84631 C0FS4U 10094458 IC50 = 840 nM T84631 CMHD92 10094532 IC50 = 66000 nM T84631 CRXD40 10095024 Ki = 2800 nM T84631 CQP65H 10095093 Ki = 3600 nM T84631 C6PVA7 10095315 IC50 = 530 nM T84631 C3TWI1 10095455 Ki = 1 nM T84631 C3OG5U 10095865 Ki = 2 nM T84631 C0JE3C 10096795 IC50 = 150 nM T84631 C3XBN4 10097126 IC50 = 27 nM T84631 C8L7HY 10097631 Ki = 2330 nM T84631 C3IRT4 10098156 Ki = 5400 nM T84631 CRS8D1 10098302 Ki = 2.2 nM T84631 C6V2QM 10098361 Ki = 0.11 nM T84631 COSB36 10098572 Ki = 0.02 nM T84631 C9TN8U 10098702 Ki = 380 nM T84631 CD3VB0 10099008 Ki = 0.074 nM T84631 CX8A6G 10099038 Ki > 8000 nM T84631 CO8G7N 10099218 IC50 = 2 nM T84631 CP39AO 10099570 IC50 = 4.8 nM T84631 CO7J9C 10099638 Ki = 26 nM T84631 CV6NQ3 10099674 Ki > 8000 nM T84631 CW6IS3 10113744 IC50 = 20 nM T84631 C7HKG1 10114497 IC50 < 0.5 nM T84631 CH4Z6B 10116752 Ki = 0.14 nM T84631 CW4RZ5 10116936 IC50 > 450 nM T84631 C1VT4F 10117027 Ki = 15 nM T84631 C9V2WC 10117161 IC50 = 52 nM T84631 CK69GS 10117541 Ki = 0.24 nM T84631 CXCR46 10117543 Ki > 75000 nM T84631 C1XZ8N 10117556 IC50 = 4 nM T84631 CM34QP 10118017 Ki = 4 nM T84631 CL9RB8 10118144 Ki = 0.28 nM T84631 CB4QC8 10118358 Ki = 0.97 nM T84631 C9PG6D 10119254 Ki = 0.001 nM T84631 CX9VL6 10119957 Ki = 300 nM T84631 CV5E4L 10121049 Ki > 75400 nM T84631 C4TB7E 10121121 Ki = 15 nM T84631 CL68QZ 10121795 IC50 = 128 nM T84631 CS32UJ 10128374 Ki = 0.3 nM T84631 C3JPD6 10128550 Ki = 44.5 nM T84631 C1BA9E 10128598 Ki = 2 nM T84631 CJP02S 10128788 Ki = 5.3 nM T84631 C6AET3 10128907 Ki = 19 nM T84631 C0KQ9U 10129004 Ki = 2 nM T84631 C4FV1T 10129354 Ki = 1 nM T84631 CR03NV 10131788 Ki > 1000000 nM T84631 CN9F5G 10137016 Ki = 0.044 nM T84631 CJYD93 10137523 IC50 = 187 nM T84631 C7QB2E 10138114 IC50 = 32 nM T84631 CUCF82 10139899 Ki = 0.97 nM T84631 CVA35H 10140425 Ki = 178.6 nM T84631 CMFW67 10140911 Ki = 0.51 nM T84631 C67VZS 10141105 IC50 = 2 nM T84631 CF68DH 10141182 Ki = 3 nM T84631 CWF4I3 10141502 Ki = 5400 nM T84631 CN2WO7 10141594 Ki = 2.8 nM T84631 C1Q3KU 10141691 Ki = 0.73 nM T84631 CRH46O 10142203 Ki = 0.013 nM T84631 C1SKF3 10142819 IC50 = 6.7 nM T84631 C17YOT 10142920 Ki = 2 nM T84631 C54YQM 10143087 IC50 = 1320 nM T84631 C31QAL 10143532 Ki = 0.21 nM T84631 CYCG10 10151574 Ki = 24 nM T84631 CJ52ND 10152434 Ki = 2 nM T84631 C6XYM8 10152710 Ki = 11 nM T84631 CJ93LZ 10152785 Ki = 7 nM T84631 C86MJA 10152813 Ki = 1 nM T84631 C7HW4S 10161422 IC50 = 90 nM T84631 C95PMZ 10161902 IC50 = 26 nM T84631 CVZ23C 10162019 Ki = 53 nM T84631 C5IQ3M 10162145 IC50 = 1.5 nM T84631 C4K3WG 10162441 Ki = 96.4 nM T84631 CV27BE 10162765 Ki = 189 nM T84631 CT65YJ 10162799 Ki = 5300 nM T84631 CBHY78 10163266 Ki = 248.6 nM T84631 CF82TK 10163421 Ki = 6.3 nM T84631 C75ADN 10164065 Ki = 0.92 nM T84631 CM6PS4 10165173 Ki = 111000 nM T84631 C1QBH5 10165288 Ki = 11 nM T84631 C5WB4J 10165649 Ki > 75400 nM T84631 C7G4JC 10166616 Ki > 75400 nM T84631 CEPJ05 10166622 Ki > 75400 nM T84631 C5I0YH 10168444 Ki = 20 nM T84631 C24FCQ 10174464 Ki = 2 nM T84631 CD60LF 10174479 Ki = 6.8 nM T84631 CG2B8A 10174487 Ki = 15 nM T84631 CHPZ12 10174488 Ki = 3 nM T84631 CL0BI3 10174813 Ki = 78 nM T84631 CB17JX 10174938 Ki = 19 nM T84631 CMX71K 10174991 Ki = 2 nM T84631 C86UTO 10175171 Ki = 3 nM T84631 COVN41 10175189 Ki = 6.9 nM T84631 CG37YX 10181104 IC50 > 30000 nM T84631 CN2ZL1 10182437 IC50 = 8.2 nM T84631 COD9C2 10183134 IC50 = 3 nM T84631 CX9NV0 10183250 Ki = 16 nM T84631 CF4S8B 10183471 Ki = 0.6 nM T84631 CT31ZH 10183608 Ki = 152.7 nM T84631 CM0X5B 10184785 Ki = 1.4 nM T84631 C5K2GS 10185181 IC50 = 1.3 nM T84631 C7PC2K 10185292 IC50 > 170 nM T84631 CK5WD2 10185323 Ki = 15 nM T84631 C93EKT 10185327 Ki = 76.8 nM T84631 C3U1NL 10185372 Ki = 600 nM T84631 CTA49K 10185508 IC50 = 12 nM T84631 CFIH78 10185526 IC50 = 100 nM T84631 C7U3IT 10185995 Ki = 0.057 nM T84631 CU24HL 10186048 Ki = 16 nM T84631 C14TNW 10187006 Ki = 1 nM T84631 C1DN4F 10187311 Ki = 82100 nM T84631 CZ9KS7 10188952 Ki = 46 nM T84631 CG9T8S 10189755 IC50 = 1548 nM T84631 CKI5B8 10195400 Ki = 11 nM T84631 CK2Z4I 10195824 Ki = 7 nM T84631 C4P6BM 10195843 Ki = 2 nM T84631 CE3PG5 10196628 Ki = 81 nM T84631 CY5XQ6 10196732 Ki = 1 nM T84631 CO6VM1 10196955 Ki = 7396.05 nM T84631 CF2E6U 10198683 IC50 = 32000 nM T84631 CZ09JV 10202260 IC50 = 4 nM T84631 CHY62J 10203373 Ki = 2.9 nM T84631 CCV6X8 10203976 IC50 = 0.8 nM T84631 CO51ZR 10205659 Ki = 0.06 nM T84631 C2CWI1 10206231 Ki = 370 nM T84631 CFS69U 10206365 Ki = 2.4 nM T84631 CO4QT2 10207346 IC50 = 3250 nM T84631 COY39X 10207569 IC50 = 6.7 nM T84631 CW62PU 10207853 Ki = 1.6 nM T84631 CRL6T9 10207889 IC50 = 8.7 nM T84631 CT0S2D 10208075 Ki = 5 nM T84631 C1H2FS 10208201 Ki = 0.3 nM T84631 C01QTR 10209142 Ki > 75400 nM T84631 CP69QR 10212999 IC50 = 80 nM T84631 C7FTD2 10217291 Ki = 200 nM T84631 C1YOJ4 10217652 Ki = 5 nM T84631 CJRS38 10217801 Ki = 3 nM T84631 C42CUP 10217822 Ki = 370 nM T84631 CML04S 10218126 Ki = 6 nM T84631 C0DPK8 10218244 Ki = 4.8 nM T84631 CG8NY9 10218368 Ki = 73 nM T84631 C3P2VS 10218446 Ki = 2 nM T84631 CG7OS8 10225234 IC50 = 1.4 nM T84631 C6HAC0 10227428 Ki = 0.98 nM T84631 CM8O7V 10227632 Ki = 10 nM T84631 CYR45Q 10227730 IC50 > 30000 nM T84631 CIAX57 10228506 Ki > 75000 nM T84631 CSR74M 10228660 IC50 > 100000 nM T84631 CN1PX4 10228720 Ki = 29 nM T84631 CY41MS 10228870 Ki = 10 nM T84631 C98FSX 10230007 Ki = 103000 nM T84631 CMU21W 10231661 Ki = 85200 nM T84631 C87QYI 10239204 Ki = 350 nM T84631 C7G5XE 10239342 Ki = 0.17 nM T84631 CX3DY4 10239377 Ki = 2 nM T84631 CEM6N7 10239497 Ki = 1 nM T84631 C2O5HU 10239546 Ki = 53 nM T84631 CD0X3A 10239600 Ki = 23988.33 nM T84631 CSM4Y6 10239728 Ki = 4 nM T84631 CF4ND2 10247830 Ki = 5600 nM T84631 C9QML3 10250104 Ki = 57 nM T84631 CCI28E 10250490 Ki = 1.5 nM T84631 CC04IK 10253196 IC50 = 1010 nM T84631 C7RVY1 10253674 Ki = 15 nM T84631 CG8MU6 10254797 Ki = 1.5 nM T84631 C4Z1LU 10255253 Ki = 12 nM T84631 C71RTC 10255760 IC50 = 5.2 nM T84631 CS4F5P 10256448 IC50 > 100000 nM T84631 CD6V5R 10256934 IC50 = 27 nM T84631 C4WV1A 10257345 IC50 = 0.83 nM T84631 CFBN38 10257580 IC50 = 30 nM T84631 CJN34G 10258080 Ki = 0.037 nM T84631 C91KHA 10258902 Ki = 0.02 nM T84631 CVJ0I9 10258984 Ki = 0.013 nM T84631 CAM06S 10273747 IC50 = 43 nM T84631 CYZ79T 10274887 IC50 = 140 nM T84631 CQ9ZO1 10275412 Ki = 0.11 nM T84631 C50WLH 10278497 IC50 = 4 nM T84631 CL7E8K 10280735 Ki = 0.56 nM T84631 CB1S5P 10281431 Ki > 75400 nM T84631 CSEV08 10289091 Ki = 0.25 nM T84631 CMP9A5 10289373 Ki = 260 nM T84631 CXL1S0 10289409 Ki = 75000 nM T84631 C5BRU4 10289601 Ki = 13 nM T84631 CCV2P1 10289690 Ki = 28 nM T84631 CS8E7Y 10289697 Ki = 1999.86 nM T84631 CK2R3I 10290214 Ki = 0.88 nM T84631 CZM97W 10293977 Ki = 110000 nM T84631 C0T3CN 10296435 IC50 > 100000 nM T84631 CT2A4B 10297501 IC50 = 8 nM T84631 CV10CU 10297977 Ki = 0.044 nM T84631 CM62FC 10298615 IC50 = 4060 nM T84631 C1AP6H 10298858 Ki = 0.105 nM T84631 C79BFH 10298942 Ki = 0.09 nM T84631 C03FHY 10299568 IC50 = 2 nM T84631 CPX8N9 10299701 Ki = 0.23 nM T84631 CDP9R7 10299889 Ki = 29 nM T84631 CLJ02I 10300491 Ki = 0.47 nM T84631 CDY8F9 10300557 Ki = 1100 nM T84631 CEW97F 10301102 Ki = 3000 nM T84631 C6JSB5 10301730 Ki = 3 nM T84631 C29IBW 10303308 IC50 = 6.2 nM T84631 CGTF74 10303947 Ki > 75400 nM T84631 C17RDU 10304095 Ki > 10000 nM T84631 C8PA9J 10310498 Ki = 8 nM T84631 C0PQ6I 10311006 Ki = 4 nM T84631 CVYT89 10311026 Ki = 6 nM T84631 C4DQJ1 10311346 Ki = 2600 nM T84631 CU4HS2 10311517 Ki = 11 nM T84631 CHGS42 10311669 Ki = 9 nM T84631 C9N1TU 10311760 Ki < 1 nM T84631 CFTS84 10311761 Ki = 5 nM T84631 CN8FL2 10315612 Ki = 970 nM T84631 CMR75W 10318568 IC50 > 100000 nM T84631 C25XSY 10318999 IC50 = 4100 nM T84631 CGO0R3 10321806 IC50 = 60 nM T84631 C8Y4EJ 10322243 Ki > 15000 nM T84631 CMR6Y8 10323469 Ki = 1.6 nM T84631 CC7LN6 10324201 Ki = 0.05 nM T84631 C8SQ1N 10324263 IC50 = 8 nM T84631 CX9J5U 10324635 Ki = 3.7 nM T84631 C6QPK0 10324772 Ki = 100 nM T84631 CT0FX4 10325259 Ki > 8000 nM T84631 C56PEV 10325271 IC50 > 2500 nM T84631 CJ28HS 10325481 Ki = 1.8 nM T84631 CA67OL 10325720 Ki = 730 nM T84631 C41ZLB 10326602 IC50 = 4.9 nM T84631 C53QGN 10339033 Ki > 15000 nM T84631 CN5R3I 10340020 Ki = 400 nM T84631 CZMH83 10340538 IC50 = 45000 nM T84631 C4YR1M 10342318 Ki = 12000 nM T84631 CP64HV 10342843 Ki = 980000 nM T84631 C30ODG 10342944 IC50 = 1948 nM T84631 CV8J6G 10343097 Ki = 7 nM T84631 CKSH17 10343499 IC50 = 85 nM T84631 CFL57Y 10343633 Ki = 0.44 nM T84631 CK9J7X 10343728 Ki = 154 nM T84631 C4I7DQ 10345176 Ki = 0.026 nM T84631 C8FO7Q 10345230 Ki = 0.035 nM T84631 CES6C2 10345244 Ki = 5900 nM T84631 CT9GJ0 10345579 Ki = 1.1 nM T84631 CGBX39 10346320 Ki < 0.02 nM T84631 CH0RW2 10346646 IC50 = 490 nM T84631 CZ2WV3 10347131 Ki = 23 nM T84631 C3ZS2H 10347405 Ki = 1 nM T84631 C4KER5 10347610 IC50 = 18.7 nM T84631 CI4LG1 10347624 Ki = 1.8 nM T84631 CL09QG 10349678 IC50 = 290 nM T84631 C83DLG 10361934 Ki = 0.66 nM T84631 CL07UC 10364218 Ki > 10000 nM T84631 C1XV4P 10364890 IC50 = 2794 nM T84631 CW29YO 10365461 IC50 = 310 nM T84631 CH0V8B 10366070 Ki = 13 nM T84631 C0ODK9 10366157 IC50 = 16000 nM T84631 C0XW1E 10366176 IC50 = 360 nM T84631 CO0Z6Y 10366592 Ki = 1.8 nM T84631 C10ISY 10367012 Ki = 95000 nM T84631 CJ0O5P 10367277 IC50 > 33000 nM T84631 CIQ63E 10367299 IC50 = 230 nM T84631 CG98CM 10367552 Ki = 0.7 nM T84631 C5T6DO 10367956 Ki = 0.75 nM T84631 CJWE07 10368488 IC50 = 190 nM T84631 CDO83F 10368538 Ki > 75000 nM T84631 C5PR3L 10368553 Ki = 2.5 nM T84631 C9ZD0S 10368685 Ki = 0.46 nM T84631 CNV3A1 10369141 Ki = 0.055 nM T84631 CE27CV 10370457 Ki = 4400 nM T84631 C6HML8 10371129 Ki = 0.043 nM T84631 CYBF76 10386378 Ki = 6.9 nM T84631 C26CSM 10386393 IC50 = 2200 nM T84631 C71PIO 10387118 Ki > 20 nM T84631 C7TH5Q 10387956 Ki = 3 nM T84631 CMNP39 10389039 Ki = 0.7 nM T84631 CLGF71 10389462 Ki = 9 nM T84631 CE45NM 10389524 Ki = 0.16 nM T84631 CL3F1U 10389579 Ki = 2.5 nM T84631 CM6L0W 10389769 Ki > 10000 nM T84631 C4ITG3 10389930 Ki = 1 nM T84631 C47OZV 10390121 Ki = 1.2 nM T84631 C3BR5A 10390490 Ki = 2.4 nM T84631 CXF20B 10391310 IC50 = 3000 nM T84631 CJNV62 10391699 IC50 > 33000 nM T84631 C6S4CO 10391715 Ki = 8 nM T84631 CEH4D1 10391881 Ki = 14 nM T84631 CLK08Z 10391999 Ki = 0.8 nM T84631 CNS5B3 10392083 Ki = 5 nM T84631 CF6P1M 10392348 Ki = 3500 nM T84631 C94IOU 10392838 Ki = 2 nM T84631 C6QP4U 10393267 Ki = 0.1 nM T84631 CCA45U 10394183 IC50 = 59 nM T84631 CM1WJ6 10394292 Ki = 12 nM T84631 C4FBO0 10409093 Ki = 12 nM T84631 C56NXW 10409551 IC50 = 12000 nM T84631 CO3Z5D 10409945 IC50 = 1700 nM T84631 CMQY61 10410471 Ki > 15000 nM T84631 C2L8SQ 10410499 IC50 = 4200 nM T84631 C9AM3R 10410743 IC50 = 11000 nM T84631 CL34IB 10410866 Ki = 60000 nM T84631 C70AME 10411443 IC50 = 130000 nM T84631 C7K8JS 10411444 IC50 = 2218 nM T84631 C20ZSL 10411684 Ki = 0.32 nM T84631 CD0VI1 10412365 Ki = 18 nM T84631 C03MWI 10413130 Ki = 10 nM T84631 CF8M6C 10415115 Ki = 3050 nM T84631 CVK4L6 10418061 IC50 > 100000 nM T84631 CS4DL8 10433086 Ki = 13 nM T84631 C1RE8V 10433463 IC50 = 0.18 nM T84631 C4K9QX 10433872 IC50 = 9500 nM T84631 CFIC58 10434349 Ki = 0.041 nM T84631 CK3YW7 10434792 Ki = 0.087 nM T84631 C6L5IM 10434906 Ki = 1.6 nM T84631 C6AZ8B 10435038 Ki = 500 nM T84631 CX39AB 10435238 Ki = 18 nM T84631 CHCI84 10435532 Ki > 15000 nM T84631 CUM2T7 10436294 Ki = 2.5 nM T84631 C46YOA 10437408 IC50 = 5.8 nM T84631 C4L9EK 10438017 Ki = 650 nM T84631 CG07WY 10438196 Ki = 0.15 nM T84631 CL4K2S 10447733 IC50 = 112000 nM T84631 CCU35L 10453208 IC50 = 700000 nM T84631 C9M5RI 10453763 Ki > 15000 nM T84631 C4SZV0 10454685 Ki > 10000 nM T84631 C7HOX3 10454867 IC50 = 1000 nM T84631 CV9N1X 10457101 Ki = 7.2 nM T84631 C4M7SR 10458428 IC50 = 19 nM T84631 C50FMX 10458597 Ki = 550 nM T84631 C7M5HE 10459832 Ki = 0.079 nM T84631 C9W5IS 10460210 Ki = 5800 nM T84631 C9HI6A 10460541 IC50 = 1.9 nM T84631 CI87FD 10460564 IC50 = 1.2 nM T84631 CKM0N3 10460673 IC50 = 4 nM T84631 C7O6BE 10477973 Ki = 47 nM T84631 C53XJD 10478176 Ki = 560 nM T84631 C0W7NM 10478661 Ki > 15000 nM T84631 C63GRO 10479438 IC50 = 328 nM T84631 C1MX6F 10480245 Ki > 15000 nM T84631 C45KWI 10480373 Ki = 0.7 nM T84631 CCP2N8 10480374 Ki = 21 nM T84631 CV0X6G 10480463 IC50 = 0.2 nM T84631 CN1YX8 10480534 Ki = 0.074 nM T84631 CF2G8Q 10481025 Ki = 9 nM T84631 CM5A3J 10481558 Ki = 0.1 nM T84631 CMIN26 10481978 Ki = 0.32 nM T84631 CKIQ80 10482395 Ki = 0.054 nM T84631 CJ50AY 10483408 Ki = 10 nM T84631 CEI65Z 10483775 Ki = 340 nM T84631 CKL8H3 10497634 Ki = 230 nM T84631 CQE12B 10501172 Ki = 52 nM T84631 C1F7IZ 10501283 Ki = 24400 nM T84631 C6F2ZX 10501400 Ki = 52 nM T84631 CFU1E5 10501943 Ki = 110 nM T84631 CFP53Y 10502109 IC50 > 33000 nM T84631 CKI70V 10502393 Ki = 98 nM T84631 CEKX36 10503075 Ki = 1300 nM T84631 C4O9JK 10503954 Ki = 140 nM T84631 CY16UR 10504366 Ki = 1100 nM T84631 C0U6NB 10504802 Ki = 38500 nM T84631 CG5IS0 10505288 Ki = 0.005 nM T84631 C09TUO 10506433 Ki = 21 nM T84631 CXB50R 10508061 Ki = 66 nM T84631 CQS6Y2 10523322 Ki = 200 nM T84631 CFL49H 10524222 Ki = 1800 nM T84631 C87BCM 10525391 Ki = 700 nM T84631 CJ15UC 10525392 Ki = 11900 nM T84631 CD82SZ 10525943 Ki = 130 nM T84631 CZ0E8S 10526100 Ki = 34 nM T84631 C42XPE 10526785 Ki = 240 nM T84631 C7Y0WM 10527751 Ki = 41 nM T84631 CS7UC4 10528210 Ki = 280 nM T84631 CU8I0J 10528552 Ki = 4.1 nM T84631 CT41XW 10528653 Ki = 190 nM T84631 CF1PZ4 10530789 IC50 = 2000 nM T84631 CA0QG6 10531178 Ki = 0.8 nM T84631 C1K0NS 10532026 Ki = 53 nM T84631 CKYZ01 10532259 Ki = 4.2 nM T84631 C7S9QW 10532670 IC50 = 30 nM T84631 COB07E 10543987 Ki > 30000 nM T84631 CK13IY 10546004 Ki = 550 nM T84631 CO1JW8 10546322 Ki = 420 nM T84631 CEP1L6 10547293 Ki = 140 nM T84631 CO46GQ 10548215 Ki = 29000 nM T84631 CYEN07 10548429 Ki = 600 nM T84631 CEC7J6 10549325 Ki = 2200 nM T84631 C2F6CT 10549508 Ki = 12 nM T84631 CB81VQ 10551446 Ki = 440 nM T84631 CDH1F3 10552170 Ki = 440 nM T84631 CVR3P1 10552445 Ki = 130 nM T84631 C4Q5VT 10552446 IC50 = 0.008 nM T84631 CYX1V7 10553919 Ki = 9.4 nM T84631 C4J1KI 10554052 Ki = 919 nM T84631 CE8V0B 10555065 Ki = 220 nM T84631 CWR8G9 10555769 Ki = 130 nM T84631 CGQ38W 10555959 Ki = 380 nM T84631 CQG10I 10556031 Ki = 21 nM T84631 CSK8V5 10556085 Ki = 6.8 nM T84631 CGHL47 10556206 Ki = 4.3 nM T84631 CY1JF2 10569959 Ki = 940 nM T84631 CZ6HD9 10570938 Ki = 1642 nM T84631 C52FQT 10571832 Ki = 192 nM T84631 C1HA7S 10572228 Ki = 12 nM T84631 C2VG9M 10572774 Ki = 1.3 nM T84631 CV71RX 10573919 Ki = 620 nM T84631 CS8H3A 10574097 Ki = 59 nM T84631 CSHM62 10575806 Ki = 78 nM T84631 CY5O2K 10576002 Ki = 110 nM T84631 CY1A0X 10576138 Ki = 330 nM T84631 C9MN1H 10579028 Ki = 890 nM T84631 C6LO8Q 10580222 Ki = 0.32 nM T84631 C1D8GI 10580396 Ki = 0.44 nM T84631 C42LVU 10580437 Ki = 3.5 nM T84631 C02RYN 10592155 Ki = 5000 nM T84631 C4VMO3 10595198 Ki = 2800 nM T84631 CWJ68A 10596601 Ki = 95 nM T84631 CO3N1I 10597592 Ki > 10000 nM T84631 CI5CH1 10597827 Ki = 0.46 nM T84631 CT2E6F 10598802 Ki = 2.5 nM T84631 CJZF07 10599669 Ki = 7000 nM T84631 C7SEQ9 10599734 Ki = 2600 nM T84631 CD6L3E 10600145 Ki = 1100 nM T84631 CCQU28 10600245 Ki = 3.1 nM T84631 C8L9FV 10600329 Ki = 1200 nM T84631 CVEH84 10600484 Ki = 240000 nM T84631 C0SD6T 10603555 Ki = 1600 nM T84631 CP69LR 10604270 Ki = 68 nM T84631 C8CQY2 10604382 Ki < 5 nM T84631 CY1J0N 10604774 Ki = 2.1 nM T84631 C1RH3P 10621200 Ki = 654 nM T84631 CC26YF 10622456 Ki > 5000 nM T84631 CO83BP 10622800 IC50 = 120 nM T84631 C39IFP 10623057 Ki = 180 nM T84631 C5K8QJ 10623402 Ki > 100000 nM T84631 CXD95O 10623670 Ki = 720 nM T84631 CSP20T 10623756 Ki = 83 nM T84631 CZJL67 10623842 Ki = 7 nM T84631 CV0I5Y 10623890 Ki = 41 nM T84631 C3OJ4U 10623965 Ki = 0.04 nM T84631 C69VAT 10624206 Ki = 6 nM T84631 C1ZW5F 10624489 Ki = 100 nM T84631 C8SUZ9 10624948 Ki = 640 nM T84631 C8S6QZ 10625945 Ki = 1300 nM T84631 C8PHU2 10626697 Ki = 27000 nM T84631 CJ62ZG 10626722 Ki > 100000 nM T84631 CK25AY 10626893 Ki = 160000 nM T84631 CQ7F0T 10627268 Ki = 480 nM T84631 C03CIN 10628066 Ki = 2.4 nM T84631 C1PX0H 10642149 Ki = 18 nM T84631 CF3P4J 10642387 Ki = 53 nM T84631 C4KMJ8 10644692 Ki = 390 nM T84631 CZ9L8T 10644693 Ki = 18 nM T84631 C4M0QB 10645022 Ki = 140 nM T84631 C0QP4O 10645136 Ki = 9900 nM T84631 C3S0GW 10645345 Ki = 640 nM T84631 CFNH06 10645807 IC50 = 53 nM T84631 C72XTB 10646342 Ki = 225 nM T84631 CNC25X 10646757 Ki = 130 nM T84631 CRMG36 10647285 Ki = 1000 nM T84631 C1XDA6 10647609 IC50 = 950 nM T84631 CR1Y2D 10647704 Ki = 2.3 nM T84631 C76RFN 10647907 Ki = 22 nM T84631 CR5EX8 10648196 Ki = 820 nM T84631 C41KHW 10648454 Ki = 4 nM T84631 C1KVB3 10650805 Ki > 200000 nM T84631 C2OSA9 10651120 Ki > 100000 nM T84631 C6E4WZ 10651873 Ki = 2.2 nM T84631 CG40SW 10661464 Ki = 5100 nM T84631 CRDG85 10665326 Ki = 130 nM T84631 C4WCH6 10668443 Ki = 660 nM T84631 CUD8A7 10669525 Ki = 1100 nM T84631 C7CVW2 10669933 IC50 = 240 nM T84631 CD2C0U 10670479 Ki = 5.2 nM T84631 C6PAD8 10670666 Ki = 500 nM T84631 CZO1K8 10671210 Ki = 210 nM T84631 C4LJO3 10671702 Ki > 100000 nM T84631 CIKJ09 10672223 Ki = 7 nM T84631 CW1G9B 10672666 IC50 > 10000 nM T84631 CP6RF7 10673965 IC50 = 333 nM T84631 CM1Y2D 10675086 Ki = 62 nM T84631 C4TIU1 10675632 Ki = 0.008 nM T84631 C8P2UC 10675884 Ki = 8.8 nM T84631 CFQ5V2 10690751 Ki = 1850 nM T84631 CVE95Z 10691360 Ki = 24 nM T84631 CI48CW 10692578 Ki = 230 nM T84631 CD8S2B 10692579 Ki = 60 nM T84631 C4KBY2 10692711 IC50 = 6216 nM T84631 CID1F6 10693808 Ki > 33700 nM T84631 CZ53XC 10693841 Ki > 5000 nM T84631 CS08UM 10694720 Ki = 690 nM T84631 CVR1F9 10694772 Ki = 160 nM T84631 CIB63V 10694800 Ki = 3.1 nM T84631 C5VB1U 10695159 Ki = 8700 nM T84631 C2W4YZ 10695208 Ki = 220 nM T84631 CW8RV0 10696389 Ki = 8 nM T84631 CP4QC5 10696511 Ki > 1000000 nM T84631 C3QH0L 10697320 Ki = 5 nM T84631 C3WC0Q 10698376 Ki = 230000 nM T84631 CWX87E 10698758 Ki > 100000 nM T84631 C4B1DG 10712659 Ki > 5000 nM T84631 CY0P5F 10714145 Ki = 220 nM T84631 CF6TZ2 10715258 Ki = 1150 nM T84631 CK2WI6 10715476 Ki = 59 nM T84631 CZB24K 10715861 Ki = 280 nM T84631 C0TE1Z 10716448 Ki = 2400 nM T84631 C49JDV 10717698 Ki = 3300 nM T84631 CFG6T3 10717789 Ki = 100 nM T84631 CPGV87 10718240 Ki = 18000 nM T84631 CCP58N 10718840 Ki = 3.4 nM T84631 C82FPL 10718889 Ki = 120 nM T84631 CFH75T 10718950 Ki = 380 nM T84631 C1Z3PF 10719336 Ki = 0.007 nM T84631 COA5Z1 10719523 Ki = 43 nM T84631 CIKF89 10719580 Ki = 220000 nM T84631 CLXN90 10721219 Ki = 41 nM T84631 CM58XP 10721501 IC50 = 700 nM T84631 CMUX37 10722043 Ki = 240 nM T84631 CAS17I 10722747 Ki = 0.8 nM T84631 CUTA38 10723163 Ki = 0.92 nM T84631 CF9VZ0 10738109 Ki > 500 nM T84631 CZ0G6W 10738922 Ki = 130 nM T84631 C1GCY4 10739768 Ki = 2.8 nM T84631 CL7RC5 10742017 IC50 > 33000 nM T84631 C64AUD 10742143 Ki = 150 nM T84631 CK26FW 10742542 Ki = 11 nM T84631 C5L7HE 10745242 Ki > 100000 nM T84631 CAUM51 10745299 Ki = 0.01 nM T84631 CU5OG9 10746409 Ki = 6780 nM T84631 C8C1BP 10746437 Ki = 74131.02 nM T84631 C3V8JP 10746573 Ki = 0.06 nM T84631 C8J9PM 10761427 Ki = 22900 nM T84631 C9JLQ7 10761484 Ki = 2400 nM T84631 CHA46Q 10764382 Ki > 500 nM T84631 C0FTS9 10764466 Ki = 32 nM T84631 C9SDJ1 10765420 Ki = 120 nM T84631 CD51XL 10765919 Ki = 130 nM T84631 CQUM96 10765972 Ki = 370 nM T84631 C2YPX5 10766061 Ki = 0.047 nM T84631 CJSW62 10767268 Ki = 150 nM T84631 CKOQ35 10767421 Ki = 7100 nM T84631 C9SQB5 10767957 Ki = 0.009 nM T84631 CCK3E5 10768801 Ki = 8 nM T84631 C5DYQ3 10769476 Ki = 2.7 nM T84631 C62KFB 10769759 Ki = 4.1 nM T84631 C24ZSE 10769921 Ki = 11 nM T84631 C5E6AY 10770527 Ki = 2.9 nM T84631 C4Z2LQ 10770606 Ki = 1.7 nM T84631 CQW74C 10770621 Ki = 1.6 nM T84631 CCZ9U0 10770773 Ki = 1 nM T84631 C3W7TF 10770845 Ki = 1.7 nM T84631 C7VXA1 10784195 Ki = 2800 nM T84631 CJ7O1H 10785523 Ki = 5.6 nM T84631 CI9BZ1 10786604 Ki = 42 nM T84631 CQRZ02 10787180 Ki = 320 nM T84631 CD1CF3 10787181 Ki = 350 nM T84631 C0AUV8 10788046 Ki > 5000 nM T84631 C4CAT2 10788047 Ki = 4.8 nM T84631 CRHE34 10788206 Ki = 190 nM T84631 CD21MW 10788364 Ki = 9800 nM T84631 CKLU46 10788963 Ki = 395 nM T84631 C0RL4C 10789777 Ki = 250 nM T84631 CMX5V9 10789805 Ki = 970 nM T84631 CT8M1C 10790019 Ki = 310 nM T84631 CL73OX 10791003 Ki = 160000 nM T84631 C5TID3 10791816 Ki = 120 nM T84631 CBNP58 10792157 Ki = 56 nM T84631 CRD65S 10792619 Ki > 200000 nM T84631 CLWY92 10793236 Ki = 14000 nM T84631 C5ENU2 10794450 Ki = 0.11 nM T84631 C64ZVF 10794532 Ki = 4.2 nM T84631 CC95IV 10794535 Ki = 8.5 nM T84631 CD6U1P 10806942 Ki = 1400 nM T84631 CR51LN 10807566 Ki = 4579 nM T84631 CYAJ14 10810195 Ki = 4.6 nM T84631 CL9O0C 10810196 Ki = 500 nM T84631 CUQX02 10810754 Ki = 340 nM T84631 C74QCG 10811600 Ki = 1200 nM T84631 C0U7PJ 10811747 Ki = 510 nM T84631 CYS08X 10813043 Ki = 14 nM T84631 CQK97I 10813230 Ki = 49 nM T84631 C3WX4F 10813359 Ki = 2.4 nM T84631 C13KAX 10813709 Ki = 70 nM T84631 CZA0D1 10814968 Ki = 0.02 nM T84631 CE1DT2 10815540 Ki = 25 nM T84631 CV1U5L 10816337 Ki = 31 nM T84631 CL8YB0 10816451 Ki = 34 nM T84631 CPRS52 10817210 Ki = 7600 nM T84631 CSZR21 10817699 Ki = 9.9 nM T84631 CUS6D0 10818009 Ki = 19 nM T84631 C0M3XB 10831506 Ki = 53 nM T84631 C9HPZ8 10831834 IC50 = 6300 nM T84631 CE2LP4 10832026 Ki > 5000 nM T84631 CLXP56 10833102 Ki = 1400 nM T84631 C6NW5I 10833234 Ki > 5000 nM T84631 CJ2M4I 10835535 Ki = 23 nM T84631 CW8OT1 10835646 Ki = 110 nM T84631 C2KXJ7 10835995 Ki = 750 nM T84631 CH0RG9 10836919 Ki = 570 nM T84631 C67FIC 10837478 Ki = 55 nM T84631 CW3YA2 10837929 Ki = 120 nM T84631 C1FTR2 10837980 Ki = 6 nM T84631 C5FSB0 10838473 Ki = 62 nM T84631 CM13CR 10840852 Ki = 0.6 nM T84631 CYX51H 10840933 Ki = 7.2 nM T84631 CZVR32 10841125 Ki = 10000 nM T84631 COLC79 10841532 Ki = 52000 nM T84631 C6QF7T 10841535 Ki = 17800 nM T84631 C2R7OQ 10841758 Ki = 3.3 nM T84631 CJRU60 10860637 Ki = 948 nM T84631 CBK06L 10861643 IC50 > 60000 nM T84631 C6F2ZP 10863119 Ki = 10000 nM T84631 C7U4IT 10863260 Ki = 1720 nM T84631 CB38YZ 10863406 Ki > 5000 nM T84631 CK7VC8 10863579 Ki = 820 nM T84631 C07BLI 10864217 Ki = 50 nM T84631 C62IPV 10864710 Ki = 11 nM T84631 C02XLH 10865109 IC50 = 240 nM T84631 CZX59B 10865289 Ki = 14 nM T84631 C9LEJ0 10865386 IC50 = 1700 nM T84631 C1BOZ5 10865461 IC50 = 270 nM T84631 CN2CE8 10865462 IC50 = 610 nM T84631 CLB15C 10871563 Ki > 75000 nM T84631 CWVZ13 10873723 Ki = 262 nM T84631 CD7I4A 10873871 Ki = 1800 nM T84631 CPSW72 10873946 Ki = 45 nM T84631 C0KIZ5 10874086 Ki = 220 nM T84631 CXG62W 10874449 Ki = 38 nM T84631 C3Z6PT 10874628 IC50 > 30000 nM T84631 C2TH3I 10875009 Ki = 154 nM T84631 C7YEP4 10875960 IC50 = 2400 nM T84631 C80WCU 10883641 Ki = 1700 nM T84631 CTAF76 10884388 Ki = 19 nM T84631 CAR7T6 10884739 Ki = 5310 nM T84631 CZP9L7 10884798 Ki = 1556 nM T84631 CJWL05 10884908 Ki = 798 nM T84631 C1PNQ4 10885181 Ki > 5000 nM T84631 C27LWG 10885612 Ki = 99 nM T84631 C8EG3O 10886723 Ki = 226 nM T84631 CK6T4L 10892244 Ki = 10000 nM T84631 CCA1Q7 10894246 Ki = 6890 nM T84631 CU8J0C 10894269 Ki = 28 nM T84631 CNL3H2 10894415 Ki = 2000 nM T84631 CJGS43 10894874 Ki = 26 nM T84631 CW9MC1 10894892 Ki = 5800 nM T84631 C49BRD 10894895 Ki = 320 nM T84631 CW7Q2U 10895700 IC50 > 250000 nM T84631 C16NXJ 10896126 Ki = 13 nM T84631 CKY20H 10896140 Ki > 5000 nM T84631 CMP45U 10896308 Ki = 2700 nM T84631 C1YPJ0 10896662 Ki = 42 nM T84631 C39AVR 10897080 Ki = 7 nM T84631 C59ETF 10897550 Ki = 23 nM T84631 C2GPU4 10897682 IC50 = 1030 nM T84631 CQTC02 10903566 Ki = 6800 nM T84631 C8J1TX 10904089 Ki <= 11000 nM T84631 CR9G0E 10905722 Ki = 1200 nM T84631 CB1HW4 10905809 IC50 > 30000 nM T84631 C1F8UV 10905825 Ki = 3600 nM T84631 C9C6UE 10906426 Ki = 600 nM T84631 CH2G5Q 10906977 Ki > 75000 nM T84631 CTM36K 10907121 Ki = 5500 nM T84631 C3FY5S 10907552 Ki = 133 nM T84631 CPJ1Q7 10908669 IC50 = 160 nM T84631 C9E7RY 10908791 IC50 = 1250 nM T84631 C2BXU9 10908808 IC50 = 300 nM T84631 C5I7SU 10916321 Ki = 530 nM T84631 CA1IB4 10916653 Ki = 4000 nM T84631 CX3FP2 10917491 Ki > 5000 nM T84631 C7K5SQ 10918066 Ki = 160 nM T84631 COQY14 10918387 Ki = 2064 nM T84631 CCDO06 10919424 Ki = 84 nM T84631 C5A8NU 10919581 IC50 = 570 nM T84631 CMK60F 10927859 Ki = 720 nM T84631 CKI49C 10928313 Ki = 21000 nM T84631 CR5VW1 10928435 Ki = 15 nM T84631 CMK6P8 10928757 IC50 > 30000 nM T84631 CK6E0Q 10928936 Ki = 840 nM T84631 C7Z6JY 10929059 Ki = 6790 nM T84631 C1KV7H 10929853 Ki = 28 nM T84631 CT5H0B 10929908 Ki = 50 nM T84631 C1Q9WZ 10930326 IC50 = 2120 nM T84631 CL20KX 10930722 IC50 = 1070 nM T84631 CG7NA5 10938859 Ki > 1200 nM T84631 C8RF5U 10938960 Ki = 500 nM T84631 CMD6C0 10939317 Ki = 26 nM T84631 CC81OU 10939381 Ki = 1300 nM T84631 CT4G3S 10939409 Ki = 2700 nM T84631 CDSU98 10939678 Ki > 5000 nM T84631 C3MY5I 10940389 Ki = 85 nM T84631 CG5BN9 10940660 Ki = 160 nM T84631 CSZX24 10941224 Ki = 24 nM T84631 C5ED3R 10946700 Ki = 7910 nM T84631 C8OA1L 10946869 Ki = 43000 nM T84631 CUN98K 10949030 Ki = 1350 nM T84631 C3NR1O 10949672 Ki = 131 nM T84631 CCM7H1 10949960 Ki = 400 nM T84631 CJDM01 10950292 Ki = 2400 nM T84631 C95WOX 10950363 Ki = 1800 nM T84631 CUWF38 10950398 Ki = 68 nM T84631 CWN81P 10950417 Ki = 20 nM T84631 CT3BN9 10951324 Ki = 18 nM T84631 C2TBO9 10959252 Ki = 26000 nM T84631 C0B9VT 10960935 Ki = 1400 nM T84631 CB9KP4 10961420 Ki = 21 nM T84631 C6ZT5K 10961564 Ki = 1200 nM T84631 C8MSV2 10961726 Ki = 325 nM T84631 C9RTW1 10961857 Ki > 1200 nM T84631 CITU70 10962439 Ki > 75000 nM T84631 CCE31H 10963578 IC50 = 185 nM T84631 CJ29QP 10972004 Ki = 183 nM T84631 CH0VN7 10972370 IC50 > 30000 nM T84631 CFC7J3 10972388 Ki = 300 nM T84631 CT6Q7Z 10972928 Ki = 39 nM T84631 CIU42D 10973463 IC50 > 30000 nM T84631 C6HG4P 10974490 IC50 = 2700 nM T84631 CVT26S 10974535 IC50 = 540 nM T84631 CH41ZW 10974733 IC50 = 2400 nM T84631 CE0F1L 10983499 Ki > 1200 nM T84631 CPO91R 10983794 Ki = 13 nM T84631 CL9V7T 10984300 Ki = 18 nM T84631 CWVR40 10985371 IC50 = 2000 nM T84631 C9Y8LS 10991007 Ki = 6 nM T84631 CB79YS 10993022 Ki = 3327 nM T84631 C3RCS5 10994039 Ki = 900 nM T84631 CN0T4L 10994091 Ki = 690 nM T84631 CM5Y6J 10994432 IC50 > 30000 nM T84631 C4VA7K 10994660 IC50 > 30000 nM T84631 CZM0S7 10995244 Ki = 360 nM T84631 CT7L2Q 10996309 IC50 = 1000 nM T84631 C43SNO 11004109 Ki = 89 nM T84631 CF26JG 11004176 Ki = 280 nM T84631 CK3N5I 11004200 Ki = 620 nM T84631 CV86TU 11004465 Ki = 370 nM T84631 CP68KV 11004693 Ki = 460 nM T84631 C8AG4Z 11005226 IC50 > 30000 nM T84631 C12REQ 11005350 Ki = 918 nM T84631 CWHG91 11005419 Ki = 180 nM T84631 C0FG9E 11006294 Ki = 60 nM T84631 CC39SB 11009950 Ki = 125000 nM T84631 C3HW2I 11014107 Ki = 3300 nM T84631 CYZL25 11015002 Ki = 210 nM T84631 CFO15P 11015356 IC50 > 30000 nM T84631 CE7BX4 11015410 Ki = 1230 nM T84631 C56HDX 11015700 Ki > 5000 nM T84631 C5IS6E 11016482 Ki = 23 nM T84631 CV8O4G 11016622 Ki = 3 nM T84631 C49NMW 11022696 Ki = 5650 nM T84631 CM37HW 11025449 Ki = 1300 nM T84631 C71KSB 11026329 Ki > 1200 nM T84631 C4EX2J 11026555 Ki > 5000 nM T84631 CYKF85 11026584 Ki = 810 nM T84631 C21MKH 11026850 Ki = 140 nM T84631 CD4LJ1 11027118 IC50 > 30000 nM T84631 C46ZEX 11027375 Ki = 19 nM T84631 CI0VR4 11028729 Ki = 82 nM T84631 C2RG6V 11028969 IC50 = 180 nM T84631 CMQ65P 11035180 Ki = 2986 nM T84631 C3QG7H 11036285 Ki = 20 nM T84631 CV1F8Q 11036379 Ki = 170 nM T84631 C5KTL2 11037540 Ki = 89 nM T84631 CXO97Q 11037642 Ki = 25 nM T84631 CDGL91 11037810 Ki = 2043 nM T84631 C7PDA1 11037845 Ki = 17350 nM T84631 C9KL0E 11037866 Ki = 7030 nM T84631 C4LPB1 11039096 Ki > 5000 nM T84631 C7RM5W 11039881 IC50 = 210 nM T84631 C7P5EN 11039916 IC50 = 2180 nM T84631 C7VX2Y 11046972 Ki = 3200 nM T84631 CSQT80 11048143 Ki = 1118 nM T84631 CMBL62 11048452 Ki = 9 nM T84631 CA1U0X 11048482 Ki = 10000 nM T84631 CJL15S 11048586 Ki = 63 nM T84631 CF01BA 11049038 Ki = 19 nM T84631 C4SW1T 11049045 Ki = 1022 nM T84631 C4UY7P 11050903 IC50 = 770 nM T84631 CD9WJ8 11057540 Ki = 340 nM T84631 C2Y6VW 11057779 Ki = 14 nM T84631 CQ61ZR 11059085 IC50 > 30000 nM T84631 CJZ10A 11059370 Ki = 3000 nM T84631 C7IA8Y 11059381 Ki = 3804 nM T84631 CZ43QG 11059512 Ki = 1400 nM T84631 CX09AC 11059549 Ki > 5000 nM T84631 CH1OX5 11059588 Ki = 4 nM T84631 C8BC4U 11059598 Ki > 1200 nM T84631 CXW4P2 11059783 Ki = 160 nM T84631 C8L9KE 11059896 IC50 > 30000 nM T84631 CYG09F 11059945 Ki = 370 nM T84631 CRK76W 11060981 Ki = 140 nM T84631 CVGU32 11067332 Ki = 13000 nM T84631 C3HNB2 11068806 Ki = 78 nM T84631 CU02AK 11069944 Ki = 959 nM T84631 CJ4U7M 11069959 Ki = 5200 nM T84631 C7CX9Y 11070206 Ki = 128 nM T84631 C5D6CK 11070239 Ki = 77 nM T84631 CZY36H 11071021 Ki = 1628 nM T84631 CZU7P2 11071979 Ki = 94 nM T84631 C7YDH0 11072681 IC50 = 150 nM T84631 CDKX73 11080299 Ki = 263 nM T84631 CW3QV0 11080411 Ki = 2100 nM T84631 CZ5PW9 11080476 Ki = 308 nM T84631 CSE89U 11081058 Ki = 1219 nM T84631 CZ73WT 11081112 Ki = 3 nM T84631 C0FVC8 11082011 Ki = 61 nM T84631 CRIM63 11082881 Ki = 245 nM T84631 C2XYV1 11091496 Ki = 970 nM T84631 CB21LS 11092876 Ki = 1820 nM T84631 CXO16G 11092974 Ki = 14 nM T84631 CUX7H5 11098880 Ki = 7160 nM T84631 C0UP3R 11101386 Ki = 2032 nM T84631 C9CUO6 11102065 IC50 > 30000 nM T84631 C2XAM1 11102245 Ki = 650 nM T84631 CM1F6C 11102508 Ki = 2200 nM T84631 CY3M6F 11102509 Ki = 2400 nM T84631 C7DF0B 11102544 Ki = 193 nM T84631 C8R5EM 11102680 Ki = 476 nM T84631 CVB8L0 11102692 Ki = 37 nM T84631 C1U0NG 11102698 Ki = 841 nM T84631 C1GY8M 11102714 Ki = 1400 nM T84631 CU53EA 11104490 IC50 = 250 nM T84631 C41PZK 11112423 Ki = 64 nM T84631 C9KE6A 11112625 Ki = 210 nM T84631 C59EGY 11112713 Ki = 240 nM T84631 CI3N0C 11112769 Ki = 1360 nM T84631 CPD34Y 11112824 Ki = 48 nM T84631 CZV69J 11112866 Ki = 1200 nM T84631 CANW92 11112933 IC50 > 30000 nM T84631 CC37UH 11113237 Ki = 274 nM T84631 CAGC62 11113397 Ki = 304 nM T84631 CKL74M 11113517 Ki = 3 nM T84631 CS14TD 11113557 Ki = 318 nM T84631 CBY3A4 11113676 Ki > 5000 nM T84631 C30NPX 11113694 Ki = 2800 nM T84631 CEP79U 11122516 Ki > 5000 nM T84631 CDIS79 11122714 Ki = 1600 nM T84631 C03CFY 11122823 Ki > 5000 nM T84631 CALC18 11123099 Ki = 2000 nM T84631 CE4DH7 11123192 Ki = 173 nM T84631 CJBF29 11123629 Ki = 117 nM T84631 C39ATZ 11124077 Ki = 5000 nM T84631 CT50NB 11124237 Ki = 170 nM T84631 C47UEP 11125405 IC50 = 900 nM T84631 CD71SV 11125697 IC50 = 500 nM T84631 C0KYJ6 11133405 Ki = 1608 nM T84631 C39IZS 11134001 Ki = 4500 nM T84631 CT7S6O 11134002 Ki > 5000 nM T84631 CQ7X3J 11134090 Ki = 707 nM T84631 CY7E9X 11135514 Ki = 610 nM T84631 CD56CJ 11135734 Ki = 141 nM T84631 C0SG9J 11136398 IC50 = 250 nM T84631 C9KL8Y 11144992 Ki > 1200 nM T84631 CMX1S2 11146905 IC50 = 330 nM T84631 CWMD96 11146965 IC50 = 2770 nM T84631 C1NMK4 11146971 IC50 = 310 nM T84631 CS1K9H 11156015 Ki = 225200 nM T84631 C2TL3I 11156562 Ki = 110 nM T84631 CK3RG5 11157000 Ki = 2.9 nM T84631 CT2ML6 11157065 Ki = 10000 nM T84631 CJ4X7R 11158066 IC50 = 65000 nM T84631 C83DUK 11164311 IC50 = 3340 nM T84631 C5KG1A 11164549 Ki > 10000 nM T84631 CRD42J 11168063 Ki = 7.1 nM T84631 C3WKQ1 11168297 Ki = 2.8 nM T84631 CRG25K 11168660 IC50 = 190 nM T84631 C8KQY0 11168755 Ki = 10000 nM T84631 C58IYE 11169197 Ki = 17300 nM T84631 CIF5K2 11178928 Ki = 2 nM T84631 CZC46I 11179149 IC50 = 26 nM T84631 COM9K4 11179316 IC50 = 4300 nM T84631 CTM80Q 11179758 IC50 = 74 nM T84631 CEO0A3 11179888 Ki = 7 nM T84631 CU9K4E 11180045 IC50 = 22 nM T84631 C9X4JY 11181893 Ki = 0.37 nM T84631 CR0S7Z 11188883 Ki = 7800 nM T84631 CY70EN 11191165 IC50 > 10000 nM T84631 CB25UF 11191236 Ki = 1.1 nM T84631 C2RVF5 11191430 IC50 = 320 nM T84631 C68FEJ 11191721 IC50 = 105 nM T84631 CER29V 11197304 IC50 > 5000 nM T84631 CWA6L1 11202766 IC50 = 230 nM T84631 CAM0I3 11203305 Ki = 54 nM T84631 CJ6CW4 11203935 Ki = 38 nM T84631 C9J5HC 11212885 Ki = 87 nM T84631 CVG72J 11213445 Ki = 2221 nM T84631 CR5S8A 11214337 Ki = 2518 nM T84631 C9BY1M 11214717 Ki = 950 nM T84631 CO7H9G 11214939 Ki = 16590 nM T84631 CKH8E1 11215005 Ki = 71 nM T84631 C8BRJ1 11225386 Ki = 5.3 nM T84631 CSJW59 11226109 Ki = 7 nM T84631 CYQ3J1 11226153 Ki = 4327 nM T84631 C7MT4K 11226168 Ki = 5755 nM T84631 C7DJT1 11226460 Ki = 8 nM T84631 CP51FI 11226542 Ki = 1.7 nM T84631 CQZ7S2 11236581 Ki = 140 nM T84631 CVK0I4 11237021 IC50 = 1980 nM T84631 CLA93S 11237163 Ki = 0.67 nM T84631 CB29QS 11237358 Ki = 1540 nM T84631 CY8O2E 11237428 Ki = 7700 nM T84631 C37VTL 11238193 Ki = 62 nM T84631 CA3IS9 11248439 Ki = 2.8 nM T84631 CI0NE7 11248994 Ki = 9 nM T84631 CUP5C4 11249230 Ki = 1 nM T84631 C98HOZ 11249318 Ki = 1.8 nM T84631 C75IPG 11249648 Ki = 124 nM T84631 CE2JK3 11249816 Ki = 264 nM T84631 CHQ50D 11260319 IC50 = 420 nM T84631 CI9D8E 11260802 Ki = 10000 nM T84631 CN0EI2 11260937 Ki = 1051 nM T84631 CF0WU1 11261069 Ki = 4883 nM T84631 C7WIZ3 11261098 IC50 = 2900 nM T84631 C9MJA2 11271356 Ki = 2820 nM T84631 C2AFH8 11271916 IC50 = 230 nM T84631 CRDU42 11271947 Ki = 15 nM T84631 CYRO76 11272254 IC50 = 60 nM T84631 CW4OK6 11272980 Ki = 18 nM T84631 C92KFX 11273269 IC50 = 110 nM T84631 C73WSC 11273795 IC50 > 20000 nM T84631 CQP45I 11283566 Ki = 2 nM T84631 CZJ9C8 11283614 IC50 = 718 nM T84631 C91BDA 11284460 IC50 = 1900 nM T84631 CSH76U 11284767 Ki = 54600 nM T84631 CJ82SB 11294750 IC50 = 493 nM T84631 CO7LS5 11294802 Ki = 26 nM T84631 CEF02R 11294993 Ki = 0.53 nM T84631 CXQO17 11295553 Ki = 2574 nM T84631 C2WG5Z 11295972 Ki = 8 nM T84631 C3ZX2E 11295984 Ki = 810 nM T84631 CL79GU 11303092 IC50 = 4060 nM T84631 CTZ7X4 11306388 Ki = 2 nM T84631 CNCL81 11306615 Ki = 21 nM T84631 CA80VZ 11306712 Ki = 16 nM T84631 CL2GZ0 11306789 IC50 = 160 nM T84631 C71PYV 11307226 IC50 = 22 nM T84631 C72IDM 11307246 Ki = 47 nM T84631 C7L9MF 11307344 Ki = 421 nM T84631 C0TUI9 11307532 Ki = 0.54 nM T84631 CF9RM8 11307929 Ki = 17 nM T84631 CNUP65 11316684 Ki = 1.1 nM T84631 C5ZC1G 11317814 Ki = 2 nM T84631 C3L6GK 11318187 IC50 = 230 nM T84631 CP08JC 11318191 IC50 = 550 nM T84631 C7ZS2B 11320069 Ki = 0.7 nM T84631 CY87CQ 11329232 Ki = 5410 nM T84631 C14AWK 11329397 Ki = 1412 nM T84631 CTXB71 11329441 IC50 = 270 nM T84631 CUCB51 11329534 Ki = 3 nM T84631 C4K3SW 11329788 Ki = 3925 nM T84631 C3J7WN 11329826 IC50 = 255 nM T84631 CB46ZC 11329971 IC50 = 210 nM T84631 CVAI21 11330048 Ki = 3.6 nM T84631 CC6O0W 11340558 Ki = 8.1 nM T84631 CJI8G5 11340774 IC50 = 800 nM T84631 CSJZ70 11341303 Ki = 960 nM T84631 CW7E9F 11341378 Ki = 2184 nM T84631 C64EOX 11341794 Ki = 28 nM T84631 CR8NW9 11351302 Ki = 1.5 nM T84631 CK28PW 11351714 Ki = 173 nM T84631 CY9D3C 11352421 IC50 = 5.5 nM T84631 C12OTG 11352538 Ki = 20 nM T84631 C3FC4B 11352678 Ki = 17 nM T84631 CSIM71 11353123 Ki = 20 nM T84631 C1HON4 11353394 Ki = 153 nM T84631 C1V5ES 11363818 IC50 = 1350 nM T84631 CQ9BZ3 11363906 Ki = 42 nM T84631 CVA12Y 11363985 Ki = 3 nM T84631 CK51RW 11364032 Ki = 24 nM T84631 CT83NF 11364269 Ki = 22 nM T84631 C1ZGT7 11364310 Ki = 10000 nM T84631 CR04CN 11364346 Ki = 0.7 nM T84631 CY2HW5 11365859 Ki = 4.5 nM T84631 CBU78I 11373015 IC50 = 510 nM T84631 C4U9OQ 11374975 IC50 = 510 nM T84631 C52YOA 11375433 IC50 = 390 nM T84631 CDS70L 11375712 IC50 = 247 nM T84631 CUNB34 11377164 IC50 = 83 nM T84631 CJBD34 11386051 Ki = 2.6 nM T84631 CWUY06 11386385 Ki = 5 nM T84631 CB41UN 11386766 Ki = 1265 nM T84631 CIWL90 11386810 Ki = 10 nM T84631 COQH61 11387388 Ki = 55 nM T84631 C8URO7 11387451 Ki = 0.88 nM T84631 C6U5OI 11387989 Ki = 61 nM T84631 CDC76X 11396607 Ki = 9.5 nM T84631 CZ4EM5 11397605 Ki = 4.4 nM T84631 C5MYX8 11397764 Ki = 2.6 nM T84631 CV4I7J 11397824 IC50 = 6200 nM T84631 CVU08E 11397915 IC50 = 3.5 nM T84631 CU5H0T 11398145 IC50 = 270 nM T84631 C1MS0G 11398207 Ki = 6200 nM T84631 C2M1OW 11398411 Ki = 970 nM T84631 CM34VR 11398878 Ki = 10000 nM T84631 CR9Q3O 11399867 IC50 = 1400 nM T84631 C3O9MG 11408346 Ki = 4219 nM T84631 CS8TK0 11408450 Ki = 1.8 nM T84631 CR9Y7U 11408532 Ki = 4.7 nM T84631 C3DQ7J 11409073 IC50 = 120 nM T84631 C3KYM8 11409900 IC50 = 190 nM T84631 CPF6V4 11410761 Ki = 10000 nM T84631 C8WZ0P 11416498 Ki > 10000 nM T84631 CJI48N 11419907 Ki = 9345 nM T84631 CAI3Y6 11420126 Ki = 74 nM T84631 CODR29 11420832 Ki > 75000 nM T84631 CR9OZ8 11420936 Ki = 14 nM T84631 C8R5QT 11420982 Ki = 10000 nM T84631 CUHD35 11421628 Ki = 800 nM T84631 CTY4I2 11431806 Ki = 230 nM T84631 C9HIK8 11432017 Ki = 1128 nM T84631 C9UE5W 11432325 Ki = 5 nM T84631 CZ3C9N 11432971 Ki = 9 nM T84631 CH74DF 11433275 Ki = 835 nM T84631 CLH6X5 11433511 Ki = 1 nM T84631 CCPU80 11434124 Ki = 7.7 nM T84631 CN46CG 11441985 IC50 = 56 nM T84631 CW36NJ 11442160 Ki = 406 nM T84631 C9DQ6J 11443267 Ki = 34 nM T84631 CSI0R8 11443686 Ki = 3040 nM T84631 CNU51Z 11443953 Ki = 1484 nM T84631 CZ2YU6 11444061 Ki = 10000 nM T84631 CH7X6T 11444549 Ki = 10000 nM T84631 CIQH43 11445130 IC50 = 3600 nM T84631 CM7DK5 11445304 Ki = 0.16 nM T84631 C10PTA 11454249 Ki = 1 nM T84631 CFL61Z 11454667 Ki = 270 nM T84631 CB60QJ 11455408 Ki = 15 nM T84631 COC38U 11455413 Ki = 6217 nM T84631 C05LOJ 11455486 IC50 = 86 nM T84631 CG8H7N 11465140 IC50 = 5.5 nM T84631 CNF2M3 11465752 Ki = 650 nM T84631 CWC4B0 11465955 Ki = 3.7 nM T84631 C7B1LU 11466448 Ki = 10000 nM T84631 CYSI10 11466604 Ki = 13 nM T84631 CX31CK 11466687 Ki = 57 nM T84631 C89DVO 11466821 Ki = 1247 nM T84631 C8KJ1G 11466928 Ki = 110 nM T84631 C13CGX 11466988 Ki = 31 nM T84631 CU9LH8 11466995 IC50 = 400 nM T84631 C0T6CN 11467119 Ki = 600 nM T84631 CH4V9C 11468062 Ki = 0.1 nM T84631 CUF04L 11468141 Ki = 163 nM T84631 CJ6TL8 11468217 Ki = 0.52 nM T84631 C6P9OD 11477087 IC50 = 1300 nM T84631 CAC5N9 11477894 Ki = 2.3 nM T84631 CD31BU 11478099 IC50 = 5440 nM T84631 CLO07F 11478314 Ki = 10000 nM T84631 CU04WZ 11478333 Ki = 2.4 nM T84631 C85JCH 11478408 Ki = 130 nM T84631 C73GXV 11479028 Ki = 18 nM T84631 CVI82D 11479420 Ki = 0.09 nM T84631 CDKN64 11488503 Ki = 4.2 nM T84631 CGY6X5 11488924 Ki = 407 nM T84631 CB1PG7 11489024 IC50 = 640 nM T84631 CF15XY 11489042 IC50 = 920 nM T84631 C5DFC7 11489269 IC50 = 1200 nM T84631 CC5DO0 11489287 IC50 = 2200 nM T84631 CU2JO0 11489417 Ki = 463 nM T84631 C50FQZ 11489885 Ki > 200000 nM T84631 CI65TJ 11490312 IC50 = 80 nM T84631 C9R6LC 11496149 Ki = 4 nM T84631 C84NJM 11496686 IC50 = 3.6 nM T84631 CZ30GX 11497599 Ki = 5.5 nM T84631 C81ZHR 11503981 Ki = 0.33 nM T84631 CK34OX 11509611 Ki > 8180 nM T84631 CO1AY9 11509879 Ki = 223 nM T84631 CJZ09N 11512593 Ki = 5100 nM T84631 C28BMR 11513105 Ki = 4900 nM T84631 CLN0W3 11517577 IC50 = 1170 nM T84631 C1BV2R 11518043 IC50 = 197 nM T84631 C13UZL 11518307 Ki = 0.19 nM T84631 CLT1I0 11518907 Ki = 0.033 nM T84631 CKAE28 11519499 Ki = 3 nM T84631 CV6JF2 11523750 IC50 = 74 nM T84631 CO68MA 11524737 Ki > 8180 nM T84631 C0A6TY 11524901 IC50 = 2300 nM T84631 CKN8R7 11525275 IC50 = 1900 nM T84631 C20NQD 11525292 IC50 = 1.4 nM T84631 CRNU10 11534959 Ki = 4100 nM T84631 C9M6JZ 11538422 Ki = 2900 nM T84631 CUY97G 11539245 IC50 = 94 nM T84631 CD1A6T 11542037 Ki = 2800 nM T84631 CA8KD7 11542038 Ki = 1200 nM T84631 CKY49D 11546456 IC50 = 2000 nM T84631 CDS27O 11553603 IC50 = 40 nM T84631 CLQ1A9 11554212 IC50 = 8.5 nM T84631 CBP69L 11557024 Ki = 9500 nM T84631 CE4DV8 11561857 Ki = 5 nM T84631 CKJC51 11561914 Ki = 6 nM T84631 C2KM3Z 11562451 IC50 = 1 nM T84631 C3EMG1 11562571 IC50 = 2.3 nM T84631 CCG84F 11563457 Ki = 2300 nM T84631 CV46NL 11563632 Ki > 1000000 nM T84631 C4JLC8 11569203 IC50 = 0.4 nM T84631 CEAZ46 11569930 Ki = 66000 nM T84631 C3TJ7M 11570580 Ki = 1800 nM T84631 C6RHD8 11570700 Ki = 13000 nM T84631 C1DN2L 11570759 Ki = 80000 nM T84631 C9R6VJ 11575714 IC50 = 1260 nM T84631 C6FG8V 11577055 Ki = 76000 nM T84631 CIY34V 11577968 Ki = 8300 nM T84631 CJ38EP 11577970 Ki = 10500 nM T84631 C7MF9N 11578158 Ki = 3200 nM T84631 C6A0XP 11583256 IC50 = 2.5 nM T84631 C5W7FH 11583355 Ki = 5 nM T84631 C76BVQ 11583800 IC50 = 9.1 nM T84631 CTSK74 11584729 Ki = 21000 nM T84631 C96GNS 11585914 IC50 = 9500 nM T84631 C5W4SM 11590677 Ki = 0.3 nM T84631 C1RQ6P 11592130 Ki = 23000 nM T84631 CBC84M 11592593 Ki = 13000 nM T84631 C7ZS8L 11592600 Ki = 4600 nM T84631 C7QTY8 11606981 Ki = 2000 nM T84631 CU07NO 11607091 Ki = 17000 nM T84631 CC94FI 11612290 Ki = 0.028 nM T84631 CL9TZ2 11614477 Ki = 5000 nM T84631 C78TFB 11618984 IC50 = 290 nM T84631 CA56HC 11619782 IC50 = 1200 nM T84631 CB4O2Q 11621579 Ki = 2800 nM T84631 CD3R1E 11627899 Ki = 35000 nM T84631 CB9P0Q 11628768 Ki = 10000 nM T84631 CO3Q9N 11635973 Ki = 9000 nM T84631 CRX98P 11636026 Ki = 2800 nM T84631 C8N5CR 11638121 Ki = 1 nM T84631 CMC85Y 11641579 Ki = 3 nM T84631 CW10CL 11642802 Ki = 25000 nM T84631 C1O5ZV 11648797 Ki = 314000 nM T84631 CE3D4T 11650066 IC50 = 7.6 nM T84631 CZL5O6 11650704 Ki = 5.2 nM T84631 C7NG4M 11652744 Ki = 1 nM T84631 C2W5XF 11656797 Ki = 15000 nM T84631 C4SAR0 11657278 Ki = 1300 nM T84631 CVQ16C 11664107 Ki = 34000 nM T84631 CPZG49 11664334 Ki = 130000 nM T84631 CT9E0G 11664643 Ki = 2900 nM T84631 CWV87X 11671266 Ki = 15000 nM T84631 CE0A6N 11671776 Ki = 5300 nM T84631 C85GCY 11671956 Ki = 5800 nM T84631 C1IMQ2 11677338 Ki = 0.06 nM T84631 C1DHO6 11678360 Ki = 24000 nM T84631 C4IBO3 11678764 Ki = 2200 nM T84631 CJP9O1 11684611 Ki = 6390 nM T84631 C69YSR 11693028 Ki = 6300 nM T84631 CCQY30 11693049 Ki = 4000 nM T84631 CS27RX 11697174 Ki = 175 nM T84631 C0YO6U 11698686 Ki = 0.2 nM T84631 CPFW75 11699600 Ki = 13000 nM T84631 C3VS2H 11699903 Ki = 2300 nM T84631 CNV09Z 11699913 Ki = 1000 nM T84631 CI96PN 11704628 Ki = 124 nM T84631 C89KHJ 11707555 IC50 = 9600 nM T84631 CCVY81 11711363 IC50 = 4.2 nM T84631 CM57QZ 11718954 IC50 = 29 nM T84631 CKQ4O2 11721188 Ki = 56000 nM T84631 C4UB2X 11721375 Ki = 10000 nM T84631 C4M0XP 11725377 IC50 = 940 nM T84631 CJZA24 11729069 Ki = 2500 nM T84631 CL4CN3 11729890 Ki = 208 nM T84631 CS12RM 11730232 Ki = 45 nM T84631 CBJ4R6 11730277 Ki = 12000 nM T84631 CQ0ZP6 11730472 Ki > 1200 nM T84631 CL8HU6 11730709 IC50 > 30000 nM T84631 C7D8HR 11731179 Ki = 99 nM T84631 CN70PY 11732209 Ki = 1112 nM T84631 CW1U7K 11732650 Ki = 2190 nM T84631 C0VO1S 11732813 Ki = 191 nM T84631 C8K1ZJ 11733007 Ki = 720 nM T84631 C7LW3O 11734113 Ki = 100 nM T84631 CNZ04Q 11740591 Ki = 1400 nM T84631 CR53AD 11742672 Ki = 3 nM T84631 C8QZK0 11743193 Ki = 80 nM T84631 CO12HL 11743369 Ki = 495 nM T84631 C5VN3J 11744466 Ki = 2.7 nM T84631 CM95SZ 11744578 IC50 = 1 nM T84631 C7DHE6 11752478 Ki = 6515 nM T84631 C27LUA 11752612 IC50 = 160 nM T84631 CCBH57 11752638 Ki = 306 nM T84631 C5C3BR 11752747 Ki = 24 nM T84631 CX18BY 11752965 Ki = 4.2 nM T84631 CQ81KJ 11753784 IC50 = 122 nM T84631 CP3FI1 11753847 Ki > 15000 nM T84631 C1LPF4 11754261 IC50 = 14 nM T84631 CV62MN 11754356 IC50 = 58 nM T84631 CZ2W6F 11754502 Ki = 3300 nM T84631 C8GJO7 11754872 IC50 = 9.3 nM T84631 CNPW05 11755188 Ki = 0.7 nM T84631 CUMO51 11756555 IC50 = 58 nM T84631 CTOM97 11756558 Ki = 169 nM T84631 C9XAJ5 11756561 Ki = 0.12 nM T84631 CS0JR2 11756961 Ki = 0.83 nM T84631 CMR6A0 11758260 Ki > 8000 nM T84631 C7P4CG 11758475 Ki = 5900 nM T84631 CMD7Z1 11760447 Ki = 5000 nM T84631 CG82LK 11761121 Ki = 1400 nM T84631 CZ7QI3 11761613 Ki = 125 nM T84631 C82ULR 11761706 Ki = 700 nM T84631 CDLZ28 11761967 Ki = 44 nM T84631 CJVR18 11762113 Ki = 1300 nM T84631 CHQ58K 11762202 Ki = 131 nM T84631 C0C9KI 11762303 Ki > 1200 nM T84631 CL53HV 11762323 Ki = 4 nM T84631 CZ91LI 11762766 Ki > 75000 nM T84631 COM9B5 11763170 IC50 > 30000 nM T84631 CWR03Q 11766372 IC50 = 210 nM T84631 CR2E9T 11782463 Ki = 43 nM T84631 C9LC5W 11784323 Ki = 5000 nM T84631 CRH1M7 11784791 Ki = 0.7 nM T84631 C7M3TO 11785263 Ki = 3 nM T84631 CL7QS3 11785424 Ki = 4035 nM T84631 C85MUK 11785772 Ki = 1378 nM T84631 C1EQX3 11785872 Ki = 167 nM T84631 CN3IG5 11785929 Ki = 10 nM T84631 CK4CH2 11786303 Ki = 10 nM T84631 CU9RW5 11792439 Ki = 2700 nM T84631 C8LD7W 11793807 Ki > 5000 nM T84631 CAGC25 11795137 Ki = 160 nM T84631 CZ62LI 11796080 Ki = 960 nM T84631 CW6DG1 11796805 Ki = 1600 nM T84631 CF1S2R 11796942 Ki > 5000 nM T84631 CIS51A 11797515 Ki = 94000 nM T84631 CZM62X 11797951 Ki = 110 nM T84631 CNO67W 11798089 Ki = 5200 nM T84631 CH2Z1N 11798267 Ki = 89 nM T84631 CK8MI3 11798429 Ki = 420000 nM T84631 CK31IT 11800766 Ki = 19 nM T84631 CL6Z3G 11801417 Ki = 16000 nM T84631 C68VNG 11801427 Ki = 210 nM T84631 CL01GT 11801580 Ki = 7.2 nM T84631 CVZ82O 11801725 Ki = 200 nM T84631 CFP36D 11802531 Ki = 13 nM T84631 CY46UZ 11802721 Ki = 5.3 nM T84631 C09WKB 11813114 Ki = 2400 nM T84631 C9VW2P 11813305 Ki = 8 nM T84631 C6W0VT 11813820 Ki = 66 nM T84631 C47BFQ 11813993 Ki = 76 nM T84631 C1Y5NB 11814014 Ki = 144 nM T84631 CUN1S4 11814234 Ki = 134 nM T84631 C8INH6 11814686 IC50 = 3140 nM T84631 C7JO4I 11823405 Ki = 8800 nM T84631 C98ZOR 11824040 Ki = 19000 nM T84631 CYX74A 11824584 Ki = 5200 nM T84631 CCT84E 11825785 Ki > 5000 nM T84631 CEYP62 11826299 Ki = 51 nM T84631 C79MQD 11826825 IC50 > 30000 nM T84631 C3EFY7 11826875 Ki = 61 nM T84631 C93TLO 11827247 Ki = 26 nM T84631 C9R2OA 11828043 Ki = 103 nM T84631 C61GPA 11828451 IC50 = 2100 nM T84631 CW6E7I 11828640 IC50 = 210 nM T84631 C4DTE8 11849112 Ki = 1 nM T84631 CY8T0B 11950081 Ki = 0.6 nM T84631 CQ74TC 11950083 Ki = 1 nM T84631 CN27JS 11950249 Ki = 1 nM T84631 CGY83S 11950253 Ki = 10 nM T84631 C6XW2E 11950427 Ki = 8 nM T84631 CRD0A6 11950428 Ki = 15 nM T84631 CTJ3A8 11950431 Ki = 1.3 nM T84631 CXH68R 11950432 Ki = 0.6 nM T84631 C9PV4Y 11950602 Ki = 2 nM T84631 CYX53O 11950605 Ki = 2 nM T84631 C86SCE 11950606 Ki = 1 nM T84631 CTZ4B6 11956166 Ki = 100 nM T84631 C6XRH4 11966394 Ki = 40 nM T84631 C5SEB3 11967063 IC50 = 1800 nM T84631 CTB2C9 11967128 IC50 = 380 nM T84631 CS92GP 11979006 Ki = 10 nM T84631 C12IZN 11979007 Ki = 3 nM T84631 C34NUJ 11979125 Ki = 10 nM T84631 CE04WI 11979126 Ki = 22 nM T84631 C69HNO 11984565 Ki = 7200 nM T84631 CPR4I1 12047383 Ki = 87000 nM T84631 C5U0FJ 12047384 Ki = 87000 nM T84631 C5FU3H 12047385 Ki = 45000 nM T84631 CX98PQ 12082573 IC50 = 500 nM T84631 CT7IR8 12110710 IC50 > 100000 nM T84631 CLJ15H 12222233 Ki = 6.8 nM T84631 C1TK9C 12972260 IC50 = 106 nM T84631 C1IT4G 12972261 IC50 = 62.6 nM T84631 C84CJL 12986348 IC50 = 260 nM T84631 CYN6H0 12988920 Ki = 0.72 nM T84631 CO5Z4Y 12989060 Ki = 0.29 nM T84631 CQ8OU1 13755335 Ki = 1800 nM T84631 C45LTS 13755337 Ki = 1300 nM T84631 C60TVD 15392306 IC50 = 6 nM T84631 C7ZV8R 15392323 IC50 = 6 nM T84631 C3HYW7 15431805 IC50 > 2500 nM T84631 CZBD56 15435386 Ki = 94 nM T84631 C9KJ5Y 15461560 Ki = 0.33 nM T84631 CM2RN1 15461564 Ki = 0.015 nM T84631 C5CQ6R 15463576 Ki = 3.4 nM T84631 CCN18Q 15463577 Ki = 13 nM T84631 CZ4L6O 15463578 Ki = 400 nM T84631 CF9H3Z 15463579 Ki = 460 nM T84631 CY2S1U 15463580 Ki = 12 nM T84631 CQTF26 15463581 Ki = 26 nM T84631 CX5S1Z 15511974 Ki = 2.1 nM T84631 CW2QY0 15515689 IC50 = 4100 nM T84631 CG9Q0P 15515690 IC50 = 2500 nM T84631 C54SUM 15515691 IC50 = 16000 nM T84631 C60JFG 15521694 Ki = 1450 nM T84631 CP63GF 15534822 IC50 > 2500 nM T84631 CPJT95 15545832 Ki = 180 nM T84631 CKQ8M6 15546794 Ki = 6 nM T84631 CI6G0C 15736732 IC50 = 2500 nM T84631 CL9T7Y 15870100 Ki = 2100 nM T84631 CB3T9P 15870101 Ki = 400 nM T84631 C9EH2Y 15887336 IC50 = 230 nM T84631 C6VZ1N 15942655 Ki = 125000 nM T84631 CA86KZ 15947513 Ki = 8100 nM T84631 CU0O5N 15947601 Ki = 3900 nM T84631 CQ3RF8 15947602 Ki = 1800 nM T84631 CS8HY6 15947811 Ki = 4100 nM T84631 CCMQ45 15947923 Ki = 7600 nM T84631 CUGI75 15947926 Ki = 6200 nM T84631 CSV70B 15948627 Ki = 7200 nM T84631 C7VH6K 15950345 Ki = 0.16 nM T84631 C4EW6F 15965462 IC50 = 4 nM T84631 CMYR94 15976119 Ki = 5077 nM T84631 CLP2D3 16004672 Ki = 0.033 nM T84631 CX7KR1 16040261 Ki = 534 nM T84631 CA8Y1K 16046152 Ki = 0.27 nM T84631 CNBJ60 16046153 Ki = 0.37 nM T84631 CC7Y0D 16066741 IC50 > 200000 nM T84631 C3EUJ6 16086336 IC50 = 33500 nM T84631 CDSM46 16098887 IC50 = 14000 nM T84631 CFK98M 16098895 IC50 = 1700 nM T84631 C6BQ0G 16098896 IC50 > 200000 nM T84631 C1ZXL4 16098897 IC50 = 8500 nM T84631 CP6Y7Q 16098898 IC50 = 22000 nM T84631 C3J6LO 16098899 IC50 > 200000 nM T84631 CQ4YJ8 16098900 IC50 = 15000 nM T84631 CDL2X5 16098901 IC50 = 13000 nM T84631 C53ZXO 16098902 IC50 > 20000 nM T84631 CUJ5A9 16098903 IC50 > 20000 nM T84631 CZ3WM4 16098905 IC50 > 200000 nM T84631 CVN8Y1 16098906 IC50 = 2700 nM T84631 CTY5W9 16098907 IC50 = 14900 nM T84631 C53YRO 16098910 IC50 = 1600 nM T84631 C91CQM 16098911 IC50 = 250 nM T84631 C0W5NR 16098912 IC50 = 1600 nM T84631 CS21OE 16098913 IC50 = 2100 nM T84631 CO08FM 16112849 Ki = 1 nM T84631 CTW28E 16124699 Ki = 109 nM T84631 CSG06K 16124700 Ki = 165 nM T84631 CO69AB 16124701 Ki = 163 nM T84631 C91VBY 16124702 Ki = 2898 nM T84631 C41KQS 16124703 Ki > 15800 nM T84631 CP82YG 16124704 Ki = 285 nM T84631 CY3F2H 16124761 Ki = 4160 nM T84631 CM3Q6R 16124762 Ki = 112 nM T84631 CPD7L0 16124763 Ki = 170 nM T84631 CA53KN 16124764 Ki = 5 nM T84631 CX2BE1 16125613 Ki = 314 nM T84631 CM3P5C 16125614 Ki = 3670 nM T84631 C6E7RC 16125615 Ki = 3225 nM T84631 C8SNI9 16125616 Ki = 782 nM T84631 CBH64D 16125617 Ki = 1200 nM T84631 CIQ7S3 16125671 Ki = 2 nM T84631 CU5YJ0 16125672 Ki = 24 nM T84631 CJ7E2X 16204383 IC50 = 1.2 nM T84631 CL7Z6K 16215018 IC50 = 3.9 nM T84631 CN6CJ2 16220264 IC50 = 6470 nM T84631 CZ7FS4 16284785 IC50 > 200000 nM T84631 C56TPZ 16285203 IC50 > 200000 nM T84631 C1KZB9 16289649 IC50 > 200000 nM T84631 CQ0EK7 16660960 IC50 = 2.1 nM T84631 CX4UT5 16660962 IC50 = 37 nM T84631 CL2W9Q 16660964 IC50 = 5.7 nM T84631 CG2Q8U 16660966 IC50 = 3.3 nM T84631 CX36RF 16660968 IC50 = 6.5 nM T84631 C27COL 16661109 IC50 = 0.43 nM T84631 CPK67M 16664096 Ki = 0.35 nM T84631 CU28CE 16718713 IC50 = 30000 nM T84631 CC20PS 16718760 IC50 = 250000 nM T84631 CCKO80 16718762 IC50 = 27000 nM T84631 CTZ74D 16718807 IC50 > 250000 nM T84631 C37MRI 16718808 IC50 > 10000 nM T84631 CUL0B3 16720561 Ki = 15.9 nM T84631 CJL72U 16731819 Ki = 0.43 nM T84631 C05JSB 16731821 Ki = 0.16 nM T84631 C6SN2Q 16731823 Ki = 0.36 nM T84631 CG49VM 16731824 Ki = 1 nM T84631 C8ZFY6 16731827 Ki = 0.4 nM T84631 CN60KL 16731975 Ki = 1.4 nM T84631 CB01OR 16731976 Ki = 0.22 nM T84631 C7MR9E 16731977 Ki = 1.4 nM T84631 CF4V3D 16731978 Ki = 0.52 nM T84631 CS2QJ8 16731979 Ki = 2.2 nM T84631 CYB1E0 16731980 Ki = 0.24 nM T84631 CD64LP 16732121 Ki = 0.18 nM T84631 CWU9D7 16732123 Ki = 0.4 nM T84631 CH2U5Z 16732125 Ki = 0.71 nM T84631 CSB43R 16732126 Ki = 0.26 nM T84631 CK74UL 16732127 Ki = 0.024 nM T84631 C4A1RO 16732128 Ki = 0.019 nM T84631 C9BD4C 16732263 Ki = 0.045 nM T84631 CZ3M6S 16732265 Ki = 0.026 nM T84631 C3DW7C 16732266 Ki = 0.02 nM T84631 CBO97E 16732268 Ki = 0.05 nM T84631 C7QBR0 16732402 Ki = 0.036 nM T84631 C6RPF4 16732404 Ki = 0.022 nM T84631 CN3D9T 16732406 Ki = 0.012 nM T84631 C1HFQ6 16732407 Ki = 2.2 nM T84631 CGC0Q2 16732555 Ki = 0.12 nM T84631 C7SUK0 16732557 Ki = 0.26 nM T84631 CT4K0V 16732559 Ki = 0.12 nM T84631 CKAZ40 16732560 Ki = 0.031 nM T84631 CKN73Z 16732562 Ki = 0.012 nM T84631 CLF90N 16732707 Ki = 0.026 nM T84631 CR3K2E 16732708 Ki = 0.024 nM T84631 C2EOR6 16732711 Ki = 0.004 nM T84631 CPK8Z7 16732713 Ki <= 0.01 nM T84631 CUHT92 16732866 Ki <= 0.01 nM T84631 C07OPV 16732868 Ki <= 0.01 nM T84631 C3Y2HE 16732871 Ki = 0.004 nM T84631 C47UEZ 16732873 Ki <= 0.01 nM T84631 CL4EW1 16733006 Ki = 0.004 nM T84631 CNYA03 16733007 Ki <= 0.01 nM T84631 C7XU2R 16733008 Ki <= 0.01 nM T84631 CRBI26 16733010 Ki = 0.022 nM T84631 CUEL18 16733012 Ki <= 0.01 nM T84631 C6OK0W 16733013 Ki = 0.006 nM T84631 C0G7KW 16733150 Ki = 0.02 nM T84631 C54HKA 16734339 Ki = 1.3 nM T84631 CJ3MX8 16734340 Ki = 0.8 nM T84631 C08JWR 16734545 Ki = 0.8 nM T84631 CF8S7J 16734546 Ki = 0.8 nM T84631 C7CSO3 16741235 IC50 = 0.16 nM T84631 COZ62I 16748993 IC50 = 0.38 nM T84631 CYDU97 16749087 IC50 = 18 nM T84631 CJG13M 17756142 IC50 = 4.6 nM T84631 C2K9GC 17788740 Ki = 170 nM T84631 CVB82P 17809181 IC50 = 880 nM T84631 CB6R1Z 17809213 IC50 = 6.63 nM T84631 C9PVW1 17822583 Ki = 2100 nM T84631 CF4K6R 17843517 IC50 = 123 nM T84631 C2IEC4 17851729 IC50 = 120 nM T84631 CA91IM 17851931 IC50 = 110 nM T84631 C16XHL 17852016 IC50 = 63 nM T84631 C72GHY 17852042 IC50 = 79 nM T84631 C5RSD3 18318130 Ki = 0.17 nM T84631 CL13IP 18318139 Ki = 0.56 nM T84631 C3P0VK 18318146 Ki = 6.8 nM T84631 COJ9F3 18318187 Ki = 0.55 nM T84631 C1S3MX 18318188 Ki = 0.88 nM T84631 CGNJ35 18318198 Ki = 7.5 nM T84631 CE7RZ4 18318201 Ki = 4.1 nM T84631 CBS40I 18318220 Ki = 0.27 nM T84631 COC54Y 18327622 Ki = 250000 nM T84631 CI5J3Y 18376546 Ki = 15 nM T84631 CMU9A3 18376555 Ki = 470 nM T84631 CFQE53 18376558 Ki = 26 nM T84631 CLUC36 18376562 Ki = 6.2 nM T84631 C76KJP 18376565 Ki = 54 nM T84631 CC94AD 18376598 Ki = 3.7 nM T84631 CJ7K3O 18376605 Ki = 10 nM T84631 C1UT4K 18376606 Ki = 1.6 nM T84631 CU98XE 18376618 Ki = 1.9 nM T84631 CCH92J 18376625 Ki = 34 nM T84631 C25PXL 18376627 Ki = 11 nM T84631 CL4UC9 18376641 Ki = 0.005 nM T84631 C4TCP6 18376642 Ki = 0.6 nM T84631 C0D1EH 18376656 Ki = 12 nM T84631 CN8CI1 18376659 Ki = 6 nM T84631 CTA57Y 18376663 Ki = 10 nM T84631 CHO4P2 18376665 Ki = 14 nM T84631 CPGX36 18376669 Ki = 0.8 nM T84631 CG0N9Q 18376671 Ki = 25 nM T84631 CU7V4F 18376679 Ki = 12 nM T84631 CIJG48 18376696 Ki = 2 nM T84631 C27NVA 18376714 Ki = 3.5 nM T84631 CR1C3F 18376717 Ki = 19 nM T84631 CSJZ89 18376719 Ki = 0.52 nM T84631 CUE92D 18376730 Ki = 73 nM T84631 CPT6W5 18376743 Ki = 58 nM T84631 CZ7HJ6 18376748 Ki = 24 nM T84631 CXW37R 18376768 Ki = 130 nM T84631 CBO4I0 18376780 Ki = 4.8 nM T84631 C7JF8K 18376782 Ki = 5.9 nM T84631 C86WAR 18376800 Ki = 2.3 nM T84631 CUZ8V3 18376816 Ki = 5 nM T84631 CAQ7X0 18376821 Ki = 590 nM T84631 C7Y8FD 18376826 Ki = 9.5 nM T84631 CRA3Y5 18376827 Ki = 7.2 nM T84631 C4I9XE 18376832 Ki = 0.45 nM T84631 C0S9XW 18376837 Ki = 24 nM T84631 CG98XS 18376838 Ki = 7.2 nM T84631 C4JE8S 18376839 Ki = 0.8 nM T84631 CN1ZX0 18376843 Ki = 2.1 nM T84631 C8YF1V 18376848 Ki = 16 nM T84631 CS79AF 18376858 Ki = 1.8 nM T84631 C9FDM4 18376865 Ki = 100 nM T84631 CUIC43 18376871 Ki = 2.1 nM T84631 CJL9E5 18376880 Ki = 1.4 nM T84631 C8KTW9 18376881 Ki = 22 nM T84631 C63EFY 18376882 Ki = 1.4 nM T84631 CE2BH4 18376888 Ki = 5.6 nM T84631 CE43LC 18376891 Ki = 21 nM T84631 C9V3HX 18376897 Ki = 18 nM T84631 C1ZKY8 18376901 Ki = 0.95 nM T84631 CH8R6S 18376905 Ki = 0.38 nM T84631 CUJP51 18376916 Ki = 260 nM T84631 CLE27U 18376919 Ki = 7.5 nM T84631 C3EN2U 18376921 Ki = 4.6 nM T84631 CM6NT1 18376930 Ki = 2.7 nM T84631 CG8Y0C 18376939 Ki = 5.2 nM T84631 C1SZ9Q 18376940 Ki = 210 nM T84631 CWG72T 18376950 Ki = 26 nM T84631 CV3ZE2 18376959 Ki = 14 nM T84631 CWI0E3 18376970 Ki = 2.2 nM T84631 C1OM7T 18376973 Ki = 0.3 nM T84631 C1T3VP 18376976 Ki = 1.6 nM T84631 C7SO8U 18376989 Ki = 150 nM T84631 CF0GR6 18376995 Ki = 7 nM T84631 CN2JE5 18376999 Ki = 30 nM T84631 CC9ZE2 18377002 Ki = 20 nM T84631 C53XHD 18377003 Ki = 1.7 nM T84631 C94LUS 18377010 Ki = 18 nM T84631 C79ZIE 18377020 Ki = 16 nM T84631 C3FYR1 18377031 Ki = 22 nM T84631 CI5U7D 18377033 Ki = 7 nM T84631 CEH2K1 18377041 Ki = 160 nM T84631 CX8RE3 18377048 Ki = 0.82 nM T84631 CN87FW 18474271 Ki = 2700 nM T84631 C3V9EC 18549309 Ki = 0.009 nM T84631 C63ILO 18549509 Ki = 0.09 nM T84631 C09CBT 18675029 IC50 = 26000 nM T84631 C0OPG9 18675052 IC50 = 5600 nM T84631 CRE8M4 18675059 IC50 = 27000 nM T84631 C9NB0Z 18675062 IC50 = 12 nM T84631 C09KIY 18675079 IC50 = 48 nM T84631 C29WYS 18675086 IC50 = 3 nM T84631 CR6I5L 18675103 IC50 = 16000 nM T84631 CLZ97R 18675188 IC50 = 7900 nM T84631 CFU8B9 18675209 IC50 = 66000 nM T84631 C17EDK 18675223 IC50 = 4900 nM T84631 C9NFX4 18675228 IC50 = 34000 nM T84631 CK6U1I 18675238 IC50 = 1600 nM T84631 CN0LW2 18675252 IC50 = 840 nM T84631 CM5VX3 18675291 IC50 = 23000 nM T84631 CD9UE4 18675298 IC50 = 68 nM T84631 CB01HJ 18675385 IC50 = 17000 nM T84631 CV5EG7 18727564 IC50 = 6 nM T84631 CWS58B 18727568 IC50 = 19 nM T84631 C2P5HW 18727569 IC50 = 1.2 nM T84631 C8ZP2O 18727570 IC50 = 1.5 nM T84631 C91FXK 18727571 IC50 = 16 nM T84631 COB7U9 18727572 IC50 = 12 nM T84631 CU3G4Q 18727574 IC50 = 4.8 nM T84631 CS8Y6P 18727576 IC50 = 10 nM T84631 C43RUO 18727577 IC50 = 5.4 nM T84631 CF4W5D 18727604 IC50 = 4 nM T84631 CB0IQ4 18727607 IC50 = 10 nM T84631 C6QZL7 18727622 IC50 = 1.2 nM T84631 CK2N1A 18727717 IC50 = 67 nM T84631 CNIB76 18727776 IC50 = 7.7 nM T84631 C9HXV5 18727777 IC50 = 370 nM T84631 C8AXM2 18727805 IC50 = 0.7 nM T84631 C31ZAL 18727831 IC50 = 15 nM T84631 CJY67O 18727833 IC50 = 2 nM T84631 C02HEA 18727834 IC50 = 15 nM T84631 CJSL38 18727836 Ki = 0.3 nM T84631 C8AMY9 18727838 IC50 = 7 nM T84631 CDO92V 18727840 IC50 = 2 nM T84631 CY8AC3 18727841 IC50 = 140 nM T84631 CB68ZV 18727844 IC50 = 0.6 nM T84631 C2M7ZO 18727846 IC50 = 0.6 nM T84631 C1IL8E 18727847 IC50 = 1.3 nM T84631 CD02TK 18727852 IC50 = 17 nM T84631 C1JMX5 18727855 IC50 = 16 nM T84631 CP7HL9 18727867 IC50 = 0.5 nM T84631 CQI72L 18727923 IC50 = 6060 nM T84631 CJM5I3 18727924 IC50 = 1810 nM T84631 C8GR2Q 18727965 IC50 = 78 nM T84631 CD51CF 18727967 IC50 = 714 nM T84631 CC0U9I 18727969 IC50 = 23 nM T84631 CL4B1V 18728102 IC50 = 226 nM T84631 C24ZCT 18728106 IC50 = 316 nM T84631 CKX4D1 18728109 IC50 = 7 nM T84631 CZ0XE6 18728123 IC50 = 0.7 nM T84631 C4DPW0 18728129 IC50 = 38 nM T84631 C0V4HL 18728139 IC50 = 26 nM T84631 C9OGD1 18728140 IC50 = 23 nM T84631 CJ4WA9 18728144 IC50 = 2 nM T84631 CE0ZU2 18728158 IC50 = 18 nM T84631 CNUR53 18800583 Ki = 400 nM T84631 C5MR0U 20585828 IC50 = 20 nM T84631 C7P4UB 20585829 IC50 = 10 nM T84631 CO2JG4 20595081 IC50 = 45 nM T84631 CGJN85 20595087 IC50 = 46 nM T84631 C9MN8Y 20595088 IC50 = 36 nM T84631 CM7BH1 20595091 IC50 = 24 nM T84631 CCH5N1 20595225 IC50 = 545 nM T84631 C70TFO 20595245 IC50 = 110 nM T84631 CX68HR 20595247 IC50 = 31 nM T84631 CX9YN6 20595251 Ki = 3.9 nM T84631 CKYA19 20595257 IC50 = 14 nM T84631 C2ID8R 20595260 Ki = 1.7 nM T84631 CH3D0Y 20595264 IC50 = 134 nM T84631 C8DXS5 20595268 IC50 = 28 nM T84631 C1HAM4 20595273 IC50 = 15 nM T84631 CM78XE 20595304 IC50 = 777 nM T84631 C10EGW 20595308 IC50 = 50 nM T84631 C0A9HN 20595310 IC50 = 50 nM T84631 CUS20T 20595326 IC50 = 16 nM T84631 CMT46A 20595328 Ki = 3.9 nM T84631 C9U2QS 20595336 IC50 = 18 nM T84631 C43UDK 20608737 IC50 > 30000 nM T84631 CW3I9O 20608738 IC50 > 30000 nM T84631 C4UZO0 20608741 IC50 > 30000 nM T84631 C9Z2VH 20608755 IC50 > 30000 nM T84631 C3OF2S 20608756 IC50 > 30000 nM T84631 CMX4Q6 20608776 IC50 > 30000 nM T84631 CXH09O 20631502 IC50 = 0.01 nM T84631 C2YDK5 20641721 IC50 = 4 nM T84631 CT7I1B 20641743 IC50 = 13 nM T84631 C7LHE8 20641745 Ki = 2.7 nM T84631 CTY8G2 20707887 Ki = 1.2 nM T84631 C0BKY3 20707927 IC50 = 2700 nM T84631 CB0X8I 20707929 IC50 = 650 nM T84631 C2BM9Q 20708041 IC50 = 1200 nM T84631 C7LX8J 20708044 IC50 = 1100 nM T84631 C0FRB4 20708055 IC50 = 60 nM T84631 CLM02X 20708056 IC50 = 380 nM T84631 C74LUP 20708058 IC50 = 50 nM T84631 CI6ZK4 20708066 IC50 = 180 nM T84631 CC3I4M 20708069 IC50 = 110 nM T84631 CJL5M6 20708073 IC50 = 360 nM T84631 CS57OI 20708074 IC50 = 890 nM T84631 CRK8N0 20708078 IC50 = 120 nM T84631 CC50OV 20708079 IC50 = 90 nM T84631 CK2V5A 20708094 IC50 = 700 nM T84631 CC7OB1 20708098 IC50 = 790 nM T84631 C6DN0A 20708099 IC50 = 160 nM T84631 C7JMO0 20708106 IC50 = 110 nM T84631 CR18VG 20708107 IC50 = 60 nM T84631 C02MHB 20708108 IC50 = 240 nM T84631 CL13GC 20708219 IC50 = 540 nM T84631 CWH2Z7 20747446 IC50 = 31 nM T84631 CXA98P 20747457 IC50 = 21 nM T84631 CV6KT1 20747459 IC50 = 61 nM T84631 CLZ5O4 20747496 IC50 = 93 nM T84631 CD2JP6 20747497 IC50 = 10 nM T84631 C2F4CK 20747503 IC50 = 256 nM T84631 C4CL5Y 20751605 IC50 = 64 nM T84631 CZ6KH9 20760195 Ki = 0.74 nM T84631 CH9J6I 20760215 Ki = 0.6 nM T84631 C7P9YE 20760216 Ki = 0.6 nM T84631 CR05LA 20760219 Ki = 3.6 nM T84631 C6ZUX8 20760222 Ki = 1.6 nM T84631 CMT78G 20760223 Ki = 3.8 nM T84631 CFY3L6 20801005 Ki = 474 nM T84631 C6IC3V 20801009 Ki = 73 nM T84631 C1DBA6 20801019 Ki = 57 nM T84631 CS29FI 20801029 Ki = 2230 nM T84631 CW0KR1 20801030 Ki = 400 nM T84631 CDIB13 20801031 Ki = 3 nM T84631 C65FLV 20801045 Ki = 654 nM T84631 C02ZCV 20801048 Ki = 9010 nM T84631 CTF5N7 20801076 Ki = 2500 nM T84631 CXQ3N0 20801082 Ki = 2100 nM T84631 CXR5A9 20801095 Ki = 810 nM T84631 C9RG0H 20801097 Ki = 4 nM T84631 CMI8H7 20801110 Ki = 220 nM T84631 CT7NZ2 20801115 Ki = 131 nM T84631 CUKR42 20801117 Ki = 64 nM T84631 C8KYF3 20801119 Ki = 106 nM T84631 CFJ13A 20801120 Ki = 71 nM T84631 CIM9C3 20801121 Ki = 27 nM T84631 CZW87C 20801125 Ki = 142 nM T84631 CB84ZQ 20801132 Ki = 20 nM T84631 CG51FK 20801137 Ki = 161 nM T84631 CC1Y0R 20801139 Ki = 40 nM T84631 CCO9S7 20801141 Ki = 125 nM T84631 C4V8ZR 20801142 Ki = 64 nM T84631 CCY5O7 20801143 Ki = 95 nM T84631 CY39JK 20801144 Ki = 95 nM T84631 COAC01 20801159 Ki = 15 nM T84631 CS3HB4 20801160 Ki = 40 nM T84631 CVSI76 20801207 Ki = 763 nM T84631 CCZJ48 20801208 Ki = 1075 nM T84631 CVNJ41 20801210 Ki > 10000 nM T84631 C3QBC1 20801212 Ki = 2480 nM T84631 CGD57F 20802932 IC50 > 30000 nM T84631 CO2FM4 20802944 IC50 > 30000 nM T84631 C1P0WC 20802959 IC50 > 30000 nM T84631 CBL6N1 20802966 IC50 > 30000 nM T84631 C27ZJT 20802995 IC50 > 100000 nM T84631 C3B4MA 20824147 IC50 = 8 nM T84631 C5ACM1 20843251 IC50 = 55000 nM T84631 C3RTJ2 20872059 Ki = 0.36 nM T84631 CG0RD2 21071205 Ki = 0.13 nM T84631 C95DUQ 21071251 Ki = 2.4 nM T84631 CR6C2I 21218691 Ki = 270 nM T84631 CS5L2M 21218709 Ki = 117 nM T84631 CEQ6B2 21218732 Ki = 20 nM T84631 C79ZNM 21218751 Ki = 143 nM T84631 CLT36V 21250176 IC50 = 500 nM T84631 CRYB96 21250293 IC50 = 400 nM T84631 C0ECB5 21250297 IC50 > 100000 nM T84631 CLV49W 21250386 IC50 = 9200 nM T84631 CN2YE9 21250416 IC50 = 46000 nM T84631 CRD4V1 21250427 IC50 = 1400 nM T84631 C3T5SA 21250434 IC50 = 31000 nM T84631 C9H7ZI 21250518 IC50 = 10600 nM T84631 CCY2M5 21366447 IC50 = 76 nM T84631 C27VLD 21366448 IC50 = 24 nM T84631 C1JQY7 21366475 IC50 = 15 nM T84631 C82SUW 21366478 IC50 = 8 nM T84631 CSG82H 21366479 IC50 = 7 nM T84631 CP0CR1 21366482 Ki = 0.7 nM T84631 CNTI15 21366511 IC50 = 143 nM T84631 C5S8ZW 21366513 IC50 = 24 nM T84631 CNC0E1 21366553 IC50 = 81 nM T84631 C9GAE1 21366554 IC50 = 39 nM T84631 C1CVM9 21366560 Ki = 5.2 nM T84631 C2LJ6Y 21366561 IC50 = 11 nM T84631 CQM6Y9 21366562 Ki = 4.1 nM T84631 C59WZX 21366563 IC50 = 10 nM T84631 C0H8KE 21366566 IC50 = 27 nM T84631 C67QCO 21366574 IC50 > 11000 nM T84631 CS2L1Y 21366575 IC50 = 483 nM T84631 CX1WM9 21366579 IC50 = 1650 nM T84631 C5XU1Y 21366636 Ki = 1.4 nM T84631 C0MXT9 21366640 Ki = 1.9 nM T84631 C0H3EX 21366644 Ki = 1 nM T84631 CYVC46 21366645 Ki = 1.2 nM T84631 C8OL1C 21366646 Ki = 1.8 nM T84631 C0U5PX 21366647 IC50 = 3 nM T84631 CP91WB 21366649 IC50 = 7 nM T84631 C8BLF5 21366650 IC50 = 4 nM T84631 CR8QB1 21366651 IC50 = 7 nM T84631 CKE17U 21366652 IC50 = 2 nM T84631 CV16OC 21366654 Ki = 0.9 nM T84631 CTND64 21578548 Ki = 27558 nM T84631 C7Z8YR 21845821 Ki = 6.31 nM T84631 C3HY2D 21845878 Ki = 1258.93 nM T84631 CI0SJ2 21967345 Ki = 5 nM T84631 CK5I4A 21968289 Ki = 170 nM T84631 CXV3I1 22017200 Ki = 320 nM T84631 C0MI4Y 22038750 Ki > 7500 nM T84631 CAS92P 22038873 Ki = 12200 nM T84631 CJ81IS 22039255 Ki = 730 nM T84631 C7VD8G 22039455 Ki = 790 nM T84631 CD2I7L 22039678 Ki = 1400 nM T84631 CK6E8W 22052309 Ki = 48 nM T84631 C4QDG0 22052319 Ki = 50 nM T84631 C0OE1R 22052320 Ki = 29 nM T84631 CX0FL5 22052323 Ki = 13 nM T84631 CHQ1R5 22052325 Ki = 61 nM T84631 CXPM37 22052326 Ki = 316 nM T84631 C6T8ZN 22052336 Ki = 86 nM T84631 C1YH0L 22052339 Ki = 54 nM T84631 COW3F2 22052347 Ki = 140 nM T84631 CSJW40 22052358 Ki = 25 nM T84631 CTNL12 22052361 Ki = 12.59 nM T84631 C4L1XD 22052368 Ki = 106 nM T84631 CC52AE 22052371 Ki = 39.81 nM T84631 C29PIU 22052373 Ki = 37 nM T84631 CA5T8Z 22052377 Ki = 1763 nM T84631 C8C7PW 22052392 Ki = 233 nM T84631 C9L5AD 22052419 Ki = 263 nM T84631 CC6Z8A 22052426 Ki = 19.95 nM T84631 CJ9W2M 22052436 Ki = 76 nM T84631 C8D7FS 22052452 Ki = 28 nM T84631 CTO8P4 22052453 Ki = 398.11 nM T84631 CV7O1I 22052465 Ki = 1554 nM T84631 C17HKB 22052478 Ki = 20 nM T84631 C1O9GL 22052482 Ki = 39.81 nM T84631 CGNH32 22052484 Ki = 75 nM T84631 CQ5VT0 22052485 Ki = 44 nM T84631 CN6YR8 22052493 Ki = 314 nM T84631 C7FYD1 22086911 Ki = 2.8 nM T84631 C5VIU4 22086968 Ki = 1.7 nM T84631 CYEU57 22086972 Ki = 0.53 nM T84631 C5K6SW 22086973 Ki = 0.55 nM T84631 CQC51W 22086974 Ki = 0.35 nM T84631 C9LI4W 22086975 Ki = 0.25 nM T84631 CB6IP5 22086976 Ki = 0.04 nM T84631 C3O8DP 22086978 Ki = 1.5 nM T84631 CDVH80 22086981 Ki = 0.35 nM T84631 CLH7A0 22086982 Ki = 0.15 nM T84631 C17KGP 22086987 Ki = 1.3 nM T84631 CG4ZH7 22086988 Ki = 0.31 nM T84631 CVM24X 22086990 Ki = 2.8 nM T84631 CJ5D8V 22086991 Ki = 1.4 nM T84631 C5V2HO 22086992 Ki = 1.9 nM T84631 CZ5O0I 22087006 Ki = 0.85 nM T84631 COK2S6 22087007 Ki = 0.81 nM T84631 CJ8D4K 22087014 Ki = 2.1 nM T84631 CKT23G 22125586 Ki = 30 nM T84631 CA3I4Y 22280766 Ki = 4.6 nM T84631 C40XEN 22313515 Ki = 450 nM T84631 CH9E3I 22313526 Ki = 560 nM T84631 C04OMK 22318549 Ki = 1 nM T84631 CS01PB 22318550 Ki = 23 nM T84631 CSQ96D 22336121 IC50 = 19.41 nM T84631 C7R9CD 22336127 IC50 = 0.64 nM T84631 C1R9CX 22336133 IC50 = 5.22 nM T84631 CHOQ30 22336142 IC50 = 8.15 nM T84631 CVG29W 22336143 IC50 = 0.12 nM T84631 CB7N4X 22336146 IC50 = 0.15 nM T84631 C8URK9 22336148 IC50 = 59 nM T84631 C3QEL8 22336150 IC50 = 0.15 nM T84631 C5O7VB 22336151 IC50 = 0.04 nM T84631 C19NAE 22336153 IC50 = 0.35 nM T84631 CHG0A5 22336163 IC50 = 1.65 nM T84631 CTOR48 22336172 IC50 = 0.45 nM T84631 C51FCG 22336174 IC50 = 0.23 nM T84631 CXZ92L 22336180 IC50 = 1.9 nM T84631 C85UYR 22336181 IC50 = 0.05 nM T84631 CU3T0V 22394327 Ki = 2900 nM T84631 CN6P9I 22394409 Ki = 18 nM T84631 CYLS84 22394472 Ki = 2997 nM T84631 CIT61O 22458350 IC50 = 3.6 nM T84631 CCD92W 22458360 IC50 = 3120 nM T84631 CRHI62 22458366 IC50 = 184 nM T84631 CCM12G 22458368 IC50 = 270 nM T84631 CT2IM0 22458374 IC50 = 920 nM T84631 CYOX21 22458381 IC50 = 880 nM T84631 COLY72 22556932 Ki = 2 nM T84631 C2V1NP 22556955 Ki = 2 nM T84631 C4YL7S 22556963 Ki = 0.7 nM T84631 C9VXC8 22556983 Ki = 20 nM T84631 CY4J8E 22596314 IC50 = 12 nM T84631 CLA45C 22596321 IC50 = 48 nM T84631 CF2RK6 22596324 IC50 = 2.5 nM T84631 C2KTB6 22596330 IC50 = 1.9 nM T84631 C9FVL3 22596339 IC50 = 49 nM T84631 C1B0NE 22596349 IC50 = 1.8 nM T84631 CC7LV3 22596380 IC50 = 4.4 nM T84631 CTG8D5 22596389 IC50 = 2.5 nM T84631 CZ4T5U 22596395 IC50 = 7.7 nM T84631 C32GEK 22596430 IC50 = 4.6 nM T84631 CA3FT7 22612508 Ki = 390 nM T84631 CUXK90 22628841 Ki = 60 nM T84631 C4W0GT 22713568 Ki > 10000 nM T84631 CJY09H 22861145 Ki = 130016.96 nM T84631 CN3ZI2 22883539 Ki = 90 nM T84631 CW8EH6 22883547 Ki = 39 nM T84631 CA3N9L 22883564 Ki = 31 nM T84631 C9DB7V 22883573 Ki = 120 nM T84631 CVZ15N 22883583 Ki = 88 nM T84631 C1R0UD 22883585 Ki = 26 nM T84631 C13-JAN 22883594 Ki = 3 nM T84631 C1KG8E 22945874 IC50 = 110 nM T84631 C3VZ7S 23283289 Ki = 19000 nM T84631 CV5NL8 23283331 Ki = 30000 nM T84631 C2K7VO 23396194 Ki = 588 nM T84631 CU01TZ 23396195 Ki = 241 nM T84631 CR6CQ9 23396199 Ki = 50 nM T84631 CY32CO 23396230 Ki = 37 nM T84631 CXD84O 23396232 Ki = 125 nM T84631 C9BUH2 23396254 Ki = 630.96 nM T84631 CEVA63 23396255 Ki = 36 nM T84631 C71ZYM 23396256 Ki = 71 nM T84631 CG3VZ4 23396258 Ki = 41 nM T84631 C3Z2EI 23396259 Ki = 4605 nM T84631 C5B8YE 23396265 Ki > 10000 nM T84631 C16WGD 23396266 Ki > 10000 nM T84631 CW3VI5 23396282 Ki = 1931 nM T84631 C3EH5R 23396283 Ki = 2494 nM T84631 C2P7KJ 23396286 Ki = 1552 nM T84631 C0Z3IW 23396287 Ki = 100 nM T84631 CI76UO 23396288 Ki = 124 nM T84631 CO63QT 23396289 Ki = 3162.28 nM T84631 C9ZAU2 23396290 Ki = 199.53 nM T84631 C0GWO4 23396291 Ki = 307 nM T84631 C7ICP0 23396292 Ki = 199.53 nM T84631 CCA13I 23396298 Ki = 39 nM T84631 C9VZK5 23396327 Ki = 4531 nM T84631 CN1H6K 23396328 Ki > 10000 nM T84631 CR2Y5O 23442128 Ki = 650 nM T84631 CQ70HF 23586156 IC50 = 995 nM T84631 C1JXS8 23634638 Ki = 1.7 nM T84631 C0W2EP 23634640 Ki = 0.33 nM T84631 CD7C1W 23634756 Ki = 9.6 nM T84631 C2KJ0P 23634757 Ki = 6.7 nM T84631 C6Z9WS 23634758 Ki = 2 nM T84631 C92VIM 23634877 Ki = 1.7 nM T84631 CY3NC8 23634878 Ki = 0.31 nM T84631 CP6Y7K 23634881 Ki = 0.63 nM T84631 C61GCE 23635132 Ki = 0.48 nM T84631 C75GTN 23635133 Ki = 0.85 nM T84631 C7HOG9 23635260 Ki = 1.1 nM T84631 CR9BK5 23635261 Ki = 1584.89 nM T84631 CDHQ47 23635262 Ki = 180 nM T84631 C1KCZ6 23635264 Ki = 0.5 nM T84631 CR8AK4 23635386 Ki = 2.1 nM T84631 C7U9XO 23635500 Ki = 0.54 nM T84631 C8URE5 23635503 Ki = 4.8 nM T84631 CH9F4R 23635626 Ki = 0.67 nM T84631 CA07TV 23635750 Ki = 0.25 nM T84631 CA7Q4T 23635752 Ki = 610 nM T84631 C06FJI 23635753 Ki = 6 nM T84631 CTS9W8 23636240 Ki = 0.25 nM T84631 C50TMW 23636367 Ki = 3.9 nM T84631 C04CKF 23636368 Ki = 7.6 nM T84631 CZO8U6 23636369 Ki = 0.08 nM T84631 C10EHQ 23636370 Ki = 0.3 nM T84631 C7JF0K 23636371 Ki = 0.07 nM T84631 CCD8R5 23644670 Ki = 82 nM T84631 CEL6C2 23644671 Ki = 0.38 nM T84631 C6KY5R 23644672 Ki = 0.66 nM T84631 CJ1QC3 23646071 Ki = 7 nM T84631 CXIY21 23646108 Ki = 346 nM T84631 C6F3VD 23646109 Ki = 56 nM T84631 C83WUS 23646110 Ki = 2720 nM T84631 C4SB7E 23646111 Ki = 22 nM T84631 C6WB0S 23646112 Ki = 136 nM T84631 CM29UX 23646113 Ki = 57 nM T84631 CN18XI 23646114 Ki = 73 nM T84631 CET26V 23646115 Ki = 27 nM T84631 C1V0EW 23646116 Ki = 24 nM T84631 C1NO3E 23646117 Ki = 4100 nM T84631 C0GT7A 23646118 Ki = 15 nM T84631 CZ7U0G 23646119 Ki = 11 nM T84631 CF52TJ 23646120 Ki = 39000 nM T84631 CE71BT 23646121 Ki = 3 nM T84631 CTD16K 23646122 Ki = 2 nM T84631 CZ8CT7 23646123 Ki < 1 nM T84631 C5FG7J 23646124 Ki = 1 nM T84631 C4SL3W 23646125 Ki = 1 nM T84631 CQA78Z 23646126 Ki < 1 nM T84631 C8VA1Z 23646127 Ki = 60 nM T84631 CQ21XZ 23646128 Ki = 72 nM T84631 C16JDI 23646129 Ki = 63 nM T84631 CUX4J8 23646130 Ki = 1 nM T84631 CN7X8I 23646131 Ki = 2 nM T84631 CNK52C 23646132 Ki = 10600 nM T84631 CE5QN2 23646133 Ki = 50 nM T84631 CT9U3L 23646134 Ki = 320 nM T84631 CW2GJ6 23646135 Ki = 2060 nM T84631 CC3YP4 23646136 Ki = 160 nM T84631 C38SAT 23646137 Ki = 40 nM T84631 CXD31S 23646138 Ki = 82 nM T84631 C92MUL 23646153 Ki = 1.6 nM T84631 CJ9OA4 23646154 Ki = 0.13 nM T84631 CP23GI 23646155 Ki = 0.11 nM T84631 CH1LX7 23646156 Ki < 0.1 nM T84631 C83QCW 23646157 Ki = 0.34 nM T84631 CX8FL0 23646158 Ki = 0.12 nM T84631 C05YBQ 23646159 Ki = 0.22 nM T84631 CYB83X 23646160 Ki = 0.64 nM T84631 CZS9J8 23646161 Ki = 0.71 nM T84631 C3N8QU 23646162 Ki = 0.24 nM T84631 C7OC4K 23646163 Ki = 0.16 nM T84631 CA8EP1 23646164 Ki = 0.27 nM T84631 CVF49W 23646165 Ki = 0.34 nM T84631 CM94VT 23646166 Ki = 8.4 nM T84631 CY3CP9 23646167 Ki = 45 nM T84631 CIR80B 23646168 Ki = 1.5 nM T84631 C9OS8M 23646169 Ki = 2.1 nM T84631 CLKM63 23646170 Ki = 1.8 nM T84631 C08QUL 23646171 Ki = 0.82 nM T84631 CS80IC 23646172 Ki = 2.7 nM T84631 CZ9TO3 23646173 Ki = 12 nM T84631 CGS86R 23646174 Ki = 20 nM T84631 CGE2M7 23646175 Ki = 2 nM T84631 CK0X2L 23646176 Ki = 88 nM T84631 CX3GB9 23646177 Ki = 54 nM T84631 C07LKX 23646178 Ki = 47 nM T84631 C0IVO1 23646179 Ki = 2.6 nM T84631 CLC9F3 23646180 Ki = 1.2 nM T84631 CGVJ65 23646181 Ki = 0.18 nM T84631 C7MC5Y 23646182 Ki = 0.74 nM T84631 CGFT69 23646183 Ki = 2 nM T84631 C7P4VU 23646184 Ki = 0.18 nM T84631 C6Q1CR 23646185 Ki = 0.18 nM T84631 CKB59A 23646186 Ki = 0.12 nM T84631 CA0LC6 23646187 Ki = 0.2 nM T84631 CM01LP 23646188 Ki = 0.09 nM T84631 CA3U0I 23646189 Ki = 0.02 nM T84631 CIR65F 23646190 Ki = 0.03 nM T84631 CDK0P2 23646191 Ki = 0.04 nM T84631 CJ4U2X 23646192 Ki = 0.02 nM T84631 CMYI38 23646193 Ki = 0.42 nM T84631 CZ1KO7 23646194 Ki = 0.25 nM T84631 CPF54M 23646195 Ki = 0.29 nM T84631 CP84AB 23646196 Ki = 0.27 nM T84631 C2WK4G 23646197 Ki = 0.12 nM T84631 CC1FV9 23646198 Ki = 0.08 nM T84631 CG82YE 23646199 Ki = 0.27 nM T84631 C5KWB9 23646200 Ki = 5.4 nM T84631 CY8SQ7 23646201 Ki = 0.05 nM T84631 CCMZ94 23646202 Ki = 0.58 nM T84631 C08AOH 23646204 Ki = 0.26 nM T84631 C82COD 23646205 Ki = 0.31 nM T84631 CS5AL3 23646206 Ki = 0.2 nM T84631 C0EO5K 23646207 Ki = 0.65 nM T84631 CN1Q7D 23646208 Ki = 0.63 nM T84631 CP24HW 23646209 Ki = 2.5 nM T84631 C6UM7B 23646210 Ki = 1.3 nM T84631 C7NKV6 23646211 Ki = 26 nM T84631 CGB18F 23646212 Ki = 3 nM T84631 C5J3OT 23646213 Ki = 2.2 nM T84631 C3JF1O 23646214 Ki = 2.8 nM T84631 C75SDV 23646215 Ki = 14 nM T84631 C8G0NU 23646216 Ki = 6.1 nM T84631 C84HGM 23646217 Ki = 28 nM T84631 CATE50 23646218 Ki = 4 nM T84631 CC52RE 23646219 Ki = 7 nM T84631 C7CZ2J 23646220 Ki = 18 nM T84631 CLDZ20 23646221 Ki = 19 nM T84631 CM7X3R 23646222 Ki = 5.6 nM T84631 CG3ZB2 23646223 Ki = 160 nM T84631 CQS7X6 23646224 Ki = 45 nM T84631 CHAD98 23646225 Ki = 36 nM T84631 C8XZ3J 23646226 Ki = 72 nM T84631 CP9A1B 23646227 Ki = 810 nM T84631 CJS63R 23646228 Ki = 2600 nM T84631 CJN96Y 23646229 Ki = 79 nM T84631 C01VKP 23646230 Ki = 1100 nM T84631 CL14AX 23646231 Ki = 120 nM T84631 C96UDO 23646233 Ki = 2.5 nM T84631 C6RM8B 23646234 Ki = 47 nM T84631 C2U0RB 23646236 Ki = 4 nM T84631 CPMW70 23646237 Ki = 740 nM T84631 CS5CV9 23646239 Ki = 71 nM T84631 CV1HY5 23646241 Ki = 22 nM T84631 C6BG3M 23646243 Ki = 280 nM T84631 CU2V7C 23646245 Ki = 2020 nM T84631 C93IYD 23646247 Ki = 5360 nM T84631 C5LQ0H 23646249 Ki = 450 nM T84631 CS68GZ 23646251 Ki > 8000 nM T84631 C7FEL6 23646252 Ki > 8000 nM T84631 C3ZAY1 23646254 Ki > 8000 nM T84631 C6EF4Y 23646256 Ki = 3240 nM T84631 CKM7Y4 23646258 Ki = 410 nM T84631 C0UMW5 23646268 Ki = 2700 nM T84631 C2RV5T 23646269 Ki = 5700 nM T84631 C4YPZ3 23646288 Ki = 2 nM T84631 CD7YW3 23646289 Ki = 0.27 nM T84631 C25LRJ 23646290 Ki = 0.25 nM T84631 CI0W3O 23646291 Ki = 0.34 nM T84631 CM5VS7 23646292 Ki = 0.2 nM T84631 CQI1G4 23646293 Ki = 0.3 nM T84631 CY96RK 23646294 Ki = 0.4 nM T84631 CRX19I 23646295 Ki = 0.1 nM T84631 CP4GN0 23646296 Ki = 0.2 nM T84631 CI04YH 23646297 Ki = 0.53 nM T84631 CB3JK7 23646298 Ki = 0.52 nM T84631 COV42F 23646299 Ki = 0.54 nM T84631 CJR4X5 23646300 Ki = 0.15 nM T84631 CN2D0X 23646301 Ki = 0.55 nM T84631 C8GX6A 23646302 Ki = 0.86 nM T84631 CUF86C 23646303 Ki = 1.14 nM T84631 CU1Z9L 23646304 Ki = 0.08 nM T84631 C69ZVT 23646306 Ki = 0.02 nM T84631 CZ6GK2 23646308 Ki = 0.05 nM T84631 C5NF0J 23646310 Ki = 0.5 nM T84631 C2XQ7C 23646311 Ki = 0.35 nM T84631 CCRD27 23646312 Ki = 0.17 nM T84631 CLC17N 23646313 Ki = 0.5 nM T84631 CS2RE4 23646314 Ki = 0.18 nM T84631 C1WE6B 23646315 Ki = 0.21 nM T84631 CM4NQ5 23646316 Ki = 0.35 nM T84631 CAN6D5 23646317 Ki = 0.11 nM T84631 CKO58P 23646318 Ki = 0.22 nM T84631 C25WIE 23646319 Ki = 3.2 nM T84631 CLB4D5 23646320 Ki = 0.77 nM T84631 CDYF29 23646329 IC50 = 85000 nM T84631 CQB29J 23646453 Ki = 5600 nM T84631 C74AMD 23646454 Ki = 13300 nM T84631 CZ7JM9 23646455 Ki = 2300 nM T84631 CD9UH7 23646456 Ki = 2600 nM T84631 CX5S3K 23646457 Ki = 9100 nM T84631 CEH94J 23646458 Ki = 15300 nM T84631 C1DRZ7 23646459 Ki = 1500 nM T84631 CK64IY 23646460 Ki = 2200 nM T84631 CSY57G 23646463 Ki > 74000 nM T84631 CZ48JL 23646472 Ki = 10000 nM T84631 CJR27Q 23646473 Ki = 10000 nM T84631 CY5SE6 23646474 Ki = 156 nM T84631 C73ZDQ 23646475 Ki = 1053 nM T84631 C7CXM5 23646476 Ki = 285 nM T84631 C54VIZ 23646526 Ki = 110 nM T84631 CSL27U 23646528 Ki = 4830 nM T84631 CJ5CZ8 23646530 Ki = 14480 nM T84631 C7SZ4N 23646532 Ki = 180 nM T84631 CM74YK 23646533 Ki = 1310 nM T84631 CB1GR0 23646534 Ki = 3520 nM T84631 CSFH79 23646622 Ki = 440 nM T84631 C35HJA 23646623 Ki = 520 nM T84631 C7E4SA 23646732 Ki = 130 nM T84631 C4Z6FV 23647193 Ki = 103 nM T84631 C1L9VZ 23647194 Ki = 48 nM T84631 CU2Z6T 23647195 Ki = 225 nM T84631 CSG4O2 23647196 Ki = 345 nM T84631 CWHX79 23647197 Ki = 839 nM T84631 CC29KT 23647198 Ki = 12 nM T84631 CWCR31 23647199 Ki = 2730 nM T84631 CA52KT 23647200 Ki = 287 nM T84631 C9AG8L 23647650 Ki = 0.008 nM T84631 CI6N8M 23647676 Ki > 5000 nM T84631 C2QNL5 23647679 Ki = 3.4 nM T84631 CEP2K3 23647680 Ki = 1.5 nM T84631 CS08RA 23647681 Ki = 20 nM T84631 CQDG25 23647682 Ki = 5.7 nM T84631 CJC10T 23648140 Ki = 3 nM T84631 CC1Z9L 23648141 Ki = 5.7 nM T84631 C5ZP9A 23648142 Ki = 4.9 nM T84631 CR1BX3 23648143 Ki = 2.4 nM T84631 CARL42 23648144 Ki = 1.7 nM T84631 COI95T 23648145 Ki = 92 nM T84631 CM20FT 23648146 Ki = 14 nM T84631 CY75HR 23648147 Ki = 0.61 nM T84631 C2XIJ7 23648148 Ki = 0.73 nM T84631 C8F4ET 23648149 Ki = 0.67 nM T84631 C9HKT7 23648150 Ki = 0.7 nM T84631 CQ0RX9 23648151 Ki = 0.41 nM T84631 CM16WB 23648152 Ki = 0.26 nM T84631 C8PO4L 23648153 Ki = 0.57 nM T84631 CV6LR5 23648154 Ki = 0.87 nM T84631 CJ24TP 23648155 Ki = 0.26 nM T84631 CRW32H 23648156 Ki = 3.9 nM T84631 CH1D5R 23648157 Ki = 8.8 nM T84631 CU78RG 23648158 Ki = 29 nM T84631 C81PHJ 23648159 Ki = 6.6 nM T84631 CG3W5Q 23661706 IC50 > 30000 nM T84631 C9O1MH 23704948 IC50 > 5000 nM T84631 CKH4O5 24180463 Ki = 0.5 nM T84631 C7AYO1 24748789 IC50 = 20000 nM T84631 CVO5L6 24748791 IC50 = 13700 nM T84631 CUAY58 24749175 IC50 = 100000 nM T84631 C69OVW 24752832 IC50 = 16 nM T84631 CI93ZB 24752833 IC50 = 13 nM T84631 C3S1MT 24773377 Ki = 1.4 nM T84631 CF5I9O 24773378 Ki = 2255 nM T84631 CW8MT6 24773379 Ki = 4.1 nM T84631 CEQA82 24773380 Ki = 690 nM T84631 C93BFM 24773469 Ki = 4.9 nM T84631 C6N2IV 24773892 Ki = 8.1 nM T84631 CQTD47 24773893 Ki = 147 nM T84631 C6H7KF 24773969 Ki = 4.4 nM T84631 CGB15F 24773970 Ki = 231 nM T84631 C4CN1H 24774292 Ki > 14400 nM T84631 CO5JE3 24774293 Ki = 6850 nM T84631 CD6HV2 24774371 Ki = 26 nM T84631 CWX96Z 24774372 Ki = 22.9 nM T84631 CO2U9L 24774373 Ki = 6.4 nM T84631 CSW54F 24794406 Ki = 5.5 nM T84631 C8X5FS 24836819 Ki = 0.021 nM T84631 CJSO87 24849206 Ki = 7 nM T84631 CF7VA8 24858772 Ki = 1050 nM T84631 C6W5XL 24858773 Ki = 9270 nM T84631 CES0Y3 24858774 Ki = 15900 nM T84631 C9N8CR 24858929 Ki = 1940 nM T84631 C7QK4H 24858930 Ki = 5710 nM T84631 CWX43I 24858931 Ki = 58700 nM T84631 CNAG78 24858932 Ki = 139000 nM T84631 C8RHA3 24858933 Ki = 33200 nM T84631 C0UA9T 24860449 IC50 > 50000 nM T84631 C52CJA 24860451 IC50 > 50000 nM T84631 COX4A7 24873356 Ki = 4500 nM T84631 CYU34A 24881188 IC50 = 910 nM T84631 C9R2QI 24881190 IC50 = 460 nM T84631 C70AFO 24881191 IC50 = 54 nM T84631 C3KRV6 24881192 IC50 = 6.9 nM T84631 CO06JI 24881193 IC50 = 170 nM T84631 C2ON8C 24881194 IC50 = 56 nM T84631 CB20OY 24881251 IC50 = 160 nM T84631 C0FY1U 24881252 IC50 = 1400 nM T84631 CU6NH0 24881253 IC50 = 56 nM T84631 C87LAW 24881255 IC50 = 37 nM T84631 CDH1E3 24881256 IC50 = 300 nM T84631 C9PHM0 24882178 IC50 = 12 nM T84631 CY61BZ 24882254 IC50 = 23 nM T84631 C2RA7O 24882255 IC50 = 120 nM T84631 CE2U6A 24882256 IC50 = 31 nM T84631 C62GNZ 24882257 IC50 = 230 nM T84631 CT26DH 24882258 IC50 = 170 nM T84631 CKWT73 24882259 IC50 = 1600 nM T84631 CKJ7M2 24882363 IC50 = 50 nM T84631 CYJI62 24936113 Ki < 0.1 nM T84631 CYRU05 24936173 IC50 = 1.7 nM T84631 CQ52VL 24936196 Ki < 0.4 nM T84631 CY7BX0 24936197 Ki < 0.3 nM T84631 C7H5DI 24936198 Ki = 0.2 nM T84631 C3BD4T 24997732 Ki = 55 nM T84631 CN0ZW3 24999867 Ki > 1000 nM T84631 CEM32W 25001205 Ki > 1000 nM T84631 CJ84TQ 25015739 IC50 = 8.6 nM T84631 CAO2V4 25030840 Ki = 19000 nM T84631 CU82IO 25030929 Ki = 11200 nM T84631 C7MCT6 25031099 Ki = 2100 nM T84631 C5PO7A 25031100 Ki = 18000 nM T84631 CH7Z1K 25031101 Ki = 8200 nM T84631 CEW9X2 25031102 Ki = 6100 nM T84631 C9NC4S 25031541 Ki = 10000 nM T84631 CK5R8Q 25032200 Ki = 2500 nM T84631 CG8HY2 25032202 Ki = 15000 nM T84631 CH76XK 25032204 Ki = 26000 nM T84631 CN23DH 25049955 IC50 = 0.8 nM T84631 CZ78XH 25049956 IC50 = 0.54 nM T84631 CVS5A8 25049959 IC50 = 0.48 nM T84631 CO4PK0 25050108 IC50 = 0.38 nM T84631 CJR65Q 25050945 IC50 = 6.1 nM T84631 C29CKQ 25050946 IC50 = 2.1 nM T84631 CY61SV 25051116 IC50 = 5.6 nM T84631 CX5P3Q 25051117 IC50 = 3.5 nM T84631 CQK9R2 25051277 IC50 = 2.9 nM T84631 CYG9R7 25051278 IC50 = 2 nM T84631 CP0GX3 25051281 IC50 = 0.93 nM T84631 CO1Q3B 25051600 IC50 = 4.1 nM T84631 CR81PB 25052256 IC50 = 1.3 nM T84631 CBG9P4 25052257 IC50 = 2.3 nM T84631 C4PGS3 25052258 IC50 = 10 nM T84631 C16GLV 25052749 IC50 = 10 nM T84631 C07BZQ 25107507 Ki = 50300 nM T84631 CK3FM6 25107508 Ki = 31600 nM T84631 CN3I9J 25107569 Ki = 112000 nM T84631 CB6H7T 25107570 Ki = 2670 nM T84631 CC40FO 25107571 Ki = 112000 nM T84631 C1QC4Y 25107572 Ki = 16000 nM T84631 CKJ04T 25107573 Ki = 27700 nM T84631 CN8Y0B 25107634 Ki = 9590 nM T84631 C84XCZ 25107635 Ki = 16600 nM T84631 CCY26A 25107636 Ki = 29700 nM T84631 CO03GM 25107637 Ki = 29500 nM T84631 CNR43C 25107638 Ki = 12100 nM T84631 CDAC04 25107705 Ki = 33800 nM T84631 CYS45L 25107706 Ki = 43100 nM T84631 CYS98D 25107707 Ki = 49600 nM T84631 CRV78W 25107708 Ki = 11900 nM T84631 CF85WU 25107709 Ki = 18000 nM T84631 C23YAU 25107770 Ki = 11800 nM T84631 CQZ70E 25107771 Ki = 35400 nM T84631 CEK7G5 25107772 Ki = 74700 nM T84631 C3V7JU 25107773 Ki = 31700 nM T84631 C4LUT7 25113610 Ki = 9 nM T84631 CPBC45 25138134 IC50 = 110 nM T84631 CK2WL4 25138136 IC50 = 114 nM T84631 C1XY0D 25138137 IC50 = 430 nM T84631 C72JBP 25138138 IC50 = 650 nM T84631 CN10CG 25138139 IC50 = 13700 nM T84631 CB3FJ8 25138140 IC50 = 8.9 nM T84631 C9H0OL 25138141 IC50 = 118 nM T84631 CI8HE3 25138142 IC50 = 2.4 nM T84631 CW8B3G 25138143 IC50 = 9 nM T84631 CTE97L 25138144 IC50 = 290 nM T84631 CBV14T 25138145 IC50 = 17000 nM T84631 C2H4PJ 25166809 Ki = 5200 nM T84631 CG76TR 25181493 Ki = 360 nM T84631 CAX4Q1 25198342 Ki = 550 nM T84631 C16ILQ 25198493 Ki = 911 nM T84631 C6V9TD 25198622 Ki = 9800 nM T84631 CV46JB 25198623 Ki = 56 nM T84631 C4S0ZM 25210468 IC50 = 0.1 nM T84631 C5RJ1T 25210469 IC50 = 0.08 nM T84631 CV4O1F 25222767 Ki = 1450 nM T84631 C1W3CU 25222769 Ki = 9470 nM T84631 C1U9AE 25222771 Ki = 57 nM T84631 C15CWG 25222774 Ki = 260000 nM T84631 CH92VC 25222868 Ki = 2000 nM T84631 CEC04N 25222874 Ki = 2500 nM T84631 C8WG3X 25222971 Ki = 57000 nM T84631 CBP53A 25222975 Ki = 1000 nM T84631 CHTV50 25222977 Ki = 3870 nM T84631 CJ67WP 25222979 Ki = 767 nM T84631 C9WQU4 25222981 Ki = 512 nM T84631 CMY62V 25223085 Ki = 130 nM T84631 C4DK1F 25223087 Ki = 666 nM T84631 CL1WP8 25223089 Ki = 33800 nM T84631 CQ5OP1 25224184 Ki = 126000 nM T84631 CK5RQ4 25224186 Ki = 5200 nM T84631 CYD28U 25224296 Ki = 177 nM T84631 CFRU38 25224298 Ki = 548 nM T84631 CHD01M 25224300 Ki = 1270 nM T84631 C43UCD 25268815 IC50 = 9 nM T84631 CKM7Y8 25269170 Ki = 1.1 nM T84631 C37QUZ 25269526 IC50 = 3.2 nM T84631 CT0J3X 25270897 IC50 = 11.6 nM T84631 CU5YR1 41583852 IC50 > 200000 nM T84631 C62HGQ 42628060 Ki = 8 nM T84631 CJX5A6 42628061 Ki = 95 nM T84631 C3M0RO 42628062 Ki = 93 nM T84631 C19WJB 42628063 Ki = 31 nM T84631 CVAI06 42643068 Ki = 442 nM T84631 CUF74S 42643069 Ki = 162 nM T84631 CZ03OW 42643070 Ki = 112 nM T84631 CZ7M8C 42643120 Ki = 99 nM T84631 C0KN2D 42643121 Ki = 32 nM T84631 CL6GN4 42643122 Ki = 18 nM T84631 C6U1KC 42643173 Ki = 74 nM T84631 CC0XK4 42643174 Ki = 6 nM T84631 CV4EW7 42643175 Ki = 175 nM T84631 CN70MF 42643176 Ki = 1272 nM T84631 CHBR63 42643177 Ki = 11 nM T84631 CR1DQ2 42643222 Ki = 20 nM T84631 CH3IF2 42643277 Ki = 27 nM T84631 CRLZ98 42643388 Ki = 94 nM T84631 CQLA03 42643389 Ki = 132 nM T84631 C8ZJ0B 44156919 IC50 = 3280 nM T84631 CPX15D 44188281 IC50 = 7.1 nM T84631 CR8W6M 44200855 IC50 = 1.8 nM T84631 C4TZ2X 44201094 IC50 = 1.1 nM T84631 C9OMR4 44264598 Ki = 8700 nM T84631 CPRE58 44264710 Ki = 193 nM T84631 CA8N9H 44264719 Ki = 120 nM T84631 CW1G8N 44264814 Ki = 200 nM T84631 CF49JR 44264817 Ki = 59000 nM T84631 C6IDX1 44264832 Ki = 5000 nM T84631 CT40BD 44264834 Ki = 100000 nM T84631 C2XLN7 44264885 Ki = 7.1 nM T84631 CW4R8J 44264888 Ki = 2.2 nM T84631 CT2V6S 44264889 Ki = 3 nM T84631 CDNH87 44264912 Ki = 130 nM T84631 CZDW40 44264920 Ki = 3.3 nM T84631 C9RZ0O 44264921 Ki = 3.7 nM T84631 CXQ1H9 44264935 Ki = 14 nM T84631 C6O5VF 44264936 Ki = 2.5 nM T84631 CVBG38 44264940 Ki = 1.7 nM T84631 C63WPN 44264954 Ki = 34 nM T84631 CB3AQ1 44264955 Ki = 10 nM T84631 CGCI69 44264981 Ki = 1.2 nM T84631 C78WPK 44264995 Ki = 69 nM T84631 C01WIT 44265005 Ki = 15 nM T84631 C1BP7E 44265006 Ki = 11 nM T84631 CQNX29 44265034 Ki = 5.5 nM T84631 CQGC19 44265371 Ki = 43 nM T84631 CW6G5E 44271568 Ki = 2 nM T84631 CD2Z4T 44271573 Ki = 2 nM T84631 C65YHR 44271609 Ki = 25 nM T84631 CA18XV 44271621 Ki = 180 nM T84631 C13CDQ 44271631 Ki = 2 nM T84631 CA53QR 44271633 Ki = 35 nM T84631 C8BRO7 44271634 Ki = 48 nM T84631 C0SNH2 44271651 Ki = 75 nM T84631 CM4HK1 44271680 Ki = 1 nM T84631 C8U9EQ 44271692 Ki = 80 nM T84631 CC8G0D 44271702 Ki = 75 nM T84631 C4A5XW 44271749 Ki = 14 nM T84631 C9TD2K 44271760 Ki = 135 nM T84631 CU51BQ 44271777 Ki = 9 nM T84631 C7AS8L 44271778 Ki = 10 nM T84631 CMCS75 44272530 Ki = 36 nM T84631 C6GRO0 44272532 Ki = 5.8 nM T84631 C96TGO 44272560 Ki = 600 nM T84631 C65SNR 44272562 Ki = 3.1 nM T84631 C8CJI6 44272581 Ki = 150 nM T84631 CKZ6O0 44272690 Ki > 338 nM T84631 CB64EA 44272825 Ki = 1810 nM T84631 C1B9MI 44273291 IC50 = 70 nM T84631 C05TZL 44273376 IC50 = 66 nM T84631 C86OEF 44273389 IC50 = 22 nM T84631 CWU7G4 44273492 IC50 = 114 nM T84631 C1Z2QU 44273493 Ki = 2.5 nM T84631 C6ABM8 44273514 IC50 = 23 nM T84631 CW59QS 44273576 IC50 = 36 nM T84631 C8H0FK 44273592 IC50 = 92 nM T84631 CP32GC 44273614 IC50 = 430 nM T84631 CH3S8F 44273615 IC50 = 40 nM T84631 CYUQ93 44273643 IC50 = 13 nM T84631 C7EK0N 44273644 IC50 = 15 nM T84631 CV9C7T 44273645 Ki = 2.9 nM T84631 CR5A3C 44273666 IC50 = 108 nM T84631 CE3C6Q 44273679 IC50 = 26 nM T84631 CKUI85 44273680 IC50 = 380 nM T84631 C2S5UM 44273701 Ki = 1.1 nM T84631 CI9QM8 44273702 Ki = 0.5 nM T84631 CQ0HZ4 44273703 Ki = 0.3 nM T84631 CRA47X 44273704 IC50 = 39 nM T84631 CR6U4L 44273709 IC50 = 75 nM T84631 CZC9Q2 44273733 IC50 = 130 nM T84631 CJP8C0 44273734 IC50 = 112 nM T84631 CC30SE 44273735 IC50 = 215 nM T84631 CV13XP 44273736 IC50 = 94 nM T84631 CIQP84 44273737 IC50 = 131 nM T84631 C1HC0I 44273738 IC50 = 88 nM T84631 CZ5T6O 44273748 IC50 = 2100 nM T84631 C0A4ME 44273753 IC50 = 166 nM T84631 C2DJG4 44273754 Ki = 1.8 nM T84631 C8C1WF 44273817 IC50 = 3600 nM T84631 CCJN68 44273818 IC50 = 54000 nM T84631 CUG08B 44273828 IC50 = 680 nM T84631 CR3V4S 44273853 IC50 = 5200 nM T84631 CN4HE5 44273854 IC50 = 2900 nM T84631 C90AKQ 44273901 IC50 = 1100 nM T84631 CM3F7J 44273935 Ki = 1.1 nM T84631 CY4V8B 44273945 Ki = 2.8 nM T84631 C8ON3U 44273946 IC50 = 80 nM T84631 CI93OZ 44273947 IC50 = 48 nM T84631 CMD47X 44274011 Ki = 3.2 nM T84631 CL7NY5 44274017 Ki = 1.5 nM T84631 C68AOF 44274019 IC50 = 27 nM T84631 C7D5GB 44274020 IC50 = 47 nM T84631 C20PYG 44274030 IC50 = 110 nM T84631 C2BF3P 44274045 IC50 = 58 nM T84631 C41EMW 44274046 Ki = 0.5 nM T84631 CBAD49 44274051 IC50 = 479 nM T84631 CA10KD 44274052 IC50 = 377 nM T84631 C89BIR 44274053 IC50 = 34 nM T84631 CP1GC0 44274058 Ki = 1.8 nM T84631 C7I2DQ 44274065 IC50 = 7800 nM T84631 CI9E6O 44274072 IC50 = 13 nM T84631 COHA75 44274088 IC50 = 41 nM T84631 CMG90C 44274089 IC50 = 2 nM T84631 C6GKD2 44274282 IC50 = 22 nM T84631 CO7Z3E 44274843 Ki = 0.3 nM T84631 C7FP2X 44274865 Ki = 0.28 nM T84631 CNZ83L 44274886 Ki = 4 nM T84631 C9UP2G 44274929 Ki = 0.1 nM T84631 C9WDV8 44274930 Ki = 0.31 nM T84631 C3U8OC 44274931 Ki = 0.4 nM T84631 C2U5SO 44274945 Ki = 58 nM T84631 C5VE6G 44275194 Ki = 0.2 nM T84631 CT2J0P 44275195 Ki = 5 nM T84631 C42RVS 44275227 Ki = 13 nM T84631 CQ12EP 44275238 Ki = 74 nM T84631 C3OM8S 44275239 Ki = 0.1 nM T84631 CGOH67 44275240 Ki = 1.3 nM T84631 CU52WR 44275243 Ki = 8 nM T84631 C2HO4D 44275249 Ki = 0.028 nM T84631 C1N5GM 44275254 Ki = 0.46 nM T84631 CX1C4Q 44275257 Ki = 0.08 nM T84631 C9EKZ2 44275271 Ki = 64 nM T84631 C4TBU7 44275275 Ki = 50 nM T84631 C2D9YK 44275287 Ki = 2.2 nM T84631 CPBU68 44275289 Ki = 180 nM T84631 CL4D3K 44275297 Ki = 260 nM T84631 C3LS5P 44275326 Ki = 670 nM T84631 CHJC81 44275330 Ki = 34 nM T84631 C4SO5M 44275345 Ki = 150 nM T84631 CBA9T0 44275361 Ki = 17 nM T84631 CEWU09 44275365 Ki = 50 nM T84631 CVU1T9 44277085 IC50 > 2500 nM T84631 C19OGX 44278104 Ki = 385 nM T84631 C4A1ZJ 44282153 Ki > 10000 nM T84631 C5DZ4L 44282601 Ki > 10000 nM T84631 CRT93X 44282678 Ki > 10000 nM T84631 CA6X2L 44283195 Ki > 10000 nM T84631 CK29QN 44284451 IC50 = 7 nM T84631 CR09BC 44284461 IC50 = 362 nM T84631 CI65CK 44284478 IC50 = 35 nM T84631 CFJ9X2 44284522 IC50 = 245 nM T84631 CMU9A4 44284541 IC50 = 0.5 nM T84631 CI9H5W 44284543 IC50 = 5 nM T84631 CXK3M6 44284559 IC50 = 0.2 nM T84631 C6MUA4 44284604 IC50 = 759 nM T84631 C2JXL4 44284641 IC50 = 99 nM T84631 C96SRI 44284734 IC50 = 7 nM T84631 C36PXQ 44284752 IC50 = 99 nM T84631 CDAO90 44284753 IC50 = 664 nM T84631 C26YIW 44284754 IC50 = 628 nM T84631 C9DE2B 44284786 Ki = 0.18 nM T84631 CM4B7C 44284787 IC50 = 1.5 nM T84631 C41JHD 44284797 IC50 = 0.75 nM T84631 CUC1P9 44284803 IC50 = 2.6 nM T84631 CDM4W1 44284804 IC50 = 3 nM T84631 CEG25W 44284810 IC50 = 234 nM T84631 C4XE0Z 44284859 IC50 = 3.7 nM T84631 C2RCE1 44284893 IC50 = 9 nM T84631 C1IQY7 44284894 IC50 = 53 nM T84631 CR26VN 44284895 IC50 = 48 nM T84631 C31KIT 44284934 IC50 = 15 nM T84631 CU57SJ 44284940 IC50 = 17 nM T84631 C6Y7AO 44284957 IC50 = 18 nM T84631 C0KF4D 44284959 IC50 = 6470 nM T84631 CMZ71H 44284992 Ki = 0.58 nM T84631 CQ3N4P 44285111 IC50 = 13 nM T84631 C5NU9L 44285118 Ki = 13 nM T84631 CZ89KE 44285126 IC50 = 191 nM T84631 CFDP09 44285127 IC50 = 10 nM T84631 C9UP4E 44285152 IC50 = 4 nM T84631 CB45NT 44285154 IC50 = 215 nM T84631 CU9G2F 44285211 Ki = 2.6 nM T84631 C0FPN1 44285253 Ki = 7.2 nM T84631 C9N1ZL 44285281 Ki = 1.2 nM T84631 C5PX3O 44285312 Ki = 4.3 nM T84631 C9LRW8 44285352 Ki = 23 nM T84631 CQ82ZW 44286426 IC50 = 2500 nM T84631 COPR02 44286428 IC50 = 905 nM T84631 CS5U7F 44286453 IC50 = 447 nM T84631 CPK5M6 44286709 Ki = 69000 nM T84631 CQ2A3R 44286878 Ki = 66000 nM T84631 CJP7K9 44286879 Ki > 75000 nM T84631 CRK53N 44286978 Ki = 53000 nM T84631 C0DG5R 44287043 Ki = 92000 nM T84631 C63JTG 44287260 IC50 = 11000 nM T84631 CB9D2R 44287527 IC50 = 3000 nM T84631 CCXM09 44287610 IC50 = 550 nM T84631 CB8IQ5 44287628 IC50 = 27 nM T84631 CT4N0L 44287629 IC50 = 28 nM T84631 CS5D4G 44287745 IC50 = 15 nM T84631 CL5I1S 44287757 IC50 = 140 nM T84631 C3QD4W 44287797 Ki = 120000 nM T84631 C5W7SA 44287798 Ki = 29000 nM T84631 CX47AK 44287838 IC50 = 60000 nM T84631 C5Q9OJ 44287854 IC50 = 46 nM T84631 C5UT7J 44287855 IC50 = 20 nM T84631 C02ARM 44287937 Ki > 200000 nM T84631 CP90NM 44288029 Ki = 110000 nM T84631 CZRH12 44290033 IC50 = 21 nM T84631 CUY95P 44290108 IC50 = 7820 nM T84631 CS76AC 44290361 IC50 = 9900 nM T84631 C3WR2N 44290375 IC50 = 3.6 nM T84631 CMY82L 44290376 IC50 > 20000 nM T84631 CHL9Y6 44290377 IC50 > 100000 nM T84631 CLDH85 44290378 IC50 = 3600 nM T84631 CXO05N 44290379 IC50 > 200000 nM T84631 CCH40M 44290403 IC50 = 25 nM T84631 CJ20SI 44290431 IC50 = 22 nM T84631 C0E3FW 44290444 IC50 = 226 nM T84631 C9D7QK 44290445 IC50 = 623 nM T84631 CD8E0V 44290452 IC50 = 3.4 nM T84631 C9ZYO2 44290453 IC50 = 5.6 nM T84631 CUH6W4 44290457 IC50 = 16 nM T84631 CNWI90 44290501 IC50 > 200000 nM T84631 CBE24K 44290502 IC50 > 100000 nM T84631 C94BSK 44290516 IC50 = 20000 nM T84631 CAXB95 44290518 IC50 > 50000 nM T84631 C49EPA 44290519 IC50 = 2200 nM T84631 C37IJH 44290520 IC50 = 3700 nM T84631 CU17NH 44290529 IC50 = 5600 nM T84631 CC8YQ3 44290530 IC50 = 74 nM T84631 CN04WY 44290542 IC50 = 14000 nM T84631 CF8JK0 44290543 Ki = 11 nM T84631 C05EYJ 44290555 IC50 = 120 nM T84631 C10ANS 44290556 IC50 = 26000 nM T84631 CO9JQ0 44290557 Ki = 6 nM T84631 CY60EW 44290560 Ki = 2 nM T84631 C70XKC 44290569 Ki = 2.7 nM T84631 C9QS3I 44290584 Ki = 46 nM T84631 CUW14A 44290648 Ki = 4 nM T84631 COB93L 44290673 Ki = 69 nM T84631 C2UV6T 44290696 Ki = 8 nM T84631 C8LY1J 44290712 Ki = 20 nM T84631 C0SYK2 44290731 Ki = 0.4 nM T84631 CN6KP1 44290929 Ki > 1200 nM T84631 C0E1RV 44290930 Ki = 1 nM T84631 C8APX2 44290947 Ki = 0.5 nM T84631 CZ7PT1 44290965 Ki = 2 nM T84631 CTA7I1 44291034 Ki = 8 nM T84631 CH59WK 44291046 Ki = 0.89 nM T84631 CYFC04 44291049 Ki = 0.8 nM T84631 C7TNE0 44291050 Ki = 0.58 nM T84631 CC4RN5 44291077 Ki = 3 nM T84631 C0BKW7 44293012 Ki = 340 nM T84631 C18BMD 44293013 Ki = 620 nM T84631 CMN52F 44293014 Ki = 160 nM T84631 CQ0MU6 44293035 Ki = 620 nM T84631 C2RZ0Q 44293068 Ki = 97 nM T84631 C8ANR4 44293069 Ki > 1200 nM T84631 C4QNY6 44293089 Ki = 170 nM T84631 CWTU04 44293097 Ki > 1200 nM T84631 CID0Q1 44293197 Ki > 1200 nM T84631 CQ5M9L 44293198 Ki = 430 nM T84631 C4JI1E 44293369 Ki > 1200 nM T84631 C07IRQ 44293370 Ki > 1200 nM T84631 CX15SW 44293371 Ki > 1200 nM T84631 CK5H8X 44293458 Ki > 1200 nM T84631 CWV12E 44293459 Ki > 1200 nM T84631 CT7Q9E 44293503 Ki = 140 nM T84631 C2FMV6 44293504 Ki = 59 nM T84631 CV3NJ0 44293505 Ki = 250 nM T84631 C5IX3B 44293517 Ki > 1200 nM T84631 C9BT7Y 44293520 Ki = 140 nM T84631 CMG6H7 44293524 Ki = 270 nM T84631 C18JSA 44293525 Ki > 1200 nM T84631 CXV2U0 44293745 Ki = 120 nM T84631 CYHM09 44293746 Ki = 51 nM T84631 CKX76L 44294121 Ki = 1100 nM T84631 CWZ6Y0 44294144 Ki = 190 nM T84631 C5AZX1 44294161 Ki = 180 nM T84631 CQH6J3 44294201 Ki = 300 nM T84631 C5P8QF 44294202 Ki = 130 nM T84631 CI8V6A 44295540 Ki > 30000 nM T84631 CBD7K8 44295640 Ki = 2300 nM T84631 C39DAX 44295655 Ki = 2300 nM T84631 CJIA32 44295656 Ki > 30000 nM T84631 CJ9P3I 44295714 Ki = 17000 nM T84631 CPH39G 44295719 Ki = 24000 nM T84631 C46QHZ 44295721 Ki > 30000 nM T84631 C0O2PG 44295723 Ki = 10 nM T84631 CVYK28 44295735 Ki > 3000 nM T84631 CH0E5L 44295746 Ki > 30000 nM T84631 C0CDH2 44295750 Ki > 30000 nM T84631 C7F8HQ 44295757 Ki > 3000 nM T84631 C8G9EL 44295762 Ki = 26000 nM T84631 C2F7KZ 44295778 Ki > 30000 nM T84631 CH9TZ2 44295784 Ki = 490 nM T84631 C6U9CB 44295788 Ki = 1000 nM T84631 C7SN2O 44295812 Ki = 45 nM T84631 C1JYX7 44295834 Ki > 30000 nM T84631 CO4CV7 44295859 Ki = 1000 nM T84631 CQGD83 44295860 Ki = 4500 nM T84631 CSU4I8 44295861 Ki = 5900 nM T84631 CG17NR 44295877 Ki = 1800 nM T84631 C5S9RT 44295886 Ki = 2100 nM T84631 C0VBP5 44295901 Ki = 1700 nM T84631 CJCG97 44295904 Ki = 4600 nM T84631 CYFO56 44295908 Ki = 1700 nM T84631 C0N7OK 44295909 Ki = 1300 nM T84631 C4TQP8 44295912 Ki = 1700 nM T84631 CRZ24O 44295918 Ki = 17000 nM T84631 CMY02C 44295921 Ki = 1600 nM T84631 C2FK9M 44295923 Ki = 1100 nM T84631 CNI38U 44295960 Ki = 13200 nM T84631 C7JPH8 44295961 Ki = 2700 nM T84631 CN6UB9 44295962 Ki = 2500 nM T84631 C79ELR 44295964 Ki = 2400 nM T84631 CSW5Q1 44295971 Ki = 7500 nM T84631 CGDS36 44295996 Ki = 7800 nM T84631 C3ZL5P 44296008 Ki = 700 nM T84631 C1O3YJ 44296027 Ki = 20000 nM T84631 C8AY9O 44296035 Ki = 7600 nM T84631 CLK7N1 44296052 Ki = 8400 nM T84631 CQ51FN 44296074 Ki = 1200 nM T84631 CETN87 44296078 Ki = 300000 nM T84631 C3DG0L 44296128 Ki = 4 nM T84631 CPF86Z 44296129 Ki = 350 nM T84631 C38SDX 44296130 Ki = 4300 nM T84631 C1WU8B 44296135 Ki = 20 nM T84631 C3O6LY 44296148 Ki = 4100 nM T84631 CHI4G1 44296149 Ki = 10000 nM T84631 C6WNO3 44296150 Ki = 11000 nM T84631 C8WKO5 44296170 Ki = 15000 nM T84631 CV31AF 44296181 Ki > 5000 nM T84631 CW8N6G 44296281 Ki = 1900 nM T84631 CXL8T3 44296383 Ki = 3 nM T84631 C9AGW7 44297775 Ki = 290 nM T84631 C5HX1A 44297783 Ki = 2800 nM T84631 C4LMD2 44298298 Ki > 5000 nM T84631 CGBX35 44298541 Ki > 5000 nM T84631 C5YZ0H 44298559 Ki > 5000 nM T84631 CJE93G 44298563 Ki > 5000 nM T84631 CWA7D2 44298564 Ki > 5000 nM T84631 CYQN71 44298587 Ki > 5000 nM T84631 CCRS93 44298594 Ki > 5000 nM T84631 CW5NL8 44298595 Ki > 5000 nM T84631 C5ZIQ1 44298940 Ki > 5000 nM T84631 CSKI34 44298941 Ki > 5000 nM T84631 CB5UA1 44298971 Ki > 5000 nM T84631 CU3NP5 44298972 Ki > 5000 nM T84631 CERA27 44299040 Ki > 5000 nM T84631 C29MVU 44303719 Ki > 470000 nM T84631 C3FB4I 44303721 Ki > 470000 nM T84631 CQLA16 44303733 Ki = 104000 nM T84631 C5RZL0 44303743 Ki = 1700 nM T84631 CTE75P 44303769 Ki = 37000 nM T84631 C16GOI 44303778 Ki = 2800 nM T84631 C26ZUK 44303789 Ki = 5200 nM T84631 CN6V9A 44303803 Ki = 2300 nM T84631 C67ZRW 44303804 Ki = 188000 nM T84631 CB38WA 44303805 Ki = 12000 nM T84631 CL0U1A 44303806 Ki = 5700 nM T84631 CVO2D9 44303808 Ki = 99000 nM T84631 C0JZY5 44303810 Ki = 15000 nM T84631 CFJ4W3 44303811 Ki = 9400 nM T84631 CE0R9A 44303824 Ki > 470000 nM T84631 C5YF7O 44303839 Ki > 470000 nM T84631 C2LY4T 44303843 Ki = 1000 nM T84631 C3HXW6 44303858 Ki = 78 nM T84631 CYW9S8 44303912 Ki = 240000 nM T84631 CIQZ37 44303925 Ki = 88000 nM T84631 CJN72A 44303933 Ki = 2100 nM T84631 CXCY31 44303935 Ki > 78000 nM T84631 C4SN8T 44304006 Ki > 470000 nM T84631 CL16JC 44304046 Ki > 470000 nM T84631 CAM6R0 44304047 Ki > 470000 nM T84631 CR4V0L 44304084 Ki = 68000 nM T84631 CG37DH 44304086 Ki = 235000 nM T84631 C7UJH1 44304087 Ki = 55000 nM T84631 CG0R8N 44304097 Ki = 13000 nM T84631 CJ80KE 44304098 Ki > 470000 nM T84631 CG8TI6 44304099 Ki > 470000 nM T84631 C9W8QC 44304100 Ki > 470000 nM T84631 CE31BF 44304104 Ki > 470000 nM T84631 C9XIO1 44304105 Ki > 470000 nM T84631 C83YIU 44304139 Ki = 151000 nM T84631 CP5S9K 44304192 Ki = 470000 nM T84631 CKD98A 44304353 Ki = 350000 nM T84631 CDNY01 44304666 IC50 > 11000 nM T84631 CU86PQ 44304683 IC50 > 11000 nM T84631 C2WER6 44304686 IC50 = 1800 nM T84631 C8FQD7 44304721 IC50 = 250 nM T84631 C9T0AL 44304783 IC50 = 9500 nM T84631 CV5X7Z 44304784 IC50 = 1300 nM T84631 C4C5QV 44304795 IC50 > 11000 nM T84631 CK30FU 44304796 IC50 = 5700 nM T84631 CJ9ZC7 44304847 IC50 = 1100 nM T84631 C0CVL6 44304925 IC50 = 1500 nM T84631 C6VMS3 44304940 IC50 = 220 nM T84631 CH5T1S 44304949 IC50 = 14 nM T84631 CH5KL1 44304966 IC50 = 190 nM T84631 CW2ND0 44304967 IC50 > 11000 nM T84631 CX68LN 44304970 IC50 = 1 nM T84631 CR92NX 44304975 IC50 = 78 nM T84631 C9FPX1 44304983 IC50 = 14 nM T84631 CSC71I 44305011 IC50 = 7 nM T84631 CI28LX 44305020 IC50 = 140 nM T84631 CC94HD 44305021 IC50 = 1500 nM T84631 C47VUA 44305033 IC50 = 2900 nM T84631 CX6HR3 44305497 IC50 = 36 nM T84631 C1TU6Q 44305498 IC50 > 11000 nM T84631 CGM7D3 44305549 IC50 = 530 nM T84631 CM6VI1 44305564 IC50 = 41 nM T84631 C85BPT 44305569 IC50 = 590 nM T84631 C2CUS5 44305576 IC50 = 27 nM T84631 C0B8EM 44305583 IC50 = 230 nM T84631 CNE75U 44305589 IC50 = 84 nM T84631 CJ5GZ8 44305595 IC50 = 3 nM T84631 CXSN91 44305596 IC50 = 270 nM T84631 C8RXZ9 44305609 IC50 = 230 nM T84631 CJ9P6T 44305616 IC50 = 24 nM T84631 C1F5ZJ 44305618 IC50 = 27 nM T84631 CR0F5Q 44305620 IC50 = 31 nM T84631 C8WPQ1 44305624 IC50 = 12 nM T84631 CN91ZP 44305641 IC50 = 67 nM T84631 CGQA30 44305642 IC50 = 640 nM T84631 CG2K9Z 44305652 IC50 = 7 nM T84631 CJSV68 44305653 IC50 = 7 nM T84631 C13RXM 44305655 IC50 = 5 nM T84631 CJ13QC 44305697 IC50 = 12 nM T84631 C9MS8B 44305700 IC50 = 70 nM T84631 C5OT9C 44305701 IC50 = 25 nM T84631 C0OGD3 44305702 IC50 = 10 nM T84631 CO1Y2P 44305705 IC50 = 57 nM T84631 C36BTK 44305707 IC50 = 1300 nM T84631 CNBM39 44305717 IC50 = 8 nM T84631 C4OA9H 44305740 IC50 = 37 nM T84631 CF9K6V 44305751 IC50 = 150 nM T84631 CK8OA9 44305755 IC50 = 14 nM T84631 CR1B5E 44305767 IC50 = 18 nM T84631 C8I2WA 44305768 IC50 = 240 nM T84631 C6D4WM 44305778 IC50 = 390 nM T84631 CPE2R8 44305779 IC50 = 64 nM T84631 CS1T4V 44305783 IC50 = 100 nM T84631 CP5Q9V 44305791 IC50 = 8 nM T84631 CD4K9F 44305792 IC50 = 11 nM T84631 CLI7J5 44305799 IC50 = 140 nM T84631 C09VHZ 44305800 IC50 = 11 nM T84631 CWDY81 44305841 IC50 = 29 nM T84631 CLP78H 44305852 IC50 = 8 nM T84631 CKCQ26 44305853 IC50 = 8 nM T84631 C09HMY 44305854 IC50 = 15 nM T84631 COS9P8 44305862 IC50 = 7 nM T84631 C4BXN1 44305898 IC50 = 19 nM T84631 C6X1UY 44305922 IC50 = 71 nM T84631 CWL6P8 44305926 IC50 = 90 nM T84631 C2OPT7 44305934 IC50 = 120 nM T84631 CZ67XS 44305943 IC50 = 160 nM T84631 C18LVJ 44305951 IC50 = 13 nM T84631 CL1RT7 44305959 IC50 = 11 nM T84631 C9OQ6V 44305961 IC50 = 9 nM T84631 CYD8Q6 44305962 IC50 = 430 nM T84631 C30CNB 44305966 IC50 = 240 nM T84631 CP0R6L 44305992 IC50 = 6 nM T84631 CWG3K9 44306043 IC50 = 30 nM T84631 C4EBA0 44306054 IC50 = 45 nM T84631 CG0V3Z 44306077 IC50 = 6 nM T84631 C2G0UZ 44306101 IC50 = 10 nM T84631 CMIB37 44306212 IC50 = 8 nM T84631 CN97SF 44310725 Ki = 1000 nM T84631 CKP5W7 44311564 IC50 > 1100 nM T84631 C6TQ7D 44312627 IC50 = 14 nM T84631 CTW03S 44312639 IC50 = 93 nM T84631 C18PFJ 44312776 IC50 = 6.3 nM T84631 CGS74O 44312851 IC50 = 6.4 nM T84631 CM5RQ6 44312966 IC50 = 2930 nM T84631 CGND24 44312967 IC50 = 0.99 nM T84631 CRN7I3 44313020 IC50 > 10000 nM T84631 C6G0NQ 44313284 IC50 = 227 nM T84631 CYQ4I0 44313285 IC50 = 4.4 nM T84631 C2D0JU 44313317 IC50 = 170 nM T84631 CU8S5P 44313405 IC50 = 12100 nM T84631 C1KQR4 44313688 Ki = 9 nM T84631 CUA30F 44313689 Ki = 84 nM T84631 C87HJP 44313722 IC50 = 590 nM T84631 C3H5RB 44313873 IC50 = 46.4 nM T84631 C8V3IH 44313932 IC50 = 6.6 nM T84631 C6VP5I 44314000 IC50 = 7.89 nM T84631 CT2ZD9 44314001 IC50 = 13.2 nM T84631 CFXW28 44314002 IC50 = 3.26 nM T84631 CM10DN 44314053 IC50 = 0.86 nM T84631 CCK1W8 44314117 IC50 = 0.78 nM T84631 CT1X8J 44314118 IC50 = 1.87 nM T84631 C5H6VU 44314181 IC50 = 2.13 nM T84631 CSTP54 44314265 IC50 = 7.63 nM T84631 CE6B9A 44314318 IC50 = 246 nM T84631 C9IN4E 44314967 IC50 = 2900 nM T84631 C97NYB 44317783 IC50 = 2500 nM T84631 C5AK3D 44317785 IC50 > 2500 nM T84631 CW2X9Z 44318052 IC50 = 2500 nM T84631 CK58VB 44318182 IC50 = 5.78 nM T84631 CND9J7 44319469 Ki = 50.12 nM T84631 CEZ84L 44320397 IC50 = 28.9 nM T84631 CSK62O 44320493 IC50 = 49 nM T84631 CYT2Q4 44320495 IC50 = 7.2 nM T84631 CG36WH 44320752 IC50 = 3.6 nM T84631 CQ64CD 44320839 IC50 = 26.7 nM T84631 CK1EZ2 44320862 IC50 = 7.3 nM T84631 C7AMH4 44320876 IC50 = 20.6 nM T84631 CX73RG 44324726 Ki = 800 nM T84631 CMZ05T 44324727 Ki = 4900 nM T84631 CI5BY6 44324744 Ki = 7500 nM T84631 CKDN47 44324745 Ki = 2500 nM T84631 CWN4P7 44325526 Ki = 490 nM T84631 C1MT8R 44325527 Ki = 420 nM T84631 C1K5OT 44325647 Ki ~ 75 nM T84631 CG6ZC8 44325794 Ki = 36 nM T84631 CBD24R 44325803 Ki = 0.04 nM T84631 CZW79L 44325865 Ki = 240 nM T84631 C4Q8AC 44325938 Ki = 480 nM T84631 C61VAC 44325939 Ki = 510 nM T84631 CK92AD 44325940 Ki = 200 nM T84631 C6LWG3 44325946 Ki = 2470 nM T84631 C5TLH0 44325953 Ki = 720 nM T84631 CHI47Q 44325959 Ki = 240 nM T84631 C1DES8 44325967 Ki = 160 nM T84631 C5CLJ1 44325971 Ki = 28 nM T84631 CYOQ97 44325982 Ki > 1200 nM T84631 C3A2IO 44325983 Ki = 110 nM T84631 CZ9J5R 44326160 Ki = 1310 nM T84631 CO2F4Z 44326181 Ki = 380 nM T84631 CF92WZ 44326243 Ki = 37 nM T84631 CE8W2L 44326303 Ki = 3690 nM T84631 CK1EF5 44326322 Ki = 7050 nM T84631 C90VZO 44326339 Ki = 23 nM T84631 CXDN72 44326446 Ki = 2384 nM T84631 C3NCW0 44327306 Ki = 950 nM T84631 CFV5D6 44327462 Ki = 1700 nM T84631 CI56QW 44327465 Ki = 1400 nM T84631 CTDM97 44327484 Ki = 1800 nM T84631 C86YFO 44327490 Ki = 870 nM T84631 CE3UL6 44327872 Ki = 800 nM T84631 CSM3B6 44330879 IC50 = 34.8 nM T84631 CVM21A 44330906 IC50 = 635 nM T84631 CY72JW 44330907 IC50 = 34.8 nM T84631 CA4Y1P 44330934 IC50 = 1440 nM T84631 C3K6JA 44330969 IC50 = 23 nM T84631 CXW57P 44330970 IC50 = 25 nM T84631 CU9Z4M 44330999 IC50 = 7.8 nM T84631 C9KW3Q 44331002 IC50 = 842 nM T84631 CJ9Y8Z 44331003 IC50 = 55 nM T84631 C1X4UM 44331004 IC50 = 3450 nM T84631 C2SK9N 44331021 IC50 = 130 nM T84631 C2CS3N 44331022 IC50 = 640 nM T84631 CAB5T7 44331052 IC50 = 45 nM T84631 CR7F8L 44331114 IC50 = 31.3 nM T84631 C4NP5G 44331140 IC50 = 676 nM T84631 CSDQ73 44331145 IC50 = 2770 nM T84631 C4CJ5M 44331146 IC50 > 10000 nM T84631 CFK17Y 44331147 IC50 = 1780 nM T84631 C2BS5N 44331180 IC50 = 96.7 nM T84631 C1NR3B 44331189 IC50 = 10000 nM T84631 CF13OL 44331190 IC50 = 644 nM T84631 CE69GW 44331194 IC50 = 3 nM T84631 C3SU1R 44331210 IC50 = 762 nM T84631 CW5S8K 44332563 IC50 = 750 nM T84631 CB3XG7 44332586 IC50 = 490 nM T84631 C0WEP3 44332603 IC50 = 1590 nM T84631 CN5Q6W 44332607 IC50 = 1180 nM T84631 C9ECP7 44332620 IC50 = 5910 nM T84631 CKZ57W 44332622 IC50 = 420 nM T84631 C37XNC 44332629 IC50 = 440 nM T84631 CKJ49D 44332675 IC50 = 253 nM T84631 CQ7SG4 44332689 IC50 = 1 nM T84631 CNK6Z7 44332698 IC50 = 890 nM T84631 CZA7S5 44332713 IC50 = 3790 nM T84631 C89GTH 44332752 IC50 = 1610 nM T84631 CXO92K 44332753 IC50 = 890 nM T84631 CXUK98 44332765 IC50 = 110 nM T84631 CZ64UF 44332770 IC50 = 57 nM T84631 CA1IJ0 44332771 IC50 = 41 nM T84631 C5M2LB 44333833 Ki = 5000 nM T84631 CYNL31 44333951 Ki = 80 nM T84631 C0FE1Y 44333960 Ki = 1390 nM T84631 CJ2IM6 44333972 Ki = 22 nM T84631 CNF52U 44333992 Ki = 438 nM T84631 CIO79X 44334002 Ki = 320 nM T84631 CTUX56 44334003 Ki = 130 nM T84631 CS5X8Z 44334242 Ki = 46 nM T84631 CYX2N3 44334264 Ki = 99 nM T84631 CNTU54 44334314 Ki = 62 nM T84631 CDMP53 44334315 Ki = 15 nM T84631 CI3CT4 44334316 Ki = 392 nM T84631 CL05HM 44334318 Ki = 630 nM T84631 CN4TX8 44334349 Ki = 300 nM T84631 CQA75Y 44334374 Ki = 54 nM T84631 CI0C4V 44334382 Ki = 810 nM T84631 C0O1XG 44334554 Ki = 30 nM T84631 CHM49Q 44337735 Ki = 106000 nM T84631 CV7HW5 44337751 Ki = 92000 nM T84631 C39GBZ 44337785 Ki = 95000 nM T84631 CX35DM 44337794 Ki = 87300 nM T84631 CN1WI2 44337821 Ki = 90200 nM T84631 C61CGV 44337884 IC50 = 50 nM T84631 C4EFA8 44337894 IC50 = 210 nM T84631 C0HP3T 44337899 IC50 = 190000 nM T84631 CH0K1J 44337917 IC50 = 1400 nM T84631 CG6T9S 44337925 IC50 = 81000 nM T84631 CA10BE 44337935 IC50 = 20000 nM T84631 C4ATV2 44337945 IC50 = 1400 nM T84631 C2AN5G 44337986 IC50 = 69 nM T84631 CFH80Q 44337989 IC50 = 27000 nM T84631 CTD5Q8 44338012 IC50 = 33000 nM T84631 C5OVP7 44338032 IC50 = 31000 nM T84631 CI8U6O 44338109 IC50 = 698 nM T84631 CHX17O 44339365 Ki = 200000 nM T84631 CSA5H1 44339376 Ki = 179000 nM T84631 CZR56N 44339399 Ki = 69000 nM T84631 C9B0SQ 44339404 Ki = 228000 nM T84631 CC2K4G 44339417 Ki = 80000 nM T84631 C5WZ9O 44339442 Ki > 500000 nM T84631 C0G3LP 44339443 Ki = 81000 nM T84631 C4CZ2V 44339453 Ki > 200000 nM T84631 C7E4KL 44339464 Ki = 176400 nM T84631 CV53DA 44339470 Ki = 131000 nM T84631 CB6R0I 44339610 Ki = 370600 nM T84631 C7TOG2 44339650 Ki = 252000 nM T84631 CKA1T3 44341287 IC50 = 290 nM T84631 CZ9BF5 44341288 IC50 > 2500 nM T84631 C4XEK1 44341417 IC50 = 29.7 nM T84631 CXL2Q8 44341827 Ki = 149000 nM T84631 CQ2PR0 44342242 Ki = 26 nM T84631 CC0Z8V 44343581 IC50 = 6.1 nM T84631 CW76HT 44343582 IC50 = 15 nM T84631 CD0TW8 44343615 IC50 = 5 nM T84631 C9NZE1 44343799 IC50 = 0.7 nM T84631 CAIZ35 44343800 IC50 = 168.8 nM T84631 C0W6EI 44343845 IC50 = 311 nM T84631 C46IGW 44343852 IC50 = 312.5 nM T84631 C5H3NY 44343853 IC50 = 312.5 nM T84631 C7B5GK 44343857 IC50 > 2500 nM T84631 C40EHX 44343858 IC50 = 44.4 nM T84631 C91PVF 44343859 IC50 = 5.6 nM T84631 C4MS5Q 44343972 IC50 = 106 nM T84631 C3ZI7A 44343993 IC50 = 106 nM T84631 CMEI89 44343994 IC50 = 20.5 nM T84631 CEA17Z 44344039 IC50 = 346.3 nM T84631 CUO74X 44344054 IC50 = 10.6 nM T84631 C60GZW 44344100 IC50 = 10.6 nM T84631 CREZ48 44344153 IC50 = 79.1 nM T84631 CM2YO1 44345652 Ki = 900 nM T84631 CAY34C 44347478 Ki = 400000 nM T84631 CT0QN1 44347480 Ki > 1000000 nM T84631 CV6KA1 44347491 IC50 > 2500 nM T84631 C2EH3B 44347493 IC50 = 451 nM T84631 C65ORY 44347498 IC50 = 369 nM T84631 CN7L4W 44347532 IC50 = 627 nM T84631 C1UN9I 44347534 Ki = 370000 nM T84631 CM3P8Z 44347559 IC50 > 2500 nM T84631 CJ5A8E 44347561 IC50 > 2500 nM T84631 C0V2FL 44347624 Ki = 1000000 nM T84631 CTQ93K 44347853 Ki = 3.3 nM T84631 CA7C9J 44347854 Ki = 0.39 nM T84631 CE2SA3 44347864 IC50 = 470 nM T84631 CDMG63 44347916 Ki > 10000 nM T84631 CEP6C1 44347929 Ki > 10000 nM T84631 CC50UP 44347950 Ki > 10000 nM T84631 C0PR3S 44347951 Ki = 4600 nM T84631 CW2B1L 44347973 Ki > 10000 nM T84631 C7F6BG 44347997 Ki = 19 nM T84631 CKBN18 44348006 Ki > 10000 nM T84631 CX85LK 44348013 Ki > 10000 nM T84631 CQTB91 44348014 Ki = 6230 nM T84631 CXN6O9 44348021 Ki > 10000 nM T84631 C64JUL 44348030 Ki > 10000 nM T84631 C58MFB 44348077 IC50 = 5.6 nM T84631 C2AQR9 44348078 IC50 = 78 nM T84631 CJ1XO7 44348087 Ki = 8 nM T84631 C95OVC 44348092 Ki = 1.2 nM T84631 CQ8CK5 44348093 Ki = 13 nM T84631 CEL8P9 44348097 IC50 = 17 nM T84631 C31JWA 44348108 Ki = 5.4 nM T84631 CPV7C4 44348111 Ki > 10000 nM T84631 CO5Y7S 44348145 Ki > 10000 nM T84631 C6O8NQ 44348177 Ki > 10000 nM T84631 CQM0O4 44348226 Ki > 10000 nM T84631 CPD32J 44348228 Ki = 10700 nM T84631 CH61QP 44348436 IC50 = 8.4 nM T84631 CA74EQ 44348505 IC50 = 180 nM T84631 C2M6TU 44348587 IC50 = 32 nM T84631 CED0Q4 44348616 IC50 = 15 nM T84631 CZI93S 44348618 IC50 = 5900 nM T84631 CR68KY 44348619 IC50 = 41 nM T84631 C5H7ZW 44348620 IC50 = 63 nM T84631 C94NSH 44348621 IC50 = 980 nM T84631 CYS5G0 44348624 IC50 = 8.2 nM T84631 CFWR38 44348631 IC50 = 10 nM T84631 CV5F9W 44348635 IC50 = 7.6 nM T84631 C6QXM9 44348648 IC50 = 7 nM T84631 C04CQG 44348722 IC50 = 20 nM T84631 CBR0V8 44348733 IC50 = 440 nM T84631 CP2H0Q 44348745 IC50 = 1200 nM T84631 CT49QY 44351237 Ki = 12 nM T84631 CRY7N5 44351253 Ki = 1400 nM T84631 C2XC3I 44353392 IC50 = 28000 nM T84631 CE8S5Y 44353433 IC50 = 2800 nM T84631 C8WAB5 44353443 IC50 = 1500 nM T84631 C8BC3Z 44358436 Ki = 3900 nM T84631 CZA62D 44358571 Ki = 38000 nM T84631 CPO39C 44358576 Ki = 0.71 nM T84631 CI24PJ 44358733 Ki = 94 nM T84631 C4ZW0K 44359352 IC50 = 580 nM T84631 CVJ38H 44359353 IC50 = 1220 nM T84631 CB5T2W 44359354 IC50 = 460 nM T84631 CG0MW7 44359453 IC50 = 90 nM T84631 C1KL4Q 44359454 IC50 = 80 nM T84631 CMA5R7 44359487 IC50 = 1970 nM T84631 CZ9E1S 44359501 IC50 = 1130 nM T84631 CPU61I 44359598 IC50 = 390 nM T84631 CZ2T4O 44359609 IC50 = 4400 nM T84631 C6AFY1 44359621 IC50 = 600 nM T84631 C2Q1NY 44359626 IC50 = 360 nM T84631 C5GZ0D 44359648 IC50 = 1120 nM T84631 C82XKL 44359703 IC50 = 2500 nM T84631 C29ANK 44359723 IC50 = 2500 nM T84631 CQ5F0T 44359724 IC50 = 2500 nM T84631 C4Y5HK 44359726 IC50 = 2500 nM T84631 CIKY14 44359730 IC50 = 20.6 nM T84631 C40POZ 44359735 IC50 = 290 nM T84631 CF0V6J 44359754 IC50 = 2500 nM T84631 C5P3UG 44359755 IC50 = 2500 nM T84631 C5UKJ2 44359756 IC50 = 2500 nM T84631 CQ10VZ 44359794 IC50 = 2500 nM T84631 C5ES1X 44359805 IC50 = 1950 nM T84631 C5CTA0 44359810 IC50 = 471 nM T84631 CSV16F 44359885 IC50 > 2500 nM T84631 CD3R9Q 44359906 IC50 = 479 nM T84631 CMDB96 44360123 IC50 = 1100 nM T84631 C79GAF 44362167 Ki = 3499.45 nM T84631 C4Y0TJ 44362180 Ki = 34994.52 nM T84631 C3UYO8 44362181 Ki = 33113.11 nM T84631 CBFW89 44362183 Ki = 2301.44 nM T84631 CM4UL0 44362193 Ki = 25118.86 nM T84631 CA8B0F 44362198 Ki = 95499.26 nM T84631 CKY09S 44362201 Ki = 15995.58 nM T84631 CDM7W1 44362220 Ki = 39994.47 nM T84631 CH8S3E 44362221 Ki = 10964.78 nM T84631 CVY70U 44362237 Ki = 13001.7 nM T84631 CS6CA2 44362238 Ki = 2511.89 nM T84631 C7BEC4 44362239 Ki = 51999.6 nM T84631 C6W3XA 44362244 Ki = 70957.78 nM T84631 CK8PS0 44362245 Ki = 76032.63 nM T84631 CH5GN7 44362276 Ki = 15995.58 nM T84631 C7R6GJ 44362294 Ki = 57942.87 nM T84631 C47UOB 44362295 Ki = 41975.9 nM T84631 C9Y4GO 44362301 Ki = 79983.43 nM T84631 C8V2SK 44362302 Ki = 119949.93 nM T84631 CC8S0D 44362303 Ki = 77624.71 nM T84631 CH2JG8 44362312 Ki = 43351.09 nM T84631 C4OGX6 44362314 Ki = 76032.63 nM T84631 C7ZC4W 44362327 Ki = 16982.44 nM T84631 CL8FT9 44362329 Ki = 41495.4 nM T84631 C2BSP7 44362336 Ki = 26001.6 nM T84631 CO3T2F 44362337 Ki = 179887.09 nM T84631 C4DTY9 44362338 Ki = 2600.16 nM T84631 CVG80E 44362342 Ki = 17988.71 nM T84631 CL9CY2 44362343 Ki = 3198.9 nM T84631 C0D3TA 44362364 Ki = 2301.44 nM T84631 CW8BP5 44362367 Ki = 359749.34 nM T84631 CWZ91O 44362370 Ki = 17988.71 nM T84631 CR1W2C 44362374 Ki = 53951.06 nM T84631 CAR1I5 44362386 Ki = 26001.6 nM T84631 C3VU1F 44362388 Ki = 7603.26 nM T84631 CM43VS 44362389 Ki = 2511.89 nM T84631 C2JF6K 44362390 Ki = 46773.51 nM T84631 CC10SF 44362395 Ki = 38018.94 nM T84631 CC19SB 44362401 Ki = 64565.42 nM T84631 CC3LE4 44362404 Ki = 43651.58 nM T84631 CQ6HR5 44362406 Ki = 8090.96 nM T84631 CBP5C2 44362409 Ki = 100000 nM T84631 CFTC83 44362421 Ki = 35974.93 nM T84631 CE9I1R 44362422 Ki = 26977.39 nM T84631 C7GC4F 44362435 Ki = 19010.78 nM T84631 C2JPQ1 44362436 Ki = 8590.14 nM T84631 CIRJ69 44362445 Ki = 60255.96 nM T84631 C6IJ9O 44362457 Ki = 899.5 nM T84631 CG5X8L 44362464 Ki = 2197.86 nM T84631 CRZO54 44362466 Ki = 1513.56 nM T84631 C3UQ2G 44362474 Ki = 9705.1 nM T84631 CP7K9D 44362494 Ki = 46025.66 nM T84631 CNV52T 44362496 Ki = 16982.44 nM T84631 CZO9L1 44362497 Ki = 50003.45 nM T84631 CQM36L 44362517 Ki = 13001.7 nM T84631 CWVC27 44362544 Ki = 26977.39 nM T84631 CTXH42 44362558 Ki = 83176.38 nM T84631 CL5N9S 44362560 Ki = 21978.6 nM T84631 CD95NC 44362564 Ki = 7762.47 nM T84631 CG6MS9 44362581 Ki = 34994.52 nM T84631 CVR0L5 44362589 Ki = 130016.96 nM T84631 CA2PW9 44362609 Ki = 230144.18 nM T84631 C13XMI 44362611 Ki = 14125.38 nM T84631 CJD6N8 44362617 Ki = 10000 nM T84631 C3PWL5 44362648 Ki = 11994.99 nM T84631 C1N8AG 44362663 Ki = 21978.6 nM T84631 C74DSW 44362679 Ki = 6760.83 nM T84631 CX30CV 44362681 Ki = 19998.62 nM T84631 CSXG35 44362682 Ki = 109900.58 nM T84631 CC7TB6 44362760 Ki = 41020.41 nM T84631 CCAS16 44362802 Ki = 190107.83 nM T84631 C17REG 44362803 Ki = 1000000 nM T84631 CPF78Q 44362805 Ki = 639734.84 nM T84631 CJ6M0W 44362819 Ki = 3097.42 nM T84631 C2P6RJ 44364043 Ki = 200 nM T84631 C06RPS 44364101 Ki = 1000 nM T84631 C8H3IU 44364106 Ki = 200 nM T84631 C0B3TG 44364107 Ki = 80 nM T84631 CN46VL 44364123 Ki = 200 nM T84631 C1P0MS 44364177 Ki = 400 nM T84631 CYK89L 44364205 Ki = 3000 nM T84631 CP7K4W 44364302 Ki = 2000 nM T84631 C4LH6Q 44364310 Ki = 3000 nM T84631 CB85LE 44364311 Ki = 200 nM T84631 CDE32K 44364319 Ki = 30 nM T84631 CTC3O5 44364320 Ki = 2000 nM T84631 CSI3V9 44364329 Ki = 3000 nM T84631 CUM70S 44364371 Ki = 2000 nM T84631 C9Z7JD 44364382 Ki = 44 nM T84631 CT8QM1 44364445 Ki = 30 nM T84631 CTB86G 44364486 Ki = 55 nM T84631 C1ELX6 44364487 Ki = 1000 nM T84631 CQ1LM8 44364504 Ki = 100 nM T84631 CS2D1R 44364505 Ki = 400 nM T84631 CQE3K8 44364506 Ki = 200 nM T84631 CT10GM 44364862 Ki = 7.1 nM T84631 CDIR32 44364938 Ki = 210 nM T84631 CL1O0R 44364939 Ki > 5000 nM T84631 CYD1M4 44364940 Ki = 78 nM T84631 CXD05A 44364941 Ki = 960 nM T84631 COJ03I 44364946 Ki > 5000 nM T84631 C5M2CT 44364948 Ki > 5000 nM T84631 CM87YB 44364952 Ki > 5000 nM T84631 CD93ET 44364982 Ki > 5000 nM T84631 CG4RV3 44364999 Ki > 500 nM T84631 CTVZ78 44365103 Ki > 5000 nM T84631 CNO4X7 44365111 Ki > 5000 nM T84631 CIDS76 44365112 Ki = 4700 nM T84631 C4OE2C 44365192 Ki > 5000 nM T84631 CEH1M4 44365200 Ki > 5000 nM T84631 CFZ2T9 44365277 Ki = 280 nM T84631 C3GA5J 44365287 Ki = 1400 nM T84631 CN4D2F 44365289 Ki > 5000 nM T84631 C5YT9W 44366105 Ki = 1 nM T84631 CT1F2W 44366339 Ki = 0.46 nM T84631 C0L3YP 44367992 IC50 = 1570 nM T84631 CRD97F 44368086 IC50 = 7 nM T84631 C0HVT6 44368087 IC50 = 3 nM T84631 COQ97A 44368088 IC50 = 9 nM T84631 CZY31U 44368261 IC50 = 14900 nM T84631 C4B9CA 44368277 IC50 = 1050 nM T84631 C01GQT 44368278 IC50 = 6920 nM T84631 CJ4O0M 44368282 IC50 > 10000 nM T84631 C67DWF 44368293 IC50 = 14 nM T84631 CGQA02 44368299 IC50 = 3 nM T84631 C78XDG 44368377 IC50 = 25 nM T84631 C1LST9 44368378 IC50 = 31 nM T84631 CH3E9V 44368542 IC50 = 4060 nM T84631 CC2F9Z 44368575 IC50 = 6 nM T84631 C6OF4C 44368576 IC50 = 0.8 nM T84631 C37ZDX 44368590 IC50 = 7000 nM T84631 CCN24M 44368609 IC50 = 934 nM T84631 CTPD09 44368610 IC50 = 3933 nM T84631 CBT5V7 44368623 IC50 = 7 nM T84631 C62DWQ 44368626 IC50 = 153 nM T84631 CR12CY 44368637 IC50 = 500 nM T84631 CM2CE0 44368638 IC50 = 191 nM T84631 CAGX61 44368877 Ki = 2100 nM T84631 C8ABU5 44368882 Ki = 1400 nM T84631 C3PHI0 44369086 Ki = 0.15 nM T84631 CWK6U8 44369271 Ki = 0.013 nM T84631 C1HBT5 44369288 Ki < 0.005 nM T84631 C6XB0Y 44371477 Ki = 2900 nM T84631 C3T0PF 44372395 Ki = 0.82 nM T84631 CAJ92B 44372499 Ki = 2.3 nM T84631 CI32UH 44372518 Ki = 0.4 nM T84631 C7I3HS 44372533 Ki = 0.2 nM T84631 CJE89V 44372620 Ki = 8.2 nM T84631 C39FZP 44372663 Ki = 15000 nM T84631 C9I0BE 44372667 Ki = 500 nM T84631 CQLA75 44372683 Ki = 100000 nM T84631 CKFN05 44372724 Ki > 1000000 nM T84631 CTD36H 44372738 Ki = 140000 nM T84631 CI6MQ5 44372778 Ki = 10600 nM T84631 CUVD59 44372831 Ki = 6 nM T84631 CBLZ18 44372833 Ki = 1.1 nM T84631 CFH41R 44372839 Ki = 2000 nM T84631 C9COY7 44372840 Ki > 1000000 nM T84631 C34AWY 44372863 Ki = 140000 nM T84631 CZE15A 44372864 Ki = 28000 nM T84631 C7X5BE 44372865 Ki = 2000 nM T84631 C2E6TP 44372889 Ki = 28000 nM T84631 CNOV-41 44372899 Ki = 0.3 nM T84631 C36XWM 44372903 Ki = 410 nM T84631 C01VKC 44374066 Ki = 0.8 nM T84631 C3MX0H 44374677 Ki = 2.3 nM T84631 C4HSA0 44374690 Ki = 1.8 nM T84631 C2Y0SC 44375908 IC50 = 24000 nM T84631 C3C2XE 44375967 IC50 = 69 nM T84631 C69QAS 44375986 IC50 = 2 nM T84631 C34XTM 44375987 Ki = 0.013 nM T84631 CZVP71 44376028 IC50 = 1 nM T84631 CZA1N6 44376029 IC50 = 0.7 nM T84631 C58WMI 44376046 IC50 = 3 nM T84631 C74KVW 44376051 IC50 = 17 nM T84631 C6SC3T 44376056 IC50 = 771 nM T84631 C2NHP9 44376074 IC50 = 2 nM T84631 CE9N6S 44376077 IC50 = 21 nM T84631 C6QTS8 44376079 IC50 = 8 nM T84631 CEKQ15 44376084 IC50 = 0.62 nM T84631 C9T2QI 44376089 IC50 = 3 nM T84631 CD0W7C 44376100 IC50 = 2 nM T84631 CG78SI 44376101 IC50 = 320 nM T84631 CG9KH1 44376121 IC50 = 118 nM T84631 C23ZRU 44376219 IC50 = 510 nM T84631 C5PH2E 44376249 IC50 = 58 nM T84631 C0Y8QD 44376252 IC50 = 0.79 nM T84631 CD03ZI 44376253 IC50 = 38 nM T84631 CX98EC 44376254 IC50 = 85 nM T84631 C1F2JZ 44376255 IC50 = 116 nM T84631 C0MS6T 44376257 IC50 = 2 nM T84631 C7BS3N 44376258 IC50 = 13 nM T84631 C63JEF 44376259 IC50 = 0.9 nM T84631 C0Z9CS 44376264 IC50 = 1 nM T84631 CSRZ57 44376273 IC50 = 10 nM T84631 CCY74M 44376286 IC50 = 6 nM T84631 CP9IY1 44376287 IC50 = 6 nM T84631 C0S9XG 44376288 IC50 = 10 nM T84631 COX13N 44376289 IC50 = 1 nM T84631 CNC7F4 44376290 IC50 = 32 nM T84631 C6X7UG 44376311 IC50 = 0.89 nM T84631 C4TGW5 44376318 IC50 = 4 nM T84631 C28ZIJ 44376322 IC50 = 37 nM T84631 C51GPZ 44376323 IC50 = 154 nM T84631 C5Y6JB 44376326 IC50 = 1 nM T84631 CA59MK 44376327 IC50 = 5 nM T84631 C5R2PM 44376328 Ki = 0.17 nM T84631 CTZR83 44376339 Ki = 800 nM T84631 CDM65F 44376342 IC50 = 4 nM T84631 C6R5AG 44376343 IC50 = 2 nM T84631 C8M2PZ 44376385 IC50 = 65 nM T84631 CH95MO 44376405 Ki = 33900 nM T84631 CB87VR 44376416 IC50 = 2 nM T84631 C5VDG0 44376417 IC50 = 2 nM T84631 C1S5KV 44376423 IC50 = 29 nM T84631 CG64YQ 44376426 Ki = 1.4 nM T84631 COAE61 44376427 IC50 = 5 nM T84631 CXEG05 44376429 IC50 = 459 nM T84631 CP7CO4 44376432 IC50 = 144 nM T84631 CKI3R7 44376454 Ki = 300 nM T84631 CT8KB1 44376468 IC50 = 22000 nM T84631 CI03DP 44376475 IC50 = 3 nM T84631 CUVH30 44376476 IC50 = 4 nM T84631 CSW71I 44376504 Ki = 850 nM T84631 C7WTQ1 44376505 Ki = 7800 nM T84631 C9SW1H 44376514 IC50 = 11 nM T84631 CM75ZP 44376515 IC50 = 31 nM T84631 C51GQP 44376523 Ki = 910 nM T84631 CA7GW4 44376525 Ki = 500 nM T84631 CHW87S 44376544 IC50 = 7 nM T84631 CKHG50 44376548 Ki = 2300 nM T84631 CZ68PY 44376566 Ki = 2500 nM T84631 C3DLJ9 44376572 IC50 = 32 nM T84631 C41SQG 44376585 Ki = 10500 nM T84631 C1PK0O 44376651 Ki = 16 nM T84631 CXG42V 44376671 Ki = 6600 nM T84631 CJBO94 44376700 IC50 = 21 nM T84631 C3K7NA 44376701 IC50 = 3 nM T84631 CKSV26 44376702 IC50 = 13 nM T84631 CXZP98 44376712 Ki = 282 nM T84631 CUFO93 44376713 Ki = 120 nM T84631 C1Z3BF 44376731 IC50 = 11 nM T84631 CEKG07 44376754 Ki = 30 nM T84631 CQX98K 44376755 Ki = 28 nM T84631 C2JKH1 44376756 Ki = 42 nM T84631 CITM85 44376766 Ki = 25700 nM T84631 CV7I3K 44376788 Ki = 500 nM T84631 CV5J1M 44376828 Ki = 38000 nM T84631 C8P5YZ 44376949 IC50 = 6 nM T84631 C4XJD0 44377015 IC50 = 888 nM T84631 CQB2G9 44377016 IC50 = 370 nM T84631 C6QG0C 44377053 Ki = 100 nM T84631 C6A7VL 44377057 Ki = 145 nM T84631 CZ6W0S 44377280 Ki > 338 nM T84631 CVS76R 44377281 Ki = 49.2 nM T84631 CI2GS0 44377287 IC50 = 0.94 nM T84631 CKX32Z 44377301 Ki > 338 nM T84631 C7W2GD 44377304 IC50 = 1.08 nM T84631 C6RA4Q 44377310 Ki > 338 nM T84631 CG0S9N 44377311 Ki = 52.7 nM T84631 CP0V6X 44377320 IC50 = 2.2 nM T84631 C4KSG5 44377322 IC50 = 0.9 nM T84631 CH1NM4 44377327 Ki = 23 nM T84631 CTP28F 44377331 IC50 = 1.1 nM T84631 CN42TW 44377336 Ki > 338 nM T84631 CPE23W 44377369 Ki > 338 nM T84631 C30VGP 44377425 IC50 = 0.9 nM T84631 C39PST 44377471 Ki = 93 nM T84631 C5Q1LA 44377475 Ki > 338 nM T84631 CVHL28 44377478 Ki = 40 nM T84631 CT0G2D 44377544 Ki = 16 nM T84631 CK6I3F 44377546 IC50 = 2.6 nM T84631 CNUL43 44377548 IC50 = 4.3 nM T84631 CZBJ51 44377550 IC50 = 5.3 nM T84631 CHU5T4 44377558 IC50 = 2.1 nM T84631 CU49MW 44377570 Ki > 338 nM T84631 C1TVZ9 44377573 Ki > 338 nM T84631 C3LE7S 44377608 Ki > 338 nM T84631 C7Y4QI 44377622 Ki = 315 nM T84631 CXLT41 44377644 Ki > 338 nM T84631 CO7N6Y 44378546 Ki = 57600 nM T84631 CLXH02 44378887 Ki = 111000 nM T84631 CC4MP1 44380667 Ki > 6000 nM T84631 C5XC2T 44381273 Ki = 17000 nM T84631 CJ6M5B 44382389 IC50 = 2500 nM T84631 CTF4N6 44382391 IC50 = 2500 nM T84631 CAI65F 44382441 IC50 > 2500 nM T84631 CB5J9R 44383041 Ki >> 1200 nM T84631 C6LH5V 44383081 IC50 = 2500 nM T84631 C9SD3E 44383242 Ki = 10 nM T84631 CFN18Q 44383278 Ki >> 1200 nM T84631 C2Y8NB 44383311 Ki = 40 nM T84631 C2NG7K 44383318 Ki >> 1200 nM T84631 CL5D3K 44383321 Ki = 120 nM T84631 CTNC21 44383351 Ki > 1200 nM T84631 C5PW9E 44383425 IC50 > 2500 nM T84631 CLQ19H 44383460 Ki = 1200 nM T84631 C43KTU 44383519 Ki = 24 nM T84631 CNBG48 44383542 IC50 > 2500 nM T84631 C2IX5U 44383543 IC50 = 2360 nM T84631 C4YS2W 44383629 Ki = 390 nM T84631 CX8CZ4 44383764 Ki = 1200 nM T84631 CKOW56 44383765 Ki >> 1200 nM T84631 CJH1T9 44383975 Ki >> 1200 nM T84631 CL5HW0 44383976 Ki >> 1200 nM T84631 C5CF2Z 44383985 Ki = 1200 nM T84631 CG8V5P 44384040 Ki = 290 nM T84631 CTLY83 44384041 Ki = 17 nM T84631 CS0IP4 44384198 Ki = 0.8 nM T84631 C6IX3V 44384674 Ki = 30 nM T84631 CP74XU 44384744 Ki = 80 nM T84631 CGI1H8 44384745 Ki = 370 nM T84631 CHK87Y 44384746 Ki = 0.46 nM T84631 CR2VG0 44384747 Ki = 0.3 nM T84631 CUR5K2 44384798 Ki = 3.6 nM T84631 CQ1D0K 44384799 Ki = 5.9 nM T84631 CVYI62 44385066 Ki = 1.3 nM T84631 CJ01YE 44385090 Ki = 20 nM T84631 CV4N1P 44385091 Ki = 3.5 nM T84631 C1ZV8A 44385092 Ki = 0.6 nM T84631 COQ8S6 44385134 Ki = 22 nM T84631 CVGJ91 44385135 Ki = 417 nM T84631 CLWT03 44385136 Ki = 300 nM T84631 CT42KF 44385150 Ki = 3 nM T84631 CALR98 44385151 Ki = 1.1 nM T84631 CNH87R 44385152 Ki = 420 nM T84631 C43MAX 44385153 Ki = 300 nM T84631 CDT45B 44385195 Ki = 0.23 nM T84631 C7U0HZ 44385205 Ki = 4.6 nM T84631 CTX13E 44385259 Ki = 1050 nM T84631 CI91SG 44385260 Ki = 6 nM T84631 C4RV6U 44385263 Ki = 5 nM T84631 CNMA50 44385268 Ki = 370 nM T84631 C3DF2V 44385269 Ki = 80 nM T84631 C9Z1OC 44385301 Ki = 0.12 nM T84631 CHPL94 44385310 Ki = 840 nM T84631 C6VZ5Y 44385361 Ki = 340 nM T84631 CCR46P 44385364 Ki = 6.3 nM T84631 CPV5B7 44385418 Ki = 190 nM T84631 C8CE6A 44385432 Ki = 160 nM T84631 C56GNK 44385447 Ki = 0.8 nM T84631 CR47ZA 44385448 IC50 = 32 nM T84631 CG35IX 44385449 Ki = 1.8 nM T84631 C1QOM8 44385484 IC50 = 1.3 nM T84631 CG7LT1 44385488 IC50 = 53 nM T84631 C7B5NP 44385500 Ki = 0.1 nM T84631 C94GZU 44385541 IC50 = 76 nM T84631 CQ7G9I 44385552 Ki = 0.1 nM T84631 CUQ30E 44385556 IC50 = 23 nM T84631 CH0EJ5 44385561 Ki = 0.9 nM T84631 CZ9KO4 44385566 IC50 = 16 nM T84631 C3T9XK 44385607 IC50 = 6.3 nM T84631 CKY0P4 44385611 IC50 = 3.8 nM T84631 C8MF3J 44385614 IC50 = 39 nM T84631 CUS20V 44385673 IC50 = 40 nM T84631 CZ8XL6 44385679 Ki = 0.5 nM T84631 CL5BA4 44385729 Ki = 0.3 nM T84631 CQ1CH4 44385753 Ki = 0.7 nM T84631 C3DSN7 44385768 IC50 = 30 nM T84631 C8USN9 44385769 IC50 = 552 nM T84631 C2E8DS 44385771 IC50 = 10 nM T84631 C2VFC6 44385772 IC50 = 1.5 nM T84631 CN8V0W 44385779 IC50 = 2 nM T84631 CO2K6D 44385783 IC50 = 2.8 nM T84631 CIHV71 44385786 Ki = 2.8 nM T84631 CPOS98 44385789 Ki = 4.5 nM T84631 C2WYO3 44385799 Ki = 2.9 nM T84631 CJ5B9H 44385803 Ki = 30 nM T84631 C7ZNB9 44385807 IC50 = 66 nM T84631 CBEA65 44385842 IC50 = 0.8 nM T84631 CN5Q1G 44385864 Ki = 2 nM T84631 C4XY8T 44385865 Ki = 60 nM T84631 CC9M7E 44385869 IC50 = 136 nM T84631 C8WK4A 44385891 IC50 = 1.1 nM T84631 C3VSU7 44385892 IC50 = 1.8 nM T84631 C8T1ZD 44385893 Ki = 0.012 nM T84631 CY81KI 44385894 IC50 = 7 nM T84631 C42JCS 44385915 Ki = 2 nM T84631 C9F6LP 44385922 IC50 = 9.5 nM T84631 C37ZQR 44385924 Ki = 1.8 nM T84631 C3D2CL 44385935 Ki = 1.3 nM T84631 CUAY63 44385953 Ki = 1 nM T84631 CX1C3I 44385963 Ki = 3.3 nM T84631 CFPH43 44385967 Ki = 4 nM T84631 CW08OY 44385998 Ki = 0.2 nM T84631 CV6KG4 44386059 Ki = 0.1 nM T84631 CWR4Q6 44386101 Ki = 6.2 nM T84631 CJ48AC 44386102 Ki = 1 nM T84631 CV13WD 44386116 Ki = 0.3 nM T84631 CGU69V 44386179 IC50 = 6.9 nM T84631 CS65LH 44386185 IC50 = 230 nM T84631 CU0P5T 44386242 IC50 = 6.8 nM T84631 CU9J0D 44386250 IC50 = 171 nM T84631 C7NF2L 44386266 IC50 = 60 nM T84631 C0Z3LF 44386268 IC50 = 22 nM T84631 C9G7QW 44386322 IC50 = 156 nM T84631 C31CUG 44386326 IC50 = 11 nM T84631 CX58AM 44386358 Ki = 0.23 nM T84631 C2WCE4 44386371 IC50 = 176 nM T84631 CDR14L 44386384 IC50 = 3.5 nM T84631 C52POK 44386417 IC50 = 12 nM T84631 CRX1I9 44386418 IC50 = 35 nM T84631 CI23WQ 44386419 Ki = 0.2 nM T84631 CFQV46 44386424 IC50 = 74 nM T84631 CIBD76 44386484 IC50 = 82 nM T84631 C8ME4O 44386493 IC50 = 5.8 nM T84631 CD4AH3 44386540 IC50 = 2.3 nM T84631 CHAO48 44386542 IC50 = 15 nM T84631 C2D6XI 44386633 IC50 = 4.1 nM T84631 CLNO15 44386637 IC50 = 35 nM T84631 C81IMH 44386642 IC50 = 40 nM T84631 C8SYK9 44386783 Ki = 210000 nM T84631 C4JB0M 44386841 IC50 = 1.3 nM T84631 CJC27L 44386868 IC50 = 5.3 nM T84631 C5FI9N 44386929 IC50 = 2.8 nM T84631 C5MR1F 44386934 Ki = 0.6 nM T84631 C8K5HM 44387041 IC50 = 2.3 nM T84631 CA45DZ 44387044 IC50 = 3.6 nM T84631 C7IG6P 44387096 IC50 = 4.1 nM T84631 C07CMU 44387102 IC50 = 1.9 nM T84631 C39LUW 44387104 IC50 = 5 nM T84631 CK0A4V 44387120 Ki = 1 nM T84631 CJ9ED7 44387165 Ki = 0.2 nM T84631 C2QD1K 44387206 IC50 = 1.4 nM T84631 C6SV1C 44387258 IC50 = 38000 nM T84631 CN2GR5 44390800 Ki = 12400 nM T84631 CW3G5V 44390801 Ki = 19000 nM T84631 CESM50 44392171 Ki = 270 nM T84631 CRYN03 44392172 Ki = 300 nM T84631 C9FUI3 44392182 Ki > 180 nM T84631 CT1AO2 44392186 Ki = 90 nM T84631 CG8V4B 44392189 Ki > 9000 nM T84631 CVK58T 44392197 Ki = 130 nM T84631 C4CU6F 44392199 Ki = 65 nM T84631 C1K6IY 44392201 Ki > 9000 nM T84631 CKO0E4 44392205 Ki = 530 nM T84631 CAE80C 44392206 Ki = 270 nM T84631 CJC84M 44392224 Ki > 9000 nM T84631 CP1CF2 44392233 Ki = 200 nM T84631 CHQG45 44392249 Ki = 19 nM T84631 C45EDM 44392250 Ki = 120 nM T84631 CLM10G 44393633 IC50 = 300 nM T84631 COS35W 44393635 IC50 = 2000 nM T84631 C54IJH 44393646 IC50 = 30 nM T84631 C4J5YZ 44393648 IC50 = 30 nM T84631 C7F1EZ 44393650 IC50 = 200 nM T84631 CM15TG 44393671 IC50 = 200 nM T84631 CW2B4G 44393673 IC50 = 200 nM T84631 CAYT14 44393675 IC50 = 6 nM T84631 CI7OZ9 44393679 IC50 = 100 nM T84631 CO3B6P 44393688 IC50 = 400 nM T84631 C5BWQ3 44393690 IC50 = 100 nM T84631 CW7T2D 44393692 IC50 = 60 nM T84631 CD0O9Q 44393694 IC50 = 100 nM T84631 CU47SD 44393720 IC50 = 3000 nM T84631 C2Q6CA 44393722 IC50 = 40 nM T84631 C95LDV 44393724 IC50 = 300 nM T84631 CUFO09 44395404 Ki = 0.19 nM T84631 CJ45KG 44395699 IC50 = 11000 nM T84631 CN04TX 44395725 IC50 = 26000 nM T84631 CN7Y2C 44395728 IC50 = 12000 nM T84631 C81TGP 44395751 IC50 = 29000 nM T84631 CS7UY1 44395771 IC50 = 29000 nM T84631 COD05Q 44395835 IC50 = 13000 nM T84631 CA0ZU3 44395871 IC50 = 10000 nM T84631 C1G7ZQ 44395885 IC50 = 14000 nM T84631 CIB17E 44395901 IC50 = 22000 nM T84631 C4SUD5 44396124 IC50 = 59000 nM T84631 CCL3J1 44396183 IC50 = 12000 nM T84631 CEC5X2 44396195 IC50 = 20000 nM T84631 C9P1FN 44398617 Ki = 25 nM T84631 CD5SQ2 44398699 Ki = 3 nM T84631 CQH41I 44398720 Ki = 0.1 nM T84631 CE5S0J 44400525 IC50 = 1130 nM T84631 CB0N5T 44400527 Ki = 19 nM T84631 CH9TP3 44402039 Ki = 512 nM T84631 C49CME 44402191 Ki = 137 nM T84631 CL80DH 44402364 Ki = 417 nM T84631 CQ4J2A 44402383 Ki = 264 nM T84631 C8WR3I 44402428 Ki = 111 nM T84631 CJQ8X6 44402429 Ki = 104 nM T84631 C6CZ8H 44402442 Ki = 136 nM T84631 CPLF17 44402521 Ki = 442 nM T84631 C5JK1T 44402528 Ki = 731 nM T84631 C9CWT3 44402591 Ki = 40 nM T84631 CV0S6N 44402617 Ki = 632 nM T84631 C0EWM8 44402974 IC50 < 10000 nM T84631 CD16XV 44402976 IC50 = 51000 nM T84631 C90VXC 44402978 IC50 = 4800 nM T84631 CPLH23 44402980 IC50 = 29000 nM T84631 C3T9OL 44402982 IC50 = 3300 nM T84631 C0Z2RO 44402984 IC50 = 11000 nM T84631 C27KPR 44402986 IC50 = 4500 nM T84631 CX90NG 44402988 IC50 = 9600 nM T84631 CQT09E 44402990 IC50 = 8000 nM T84631 C3P2QU 44402994 IC50 = 11000 nM T84631 C9E6KX 44402996 IC50 = 12000 nM T84631 C7QC1J 44402998 IC50 = 26000 nM T84631 C59QOU 44403000 IC50 = 17000 nM T84631 CF4IG0 44403002 IC50 = 11000 nM T84631 COW8T1 44403004 IC50 = 17000 nM T84631 CPU19J 44403006 IC50 = 4100 nM T84631 CW3HV4 44403010 IC50 = 4300 nM T84631 CFI1B8 44403012 IC50 = 20000 nM T84631 C61JGY 44403016 IC50 = 59000 nM T84631 C7L6YO 44403018 IC50 = 5700 nM T84631 C8PE3F 44403020 IC50 = 13000 nM T84631 C7IP1V 44403898 IC50 = 120 nM T84631 CG5V0X 44403903 IC50 = 20 nM T84631 C4F8BL 44404188 Ki = 14 nM T84631 CB6JW0 44407541 Ki = 6 nM T84631 CZD4O6 44407546 Ki = 3 nM T84631 CJ7W6K 44407547 Ki = 3 nM T84631 C1G4BC 44407625 Ki = 46 nM T84631 CA6Q9U 44407762 Ki = 140 nM T84631 CK54BG 44407769 Ki = 80 nM T84631 CC9Z0M 44407770 Ki = 2 nM T84631 C8J5OE 44407777 Ki = 40 nM T84631 CP67EA 44411094 IC50 = 251 nM T84631 CM8OZ0 44411137 IC50 > 45000 nM T84631 C3BX5Y 44412781 Ki > 150000 nM T84631 CF5XO4 44413343 Ki = 3700 nM T84631 CTD42X 44413355 Ki = 1100 nM T84631 C9KQM2 44413356 Ki = 1300 nM T84631 CQDX92 44413619 Ki = 4600 nM T84631 C9S8YL 44413733 Ki = 13 nM T84631 CO8A0Y 44414333 Ki = 100000 nM T84631 CG6H0U 44415561 Ki = 30000 nM T84631 C3LCV6 44415581 Ki = 54000 nM T84631 CJ20PN 44416510 IC50 > 200000 nM T84631 CZK3N4 44416547 IC50 = 175400 nM T84631 CQA4B5 44416549 IC50 = 129000 nM T84631 CMVF02 44416571 IC50 = 43600 nM T84631 C3TJK6 44418750 IC50 = 14200 nM T84631 C9G1VL 44418752 IC50 = 14300 nM T84631 CHK10G 44418753 IC50 = 15400 nM T84631 C9OZ1M 44418754 IC50 > 20000 nM T84631 CRM0E4 44419084 IC50 = 2 nM T84631 C8LV0Y 44419092 IC50 < 0.5 nM T84631 CQ7PD9 44419104 IC50 = 0.7 nM T84631 CID32E 44419109 IC50 = 2 nM T84631 C54KZH 44419113 IC50 = 0.9 nM T84631 C18PXN 44419484 Ki = 0.04 nM T84631 CVJ85S 44421826 IC50 > 200000 nM T84631 CWVX31 44421837 IC50 > 200000 nM T84631 CD58ZY 44421845 IC50 > 200000 nM T84631 C48NZW 44426214 Ki = 0.32 nM T84631 COUZ56 44426215 Ki = 21 nM T84631 C3F2PN 44426216 Ki = 3900 nM T84631 CZ91LH 44426217 Ki = 3.3 nM T84631 CEV53U 44426218 Ki = 2.55 nM T84631 C8O6HV 44426219 Ki = 0.095 nM T84631 CJH6E4 44426220 Ki = 32 nM T84631 C3E2FT 44426221 Ki = 53 nM T84631 CW3G0D 44426222 Ki = 52 nM T84631 CN6VL5 44426224 Ki = 0.35 nM T84631 CG9XF0 44426226 Ki = 0.36 nM T84631 CQ7CF9 44426227 Ki = 3.4 nM T84631 CL4N6J 44426228 Ki = 0.76 nM T84631 CJ3B7D 44426229 Ki = 1.6 nM T84631 C5Q8HB 44426230 Ki = 4.9 nM T84631 C6RNO7 44426232 Ki = 4.9 nM T84631 CCGR09 44426234 Ki = 200 nM T84631 CD06OJ 44426235 Ki = 65 nM T84631 CR4D0U 44426236 Ki = 16 nM T84631 CIT7D5 44426237 Ki = 0.084 nM T84631 CW71LJ 44426238 Ki = 0.25 nM T84631 CY5Z6P 44426239 Ki = 0.059 nM T84631 CI0N7E 44426240 Ki = 0.24 nM T84631 C35VBM 44426241 Ki = 0.52 nM T84631 C0LIG6 44426243 Ki = 0.049 nM T84631 C9V2JR 44426244 Ki = 0.08 nM T84631 C72TBW 44426245 Ki = 0.87 nM T84631 CZ2GS7 44426246 Ki = 0.63 nM T84631 CPKM97 44426247 Ki = 1.7 nM T84631 C1MVS4 44426248 Ki = 0.92 nM T84631 C5W1RJ 44426249 Ki = 1 nM T84631 C8H5OR 44426250 Ki = 0.94 nM T84631 C8BE9L 44426251 Ki = 2.9 nM T84631 CT6C5J 44426252 Ki = 1.5 nM T84631 CCN6T9 44426253 Ki = 17 nM T84631 C1UYG6 44426254 Ki = 8.3 nM T84631 CGV1I0 44426657 IC50 = 40 nM T84631 CXI16J 44426658 IC50 = 50 nM T84631 CZ9O0J 44426660 IC50 > 30000 nM T84631 CJN3M1 44426799 IC50 > 30000 nM T84631 CO9Q4B 44427316 IC50 > 30000 nM T84631 CD9O6E 44427319 IC50 > 30000 nM T84631 C53IBP 44428362 Ki = 2.2 nM T84631 CI6QX0 44429068 IC50 = 90 nM T84631 CED2A3 44429069 IC50 > 100000 nM T84631 CG9DX2 44429071 IC50 > 100000 nM T84631 C58ODU 44429073 IC50 = 850 nM T84631 C9QB7L 44429075 IC50 = 950 nM T84631 CEP2S5 44429076 IC50 = 350 nM T84631 CP7AD2 44429077 IC50 = 250 nM T84631 CEQ2U3 44429078 IC50 = 49 nM T84631 C0OH9V 44429079 IC50 > 100000 nM T84631 CHE96M 44429080 IC50 = 1600 nM T84631 CNZF48 44429082 IC50 = 800 nM T84631 C1EGK3 44429083 IC50 = 170 nM T84631 CA6U4B 44429085 IC50 = 200 nM T84631 C4E3TU 44429087 IC50 = 1700 nM T84631 CRJ2G1 44429088 IC50 = 2300 nM T84631 CPT8U9 44429090 IC50 > 100000 nM T84631 CGHK29 44429092 IC50 > 100000 nM T84631 C2G5ZK 44429093 IC50 > 100000 nM T84631 CMWU43 44429094 IC50 = 560 nM T84631 CG7MW6 44429096 IC50 = 190 nM T84631 CS29AL 44429097 IC50 = 65 nM T84631 CWA2F9 44429098 IC50 = 100 nM T84631 CTUO84 44429099 IC50 = 39 nM T84631 CQS80V 44429101 IC50 = 58 nM T84631 C1Q0EO 44429102 IC50 = 11 nM T84631 CV7A9L 44429104 IC50 = 12 nM T84631 CL32QO 44429105 IC50 = 590 nM T84631 CB27IK 44429106 IC50 = 13 nM T84631 CH6Z7Y 44429108 IC50 = 8.1 nM T84631 C8IHX6 44429109 IC50 = 10 nM T84631 CO78JZ 44429110 IC50 = 13 nM T84631 C0PE1M 44432470 Ki = 1.7 nM T84631 CPER15 44432471 Ki = 3.2 nM T84631 CJO6Z9 44432472 Ki = 2.1 nM T84631 C3O9RC 44432473 Ki = 2.5 nM T84631 C4BSJ6 44432474 Ki = 10 nM T84631 C0D6SL 44432475 Ki = 1.3 nM T84631 CP2LI4 44432476 Ki = 3.9 nM T84631 CBAV03 44432477 Ki = 4.8 nM T84631 CN4QV7 44432489 Ki = 1 nM T84631 CE8NY0 44432490 Ki = 7.3 nM T84631 CZ20YU 44432491 Ki = 23 nM T84631 C3DK8P 44432494 Ki = 266 nM T84631 C5D3TL 44432495 Ki = 288 nM T84631 CF9Q5N 44432496 Ki = 27 nM T84631 CIH6B5 44432497 Ki = 36 nM T84631 CP84FK 44432498 Ki = 1220 nM T84631 C3YOB9 44432499 Ki = 7.92 nM T84631 CF8G5U 44432501 Ki = 170 nM T84631 C7BP9C 44432503 Ki = 124 nM T84631 CJ59VG 44432505 Ki = 1186 nM T84631 C8AJS7 44432506 Ki = 2610 nM T84631 C2M7XN 44432507 Ki = 138 nM T84631 C1YZ9P 44432508 Ki = 892 nM T84631 C14LPX 44432509 Ki = 226 nM T84631 C68JTP 44432510 Ki = 433 nM T84631 C8VC2O 44432511 Ki = 129 nM T84631 CAJ8R2 44432512 Ki = 360 nM T84631 CW0KC9 44432514 Ki = 603 nM T84631 C5LA6U 44432515 Ki = 7420 nM T84631 C2D5US 44432516 Ki = 8560 nM T84631 C05QPV 44432517 Ki = 14 nM T84631 CVX41Y 44432522 Ki = 37 nM T84631 C0BU8P 44432527 Ki = 0.94 nM T84631 C65WMJ 44432528 Ki = 4 nM T84631 CHC7Y5 44432529 Ki = 107 nM T84631 CO9E0L 44432534 Ki = 2.4 nM T84631 CXEL19 44432536 Ki = 0.44 nM T84631 CVO5Q1 44432538 Ki = 0.51 nM T84631 CMX28G 44432539 Ki = 0.95 nM T84631 CRO15T 44432542 Ki = 10 nM T84631 CEIG96 44432570 Ki = 82 nM T84631 C7L4YU 44432571 Ki = 11500 nM T84631 C4TO1Y 44432573 Ki = 4.2 nM T84631 CZ5WC2 44432574 Ki = 929 nM T84631 C0KJ7B 44432576 Ki = 1.3 nM T84631 CMP70C 44432577 Ki = 0.71 nM T84631 C4NWL3 44434801 Ki = 0.21 nM T84631 C90KHC 44434802 Ki = 0.84 nM T84631 CDI09P 44434803 Ki = 27 nM T84631 CYKG20 44434804 Ki = 7.9 nM T84631 CAB7R9 44434805 Ki = 10870 nM T84631 CHZ0U3 44434806 Ki = 1 nM T84631 CS6ZY1 44434807 Ki = 0.27 nM T84631 CR16BF 44434808 Ki = 0.56 nM T84631 CQIX73 44434809 Ki = 1.9 nM T84631 CFLI30 44434810 Ki = 2.1 nM T84631 C1GZT7 44434811 Ki = 1.6 nM T84631 C2TK5Q 44434812 Ki = 1.6 nM T84631 CM3T0U 44434813 Ki = 0.39 nM T84631 C4HL3O 44434814 Ki = 3 nM T84631 C5R8HJ 44434815 Ki = 2.6 nM T84631 CPA5X7 44434816 Ki = 2.6 nM T84631 C7FJR9 44434817 Ki = 18 nM T84631 COG34X 44434818 Ki = 0.58 nM T84631 CRW87S 44434819 Ki = 3.9 nM T84631 CZ27MI 44434820 Ki = 2.8 nM T84631 CAZ59V 44434822 Ki = 2 nM T84631 C27VMW 44434824 Ki = 1.3 nM T84631 C51RUQ 44434825 Ki = 1.7 nM T84631 CH2L5P 44434826 Ki = 2.1 nM T84631 C9JD8H 44434829 Ki = 2.2 nM T84631 CYHV92 44434830 Ki = 0.36 nM T84631 CT6XL4 44434831 Ki = 0.74 nM T84631 CWA82Q 44434833 Ki = 0.93 nM T84631 C7PF0V 44434834 Ki = 0.44 nM T84631 C9T1DP 44434835 Ki = 0.64 nM T84631 CE3R5S 44434836 Ki = 1.7 nM T84631 C2OCL7 44434838 Ki = 1.7 nM T84631 CY0Z4T 44434840 Ki = 0.56 nM T84631 C4ADI5 44435823 Ki = 2.3 nM T84631 C30CFX 44436704 IC50 > 10000 nM T84631 CLU2J3 44441275 IC50 = 270 nM T84631 CJ67AP 44441276 IC50 > 10000 nM T84631 CKJ61O 44441277 IC50 = 3200 nM T84631 C53IBS 44441278 IC50 > 10000 nM T84631 C5DKP6 44441279 IC50 = 4400 nM T84631 CBV16E 44441280 IC50 > 10000 nM T84631 C97RGS 44441281 IC50 > 10000 nM T84631 C1N8RW 44441282 IC50 = 265 nM T84631 C2ZO6L 44441283 IC50 = 2000 nM T84631 CHB06C 44441284 IC50 = 118 nM T84631 C8WL7U 44441285 IC50 = 86 nM T84631 C3BPD0 44441286 IC50 = 175 nM T84631 CVIO95 44441287 IC50 = 11.3 nM T84631 C0D1CR 44441288 IC50 > 1400 nM T84631 CIK8L7 44441289 IC50 > 10000 nM T84631 CB49OX 44441290 IC50 = 753 nM T84631 CS90XV 44443528 IC50 = 1100 nM T84631 C0IPW3 44443531 IC50 = 150 nM T84631 CV5CK0 44443532 IC50 = 18 nM T84631 CFW4B7 44443548 IC50 = 436 nM T84631 CD1WV5 44443552 IC50 = 70 nM T84631 C20ZPQ 44443557 IC50 = 61 nM T84631 CL7O4R 44443558 IC50 = 130 nM T84631 CL68HN 44443560 IC50 = 40 nM T84631 CW31AS 44443863 Ki = 4 nM T84631 CZTC23 44444412 Ki = 1400 nM T84631 CT0K6W 44444413 Ki = 0.82 nM T84631 C2GQ4X 44444414 Ki = 19 nM T84631 CG3IT9 44444415 Ki = 1 nM T84631 CN7U2V 44444416 Ki = 0.63 nM T84631 C5DHI1 44444417 Ki = 1400 nM T84631 C50JGC 44444418 Ki = 2.2 nM T84631 C5TG0M 44446364 Ki = 1.1 nM T84631 CX02SN 44446365 Ki = 0.7 nM T84631 CUN0M5 44446366 Ki = 8.9 nM T84631 C0NB1S 44446367 Ki = 2.7 nM T84631 CGC4U3 44446368 Ki = 4.4 nM T84631 CEQ3K7 44446375 Ki = 6.3 nM T84631 C90HMC 44446376 Ki = 15.5 nM T84631 C14UGA 44446377 Ki = 74.6 nM T84631 CDJH35 44446378 Ki = 215 nM T84631 CZ07YI 44446379 Ki = 80 nM T84631 C2H1ZM 44446380 Ki = 0.2 nM T84631 CS59RX 44446381 Ki = 0.1 nM T84631 CUT3E2 44446382 Ki = 2 nM T84631 CVQ2A5 44446383 Ki = 1.1 nM T84631 CQYA21 44446384 Ki = 6.2 nM T84631 CLX79F 44446385 Ki < 0.4 nM T84631 C63ALD 44446386 Ki < 0.3 nM T84631 C15NOL 44446387 Ki = 14 nM T84631 CHV7B9 44446388 Ki = 0.4 nM T84631 C1K3BV 44446389 Ki = 1.8 nM T84631 CZA52B 44446390 Ki = 11.8 nM T84631 C7AJ3M 44446391 Ki = 6 nM T84631 C7X4ZE 44446392 Ki = 9.1 nM T84631 CPB7H6 44446393 Ki = 180 nM T84631 C78RKU 44446394 Ki = 2334 nM T84631 CN8SC7 44446622 Ki = 1.5 nM T84631 CXT60W 44446625 Ki = 0.68 nM T84631 C8PW5C 44446626 Ki = 0.53 nM T84631 C2OX0A 44446627 Ki = 0.07 nM T84631 CGE82I 44446629 Ki = 0.16 nM T84631 CKJV95 44446630 Ki = 4.7 nM T84631 C4RVO9 44446632 Ki = 22 nM T84631 C4WFK6 44446634 Ki = 2.8 nM T84631 C1HOX5 44446638 Ki = 2.3 nM T84631 C5WH9G 44446642 Ki = 0.97 nM T84631 C47NBK 44446644 Ki = 0.57 nM T84631 CU3YD7 44446648 Ki = 0.32 nM T84631 CC9LB6 44446651 Ki = 0.34 nM T84631 CSR9L5 44446652 Ki = 12 nM T84631 CH27CY 44446654 Ki = 6.9 nM T84631 CNX71T 44446656 Ki = 3.3 nM T84631 C8T7LJ 44446659 Ki = 1 nM T84631 CVQN67 44449252 Ki = 0.14 nM T84631 CS0M1X 44449283 Ki = 0.45 nM T84631 C0ER8M 44449284 Ki = 2 nM T84631 CO06UN 44449312 Ki = 0.14 nM T84631 CH2KY6 44449344 Ki = 2.2 nM T84631 CM7Z2Y 44449346 Ki = 7670 nM T84631 CI19PT 44449347 Ki = 0.12 nM T84631 CO8DL4 44449376 Ki = 1.1 nM T84631 CTY1O5 44449377 Ki = 59 nM T84631 CX7VI4 44449404 Ki = 0.62 nM T84631 CM79OK 44449405 Ki = 0.21 nM T84631 CBT6Y9 44449406 Ki = 4.2 nM T84631 CW0K7B 44449442 Ki = 1560 nM T84631 CVQA35 44449443 Ki = 0.14 nM T84631 CT1EI5 44449445 Ki = 0.58 nM T84631 C5Y9CT 44449469 Ki = 43 nM T84631 C0JD6K 44449470 Ki = 1 nM T84631 CP23WS 44449471 Ki = 3 nM T84631 CQ0P1T 44449498 Ki = 1.2 nM T84631 CEN98O 44449697 Ki = 0.005 nM T84631 CLNS10 44449700 Ki = 0.24 nM T84631 C1ATS9 44449734 Ki = 0.065 nM T84631 C8IC1F 44449735 Ki = 0.047 nM T84631 C0Y6AD 44450537 IC50 = 12 nM T84631 C15UNI 44450551 IC50 = 35 nM T84631 CY6WC9 44450552 IC50 = 24 nM T84631 C04NRS 44450553 IC50 = 21 nM T84631 CV0LM3 44450559 IC50 = 29 nM T84631 CFWS94 44450560 IC50 = 24 nM T84631 CTU6D5 44450561 IC50 = 78 nM T84631 CF8KZ6 44450562 IC50 = 840 nM T84631 C6LQ5H 44450623 IC50 = 18 nM T84631 C6RP8L 44450625 IC50 = 22 nM T84631 CQC3K0 44450638 IC50 = 41 nM T84631 CSQ67W 44450639 IC50 = 45 nM T84631 CN12UB 44450640 IC50 = 87 nM T84631 C2RS0U 44450654 IC50 = 57 nM T84631 CKT83Q 44450655 IC50 = 20 nM T84631 CPM47O 44450667 IC50 = 18 nM T84631 CTI72P 44450668 IC50 = 93 nM T84631 CC6A4Y 44453083 IC50 = 110 nM T84631 C06BVN 44453135 IC50 = 21 nM T84631 C94URG 44453211 IC50 = 0.6 nM T84631 CCR38H 44453230 Ki = 0.43 nM T84631 C0L4EK 44453237 IC50 = 2700 nM T84631 CRZ3U1 44453240 IC50 = 2 nM T84631 C12TPH 44453241 IC50 = 2 nM T84631 C5Y7AL 44453264 Ki = 2.7 nM T84631 CVQ68S 44453294 Ki = 1.1 nM T84631 CCO3E0 44453323 Ki = 2.2 nM T84631 CUAC72 44453324 Ki = 0.84 nM T84631 C4D2EV 44453334 IC50 = 17 nM T84631 CU3BS5 44453335 IC50 = 4 nM T84631 C2SH5L 44453374 IC50 = 320 nM T84631 CSC10P 44453375 IC50 = 8 nM T84631 CHRV89 44453404 Ki = 2.3 nM T84631 CH13TZ 44453406 Ki = 2.2 nM T84631 C0U3TE 44453410 IC50 = 770 nM T84631 CDZJ38 44453414 IC50 = 2 nM T84631 CK3HE8 44453438 Ki = 3200 nM T84631 C0V3FO 44453445 IC50 = 3 nM T84631 CN65UR 44453506 IC50 = 380 nM T84631 CMQ7F1 44453531 Ki = 61 nM T84631 CMNY25 44453560 Ki = 160 nM T84631 C39RNM 44453561 Ki = 420 nM T84631 CVKT34 44453567 IC50 = 1 nM T84631 C6FI3U 44453568 IC50 = 44 nM T84631 C7KER6 44453580 Ki = 16 nM T84631 C0OK6W 44453582 Ki = 28 nM T84631 C6WGH0 44453588 IC50 = 85 nM T84631 CV7FC4 44453589 IC50 = 8 nM T84631 CBMH30 44453593 IC50 = 28 nM T84631 C7T9XG 44453617 Ki = 0.35 nM T84631 C67GMZ 44453618 Ki = 0.21 nM T84631 COC52H 44453619 Ki = 18 nM T84631 C7KD4P 44453642 Ki = 0.71 nM T84631 CB86HU 44453827 IC50 = 2 nM T84631 C1OX5F 44454953 IC50 = 7.8 nM T84631 C9K1OZ 44454955 IC50 = 8.4 nM T84631 CH08YV 44454956 IC50 = 5.6 nM T84631 CG07OV 44454984 IC50 = 9 nM T84631 CXD79F 44455009 IC50 = 9.3 nM T84631 CYPN89 44455011 IC50 = 110 nM T84631 CD81LJ 44455042 IC50 = 4.5 nM T84631 CMU0N2 44455044 IC50 = 45 nM T84631 C8ZMQ1 44455079 IC50 = 28 nM T84631 CUP8J7 44455081 IC50 = 48 nM T84631 C6OXL4 44455113 IC50 = 8.6 nM T84631 COKJ02 44455114 IC50 = 530 nM T84631 CQ4F1I 44455154 IC50 = 62 nM T84631 C1MU6Z 44455155 IC50 = 130 nM T84631 CBI54T 44455189 IC50 = 10 nM T84631 CV6K4Z 44455262 IC50 = 41 nM T84631 C36KNH 44455401 IC50 = 26 nM T84631 COM4K5 44455402 IC50 = 56 nM T84631 C7RV6S 44455427 IC50 = 47 nM T84631 CMJK06 44455903 Ki = 895 nM T84631 C3D6IN 44455904 Ki = 0.5 nM T84631 CUF96X 44455934 Ki < 0.3 nM T84631 C7R0VC 44455936 Ki = 5.9 nM T84631 C91XPS 44455972 Ki = 4.5 nM T84631 C8T6VP 44455976 Ki = 2.3 nM T84631 C94SCR 44456008 Ki = 0.6 nM T84631 CHB84J 44456009 Ki = 0.8 nM T84631 CRI4A1 44456042 Ki < 1 nM T84631 CJ0WH2 44456043 Ki = 3.1 nM T84631 CET18J 44456076 Ki = 0.2 nM T84631 C4JW5U 44456118 Ki = 0.2 nM T84631 CG82AV 44456315 Ki = 5 nM T84631 CVP6D1 44456316 Ki = 16.4 nM T84631 CN7I5U 44456317 Ki < 1 nM T84631 C2HYR5 44456355 Ki = 0.6 nM T84631 CB80FW 44456356 Ki = 0.4 nM T84631 CQ2LF9 44456386 Ki = 1.2 nM T84631 C3YT1F 44456387 Ki = 0.4 nM T84631 CZJ84G 44456388 Ki = 14.7 nM T84631 CONZ35 44456432 Ki = 14.7 nM T84631 CPX63S 44456433 Ki = 125 nM T84631 C8P7AO 44456477 Ki = 29.3 nM T84631 CEVH54 44456525 IC50 > 5000 nM T84631 C2T6FK 44456526 IC50 > 5000 nM T84631 CSJY82 44456652 IC50 = 37 nM T84631 CSA87I 44456653 IC50 = 95 nM T84631 CEX4F8 44456675 IC50 = 85 nM T84631 CA80WD 44456676 IC50 = 60 nM T84631 CSRK86 44456702 IC50 = 120 nM T84631 C42JQR 44456704 IC50 = 54 nM T84631 C96YAC 44456722 IC50 = 64 nM T84631 C1C0LS 44456751 IC50 = 250 nM T84631 CZ5Q1B 44456777 IC50 = 160 nM T84631 C4R1JB 44456779 IC50 = 720 nM T84631 CAIN46 44456806 IC50 = 140 nM T84631 CZ7D3W 44456807 IC50 = 840 nM T84631 CEC75K 44456850 IC50 = 470 nM T84631 CPYT84 44456869 IC50 > 5000 nM T84631 C1TFA0 44456897 IC50 > 5000 nM T84631 C6ERW2 44456898 IC50 = 720 nM T84631 C6TFX8 44457896 Ki = 54 nM T84631 C2VAB4 44457926 Ki = 200 nM T84631 CPXA19 44457985 Ki = 100 nM T84631 C3H9RE 44458036 Ki = 120 nM T84631 COE83M 44458061 Ki = 1.1 nM T84631 C0GCJ3 44458084 Ki = 5800 nM T84631 CB4P1V 44458141 Ki = 17 nM T84631 C3B0TA 44458142 Ki = 110 nM T84631 CWS61M 44458143 Ki = 120 nM T84631 C5Z9CS 44458144 Ki = 360 nM T84631 CA2ZK4 44458145 Ki = 120 nM T84631 C1DBQ3 44458182 Ki = 60 nM T84631 CS1TF7 44460215 IC50 > 2500 nM T84631 CH61KG 44460246 IC50 > 2500 nM T84631 CWB04E 44462312 IC50 = 43.2 nM T84631 CIO47G 44473069 IC50 = 10 nM T84631 CFL8D2 44473070 IC50 = 12 nM T84631 C7S5LI 44473071 IC50 = 24 nM T84631 C75XDR 44473072 IC50 = 17 nM T84631 C06IAS 44473073 IC50 = 32 nM T84631 CZ13SI 44473074 IC50 = 28 nM T84631 CY64AE 44473075 IC50 = 15 nM T84631 CM3S2V 44473076 IC50 = 6 nM T84631 CL18JO 44473077 IC50 = 7 nM T84631 CJ6A4T 44473078 IC50 = 5 nM T84631 CSV5O4 44473081 IC50 = 6 nM T84631 C28UIH 44473082 IC50 = 2 nM T84631 CYZV01 44473085 IC50 = 55 nM T84631 CC75ON 44473086 IC50 = 4 nM T84631 CA2P3T 44473087 IC50 = 3 nM T84631 C3H8CB 44473088 IC50 = 50 nM T84631 CH12VF 44473089 IC50 = 4 nM T84631 CYP8O4 44473090 IC50 = 6 nM T84631 CSR40D 44473091 IC50 = 9 nM T84631 CS0HV7 44473092 IC50 = 56 nM T84631 CUZ97H 44473093 IC50 = 10 nM T84631 CSFM32 44473094 IC50 = 17 nM T84631 C2OT5K 44473095 IC50 = 4 nM T84631 C4H0DY 44473096 IC50 = 5 nM T84631 C7S8OZ 44473097 IC50 = 3.3 nM T84631 CO19AD 44473098 IC50 = 12 nM T84631 CTP32R 44473099 IC50 = 6 nM T84631 CBRX82 44520907 IC50 = 120 nM T84631 CP4XV3 44520908 IC50 = 1100 nM T84631 CTC95U 44520909 IC50 = 1900 nM T84631 CB5IC4 44520910 IC50 = 2300 nM T84631 CRPO96 44520911 IC50 = 69 nM T84631 CN5AX7 44520912 IC50 = 55 nM T84631 CZ54XV 44520913 IC50 = 1.4 nM T84631 C2IN6J 44520914 IC50 = 49 nM T84631 C4CT6V 44520915 IC50 = 3.5 nM T84631 CJY68M 44520916 IC50 = 4.8 nM T84631 CLA7J5 44520917 IC50 = 5.7 nM T84631 CEI82S 44520918 IC50 = 15 nM T84631 CGC10V 44520919 IC50 = 3.2 nM T84631 CS38ZY 44520920 IC50 = 4000 nM T84631 COT9K1 44520921 IC50 = 3 nM T84631 C8SOG1 44520922 IC50 = 4.1 nM T84631 CBLG40 44520923 IC50 = 870 nM T84631 CPY9M7 44520924 IC50 = 35 nM T84631 CUJ6F0 44520925 IC50 = 12 nM T84631 CM9HL2 44520927 IC50 = 4.9 nM T84631 C1H2DQ 44520928 IC50 = 12 nM T84631 C4V5OJ 44520929 IC50 = 9.5 nM T84631 CY9IN4 44520930 IC50 = 3.4 nM T84631 CVZW52 44537923 IC50 = 2700 nM T84631 C0SR7G 44560382 Ki = 0.14 nM T84631 CFSV74 44560383 Ki = 1.4 nM T84631 CH8F6K 44560756 Ki = 0.038 nM T84631 C7AIN2 44560776 Ki = 2.4 nM T84631 CMG1Z3 44560812 Ki = 5.8 nM T84631 CGC65N 44560813 Ki = 30 nM T84631 C68JXO 44560836 Ki = 54 nM T84631 CM6PB1 44560883 Ki = 0.57 nM T84631 CZD69W 44560918 Ki = 0.042 nM T84631 C6SI5T 44565123 Ki = 25084 nM T84631 C1F8OZ 44565598 IC50 = 2 nM T84631 CT47ME 44565599 IC50 = 0.5 nM T84631 C6CE3S 44565600 IC50 = 0.5 nM T84631 CGR65Q 44565601 IC50 = 0.5 nM T84631 CC7KE3 44565602 IC50 = 1.2 nM T84631 C8L5HU 44565603 IC50 = 0.9 nM T84631 C41GHV 44565623 IC50 = 1.3 nM T84631 CW5EX0 44565624 IC50 = 1 nM T84631 CDG04W 44565625 IC50 = 1.2 nM T84631 C0XC6Y 44565626 IC50 = 1.2 nM T84631 COJE58 44565627 IC50 = 0.9 nM T84631 C7EF2R 44565628 IC50 = 3 nM T84631 CB7WF1 44565629 IC50 < 0.5 nM T84631 C0MHX6 44565630 IC50 = 3 nM T84631 C14HKO 44565631 IC50 = 0.5 nM T84631 CR09OH 44565632 IC50 = 0.4 nM T84631 CA0XT3 44565740 IC50 < 0.5 nM T84631 CY4HL8 44565741 IC50 = 1.5 nM T84631 CD94RJ 44565746 IC50 = 1.3 nM T84631 C2EJ4X 44565747 IC50 = 1.1 nM T84631 C9XT0W 44565748 IC50 = 3 nM T84631 C5NTH8 44565757 IC50 = 6 nM T84631 CXZK47 44565758 IC50 = 1.1 nM T84631 C48BCZ 44565759 IC50 = 7 nM T84631 CBV9Z6 44565760 IC50 = 2 nM T84631 C7MSE6 44565784 IC50 = 0.7 nM T84631 CAE2K6 44565785 IC50 = 1 nM T84631 CW4DZ0 44565786 IC50 = 3 nM T84631 C4O1MU 44565787 IC50 = 1 nM T84631 C9GXH4 44565788 IC50 = 6 nM T84631 CKF9Z4 44565789 IC50 = 17 nM T84631 C4CX2F 44565790 IC50 = 10 nM T84631 CEW6G1 44569299 Ki = 10 nM T84631 C9JNT3 44569300 Ki = 1700 nM T84631 C9XE7Q 44569301 Ki = 92000 nM T84631 CZI8D7 44569333 Ki = 430000 nM T84631 CR4CP6 44569359 Ki = 55000 nM T84631 C9JF7W 44569667 Ki = 4400 nM T84631 C61IJB 44569732 Ki = 8000 nM T84631 CR36MB 44569733 Ki = 61000 nM T84631 CE25UL 44569767 Ki = 20000 nM T84631 C0CZ4I 44569768 Ki = 14000 nM T84631 CIR4M0 44569769 Ki = 5400 nM T84631 C02SHD 44569811 Ki = 700 nM T84631 CG3LE9 44569812 Ki = 5600 nM T84631 CCU7V0 44569813 Ki = 910 nM T84631 C8BR6E 44569843 Ki = 660 nM T84631 C7Q9BH 44569844 Ki = 3400 nM T84631 CZ35OW 44569845 Ki = 420 nM T84631 CHV9C1 44569846 Ki = 630 nM T84631 C5JQ4W 44569889 Ki = 1600 nM T84631 CE1O4I 44569890 Ki = 3500 nM T84631 C4JU7I 44569891 Ki = 150 nM T84631 CGS83Z 44569892 Ki = 250 nM T84631 CFKJ12 44570705 IC50 = 4.5 nM T84631 CCA09Y 44570706 IC50 = 2.6 nM T84631 C7QWX9 44570769 IC50 = 2.9 nM T84631 C64OEB 44570770 IC50 = 2.3 nM T84631 C3KF1Y 44570771 IC50 = 3.5 nM T84631 CJVS07 44570772 IC50 = 2.5 nM T84631 C60XGS 44571089 IC50 = 3.4 nM T84631 C7DBF4 44571090 IC50 = 2.2 nM T84631 CGRP54 44571091 IC50 = 4.2 nM T84631 CYKJ28 44571092 IC50 = 5.4 nM T84631 CL9XM5 44571093 IC50 = 12 nM T84631 C0RU9L 44571134 IC50 = 1.8 nM T84631 C4BN3H 44573109 Ki = 10000 nM T84631 COR57Y 44573272 Ki = 4400 nM T84631 C6DX3Y 44573273 Ki = 3400 nM T84631 CM2R1P 44573274 Ki = 44000 nM T84631 CSP1I0 44573310 Ki = 2500 nM T84631 C6EG9V 44573311 Ki = 11000 nM T84631 CYV3X2 44573378 Ki = 17000 nM T84631 CWUA41 44573379 Ki = 100 nM T84631 CYA64G 44573380 Ki = 127000 nM T84631 CLG42S 44573428 Ki = 30000 nM T84631 C5F9RK 44577595 IC50 = 400 nM T84631 CIO19Z 44577596 IC50 = 1159 nM T84631 CLUJ07 44577597 IC50 = 246 nM T84631 CU2E3N 44577598 IC50 = 208 nM T84631 CC7IV5 44577599 IC50 = 494 nM T84631 C1LM4B 44577642 IC50 = 245 nM T84631 C5Q6ZB 44577643 IC50 = 276 nM T84631 CTE9W4 44577644 IC50 = 709 nM T84631 CD6OY9 44577645 IC50 = 193 nM T84631 C1O6VJ 44577646 IC50 = 227 nM T84631 CD2NO7 44577647 IC50 = 403 nM T84631 CX14HM 44577648 IC50 = 872 nM T84631 CV21YL 44577649 IC50 = 628 nM T84631 CO19SA 44577650 IC50 = 380 nM T84631 CVMN47 44577651 IC50 = 14 nM T84631 C3YZF4 44577954 IC50 = 517 nM T84631 CMK2S5 44577955 IC50 = 371 nM T84631 CP62MY 44577956 IC50 = 198 nM T84631 CRW83N 44577957 IC50 = 835 nM T84631 C01HVO 44577990 IC50 = 373 nM T84631 CPUZ06 44577991 IC50 = 222 nM T84631 C4XKY0 44577992 IC50 = 271 nM T84631 C30CBZ 44577993 IC50 = 396 nM T84631 CU4T1V 44577994 IC50 = 267 nM T84631 C15TZO 44577995 IC50 = 294 nM T84631 C65QDR 44577996 IC50 = 546 nM T84631 CF63WE 44578029 IC50 = 256 nM T84631 CHS79J 44578030 IC50 = 368 nM T84631 C5TBZ9 44578031 IC50 = 272 nM T84631 C3W8PT 44578032 IC50 = 462 nM T84631 CPYZ70 44578033 IC50 = 386 nM T84631 C7Y1QL 44578034 IC50 = 17 nM T84631 CLT8Z4 44578035 IC50 = 1073 nM T84631 CK6UG1 44578036 IC50 = 506 nM T84631 CLT5O2 44581199 Ki = 0.043 nM T84631 C97WFB 44581200 Ki = 0.084 nM T84631 CK8MJ1 44581201 Ki = 0.14 nM T84631 CPB78V 44581202 Ki = 0.74 nM T84631 CG1A0W 44581236 Ki = 0.56 nM T84631 C90ZBV 44581286 Ki = 0.18 nM T84631 CYL1B8 44581287 Ki = 0.32 nM T84631 CUJ83A 44581288 Ki = 0.071 nM T84631 CO12AM 44581325 Ki = 0.29 nM T84631 CHM16K 44581326 Ki = 0.59 nM T84631 C5CW2I 44581328 Ki = 0.36 nM T84631 C5BIF8 44581330 Ki = 0.068 nM T84631 CR75GK 44581361 Ki = 0.24 nM T84631 CH4M0F 44581362 Ki = 0.055 nM T84631 CB1GN5 44581363 Ki = 0.15 nM T84631 C2PXK1 44581390 Ki = 0.051 nM T84631 C6JX8N 44581393 Ki = 0.054 nM T84631 CT2DU0 44581418 Ki = 0.027 nM T84631 CMHW28 44581420 Ki = 0.042 nM T84631 CN32IF 44581421 Ki = 0.093 nM T84631 C8XF5J 44581456 Ki = 0.073 nM T84631 CA54PQ 44581457 Ki = 0.24 nM T84631 C2MQ1A 44581459 Ki = 0.11 nM T84631 CR42LZ 44581460 Ki = 0.78 nM T84631 CYZN78 44581494 Ki = 0.16 nM T84631 C2M3XU 44581496 Ki = 0.085 nM T84631 CLRP24 44581497 Ki = 0.12 nM T84631 C7ZQF0 44581498 Ki = 0.14 nM T84631 CMY6U3 44581556 Ki = 5.1 nM T84631 CN69DU 44581557 Ki = 3 nM T84631 CZ4L9O 44581558 Ki = 11 nM T84631 C7IKA3 44581559 Ki = 1.5 nM T84631 C9P7CT 44581590 Ki = 2.9 nM T84631 CBE98L 44581591 Ki = 7.6 nM T84631 C4N6LC 44581592 Ki = 20 nM T84631 CXW8T5 44581593 Ki = 0.55 nM T84631 C03LRJ 44581629 Ki = 0.02 nM T84631 CYUF13 44581630 Ki = 0.02 nM T84631 C6YDN5 44581631 Ki = 0.21 nM T84631 CJL04I 44581664 Ki = 0.021 nM T84631 C0UET1 44581665 Ki = 0.16 nM T84631 C6MTH1 44581704 Ki = 4.9 nM T84631 CX0T1R 44581705 Ki = 1.1 nM T84631 C6Y7QO 44581749 Ki = 0.065 nM T84631 CH6VU9 44581750 Ki = 0.31 nM T84631 C7Q8RG 44582128 IC50 = 0.5 nM T84631 CE4F0K 44582129 IC50 = 0.18 nM T84631 CN3FT7 44582147 IC50 = 1.2 nM T84631 C2LKP1 44582148 IC50 = 0.11 nM T84631 C4LZJ3 44582149 IC50 = 0.34 nM T84631 CA2N1I 44582150 IC50 = 0.02 nM T84631 CRW3K7 44582204 IC50 = 0.54 nM T84631 CIW63Z 44582205 IC50 = 0.31 nM T84631 C3E4LY 44582206 IC50 = 0.5 nM T84631 CCU71D 44582207 IC50 = 0.18 nM T84631 C0AG3O 44582221 IC50 = 0.22 nM T84631 CU5W8N 44582222 IC50 = 0.05 nM T84631 C06BKE 44582223 IC50 = 0.16 nM T84631 CJ96RG 44582224 IC50 = 0.08 nM T84631 C18TMJ 44586926 IC50 = 110 nM T84631 CR1XF9 44586927 IC50 = 840 nM T84631 C45DAE 44586955 IC50 = 75 nM T84631 C72KMC 44586956 IC50 = 88 nM T84631 CB8T1E 44586957 IC50 = 16 nM T84631 CCU92M 44586958 IC50 = 12 nM T84631 CR6X5Q 44587208 Ki = 2700 nM T84631 C87KXE 44587209 Ki = 330 nM T84631 CGOR19 44587231 Ki = 1500 nM T84631 C8WH9R 44587232 Ki = 160 nM T84631 C3WOP7 44587261 Ki = 25000 nM T84631 CX1DP6 44587262 Ki = 1800 nM T84631 C7K6JN 44587263 Ki = 3130 nM T84631 CKL1J2 44587264 Ki = 685 nM T84631 CTF79D 44587290 Ki = 2483 nM T84631 CBXY02 44587291 Ki = 14700 nM T84631 CDBV80 44587292 Ki = 5700 nM T84631 CWZ34J 44587314 Ki = 920 nM T84631 C6Y1FA 44587835 Ki = 3000 nM T84631 C91QNS 44587836 Ki = 14000 nM T84631 C0CRG4 44589267 IC50 = 336 nM T84631 CY3VQ2 44589268 IC50 = 46 nM T84631 C10NMD 44590397 Ki = 7991 nM T84631 COQ0E6 44592399 IC50 = 35 nM T84631 CK82XN 44592400 IC50 = 290 nM T84631 C3XEW7 44592401 IC50 = 25 nM T84631 C96CWM 44592402 IC50 = 30 nM T84631 C17NRH 44592470 IC50 = 6 nM T84631 CRF34H 44592525 IC50 = 9 nM T84631 C3L1AN 44592526 IC50 = 8 nM T84631 CI5C1F 44592560 IC50 = 26.96 nM T84631 C9RWU8 44592561 IC50 = 0.31 nM T84631 CHK9G2 44592562 IC50 = 6.62 nM T84631 CNIX06 44592593 IC50 = 11.27 nM T84631 CZJ7C6 44592617 IC50 = 46.05 nM T84631 C1A8YB 44592658 IC50 = 50 nM T84631 CN7G0O 44592693 IC50 = 36.49 nM T84631 CC65UK 44592729 IC50 = 1.3 nM T84631 C9OG6N 44592765 IC50 = 0.05 nM T84631 CKC2Q8 44592831 IC50 = 0.13 nM T84631 CY2IM4 44592833 IC50 = 0.05 nM T84631 CW72YN 44592864 IC50 = 0.02 nM T84631 CD4G2B 44592865 IC50 = 0.23 nM T84631 CDLY78 44592888 IC50 = 1.75 nM T84631 C4RDW0 44592955 IC50 = 50 nM T84631 C1PLT5 44592978 IC50 = 50 nM T84631 CVS21G 44592979 IC50 = 8.14 nM T84631 C4M0KI 44593006 IC50 = 1.17 nM T84631 C9PCO6 44593008 IC50 = 7.6 nM T84631 C1Y8IM 44593413 Ki = 0.064 nM T84631 C8X3KA 44593414 Ki = 0.025 nM T84631 C97UBM 44593556 IC50 = 7.5 nM T84631 CPZR42 44607103 IC50 = 27900 nM T84631 C6MIK9 44626665 IC50 = 1023 nM T84631 C4LQW3 44629430 Ki = 11900 nM T84631 CL20GE 44629584 Ki = 0.2 nM T84631 CUK2I7 45103480 Ki = 70 nM T84631 CP6SB1 45103481 Ki = 290 nM T84631 CM16YW 45103482 Ki = 52 nM T84631 C2PVE0 45103523 Ki = 6500 nM T84631 CKN2F4 45103582 Ki = 2.6 nM T84631 C80DXA 45103583 Ki = 0.5 nM T84631 CG51EA 45103584 Ki = 1300 nM T84631 C46JPW 45103585 Ki = 250 nM T84631 C8XBZ6 45103586 Ki = 560 nM T84631 CXS6K8 45103587 Ki = 825 nM T84631 CPR1O7 45103680 Ki = 354 nM T84631 CJU8M5 45103681 Ki = 2844 nM T84631 CZ4JW1 45261445 Ki = 102 nM T84631 C3P8EA 45263195 IC50 = 600 nM T84631 CK7E3M 45264760 Ki = 220 nM T84631 C3Y8WE 45266133 Ki = 3900 nM T84631 C5E6AS 45267012 IC50 = 1720 nM T84631 CZ32WR 45267285 IC50 = 2882 nM T84631 C1TYA3 45267286 IC50 = 2677 nM T84631 CU3WJ8 45267299 IC50 = 21 nM T84631 C41ELS 45267302 IC50 = 928 nM T84631 C67DKE 45267303 IC50 = 195 nM T84631 CGU67A 45267836 IC50 = 2030 nM T84631 CW3SX0 45267838 IC50 = 1050 nM T84631 CT1WY2 45268147 IC50 = 780 nM T84631 C1ZWU3 45268157 IC50 = 2600 nM T84631 CCVL15 45268158 IC50 = 2939 nM T84631 CB1O0D 45268159 IC50 = 11 nM T84631 C6GDW5 45268170 IC50 = 53 nM T84631 CY75OX 45268711 IC50 = 2810 nM T84631 CZ0YE8 45269033 IC50 = 11879 nM T84631 CMSU50 45269045 IC50 = 30000 nM T84631 C9Z5TG 45269048 IC50 = 15 nM T84631 CSY60N 45269572 IC50 = 3230 nM T84631 CO18RA 45269846 IC50 = 54 nM T84631 C42QBM 45269847 IC50 = 28 nM T84631 C2QLJ7 45269887 IC50 = 2400 nM T84631 CDAM80 45269891 IC50 = 349 nM T84631 CQO6T8 45269898 IC50 > 32000 nM T84631 COA86N 45270402 IC50 = 1520 nM T84631 CFQ14D 45270405 IC50 = 800 nM T84631 CH1P5M 45270407 IC50 = 2790 nM T84631 CP7DF5 45270707 IC50 > 34000 nM T84631 C7EV9T 45270708 IC50 > 34000 nM T84631 CAMB38 45270720 IC50 = 76 nM T84631 CI49ER 45270731 IC50 = 19 nM T84631 C90JGW 45270732 IC50 = 386 nM T84631 CB2QX3 45270733 IC50 = 22 nM T84631 C6YPG9 45270763 Ki = 14 nM T84631 CU26GQ 45271227 IC50 = 1630 nM T84631 C41TXV 45271542 IC50 = 167 nM T84631 C45DVC 45271581 Ki = 43 nM T84631 CW6CB5 45272126 IC50 = 210 nM T84631 CWP6T9 45272400 IC50 = 5 nM T84631 CPBF26 45272436 IC50 > 34000 nM T84631 C96EXW 45272443 IC50 = 18759 nM T84631 C49XBD 45272455 IC50 = 940 nM T84631 C7UDO4 45273309 IC50 = 1300 nM T84631 CF97AM 45273310 IC50 = 84 nM T84631 C4N0LV 45273311 IC50 = 15538 nM T84631 C69XFH 45273319 IC50 = 2728 nM T84631 CS8U0D 45273320 IC50 = 27 nM T84631 CQ7SY8 45273327 IC50 = 14818 nM T84631 CJ73BT 45486346 Ki = 83000 nM T84631 C9ETC4 45486354 Ki = 123000 nM T84631 CVEK34 45488045 IC50 = 18 nM T84631 CK15WB 45488046 IC50 = 10 nM T84631 CE4F6R 45488047 IC50 = 3 nM T84631 CI5S4V 45488048 IC50 = 3 nM T84631 C8VOL9 46191308 Ki = 0.8 nM T84631 CCG5U1 46196561 Ki = 0.5 nM T84631 C1I0OD 46222444 IC50 = 11 nM T84631 CCP8B0 46222445 IC50 = 1.7 nM T84631 CCM09Y 46222669 IC50 = 24 nM T84631 CCH8I6 46222670 IC50 = 51 nM T84631 CQ4BV0 46222671 IC50 = 60 nM T84631 C14DQZ 46222672 IC50 = 14 nM T84631 C9LU7N 46222673 IC50 = 147 nM T84631 C5T6FE 46226298 Ki = 6.2 nM T84631 CB9O0A 46226299 Ki = 6 nM T84631 CW86BU 46226322 Ki = 5.1 nM T84631 CV1R9H 46226323 Ki = 35 nM T84631 C8JPB3 46226324 Ki = 1.5 nM T84631 C63LKZ 46226325 Ki = 0.8 nM T84631 C3WRU1 46226349 Ki = 5 nM T84631 CS7X8I 46226372 Ki = 0.8 nM T84631 C3IA0F 46226373 Ki = 2 nM T84631 CE6F8R 46226374 Ki = 1 nM T84631 C1HPB8 46226391 Ki = 5 nM T84631 CGZF19 46226392 Ki = 0.8 nM T84631 CO8I9D 46226393 Ki = 2 nM T84631 CG8LX3 46226394 Ki = 2 nM T84631 CKL39P 46226415 Ki = 4 nM T84631 CQW85G 46226416 Ki = 2 nM T84631 C3RMI8 46226796 IC50 > 5000 nM T84631 C7BQ1U 46226806 IC50 = 21 nM T84631 CM10IF 46226817 IC50 = 930 nM T84631 CW47XK 46232635 Ki = 9 nM T84631 C9L1ZS 46233075 Ki = 1560 nM T84631 CD62VO 46233076 Ki = 1270 nM T84631 C5PI6E 46233077 Ki = 1300 nM T84631 C9BLH7 46233114 Ki = 2375 nM T84631 C42DOH 46233115 Ki = 1628 nM T84631 CA7S2F 46233116 Ki = 1585 nM T84631 CQ4UF5 46233117 Ki = 2115 nM T84631 CEU41B 46233150 Ki = 1363 nM T84631 CXV4P6 46233151 Ki = 3970 nM T84631 CFA7H0 46233153 Ki = 2600 nM T84631 CH01MJ 46233194 Ki = 600 nM T84631 CR5VN4 46233261 Ki = 6200 nM T84631 CHF74W 46233262 Ki = 7300 nM T84631 C8ONP6 46233306 Ki = 4300 nM T84631 CG6QI5 46233307 Ki = 2900 nM T84631 CL0W5E 46233309 Ki = 4300 nM T84631 C8AQZ5 46233310 Ki = 13100 nM T84631 C7XT0F 46233339 Ki = 7900 nM T84631 CJ3P5N 46233341 Ki = 5700 nM T84631 CBC4Y5 46233342 Ki = 105 nM T84631 CUPC52 46233343 Ki = 55 nM T84631 CHF45Z 46233364 Ki > 100000 nM T84631 CUZW20 46233366 Ki = 3350 nM T84631 CTMN13 46233367 Ki = 1150 nM T84631 C23KIW 46233369 Ki = 45000 nM T84631 CLHX82 46233406 Ki = 13800 nM T84631 C8T5CW 46233408 Ki = 3400 nM T84631 CQ01MF 46233409 Ki = 150 nM T84631 CY92TG 46233410 Ki = 950 nM T84631 CZ7CQ8 46233411 Ki = 44 nM T84631 CPBS35 46233412 Ki = 910 nM T84631 C12SEZ 46233413 Ki = 17 nM T84631 C7VKZ8 46233414 Ki = 33 nM T84631 CCI75A 46233462 Ki = 37 nM T84631 CYG6A2 46233463 Ki = 25 nM T84631 CT5MH6 46233491 Ki = 0.6 nM T84631 CY5C1O 46233492 Ki = 4450 nM T84631 C5H2EF 46233511 Ki = 960 nM T84631 CZ46CU 46233512 Ki = 1740 nM T84631 CI8NV4 46233513 Ki = 700 nM T84631 C84HTG 46233514 Ki = 360 nM T84631 CA4Z5X 46233537 Ki = 1810 nM T84631 C5SK7C 46233538 Ki = 830 nM T84631 C0Y8IT 46233539 Ki = 550 nM T84631 C16IMD 46233540 Ki = 1300 nM T84631 CW3S0U 46233565 Ki = 1700 nM T84631 C03TRU 46233566 Ki = 1184 nM T84631 C8RCY2 46233567 Ki = 800 nM T84631 CHO28I 46233568 Ki = 600 nM T84631 CRDC20 46233603 Ki = 3773 nM T84631 CWVY84 46233604 Ki = 872 nM T84631 C7ZP4M 46233605 Ki = 1562 nM T84631 CT84CW 46233649 Ki = 1147 nM T84631 CF8Z3Q 46233651 Ki = 828 nM T84631 CX28UI 46233688 Ki = 1482 nM T84631 C9P0FC 46233689 Ki = 1303 nM T84631 CWO0V7 46233690 Ki = 2252 nM T84631 C7ET8Q 46233691 Ki = 2051 nM T84631 C8E0ZQ 46835134 Ki = 192 nM T84631 C62RBC 46835135 Ki = 9 nM T84631 CY47OV 46878192 Ki > 6000 nM T84631 CQ2G6A 46878194 Ki > 6000 nM T84631 CC6GE9 46878197 Ki = 970 nM T84631 CE79OB 46878198 Ki > 6000 nM T84631 CS07EW 46878199 Ki > 6000 nM T84631 C3HZP7 46878200 Ki = 6000 nM T84631 CF5ZQ8 46878201 Ki = 6000 nM T84631 C7ICJ0 46878202 Ki > 6000 nM T84631 CQJR51 46878203 Ki = 9 nM T84631 C9BXU7 46878204 Ki = 6000 nM T84631 CXQL63 46878205 Ki > 6000 nM T84631 CR93NC 46878206 Ki > 6000 nM T84631 C0H3UO 46878241 Ki > 5000 nM T84631 CS7B4G 46888797 IC50 = 20 nM T84631 CNS8R6 46888834 IC50 = 49 nM T84631 CPT7U3 46888835 IC50 = 28 nM T84631 CS7XO5 46889240 IC50 = 23 nM T84631 C9E3HU 46889265 IC50 = 46 nM T84631 C8U3OW 46889266 IC50 = 198 nM T84631 CNA06P 46905365 Ki = 200 nM T84631 CX2L8G 46905375 Ki = 34 nM T84631 CTR32W 46905376 Ki = 10 nM T84631 CS8GZ7 46905377 Ki = 200 nM T84631 C9W1ZK 46905378 Ki = 670 nM T84631 CR6P1E 46905379 Ki = 71 nM T84631 C75IRP 46905995 Ki = 1.3 nM T84631 CB2F7T 46978227 Ki > 62500 nM T84631 CEDL20 49796469 Ki = 80 nM T84631 C8NK1S 49796470 Ki = 800 nM T84631 C4MK5H 49796471 Ki = 7800 nM T84631 C75HOB 49796472 Ki = 900 nM T84631 CS90ZF 49796473 Ki = 24 nM T84631 CXUM36 49820499 Ki = 300 nM T84631 CX7SA8 49820500 Ki = 300 nM T84631 C6OIW8 49820657 Ki = 2300 nM T84631 CAI5S9 49827569 Ki = 7.943 nM T84631 CU1DK9 49835415 Ki = 52 nM T84631 C0OQ8N 49835557 Ki = 2.7 nM T84631 CQ23SL 49864307 Ki = 201 nM T84631 CTO73I 49864308 Ki = 22 nM T84631 CT8NM4 49864309 Ki = 46 nM T84631 C8U1HB 49864310 Ki = 40 nM T84631 C78QKE 49864328 Ki = 120 nM T84631 CFIW73 49864329 Ki = 28 nM T84631 CDZ3B0 49864350 Ki = 11 nM T84631 CLW9I6 49864373 Ki = 17 nM T84631 CSZ3P1 49864435 Ki = 46 nM T84631 CZR1W9 49864436 Ki = 34 nM T84631 C5YH3T 49864437 Ki = 44 nM T84631 CK5G4W 49864458 Ki = 11 nM T84631 CLOY62 49864459 Ki = 24 nM T84631 CR8JK9 49864483 Ki = 27 nM T84631 C42KOC 49864498 Ki = 345 nM T84631 CR3F4Q 49864657 Ki = 36 nM T84631 CIP8O4 49864658 Ki = 92 nM T84631 CWA50O 49864685 Ki = 1779 nM T84631 C9P6TE 49864704 Ki = 42 nM T84631 CM4YA0 49864705 Ki = 15 nM T84631 CRW92J 49864706 Ki = 40 nM T84631 CU0LX7 50919254 Ki = 2 nM T84631 C2LK1E 50919255 Ki = 9 nM T84631 CIZ5Y1 50919256 Ki = 2 nM T84631 CC89AZ 50919257 Ki = 4 nM T84631 CAM3V7 50939649 Ki = 50 nM T84631 CHC74O 50939651 Ki = 810 nM T84631 CT9P8Q 51041296 Ki = 0.11 nM T84631 CKCN49 51346898 Ki = 3 nM T84631 CV0IQ5 52940898 Ki < 0.3 nM T84631 C2DO1B 52940908 IC50 = 8 nM T84631 C84CYB 52940909 IC50 = 4 nM T84631 C4FDU5 52941018 IC50 = 35 nM T84631 C1DRJ2 52941698 Ki = 0.1 nM T84631 C57MVG 52942150 Ki = 3 nM T84631 CPK9R0 52943286 Ki = 0.7 nM T84631 CBO9N7 52943447 IC50 = 120 nM T84631 CQ19NI 52944468 Ki = 2 nM T84631 C1M3EC 52944526 IC50 = 3 nM T84631 C1RWG9 52944684 IC50 = 3450 nM T84631 C8XN9J 52945796 Ki = 1100 nM T84631 CR06QB 52946959 Ki = 0.55 nM T84631 CI0P3R 52947731 Ki = 0.9 nM T84631 CU90GX 52949410 Ki < 0.4 nM T84631 CVRQ75 52949419 Ki = 0.6 nM T84631 C4Y8FZ 52949515 Ki = 16000 nM T84631 CPE05T 53242224 IC50 = 2.2 nM T84631 CB8XU4 53317105 IC50 = 13 nM T84631 CS6TR3 53317106 IC50 = 48 nM T84631 COP4X3 53317127 IC50 = 9 nM T84631 CX1KR9 53317330 Ki = 1 nM T84631 CA86OS 53317375 Ki = 1000000 nM T84631 CA45BG 53317639 IC50 = 1618 nM T84631 C8U3NB 53317693 IC50 = 439 nM T84631 C68TOQ 53318416 IC50 = 1930 nM T84631 CIVY68 53318619 Ki = 15 nM T84631 CXVJ49 53318620 Ki = 6 nM T84631 CLUD64 53319727 IC50 = 4145 nM T84631 CWOK94 53321019 IC50 = 27 nM T84631 C6K1WJ 53321020 IC50 = 11 nM T84631 C79RGN 53321237 Ki = 5 nM T84631 CAYD14 53321238 Ki = 2 nM T84631 C7QEI1 53321291 Ki = 16000 nM T84631 C7CR5Q 53322361 IC50 = 6830 nM T84631 CL0SC2 53322387 IC50 = 623 nM T84631 CL6R7Y 53322388 IC50 = 204 nM T84631 CL29IO 53322566 Ki = 6 nM T84631 CFOI53 53322612 Ki = 80000 nM T84631 CR0VJ3 53323722 IC50 = 93 nM T84631 C3B1AG 53323723 IC50 = 2476 nM T84631 C0A1DL 53323905 Ki = 2 nM T84631 CWA7B3 53323948 Ki = 1000000 nM T84631 CUQ82T 53324997 IC50 = 1025 nM T84631 CJB75L 53324998 IC50 = 5675 nM T84631 CP9JT3 53324999 IC50 = 18 nM T84631 CSHU35 53325000 IC50 = 12 nM T84631 CO6TG4 53325236 Ki = 1000000 nM T84631 CO0R2M 53325237 Ki = 1000000 nM T84631 COF8N6 53325369 Ki = 3 nM T84631 CK25QS 53326291 IC50 = 642 nM T84631 CFB65G 53326292 IC50 > 10000 nM T84631 CW10IE 53326477 Ki = 100 nM T84631 CT2RQ6 53326832 Ki = 4 nM T84631 C0DYJ6 53326870 IC50 = 59 nM T84631 CA6GQ5 53341037 Ki > 13300 nM T84631 CIKQ81 53345652 Ki > 130 nM T84631 CXWS90 53345968 Ki > 1000 nM T84631 CB08CW 53379392 Ki = 129 nM T84631 C6XNM0 53380822 Ki = 1500 nM T84631 C1KFQ0 53380823 Ki = 9800 nM T84631 C7JWD0 53380936 Ki = 6660 nM T84631 C97KGD 53380937 Ki = 6800 nM T84631 CKV6Q2 53380938 Ki = 1600 nM T84631 C47WIH 53380939 Ki = 15000 nM T84631 CY3RO0 53380940 Ki = 5490 nM T84631 C3R8PW 53380941 Ki = 6000 nM T84631 CI5XO8 53388478 IC50 = 970000 nM T84631 C4HB3V 53392251 IC50 > 300000 nM T84631 CV60BK 53488415 Ki = 4.71 nM T84631 C8SCH2 53800364 IC50 = 50 nM T84631 C9GFU3 53864431 IC50 = 190 nM T84631 C16KAQ 53954748 IC50 = 56 nM T84631 CEIQ26 54352954 IC50 = 3000 nM T84631 CQNW76 54507330 IC50 = 200 nM T84631 C2FS3H 54555233 IC50 = 100 nM T84631 CI67SD 54580287 IC50 = 1600 nM T84631 C82FQT 54580288 IC50 = 3.5 nM T84631 C4C3DP 54581293 IC50 = 200 nM T84631 CXE31M 54581294 IC50 = 7.4 nM T84631 CV20EN 54581295 IC50 > 10000 nM T84631 CUY6J3 54581296 IC50 = 65 nM T84631 CE3D7F 54582336 IC50 = 1.9 nM T84631 C3EM0S 54583288 IC50 = 3945 nM T84631 CUSC68 54583289 IC50 = 7.7 nM T84631 C9IJ0M 54583290 IC50 = 170 nM T84631 C6C7NO 54584026 Ki = 0.5012 nM T84631 CH3A5X 54584246 IC50 = 1200 nM T84631 CYB6H9 54584247 IC50 = 970 nM T84631 C2H6IJ 54584248 IC50 = 110 nM T84631 C0MA2W 54584249 IC50 = 1.1 nM T84631 CSMJ20 54584250 IC50 = 2.5 nM T84631 C38YZE 54584279 IC50 = 120 nM T84631 CN7T4Q 54584280 IC50 = 100 nM T84631 CC1S7R 54585216 IC50 = 70 nM T84631 C7TEM9 54585217 IC50 = 770 nM T84631 CL86NU 54585218 IC50 = 5.6 nM T84631 CP8EA5 54585238 IC50 = 2.7 nM T84631 C7BTJ1 54586167 IC50 = 47 nM T84631 CC6AT1 54586168 IC50 = 460 nM T84631 CT8G6K 54586169 IC50 = 610 nM T84631 C5K3JQ 54586170 IC50 = 100 nM T84631 CBO8V7 54587183 IC50 = 221 nM T84631 CNO24S 54587184 IC50 = 4100 nM T84631 CQ5PV6 54587185 IC50 = 2100 nM T84631 CFLR93 54587186 IC50 = 29 nM T84631 C2GZA5 54587362 IC50 = 690 nM T84631 C9I4OP 54738720 Ki = 4400 nM T84631 CWQ17K 54751669 Ki = 146 nM T84631 CK52NT 54751670 Ki = 1620 nM T84631 C17MSO 56640092 Ki = 152 nM T84631 CGP7Y6 56640160 Ki = 21 nM T84631 C30AJK 56640226 Ki = 784 nM T84631 C9YXM2 56659587 IC50 = 1078000 nM T84631 CA32CM 56659850 Ki = 1.4 nM T84631 C6OI5V 56660094 Ki = 8000 nM T84631 CKFI81 56660095 Ki = 1200 nM T84631 CKO4M6 56663319 Ki = 37 nM T84631 C2T1WM 56665604 IC50 = 380 nM T84631 CMG9H6 56666511 IC50 > 580000 nM T84631 CCM80T 56670171 Ki = 31 nM T84631 C0M3AE 56673432 IC50 > 1480000 nM T84631 CI6RX7 56673433 IC50 > 590000 nM T84631 CGM2J4 56673694 Ki = 21 nM T84631 C4T6NO 56673695 Ki = 14.5 nM T84631 C7DE8I 56676739 IC50 > 1340000 nM T84631 CE4AT6 56676740 IC50 > 400000 nM T84631 C8CN9W 56676741 IC50 = 440000 nM T84631 C1TH3W 56677006 Ki = 565 nM T84631 CY34VE 56677007 Ki = 2.1 nM T84631 C5LVJ2 56680051 IC50 > 640000 nM T84631 CKF2M0 56680052 IC50 = 508000 nM T84631 C72IHP 56680339 Ki = 397 nM T84631 CT7U8L 56683905 Ki = 4900 nM T84631 C3CDB4 56683906 Ki = 4700 nM T84631 C14YLP 56849975 IC50 = 103 nM T84631 C5DQ2M 56849977 IC50 = 539 nM T84631 C1F8IX 56849978 IC50 = 140 nM T84631 C2V0JC 56850120 IC50 = 73.4 nM T84631 CRL87T 56850121 IC50 = 118 nM T84631 CKD9E0 56850122 IC50 = 213 nM T84631 CIDT59 56850256 IC50 = 99.2 nM T84631 CE0X3B 56850258 IC50 = 31.1 nM T84631 CFZ7P2 56850260 IC50 = 50.3 nM T84631 C06NPR 56850396 IC50 = 157 nM T84631 CN35WB 56850397 IC50 = 155 nM T84631 CLS9Y7 56850526 IC50 = 1438 nM T84631 CKNE35 56850528 IC50 = 6143 nM T84631 CX63IV 56850529 IC50 = 349 nM T84631 CN5EI8 56850671 IC50 = 64.2 nM T84631 CM2W4G 56850672 IC50 = 59.8 nM T84631 CJAK41 56850673 IC50 = 86.1 nM T84631 CDKY37 56850674 IC50 = 41.3 nM T84631 CLF6Q0 56850675 IC50 = 41.4 nM T84631 C8UHN3 56949979 IC50 = 9000 nM T84631 CH1EI8 56954620 Ki = 3430 nM T84631 C4EHU8 56954732 Ki = 9370 nM T84631 C5C8XO 56954733 Ki = 3472 nM T84631 CST4F0 56954834 Ki = 42 nM T84631 CRK92A 56954952 Ki = 1860 nM T84631 CB57DW 57391171 Ki = 7600 nM T84631 CZ6D2Q 57391429 IC50 = 4.9 nM T84631 CZ41MI 57391430 IC50 = 0.74 nM T84631 CWJ4I7 57391565 Ki = 14000 nM T84631 C36LXQ 57392276 IC50 = 20 nM T84631 CPBW48 57392333 Ki = 360000 nM T84631 CUI1W3 57392347 IC50 = 32 nM T84631 CPF25Q 57392348 IC50 = 337 nM T84631 C15EGS 57392349 IC50 = 674 nM T84631 C0DZ6H 57392472 IC50 = 7 nM T84631 C7APO2 57392934 Ki = 6500 nM T84631 CZ2A0S 57392935 Ki = 1600 nM T84631 C6M5RS 57393195 IC50 = 1.6 nM T84631 CX16KB 57393324 Ki = 4000 nM T84631 CG9AS5 57394027 IC50 = 8.3 nM T84631 C1AZB4 57394031 IC50 = 4.7 nM T84631 CR9S5P 57394086 IC50 = 129 nM T84631 CNQT87 57394087 IC50 = 1330 nM T84631 COB56U 57394088 IC50 = 22 nM T84631 C3K0VW 57394177 IC50 = 13 nM T84631 C6EWL9 57394677 Ki = 5600 nM T84631 CE2BA9 57394917 IC50 = 49 nM T84631 CG07ZY 57394918 IC50 = 1.5 nM T84631 C8T2ZJ 57395044 Ki = 790 nM T84631 CNLD49 57395793 IC50 = 5 nM T84631 CL2JE5 57395841 Ki = 310000 nM T84631 CSF3D7 57395856 IC50 = 32 nM T84631 CN0UR9 57395857 IC50 = 51 nM T84631 CI1QX2 57395858 IC50 = 14 nM T84631 C2JI3K 57397571 IC50 = 6 nM T84631 CKR94L 57397646 IC50 = 11 nM T84631 CYEK40 57397750 IC50 = 10 nM T84631 C9F4OL 57398232 Ki = 7700 nM T84631 C5OAB7 57398233 Ki = 2830 nM T84631 CY39KP 57398234 Ki = 1600 nM T84631 C83YUW 57398444 IC50 = 53 nM T84631 C9MWA3 57399250 IC50 = 4.8 nM T84631 C49TVR 57399313 IC50 = 121 nM T84631 C7F4ER 57399314 IC50 = 1957 nM T84631 CRQ19W 57399315 IC50 = 209 nM T84631 C5SK3Q 57399481 IC50 = 1110 nM T84631 CODX48 57399879 Ki = 18000 nM T84631 C93VSX 57399880 Ki = 4100 nM T84631 C5WOZ3 57399881 Ki = 3600 nM T84631 CC69OL 57400113 IC50 = 9.1 nM T84631 CUX76O 57400114 IC50 = 2.4 nM T84631 C9ZL5X 57400230 Ki = 1600 nM T84631 CPZR79 57400272 Ki = 6600 nM T84631 CKYJ43 57401018 IC50 = 6.3 nM T84631 CH2AN8 57401242 IC50 = 9750 nM T84631 CS2ZY1 57401658 Ki = 16300 nM T84631 C92EDA 57401914 IC50 = 231 nM T84631 C7F3ET 57401915 IC50 = 4.9 nM T84631 C7SM8P 57401916 IC50 = 2.9 nM T84631 CJ9TH7 57402084 IC50 = 1.2 nM T84631 CH90JO 57402841 IC50 = 130 nM T84631 C6T0ZQ 57402842 IC50 = 14 nM T84631 C0H4UQ 57402934 IC50 = 32 nM T84631 CG90KP 57403382 Ki = 7700 nM T84631 C3CKA6 57403383 Ki = 4400 nM T84631 C4OB6Z 57403384 Ki = 14000 nM T84631 CD0XJ5 57403637 IC50 = 6.9 nM T84631 CDW0N6 57403638 IC50 = 2 nM T84631 CKI4S8 57403776 Ki = 9800 nM T84631 C5MX2D 57404340 IC50 > 50000 nM T84631 C4R2LU 57594784 IC50 = 4.9 nM T84631 C5NC8T 57594789 IC50 = 15 nM T84631 C63FQC 57803696 Ki = 460 nM T84631 CLV91D 57803729 Ki = 4070 nM T84631 CEH39Z 57803776 Ki = 2330 nM T84631 C2W7GY 57803799 Ki = 560 nM T84631 CU4N3X 57803861 Ki = 680 nM T84631 CEG27C 57803875 Ki = 450 nM T84631 CI6U8B 57803906 Ki = 760 nM T84631 C6X3ER 57803948 Ki = 540 nM T84631 CH2QT8 57804013 Ki = 430 nM T84631 C45OXB 57804023 Ki = 2190 nM T84631 CFMO72 57804069 Ki = 430 nM T84631 CTE30K 57842560 Ki = 4800 nM T84631 C0C6UB 57842624 Ki = 3300 nM T84631 C7XY5A 57842673 Ki > 9000 nM T84631 CU9S6K 57842710 Ki = 2600 nM T84631 CL8T7M 57842742 Ki = 610 nM T84631 C41NSR 57842812 Ki = 5500 nM T84631 C9XW1C 57842830 Ki = 5800 nM T84631 CWF0C3 57842850 Ki = 3200 nM T84631 C73CPB 57842913 Ki = 1000 nM T84631 CB5F0H 57942680 Ki = 4500 nM T84631 C8GXF1 57942687 Ki = 6000 nM T84631 CO52PA 57942693 Ki = 6400 nM T84631 CS23DW 57942743 Ki = 5200 nM T84631 C0DO5P 57942817 Ki = 5200 nM T84631 CV0KZ6 57942834 Ki = 3700 nM T84631 C0KRC1 57942835 Ki = 2900 nM T84631 C60HCV 57976401 Ki > 13300 nM T84631 CHB27Y 57976410 Ki = 1128 nM T84631 CM8UJ7 57976444 Ki > 1000 nM T84631 CQ71KE 57976446 Ki = 1500 nM T84631 CXL75F 58630486 Ki > 15000 nM T84631 C3OA5C 58789089 Ki = 3500 nM T84631 C2W1UT 58789135 Ki = 2800 nM T84631 CT9C1Z 58789193 Ki = 8200 nM T84631 C1C8SA 59019689 Ki = 1.5 nM T84631 CP2WM6 59019709 Ki = 0.15 nM T84631 CCM38Z 59020027 Ki = 0.2 nM T84631 C4R9VT 59020061 Ki = 0.05 nM T84631 C7NUC3 59020071 Ki = 1.22 nM T84631 C5ICF9 59020139 Ki = 0.06 nM T84631 CL6EP7 59020154 Ki = 0.48 nM T84631 CSC0L5 59020200 Ki = 0.66 nM T84631 C56MGU 59020231 Ki = 0.05 nM T84631 CDMI79 59020246 Ki = 0.07 nM T84631 CYF20E 59020269 Ki = 9.27 nM T84631 C91APY 59095797 IC50 = 270 nM T84631 C69SED 59095888 IC50 = 1700 nM T84631 CN09MI 59108388 IC50 = 68 nM T84631 C1BHM8 59108407 IC50 = 6.9 nM T84631 CPW2H7 59315536 Ki = 2800 nM T84631 CO38AC 59402011 Ki > 9000 nM T84631 CMU38J 59432238 IC50 = 1.5 nM T84631 CA83BF 59432241 IC50 = 66 nM T84631 C7IO5P 60150643 Ki = 900 nM T84631 C6JP8Q 60154989 Ki = 340 nM T84631 CE5A7B 60162406 Ki > 10000 nM T84631 C8TWY6 66554641 Ki = 6900 nM T84631 CUWT16 66554643 Ki = 0.25 nM T84631 C1W8HF 66554816 Ki = 0.09 nM T84631 CA8L6M 66573468 IC50 = 19000 nM T84631 C2CX0G 66573469 IC50 = 221000 nM T84631 C71CLE 66573471 IC50 = 12800 nM T84631 C8R7DY 66573472 IC50 = 19000 nM T84631 CG0O8A 66573532 IC50 = 20000 nM T84631 CP6JT5 66573533 IC50 = 6000 nM T84631 C6C3MI 66573535 IC50 = 42000 nM T84631 C9N5SP 66573536 IC50 = 56000 nM T84631 C5XP9E 66573589 IC50 = 209000 nM T84631 C8V9FN 66573590 IC50 = 19000 nM T84631 CP30LR 66573591 IC50 = 1300 nM T84631 CWT42D 66573592 IC50 = 14000 nM T84631 CJMT47 66573593 IC50 = 34000 nM T84631 CIR14C 66573637 IC50 = 197000 nM T84631 C2ELC3 66573638 IC50 = 85000 nM T84631 C1XS3L 66573639 IC50 = 335000 nM T84631 CQT4K0 66573640 IC50 = 246000 nM T84631 CTVP01 66573641 IC50 = 18000 nM T84631 C5JOZ8 66573709 IC50 = 900 nM T84631 CEJ02R 66573710 IC50 = 311000 nM T84631 CD86QN 66573711 IC50 = 13300 nM T84631 C2H9VX 66573712 IC50 = 103000 nM T84631 C8VZC9 66573779 IC50 = 1300 nM T84631 CM0DX8 66573780 IC50 = 36000 nM T84631 CKJG43 66573781 IC50 = 1100 nM T84631 CKY92Q 66573782 IC50 = 5400 nM T84631 C27HBF 66573783 IC50 = 190000 nM T84631 CA61DQ 66573843 IC50 > 500000 nM T84631 CZ6N3E 66573844 IC50 = 1600 nM T84631 CWCA65 66573845 IC50 = 270 nM T84631 C8MNG4 66573846 IC50 > 500000 nM T84631 CDL02G 66573847 IC50 = 2900 nM T84631 CH6VF3 66573909 IC50 > 500000 nM T84631 C5N8TC 66573910 IC50 = 151000 nM T84631 CXZ02D 66573911 IC50 > 500000 nM T84631 CY17TB 66573912 IC50 > 500000 nM T84631 CL9B6F 66573973 IC50 = 7800 nM T84631 CT4CR3 66573974 IC50 = 54000 nM T84631 CJG14M 66574033 IC50 > 500000 nM T84631 CR5IJ8 66574034 IC50 = 69000 nM T84631 CPV28L 66574037 IC50 = 371000 nM T84631 C3PV1H 66574099 IC50 = 358000 nM T84631 C5RZE9 66574100 IC50 = 99000 nM T84631 CNG0E4 66574102 IC50 = 23000 nM T84631 CFR0J7 66574158 IC50 = 9000 nM T84631 CBE3G1 66574160 IC50 = 10000 nM T84631 CS1B2I 66574390 IC50 = 9900 nM T84631 C09HIT 66574391 IC50 = 16400 nM T84631 C3LT2W 66674079 Ki > 8180 nM T84631 C23QOJ 66674821 Ki > 8180 nM T84631 CWOD93 66744646 Ki > 13300 nM T84631 CSAQ19 66818162 Ki = 400 nM T84631 C89BXR 66818555 Ki = 300 nM T84631 C9LTK3 66818589 Ki = 600 nM T84631 C41RKZ 66818743 Ki = 1500 nM T84631 CRH5O7 66818889 Ki = 200 nM T84631 CE6JP2 66911194 IC50 = 2.6 nM T84631 CGH09I 66911211 IC50 = 3.4 nM T84631 CKWQ82 67155200 Ki = 1 nM T84631 CY05ND 67155277 IC50 = 145 nM T84631 CA0GE1 67155403 IC50 = 1.1 nM T84631 CN51PD 67155431 IC50 = 1 nM T84631 C0SDB3 68020667 Ki = 7357 nM T84631 C17JAZ 68284084 IC50 > 30000 nM T84631 CE79VS 68440006 Ki = 5400 nM T84631 CA5DG8 69249482 Ki = 1300 nM T84631 CQY32W 69295008 Ki = 7300 nM T84631 CFPM31 69442778 IC50 = 150 nM T84631 C3BFL4 69515911 Ki = 0.07 nM T84631 CL5MN1 69516774 Ki = 0.24 nM T84631 CO7TI8 69516837 Ki = 1.01 nM T84631 CX10QE 69516998 Ki = 0.11 nM T84631 CA49UK 69520512 Ki > 17000 nM T84631 C0KB4O 69641445 Ki > 8000 nM T84631 CO3Z8Y 69654811 Ki > 15000 nM T84631 C6AU1R 70252985 Ki = 840 nM T84631 CTO5I6 70253788 Ki > 3000 nM T84631 C8A7ZJ 70306716 Ki = 45 nM T84631 C0WKD9 70662368 IC50 = 3000 nM T84631 C4IFW3 70683249 Ki = 42 nM T84631 C28CEG 70685001 IC50 = 3 nM T84631 C7U9OA 70687171 IC50 = 80 nM T84631 CN38UY 70687492 Ki = 220 nM T84631 C9EL3C 71260387 Ki = 3660 nM T84631 C28RBT 71449502 IC50 = 3.4 nM T84631 C45SHM 71451304 Ki = 1.5 nM T84631 C15ECT 71451305 IC50 = 2.4 nM T84631 C74KFY 71454853 IC50 = 4 nM T84631 CAM29T 71454854 IC50 = 5.6 nM T84631 C53FKA 71458482 IC50 = 5.4 nM T84631 CX4HG2 71458531 IC50 = 740000 nM T84631 CR1WC4 71461267 IC50 = 6400 nM T84631 C8RPG9 71462026 IC50 = 6.4 nM T84631 CVD3W9 71495381 Ki = 32 nM T84631 CNVH43 71495466 Ki = 170 nM T84631 CA5N2S 71495467 Ki = 260 nM T84631 CQ98NY 71495468 Ki = 1100 nM T84631 CE15GB 71495559 Ki = 3050 nM T84631 CW1Y2L 71495560 Ki = 3200 nM T84631 C5Q9BD 71495561 Ki = 1120 nM T84631 C36MRI 71495659 Ki = 60 nM T84631 C7PDA9 71495660 Ki = 110 nM T84631 CF3C8E 71495661 Ki = 580 nM T84631 CECD13 71495765 Ki = 230 nM T84631 C7LXK1 71495766 Ki = 370 nM T84631 CKQ82B 71495974 Ki = 13900 nM T84631 CSV38K 71495975 Ki = 14100 nM T84631 C7QPA0 71495976 Ki = 16900 nM T84631 CI4P9Z 71495977 Ki = 8890 nM T84631 CE03BA 71496089 Ki = 1200 nM T84631 CLO24G 71496201 Ki = 3410 nM T84631 CIE7A6 71496202 Ki = 2450 nM T84631 CAM0I4 71496204 Ki = 550 nM T84631 CJPF90 71548883 Ki > 9000 nM T84631 C30ZKJ 71561420 Ki = 25000 nM T84631 CH32TL 71561557 Ki = 2510 nM T84631 C83ZNH 71562308 IC50 = 266 ug.mL-1 T84631 C8RW7E 71562631 Ki = 12.3 nM T84631 C4UHB2 71562760 Ki = 415 nM T84631 C0EM6D 71562761 Ki = 237 nM T84631 CNS21T 71562882 Ki = 1260 nM T84631 C3SBE2 71562883 Ki = 8500 nM T84631 C2NY0B 71563006 Ki = 14042 nM T84631 CG46AZ 71563007 Ki = 3700 nM T84631 C2O4SB 71563124 Ki = 9000 nM T84631 C4CT8O 71563125 Ki = 3250 nM T84631 C6I9DJ 71567884 Ki = 650 nM T84631 CC7Z0N 71567885 Ki = 1000 nM T84631 C40CRP 71567886 Ki = 2200 nM T84631 CG8X1C 71567887 Ki > 15000 nM T84631 C5DU6Q 71568014 Ki = 1100 nM T84631 C4ICT8 71568015 Ki = 3700 nM T84631 C9BSO1 71568137 Ki = 290 nM T84631 C9TBN3 71568263 Ki > 15000 nM T84631 CXYQ68 71568403 Ki > 15000 nM T84631 C53BYN 71580813 Ki = 16 nM T84631 C57PCL 71580892 Ki = 1500 nM T84631 CRD4I9 71625797 Ki > 25000 nM T84631 CG1V9P 71627416 Ki > 8000 nM T84631 C9J7NH 71652207 Ki = 5080 nM T84631 CLH52G 71654374 Ki = 2150 nM T84631 C8GDV7 71654376 Ki = 1510 nM T84631 CY29LR 71654530 Ki = 637 nM T84631 C3K6PT 71654532 Ki = 2700 nM T84631 C3X7FP 71654534 Ki = 5190 nM T84631 CCGP56 71654535 Ki = 1960 nM T84631 CZG3Y9 71654536 Ki = 1270 nM T84631 C62ZTJ 71660643 IC50 > 33000 nM T84631 C5D2OL 71698598 Ki = 54400 nM T84631 CGYN76 71698686 Ki = 49300 nM T84631 CD0Z5K 71698687 Ki = 28700 nM T84631 C0DUT2 71698688 Ki = 38200 nM T84631 C60JTA 71698689 Ki = 55600 nM T84631 C35ZJV 71698690 Ki = 111000 nM T84631 C9XSB5 71698770 Ki = 48800 nM T84631 CRN95M 71698771 Ki = 47500 nM T84631 C0LW4G 71698774 Ki = 11200 nM T84631 CH26JR 71698775 Ki = 88200 nM T84631 C0WR9F 71699124 Ki > 100000 nM T84631 CZKL39 71699125 Ki > 100000 nM T84631 C27TZK 71699126 Ki = 34300 nM T84631 CD12FS 71699127 Ki = 25600 nM T84631 CFN7Q4 71699199 Ki = 43000 nM T84631 C7RTF0 71699200 Ki = 62900 nM T84631 C8JE0W 71699201 Ki = 54100 nM T84631 CRAG19 71699203 Ki = 10800 nM T84631 CYAH23 71699286 Ki = 82300 nM T84631 CM8E7F 71699287 Ki = 37000 nM T84631 C9Y3DN 71699288 Ki = 57700 nM T84631 C78DJQ 71711730 IC50 < 10000 nM T84631 CQ3K2V 71719191 Ki = 1803 nM T84631 C4TP1M 71748092 Ki = 1800 nM T84631 CVM7Y6 71748093 Ki = 4400 nM T84631 C8HZ6Q 71748094 Ki = 3700 nM T84631 C6CB0G 71748095 Ki = 3900 nM T84631 C2Z7XJ 71748113 Ki = 3100 nM T84631 CM83VP 72163524 IC50 > 10000 nM T84631 CRBH34 72164200 IC50 > 33000 nM T84631 CWNZ45 72164201 IC50 > 33000 nM T84631 CBVO02 72164443 Ki > 8000 nM T84631 C1W9NH 72164444 Ki > 8000 nM T84631 C6Z3IC 72164445 Ki > 8000 nM T84631 C0CGB5 72164564 Ki > 8000 nM T84631 CN37EY 72164565 Ki = 8200 nM T84631 CIT3O5 72164566 Ki > 8000 nM T84631 C80OFE 72164567 Ki > 8000 nM T84631 CD01PR 72164568 Ki > 8000 nM T84631 C85RCG 72164697 Ki = 7000 nM T84631 CP4M2G 72164698 Ki = 7200 nM T84631 C0EWD8 72164699 Ki = 5600 nM T84631 C9G4PK 72200999 IC50 = 0.5 nM T84631 CG8Z7P 72206621 IC50 = 0.2 nM T84631 CK34ZH 72550138 Ki = 6200 nM T84631 CT45ER 72550807 Ki = 3900 nM T84631 C46TNC 72550811 Ki = 4300 nM T84631 CXM6C2 72550813 Ki = 6650 nM T84631 CLI36U 72551247 Ki = 4000 nM T84631 C7OF4T 72711856 Ki = 57300 nM T84631 C4Z2RL 72711858 Ki > 250000 nM T84631 C14KIG 72711859 Ki = 47100 nM T84631 CN08OJ 72711860 Ki = 91600 nM T84631 C0BCJ7 72711861 Ki = 78000 nM T84631 C4CG6J 72711863 Ki = 63500 nM T84631 C8NCB1 72712043 Ki = 7460 nM T84631 CIO50P 72712044 Ki > 250000 nM T84631 CK4H1G 72712045 Ki = 25100 nM T84631 CDY10L 72712046 Ki = 3830 nM T84631 CH9MT7 72712048 Ki = 23600 nM T84631 CW3QR2 72712049 Ki = 1100 nM T84631 CAL2W7 72712050 Ki = 5640 nM T84631 C2A4TH 72712051 Ki = 6830 nM T84631 CJX7H1 72712052 Ki = 8800 nM T84631 CN73TI 72712053 Ki = 27000 nM T84631 C7W6OH 72712054 Ki = 29600 nM T84631 CT1F6W 72712055 Ki > 250000 nM T84631 CK6BL5 72712056 Ki = 37100 nM T84631 C8L3AV 72712057 Ki = 6310 nM T84631 C6NB1T 72712058 Ki = 6000 nM T84631 C2ZKR0 72712059 Ki = 6730 nM T84631 CZ80WI 72712060 Ki = 7730 nM T84631 C2CBY8 72712061 Ki = 15600 nM T84631 C0U7QR 72712062 Ki = 35100 nM T84631 CB0F1O 72712063 Ki = 48500 nM T84631 CAQ0T5 72712064 Ki = 25000 nM T84631 CS0PO5 72712065 Ki = 36100 nM T84631 CM8QC1 72712066 Ki = 12200 nM T84631 C0YW7A 72712067 Ki = 11100 nM T84631 CHJ25Y 72712068 Ki = 7230 nM T84631 CP4BS0 72712069 Ki = 16400 nM T84631 C3J8RV 72712070 Ki = 606 nM T84631 CQI5T2 72712071 Ki = 37700 nM T84631 COQ58Y 72712072 Ki = 44100 nM T84631 CU4I2F 72712250 Ki = 126000 nM T84631 C64SNL 72712251 Ki = 3720 nM T84631 CI2E4L 72712252 Ki = 133 nM T84631 C9BX1Q 72712253 Ki = 2140 nM T84631 CC73NU 72712254 Ki = 774 nM T84631 CF80WL 72712255 Ki > 250000 nM T84631 CAZ5R4 72725806 Ki = 3000 nM T84631 CPW7T3 72725807 Ki = 57 nM T84631 CM1OK7 72792543 IC50 = 39 nM T84631 CBP05V 72792607 IC50 = 13 nM T84631 CYXT24 72792608 IC50 = 0.6 nM T84631 CO89NF 72792609 IC50 = 0.5 nM T84631 CC50RS 72792610 IC50 = 1 nM T84631 CCEZ71 72792672 IC50 = 3.4 nM T84631 CFRI96 72792673 IC50 = 1.2 nM T84631 C86RTS 72792674 IC50 = 1.4 nM T84631 CI5U3J 72792675 IC50 = 1.4 nM T84631 CQ08NT 72792744 IC50 = 1.9 nM T84631 CWB62R 72792745 IC50 = 2.99 nM T84631 CA8WG3 72792746 IC50 = 1.8 nM T84631 CR17NL 72792747 IC50 = 1.1 nM T84631 CW84BZ 73345684 IC50 = 100 nM T84631 CT21AC 73345685 IC50 = 224 nM T84631 C4FQ0W 73345765 Ki > 6000 nM T84631 CCD54H 73345766 Ki > 6000 nM T84631 CO4A1M 73345767 Ki > 6000 nM T84631 CC2FW1 73345771 Ki > 6000 nM T84631 C3JN8A 73347180 IC50 = 550 nM T84631 CQF46R 73348759 Ki > 6000 nM T84631 CJG30R 73348764 Ki = 4200 nM T84631 CUD26E 73348765 Ki > 6000 nM T84631 CSQ41U 73348767 Ki = 760 nM T84631 C7Y3ZB 73348933 Ki = 88.7 nM T84631 CAJ7O5 73350148 Ki > 1000000 nM T84631 CYL2K9 73350270 IC50 = 167 nM T84631 C1EPR4 73350271 IC50 = 220 nM T84631 CHF47P 73350338 Ki > 6000 nM T84631 C5VP6W 73350339 Ki > 6000 nM T84631 CK45HD 73350340 Ki = 4900 nM T84631 C60BNQ 73350342 Ki > 6000 nM T84631 CL8EG7 73350757 Ki = 2250 nM T84631 C36EPY 73351772 IC50 = 12000 nM T84631 COBX03 73351777 IC50 = 2000 nM T84631 C2NEV3 73351853 Ki > 6000 nM T84631 CX1WJ7 73351856 Ki = 1600 nM T84631 C4CD7U 73351857 Ki > 6000 nM T84631 C69BHN 73353326 Ki > 6000 nM T84631 C26QPS 73353327 Ki > 6000 nM T84631 C7DGZ9 73353328 Ki > 6000 nM T84631 CA2P1B 73353330 Ki > 6000 nM T84631 CPS6J3 73354766 IC50 = 1000 nM T84631 CNRW95 73354848 Ki > 6000 nM T84631 COF2K0 73354849 Ki > 6000 nM T84631 C3VFD6 73354850 Ki = 4300 nM T84631 CL34CV 73354863 Ki > 6000 nM T84631 C5U9CI 73355715 Ki = 0.0042 nM T84631 CXG0B8 73356296 IC50 = 230 nM T84631 C8N4RM 73356390 Ki = 6000 nM T84631 C5MVT3 76310068 Ki = 1200 nM T84631 CH1BJ2 76311085 Ki = 970 nM T84631 C9OKI1 76311087 Ki = 1140 nM T84631 CZU72O 76311088 Ki = 3980 nM T84631 CE3ZI8 76311089 Ki = 6700 nM T84631 C29QNE 76311090 Ki = 4100 nM T84631 C3R8LG 76311091 Ki = 2250 nM T84631 CD4AZ2 76311332 Ki = 769 nM T84631 CSBD17 76314701 Ki = 5810 nM T84631 C6FQ0C 76314925 Ki = 62.2 nM T84631 C9J0BH 76317785 Ki = 9000 nM T84631 C9C4BV 76317871 Ki = 14000 nM T84631 CSY3T8 76318271 Ki = 1940 nM T84631 CI7MO1 76318272 Ki > 15000 nM T84631 C28QGR 76318273 Ki = 6400 nM T84631 C4WUP1 76318274 Ki = 8350 nM T84631 CWZA05 76320988 Ki = 100 nM T84631 C9PJ1H 76321975 Ki = 2060 nM T84631 C7UP8I 76321976 Ki = 641 nM T84631 CP1MR4 76322205 Ki = 21.9 nM T84631 CO28RN 76325189 Ki = 8000 nM T84631 CHNJ05 76325595 Ki = 1100 nM T84631 C6UR1G 76325596 Ki = 24 nM T84631 CDB4R0 76325821 Ki = 62.4 nM T84631 CJ10YI 76328088 IC50 = 3500 nM T84631 C3W5PN 76329159 Ki = 9300 nM T84631 CJ9D8H 76329160 Ki = 880 nM T84631 C6CW8M 76332426 Ki > 43000 nM T84631 CL09IJ 76332819 Ki = 130 nM T84631 CXKG18 76332820 Ki > 15000 nM T84631 CYCA26 76332821 Ki = 1480 nM T84631 CADC95 76336441 Ki = 606 nM T84631 CZ4N5I 76336442 Ki = 1310 nM T84631 C7TNX2 76336443 Ki = 1810 nM T84631 CO54FL 76336676 Ki = 337 nM T84631 C10OJP 76336677 Ki = 1220 nM T84631 CAT95V 76685067 IC50 = 3.41 nM T84631 CMD5V7 86583041 Ki > 9000 nM T84631 CWP85J 87360663 IC50 > 10000 nM T84631 CO6U9I 88582319 Ki = 200 nM T84631 CMC3L7 89399327 Ki = 2610 nM T84631 CKR2A0 90295536 IC50 = 590 nM T84631 C9FDP4 90295556 IC50 = 2510 nM T84631 CM3LT0 90295602 IC50 = 46.64 nM T84631 CSJY38 90295614 IC50 = 57.81 nM T84631 CQ6D0F 90295617 IC50 > 100000 nM T84631 C7OL1W 90295621 IC50 = 130 nM T84631 CD8O6C 90295622 IC50 > 100000 nM T84631 CNOB68 90295624 IC50 = 1220 nM T84631 C9ZC5G 90295630 IC50 = 40.56 nM T84631 C7B6FC 90295663 IC50 = 1860 nM T84631 C8YCR2 90295664 IC50 = 730 nM T84631 CE09FR 90295757 IC50 = 87.17 nM T84631 C97WGT 90295764 IC50 = 190 nM T84631 C6SK4I 90664135 IC50 > 1000 ug.mL-1 T84631 CE60BJ 90664137 IC50 > 1000 ug.mL-1 T84631 CYB39G 90664139 IC50 > 1000 ug.mL-1 T84631 C6KU0A 90664141 IC50 > 1000 ug.mL-1 T84631 C0T4MS 90665251 IC50 > 1000 ug.mL-1 T84631 CD53HR 90665253 IC50 > 1000 ug.mL-1 T84631 C1SAZ8 90666139 Ki = 180 nM T84631 C2ERV8 90666140 Ki = 7070 nM T84631 CSO5R7 90666141 Ki = 4790 nM T84631 C3F0PB 90666142 Ki = 6450 nM T84631 CG1W0R 90666143 Ki = 5520 nM T84631 CI3AX1 90666144 Ki = 51 nM T84631 C43YWM 90666145 Ki = 29 nM T84631 CT45NA 90666146 Ki = 11 nM T84631 C56KQL 90666147 Ki = 20 nM T84631 COH41Y 91666660 Ki = 1400 nM T84631 CUC01L 91799239 Ki = 105 nM T84631 CA90QH 91827690 IC50 = 380 nM T84631 CE28SQ 91972030 IC50 > 100000 nM T84631 CISE50 101353098 IC50 = 7165 nM T84631 C6A3ZK 101886607 Ki = 11600 nM T84631 CTG2Q1 117987029 IC50 = 60.56 nM T84631 C4G7NE 117987044 IC50 = 2210 nM T84631 C3PS6Y 118098650 Ki = 1800 nM T84631 CYH43T 118456915 IC50 > 100000 nM T84631 CM39QL 118456920 IC50 > 100000 nM T84631 C1C3HV 118456930 IC50 > 30000 nM T84631 CKST03 118456931 IC50 = 25000 nM T84631 C4CJM6 118456935 IC50 > 100000 nM T84631 C6EJB5 118456946 IC50 > 100000 nM T84631 C6ZS9A 118456950 IC50 > 100000 nM T84631 CQ43TO 118456975 IC50 = 29000 nM T84631 CL4K5X 118456998 IC50 > 100000 nM T84631 CCR4Y5 118457019 IC50 > 100000 nM T84631 C26CAL 118457021 IC50 > 100000 nM T84631 COY1V8 118457032 IC50 = 22000 nM T84631 CWY2B9 118457044 IC50 = 26000 nM T84631 CS05DP 118457052 IC50 > 100000 nM T84631 CO72PX 118519577 IC50 = 88.53 nM T84631 CFCN48 118519579 IC50 = 20.22 nM T84631 C1FG2P 118519580 IC50 = 1750 nM T84631 C28MKY 118519581 IC50 > 100000 nM T84631 C21COH 118519584 IC50 = 8080 nM T84631 C52CRZ 118519585 IC50 = 74.77 nM T84631 C5X2KG 118519586 IC50 = 25880 nM T84631 CH1ON2 118519588 IC50 > 100000 nM T84631 CVJ3D6 118519593 IC50 = 32.08 nM T84631 CGA28Y 118519594 IC50 = 5530 nM T84631 CH8B3W 118519596 IC50 = 160 nM T84631 CWH39U 118519597 IC50 = 52690 nM T84631 CVEF90 118519598 IC50 = 11360 nM T84631 CZ8N3W 118519604 IC50 > 100000 nM T84631 C3TB4X 118519607 IC50 = 4180 nM T84631 CLE03N 118519608 IC50 = 710 nM T84631 CXK35R 118519612 IC50 > 100000 nM T84631 C46MSP 118542774 Ki = 740 nM T84631 C20WBY 118542785 Ki = 240 nM T84631 CI65YK 118542879 Ki = 200 nM T84631 CEH93P 118542958 Ki = 250 nM T84631 CITU59 118548755 Ki = 750 nM T84631 CMF5R6 118548758 Ki = 850 nM T84631 C1IH2W 118548759 Ki = 1230 nM T84631 C6LZQ3 118548760 Ki = 510 nM T84631 C62ZNW 118548761 Ki = 610 nM T84631 C3WQ9D 118548776 Ki = 1550 nM T84631 CU01RP 118548813 Ki = 660 nM T84631 C2N1YG 118574661 IC50 = 560 nM T84631 CAB58Q 118574662 IC50 = 310 nM T84631 CK75GJ 118574663 IC50 = 37.65 nM T84631 CW82NL 118574664 IC50 = 15770 nM T84631 C3IU6A 118574693 IC50 = 1210 nM T84631 CIU5Z9 118584716 IC50 = 7060 nM T84631 C51RJX 118707613 Ki = 0.32 nM T84631 CM7GL3 118713017 IC50 = 4780 nM T84631 CKS29X 118713018 IC50 = 2.51 nM T84631 CNA91K 118713019 IC50 = 4.89 nM T84631 CV0Y1I 118713020 IC50 = 45.22 nM T84631 C9SK5T 118713021 IC50 = 63.96 nM T84631 CUN3T1 118713022 IC50 = 17.37 nM T84631 C9OU4J 118713023 IC50 = 50.52 nM T84631 C1Z7LV 118713024 IC50 = 20.87 nM T84631 CEJ56B 118713025 IC50 = 1610 nM T84631 CRF62H 118713026 IC50 = 4.71 nM T84631 CY9KW3 118713027 IC50 = 6.59 nM T84631 CRA2J1 118713028 IC50 = 8180 nM T84631 CAS3L5 118713029 IC50 = 5.06 nM T84631 CFHP98 118713030 IC50 = 15.2 nM T84631 CUS29V 118716986 Ki = 18300 nM T84631 C0GRU4 118718129 Ki = 3.1 nM T84631 C3MVG0 118720988 Ki > 8180 nM T84631 C9M2IH 118720990 Ki > 8180 nM T84631 C1E6GW 118720991 Ki > 8180 nM T84631 C9BVI5 118720993 Ki > 8180 nM T84631 C1FQZ6 118720994 Ki > 9000 nM T84631 C0WZA2 118720996 Ki > 8180 nM T84631 CE89KB 118720997 Ki > 8180 nM T84631 CIAL50 118720998 Ki > 8180 nM T84631 C4HLM3 118720999 Ki > 8180 nM T84631 CLD6I3 118721000 Ki > 8180 nM T84631 C0XG7H 118721001 Ki > 8180 nM T84631 CZC53M 118721002 Ki > 8180 nM T84631 C8FZ2L 118721003 Ki > 8180 nM T84631 C0M4IQ 118721004 Ki > 9000 nM T84631 CLRB29 118721005 Ki = 1370 nM T84631 C9B1FX 118721007 Ki > 8180 nM T84631 CRV5Y1 118721008 Ki = 6390 nM T84631 CH6AQ9 118721009 Ki > 8180 nM T84631 CI7YD4 118723652 IC50 = 140 nM T84631 C7ZX1R 118723654 IC50 = 61 nM T84631 CC5L2H 118723655 IC50 = 68 nM T84631 CSE75C 118723704 IC50 = 220 nM T84631 CA41EG 118723706 IC50 = 290 nM T84631 CC52MF 118723708 IC50 = 16 nM T84631 CTF5U9 118723709 IC50 = 3.6 nM T84631 C4U2AW 118723894 IC50 = 352000 nM T84631 CV5JG3 118723904 IC50 = 195000 nM T84631 CP98JL 118723906 IC50 = 229000 nM T84631 C0UO7Q 118723908 IC50 = 344000 nM T84631 C3IA9S 118726913 IC50 = 13 nM T84631 CABH86 118726934 IC50 = 18 nM T84631 COB7H3 118731959 IC50 = 27 nM T84631 CR67JK 118731960 Ki = 90 nM T84631 CMKI65 118731961 IC50 = 298 nM T84631 C4O2IH 118731962 IC50 = 1120 nM T84631 C8OC5Y 118731963 IC50 = 798 nM T84631 C17ARY 118731964 IC50 = 621 nM T84631 CR4O3V 118731965 IC50 = 452 nM T84631 C7Q0EA 118731966 IC50 = 678 nM T84631 CUQ32B 118731967 IC50 = 828 nM T84631 CCV65S 118731968 IC50 = 612 nM T84631 CW5ZV9 118731969 IC50 = 67 nM T84631 CGQW74 118731970 IC50 = 521 nM T84631 CO5X2B 118731971 IC50 = 23 nM T84631 C34UOK 118731972 IC50 = 183 nM T84631 CDX2R9 118731973 IC50 = 286 nM T84631 CYN2A9 118731974 IC50 = 378 nM T84631 C60SWE 118733712 IC50 = 610 nM T84631 C17VDS 118733713 IC50 = 2.01 nM T84631 CWRX39 118733714 IC50 = 1310 nM T84631 C7OU0X 118733715 IC50 = 1420 nM T84631 C1LK8Q 118733716 IC50 = 2620 nM T84631 CN25YW 118733717 IC50 = 2930 nM T84631 CXUG54 118733718 IC50 = 3220 nM T84631 C2YF0P 118733719 IC50 = 3800 nM T84631 COH5X2 118733720 IC50 = 6.58 nM T84631 CO8B5R 118733721 IC50 = 3.25 nM T84631 CV04QG 118733722 IC50 = 2210 nM T84631 C9AVB2 118733723 IC50 = 1830 nM T84631 CU36GW 118733724 IC50 = 1510 nM T84631 C64ALF 118733725 IC50 = 3060 nM T84631 CA8HY2 118733726 IC50 = 5780 nM T84631 CH2EA0 118733727 IC50 = 5320 nM T84631 CKUY41 118733728 IC50 = 10120 nM T84631 CU6F3L 118733729 IC50 = 11020 nM T84631 CY2Z4Q 118733730 IC50 = 10450 nM T84631 CJ5HT0 118733731 IC50 = 11290 nM T84631 C9P2UN 118733732 IC50 = 1870 nM T84631 C0SBJ9 118733733 IC50 = 870 nM T84631 C9YI0Z 118733734 IC50 = 650 nM T84631 CLKN48 118733735 IC50 = 9.46 nM T84631 CQ84KH 118733736 IC50 = 2420 nM T84631 CVYW12 118733737 IC50 = 2720 nM T84631 CW64OQ 118733738 IC50 = 3030 nM T84631 CY0JV9 118733739 IC50 = 3850 nM T84631 CZW8Q0 118733740 IC50 = 3600 nM T84631 CPH87E 118736125 Ki > 62500 nM T84631 C32KLW 118736129 Ki = 12000 nM T84631 CPN2Q3 118736138 Ki = 390 nM T84631 CHQ5P7 118987013 Ki > 9000 nM T84631 CRI9U5 121399126 Ki = 245 nM T84631 CNXI35 121399185 Ki > 28890 nM T84631 CNF2P3 121399230 Ki > 28890 nM T84631 CPHN78 121399237 Ki = 2473 nM T84631 C2TIC0 121399249 Ki > 28890 nM T84631 C3F7RH 121399265 Ki = 340 nM T84631 CV9TX1 121399281 Ki = 2798 nM T84631 C1ZYC9 121399296 Ki = 195 nM T84631 C4Q0HT 121399308 Ki = 544 nM T84631 C2WD1Q 121407246 Ki = 20720 nM T84631 C3WC9Y 121488127 IC50 = 72000 nM T84631 C3YVQ8 122164611 Ki = 850 nM T84631 CY1S5D 122164612 Ki = 900 nM T84631 CKJN32 122164799 IC50 > 30000 nM T84631 CCE7R9 122187957 IC50 = 17.1 nM T84631 CWV2C7 122187958 IC50 = 28.6 nM T84631 CDH51U 122187961 IC50 = 25.9 nM T84631 CT2Q7L 122187963 IC50 = 15.6 nM T84631 CQ2W6H 122187967 IC50 = 6.5 nM T84631 C9KL5N 122192970 Ki = 412 nM T84631 C6SAE8 122192971 Ki = 1010 nM T84631 CZQ6W3 122192972 Ki = 1507 nM T84631 CX7K5B 122192988 Ki = 15160 nM T84631 C1MVP5 122192989 Ki = 1932 nM T84631 CLHV68 122192990 Ki > 28890 nM T84631 CXU4S3 122193791 Ki = 2259 nM T84631 C23NAU 122193792 Ki = 2145 nM T84631 CX79CM 122193793 Ki = 662 nM T84631 C9ASN2 122193794 Ki = 2036 nM T84631 C9Y6SO 122193795 Ki = 28890 nM T84631 CX9T3D 122193796 Ki = 10710 nM T84631 C2FS4M 122193797 Ki = 4227 nM T84631 COMK61 122193798 Ki = 1006 nM T84631 CZL3W8 122193799 Ki = 258 nM T84631 C90QDF 122193800 Ki = 605 nM T84631 CGQA72 122193881 Ki = 378 nM T84631 C9WT4R 122193882 Ki = 246 nM T84631 CSB1Q5 122193883 Ki = 1682 nM T84631 C9BLF1 122193884 Ki = 1553 nM T84631 CM0TS7 122193885 Ki = 1110 nM T84631 CLI82V 122193886 Ki = 1540 nM T84631 CEN5J7 122193887 Ki = 743 nM T84631 CIJ85X 122193888 Ki = 590 nM T84631 C13UCF 122193889 Ki = 518 nM T84631 CJS68F 122193891 Ki = 1748 nM T84631 CTGN19 122193892 Ki = 1416 nM T84631 C62TVJ 122193893 Ki = 3283 nM T84631 CQO8Z9 122193894 Ki = 1082 nM T84631 C9K8SJ 122193895 Ki = 193 nM T84631 C5R8SG 122193896 Ki = 397 nM T84631 C5LR2A 122193897 Ki > 5000 nM T84631 CH2VR6 122193898 Ki = 337 nM T84631 CI6HC5 122193899 Ki = 507 nM T84631 COZP50 122193900 Ki = 257 nM T84631 CH46TB 122194031 Ki = 5315 nM T84631 CGD97N 122194032 Ki = 1035 nM T84631 C6HX9J 122194033 Ki = 234 nM T84631 CN76EH 122194035 Ki = 1053 nM T84631 CU6QD5 122194036 Ki = 409 nM T84631 CR7MG0 122224465 IC50 > 250000 nM T84631 CAI69W 123238067 Ki = 920 nM T84631 C76BAD 123424620 Ki = 180 nM T84631 CK0W2P 127027635 Ki > 9000 nM T84631 CJ6DA9 127028140 IC50 > 10000 nM T84631 CD9KI3 127028141 IC50 > 10000 nM T84631 CPC0M8 127031390 Ki > 9000 nM T84631 CA30BN 127033248 Ki = 25500 nM T84631 CO7PY0 127033521 Ki = 49400 nM T84631 CE0QZ4 127033522 Ki = 22800 nM T84631 C7ZIR9 127034099 Ki = 400 nM T84631 CN4U9B 127037807 IC50 = 51580 nM T84631 C85ROH 127041472 IC50 > 100000 nM T84631 C4T9KU 127045502 Ki = 6800 nM T84631 C4RFP7 127045503 Ki > 13300 nM T84631 C2IOG9 127045504 Ki > 13300 nM T84631 CHK80O 127045505 Ki > 13300 nM T84631 CL6W5N 127045506 Ki > 13300 nM T84631 CE26HW 131955087 IC50 = 71000 nM T84631 CWQ14N 132578544 IC50 = 150 nM T84631 CPSU28 132938122 IC50 = 140 nM T84631 CT2RV6 134130781 IC50 > 1000000 nM T84631 CWV3G6 134131077 IC50 > 200000 nM T84631 CS8FV1 134131084 IC50 > 200000 nM T84631 C92RTL 134131303 IC50 > 200000 nM T84631 CL37SG 134131589 IC50 > 200000 nM T84631 CPQ04R 134132204 Ki > 10000 nM T84631 CC7UO1 134133660 Ki = 1400 nM T84631 C6DPW7 134141496 Ki > 9000 nM T84631 CIRU10 134145163 Ki = 2000 nM T84631 CHA7X9 134146314 Ki = 2500 nM T84631 C9UZI0 134148669 Ki = 3000 nM T84631 CTG65U 134148771 Ki = 1000 nM T84631 CNR48I 134149150 IC50 = 2400 nM T84631 CR6V9U 134150310 Ki = 1050 nM T84631 CNAR93 134150771 IC50 = 1990 nM T84631 C3QEO5 134151811 Ki = 4800 nM T84631 CJZ50O 134153212 IC50 = 2400 nM T84631 CG9UL4 134156593 Ki = 1800 nM T84631 C9JF0Q 134157000 IC50 = 850 nM T84631 CYJ61L 134157128 IC50 = 350 nM T84631 CD06PE 134313025 IC50 = 3800 nM T84631 C6HTD5 135393470 IC50 > 50000 nM T84631 C7NA6E 135393474 IC50 > 50000 nM T84631 CBW03G 135404142 Ki = 810 nM T84631 C8GE5V 135404808 Ki = 8 nM T84631 CD53CZ 135404951 Ki = 0.75 nM T84631 C9YUQ1 135405121 Ki = 0.07 nM T84631 C9SY8U 135406499 Ki = 26 nM T84631 CQEZ96 135406539 Ki = 983 nM T84631 C94GZP 135406646 Ki = 0.31 nM T84631 CP7Z3S 135407592 Ki = 13 nM T84631 C5XA6H 135407717 Ki = 9400 nM T84631 C0OX6T 135407736 Ki = 7800 nM T84631 CA8X0V 135409826 Ki = 3 nM T84631 CD48MU 135415156 Ki = 3.1 nM T84631 CNIE32 135426905 Ki = 0.41 nM T84631 CK1AD7 135426949 Ki = 0.71 nM T84631 C61XOA 135427245 Ki = 16000 nM T84631 CL25SO 135427324 Ki = 8.4 nM T84631 C2I6WX 135430716 Ki = 320 nM T84631 CHMD42 135431470 Ki = 3500 nM T84631 C8WS4O 135443730 Ki = 16000 nM T84631 CTP5V8 135444609 Ki = 2100 nM T84631 C3SMN4 135444666 IC50 = 0.7 nM T84631 C4M5BF 135450980 Ki > 75000 nM T84631 CKA3D2 135451808 Ki = 0.26 nM T84631 C9KLD3 135455964 Ki = 2 nM T84631 CSK06Y 135456121 Ki = 5 nM T84631 CJWC64 135462427 Ki = 3 nM T84631 CXS6B9 135471524 Ki = 5000 nM T84631 C5PO0Q 135471605 Ki = 78 nM T84631 CU8IC7 135474643 Ki = 6 nM T84631 C2PFI8 135475618 Ki = 1300 nM T84631 CI8Z4U 135479981 Ki = 23 nM T84631 C50EKI 135484100 Ki = 0.28 nM T84631 C37PHT 135487779 IC50 = 4.4 nM T84631 CBE9G0 135490854 Ki = 9900 nM T84631 CZGI04 135490911 Ki = 12 nM T84631 C9T1IA 135492878 Ki > 5000 nM T84631 CRNB95 135492887 Ki > 5000 nM T84631 C9TA2B 135501173 Ki = 0.33 nM T84631 CO5UV8 135501194 Ki = 0.43 nM T84631 CMQ6O0 135501618 Ki = 10000 nM T84631 C47UGJ 135503965 Ki = 3 nM T84631 CVA61N 135512760 Ki = 5700 nM T84631 CLO72H 135514651 Ki = 0.42 nM T84631 CP51ZM 135515290 Ki = 0.24 nM T84631 CW7TI2 135515464 Ki = 29 nM T84631 C3MLP1 135517489 Ki = 106 nM T84631 CSW47P 135528873 Ki = 2700 nM T84631 CW9YX8 135530632 Ki = 5.7 nM T84631 CET9Q2 135530746 Ki = 0.5 nM T84631 C4OW8A 135531345 Ki = 0.65 nM T84631 CK97FT 135533257 Ki = 940 nM T84631 CAD75F 135535997 Ki = 30000 nM T84631 C3E4CU 135537603 Ki = 1.2 nM T84631 C67TIA 135544099 IC50 = 2.2 nM T84631 CDT59O 135544137 Ki = 2 nM T84631 CCH49A 135544551 Ki = 890 nM T84631 CKLD47 135544579 Ki = 25000 nM T84631 CSO35D 135546147 Ki = 85 nM T84631 C5RG6Z 135546170 Ki = 2.4 nM T84631 CD9AO5 135548205 Ki = 9 nM T84631 C7Q9YK 135559071 Ki > 150000 nM T84631 CAU8S4 135559072 Ki > 150000 nM T84631 C9D1MQ 135581665 Ki = 44 nM T84631 CB6L5Y 135581668 Ki = 0.1 nM T84631 C5ZFS3 135581673 Ki = 0.34 nM T84631 CYG47F 135581674 Ki = 3 nM T84631 C94JBX 135581677 Ki = 18.5 nM T84631 C05ONT 135581679 Ki = 7.3 nM T84631 CUL71O 135581680 Ki = 0.1 nM T84631 C5YW3X 135581684 Ki = 0.58 nM T84631 CC72AJ 135610111 Ki = 51 nM T84631 C09QFL 135667566 Ki = 10 nM T84631 CR82IN 135677712 Ki = 62 nM T84631 CUX2R7 135677713 Ki = 9.7 nM T84631 C58PSA 135740053 Ki = 1.1 nM T84631 C4VL1K 135740054 Ki = 0.4 nM T84631 CZL58Y 135740055 Ki = 2.2 nM T84631 CR05YT 135740056 Ki = 2 nM T84631 C2O7PT 135740057 Ki = 0.25 nM T84631 C6MZP7 135763271 Ki = 59 nM T84631 C68GTN 135763273 Ki = 61 nM T84631 C91UXW 135802775 Ki = 7 nM T84631 C0AX3J 135802853 Ki = 81 nM T84631 CRB42G 135802854 Ki = 19 nM T84631 CQD2Z1 135855944 Ki = 0.5 nM T84631 C5ZL2K 135857416 IC50 = 1.4 nM T84631 CMJ0B6 135962022 Ki = 58 nM T84631 CUV6M0 135972471 IC50 = 511 nM T84631 CC54EI 135986123 IC50 = 1.5 nM T84631 C9G7TE 135995982 Ki = 10 nM T84631 C78ZVN 136000585 Ki = 1000 nM T84631 CRG5N4 136000680 Ki = 3.162 nM T84631 C1OXJ5 136029174 Ki = 810 nM T84631 C6S5OL 136034781 Ki = 94000 nM T84631 CPSO31 136045813 Ki = 100 nM T84631 CL1K8S 136045814 Ki = 27 nM T84631 C5KO1C 136045815 Ki = 59 nM T84631 C2MDW7 136045816 Ki = 7300 nM T84631 CJIP97 136045817 Ki = 14 nM T84631 C39YHK 136045818 Ki = 7000 nM T84631 CZE5Y4 136045819 Ki = 3700 nM T84631 CT2UQ9 136045820 Ki > 10000 nM T84631 C1S4QD 136045821 Ki = 3500 nM T84631 CYQ70K 136053621 IC50 = 3.5 nM T84631 C46VRO 136058172 Ki = 20 nM T84631 C6Q4FB 136058174 Ki = 37 nM T84631 C34UZI 136058175 Ki = 12 nM T84631 CUX79V 136058176 Ki = 38 nM T84631 CBY56D 136058177 Ki = 254 nM T84631 C4YO6Q 136058178 Ki = 181 nM T84631 CB39EK 136058180 Ki = 51 nM T84631 C8PLB3 136058181 Ki = 88 nM T84631 CSU6X4 136058182 Ki = 184 nM T84631 C0Y3CA 136058183 Ki = 2 nM T84631 C8IH1Z 136058184 Ki = 9 nM T84631 C4LG7S 136058185 Ki = 131 nM T84631 CCX30L 136058186 Ki = 5 nM T84631 C6KG8F 136058187 Ki = 128 nM T84631 CHS25L 136058188 Ki = 19 nM T84631 C8G4TI 136066129 Ki = 0.84 nM T84631 CY6XD7 136066130 Ki = 8.1 nM T84631 CN70IU 136092208 Ki > 75000 nM T84631 C5N3KP 136092209 Ki = 38000 nM T84631 C1BUH6 136092210 Ki = 125000 nM T84631 CFQ2C8 136092211 Ki = 38000 nM T84631 CX5R9J 136092212 Ki = 83000 nM T84631 C35PXN 136092213 Ki = 32000 nM T84631 CEXJ30 136092214 Ki = 41000 nM T84631 CS6QH0 136092215 Ki = 43000 nM T84631 CMR7L4 136092216 Ki = 167000 nM T84631 CN0WR7 136092217 Ki = 13000 nM T84631 COCN35 136092218 Ki = 34000 nM T84631 CA79JC 136092219 Ki = 6800 nM T84631 C5ST7C 136094220 Ki = 20000 nM T84631 CE0JY5 136094222 Ki > 30000 nM T84631 CJ8GD5 136094223 Ki > 30000 nM T84631 CFL8T4 136094224 Ki = 22000 nM T84631 CQW40T 136104458 IC50 > 100000 nM T84631 CI7XJ3 136104459 IC50 > 100000 nM T84631 C5FHI3 136180800 IC50 = 25 nM T84631 CPK6X2 136198635 Ki = 1.5 nM T84631 CRJ5S4 136198636 Ki = 5 nM T84631 C7WE2G 136198637 Ki = 2 nM T84631 C12UWY 136198638 Ki = 3 nM T84631 CT1QN2 136224837 Ki = 89700 nM T84631 CN8BW0 136224847 Ki > 100000 nM T84631 C7KE9J 136224848 Ki > 100000 nM T84631 C7R1TS 136224849 Ki > 100000 nM T84631 CG24CQ 136224854 Ki = 94800 nM T84631 CK4CM2 137028369 Ki > 28890 nM T84631 C3FRZ4 137629177 Ki = 0.034 nM T84631 C6OVC4 137631541 IC50 = 532 nM T84631 C2JT1W 137632528 IC50 = 212000 nM T84631 CL9C4Z 137633250 IC50 = 887 nM T84631 C64QCY 137633331 IC50 = 546000 nM T84631 CTV82J 137635086 IC50 = 127 nM T84631 CZB61A 137635154 IC50 = 165 nM T84631 CSI03M 137635473 IC50 = 243000 nM T84631 C5BOV8 137635960 IC50 = 157 nM T84631 CDQ62V 137637214 Ki > 50000 nM T84631 C9C4IS 137638370 IC50 = 234 nM T84631 C7W4AS 137638513 IC50 > 100000 nM T84631 CI7G6V 137639337 IC50 = 0.00188 ug.mL-1 T84631 C2K8JV 137639385 Ki = 23000 nM T84631 C89DPN 137639579 IC50 = 717 nM T84631 CGT80B 137640248 IC50 > 100000 nM T84631 CZWT21 137640786 IC50 = 360 nM T84631 CKYM10 137641934 IC50 = 354000 nM T84631 CE1XH0 137642026 IC50 = 1.473 ug.mL-1 T84631 C1RG9N 137642543 IC50 = 4065 nM T84631 C7YI0J 137643322 IC50 = 21 nM T84631 CIX05F 137645194 IC50 = 0.00169 ug.mL-1 T84631 CPY2W8 137646429 IC50 = 0.00287 ug.mL-1 T84631 CNO2T8 137647340 IC50 = 505000 nM T84631 C9EO5K 137647755 IC50 = 52000 nM T84631 CA1WS5 137647866 IC50 = 1414 nM T84631 CTJW91 137647903 IC50 = 345 nM T84631 C8RQW5 137647928 IC50 = 78000 nM T84631 CX5PU9 137648045 IC50 = 0.0315 ug.mL-1 T84631 C9F8HU 137648149 IC50 = 0.00527 ug.mL-1 T84631 C37KPL 137648430 IC50 > 100000 nM T84631 CDN2G1 137650387 IC50 = 0.03336 ug.mL-1 T84631 CVC4G9 137652563 IC50 = 42 nM T84631 CTZJ47 137653030 IC50 = 1267 nM T84631 CCH72E 137653236 IC50 = 0.803 ug.mL-1 T84631 CWO52T 137653817 IC50 = 20000 nM T84631 CNX46H 137654508 Ki > 50000 nM T84631 CS0XG8 137654871 IC50 = 113000 nM T84631 C1OXG8 137655944 IC50 = 31000 nM T84631 CG1AP0 137656734 IC50 = 179000 nM T84631 CYEK02 137658233 IC50 > 100000 nM T84631 CL8JG7 137658848 IC50 = 498 nM T84631 CY17AJ 137658996 IC50 = 2212 nM T84631 CYR84Z 137660177 IC50 = 1345 nM T84631 C68LGV 137661693 IC50 = 0.01692 ug.mL-1 T84631 CUZ35A 138115400 IC50 > 100000 nM T84631 CO51HN 139030452 IC50 > 50000 nM T84631 CX07YE 139592452 Ki > 9000 nM T84631 CE6C0A 145970642 Ki = 1940 nM T84631 CVU38Y 145979005 IC50 = 3026 nM T84631 C9QVU2 145981403 IC50 = 81 nM T84631 CZ1R3B 145982984 Ki = 45 nM T84631 CY53BG 145987654 IC50 = 5617 nM T84631 C5ST3M 145987720 IC50 = 1067 nM T84631 C0UIH3 145991316 IC50 = 5735 nM T84631 CM83CB 145993920 IC50 = 8451 nM T84631 C4HLX8 146029523 IC50 > 50000 nM T84631 CSBC71 146680900 IC50 = 31000 nM T84631 CH59QO 155510375 Ki > 100000 nM T84631 CZ28WP 155510611 IC50 = 246 nM T84631 CICU31 155511394 Ki = 28 nM T84631 CZR36C 155511554 IC50 > 100000 nM T84631 C1S8NW 155511576 Ki = 4861 nM T84631 CA81QV 155512709 Ki = 77600 nM T84631 C2VX3G 155512946 Ki > 13300 nM T84631 CTWK05 155513086 Ki = 321 nM T84631 C5K2RF 155513099 IC50 = 272 nM T84631 C52CEV 155513763 IC50 = 981 nM T84631 CZ9S2L 155513899 IC50 = 3189 nM T84631 C2CI8S 155513907 Ki = 15 nM T84631 CYT20V 155514020 Ki > 50000 nM T84631 C4MUP2 155514223 IC50 = 18 nM T84631 CAT98N 155514640 Ki = 460 nM T84631 C37MUL 155515203 IC50 = 3.5 nM T84631 CG9H4N 155515624 Ki = 113900 nM T84631 C7ZM4R 155515728 Ki = 16150 nM T84631 CPUG37 155516479 Ki > 17000 nM T84631 CFRS54 155516565 Ki = 28890 nM T84631 C57VQG 155516820 Ki = 785 nM T84631 CWI23M 155516948 Ki = 9877 nM T84631 CXY80S 155517048 Ki = 4674 nM T84631 C1ZSV0 155517054 Ki = 20480 nM T84631 C7N3OG 155517516 Ki = 20984 nM T84631 CZ7U1E 155517733 IC50 = 315 nM T84631 C5OG8J 155518396 Ki = 211 nM T84631 CF96DM 155518671 Ki = 96000 nM T84631 C4P9BA 155519561 Ki = 20671 nM T84631 C6NX4K 155519661 IC50 = 1584.89 nM T84631 C4MS1B 155519676 IC50 = 63095.73 nM T84631 CEID74 155519809 IC50 = 1079 nM T84631 C7DUX3 155520916 Ki > 100000 nM T84631 CW8JF0 155521080 IC50 = 77 nM T84631 CBA58W 155522743 Ki = 6169 nM T84631 CE01NY 155523107 IC50 > 20000 nM T84631 CSNL72 155523159 IC50 = 6100 nM T84631 CHW08G 155523201 Ki = 2654 nM T84631 CW9K3R 155523263 IC50 > 20000 nM T84631 CGMP07 155523803 IC50 = 260 nM T84631 CH0N9A 155523885 Ki = 7900 nM T84631 C5N4UF 155524709 Ki = 515 nM T84631 C7FXS3 155524763 IC50 = 7900 nM T84631 CYL8M0 155526377 Ki = 104200 nM T84631 CDT90I 155526882 Ki = 4333 nM T84631 C8F0RX 155526963 IC50 = 234 nM T84631 CX7CO2 155527010 Ki = 7400 nM T84631 CES4H0 155527736 Ki = 13342 nM T84631 CN3BH5 155527998 IC50 = 50118.72 nM T84631 CHYW65 155528639 IC50 = 5011.87 nM T84631 CG68UH 155529134 IC50 > 20000 nM T84631 CD7O2G 155530095 IC50 = 63095.73 nM T84631 CA82SM 155530516 Ki = 29 nM T84631 CT0N2L 155530721 IC50 = 18500 nM T84631 C35QWO 155531023 IC50 = 3981.07 nM T84631 CAU5B6 155531331 Ki = 1931 nM T84631 CP8K2J 155531811 Ki = 11530 nM T84631 C0UR8Q 155531991 Ki = 134400 nM T84631 C3AL6D 155533619 IC50 = 10 nM T84631 CY3FE6 155533938 IC50 = 4.8 nM T84631 C6F4JA 155534286 IC50 = 653 nM T84631 C7M2UT 155534310 IC50 = 6500 nM T84631 C2JC8E 155534627 Ki = 360 nM T84631 CN3K2L 155534709 Ki = 10697 nM T84631 CWS27U 155535533 IC50 = 1543 nM T84631 CLZO23 155535564 IC50 = 2087 nM T84631 CIHM01 155535907 Ki > 100000 nM T84631 C12HON 155536142 IC50 = 31622.78 nM T84631 CAK5R1 155536805 Ki = 2636 nM T84631 CGP82O 155536856 IC50 = 1700 nM T84631 C6S1JG 155537077 Ki = 8607 nM T84631 CUD5Y4 155537271 Ki = 2693 nM T84631 C7JMK4 155538439 Ki > 13000 nM T84631 C9QE5N 155538514 Ki > 100000 nM T84631 CD9J2M 155538805 Ki = 1612 nM T84631 CX9Q2L 155539448 IC50 = 45 nM T84631 CRT3D4 155540148 Ki = 50730 nM T84631 CT2VP1 155540521 Ki = 1913 nM T84631 CL90DN 155540666 Ki > 10000 nM T84631 CY6DK3 155540964 IC50 = 1995.26 nM T84631 C4CHR9 155542229 Ki = 188400 nM T84631 CI1G4S 155543248 IC50 = 1387 nM T84631 CY3T7E 155544010 IC50 = 220 nM T84631 C2MDQ4 155544600 Ki = 2875 nM T84631 CT4S3M 155544624 IC50 = 9000 nM T84631 CD9C5J 155545050 Ki = 26433 nM T84631 C4Q8CE 155545465 Ki = 1941 nM T84631 CU52QS 155545897 Ki > 10000 nM T84631 CQ51DI 155546002 IC50 = 2000 nM T84631 CJR8Y9 155546116 IC50 = 20 nM T84631 CLRJ05 155546124 Ki = 10276 nM T84631 CET91Y 155546188 IC50 = 179 nM T84631 CH2S6R 155546346 Ki = 520 nM T84631 CK6IX7 155547422 Ki = 12136 nM T84631 C5MB9R 155547962 IC50 = 10000 nM T84631 C0D5YW 155548172 IC50 > 2000 nM T84631 CLFB25 155548371 IC50 = 31622.78 nM T84631 CSI5J1 155548907 Ki = 201800 nM T84631 C2H3XJ 155549088 Ki = 2492 nM T84631 C8M9HD 155550013 Ki = 4177 nM T84631 CWC8X9 155550748 IC50 > 100000 nM T84631 C5X4OZ 155550860 Ki = 4025 nM T84631 CU9FL4 155551858 Ki > 50000 nM T84631 COM52R 155551892 IC50 = 5011.87 nM T84631 CA5VG2 155552651 Ki = 404500 nM T84631 C5S6HO 155553129 Ki = 47400 nM T84631 CZT5N7 155553153 Ki = 1809 nM T84631 CJ3FI5 155553630 IC50 = 79432.82 nM T84631 CA3W7F 155554002 Ki = 570 nM T84631 C5TV4J 155554082 Ki = 20640 nM T84631 CO60RZ 155555054 Ki = 9253 nM T84631 C82AXQ 155555647 Ki = 1643 nM T84631 CJW0Q5 155555987 Ki = 1974 nM T84631 CV0R8Y 155556453 Ki = 24000 nM T84631 CFU32P 155557286 IC50 = 4700 nM T84631 C3GWK1 155557690 Ki = 1980 nM T84631 CSW48V 155557718 IC50 = 398.11 nM T84631 CXL5D4 155558368 Ki > 100000 nM T84631 C9U2VZ 155558446 IC50 = 17800 nM T84631 CUA52W 155559155 IC50 = 960 nM T84631 CNZ1K5 155559920 Ki = 500 nM T84631 C3R5JK 155561209 IC50 = 7400 nM T84631 C3SXY1 155561904 Ki = 39520 nM T84631 C1EOR9 155561935 Ki = 1023 nM T84631 CX5O7K 155562968 Ki > 15000 nM T84631 C87WSX 155563035 Ki = 5500000 nM T84631 CQ6N8F 155564027 IC50 = 513 nM T84631 CD0OB4 155564213 Ki = 3603 nM T84631 C5I0YM 155564398 IC50 = 24 nM T84631 C2ZSL7 155565147 IC50 = 7200 nM T84631 CV6KA7 155565165 Ki = 9786 nM T84631 CM8XB1 155565537 IC50 = 7943.28 nM T84631 CTF0S7 155566456 Ki = 447 nM T84631 CS6XQ9 155566619 Ki = 18087 nM T84631 CGD4R1 155566743 IC50 = 30 nM T84631 CP4F1U 155567613 Ki > 50000 nM T84631 CEZ8B9 155568406 Ki > 100000 nM T84631 CK0EA2 155568484 Ki = 34400 nM T84631 CVK8X3 44338049 IC50 = 4.6 nM T84631 CY8D1H 54585929 Ki = 1258.93 nM T84631 D00KJP 10322586 Ki = 7 nM T84631 D00QDR 65238 IC50 = 170 nM T84631 D01LCS 447480 Ki = 1500 nM T84631 D01RTU 448763 Ki > 1000000 nM T84631 D02AVL 18376720 Ki = 0.005 nM T84631 D02KKL 1282 Ki = 1 nM T84631 D02PAU 16731825 Ki = 0.21 nM T84631 D02XPB 23646462 Ki = 1200 nM T84631 D02YIW 1794 IC50 > 50000 nM T84631 D03QAQ 9869498 Ki = 0.01 nM T84631 D03ZUM 6917805 IC50 = 1600 nM T84631 D06HOI 44249821 IC50 = 6.5 nM T84631 D06MTX 1506 Ki = 14000 nM T84631 D07HWB 10417809 IC50 = 280 nM T84631 D07IBU 10696098 IC50 > 20000 nM T84631 D07SFI 2332 Ki = 200 nM T84631 D07ZRG 46899577 Ki = 2.4 nM T84631 D0C1TS 44272875 Ki = 674 nM T84631 D0CT8A 23646461 Ki = 39000 nM T84631 D0F6EZ 44436702 Ki > 1000000 nM T84631 D0FV9Y 44453269 IC50 = 6 nM T84631 D0G4LX 46233650 Ki = 583 nM T84631 D0I1UF 14035442 Ki = 450 nM T84631 D0J1CC 11948634 Ki = 11400 nM T84631 D0J1QT 44473100 Ki = 5.2 nM T84631 D0JU9N 6914623 Ki = 0.03 nM T84631 D0K7YL 447476 Ki = 78 nM T84631 D0LX0D 46233193 Ki = 14800 nM T84631 D0M1BF 9803617 Ki = 96 nM T84631 D0M4VZ 10456438 IC50 = 1900 nM T84631 D0MQ6K 10574241 Ki = 80 nM T84631 D0O0GT 44272797 Ki = 192 nM T84631 D0ON2Z 204102 Ki = 0.19 nM T84631 D0P7NY 23661637 IC50 = 100000 nM T84631 D0R5KV 4322 Ki = 0.1 nM T84631 D0R9CH 3400921 Ki = 0.007 nM T84631 D0SP2I 6852210 Ki = 27000 nM T84631 D0V7TH 76328755 Ki > 15000 nM T84631 D0Y4KJ 46233192 Ki = 3700 nM T84631 D0Y5IQ 44255320 IC50 = 10000 nM T84631 D0Y8QU 9869156 IC50 > 2500 nM T84631 D0Y9PH 45486355 Ki = 40000 nM T84631 D0Z2PJ 24859718 Ki = 6000 nM T84631 D0Z2TG 442688 IC50 = 560 nM T90985 D05ICT 132010322 Ki = 1 nM T90985 D0G8BM 16722836 IC50 = 340 nM T90985 D0M2TS 71600087 Ki = 2.2 nM T90985 D0O0LQ 11364421 IC50 = 260 nM T90985 D0PH9I 118693659 Ki = 100 nM T90985 D0ZW4W 46907787 IC50 = 103 nM T90985 D0D3PX 46926350 IC50 = 37000 nM T90985 CNQ59G 719444 IC50 = 68000 nM T90985 CS1EI8 4541508 Ki > 40000 nM T90985 CB45RH 4794457 Ki > 40000 nM T90985 CY71BJ 4800411 Ki = 1400 nM T90985 CHU94T 6484105 IC50 = 140000 nM T90985 C81LRG 9581822 IC50 = 120000 nM T90985 C0BW3Q 11260691 IC50 = 342 nM T90985 CMJ01U 11283298 IC50 = 560 nM T90985 C6ONU5 16251975 Ki > 40000 nM T90985 CP60ON 16258758 Ki = 2400 nM T90985 CE3X0C 16265714 Ki <= 450 nM T90985 C6WU8Z 16414715 IC50 = 130000 nM T90985 CBX53R 16457178 IC50 = 220000 nM T90985 C4TC3X 16722832 IC50 = 230 nM T90985 CGFA68 16822024 Ki = 1100 nM T90985 CVGU58 18536615 IC50 = 13000 nM T90985 C6Y4GF 18536633 IC50 = 18000 nM T90985 CDS15V 18536647 IC50 = 88000 nM T90985 C1C3QM 44269241 IC50 > 250000 nM T90985 C98BLM 49871817 IC50 = 110 nM T90985 CG3PR6 52912222 IC50 = 31622.78 nM T90985 CF8B4E 60498769 IC50 = 100000 nM T90985 CIPN50 71760902 Ki = 110 nM T90985 C5TB9S 77843982 Ki = 140 nM T90985 COZ8S1 78319129 Ki = 490 nM T90985 C4IF8T 78425807 Ki = 0.69 nM T90985 CFE7R3 86270928 Ki = 4.2 nM T90985 CDG13U 86295201 IC50 = 3513 nM T90985 C1W3XP 112499930 IC50 = 2300 nM T90985 C3QJ5L 122181550 IC50 = 31622.78 nM T90985 CD24VL 122187519 IC50 = 25990 nM T90985 CH14FC 127032939 IC50 = 7900 nM T90985 CS4NG8 127033568 IC50 > 100000 nM T90985 CSO7R6 135530212 IC50 = 220000 nM T90985 C5F3LV 135567026 IC50 > 100000 nM T90985 CO71RI 137285009 IC50 = 3082 nM T90985 CS9MR6 137285011 IC50 = 2781 nM T90985 CFXE14 137321203 IC50 = 501.19 nM T90985 CXN4U1 137321204 IC50 = 199.53 nM T90985 CR5FO2 137632087 Ki > 40000 nM T90985 C7F4MJ 137632577 Ki = 230 nM T90985 CA2D8W 137632690 Ki > 40000 nM T90985 C12WYV 137633398 IC50 = 67000 nM T90985 CO08EU 137636712 Ki = 5600 nM T90985 CVK32T 137639306 Ki <= 450 nM T90985 CVQE64 137643147 Ki > 40000 nM T90985 CD8VQ1 137643820 Ki > 40000 nM T90985 CRJ2W3 137644677 IC50 = 2200 nM T90985 C8QO2D 137648257 Ki = 200 nM T90985 CA4WO8 137653484 Ki = 220 nM T90985 CZ1K6N 137654718 Ki = 23000 nM T90985 CVH74T 137655200 Ki = 4700 nM T90985 C1YOL6 137657448 Ki = 200 nM T90985 CPRY31 137661484 IC50 = 87000 nM T90985 CU5N8O 137701509 IC50 = 3500 nM T90985 CYV4O3 138756791 IC50 = 4700 nM T90985 CQ6XB7 139030526 IC50 = 15848.93 nM T90985 CD6U7X 145925666 IC50 = 357.1 nM T90985 CC17DU 145964393 IC50 = 933 nM T90985 CH06LF 145964543 IC50 = 392 nM T90985 CCW5X8 145965219 IC50 = 378 nM T90985 CE4D5F 145966579 IC50 = 1951 nM T90985 CXWZ04 145967512 IC50 = 978 nM T90985 CV83ED 145972103 Ki = 5.9 nM T90985 CN70KV 145972360 IC50 = 289 nM T90985 C2RTO8 145972845 IC50 = 229 nM T90985 C6R2YM 145975649 IC50 = 8468 nM T90985 CTAZ41 145975701 IC50 > 50000 nM T90985 CW56PH 145975703 IC50 = 102 nM T90985 CN4O0K 145976012 IC50 = 750 nM T90985 CR28YS 145976646 IC50 = 245 nM T90985 CVJ61U 145977109 IC50 = 3543 nM T90985 CB9F1X 145977980 IC50 = 369 nM T90985 C0MD9U 145978238 IC50 = 558 nM T90985 C9FIY4 153534005 IC50 > 20000 nM T90985 CFD6H1 155352361 IC50 = 36000 nM T90985 CFK2B1 155352401 IC50 = 110000 nM T90985 C27LFN 155514936 IC50 = 1600 nM T90985 D00XRH 91820725 IC50 = 25118.86 nM T90985 D0F5TZ 91827383 IC50 = 31622.78 nM T90985 D0VC0I 5169 IC50 = 20000 nM T90985 D0Y3OO 11327430 IC50 = 3500 nM T31818 CVPF30 11839482 EC50 = 22000 nM T31818 CM5X2F 59821830 EC50 = 20000 nM T31818 C4RKS8 90665331 EC50 = 17000 nM T31818 CE2SV0 90665332 EC50 = 20000 nM T31818 CU8HX1 90665337 EC50 = 19000 nM T31818 CM87PA 90665339 EC50 = 16000 nM T31818 C9SBM0 90665340 EC50 = 40000 nM T31818 CV03RS 90665341 EC50 = 11000 nM T79747 D05FKU 86280523 IC50 = 2.9 nM T79747 D0J5HR 46926973 IC50 = 0.4 nM T79747 C5R1AG 2155128 IC50 = 157 nM T79747 CO9UQ2 3423911 IC50 = 60 nM T79747 CFL8J3 4786512 IC50 = 15 nM T79747 C7SH6B 4993304 IC50 = 8 nM T79747 CX91ZA 9114840 IC50 = 24 nM T79747 C1Y3XQ 57519544 IC50 = 0.074 nM T79747 CMKO61 86303027 IC50 = 1 nM T79747 C3Y9KN 86303187 IC50 = 2 nM T79747 CS5DT3 86303342 IC50 > 50000 nM T79747 C2EOJ5 86763941 IC50 = 0.5 nM T79747 CNB7A0 86763942 IC50 = 5400 nM T79747 CP9N7S 86764709 IC50 = 0.4 nM T79747 CK6E0W 91810397 IC50 = 12 nM T79747 CWM43E 117668573 IC50 = 33000 nM T79747 CL5OI9 117668598 IC50 = 42 nM T79747 CJ94UW 117668684 IC50 > 50000 nM T79747 C2RS7Z 117668802 IC50 = 40 nM T79747 C5IO0K 117671078 IC50 = 10 nM T79747 CE8SK5 117671214 IC50 = 4 nM T79747 CWL5J8 118174040 IC50 = 12 nM T79747 CS6Y1X 118174075 IC50 = 29 nM T79747 CT24YC 118174086 IC50 = 12 nM T79747 CYAX71 118174089 IC50 = 1 nM T79747 CCK2H9 118174109 IC50 = 67 nM T79747 C12LXT 118174114 IC50 = 8 nM T79747 CF38UC 118174137 IC50 = 29 nM T79747 CKXC27 118174156 IC50 = 15 nM T79747 CZ46TY 118174196 IC50 = 1 nM T79747 CZ3A6L 118174200 IC50 = 72 nM T79747 C7GU0A 118174229 IC50 = 11 nM T79747 CDA16S 118174232 IC50 = 11 nM T79747 CS7ER1 118174312 IC50 = 9 nM T79747 C6E8OG 121237481 IC50 = 0.38 nM T79747 C0FQX3 122192846 IC50 = 5 nM T79747 CF0S3G 122192847 IC50 = 2.2 nM T79747 CMXO16 122192848 IC50 = 0.23 nM T79747 C8V4CD 122192849 IC50 = 188 nM T79747 CE68BP 122192850 IC50 = 164 nM T79747 C8V5YM 122192851 IC50 = 40 nM T79747 C19VFK 122192852 IC50 = 30 nM T79747 C15UAX 122192853 IC50 > 1000 nM T79747 CRBE37 122192854 IC50 > 1000 nM T79747 C36ZXY 122192855 IC50 > 1000 nM T79747 CS34WY 122192856 IC50 > 1000 nM T79747 C1JR4U 122192857 IC50 > 1000 nM T79747 CN4RC0 122192858 IC50 > 1000 nM T79747 CO3KE8 122192859 IC50 > 1000 nM T79747 CCVR74 122192860 IC50 = 2.7 nM T79747 CK4BO2 122192861 IC50 = 485 nM T79747 C5JOZ0 122192862 IC50 = 24 nM T79747 CO2WJ4 122192863 IC50 = 483 nM T79747 CN52YT 122192864 IC50 = 0.96 nM T79747 CI9WG3 122192865 IC50 = 0.67 nM T79747 CV2KN5 122192866 IC50 = 0.53 nM T79747 CV4PZ3 122192867 IC50 = 0.19 nM T79747 C5B2DY 122192868 IC50 = 0.11 nM T79747 CB97PK 122195558 IC50 = 27 nM T79747 CF20MA 122195559 IC50 = 5 nM T79747 C98ECK 122234471 IC50 = 130 nM T79747 CL2MT3 122234472 IC50 = 5 nM T79747 CX6NG2 122234473 IC50 = 689 nM T79747 C2R4UL 122234474 IC50 = 7 nM T79747 C32PNV 122234475 IC50 = 1 nM T79747 C4OW0K 122652940 IC50 = 6 nM T79747 C5I6CL 137635434 IC50 = 15 nM T79747 C0Y9EA 137642070 IC50 = 60 nM T79747 CM43SF 137648320 IC50 = 30 nM T79747 CCEM45 137661947 IC50 = 42 nM T79747 C9T0SR 145976580 IC50 = 710 nM T79591 D0L5WM 2157 IC50 = 650 nM T79591 D0S6JG 5920 Ki = 0.22 nM T79591 D0Z4EI 55245 Ki > 1250 nM T79591 D01QXY 9862248 Ki = 1.09 nM T79591 D03MYO 15981237 EC50 = 3740 nM T79591 D07ZTD 15942005 Ki = 12500 nM T79591 D0J6XC 5803 IC50 = 0.14 nM T79591 D0V5FQ 166559 Ki = 40 nM T79591 D02WGY 10299876 Ki = 9.6 nM T79591 D07EGS 9874938 Ki = 0.51 nM T79591 CLSK17 5804 IC50 = 0.04074 nM T79591 C47GSU 79170 IC50 = 9200 nM T79591 C57HCR 652088 IC50 = 85300 nM T79591 CB6HQ4 656928 IC50 = 15.14 nM T79591 C5T8GU 2249170 IC50 = 18100 nM T79591 CG59SJ 2404806 IC50 = 47700 nM T79591 CJN3P5 4266779 IC50 = 16600 nM T79591 CU1I3O 4652254 IC50 > 100000 nM T79591 CRQ1O4 9819350 Ki = 0.7 nM T79591 C4PCB9 9825337 EC50 = 23 nM T79591 C3MZ1Y 9843007 Ki = 172 nM T79591 CJ6E2M 9847869 Ki = 20 nM T79591 CA27CJ 9862799 IC50 = 128.82 nM T79591 CZ82PF 9863447 EC50 = 4.5 nM T79591 CC64MT 9869395 IC50 = 1600 nM T79591 CZ1U7X 9932398 IC50 = 9.7 nM T79591 CY01RH 9933119 EC50 = 0.38 nM T79591 CHG6L7 9933993 IC50 = 630 nM T79591 C46NXU 9951790 IC50 = 1.4 nM T79591 CX4MZ9 9980722 IC50 = 19 nM T79591 CZ96GN 10030727 IC50 = 88 nM T79591 CJ05DK 10049652 IC50 = 13 nM T79591 CP1R7A 10113366 IC50 = 360 nM T79591 C72HTV 10135986 IC50 = 420 nM T79591 CMY69T 10137392 IC50 = 600 nM T79591 CGE9I7 10151760 Ki = 228 nM T79591 C1Y3FJ 10174187 Ki = 186 nM T79591 CD4SX7 10202877 IC50 = 2600 nM T79591 CNPD04 10216950 Ki = 69.3 nM T79591 CDY6F5 10238439 Ki = 30.5 nM T79591 C1DYU9 10269704 Ki = 147 nM T79591 CJB2E3 10274474 Ki = 3 nM T79591 C7UYX0 10276774 Ki = 2.1 nM T79591 CH5NX1 10279835 Ki = 126 nM T79591 CW26FQ 10287060 Ki = 2.45 nM T79591 CIB52S 10297431 IC50 = 3300 nM T79591 CSC3T4 10299993 IC50 = 616.6 nM T79591 C81BSZ 10309431 Ki = 127 nM T79591 C09IJX 10310671 Ki > 10000 nM T79591 CT13FC 10310672 Ki > 10000 nM T79591 C0VMH3 10321482 IC50 = 5000 nM T79591 C7TGL0 10322653 Ki = 8 nM T79591 CP8O0Q 10455127 IC50 = 101 nM T79591 C3UAD9 10456672 IC50 = 5.4 nM T79591 C5N7BD 10456830 IC50 = 0.1 nM T79591 C34MFS 10457976 IC50 = 62 nM T79591 C4T6ZH 10479778 IC50 = 4.3 nM T79591 CM4ED8 10479779 IC50 = 2.512 nM T79591 CU42IL 10897325 IC50 = 1400 nM T79591 CX2RY1 10904700 EC50 = 0.3 nM T79591 CZ3SX1 10918755 IC50 = 820 nM T79591 CD9G7N 11164881 IC50 = 12882.5 nM T79591 C6OX1A 11209929 IC50 = 160000 nM T79591 CPY31C 11247142 IC50 = 460 nM T79591 CA8Z1T 11281247 IC50 = 1584.89 nM T79591 CY0M1L 11395277 IC50 = 4365.16 nM T79591 C48UZO 11463526 IC50 = 820 nM T79591 C5CZ2Q 11998611 Ki = 12500 nM T79591 CRJ1N9 11999781 Ki = 42.1 nM T79591 C7N4HR 11999783 Ki = 10.3 nM T79591 CW01OG 12001110 EC50 = 330 nM T79591 C1AU0V 13958302 Ki = 8.72 nM T79591 CDB93J 15219550 IC50 = 19200 nM T79591 CDKZ56 15940421 Ki = 143 nM T79591 CM17XO 15941848 Ki = 35.2 nM T79591 C1QZ3U 15941849 Ki = 285 nM T79591 CRK5V2 15941850 Ki = 1416 nM T79591 C7PV1O 15941997 Ki = 18.6 nM T79591 C7BD0S 15941998 Ki = 186 nM T79591 C93MUZ 15942131 Ki = 30.5 nM T79591 CNCW45 15942413 Ki = 28.4 nM T79591 CEQ1J5 15981204 EC50 = 15640 nM T79591 CZEJ29 15981205 EC50 = 12000 nM T79591 C47AYJ 15981206 EC50 = 3280 nM T79591 CRF9T7 15981207 EC50 = 7010 nM T79591 C4XF0E 15981234 EC50 = 390 nM T79591 C7U4OQ 15981235 EC50 = 700 nM T79591 CT9N6B 15981236 EC50 = 210 nM T79591 CTI37Q 15981238 EC50 = 410 nM T79591 CIM62O 15981239 EC50 = 780 nM T79591 CB6UE5 15981240 EC50 = 2750 nM T79591 CL0FG1 15981241 EC50 = 820 nM T79591 C4BU2G 15981272 EC50 = 4290 nM T79591 C5BO7H 15981273 EC50 = 750 nM T79591 CES0V2 15981274 EC50 = 8880 nM T79591 C2SR1B 15981276 EC50 = 14390 nM T79591 CIB52A 15981279 EC50 = 1250 nM T79591 CWK35C 16730429 IC50 = 99 nM T79591 C7G2AM 18415120 Ki = 235 nM T79591 CD0L4R 21110667 Ki = 201 nM T79591 C0AQU8 21110669 Ki = 814 nM T79591 CZI6V2 21110670 Ki = 1366 nM T79591 C47HQO 21110672 Ki = 1645 nM T79591 CV3FE0 21110673 Ki = 429 nM T79591 CCGP69 21110677 Ki = 710 nM T79591 CM0DL5 21110680 Ki > 10000 nM T79591 CHN91T 21110689 Ki = 1431 nM T79591 CHT5Y9 21110691 Ki = 154 nM T79591 C7TN9A 21110692 Ki = 1638 nM T79591 CX5I2A 21636517 IC50 = 71000 nM T79591 CF2X6V 22339458 EC50 = 12 nM T79591 CF2CQ7 22372339 IC50 > 100000 nM T79591 CFV3P7 23635238 IC50 = 3600 nM T79591 CWE74Y 23635239 IC50 = 3000 nM T79591 CM6S4G 23635240 IC50 = 4100 nM T79591 CPR67K 23635363 IC50 = 6300 nM T79591 CI6D4Y 23635365 IC50 = 22600 nM T79591 CAHT12 23635366 IC50 = 16500 nM T79591 C1G2TO 23635477 IC50 = 52900 nM T79591 C17PKJ 23635478 IC50 > 100000 nM T79591 CC3VU5 23635479 IC50 > 100000 nM T79591 CGU3Z0 23635480 IC50 > 100000 nM T79591 C82WJG 23635600 IC50 > 100000 nM T79591 C18SZO 23635729 IC50 = 21600 nM T79591 C7BLC2 23635731 IC50 > 100000 nM T79591 CE6DP7 23635732 IC50 > 100000 nM T79591 CGL6T0 23635852 IC50 > 100000 nM T79591 CK4XI2 23635853 IC50 > 100000 nM T79591 CY80FR 23635854 IC50 > 100000 nM T79591 C7NAV1 23635855 IC50 = 68900 nM T79591 CU81CL 23635857 IC50 > 100000 nM T79591 C31FPX 23635859 IC50 > 100000 nM T79591 CQ2E7G 23642624 IC50 > 100000 nM T79591 CB38IZ 23644731 IC50 = 269.15 nM T79591 CT5QC3 23648079 IC50 = 0.14 nM T79591 CP7SV3 23648080 IC50 = 26 nM T79591 CYU20W 23648081 IC50 = 10 nM T79591 C3V1BH 23648082 IC50 = 83 nM T79591 C1JIZ5 23648083 IC50 = 4.3 nM T79591 C3QR1F 23648084 IC50 = 9.8 nM T79591 C0N2YD 23648085 IC50 = 7.5 nM T79591 C08JWQ 23648086 IC50 = 5.5 nM T79591 C5INJ3 23648087 IC50 = 460 nM T79591 CTJK20 23648089 IC50 = 670 nM T79591 CE4R6V 23648090 IC50 = 1500 nM T79591 C84TAV 23648093 IC50 = 1300 nM T79591 CB7OK8 23648094 IC50 = 370 nM T79591 C45JQX 23648095 IC50 = 500 nM T79591 C80CEB 23648096 IC50 = 480 nM T79591 C1DLP6 23648097 IC50 = 930 nM T79591 C4LY6R 23648098 IC50 = 39000 nM T79591 C4KX5O 23648099 IC50 = 1800 nM T79591 C9N7IR 23648100 IC50 = 69000 nM T79591 CV20UI 23648101 IC50 = 12.88 nM T79591 CIKD57 23648102 IC50 = 240 nM T79591 CV91YT 23648103 IC50 = 1288.25 nM T79591 C5WKV2 23648104 IC50 = 1200 nM T79591 C5V6OQ 23648105 IC50 = 128.82 nM T79591 C91FSP 23648106 IC50 = 18.2 nM T79591 CBD9J5 23648107 IC50 = 39.81 nM T79591 C1SXM0 23648109 IC50 = 123.03 nM T79591 C98FIL 23648110 IC50 = 457.09 nM T79591 C7R2XE 23648111 IC50 = 295.12 nM T79591 CR85SZ 23648112 IC50 = 30.2 nM T79591 CN2YX0 23648113 IC50 = 100 nM T79591 CC69AB 23648114 IC50 = 1047.13 nM T79591 COP12V 23648115 IC50 = 1174.9 nM T79591 CN5T8D 23648116 IC50 = 851.14 nM T79591 C7ON2Q 23648118 IC50 = 812.83 nM T79591 CXTZ50 23648122 IC50 = 123.03 nM T79591 CZ8J0T 23648123 IC50 = 245.47 nM T79591 C12HDM 23648124 IC50 = 50.12 nM T79591 CFA1Y6 23648126 IC50 = 501.19 nM T79591 C35AZQ 23648127 IC50 = 1479.11 nM T79591 CR1S4E 23648128 IC50 = 549.54 nM T79591 C0WY3I 23648129 IC50 = 239.88 nM T79591 CL60SF 23648130 IC50 = 426.58 nM T79591 C72TJZ 23648131 IC50 = 85.11 nM T79591 COL8Q7 23648132 IC50 = 204.17 nM T79591 CNWC43 23648133 IC50 = 281.84 nM T79591 C4SW8I 23648134 IC50 = 229.09 nM T79591 CQ7M3I 23648135 IC50 = 93.33 nM T79591 CQW43F 23648136 IC50 = 95.5 nM T79591 C62YFJ 23648137 IC50 = 18.2 nM T79591 CICP87 23648138 IC50 = 1148.15 nM T79591 CTE1N2 24748569 EC50 > 10000 nM T79591 C5XD8Q 24830528 IC50 = 230 nM T79591 CR2A9H 24830680 IC50 = 5200 nM T79591 CD6EI3 24830686 IC50 = 190 nM T79591 CKDP62 24830833 IC50 = 5200 nM T79591 CO9E2H 24894049 EC50 = 1056 nM T79591 C5BS8M 25149230 Ki = 16 nM T79591 CJ6LC2 25149503 Ki = 61.6 nM T79591 CT0J6H 25149504 Ki = 1165 nM T79591 CFW74J 25149505 Ki = 3296 nM T79591 C5MFE8 25149592 Ki = 303 nM T79591 CLSD47 25149598 Ki = 183 nM T79591 CZP70F 25150124 Ki = 897 nM T79591 C4MT7I 25150127 Ki = 594 nM T79591 C7G5CL 25150225 Ki = 1760 nM T79591 C57AUE 25150325 Ki = 1.84 nM T79591 CLZ86A 25150424 Ki = 3.74 nM T79591 CRW82I 44136896 IC50 = 8200 nM T79591 CQAT73 44186032 IC50 = 5300 nM T79591 CC0YN9 44186033 IC50 > 50000 nM T79591 C7VZI4 44186034 IC50 = 3500 nM T79591 CR1D9P 44186035 IC50 = 4000 nM T79591 CC32IS 44186097 IC50 = 3800 nM T79591 C2MG6T 44186098 IC50 = 22200 nM T79591 C4XV1B 44186099 IC50 = 4300 nM T79591 CFJ0P8 44186100 IC50 > 50000 nM T79591 C31NSX 44186101 IC50 = 3500 nM T79591 CBM5Z6 44186102 IC50 = 3200 nM T79591 CX10SK 44186103 IC50 = 2300 nM T79591 C8TU3K 44186104 IC50 = 1200 nM T79591 CWY0A2 44186168 IC50 = 9300 nM T79591 CO65HR 44186169 IC50 = 3400 nM T79591 C1TU5I 44186170 IC50 = 1400 nM T79591 CC49MP 44186171 IC50 = 7700 nM T79591 C3M4KR 44186172 IC50 = 3000 nM T79591 C4COU6 44186173 IC50 = 600 nM T79591 C40ENX 44186175 IC50 = 14800 nM T79591 CIL71S 44186232 IC50 > 50000 nM T79591 CP1A5G 44186233 IC50 > 50000 nM T79591 C4CMU9 44186234 IC50 > 50000 nM T79591 CM9V8Z 44186235 IC50 = 1900 nM T79591 CDI86U 44186236 IC50 = 1300 nM T79591 C2YL8N 44186237 IC50 = 4800 nM T79591 CYO36K 44186238 IC50 = 19800 nM T79591 CRHL62 44186239 IC50 = 3000 nM T79591 CS2N6F 44186298 IC50 > 50000 nM T79591 CES48R 44186299 IC50 > 50000 nM T79591 C6XEM3 44186300 IC50 > 50000 nM T79591 C35QER 44186301 IC50 = 30900 nM T79591 CREP27 44186302 IC50 > 50000 nM T79591 CPLW35 44186303 IC50 = 6200 nM T79591 C1PFT0 44186305 IC50 = 33300 nM T79591 CA1EV7 44186421 IC50 = 5800 nM T79591 CU64OD 44186422 IC50 = 5400 nM T79591 C9J0YD 44186423 IC50 = 2600 nM T79591 C25UOE 44186424 IC50 = 1100 nM T79591 CX9U3Q 44186425 IC50 = 1900 nM T79591 C0Z9OK 44186469 IC50 = 4700 nM T79591 CTJ1O5 44186470 IC50 = 3700 nM T79591 CN8QS2 44186471 IC50 = 1300 nM T79591 C78TSP 44186472 IC50 = 810 nM T79591 CL17KI 44186473 IC50 = 7100 nM T79591 COL0S6 44186474 IC50 = 4100 nM T79591 C75UOJ 44186475 IC50 = 13400 nM T79591 C1KVH2 44186476 IC50 > 50000 nM T79591 C3SH2I 44186517 IC50 = 1900 nM T79591 C8X1EA 44186518 IC50 = 6300 nM T79591 CS7K3Y 44186519 IC50 = 8400 nM T79591 CHW5K6 44186520 IC50 > 50000 nM T79591 C58YWK 44186521 IC50 > 50000 nM T79591 CJPO14 44186523 IC50 = 6800 nM T79591 C2NPV9 44186562 IC50 = 9800 nM T79591 CYH38F 44186563 IC50 > 50000 nM T79591 CGXM40 44349576 EC50 = 1500 nM T79591 CB1P0S 44396251 Ki > 1250 nM T79591 CHY1C3 44396271 Ki = 1200 nM T79591 C29MBI 44396272 Ki = 1100 nM T79591 C4TQ6N 44396282 Ki = 670 nM T79591 CH2Y3L 44396283 Ki > 1250 nM T79591 CWZB52 44396284 Ki > 1250 nM T79591 CD80LM 44396296 Ki = 790 nM T79591 C6SI5L 44396297 Ki > 1250 nM T79591 CR4H1E 44396316 Ki > 1250 nM T79591 C45LRH 44396317 Ki > 1250 nM T79591 CA8V4G 44396331 Ki > 1250 nM T79591 CA8OB7 44400181 IC50 = 650 nM T79591 C4G9CF 44403605 IC50 = 3605 nM T79591 CW6EH8 44403606 IC50 = 109 nM T79591 C0L3WU 44403607 IC50 = 1538 nM T79591 COU4B6 44403627 IC50 = 48 nM T79591 CVH75N 44403628 IC50 = 125 nM T79591 CTQ48J 44403634 IC50 = 14 nM T79591 C3SZ4I 44408427 EC50 = 83 nM T79591 CDE12F 44408544 EC50 = 4.1 nM T79591 C3TAU6 44408607 IC50 = 251.19 nM T79591 CM27EY 44417461 IC50 = 460 nM T79591 CC9BF0 44433089 IC50 = 168 nM T79591 CP7C9J 44435761 IC50 > 100000 nM T79591 CWG53Q 44435778 IC50 = 60900 nM T79591 CH56GJ 44435779 IC50 = 69600 nM T79591 CB1UR7 44435786 IC50 = 75600 nM T79591 CL3FT4 44445692 IC50 = 125.89 nM T79591 C20LCQ 44445716 IC50 = 2691.53 nM T79591 C1EGS9 44445719 IC50 = 457.09 nM T79591 CHT8I1 44445726 IC50 = 38.02 nM T79591 C9U7HY 44445727 IC50 = 3467.37 nM T79591 C31JKD 44445730 IC50 = 338.84 nM T79591 C0NH4Z 44445731 IC50 = 616.6 nM T79591 CEX30A 44452442 EC50 = 11 nM T79591 CR5SI0 44476535 EC50 > 10000 nM T79591 CD38FN 44567764 EC50 = 222 nM T79591 CV1W9E 44589465 Ki = 378 nM T79591 C9K7HA 45270610 IC50 > 50000 nM T79591 CUD91T 49862248 EC50 > 10000 nM T79591 CM7BY6 53385590 IC50 = 4500 nM T79591 C6Z7WI 60204885 IC50 = 1200 nM T79591 C05ZRG 69428069 Ki = 91.8 nM T79591 CR2M8J 69844039 Ki = 503 nM T79591 C5SRF8 70681735 Ki = 195 nM T79591 C3A0DO 70682526 IC50 = 5600 nM T79591 CLJU20 70682537 IC50 = 430 nM T79591 C2SVR8 70682538 IC50 = 2500 nM T79591 CBVQ29 70683842 Ki = 24.4 nM T79591 CVON79 70683843 Ki = 300 nM T79591 C9R0NB 70683844 Ki = 1246 nM T79591 CG40IU 70684617 IC50 = 1100 nM T79591 CO1MQ8 70684618 IC50 = 1000 nM T79591 CU5VH3 70684619 IC50 = 3200 nM T79591 CARO49 70685018 Ki > 1250 nM T79591 CVK46F 70686763 IC50 = 4700 nM T79591 CWJ6U3 70686764 IC50 = 100 nM T79591 C70SIB 70688836 IC50 = 1100 nM T79591 CLF25D 70690926 IC50 = 1100 nM T79591 CB3ZC2 70690927 IC50 = 300 nM T79591 C6FA0H 70690939 IC50 = 1600 nM T79591 C90XVL 70693065 IC50 = 2400 nM T79591 CC2EK8 70693080 IC50 = 2500 nM T79591 C2WC4V 70695111 IC50 = 3500 nM T79591 C92QMH 70695112 IC50 = 460 nM T79591 CMNE57 70695113 IC50 = 190 nM T79591 CTQ37A 70697163 IC50 = 2600 nM T79591 CLU28H 71461159 EC50 = 18 nM T79591 CL8K9N 71523879 Ki > 10000 nM T79591 CQ0C5S 71523924 Ki > 10000 nM T79591 C8DI5U 71523925 Ki = 6751 nM T79591 CTU1K7 71523963 Ki = 4866 nM T79591 CGHD73 71570928 IC50 = 9600 nM T79591 C49SBQ 71571065 IC50 = 4200 nM T79591 CE06XT 71571066 IC50 = 1900 nM T79591 CR92GT 71571067 IC50 = 1700 nM T79591 CTUC72 71571068 IC50 > 60000 nM T79591 C7UHM3 71571069 IC50 > 60000 nM T79591 C1P5HY 71571070 IC50 > 60000 nM T79591 C4CNP2 71571213 IC50 > 60000 nM T79591 CAV18D 71571215 IC50 > 60000 nM T79591 C97ISQ 71571216 IC50 > 60000 nM T79591 C5ZT9O 71716541 IC50 > 60000 nM T79591 C1TN8C 71716542 IC50 > 60000 nM T79591 CPJ4T2 71716543 IC50 > 60000 nM T79591 CP9B4C 71716544 IC50 > 60000 nM T79591 C4OE3H 71716545 IC50 > 60000 nM T79591 CIJ84X 71716546 IC50 = 29000 nM T79591 C4XL7Z 71716547 IC50 > 60000 nM T79591 C7BMG8 71716548 IC50 > 60000 nM T79591 C8O2NJ 71716549 IC50 > 60000 nM T79591 CA1Q0X 71716550 IC50 > 60000 nM T79591 CM6ZN5 71716551 IC50 > 60000 nM T79591 CX6RH7 71716552 IC50 > 60000 nM T79591 CTI7H2 71716553 IC50 > 60000 nM T79591 C8YEZ6 71716554 IC50 > 60000 nM T79591 CT3D1M 71717145 IC50 > 60000 nM T79591 CSHP85 71717146 IC50 > 60000 nM T79591 C5K3QG 71717147 IC50 > 60000 nM T79591 C6B5DO 71717148 IC50 > 60000 nM T79591 CK0ZQ9 71717149 IC50 > 60000 nM T79591 C96GSC 71717150 IC50 > 60000 nM T79591 C36SFW 71717155 IC50 > 60000 nM T79591 CLR58A 71717156 IC50 > 60000 nM T79591 CN4A9V 71717771 IC50 > 60000 nM T79591 CPLW58 71717772 IC50 > 60000 nM T79591 CIL03B 71717773 IC50 = 44000 nM T79591 C63QLG 71717774 IC50 = 33000 nM T79591 CV0I1H 71717775 IC50 = 33000 nM T79591 CUN4O0 71717776 IC50 > 60000 nM T79591 CSO2X5 71717777 IC50 > 60000 nM T79591 C52BZC 71717778 IC50 > 60000 nM T79591 CIE8V5 71717779 IC50 > 60000 nM T79591 C46ICD 71717780 IC50 > 60000 nM T79591 CPH02C 71718378 IC50 > 60000 nM T79591 COX71E 71718379 IC50 > 60000 nM T79591 CC94QZ 71718380 IC50 = 58000 nM T79591 CG2TH9 71718381 IC50 = 37000 nM T79591 C6G4BT 71718382 IC50 = 32000 nM T79591 CQ8AI1 71718383 IC50 > 60000 nM T79591 C4KOT9 71718386 IC50 > 60000 nM T79591 CH2TV1 71718387 IC50 > 60000 nM T79591 CXO1S7 71718388 IC50 > 60000 nM T79591 CI6AN0 71718985 IC50 > 60000 nM T79591 C5U7IR 71718986 IC50 > 60000 nM T79591 C0CJ8S 71718987 IC50 > 60000 nM T79591 C4KAZ7 71718988 IC50 > 60000 nM T79591 CIN3V1 71718992 IC50 > 60000 nM T79591 CZ3WG5 71718993 IC50 > 60000 nM T79591 CE6X2K 71718994 IC50 > 60000 nM T79591 C1IH2Q 71718995 IC50 > 60000 nM T79591 CN1RW4 71718996 IC50 > 60000 nM T79591 CKA36P 71718997 IC50 > 60000 nM T79591 C8LWP5 71719585 IC50 > 60000 nM T79591 CQ6BL0 71719586 IC50 > 60000 nM T79591 CFO1J2 71719587 IC50 > 60000 nM T79591 CT0DH9 71719588 IC50 > 60000 nM T79591 C3BT7V 71719589 IC50 > 60000 nM T79591 CBY36L 71719590 IC50 > 60000 nM T79591 C5SPB2 71719591 IC50 > 60000 nM T79591 CYNI30 71719592 IC50 > 60000 nM T79591 CJ5O6Q 71719593 IC50 > 60000 nM T79591 C7EKV1 71719594 IC50 > 60000 nM T79591 CB7O4D 71719597 IC50 > 60000 nM T79591 CD98PS 71719598 IC50 > 60000 nM T79591 CQ7U4O 71719599 IC50 > 60000 nM T79591 CXDE81 71719600 IC50 > 60000 nM T79591 CDM58X 71719601 IC50 > 60000 nM T79591 CCV8I1 71719602 IC50 > 60000 nM T79591 CH1EB5 71719603 IC50 > 60000 nM T79591 CX46KH 71719604 IC50 > 60000 nM T79591 C7KER0 71720182 IC50 = 44000 nM T79591 C0DYJ3 71720183 IC50 = 25000 nM T79591 CY4J2C 71720184 IC50 = 29000 nM T79591 C4Z0VS 71720185 IC50 > 60000 nM T79591 C5H0WP 71720186 IC50 > 60000 nM T79591 C9B4SP 71720187 IC50 > 60000 nM T79591 CHFZ51 71720188 IC50 > 60000 nM T79591 C2FM0U 71720189 IC50 > 60000 nM T79591 CUG52N 71720190 IC50 > 60000 nM T79591 CV1US9 71720192 IC50 > 60000 nM T79591 C7X8QB 71720193 IC50 > 60000 nM T79591 CB56IU 71720826 IC50 > 60000 nM T79591 CS5R7G 71720827 IC50 > 60000 nM T79591 CTF8D3 71720828 IC50 > 60000 nM T79591 CZ71PL 71720830 IC50 > 60000 nM T79591 C0Y9CT 71720831 IC50 > 60000 nM T79591 CP0G7O 73054742 EC50 = 450 nM T79591 CBJ8C9 73055020 EC50 = 39 nM T79591 CCO4X8 73055021 EC50 = 180 nM T79591 CZ8RJ5 73055022 EC50 = 100 nM T79591 C36LIJ 73055023 IC50 > 10000 nM T79591 C25DRF 73055024 IC50 = 230 nM T79591 C27TWJ 76313972 IC50 > 30000 nM T79591 CO3KL0 118726602 Ki = 13.45 nM T79591 C45QSH 118726603 Ki = 16.33 nM T79591 CWQE31 118726604 Ki = 7.74 nM T79591 CZOI45 118726605 Ki = 1.09 nM T79591 C1QZ8J 118726606 Ki = 0.35 nM T79591 C0A9JB 118726607 Ki = 2.05 nM T79591 C94RVF 118726608 Ki = 0.38 nM T79591 C8IDF7 118726609 Ki = 2.77 nM T79591 C4KY2I 118726610 Ki = 0.51 nM T79591 CEW5K8 118726611 Ki = 9.98 nM T79591 CM2R8J 118726612 Ki = 36.53 nM T79591 CZM9O6 118726613 Ki = 32.33 nM T79591 CK8RB5 118726614 Ki = 46.55 nM T79591 CJA6K2 118726615 Ki = 89.89 nM T79591 C2J8PF 118726616 Ki = 199.97 nM T79591 CH1FA8 135528521 IC50 = 32 nM T79591 C0FWQ7 135559141 IC50 = 1513.56 nM T79591 CU20KW 135559142 IC50 = 144.54 nM T79591 CW9R4B 135559143 IC50 = 562.34 nM T79591 CCF02H 145964530 IC50 = 8400 nM T79591 C56SHA 145964597 IC50 = 5400 nM T79591 C5H8EZ 145965425 IC50 = 4200 nM T79591 C98CHS 145977976 IC50 = 10100 nM T79591 D01HAZ 23635364 IC50 = 6900 nM T79591 D01NTN 11350323 IC50 = 1096.48 nM T79591 D01WVE 9872203 IC50 = 2200 nM T79591 D02CGG 44435789 IC50 = 39100 nM T79591 D03VOM 3092218 IC50 = 10600 nM T79591 D03XCG 23635367 IC50 = 25800 nM T79591 D05FRX 11153607 IC50 = 700 nM T79591 D05XMM 44186304 IC50 = 16800 nM T79591 D05ZJC 9925361 IC50 = 26000 nM T79591 D06IJW 23635362 IC50 = 4100 nM T79591 D07MAF 21653696 IC50 = 7400 nM T79591 D08BQI 11291923 IC50 = 19952.62 nM T79591 D09XOC 23635858 IC50 = 4200 nM T79591 D0A5XG 10027822 IC50 = 950 nM T79591 D0G7HF 23635860 IC50 = 33200 nM T79591 D0H6BV 24843916 IC50 = 7700 nM T79591 D0I2GK 71212 IC50 = 0.24 nM T79591 D0I7DH 23635476 IC50 = 18900 nM T79591 D0J0MD 23635730 IC50 = 17500 nM T79591 D0Q9ZN 23648092 IC50 = 680 nM T79591 D0U0GY 44435784 IC50 = 23000 nM T79591 D0U9JC 44435785 IC50 = 21400 nM T79591 D0YU9Z 14899645 IC50 = 28100 nM T79591 D0ZX0Y 23635856 IC50 = 16700 nM T25608 D0Q5XX 445580 EC50 = 11700 nM T25608 D0UE9X 5280933 EC50 = 4620 nM T25608 D0EO2C 51049992 Ki = 4.7 nM T25608 D0V1WQ 24857286 EC50 = 1.9 nM T25608 CKRG59 10466 EC50 = 20892.96 nM T25608 CWY93I 37289 EC50 = 18620.87 nM T25608 C80LUR 154005 EC50 = 2190 nM T25608 CXH9K8 169433 EC50 > 100000 nM T25608 CF1W7M 233085 EC50 > 50118.72 nM T25608 CC05OD 561372 EC50 = 457.09 nM T25608 C19ADF 643684 EC50 = 11481.54 nM T25608 CA9GQ6 674995 IC50 = 12882.5 nM T25608 CZN6S9 743974 EC50 > 31622.78 nM T25608 C5IW8B 763016 EC50 = 24600 nM T25608 CK4OG8 797771 EC50 = 16700 nM T25608 C8MF6P 805130 IC50 = 2800 nM T25608 CQE21M 818213 EC50 = 16100 nM T25608 CS4H3F 853224 EC50 = 970 nM T25608 C1M7UY 1201156 EC50 = 16800 nM T25608 C4H7CT 1201222 EC50 = 22600 nM T25608 C1ZC6G 1202260 EC50 = 19000 nM T25608 CAIT59 1622278 EC50 = 3200 nM T25608 CP29AK 1646307 EC50 = 12200 nM T25608 C3HK9O 1855223 EC50 = 15100 nM T25608 C9T2OI 2214962 EC50 = 14500 nM T25608 CDU19P 2233248 IC50 = 5300 nM T25608 CB53NT 2843133 IC50 = 8128.31 nM T25608 CTUP01 3514336 EC50 = 5000 nM T25608 CG62ZB 4671033 IC50 = 10000 nM T25608 CQC0E6 4987566 EC50 = 8200 nM T25608 COT13S 5312743 EC50 > 100000 nM T25608 C7ASQ0 5312744 EC50 > 100000 nM T25608 C5YM6G 5332902 IC50 = 251.19 nM T25608 CMZY13 5353640 EC50 = 240 nM T25608 CED08V 9889284 EC50 > 10000 nM T25608 C13JXE 10131213 EC50 = 1258.93 nM T25608 CNZ5W7 10176767 EC50 > 100000 nM T25608 CZ2TJ7 10266133 EC50 = 8810 nM T25608 C15GQR 10292451 EC50 = 7.2 nM T25608 CN2WQ6 11190525 EC50 = 14 nM T25608 CZ3I5E 11203294 Ki = 16 nM T25608 COJW03 11226058 Ki = 15 nM T25608 CNS3C5 11236925 Ki = 20 nM T25608 CE6P9V 11245322 EC50 = 12.3 nM T25608 CG76JQ 11265145 EC50 = 9332.54 nM T25608 C8FV4O 11271473 Ki = 43 nM T25608 CRB69Z 11316164 EC50 = 288.4 nM T25608 CT68IQ 11327107 EC50 = 49 nM T25608 C3N5JU 11398822 EC50 = 15 nM T25608 CV9HT4 11489259 Ki = 21 nM T25608 CWR98I 11507535 EC50 = 8890 nM T25608 C8D7IB 11674915 EC50 = 6.7 nM T25608 CKV9W3 11739868 EC50 = 562.34 nM T25608 C49KIE 11750823 EC50 = 302 nM T25608 CWC60K 11773976 EC50 = 12.59 nM T25608 CIQ15K 11961321 EC50 = 7.6 nM T25608 CP1Q3H 12002185 Ki = 20 nM T25608 CDG28M 12002201 Ki = 19 nM T25608 C2RG8P 12002202 Ki = 18 nM T25608 CBJ23P 14454530 EC50 > 100000 nM T25608 C8GT5Q 15602772 EC50 = 3.8 nM T25608 CZ2SC0 15603739 EC50 = 61 nM T25608 CIK6A2 15603842 EC50 = 11 nM T25608 CF8Q7T 15603946 EC50 = 16 nM T25608 CHYT81 15603947 EC50 = 65 nM T25608 C9B1IW 15604310 EC50 = 1.3 nM T25608 C4QI2Y 15604434 EC50 = 69 nM T25608 CVT35C 15659412 EC50 = 8000 nM T25608 C59DBZ 15659413 EC50 = 6000 nM T25608 CP0SB8 16110418 EC50 > 10000 nM T25608 C3JYS8 16661950 IC50 = 6300 nM T25608 CECK07 17754443 EC50 = 0.1 nM T25608 CQS7M8 19705952 EC50 = 3500 nM T25608 CX2Z9H 20331242 EC50 = 1000 nM T25608 C5A4VN 20993091 EC50 = 1358 nM T25608 CV2BL0 21322577 EC50 = 2484 nM T25608 C46RPA 22036572 EC50 = 3200 nM T25608 C0M3CA 23082739 EC50 = 35 nM T25608 C1GQ3U 23082789 EC50 = 3500 nM T25608 CQK3G8 23082861 EC50 = 1700 nM T25608 C2DB9E 23082877 EC50 = 20 nM T25608 CPL70G 23083015 Ki = 520 nM T25608 C40SFL 23083189 EC50 = 40 nM T25608 CLPE35 23083190 EC50 = 47 nM T25608 CMYD48 23083193 EC50 = 38 nM T25608 CL26XS 23111666 EC50 = 39 nM T25608 C1HEB2 23111668 EC50 = 28 nM T25608 CPFD82 23111671 EC50 = 180 nM T25608 CTK9V6 23111682 Ki = 18 nM T25608 CC3H7G 23111689 EC50 = 29 nM T25608 C27VQJ 23111693 EC50 = 24 nM T25608 CPOD26 23111694 Ki = 6.9 nM T25608 CHT0Q8 23111704 EC50 = 23 nM T25608 C1JK5B 23111708 EC50 = 1700 nM T25608 CT38PB 23111732 EC50 > 10000 nM T25608 C1L6RM 23111734 EC50 = 28 nM T25608 CT32AF 23111754 EC50 = 540 nM T25608 C29JHR 23111764 Ki > 10000 nM T25608 CPSD80 23111766 EC50 = 33 nM T25608 CRY9S6 23111781 EC50 = 22 nM T25608 CE71HA 23111791 EC50 = 21 nM T25608 CA1OT7 23136315 EC50 = 1100 nM T25608 CE3JI2 23136363 EC50 = 34 nM T25608 CV2HD8 23136401 EC50 = 3837 nM T25608 CD4VG3 23136411 EC50 = 134.9 nM T25608 CW3AM0 23136477 EC50 = 1905.46 nM T25608 CJGL28 23157191 EC50 = 6.3 nM T25608 CS7T9B 23157282 Ki = 18 nM T25608 CXSW42 23157589 EC50 = 520 nM T25608 CTE01K 23159839 EC50 = 2700 nM T25608 CQDI97 23159846 EC50 = 2700 nM T25608 CSO9X7 23159951 EC50 = 530 nM T25608 CTQ53W 23346507 EC50 = 758.58 nM T25608 C54OXK 23642299 EC50 = 16 nM T25608 CIA3X8 23699039 EC50 > 100000 nM T25608 CI2K8W 24825479 EC50 = 50.12 nM T25608 C4UM5N 24825480 EC50 = 398.11 nM T25608 C0JYX7 24825481 EC50 = 1122.02 nM T25608 CATZ28 24825482 EC50 = 16595.87 nM T25608 CI30KR 24825483 EC50 = 3981.07 nM T25608 CY0F4L 24825484 EC50 = 218.78 nM T25608 CCG12J 24825485 EC50 = 39.81 nM T25608 C1IZD5 24825486 EC50 = 501.19 nM T25608 C06XPY 24825487 EC50 = 1584.89 nM T25608 CK91WQ 24825488 EC50 < 31622.78 nM T25608 CI7A0X 24825489 EC50 = 12302.69 nM T25608 CQJV71 24825490 EC50 = 251.19 nM T25608 CF80AP 24825491 EC50 = 794.33 nM T25608 CHX09F 24825492 EC50 = 173.78 nM T25608 C49IJM 24825493 EC50 = 1995.26 nM T25608 CTG8N0 24825494 EC50 = 1995.26 nM T25608 C18UWB 24825495 EC50 = 3981.07 nM T25608 CVT5A0 24825496 EC50 = 3981.07 nM T25608 CJS5P6 24825497 EC50 = 5011.87 nM T25608 CWX6U2 24825498 EC50 = 5011.87 nM T25608 C9YCR5 24825499 EC50 < 31622.78 nM T25608 CBG1E0 24825500 EC50 < 31622.78 nM T25608 C9S8OB 24825501 EC50 < 31622.78 nM T25608 C8WMP2 24825502 EC50 < 31622.78 nM T25608 C2L0ON 24825503 EC50 < 31622.78 nM T25608 C9WHV1 24825504 EC50 < 31622.78 nM T25608 CDZ26M 24825505 EC50 = 1258.93 nM T25608 C37KYZ 24825506 EC50 < 31622.78 nM T25608 CG7E5P 24825507 EC50 < 31622.78 nM T25608 CW0VI4 24825508 EC50 < 31622.78 nM T25608 C56XKE 24825509 EC50 = 97.72 nM T25608 CK12YG 24857285 EC50 = 13 nM T25608 C31OGF 24857375 EC50 = 16 nM T25608 CJ1V3Z 24857376 Ki = 12 nM T25608 CK1E7M 24860552 EC50 = 302 nM T25608 C2L8YX 24897670 EC50 = 3.6 nM T25608 CS8T2B 25109512 EC50 = 21000 nM T25608 C32MTA 25149900 EC50 = 5623.41 nM T25608 CZ39BV 25149901 EC50 = 95.5 nM T25608 CK8IX2 25150011 EC50 = 354.81 nM T25608 C5JO1X 25150012 EC50 = 91.2 nM T25608 CG40IY 25150013 EC50 = 89.13 nM T25608 C3FM2H 25150015 EC50 = 87.1 nM T25608 CE7O1K 25150016 EC50 = 74.13 nM T25608 C61UMS 25150018 EC50 = 3715 nM T25608 CMS8T4 25150113 EC50 = 1096.48 nM T25608 CY51JZ 25150114 EC50 = 512.86 nM T25608 CD25SW 25150117 EC50 = 891.25 nM T25608 C1LDN0 25150118 EC50 = 58.88 nM T25608 CYA5N2 25150119 EC50 = 154.88 nM T25608 CYO95C 25150120 EC50 = 43.65 nM T25608 CQB54I 25150121 EC50 = 107.15 nM T25608 C4B8YC 25261464 EC50 = 1100 nM T25608 C6PAV0 25261467 EC50 = 2100 nM T25608 CJZ51K 25272661 IC50 = 2100 nM T25608 CBXQ30 25766502 EC50 = 18800 nM T25608 C5J3YP 42603138 EC50 = 260 nM T25608 C7SGQ2 44223813 EC50 = 500 nM T25608 CL6SX0 44244518 IC50 = 20 nM T25608 CBKM86 44409608 EC50 < 10000 nM T25608 CYB4F6 44409612 EC50 < 10000 nM T25608 CT5AW0 44409664 EC50 = 48.98 nM T25608 CM5VG7 44409665 EC50 = 39.81 nM T25608 C5YKA3 44409670 EC50 = 100 nM T25608 CDRN85 44409676 EC50 = 14.79 nM T25608 CRJZ90 44409677 EC50 = 6.918 nM T25608 CCY03M 44409690 EC50 = 67.61 nM T25608 CLK8N5 44409695 EC50 < 10000 nM T25608 C9YVL7 44409697 EC50 = 323.59 nM T25608 C3Y8JC 44409698 EC50 = 173.78 nM T25608 CDZ92U 44409699 EC50 = 125.89 nM T25608 C8X0EI 44409702 EC50 = 114.82 nM T25608 C0HB4O 44409703 EC50 = 4.467 nM T25608 CMOF79 44409722 EC50 = 2.455 nM T25608 CO6ZV2 44409728 EC50 = 100 nM T25608 C54KUR 44409729 EC50 = 354.81 nM T25608 CIAY19 44409843 EC50 = 10.96 nM T25608 CU92HA 44409844 EC50 = 66.07 nM T25608 CS6RX1 44409877 EC50 = 51.29 nM T25608 C1IT3N 44409878 EC50 = 12.88 nM T25608 CIKM52 44409883 EC50 = 204.17 nM T25608 CFH0P9 44409906 EC50 = 2041 nM T25608 CR0M8C 44409915 EC50 < 10000 nM T25608 C6NF2X 44409916 EC50 = 58.88 nM T25608 CSO5Z9 44409926 EC50 = 9.12 nM T25608 C5RV8P 44409927 EC50 = 53.7 nM T25608 CP6CR2 44409928 EC50 < 10000 nM T25608 C6EL9I 44409929 EC50 = 144.54 nM T25608 CQ8W9J 44409933 EC50 = 36.31 nM T25608 CK8X5D 44571477 EC50 = 970 nM T25608 CX42DJ 44572033 EC50 = 19 nM T25608 CA3JQ8 44572094 EC50 = 260 nM T25608 CVS9U3 44572096 EC50 < 100 nM T25608 CMO3C5 44572097 EC50 = 10 nM T25608 C5KRH4 44589697 EC50 = 85.11 nM T25608 C0LQS4 44591612 IC50 = 10 nM T25608 C3DOW2 44591613 IC50 = 12 nM T25608 CR35KT 44591627 IC50 = 96 nM T25608 CAK8V6 44591628 IC50 = 2 nM T25608 CCWB82 44591629 IC50 = 3 nM T25608 CWR61H 44591630 IC50 = 29 nM T25608 CP4BC2 44591651 IC50 = 156 nM T25608 CJ03XW 44591652 IC50 = 4 nM T25608 C3ZP1K 44591689 IC50 = 89 nM T25608 CT5X0J 44591690 IC50 = 228 nM T25608 C58MHZ 44591691 IC50 = 119 nM T25608 CKHA83 44591692 IC50 = 13 nM T25608 C8KZF9 44591693 IC50 = 10 nM T25608 C7FR4Z 44591719 IC50 = 10 nM T25608 CJ7L9M 44634022 EC50 = 13182.57 nM T25608 CBZG45 44634023 EC50 = 6025.6 nM T25608 CI4SA8 44634024 EC50 = 295.12 nM T25608 CIA25J 45107281 EC50 = 6.2 nM T25608 CA0B5S 45107282 EC50 = 3.9 nM T25608 C1IYL9 45107307 EC50 = 20 nM T25608 C5IAO0 45107311 EC50 = 5 nM T25608 CJN6F1 45107312 EC50 = 3.7 nM T25608 C16NSP 45107317 EC50 = 12 nM T25608 C4UQ9M 45107318 EC50 = 29 nM T25608 CYQC63 45107320 EC50 = 21 nM T25608 CYL14S 45107323 EC50 = 9.9 nM T25608 CHZ23U 45107324 EC50 = 13 nM T25608 C0AHF2 45107476 EC50 = 5.3 nM T25608 CU35QF 45254027 EC50 = 81 nM T25608 C7PRU9 45377306 EC50 > 30000 nM T25608 C3E9VN 46231386 EC50 = 6451 nM T25608 CP93KX 46232307 EC50 = 10 nM T25608 CZ7U2W 46869922 EC50 = 14 nM T25608 CYTP35 46892131 IC50 > 100000 nM T25608 C8XSB6 51031010 Ki = 39 nM T25608 CC91LO 51349860 EC50 = 300 nM T25608 CP9JN0 51349861 EC50 = 154.88 nM T25608 CW1D0B 51349990 EC50 = 300 nM T25608 CIX80K 51349991 EC50 = 260 nM T25608 CNP73Q 51349992 EC50 = 40 nM T25608 C3UA4P 51349993 EC50 = 45 nM T25608 CXR9O8 51350134 EC50 = 1800 nM T25608 CQHP45 51350135 EC50 = 170 nM T25608 CSU3C9 51350136 EC50 = 170 nM T25608 C7PVZ1 51350137 EC50 = 32 nM T25608 CAS51V 51350138 EC50 = 5.7 nM T25608 C1FC4M 51350139 EC50 = 30 nM T25608 CYUQ87 51350140 EC50 = 30 nM T25608 C5SVW3 51350270 EC50 = 120 nM T25608 CCA03I 51350271 EC50 = 240 nM T25608 C4EGI3 51350272 EC50 = 16.6 nM T25608 CO39YF 51350273 EC50 = 82 nM T25608 CRMT67 51350274 EC50 = 120 nM T25608 CYO4V0 51350404 EC50 = 20 nM T25608 C5IT1B 51350405 EC50 = 30 nM T25608 CIY29U 51350406 EC50 = 19 nM T25608 C7EUM1 51350407 EC50 = 9.9 nM T25608 CFYV70 51351414 EC50 = 320 nM T25608 CQIY23 53248846 IC50 = 12 nM T25608 C9MHR0 53248847 EC50 = 113 nM T25608 C7AI4W 54580132 EC50 = 446.68 nM T25608 C4MOV9 54580624 EC50 = 94 nM T25608 C4U8CJ 54580625 EC50 = 114 nM T25608 C3AYC2 54580626 EC50 = 2820 nM T25608 CB1E0U 54580627 IC50 = 10000 nM T25608 CYT3I8 54581632 EC50 = 970 nM T25608 CBJ8D3 54581633 IC50 = 342 nM T25608 C4YRU1 54582145 EC50 = 69.18 nM T25608 C7W8IE 54582148 EC50 = 6309.57 nM T25608 CS03YA 54582149 EC50 = 524.81 nM T25608 CKV29F 54582150 EC50 = 1071.52 nM T25608 CA3JY5 54582628 IC50 = 36 nM T25608 CXQ1S2 54582629 IC50 = 13 nM T25608 C6XPK4 54582630 EC50 = 108 nM T25608 C9K2AQ 54582631 IC50 = 433 nM T25608 C4HD9E 54583097 EC50 = 3311.31 nM T25608 CU5K1Y 54583098 EC50 = 53.7 nM T25608 CJN07Y 54583099 EC50 = 125.89 nM T25608 CYQK29 54583581 EC50 = 1578 nM T25608 C6K1CE 54583582 EC50 = 51 nM T25608 CS26NZ 54584097 EC50 = 12589.25 nM T25608 C31NYG 54584098 EC50 = 75.86 nM T25608 C2N9LK 54584570 EC50 = 686 nM T25608 CDYZ19 54585039 EC50 = 165.96 nM T25608 CHQ70W 54586010 EC50 = 21379.62 nM T25608 C03CFM 54586011 EC50 = 83.18 nM T25608 C4HWR8 54586484 IC50 = 23 nM T25608 C7A1CM 54586485 IC50 = 211 nM T25608 CKJ67Q 54586486 EC50 = 31 nM T25608 C91ENI 54586982 EC50 = 3630.78 nM T25608 CR4XH7 54586983 EC50 = 2454.71 nM T25608 C2W0GK 54586984 EC50 = 186.21 nM T25608 CXO2A9 54669771 EC50 = 40.74 nM T25608 C7WX2N 54757513 EC50 = 4073.8 nM T25608 CY51XQ 54757514 EC50 = 6165.95 nM T25608 C68IMN 54757515 EC50 = 10964.78 nM T25608 C16BGK 54757516 EC50 = 602.56 nM T25608 C7L8YN 54757517 EC50 = 707.95 nM T25608 C7Y5OB 54757518 EC50 = 660.69 nM T25608 CZ1M3Q 54757519 EC50 > 100000 nM T25608 CGL9J4 54757619 EC50 = 9120.11 nM T25608 CN87XO 54757620 EC50 = 9549.93 nM T25608 CHO24D 54757621 EC50 = 4265.8 nM T25608 CHGX78 54757622 EC50 = 2754.23 nM T25608 CV1L0F 54757623 EC50 = 3890.45 nM T25608 C3TE0M 54757624 EC50 = 251.19 nM T25608 C3BDI6 54757625 EC50 = 75.86 nM T25608 C1IHM9 54757626 EC50 = 1122.02 nM T25608 C4CFX9 54757627 EC50 = 512.86 nM T25608 CT53SC 54757732 EC50 = 524.81 nM T25608 CAN93K 54757733 EC50 = 478.63 nM T25608 C32BGX 54757734 EC50 = 186.21 nM T25608 C83TPD 54757735 EC50 = 1071.52 nM T25608 C2P9QA 54757736 EC50 = 177.83 nM T25608 CJ5UA0 54757737 EC50 = 120.23 nM T25608 CJV75N 54757738 EC50 = 134.9 nM T25608 CME5K8 54757739 EC50 = 316.23 nM T25608 C84XHT 54757829 EC50 = 794.33 nM T25608 CRU9P0 54757830 EC50 = 79.43 nM T25608 CBZ7Q3 54757831 EC50 = 43.65 nM T25608 CD8S9Y 56640072 EC50 < 10 nM T25608 CRN7Q3 56680363 EC50 = 42.66 nM T25608 C04CIX 57325674 EC50 = 69 nM T25608 C0NS2J 57325678 EC50 = 570 nM T25608 CKD80Z 57325840 EC50 = 960 nM T25608 CHW75L 57325841 EC50 = 84 nM T25608 CVKL67 57325842 EC50 = 140 nM T25608 CA7IH2 57325916 EC50 = 510 nM T25608 CU8JI5 57325917 EC50 = 91 nM T25608 C0OS7K 57325919 Ki > 10000 nM T25608 CSQB56 57390187 EC50 = 6200 nM T25608 C36RSI 57390188 EC50 = 240 nM T25608 CE48GA 57391957 EC50 = 900 nM T25608 CLQ37O 57391958 EC50 = 1200 nM T25608 CWE7D8 57391959 EC50 = 27000 nM T25608 CVCZ15 57391960 EC50 = 1200 nM T25608 CG6M0N 57393689 EC50 = 580 nM T25608 C2MPC4 57393690 EC50 = 6700 nM T25608 CH17PJ 57393691 EC50 = 64 nM T25608 C31SBK 57393692 EC50 = 25 nM T25608 C3GD1S 57394144 EC50 = 360 nM T25608 CS5X0U 57395404 EC50 = 1100 nM T25608 C81BDZ 57397248 EC50 = 3200 nM T25608 CDH46R 57398937 EC50 = 120 nM T25608 CKB1R2 57398938 EC50 = 58 nM T25608 C2FH6J 57400636 EC50 = 620 nM T25608 CUGV01 57400637 EC50 = 110 nM T25608 CC5TA0 57402427 EC50 = 180 nM T25608 C9AZJ4 57413287 Ki = 99 nM T25608 CS2CD8 57413288 EC50 = 12 nM T25608 CY7BM5 57413289 EC50 = 15 nM T25608 CQP6Y0 57413290 EC50 = 13 nM T25608 C9R1CF 57413373 EC50 = 4.5 nM T25608 CRP91W 57413375 Ki = 12 nM T25608 CRQ45D 57414267 EC50 = 16 nM T25608 CY6I2L 57414268 Ki = 280 nM T25608 CSOE32 57414401 Ki = 21 nM T25608 CI8O0Z 57414402 EC50 = 18 nM T25608 CFI28H 57414403 Ki = 270 nM T25608 C38LHP 57414404 EC50 = 39 nM T25608 CFT94Q 57414405 EC50 = 22 nM T25608 CYT0J7 57414538 EC50 = 290 nM T25608 C7LIV6 57414539 EC50 = 14 nM T25608 C35ADQ 57414540 EC50 = 17 nM T25608 C21PIC 57414542 Ki = 8.8 nM T25608 CN53WX 57414543 Ki = 12 nM T25608 CCT57F 57414676 Ki = 15 nM T25608 C3FY1L 57414677 Ki = 11 nM T25608 CQ7B5A 57414678 EC50 = 29 nM T25608 C1SAB3 57414679 EC50 = 18 nM T25608 CL0NP8 57414680 EC50 = 19 nM T25608 CY5O1Q 57521702 EC50 = 602.56 nM T25608 CDW9N4 57521808 EC50 = 524.81 nM T25608 CZL1W6 57521809 EC50 = 630.96 nM T25608 CT06GY 57521810 EC50 = 933.25 nM T25608 C9S5CH 57521811 EC50 = 512.86 nM T25608 C2DUX1 57521812 EC50 = 851.14 nM T25608 CD8G6M 57521813 EC50 = 1148.15 nM T25608 CDRW60 57521814 EC50 = 2041.74 nM T25608 C76WSM 57521913 EC50 = 4466.84 nM T25608 C9O0LB 57521914 EC50 = 630.96 nM T25608 CS6B7Q 57521915 EC50 = 3548.13 nM T25608 CV8F2A 57521916 EC50 = 602.56 nM T25608 CBTP21 57521917 EC50 = 109.65 nM T25608 CPZQ75 57521918 EC50 = 407.38 nM T25608 CH9K1N 57521919 EC50 = 954.99 nM T25608 C7PEI1 57705531 EC50 = 680 nM T25608 CEY7A5 57705555 EC50 = 110 nM T25608 C51GWM 57705575 EC50 = 1960 nM T25608 C9KPA0 57705648 EC50 = 790 nM T25608 CT8RL2 57705679 EC50 = 90 nM T25608 CGA5E7 57705719 EC50 = 740 nM T25608 C7K4VJ 57705749 EC50 = 140 nM T25608 CM17AI 57705806 EC50 = 120 nM T25608 CF7V9T 57705838 EC50 = 105 nM T25608 CLY04B 57705851 EC50 = 120 nM T25608 C86ICX 57705863 EC50 = 900 nM T25608 C6D8IA 57705880 EC50 = 76 nM T25608 C9F5IV 57705939 EC50 = 227 nM T25608 C3FY4G 57706009 EC50 = 770 nM T25608 CJ70CQ 57706031 EC50 = 690 nM T25608 CK2O3H 57706032 EC50 = 370 nM T25608 C2SFX9 57706097 EC50 = 1830 nM T25608 C8QR5G 57706220 EC50 = 147 nM T25608 C8OH5L 57706227 EC50 = 68 nM T25608 CBDC31 57706280 EC50 = 90 nM T25608 CF35CK 57706451 EC50 = 1410 nM T25608 CPV92M 57706502 EC50 = 310 nM T25608 CBYZ29 57706588 EC50 = 370 nM T25608 C49KUF 57706620 EC50 = 100 nM T25608 C5PZC7 57706642 EC50 = 420 nM T25608 CM97RW 57706720 EC50 = 2200 nM T25608 C5Z4XH 57706778 EC50 = 13 nM T25608 CTH1L7 57706902 EC50 = 88 nM T25608 CG5EK4 57707025 EC50 = 80 nM T25608 CMNJ56 57707110 EC50 = 93 nM T25608 C6V0SY 57707179 EC50 = 100 nM T25608 CQC7P4 57707214 EC50 = 114 nM T25608 CB9C0R 57787398 EC50 = 380 nM T25608 C68FGV 57839754 EC50 > 30000 nM T25608 C20WOJ 58137077 IC50 = 630.96 nM T25608 CRVQ03 58172957 EC50 = 370 nM T25608 C9T0PH 58172961 EC50 = 23 nM T25608 C01QZR 58172969 EC50 = 63 nM T25608 C70RHJ 58172971 EC50 = 1500 nM T25608 C6UOC4 58172978 EC50 = 98 nM T25608 C3WLT5 58172979 EC50 = 27 nM T25608 CYR85D 58172984 EC50 = 970 nM T25608 CUJ5W2 58172986 EC50 = 31 nM T25608 C57AXW 58172988 EC50 = 3100 nM T25608 CJIL12 58172989 EC50 = 49 nM T25608 C02LMG 58172991 EC50 = 89 nM T25608 CQBS49 58172998 EC50 = 210 nM T25608 CQH03N 58172999 EC50 = 190 nM T25608 CM6J1X 58173000 EC50 = 82 nM T25608 CO6P0D 58173002 EC50 = 12 nM T25608 C3LA7I 58218542 EC50 = 560 nM T25608 C0MKH5 58218551 EC50 = 150 nM T25608 CG8U2O 58218571 EC50 = 190 nM T25608 CM7AS3 58218581 EC50 = 360 nM T25608 C68DGL 58218607 EC50 = 140 nM T25608 CWQU02 58218608 EC50 = 67 nM T25608 CS6W8J 58218630 EC50 = 340 nM T25608 CP60JL 58218638 EC50 = 74 nM T25608 CLEV75 58218640 EC50 = 120 nM T25608 C8U1WQ 58218651 Ki = 35 nM T25608 CR0EU5 58218655 EC50 = 2300 nM T25608 C05QYV 58218671 EC50 = 1700 nM T25608 CC0R5G 58218672 EC50 = 570 nM T25608 C9R0HB 58218673 Ki = 13 nM T25608 C3AH2Y 58218694 EC50 = 74 nM T25608 CU0N5T 58218699 EC50 = 3500 nM T25608 C9SHX4 58218709 Ki = 60 nM T25608 C1YUI5 58218726 EC50 = 82 nM T25608 C19SRZ 58218740 EC50 = 150 nM T25608 CMZL87 58319089 EC50 = 2041.74 nM T25608 CUW17O 58319094 EC50 = 83.18 nM T25608 CAEP71 58319098 EC50 = 123.03 nM T25608 C6BK9A 58319107 EC50 = 1000 nM T25608 C6BEP7 58319118 EC50 = 218.78 nM T25608 CR2V9U 58319121 EC50 = 151.36 nM T25608 C6RF5S 58319126 EC50 = 186.21 nM T25608 CX6YK3 58319127 EC50 = 446.68 nM T25608 CU3T9M 58319134 EC50 = 70.79 nM T25608 CB0FY8 58319135 EC50 = 89.13 nM T25608 CB47WD 58319138 EC50 = 16218.1 nM T25608 CP7CY3 58319139 EC50 = 416.87 nM T25608 CT29VJ 58319142 EC50 = 575.44 nM T25608 CU91ZL 58379717 EC50 = 98 nM T25608 C9O4GC 58379893 EC50 = 212 nM T25608 C7OXV2 58379987 EC50 = 105 nM T25608 C5TH9M 58380220 EC50 = 250 nM T25608 CT09DC 58380255 EC50 = 92 nM T25608 COQ92J 58380284 EC50 = 820 nM T25608 CF4B2G 58380381 EC50 = 150 nM T25608 C6GZ3H 58758896 EC50 = 130 nM T25608 C1B5PX 59132613 EC50 = 120 nM T25608 CVI53W 59132740 EC50 = 400 nM T25608 CACS13 59590781 EC50 = 3.4 nM T25608 CU0K4Q 59590895 EC50 = 6.7 nM T25608 CEOP18 60195036 EC50 = 17.38 nM T25608 CS4X9Y 60195037 EC50 = 14.79 nM T25608 CR9C7I 60195038 EC50 = 9.333 nM T25608 CX30BG 60195039 EC50 = 23.44 nM T25608 C7S3HJ 60195040 EC50 = 17.78 nM T25608 CQLD97 60195125 Ki = 4.365 nM T25608 C9DH3R 66562286 EC50 = 35.48 nM T25608 C16SUO 66562287 EC50 = 81.28 nM T25608 CB75OA 66562288 EC50 = 20 nM T25608 CEK8U4 66562289 EC50 = 37.15 nM T25608 C04XUT 66562385 EC50 = 33.11 nM T25608 CI73FC 66562386 EC50 = 16.98 nM T25608 CH5JZ6 66562387 EC50 = 1445.44 nM T25608 CUI9P3 66562388 EC50 = 1949.84 nM T25608 C7D0FE 66562389 EC50 = 141.25 nM T25608 C1RBT5 66562390 EC50 = 144.54 nM T25608 CD0GO5 66562391 EC50 = 426.58 nM T25608 CI7WO1 66562392 EC50 = 38.02 nM T25608 CAU1G2 66562488 EC50 = 18.2 nM T25608 C9HQ8C 67058186 EC50 = 360 nM T25608 CM5IL7 67058222 EC50 = 13 nM T25608 CF0MW1 67058227 EC50 = 19 nM T25608 CK9N8S 67058273 EC50 = 62 nM T25608 CB8KF5 67058307 EC50 = 13 nM T25608 C6NIF3 67072752 EC50 = 19.95 nM T25608 C1BQH0 67085353 EC50 = 310 nM T25608 C5DMN9 67085761 Ki = 10 nM T25608 C6RZL9 67134965 IC50 = 2454.71 nM T25608 CN28HY 67359903 EC50 = 520 nM T25608 C13YCK 67361692 EC50 = 350 nM T25608 CPM76C 67972848 EC50 = 380 nM T25608 CYE04T 68265494 EC50 = 180 nM T25608 C3TM0C 68674201 EC50 = 330 nM T25608 CV82WY 68676271 EC50 = 190 nM T25608 C9X6PR 70522117 EC50 = 977.24 nM T25608 C61LQJ 70901463 EC50 = 3780 nM T25608 CNI46A 71257551 EC50 = 3 nM T25608 C68XRW 71449361 EC50 = 650 nM T25608 COA43P 71449362 EC50 = 2300 nM T25608 CYTQ78 71449363 EC50 = 2100 nM T25608 CEC1V0 71451164 EC50 = 1900 nM T25608 C0MW1K 71454737 EC50 = 1200 nM T25608 CP2VM5 71456495 EC50 = 2300 nM T25608 C1SNX9 71457285 Ki = 370 nM T25608 CG64XE 71458348 EC50 = 1310 nM T25608 C1AH6B 71460190 EC50 = 1200 nM T25608 CI5W0H 71460255 EC50 = 79 nM T25608 CI3Y2S 71460547 EC50 = 21.88 nM T25608 CF3T9Q 71461901 EC50 = 4000 nM T25608 CMZY24 71562312 EC50 = 1000 nM T25608 CS9BX3 71562313 EC50 = 2290.87 nM T25608 CTM07K 71562314 EC50 = 199.53 nM T25608 CVOS18 71562315 EC50 = 346.74 nM T25608 CY1H3I 71562316 EC50 = 144.54 nM T25608 CF2Y6B 71562317 EC50 = 138.04 nM T25608 C80VUQ 71562421 EC50 = 93.33 nM T25608 C0VXG7 71562422 EC50 = 309.03 nM T25608 CR38OD 71562423 EC50 = 138.04 nM T25608 C47QRK 71562424 EC50 = 524.81 nM T25608 C4OZ6V 71562526 EC50 = 338.84 nM T25608 CRP5U8 71562527 EC50 = 223.87 nM T25608 CJ7UZ1 71562637 EC50 = 95.5 nM T25608 C30LJD 71562638 EC50 = 40.74 nM T25608 CN21ZT 71562639 EC50 = 38.02 nM T25608 C6NV8H 71562640 EC50 = 812.83 nM T25608 C2YW9D 71562641 EC50 = 426.58 nM T25608 C4Y2MH 71562768 EC50 = 467.74 nM T25608 CDG40T 71562769 EC50 = 39.81 nM T25608 CKF3X1 71562770 EC50 = 190.55 nM T25608 C8TFI5 71562771 EC50 = 46.77 nM T25608 CHW16K 71562772 EC50 = 263.03 nM T25608 CY73IA 71562773 EC50 = 35.48 nM T25608 C3R0FO 71575419 EC50 = 13.5 nM T25608 CT1D2M 71612680 EC50 = 74.7 nM T25608 CXO1J4 71612681 EC50 = 73.2 nM T25608 CVN8E3 71612682 EC50 = 74.5 nM T25608 C0JNV8 71612683 EC50 = 54.7 nM T25608 C54LIA 71612684 EC50 > 10000 nM T25608 CE4CA6 71612685 EC50 = 36.4 nM T25608 CSBP81 71612894 EC50 = 105.1 nM T25608 CC41RU 71612895 EC50 = 63.7 nM T25608 CMRT56 71612896 EC50 = 55.9 nM T25608 CR1O3Q 71612897 EC50 = 282 nM T25608 C5S4OZ 71612898 EC50 = 46.5 nM T25608 CGKW10 71613092 EC50 = 67.5 nM T25608 CWM47R 71613093 EC50 = 82.4 nM T25608 CV3DW5 71613094 EC50 = 120.7 nM T25608 C1GF4I 71613095 EC50 = 94.8 nM T25608 CM98GB 71613096 EC50 = 145.2 nM T25608 CG6UJ1 71613311 EC50 = 52.9 nM T25608 C19YZB 71613312 EC50 = 30.1 nM T25608 CJY0H8 71613313 EC50 = 39.3 nM T25608 CYQ0D3 71613314 EC50 = 19.1 nM T25608 C2PX9O 71613315 EC50 = 66.7 nM T25608 CI6FY1 71613316 EC50 = 56.7 nM T25608 C7F9BO 71613515 EC50 = 111.1 nM T25608 CBI53Y 71613516 EC50 = 34.2 nM T25608 C0NPS8 71613517 EC50 = 219.8 nM T25608 CBS8D2 71613518 EC50 = 16 nM T25608 CYD54Q 71613519 EC50 = 190.5 nM T25608 C6O0IM 71613520 EC50 = 11.3 nM T25608 C36PAQ 71613521 EC50 = 30.4 nM T25608 C9L8NQ 71615467 EC50 = 122.6 nM T25608 C85KRA 71615468 EC50 = 56.2 nM T25608 C1F3EO 71615469 EC50 = 205.1 nM T25608 CD2IE1 71615470 EC50 = 125 nM T25608 CID4G7 71615666 EC50 = 65.4 nM T25608 C7G5TN 71615667 EC50 = 35.9 nM T25608 CEI6V4 71615668 EC50 = 38.7 nM T25608 CASF10 71615669 EC50 = 61.6 nM T25608 CXAC53 71615670 EC50 = 88 nM T25608 C8DUF7 71615671 EC50 = 132 nM T25608 C1PR6K 71655225 EC50 = 2137.96 nM T25608 CD6EU4 71655226 EC50 = 2511.89 nM T25608 C3XC7G 71655227 EC50 = 22.39 nM T25608 CJMF15 71655293 EC50 = 74.13 nM T25608 CL7BA0 71715951 EC50 < 100 nM T25608 C8F0DH 71816758 EC50 > 30000 nM T25608 CD15WX 71816759 EC50 > 30000 nM T25608 CN3E6S 71816760 EC50 > 30000 nM T25608 C7KN9H 71816761 EC50 = 1420 nM T25608 CMXI29 71816806 EC50 > 30000 nM T25608 CBLG16 71816808 EC50 = 2130 nM T25608 CD0AY7 73345869 EC50 = 18.2 nM T25608 C75PUZ 73345870 EC50 = 363.08 nM T25608 CQ6N0O 73348895 EC50 = 371.54 nM T25608 CPF43O 73354950 EC50 = 724.44 nM T25608 C68LKC 73356502 EC50 = 1380 nM T25608 CQ7T4B 73356514 EC50 = 616.6 nM T25608 CPMI97 73777069 EC50 > 10000 nM T25608 CC0V2Z 73777085 EC50 > 10000 nM T25608 CIX50H 73777111 EC50 > 10000 nM T25608 C9N7VS 73777135 EC50 > 10000 nM T25608 CH5CY8 73777153 EC50 = 6300 nM T25608 CAW6R9 73777156 EC50 = 2500 nM T25608 C0PV3T 73777174 EC50 > 10000 nM T25608 CEYQ78 73777175 EC50 = 8100 nM T25608 C3Y4IL 73891117 EC50 = 6 nM T25608 CR6D4C 75202601 EC50 = 2830 nM T25608 C0CH3I 75202609 EC50 = 530 nM T25608 CM68XD 75204006 EC50 = 190 nM T25608 C07LQH 75204360 EC50 = 210 nM T25608 CYEG23 75204485 EC50 = 940 nM T25608 C0B2NO 75204487 EC50 = 630 nM T25608 CY20UR 75511297 EC50 = 4000 nM T25608 CG3S0Z 75511298 EC50 = 2390 nM T25608 C2SQU1 75511299 EC50 = 2650 nM T25608 C14SZK 75511301 EC50 = 680 nM T25608 C60CGT 75511302 EC50 = 560 nM T25608 C23EHB 75511303 EC50 = 1070 nM T25608 CN3LD9 75511304 EC50 = 700 nM T25608 CX4OE5 75511305 EC50 > 100000 nM T25608 C14EYX 75511306 EC50 = 2670 nM T25608 CL1AJ5 75511307 EC50 = 1200 nM T25608 C6YA1G 75511308 EC50 = 2570 nM T25608 C6MA0F 75511310 EC50 = 210 nM T25608 CRL8X0 75511312 EC50 = 1260 nM T25608 C1W9FN 75511315 EC50 = 13100 nM T25608 C7WVJ5 75511316 EC50 = 3000 nM T25608 C9AQ8B 75511317 EC50 = 4580 nM T25608 C23YEG 76900387 EC50 = 70 nM T25608 CPT9V0 77845055 EC50 = 110 nM T25608 CI2DU6 82051616 EC50 = 11588 nM T25608 CE36PD 82051652 EC50 > 30000 nM T25608 C54DHY 85470884 EC50 = 3340 nM T25608 C6EZF9 85472225 EC50 = 3000 nM T25608 C4EVX7 85970906 EC50 = 9910 nM T25608 COJ03Z 86280676 IC50 > 100000 nM T25608 CD80NR 86288852 EC50 = 0.6 nM T25608 C86BUC 86803183 EC50 = 47500 nM T25608 CX8JY7 86803185 EC50 = 1110 nM T25608 CNFI50 86803186 EC50 = 610 nM T25608 C1KD7H 86803188 EC50 = 2120 nM T25608 CVYK05 86803191 EC50 = 1600 nM T25608 CA24JF 86803193 EC50 = 300 nM T25608 CWC61R 86803196 EC50 = 1130 nM T25608 CP7N5Z 86803219 EC50 = 30100 nM T25608 CNQ59Y 86803224 EC50 = 58 nM T25608 C0W2IX 86817649 EC50 = 500 nM T25608 CN9LT5 87054900 EC50 > 9950 nM T25608 C3L9RY 87055315 EC50 > 100000 nM T25608 CP17IF 87262743 EC50 = 170 nM T25608 CJC5L7 87265393 EC50 = 310 nM T25608 CB94OM 89671280 EC50 = 4 nM T25608 CT92HE 90150977 EC50 = 600 nM T25608 CA41EH 90151022 EC50 = 5900 nM T25608 CQN0H4 90151023 EC50 = 280 nM T25608 CRMJ40 90151177 EC50 = 620 nM T25608 C8IMX2 90151202 EC50 = 1930 nM T25608 C6P9ZY 90151205 EC50 = 440 nM T25608 CX3UW9 90151222 EC50 = 360 nM T25608 CR7G4A 90151279 EC50 = 6270 nM T25608 CDML50 90151283 EC50 = 370 nM T25608 CJ18OS 90151297 EC50 = 510 nM T25608 CI5MN6 90151309 EC50 = 3620 nM T25608 CH0SL3 90151370 EC50 = 100 nM T25608 CIFE09 90151400 EC50 = 360 nM T25608 C7OB1H 90151428 EC50 = 500 nM T25608 CV2U3J 90151435 EC50 = 190 nM T25608 C6Q9TN 90151464 EC50 = 3060 nM T25608 CEC97K 90151466 EC50 = 250 nM T25608 C2NC7J 90151501 EC50 = 150 nM T25608 CJZ8W9 90151514 EC50 = 450 nM T25608 C1U4ZE 90151518 EC50 = 1340 nM T25608 C76OPC 90151527 EC50 = 800 nM T25608 CQ76FH 90151529 EC50 = 480 nM T25608 C31BQW 90151537 EC50 = 2550 nM T25608 C5U6ES 90151568 EC50 = 1180 nM T25608 CP1N2O 90151624 EC50 = 2610 nM T25608 C3DMG7 90151625 EC50 = 220 nM T25608 CRL0F1 90151652 EC50 = 450 nM T25608 C60MBW 90151763 EC50 = 7680 nM T25608 C0XV1D 90151764 EC50 = 110 nM T25608 CMI35V 90158812 EC50 = 37 nM T25608 C2BMT5 90161101 EC50 = 320 nM T25608 C0YQ8E 90176463 EC50 = 20 nM T25608 C72JKP 90357232 EC50 = 1.1 nM T25608 C6SG0A 90372365 EC50 = 29 nM T25608 C7M3AG 90372458 EC50 = 816 nM T25608 C4J1UE 90372616 EC50 = 5.2 nM T25608 CDJ1R8 90418278 EC50 > 5000 nM T25608 C32NHB 90644286 EC50 = 3.5 nM T25608 C71KBF 90644287 EC50 = 71 nM T25608 CN17FZ 90644288 EC50 = 32 nM T25608 CZ1OL4 90644289 EC50 = 65 nM T25608 CIP4R2 90644290 EC50 = 3.8 nM T25608 CIA9O6 90644291 EC50 = 420 nM T25608 C6LG5C 90644292 EC50 = 130 nM T25608 CSPJ89 90644293 EC50 = 9.3 nM T25608 C0HG4I 90644294 EC50 = 81 nM T25608 C0WX4B 90644295 EC50 = 2500 nM T25608 CKP0Q6 90644296 EC50 = 8.6 nM T25608 CFK6R0 90644297 EC50 = 65 nM T25608 CQG80O 90644298 EC50 = 120 nM T25608 CP06GD 90644299 EC50 = 18 nM T25608 CMUJ41 90644300 EC50 = 10 nM T25608 C0LBC3 90644301 EC50 = 14 nM T25608 C45GPE 90644302 EC50 = 230 nM T25608 CKI2V9 90644303 EC50 = 35 nM T25608 C0T3VY 90644561 EC50 = 36 nM T25608 C8CF7R 90644562 EC50 = 9 nM T25608 CX70OS 90655858 EC50 = 3700 nM T25608 CX9YU2 90655859 EC50 = 30000 nM T25608 C3A6NL 90655860 EC50 = 1.7 nM T25608 C9RXS2 90655861 EC50 = 6 nM T25608 CL0R8E 90655862 EC50 = 19 nM T25608 CYN4H6 90655863 EC50 = 22 nM T25608 C8IDE7 91801188 EC50 = 3 nM T25608 CUX4B6 91809187 EC50 = 11 nM T25608 C5G3BA 91824140 EC50 = 146 nM T25608 CR7B3W 91827421 EC50 = 0.3 nM T25608 CCE0N5 100502467 IC50 = 10715.19 nM T25608 CYH40T 102338889 EC50 > 100000 nM T25608 CR75CZ 117886639 EC50 > 10000 nM T25608 C3ZH8N 118129974 Ki = 63 nM T25608 C09KBW 118129979 EC50 = 9 nM T25608 CBM67L 118129981 Ki = 37 nM T25608 CZ3KB5 118129998 EC50 = 16 nM T25608 C7NV5G 118129999 EC50 = 2 nM T25608 CR54JA 118144953 EC50 = 151 nM T25608 CI9Z2D 118144973 EC50 = 4.5 nM T25608 CQMU81 118144976 EC50 = 64 nM T25608 CYE4A0 118144982 EC50 = 3.9 nM T25608 C8BJP0 118145019 EC50 = 2156 nM T25608 C7DWG9 118145020 EC50 = 90 nM T25608 CM5S0K 118145140 EC50 = 15 nM T25608 CCVR32 118151370 EC50 = 1 nM T25608 CV90BK 118623088 EC50 = 7 nM T25608 C7TG3X 118637972 EC50 = 23 nM T25608 C31JBK 118637973 EC50 = 165 nM T25608 C9SFI2 118637974 EC50 = 133 nM T25608 COM74C 118637996 EC50 = 1.7 nM T25608 CZDG27 118638001 EC50 = 30 nM T25608 CEOL73 118642344 EC50 = 2.6 nM T25608 CTGF27 118642372 EC50 = 19 nM T25608 CV13EP 118642379 EC50 = 56 nM T25608 C5ZQ3O 118642384 EC50 = 16 nM T25608 CJ85CQ 118642390 EC50 = 11 nM T25608 CK83MT 118642391 EC50 = 304 nM T25608 C1X5KI 118719473 EC50 = 121.1 nM T25608 CI0DV6 118719474 EC50 = 389.3 nM T25608 C7IG1W 118719717 EC50 = 153.3 nM T25608 CKJZ70 118719720 EC50 = 92.6 nM T25608 CQWP70 118719721 EC50 = 62.3 nM T25608 CH8TE4 118737971 EC50 = 69 nM T25608 CVB7Z5 118737972 EC50 = 63 nM T25608 C9AJC3 118737973 EC50 = 330 nM T25608 CH9FW6 118737974 EC50 = 2600 nM T25608 CX8ZY4 122184685 EC50 = 160 nM T25608 CXKQ09 122184686 EC50 = 540 nM T25608 CGA1I0 122185431 EC50 = 1700 nM T25608 CVZI02 122185432 EC50 = 3800 nM T25608 CZ01FD 122185433 EC50 = 580 nM T25608 CFC26W 122185434 EC50 = 1600 nM T25608 CTYZ26 122185435 EC50 = 30 nM T25608 CP3Q5Y 122185436 EC50 = 19 nM T25608 C36OFW 122185437 EC50 = 100 nM T25608 C2B7NQ 122185438 EC50 = 53 nM T25608 C1Q4MD 122185439 EC50 = 12 nM T25608 CL96RS 122185440 EC50 = 35 nM T25608 CS14ME 122185441 EC50 = 2100 nM T25608 C7VXS9 122185442 EC50 = 3200 nM T25608 CO6QC0 122185443 EC50 = 65 nM T25608 CBSQ43 122185444 EC50 = 49 nM T25608 CLEG07 122185445 EC50 = 560 nM T25608 C1JIA0 122185446 EC50 = 147 nM T25608 C52AYK 122185447 EC50 = 13 nM T25608 C0O6XU 122185448 EC50 = 7.5 nM T25608 CYP30W 122185449 EC50 = 5600 nM T25608 C7N8QL 122185450 EC50 = 120 nM T25608 C9VCR7 122185451 EC50 = 12 nM T25608 CKDT83 122185452 EC50 = 20 nM T25608 C91JIK 122185453 EC50 = 36 nM T25608 C5JQP9 122189672 EC50 = 135.3 nM T25608 C0ZWI4 122189676 EC50 = 135.9 nM T25608 C4FPH2 122189677 EC50 = 108.2 nM T25608 CXWG24 122189678 EC50 = 148.2 nM T25608 CE5FW3 122189680 EC50 = 115.6 nM T25608 CCI6Q8 122189682 EC50 = 121.7 nM T25608 CE0DI6 122189683 EC50 = 140.3 nM T25608 CQK8F3 122189685 EC50 = 147.6 nM T25608 CHOE31 122189737 EC50 = 132.9 nM T25608 C1WUV9 122193735 EC50 = 49.7 nM T25608 C1ND8B 122193736 EC50 = 65.9 nM T25608 C4IEU5 122193737 EC50 = 105.8 nM T25608 C27TUN 122193742 EC50 = 110.3 nM T25608 CUE3S5 122193743 EC50 = 103.6 nM T25608 CC5P0F 122193972 EC50 = 109.5 nM T25608 C0R5CD 122193975 EC50 = 43.6 nM T25608 C7V5SG 124011385 EC50 = 1100 nM T25608 CT3R2Q 126961699 IC50 = 158.49 nM T25608 C9U2VX 127025284 EC50 = 1150 nM T25608 CNK89Y 127025285 EC50 = 6110 nM T25608 CA5G1S 127025488 EC50 = 7730 nM T25608 C29TMV 127025858 EC50 = 23120 nM T25608 CB1UT6 127025866 EC50 = 21010 nM T25608 CQZB72 127025867 EC50 = 16600 nM T25608 C4-AUG-07 127027011 EC50 = 1890 nM T25608 C1I7VD 127027659 EC50 = 3570 nM T25608 C1EN3G 127027726 EC50 = 19580 nM T25608 C4U3QH 127027727 EC50 = 7420 nM T25608 C7ZM2B 127027728 EC50 = 8510 nM T25608 CYE4J9 127027729 EC50 = 1660 nM T25608 C90UDI 127027730 EC50 = 4110 nM T25608 C9C0LW 127029850 EC50 = 96.7 nM T25608 C06KLU 127029851 EC50 = 123.4 nM T25608 CWDA29 127030344 EC50 = 489.78 nM T25608 CZ6M9F 127030713 EC50 < 100000 nM T25608 CP60IR 127030714 EC50 = 199.53 nM T25608 CQPG95 127030715 EC50 = 416.87 nM T25608 CJLP42 127030730 EC50 = 118.5 nM T25608 C1P2AW 127031001 EC50 = 83.18 nM T25608 CL24TF 127031002 EC50 = 208.93 nM T25608 CMC5G3 127031003 EC50 = 47.86 nM T25608 CN38XB 127031412 EC50 = 34.7 nM T25608 CDC7F8 127031413 EC50 = 61.2 nM T25608 C32GDE 127031569 EC50 = 389.05 nM T25608 C80XOP 127032539 EC50 = 46.9 nM T25608 CS9N8K 127033020 EC50 = 512.86 nM T25608 CM9P3T 127033239 EC50 = 68.5 nM T25608 CFZ6D3 127033352 EC50 = 1445.44 nM T25608 CG8LY9 127033353 EC50 = 1819.7 nM T25608 C2OM9J 127033354 EC50 = 5011.87 nM T25608 C0P8LB 127033514 EC50 = 102 nM T25608 CCI7M6 127033818 EC50 = 73.5 nM T25608 CAEB91 127033820 EC50 = 137.5 nM T25608 CM64PE 127033821 EC50 = 85.6 nM T25608 C45XEQ 127034369 EC50 = 64.8 nM T25608 C0MH3C 127034370 EC50 = 48.7 nM T25608 CIQ4F8 127035471 EC50 = 330 nM T25608 CLF1N9 127035472 EC50 = 190 nM T25608 C8K4EU 127035636 EC50 = 23000 nM T25608 C29TRI 127035637 EC50 = 690 nM T25608 C2IAM9 127035638 EC50 = 410 nM T25608 C8EC9W 127035639 EC50 = 750 nM T25608 C5LUP7 127035667 EC50 = 43 nM T25608 C9RSG1 127035668 EC50 = 48 nM T25608 CE42KC 127035669 EC50 = 58 nM T25608 CQ0PC1 127036747 EC50 = 440 nM T25608 CWX6R0 127036748 EC50 = 112 nM T25608 CX6I0B 127036828 EC50 = 36 nM T25608 CVO35L 127036829 EC50 = 69 nM T25608 CE9U3A 127036959 EC50 = 240 nM T25608 CIA6T8 127036960 EC50 = 97 nM T25608 C3C5IY 127037608 EC50 = 43 nM T25608 CL5D9C 127037633 EC50 = 59 nM T25608 CD51PV 127037664 IC50 > 39810.72 nM T25608 C8WAB2 127038348 IC50 > 39810.72 nM T25608 C8JH5V 127038399 IC50 = 100 nM T25608 C9OGB2 127038400 IC50 = 25.12 nM T25608 C76FOP 127038401 IC50 = 501.19 nM T25608 C9D5FS 127038402 IC50 = 6309.57 nM T25608 CRU1T3 127038403 IC50 = 7.943 nM T25608 C0TQN1 127038708 IC50 = 398.11 nM T25608 CJ1S9P 127039385 IC50 = 501.19 nM T25608 CW5RV4 127039708 IC50 = 398.11 nM T25608 C36LBX 127039747 IC50 > 39810.72 nM T25608 CA7P9J 127039748 IC50 = 794.33 nM T25608 C6U4ZF 127040059 IC50 = 398.11 nM T25608 C9YW8X 127040093 IC50 = 630.96 nM T25608 C84IXF 127040094 IC50 = 398.11 nM T25608 CAC71N 127040095 IC50 = 501.19 nM T25608 CLH0B9 127040096 IC50 = 251.19 nM T25608 C69UFE 127040097 IC50 = 501.19 nM T25608 CM15FR 127040115 IC50 = 12.59 nM T25608 C1XBW9 127040116 IC50 = 316.23 nM T25608 C5PJ0H 127040117 IC50 = 79.43 nM T25608 CVL12W 127040118 IC50 = 398.11 nM T25608 CF17PH 127040388 IC50 = 316.23 nM T25608 C04LHZ 127040432 IC50 = 794.33 nM T25608 C2JGV6 127040433 IC50 = 251.19 nM T25608 CZTY30 127040434 IC50 = 1995.26 nM T25608 C17TPU 127040723 IC50 = 3162.28 nM T25608 C8S1MJ 127040748 IC50 = 1995.26 nM T25608 C17ZDX 127040749 IC50 = 7943.28 nM T25608 CG19JK 127041066 IC50 = 1584.89 nM T25608 C8H1RB 127041988 IC50 = 63.1 nM T25608 CPF9A0 127042378 IC50 = 1584.89 nM T25608 CP46OL 127042379 IC50 = 398.11 nM T25608 CI24WP 127042380 IC50 = 1258.93 nM T25608 CM63NP 127042381 IC50 = 398.11 nM T25608 C8FV9D 127042382 IC50 = 1258.93 nM T25608 C9BI7U 127042383 IC50 = 251.19 nM T25608 CDUJ24 127042700 IC50 = 10000 nM T25608 C4O1HN 127042701 IC50 = 2511.89 nM T25608 CPYF81 127042702 IC50 = 31622.78 nM T25608 C0ZGS6 127042703 IC50 > 39810.72 nM T25608 C9MFE4 127042704 IC50 > 39810.72 nM T25608 C8LYI3 127042705 IC50 > 39810.72 nM T25608 C3PIA4 127042713 IC50 = 630.96 nM T25608 C5O8PQ 127045657 EC50 = 38.9 nM T25608 C7R1DO 127045658 EC50 = 114 nM T25608 CXFL01 127045659 EC50 = 11.1 nM T25608 CU87JB 127045863 EC50 = 9.3 nM T25608 CZ32DO 127045864 EC50 = 24.3 nM T25608 CEF75Q 127045865 EC50 = 25.9 nM T25608 C5LF9Z 127045866 EC50 = 25.2 nM T25608 C0IPA3 127045888 EC50 = 214 nM T25608 CN5A8X 127046662 EC50 = 143 nM T25608 CRD1A3 127046663 EC50 = 90.9 nM T25608 CYQ21F 127046664 EC50 = 102 nM T25608 C4F5VZ 127046665 EC50 = 506 nM T25608 CG62RV 127046666 EC50 = 4980 nM T25608 C9GNL4 127046667 EC50 = 862 nM T25608 CI3YB2 127046834 EC50 = 1930 nM T25608 CH83VC 127046960 EC50 = 24.8 nM T25608 CPH9G8 127046961 EC50 = 12 nM T25608 C6OBJ0 127046962 EC50 = 33.2 nM T25608 CH9GZ7 127047527 EC50 = 15.9 nM T25608 CUL5X1 127047528 EC50 = 22.9 nM T25608 CY0E9S 127047529 EC50 = 53.1 nM T25608 CK2G8P 127047530 EC50 = 69.1 nM T25608 C64BKX 127047531 EC50 = 96.7 nM T25608 CWR93I 127047532 EC50 = 79.2 nM T25608 CM65EC 127047533 EC50 = 89.3 nM T25608 C6OPM1 127048827 EC50 = 1280 nM T25608 CH9S7P 127048842 EC50 = 760 nM T25608 CN28RD 127048843 EC50 = 1690 nM T25608 CBTU60 127048844 EC50 = 17940 nM T25608 CZ95XB 127049161 EC50 = 1770 nM T25608 C34HEA 127049498 EC50 = 10620 nM T25608 C8B4QX 127050768 EC50 = 1190 nM T25608 CC3GP9 127050769 EC50 = 4680 nM T25608 C6V3FP 127050770 EC50 = 580 nM T25608 CY1MN8 127050771 EC50 = 4300 nM T25608 CDJ7N9 127051302 EC50 = 1060 nM T25608 C7URZ3 127051657 EC50 > 10000 nM T25608 CE94RI 127051658 EC50 = 580 nM T25608 C9VUY6 127051659 EC50 = 6640 nM T25608 CE6J4T 127051660 EC50 = 1520 nM T25608 C5AJR9 127051855 EC50 > 1000 nM T25608 CV6O5J 127051856 EC50 = 187 nM T25608 CX7FO8 127051975 EC50 = 3690 nM T25608 CA0Z5S 127052270 EC50 = 1640 nM T25608 C9TX8Q 130253300 EC50 = 1200 nM T25608 CSI6R9 131842087 EC50 = 28.84 nM T25608 C1N5WO 131986027 EC50 = 13 nM T25608 C5IQ3Z 131986030 EC50 = 8 nM T25608 CB1ZH5 131986035 EC50 = 30 nM T25608 C47GLX 131986050 EC50 = 20 nM T25608 C7UQ4J 131986051 EC50 = 16 nM T25608 C5LZ8H 131986057 EC50 = 23 nM T25608 CYBU25 131986061 EC50 = 13 nM T25608 C8RL3X 131986065 EC50 = 88 nM T25608 CQW41S 131986072 EC50 = 15 nM T25608 C3HF5U 131986075 EC50 = 37 nM T25608 C4FK5N 131986082 EC50 = 67 nM T25608 CA5JX0 131986090 EC50 = 672 nM T25608 C4RI9P 131986112 EC50 = 54 nM T25608 C6WS3P 131986113 EC50 = 28 nM T25608 COCX92 131986115 EC50 = 18 nM T25608 CR13MG 131986116 EC50 = 12 nM T25608 CEZ01T 131986130 EC50 = 39 nM T25608 C6ZI8H 131986132 EC50 = 29 nM T25608 C0T6ZR 131986136 EC50 = 10 nM T25608 C6PY0T 131986140 EC50 = 19 nM T25608 C6FTO2 131986147 EC50 = 107 nM T25608 CQR4K9 131986162 EC50 = 858 nM T25608 C90AOL 131986164 EC50 = 134 nM T25608 CX91BM 131986179 EC50 = 15 nM T25608 CPGU02 131986182 EC50 = 85 nM T25608 C8W7DM 131986250 EC50 = 83 nM T25608 C3I8RE 131986294 EC50 = 9 nM T25608 C2RP7K 131986295 EC50 = 9 nM T25608 C4YV0A 131986297 EC50 = 63 nM T25608 C0L2GI 131986300 EC50 = 25 nM T25608 CF0XJ3 131986378 EC50 = 47 nM T25608 C9DIF2 131986401 EC50 = 20 nM T25608 CBXG19 132606863 EC50 = 110 nM T25608 C9IN6R 132606864 Ki = 45 nM T25608 CJ67MD 134129919 EC50 = 2.1 nM T25608 C53BMN 134129938 EC50 = 4400 nM T25608 CZBD80 134130352 EC50 = 58 nM T25608 CFH18E 134130696 EC50 = 61 nM T25608 CV7S3B 134130787 EC50 = 296 nM T25608 C0DU2R 134130822 EC50 = 1160 nM T25608 CHF3S7 134130859 EC50 = 1252 nM T25608 CSK3E0 134131511 EC50 = 7.3 nM T25608 C17CZB 134131620 EC50 > 10000 nM T25608 CW4S6G 134131874 EC50 > 10000 nM T25608 CO1RW6 134132142 EC50 > 9950 nM T25608 CXE17Y 134132711 IC50 > 100000 nM T25608 C4AB5J 134132951 EC50 > 10000 nM T25608 CB89WY 134133275 EC50 > 9950 nM T25608 C7DE1O 134133297 EC50 = 9260 nM T25608 CKTJ79 134133342 EC50 = 810 nM T25608 CG0L6Q 134133355 EC50 > 10000 nM T25608 CP92NR 134133506 EC50 > 20000 nM T25608 C2W0EY 134133675 EC50 = 3186 nM T25608 C83GOA 134133797 IC50 > 100000 nM T25608 CS3P7G 134133992 EC50 > 10000 nM T25608 CWS2G0 134134149 EC50 = 6799 nM T25608 CUEY64 134134226 EC50 > 20000 nM T25608 CJOQ95 134134229 EC50 = 1829 nM T25608 CQJ8M6 134134433 EC50 = 1.9 nM T25608 CK0NZ3 134134768 EC50 = 140 nM T25608 CNA4L8 134134846 IC50 = 173.78 nM T25608 C21VEN 134135255 EC50 > 20000 nM T25608 C96FRN 134135468 EC50 > 10000 nM T25608 CIFJ93 134135852 EC50 = 42 nM T25608 CUB2S6 134136015 EC50 = 1.4 nM T25608 CCH39I 134136175 EC50 = 6716 nM T25608 C1ECW4 134136203 EC50 = 38 nM T25608 CPBG95 134136959 EC50 = 280 nM T25608 C8LPH3 134137203 EC50 = 10 nM T25608 C2A1ZF 134137248 EC50 = 16.1 nM T25608 C7VOB4 134137619 EC50 > 9950 nM T25608 CR7P0U 134137873 EC50 = 10.5 nM T25608 CIRQ17 134137874 EC50 = 8.6 nM T25608 CXRE49 134138099 IC50 = 2884.03 nM T25608 CD9V6N 134138281 EC50 > 10000 nM T25608 CN9LG1 134138318 EC50 = 6311 nM T25608 CATP91 134138359 EC50 = 118.3 nM T25608 CF2RI3 134138706 EC50 = 16.7 nM T25608 C2J4UK 134138802 EC50 > 10000 nM T25608 C7K6EC 134138870 EC50 = 13 nM T25608 CBCK71 134139119 EC50 = 7 nM T25608 C5JM4L 134139171 EC50 = 2959 nM T25608 CPEK74 134139282 EC50 = 0.8 nM T25608 C1BMG7 134139527 EC50 = 2010 nM T25608 CTL96P 134139990 EC50 = 29.6 nM T25608 CGO7M3 134140070 EC50 > 10000 nM T25608 C5SQU0 134140073 EC50 > 9950 nM T25608 C8DM7J 134140466 EC50 = 2 nM T25608 C17WXH 134140675 EC50 = 4.4 nM T25608 C76URI 134141029 EC50 > 9950 nM T25608 CN9BG4 134141270 EC50 = 1126 nM T25608 CJ30RW 134141489 EC50 = 77 nM T25608 CI75ZW 134141650 IC50 = 3388.44 nM T25608 CO73WM 134141723 EC50 < 300 nM T25608 CNG6U9 134142024 EC50 > 20000 nM T25608 CAR2U0 134142025 EC50 > 20000 nM T25608 C35XWN 134142149 EC50 = 7.9 nM T25608 CZO53G 134142245 EC50 = 7.7 nM T25608 C6ZRV4 134142450 EC50 > 9950 nM T25608 CCDO98 134142866 EC50 = 4218 nM T25608 C4VL9A 134143163 EC50 > 9950 nM T25608 CIN93P 134143370 EC50 > 10000 nM T25608 C9LE7R 134143393 EC50 = 4540 nM T25608 C5HTX1 134143418 EC50 = 8.6 nM T25608 CBLF04 134143899 EC50 = 1391 nM T25608 C9QUR0 134144000 EC50 > 10000 nM T25608 CBW12L 134144214 EC50 = 9463 nM T25608 CL89UD 134144239 EC50 = 10 nM T25608 C0A8TH 134145071 IC50 > 100000 nM T25608 C2GH9K 134145195 EC50 > 9950 nM T25608 CYP7O1 134145412 EC50 > 9950 nM T25608 C8C1DB 134145700 EC50 > 10000 nM T25608 CU36BG 134145750 EC50 > 9950 nM T25608 C8KY5G 134145778 IC50 = 3890.45 nM T25608 C96FUD 134146021 EC50 > 9950 nM T25608 C9N5LO 134146386 EC50 > 10000 nM T25608 CY3ZF0 134146590 EC50 = 410 nM T25608 COYL20 134146720 EC50 > 10000 nM T25608 CC13ZE 134146958 EC50 > 10000 nM T25608 C1OMN0 134147174 EC50 > 9950 nM T25608 CXH3T0 134147328 IC50 = 19952.62 nM T25608 CJXK51 134147518 EC50 = 4.6 nM T25608 CUO72N 134147601 EC50 > 10000 nM T25608 CJ20TQ 134148110 EC50 > 10000 nM T25608 C6ZMV9 134148223 EC50 > 20000 nM T25608 C7XBW3 134148736 EC50 > 9950 nM T25608 CQ5R4P 134149615 EC50 = 1350 nM T25608 CA5B2J 134150245 EC50 = 1042 nM T25608 C9FZ5V 134150458 EC50 > 20000 nM T25608 C6Z7HO 134150797 EC50 = 1.9 nM T25608 C1GDK0 134150871 EC50 > 10000 nM T25608 C87ECV 134150969 EC50 > 1000 nM T25608 CLM9Q7 134151115 EC50 = 2504 nM T25608 CAG0Y1 134151150 EC50 = 55 nM T25608 CYG78X 134151354 EC50 > 20000 nM T25608 C6TP5Q 134151754 EC50 = 1270 nM T25608 CRH0A7 134151903 EC50 > 10000 nM T25608 CAY73T 134152336 EC50 > 10000 nM T25608 CF13KR 134152488 EC50 > 20000 nM T25608 C3SFX4 134152545 IC50 = 616.6 nM T25608 CNK25T 134152845 EC50 > 9950 nM T25608 CRGW59 134153067 IC50 = 44668.36 nM T25608 C82ZGH 134153148 EC50 = 71 nM T25608 CW54AS 134153222 IC50 > 100000 nM T25608 CVOE51 134153298 EC50 > 10000 nM T25608 C7U9SB 134153546 EC50 = 2000 nM T25608 C4H8UV 134153562 EC50 = 5406 nM T25608 C4O0ZM 134153986 EC50 > 10000 nM T25608 C49FKZ 134154330 EC50 > 9950 nM T25608 CV1E3G 134154415 EC50 > 10000 nM T25608 C0GYX7 134154417 EC50 > 9950 nM T25608 CM69QG 134154473 EC50 = 3600 nM T25608 C6SA1G 134154953 IC50 = 25118.86 nM T25608 CK29QG 134155067 EC50 > 10000 nM T25608 C9LNQ5 134155277 EC50 > 9950 nM T25608 CSM4R6 134155480 EC50 = 2100 nM T25608 CK7PY5 134155821 EC50 = 12 nM T25608 CA6RE0 134155847 EC50 = 2200 nM T25608 C7TO6A 134155950 EC50 > 10000 nM T25608 CK9M4A 134156096 EC50 = 3352 nM T25608 CL92ZI 134156455 EC50 > 10000 nM T25608 CA49BH 134156727 EC50 > 10000 nM T25608 CK84XB 134157015 EC50 = 1300 nM T25608 C7GDP1 134157207 EC50 > 9950 nM T25608 CJ6T8B 134157563 EC50 > 9950 nM T25608 C2GKN8 134157586 EC50 = 3586 nM T25608 CD0S5Z 134157824 EC50 > 20000 nM T25608 CUP4M1 134465730 EC50 = 2.2 nM T25608 CB0Q9N 134465732 EC50 = 0.2 nM T25608 C7V1RX 134465785 EC50 = 0.94 nM T25608 CVA5D0 134465794 EC50 = 0.25 nM T25608 CXOJ48 134538585 EC50 = 4 nM T25608 CKEP73 137529972 EC50 = 2 nM T25608 CRI0U6 137529979 EC50 = 148 nM T25608 CR4P2U 137529983 EC50 = 7 nM T25608 C8X1RQ 137631853 EC50 = 490 nM T25608 CYRS03 137632053 EC50 = 580 nM T25608 C7TA3H 137632403 EC50 > 30000 nM T25608 CBRG92 137633101 EC50 = 220 nM T25608 CUK0D4 137633394 EC50 = 150 nM T25608 C7MF0A 137633536 EC50 = 11800 nM T25608 CO0RD7 137633561 EC50 = 14800 nM T25608 C68SZA 137634330 EC50 = 81 nM T25608 CGE59Q 137634844 EC50 > 30000 nM T25608 CNUX64 137634863 EC50 > 33000 nM T25608 CL90AO 137634888 EC50 = 1260 nM T25608 C4JME8 137635143 EC50 = 2710 nM T25608 CCJ4W0 137635388 EC50 = 6400 nM T25608 C3IH5R 137635513 EC50 = 2320 nM T25608 CG8B5Y 137635715 EC50 = 260 nM T25608 COBJ62 137635907 EC50 = 70 nM T25608 COI40P 137636026 EC50 > 33000 nM T25608 CT0S7L 137636033 EC50 = 40100 nM T25608 CZ1OD2 137636167 EC50 = 1544 nM T25608 C6D7ZM 137636358 Ki = 49 nM T25608 C9GD8B 137636501 EC50 = 33500 nM T25608 CMO1E3 137636733 EC50 > 30000 nM T25608 C5QN8L 137637488 EC50 = 2100 nM T25608 CR53AY 137637576 EC50 = 3782 nM T25608 CL2DA0 137637602 EC50 = 1480 nM T25608 CWN80V 137638184 EC50 = 260 nM T25608 C3PO6D 137638269 EC50 = 220 nM T25608 CF35JS 137638341 EC50 = 180 nM T25608 CMPD78 137638355 EC50 = 18051 nM T25608 CE87QJ 137638413 EC50 = 1110 nM T25608 CT93OE 137638911 EC50 = 19952.62 nM T25608 CGD21L 137638995 EC50 = 7943.28 nM T25608 CR0IS1 137639817 EC50 = 450 nM T25608 CDMR25 137640032 EC50 = 6200 nM T25608 C0M8SI 137640301 EC50 = 1270 nM T25608 C4JOD5 137640323 EC50 > 30000 nM T25608 CI3R1P 137640417 EC50 = 32200 nM T25608 CUER14 137640728 EC50 = 3920 nM T25608 CP5U2V 137640781 EC50 = 900 nM T25608 CXL21U 137640919 EC50 = 680 nM T25608 CE9Z4L 137641343 EC50 = 19588 nM T25608 C4GVT6 137641734 EC50 = 13000 nM T25608 C0XLQ9 137642173 EC50 = 1210 nM T25608 CTW8I6 137642184 EC50 > 30000 nM T25608 CZ4KW8 137642604 EC50 = 7943.28 nM T25608 CNKP70 137642920 EC50 > 10000 nM T25608 C4QBG8 137642988 EC50 > 17000 nM T25608 CS59FT 137643339 EC50 = 10000 nM T25608 CJR49O 137643956 EC50 = 410 nM T25608 C1K4CL 137644843 EC50 = 82 nM T25608 CNK59T 137644989 EC50 = 110 nM T25608 C1XG9C 137645352 EC50 = 2560 nM T25608 CEYI29 137646043 EC50 = 11000 nM T25608 CM2C7J 137646188 EC50 > 30000 nM T25608 CU8OD6 137646308 EC50 = 640 nM T25608 CLTA84 137646337 EC50 = 6500 nM T25608 C19RYO 137646482 EC50 = 150 nM T25608 C7Y9PC 137646553 EC50 > 30000 nM T25608 C7SG5X 137646830 EC50 = 290 nM T25608 C4J7DH 137646898 EC50 > 33000 nM T25608 CIE72D 137647107 EC50 = 880 nM T25608 CQC17M 137647721 EC50 = 12589.25 nM T25608 C0OHT8 137648439 EC50 = 210 nM T25608 C3X4NA 137648780 EC50 = 240 nM T25608 C2DQ4O 137649008 Ki = 23000 nM T25608 CL1HE5 137649416 EC50 > 30000 nM T25608 CYX37M 137650524 EC50 = 2060 nM T25608 CCBI43 137652992 EC50 = 2420 nM T25608 CHD0E8 137653172 EC50 = 390 nM T25608 C9KHS5 137653756 EC50 = 3870 nM T25608 CBX4Z3 137653896 EC50 = 450 nM T25608 CFI68P 137653903 EC50 = 50 nM T25608 CP30FQ 137654021 EC50 = 210 nM T25608 CO2L0W 137654721 EC50 > 30000 nM T25608 C3Y9TQ 137655097 EC50 > 17000 nM T25608 C0XBY5 137655393 EC50 = 14700 nM T25608 CA3W9B 137655559 EC50 = 1140 nM T25608 CZLU59 137655619 EC50 = 1300 nM T25608 CT6S0B 137655758 EC50 > 33000 nM T25608 COB6K3 137656526 EC50 = 1423 nM T25608 C4E1YT 137657002 EC50 = 4600 nM T25608 CK5BX8 137657027 EC50 = 2010 nM T25608 CK9R6S 137657972 EC50 = 1584.89 nM T25608 CCW3P1 137658243 EC50 = 520 nM T25608 CCKT75 137658391 EC50 = 8900 nM T25608 CSR4W2 137658634 EC50 > 30000 nM T25608 C5YO8K 137658671 EC50 = 6490 nM T25608 CBG58K 137659266 EC50 = 260 nM T25608 CP96HY 137659517 EC50 = 680 nM T25608 CL70UQ 137659867 EC50 = 6100 nM T25608 CI21BK 137661056 EC50 = 2360 nM T25608 CT91BF 137661294 EC50 = 8 nM T25608 CZR62H 137661388 EC50 > 30000 nM T25608 CET37O 137661475 EC50 = 1700 nM T25608 CQ0GL8 137661929 EC50 = 57 nM T25608 C41OTE 141747238 EC50 = 4020 nM T25608 CDA4Z5 141747241 EC50 > 10000 nM T25608 C6K9ZT 142738539 EC50 = 9.4 nM T25608 CQ4TD1 142738540 EC50 > 25 nM T25608 CI71RX 142738543 EC50 = 1016 nM T25608 C02XYW 142738544 EC50 > 25 nM T25608 C08YVD 142738545 EC50 = 447 nM T25608 C60TYD 142738546 EC50 > 25 nM T25608 CO5ZN2 142738551 EC50 = 54.6 nM T25608 CAP4E3 142738553 EC50 = 778 nM T25608 CB7C3P 142738556 EC50 = 1308 nM T25608 CY6R9F 142738561 EC50 > 25 nM T25608 CI0E6S 142738567 EC50 = 37.8 nM T25608 C6I2JS 142738569 EC50 = 1800 nM T25608 C3R8IS 142738570 EC50 > 25 nM T25608 CCD2K8 142738574 EC50 > 25 nM T25608 CJ9B1F 142738575 EC50 = 1207 nM T25608 CBY8D4 142738578 EC50 > 25 nM T25608 C4LZ6A 142738583 EC50 = 1800 nM T25608 CQG5V4 145754982 EC50 = 41.69 nM T25608 CY0M8X 145949924 EC50 = 203 nM T25608 C74XZG 145949955 EC50 = 138 nM T25608 CN9KI4 145950126 EC50 = 172 nM T25608 C2L4ZC 145950191 EC50 = 531 nM T25608 CB7S9A 145950347 EC50 = 47 nM T25608 CYTD84 145950402 EC50 = 42 nM T25608 C8CZA1 145950447 EC50 = 54 nM T25608 CZQ1W4 145950728 EC50 = 113 nM T25608 C3UVA7 145951164 EC50 = 109 nM T25608 C0NML8 145951402 EC50 = 820 nM T25608 C09BIY 145952214 EC50 = 13 nM T25608 C6DOX5 145952673 EC50 = 50 nM T25608 CDLS51 145952700 EC50 = 1.6 nM T25608 CJ92XZ 145952952 EC50 = 20 nM T25608 CF1A8U 145953265 EC50 = 1136 nM T25608 CFP4H6 145953365 EC50 = 39 nM T25608 C7RGX9 145954367 EC50 = 94 nM T25608 C1S3NZ 145954394 EC50 > 10000 nM T25608 C6UT2R 145954794 EC50 = 155 nM T25608 CT2D7E 145954950 EC50 = 11330 nM T25608 CM3Y8D 145955179 EC50 = 308 nM T25608 CCP23Q 145955263 EC50 = 391 nM T25608 C4NM7D 145955723 EC50 = 231 nM T25608 C2O3LF 145955958 EC50 < 0.2 nM T25608 C9AJM4 145956000 EC50 > 1667 nM T25608 CLG81H 145956069 EC50 = 211 nM T25608 C2Q6IM 145956160 EC50 = 133 nM T25608 C1M5RN 145956406 EC50 < 0.2 nM T25608 C1GMP5 145956671 EC50 = 187 nM T25608 C0SLG1 145956739 EC50 = 610 nM T25608 CD6Y3Z 145956795 EC50 < 0.2 nM T25608 CLO4A7 145957072 EC50 = 97 nM T25608 CT7HW4 145957539 EC50 = 934 nM T25608 CR9J8V 145957609 EC50 = 1.1 nM T25608 CFD2Y6 145958651 EC50 > 10000 nM T25608 C36WRG 145958799 EC50 > 10000 nM T25608 C1IW4J 145958971 EC50 = 114 nM T25608 C1UB5H 145959273 EC50 = 8.2 nM T25608 CH6ZM0 145959598 EC50 = 57 nM T25608 CUG35K 145959722 EC50 = 417 nM T25608 CH8VA1 145959829 EC50 > 5000 nM T25608 CZ8E7J 145959985 EC50 = 1.7 nM T25608 CFGL96 145960084 EC50 = 1.6 nM T25608 C3A5XR 145960204 EC50 > 5000 nM T25608 CYHL49 145960453 EC50 = 21340 nM T25608 CV81UA 145960571 EC50 = 1.9 nM T25608 CMJ50D 145961418 EC50 = 0.8 nM T25608 CU14RO 145961656 EC50 = 5060 nM T25608 C9H0QO 145962064 EC50 = 144 nM T25608 CS8LJ9 145962072 EC50 = 179 nM T25608 CFUV91 145962164 EC50 = 4310 nM T25608 CD0W3C 145963128 EC50 > 25 nM T25608 C63OLJ 145963137 EC50 > 1667 nM T25608 CZ01IO 145963330 EC50 = 72 nM T25608 C9LH0Y 145963593 EC50 = 17750 nM T25608 CASW30 145963855 EC50 = 450 nM T25608 C9AQ6D 145964042 EC50 = 36.31 nM T25608 CS85LT 145964249 EC50 > 1000 nM T25608 CE09SL 145964735 EC50 > 10000 nM T25608 C6SHF7 145964802 EC50 = 426.58 nM T25608 CED62A 145964820 EC50 = 57.54 nM T25608 CH5MB9 145964866 EC50 > 1000 nM T25608 C1JR8C 145965138 EC50 = 257.04 nM T25608 C9SK7T 145965307 EC50 > 10000 nM T25608 CYT0J8 145965455 EC50 = 169.82 nM T25608 CPG7N1 145965467 EC50 = 331.13 nM T25608 CHZY25 145965661 EC50 = 52.48 nM T25608 CFX4L5 145965707 EC50 = 190.55 nM T25608 CJ1FL8 145965797 EC50 = 4120 nM T25608 CS9OA7 145965948 EC50 = 10500 nM T25608 C8RVW9 145965968 EC50 = 1411 nM T25608 CJK8U5 145965982 EC50 > 10000 nM T25608 CAL68F 145966017 EC50 = 1130 nM T25608 CE3BG0 145966029 EC50 > 10000 nM T25608 C74UGD 145966102 EC50 > 10000 nM T25608 C0L4YQ 145966167 EC50 = 457.09 nM T25608 C8R9YD 145966219 EC50 = 3260 nM T25608 C9D2XW 145966459 EC50 > 10000 nM T25608 C09WOF 145966485 EC50 = 1170 nM T25608 CG5QD9 145966540 EC50 > 1000 nM T25608 CU4GW5 145966632 EC50 = 251.19 nM T25608 C3IA4S 145966647 EC50 = 69.18 nM T25608 C2QT5B 145966699 EC50 = 213.8 nM T25608 C87MEW 145967080 EC50 > 10000 nM T25608 CNE6D4 145967091 EC50 = 66.07 nM T25608 CYC39X 145967263 EC50 = 177.83 nM T25608 CB57ZL 145967268 EC50 = 18600 nM T25608 CW6VO9 145967558 EC50 = 97.72 nM T25608 CU70AC 145967748 EC50 = 15.49 nM T25608 CX4BD7 145967778 EC50 = 75900 nM T25608 CCTO59 145967994 EC50 = 128.82 nM T25608 CIA03M 145968204 EC50 = 27.5 nM T25608 C7BTS4 145968322 EC50 = 157.1 nM T25608 C7FNC4 145969097 EC50 = 37.4 nM T25608 CR4BV2 145969373 EC50 > 10000 nM T25608 CKAL34 145969681 EC50 = 103.7 nM T25608 CMUN49 145970056 EC50 = 1020 nM T25608 CKRC96 145970067 EC50 > 1000 nM T25608 C0CVS9 145970371 EC50 = 53.7 nM T25608 CB6YO0 145970463 EC50 = 18.6 nM T25608 C7FY0C 145970728 EC50 = 28.9 nM T25608 CN4F0P 145971234 EC50 = 106 nM T25608 C1I9GA 145971547 EC50 > 10000 nM T25608 C7PCQ8 145971688 EC50 = 80 nM T25608 CIG73O 145971779 EC50 = 194.98 nM T25608 C9BZ7K 145971800 EC50 = 74.13 nM T25608 CW89VJ 145972020 EC50 = 133 nM T25608 CP0G4C 145972079 EC50 = 213.8 nM T25608 C3ZV6Y 145972304 EC50 = 1380 nM T25608 CWL07B 145973087 EC50 = 5020 nM T25608 C5ZTX4 145973102 EC50 > 10000 nM T25608 C12IJB 145973299 EC50 > 10000 nM T25608 C8X5FW 145973329 EC50 = 210 nM T25608 C2FN3Q 145973478 EC50 = 63.1 nM T25608 C96YWE 145973686 EC50 > 1000 nM T25608 C0CEN6 145973781 EC50 = 2540 nM T25608 CG28IX 145973933 EC50 > 10000 nM T25608 CAX4B9 145973937 EC50 = 1350 nM T25608 C13UBN 145973986 EC50 > 10000 nM T25608 C10LCU 145974034 EC50 > 1000 nM T25608 CQ8Z0G 145974173 EC50 = 170 nM T25608 C2NY0F 145974295 EC50 = 289 nM T25608 CI32AO 145974382 EC50 = 3670 nM T25608 CJUN-39 145974478 EC50 = 3090 nM T25608 CI50OB 145974495 EC50 = 46.77 nM T25608 CZV45O 145974509 EC50 = 2390 nM T25608 CQ9I5U 145974719 EC50 = 95.5 nM T25608 CL5TQ8 145975293 EC50 = 1520 nM T25608 C0B3CR 145975484 EC50 = 79.43 nM T25608 C0N4BC 145975522 EC50 = 5390 nM T25608 C2RPC5 145975621 EC50 = 2390 nM T25608 C4HRA6 145975628 EC50 = 288.4 nM T25608 CA21IS 145976136 EC50 = 275.42 nM T25608 CC52RT 145976145 EC50 = 194.98 nM T25608 CNL46D 145976172 EC50 = 234.42 nM T25608 C37RUC 145976267 EC50 = 1570 nM T25608 CGN2Y8 145976608 EC50 = 549.54 nM T25608 C07KYE 145976639 EC50 = 4 nM T25608 CD3R8O 145976702 EC50 = 2170 nM T25608 C2Z8KJ 145976748 EC50 = 234.42 nM T25608 CEP0I9 145976845 EC50 = 125.89 nM T25608 C59FXK 145976935 EC50 = 123.03 nM T25608 CHNC94 145976979 EC50 = 2430 nM T25608 CYI5W2 145977043 EC50 = 2710 nM T25608 C7TD1V 145977220 EC50 > 10000 nM T25608 CETA73 145977329 EC50 > 10000 nM T25608 CDTI80 145977404 EC50 = 269.15 nM T25608 C74JLM 145977668 EC50 = 363.08 nM T25608 CWA95F 145977707 EC50 = 1530 nM T25608 CS08HW 145977721 EC50 > 5000 nM T25608 CTM7A1 145977853 EC50 > 10000 nM T25608 C8MT3A 145978233 EC50 = 549.54 nM T25608 C6IU2A 145978511 EC50 = 51.29 nM T25608 C26HLU 145978559 EC50 > 1000 nM T25608 CXA80W 145978608 EC50 > 10000 nM T25608 CD67EV 145978633 EC50 = 7900 nM T25608 C0M4DC 145978849 EC50 > 1000 nM T25608 C9KC3V 145978975 EC50 = 3400 nM T25608 CLT09H 145979123 EC50 = 3980 nM T25608 C62KTQ 145979171 EC50 = 120 nM T25608 C5GLC7 145979252 EC50 = 4310 nM T25608 CC8E1Z 145979329 EC50 = 27200 nM T25608 C43IVG 145979602 EC50 = 36270 nM T25608 CXZ91W 145980154 EC50 = 10 nM T25608 CZ54IN 145980380 EC50 > 10000 nM T25608 CMUP96 145980455 EC50 = 13570 nM T25608 CN61AL 145980470 EC50 = 150 nM T25608 C0KP3F 145980573 EC50 = 3020 nM T25608 C1Q6PV 145980608 EC50 = 4260 nM T25608 CKR43C 145981599 EC50 = 3850 nM T25608 CPT0D9 145981771 EC50 = 830 nM T25608 C2SHF4 145981901 EC50 > 30000 nM T25608 CW9D3X 145981983 EC50 = 260 nM T25608 CUA9E3 145982071 EC50 = 980 nM T25608 CSW42Z 145982132 EC50 = 210 nM T25608 C87UAM 145982210 EC50 > 10000 nM T25608 CC2L9V 145982417 EC50 > 10000 nM T25608 CFY8U2 145982433 EC50 = 7620 nM T25608 C0JR7M 145982556 EC50 = 3000 nM T25608 CF34ZO 145982616 EC50 = 3500 nM T25608 CXY27B 145983006 EC50 = 61.5 nM T25608 CSW94B 145983457 EC50 = 5400 nM T25608 CO8K0Z 145983493 EC50 = 68780 nM T25608 C1CB9N 145983698 EC50 = 130 nM T25608 CAEZ16 145983824 EC50 = 3480 nM T25608 CS2A3B 145983825 EC50 = 76.4 nM T25608 CK9B5S 145984009 EC50 > 100000 nM T25608 C2IF8C 145984092 EC50 = 1200 nM T25608 C59PQC 145984275 EC50 = 800 nM T25608 C0OJ2P 145984445 EC50 > 100000 nM T25608 CT9V1W 145984594 EC50 > 100000 nM T25608 CKEB40 145984796 EC50 > 100000 nM T25608 C2V6CW 145984886 EC50 = 1030 nM T25608 CQ1TB7 145984906 EC50 = 3070 nM T25608 C67RHD 145984999 EC50 = 800 nM T25608 CK1IO9 145985116 EC50 = 2200 nM T25608 C0F2AH 145985122 EC50 = 11010 nM T25608 C9LV7A 145985123 EC50 = 93.7 nM T25608 C5C4YM 145985219 EC50 > 100000 nM T25608 CX4GB0 145985574 EC50 = 4000 nM T25608 C1HK7R 145985632 EC50 > 10000 nM T25608 CIGK40 145985686 EC50 = 24430 nM T25608 C5J4SE 145985748 EC50 > 100000 nM T25608 CX9U0T 145986046 EC50 = 29350 nM T25608 CPFW32 145986077 EC50 = 610 nM T25608 C28DAN 145986262 EC50 > 100000 nM T25608 CAE95K 145986458 EC50 > 10000 nM T25608 C0XPC2 145986478 EC50 > 50000 nM T25608 CDZG12 145986662 EC50 = 3060 nM T25608 CHL62X 145986689 EC50 = 8080 nM T25608 CW7Y4G 145986696 EC50 = 2380 nM T25608 CBOR53 145986704 EC50 > 10000 nM T25608 CT3W4M 145987015 EC50 = 100 nM T25608 C6DL2O 145987167 EC50 = 2870 nM T25608 C40HLG 145987309 EC50 = 5040 nM T25608 CB6QN4 145987484 EC50 = 7.9 nM T25608 C72DAS 145987796 EC50 = 200 nM T25608 C6MC4L 145987969 EC50 = 1800 nM T25608 CMN5R7 145987974 EC50 = 1470 nM T25608 CWZ5L7 145988414 EC50 = 39.7 nM T25608 C0G2WE 145988431 EC50 > 10000 nM T25608 CMBR98 145988551 EC50 > 10000 nM T25608 CTKM20 145988554 EC50 = 2850 nM T25608 C2ZBK5 145988796 EC50 = 210 nM T25608 CY2IL3 145989151 EC50 = 170 nM T25608 C75DSN 145989198 EC50 = 3590 nM T25608 CI94EP 145989566 EC50 = 2100 nM T25608 CHF9J1 145989900 EC50 = 2110 nM T25608 CI39OJ 145989913 EC50 > 10000 nM T25608 CQOK62 145990228 EC50 = 700 nM T25608 CJ76KD 145990303 EC50 = 2760 nM T25608 CT9WV6 145990337 EC50 = 8060 nM T25608 C7GK3H 145990715 EC50 = 46 nM T25608 C4BLV7 145990729 EC50 > 10000 nM T25608 C6OM1C 145990731 EC50 = 3770 nM T25608 CC28QH 145990980 EC50 = 110 nM T25608 C8CP3I 145991235 EC50 > 30000 nM T25608 CZQH15 145991380 EC50 = 5880 nM T25608 CVBP54 145991722 EC50 > 10000 nM T25608 CQ82EM 145991968 EC50 = 2370 nM T25608 CV2FB6 145992078 EC50 = 3450 nM T25608 C6F0LJ 145992170 EC50 = 3280 nM T25608 CP79UQ 145992176 EC50 > 10000 nM T25608 CEC30M 145992604 EC50 = 690 nM T25608 C0E2WQ 145992623 EC50 = 90 nM T25608 C87MWN 145992631 EC50 = 640 nM T25608 CDO7U1 145992642 EC50 = 2240 nM T25608 CCY19L 145992868 EC50 > 10000 nM T25608 CU3EG4 145993152 EC50 > 30000 nM T25608 CROV68 145993162 EC50 = 210 nM T25608 CX5FZ7 145993490 EC50 = 3870 nM T25608 C0T1BY 145993621 EC50 = 520 nM T25608 CFJQ16 145993644 EC50 = 280 nM T25608 C7DFI1 145994052 EC50 = 1170 nM T25608 CCV39B 145994196 EC50 = 8450 nM T25608 CC3SP5 146316684 EC50 = 6.1 nM T25608 C5BLX3 146695343 EC50 = 41.3 nM T25608 CG6T4L 146763588 EC50 = 59.8 nM T25608 CZGT59 146840871 EC50 = 40 nM T25608 C24OEI 147146439 EC50 = 4.8 nM T25608 CH2NL0 147329931 EC50 = 11.6 nM T25608 C0BDA4 147747458 EC50 = 38.7 nM T25608 C4G7NA 148173135 EC50 = 86.2 nM T25608 CIQ3X2 148485044 EC50 = 51.6 nM T25608 CP7I6Z 149144496 EC50 = 24.2 nM T25608 CDM45B 149231065 EC50 = 240 nM T25608 C1OK9A 149378333 EC50 = 225.3 nM T25608 CNWP21 149454889 EC50 = 19.3 nM T25608 CKH93B 153211729 EC50 = 196.7 nM T25608 CV53OY 153213696 EC50 = 58.5 nM T25608 C8LF3A 153272850 EC50 = 728.6 nM T25608 CM3H9E 155511380 EC50 = 220 nM T25608 C8Y9ST 155512244 EC50 = 374 nM T25608 C1N0VI 155512776 EC50 = 80 nM T25608 CYE8H1 155513821 EC50 = 59 nM T25608 C0VTM9 155515698 EC50 > 1000 nM T25608 C8RZH5 155515835 EC50 = 41.9 nM T25608 CM4TB2 155516498 EC50 = 54 nM T25608 CV53HO 155516879 EC50 = 120 nM T25608 CEZ0F1 155517179 EC50 = 1780 nM T25608 C08DTF 155517891 EC50 = 325 nM T25608 C93BFL 155519364 EC50 = 200 nM T25608 CU0L7Y 155522406 EC50 = 120 nM T25608 CT2H7E 155522452 EC50 = 460 nM T25608 C17OFD 155523655 EC50 = 1350 nM T25608 CPT9J8 155525700 EC50 = 185 nM T25608 C3P2ZK 155526024 EC50 > 10000 nM T25608 CAK2H8 155526126 EC50 = 220 nM T25608 C6RU2E 155526793 EC50 = 16 nM T25608 CWE06G 155527415 EC50 = 150 nM T25608 C26DHQ 155527487 EC50 = 60 nM T25608 CJP7Z9 155527626 EC50 = 326 nM T25608 CJI0N8 155527805 EC50 = 70 nM T25608 CR91BJ 155528372 EC50 = 2 nM T25608 C4SGK6 155528599 EC50 = 51.7 nM T25608 C34YXP 155529382 EC50 > 10000 nM T25608 CLV9W1 155529599 EC50 = 6500 nM T25608 C7NDX5 155529750 EC50 > 10000 nM T25608 C6N9YP 155530111 EC50 = 112 nM T25608 C69KEW 155530636 EC50 = 397.5 nM T25608 CT5D9K 155530726 EC50 > 10000 nM T25608 C41VZM 155533810 EC50 = 160 nM T25608 CBW2Z8 155535186 EC50 = 36.5 nM T25608 CVG6P0 155535946 EC50 > 10000 nM T25608 CXA3M2 155541840 EC50 = 536.2 nM T25608 CB14CD 155542122 EC50 = 80 nM T25608 C5W8SV 155543683 EC50 > 10000 nM T25608 CPU3Q0 155544661 EC50 = 11 nM T25608 C6PD1A 155545127 EC50 = 590 nM T25608 CX3KF2 155545207 EC50 > 10000 nM T25608 C1PO2Q 155546331 EC50 > 10000 nM T25608 CC63ZG 155547595 EC50 = 156 nM T25608 CR48CL 155547604 EC50 = 251 nM T25608 CEG6H0 155548030 EC50 = 400 nM T25608 CG3H7C 155548258 EC50 = 22.5 nM T25608 CZY63J 155549083 EC50 = 1.1 nM T25608 C9FV2A 155549085 EC50 = 36.1 nM T25608 CLI81V 155549391 EC50 = 1020 nM T25608 CAK8E6 155550483 EC50 = 45.6 nM T25608 C84OTS 155551422 EC50 = 0.11 nM T25608 CWHL51 155551584 EC50 = 16 nM T25608 CIK42F 155552554 EC50 = 290 nM T25608 CUAP95 155555299 EC50 > 10000 nM T25608 C4BSK6 155557354 EC50 > 10000 nM T25608 CY5RG0 155558174 EC50 = 69.6 nM T25608 CVH06N 155560437 EC50 > 10000 nM T25608 C7H1SI 155561223 EC50 = 155 nM T25608 CQ6VH4 155561358 EC50 = 247 nM T25608 C2NPT3 155561834 EC50 > 10000 nM T25608 C37ZFX 155563228 EC50 = 149 nM T25608 CQ7DF1 155565379 EC50 = 3 nM T25608 CG02XL 155565451 EC50 = 68 nM T25608 CS4UV7 155569570 EC50 = 300 nM T25608 C8H3WI 155569585 EC50 = 15.7 nM T25608 D01CCG 25150014 EC50 = 32 nM T25608 D01VIX 73777063 EC50 > 10000 nM T25608 D03JPL 79034 EC50 > 100000 nM T25608 D03LOG 5280450 EC50 = 540 nM T25608 D08MLH 46941175 Ki = 5.888 nM T25608 D08ZYC 11595431 EC50 = 13 nM T25608 D0C5SV 5280934 EC50 = 2884.03 nM T25608 D0J2EE 9957245 EC50 = 70 nM T25608 D0K6EG 57522038 EC50 = 5011.87 nM T25608 D0N0UC 3893 EC50 = 758.58 nM T25608 D0N9SV 25098573 EC50 = 9772.37 nM T25608 D0Q7BG 46854655 EC50 = 2.2 nM T25608 D0S0QY 66553168 EC50 = 5.888 nM T25608 D0T2CG 94216 EC50 > 100000 nM T25608 D0T4BP 97783 EC50 = 6760.83 nM T58741 D08HQK 5411 IC50 = 520 nM T58741 D0C7ET 11174599 IC50 = 2.3 nM T58741 D00BUR 216327 IC50 > 1000 nM T58741 D04PER 49836093 IC50 = 170 nM T58741 D0K9IF 71666749 IC50 > 30000 nM T58741 D0O7QA 46840946 IC50 = 160 nM T58741 D0OX9F 16046068 IC50 = 15000 nM T58741 CPN25U 998021 IC50 = 10300 nM T58741 CZK6M0 22239024 IC50 = 660 nM T58741 C3LK1F 42637004 IC50 = 1030 nM T58741 C40BIM 45139151 IC50 = 1050 nM T58741 CS5EJ1 46841648 IC50 = 1636 nM T58741 CRE97F 46841787 IC50 = 1109 nM T58741 C06OXV 52920492 IC50 = 24000 nM T58741 CMS2F7 53239561 IC50 = 3320 nM T58741 CC82DM 65459349 IC50 = 4200 nM T58741 C2MC6B 71522734 IC50 = 0.8 nM T58741 CM1B0W 71523649 IC50 = 46000 nM T58741 CJXK67 71559365 IC50 = 11 nM T58741 C9MUK3 71716856 IC50 = 510 nM T58741 CUG2V3 71716866 IC50 = 199 nM T58741 C15BSO 86270136 IC50 = 190 nM T58741 CTG76E 86687532 IC50 = 3700 nM T58741 C1BIF8 90026208 IC50 = 38 nM T58741 C26BZK 91666633 IC50 = 92 nM T58741 C7NLE8 91809347 IC50 = 480 nM T58741 CC5N9I 117737142 IC50 = 1300 nM T58741 C10BKY 117749324 IC50 = 650 nM T58741 C9KV7L 117993993 IC50 = 9400 nM T58741 C7AYV5 118540795 IC50 = 5.461 nM T58741 CR8TX9 118708662 IC50 = 26 nM T58741 C9JL4Y 118937760 IC50 = 8600 nM T58741 C9Q2ND 121333973 IC50 = 16000 nM T58741 C9K5RV 122513516 IC50 > 20000 nM T58741 C09QIY 127047645 IC50 = 5000 nM T58741 CF6L8Q 145955101 IC50 = 66 nM T58741 CCTB54 145958837 IC50 = 104 nM T58741 C38DYW 145959291 IC50 = 183 nM T58741 CK7PN3 145969142 IC50 = 1600 nM T58741 C8Q2EG 145988110 IC50 = 2100 nM T58741 COZ54G 155523716 IC50 = 1000 nM T58741 C5F9BQ 155526497 IC50 = 29000 nM T58741 CE3H4Z 155567528 IC50 = 130 nM T58741 D0P8TL 56947150 IC50 = 1.1 nM T04696 D0W0VD 3885 IC50 = 970 nM T04696 CW68ZS 61672 IC50 = 40000000 nM T04696 CH67EZ 91286 IC50 = 4100 nM T04696 CZTD26 220436 IC50 = 9000 nM T04696 CVGN02 267570 IC50 > 30000 nM T04696 CE7M6K 269624 IC50 = 40 nM T04696 CRSF26 304992 IC50 > 111000 nM T04696 CSO78Y 322478 EC50 = 870 nM T04696 CZ34CV 349435 IC50 = 25000 nM T04696 CS2B8E 397888 IC50 = 1000 nM T04696 C9WI3X 460748 EC50 = 780 nM T04696 CWYT28 460749 EC50 = 430 nM T04696 CIJ28W 555805 IC50 > 111000 nM T04696 C4BRI2 707946 IC50 > 100000 nM T04696 C6WZ2C 866938 EC50 > 30000 nM T04696 C7WC0L 930115 EC50 > 30000 nM T04696 CJ0V3O 931081 EC50 > 30000 nM T04696 CK1TD5 941846 EC50 > 30000 nM T04696 C0ME8D 951230 EC50 = 7360 nM T04696 CB0X4T 951368 EC50 > 30000 nM T04696 CBN32K 1293987 IC50 > 100000 nM T04696 C6LPN3 1313201 IC50 > 100000 nM T04696 CRL05A 1771058 IC50 = 32000 nM T04696 C35DCU 3164059 EC50 = 510 nM T04696 CNTJ89 3164066 EC50 = 1070 nM T04696 CSXC46 3164070 EC50 = 330 nM T04696 C2C9RE 4989139 EC50 = 300 nM T04696 CO01XP 5478021 IC50 = 3500 nM T04696 CO8M4Q 6411132 EC50 > 20000 nM T04696 C2BY6K 6458554 EC50 = 960 nM T04696 CVC31J 6459022 EC50 = 290 nM T04696 CC6U7A 6493950 EC50 = 280 nM T04696 C5FY6T 11266171 IC50 = 7600 nM T04696 C65MLO 11840607 IC50 = 23600 nM T04696 CHDB52 12023317 IC50 = 11000 nM T04696 C1JX2C 12023323 IC50 = 3500 nM T04696 C4RGJ6 14895314 IC50 > 111000 nM T04696 C54WZY 14895315 IC50 = 43000 nM T04696 C8Z9XB 16481078 EC50 = 200 nM T04696 CK7J6D 17756791 EC50 = 3500 nM T04696 CFBT48 46833159 EC50 = 680 nM T04696 COS86H 46834048 EC50 = 750 nM T04696 CV60DR 46834317 EC50 = 370 nM T04696 CCM26J 56837840 IC50 > 111000 nM T04696 C0DMZ7 57400600 IC50 > 111000 nM T04696 CS0Q9C 59299967 IC50 = 19000 nM T04696 CZ3Y7S 60103948 IC50 > 111000 nM T04696 CWJ46V 60104019 IC50 > 111000 nM T04696 C5BJM9 68699178 IC50 > 111000 nM T04696 CU8ZA0 71817697 EC50 = 260 nM T04696 CLD4B7 71817698 EC50 = 400 nM T04696 CZE8Q2 71817849 EC50 = 4630 nM T04696 CG2A6C 71817850 EC50 = 280 nM T04696 C2ZYW4 71817852 EC50 > 10000 nM T04696 C35QBR 71817853 EC50 = 7420 nM T04696 C8A0CS 71818002 EC50 = 670 nM T04696 CHKS75 71818003 EC50 = 1020 nM T04696 CJ3YG9 71818004 EC50 = 700 nM T04696 C8WN0H 71818005 EC50 = 640 nM T04696 C4HGP6 71818006 EC50 = 430 nM T04696 CEX8A6 71818007 EC50 = 150 nM T04696 CPB21Q 71818143 EC50 = 770 nM T04696 CTD4U6 71818144 EC50 = 250 nM T04696 C7UB6O 71818145 EC50 = 120 nM T04696 CHF45Y 71818146 EC50 = 50 nM T04696 C96AYZ 71818147 EC50 > 20000 nM T04696 CJ2OV6 71818149 EC50 > 20000 nM T04696 CLAF94 71818291 EC50 = 2100 nM T04696 CWHG19 71818293 EC50 > 150000 nM T04696 CH6BV1 71818296 EC50 > 150000 nM T04696 CHN47D 71818443 EC50 > 150000 nM T04696 CZXW74 71818444 EC50 > 150000 nM T04696 CTSD96 71818445 EC50 > 30000 nM T04696 C2WO0L 71818446 EC50 > 30000 nM T04696 C1Z9HD 71818447 EC50 > 30000 nM T04696 CG7Q6D 71818587 EC50 > 30000 nM T04696 CW8N0J 71818588 EC50 > 30000 nM T04696 C3M4FP 71818589 EC50 > 30000 nM T04696 C69KUV 71818590 EC50 > 30000 nM T04696 CT30QA 71818591 EC50 > 30000 nM T04696 C3WJ6B 71818592 EC50 > 30000 nM T04696 C7TIJ1 71818716 EC50 > 30000 nM T04696 CLU15O 71818717 EC50 > 30000 nM T04696 CF9I3P 71818718 EC50 > 30000 nM T04696 C3DTB4 71818719 EC50 > 30000 nM T04696 CI80ND 71818720 EC50 > 30000 nM T04696 COU9C7 71818721 EC50 > 30000 nM T04696 C8AR0I 71818722 EC50 = 1660 nM T04696 CB23IX 71818723 EC50 > 30000 nM T04696 CQV2B5 71818864 EC50 = 480 nM T04696 C8L1XF 71818865 IC50 = 27480 nM T04696 C5CXH0 71818866 EC50 = 2870 nM T04696 C7P2XN 71818867 EC50 = 500 nM T04696 CPK26T 71818868 IC50 = 42 nM T04696 C85OTM 71818869 EC50 = 90 nM T04696 CK6W2Z 71818870 EC50 = 250 nM T04696 C9MKT5 71819004 EC50 = 470 nM T04696 CMI5O8 71819005 EC50 = 1040 nM T04696 CG7ZN2 71819006 EC50 = 320 nM T04696 CWSE58 71819007 EC50 = 3390 nM T04696 CXG20Y 71819008 EC50 = 2740 nM T04696 CMT0Y2 71819009 EC50 = 90 nM T04696 C48DOI 71819143 EC50 = 30 nM T04696 CJC48A 71819144 EC50 = 4660 nM T04696 C7GXZ3 71819145 EC50 = 1370 nM T04696 C7Q0NF 71819146 EC50 = 290 nM T04696 C5ET9H 71819147 EC50 = 640 nM T04696 CRZ8G6 71819148 EC50 = 370 nM T04696 C19SNE 71819283 IC50 = 41 nM T04696 CB4NR9 72211790 IC50 = 9800 nM T04696 C6NQP9 73346151 EC50 = 720 nM T04696 C9CI3X 73350770 EC50 = 360 nM T04696 CRZ62F 73355036 EC50 = 24000 nM T04696 CSP7U6 118641028 IC50 > 111000 nM T04696 COJ93Q 121472570 IC50 = 11000 nM T04696 CE8KX5 121472571 IC50 = 35000 nM T04696 CU2O3F 121478289 IC50 = 11000 nM T04696 CJ1E0R 121478290 IC50 = 12000 nM T04696 C2UMF7 121478292 IC50 > 111000 nM T04696 C0SM2F 121478293 IC50 = 51000 nM T04696 C41BGD 121478294 IC50 = 15000 nM T04696 C3V9CO 121478295 IC50 = 16000 nM T04696 C7R5DK 121478296 IC50 = 66000 nM T04696 C7FYP6 121478298 IC50 > 111000 nM T04696 CIRH72 121478299 IC50 > 111000 nM T04696 CG9MA0 121478300 IC50 = 7700 nM T04696 C2NCD1 121478303 IC50 = 13000 nM T04696 CQ71GI 121478304 IC50 > 111000 nM T04696 C2JEM3 121478305 IC50 = 3300 nM T04696 CV37KR 121478306 IC50 > 111000 nM T04696 CHZ3G9 121478307 IC50 = 11000 nM T04696 C6LQR0 121478308 IC50 = 12000 nM T04696 CY52IG 121478317 IC50 = 50000 nM T04696 CD7O9U 121478318 IC50 = 24000 nM T04696 CB46CR 121478319 IC50 = 13000 nM T04696 CWN68V 121478326 IC50 = 13000 nM T04696 C5QRF9 121478327 IC50 = 14000 nM T04696 C2LGQ0 121478328 IC50 = 17000 nM T04696 COSM56 121478329 IC50 = 13000 nM T04696 CAI2T3 121478330 IC50 = 10000 nM T04696 C2UHT5 121478331 IC50 = 10000 nM T04696 C3QXM6 121478332 IC50 > 111000 nM T04696 C4GFH8 121478333 IC50 = 12000 nM T04696 CG48YT 121478334 IC50 = 8100 nM T04696 C3YM8C 121478345 IC50 = 19000 nM T04696 CUH40X 121478347 IC50 = 17000 nM T04696 CDY7B5 121478349 IC50 > 111000 nM T04696 C0P8VG 121478351 IC50 = 1900 nM T04696 CKC14X 121478358 IC50 = 37000 nM T04696 C0G9RA 121478361 IC50 = 14000 nM T04696 C27CJU 121478363 IC50 = 71000 nM T04696 CH30JX 121478365 IC50 = 22000 nM T04696 CQ3CR2 121478367 IC50 = 19000 nM T04696 CW12NY 121478368 IC50 = 68000 nM T04696 CN9UE4 121478394 IC50 = 9800 nM T04696 CCW7Y0 121478397 IC50 = 13000 nM T04696 C9B2OZ 121478399 IC50 = 11000 nM T04696 C5CN6W 121478400 IC50 = 8800 nM T04696 C1WC5X 121478401 IC50 = 18000 nM T04696 C9M1LP 121478402 IC50 = 6600 nM T04696 CN5QF3 121478403 IC50 > 111000 nM T04696 CI53LJ 121478405 IC50 = 24000 nM T04696 C12FTJ 121478406 IC50 > 111000 nM T04696 CJLG39 121478407 IC50 = 12000 nM T04696 C60YRK 121478438 IC50 > 111000 nM T04696 CT1RL3 122179149 IC50 > 111000 nM T04696 CM9AU7 122179162 IC50 > 111000 nM T04696 C98KOJ 122179163 IC50 = 37000 nM T04696 C7Q9FC 122179164 IC50 > 111000 nM T04696 CTFO36 122483585 IC50 = 5500 nM T04696 C2Q1HV 122483587 IC50 = 6500 nM T04696 CVE37N 122483588 IC50 = 13000 nM T04696 CSCZ94 122483589 IC50 = 18000 nM T04696 CU8C3T 122483590 IC50 = 7100 nM T04696 C9X8QL 122483591 IC50 = 30000 nM T04696 CM20BN 122483592 IC50 = 2600 nM T04696 COC53H 122483593 IC50 = 3200 nM T04696 CE89RT 122483594 IC50 > 37000 nM T04696 C15GNW 122483596 IC50 > 37000 nM T04696 CUGI76 122483597 IC50 = 10000 nM T04696 CCLF45 122483598 IC50 = 4500 nM T04696 CH9OJ3 122483599 IC50 > 111000 nM T04696 CIPC52 122483600 IC50 = 26000 nM T04696 C04XUJ 122483601 IC50 = 14000 nM T04696 CG3O5N 122483604 IC50 = 25000 nM T04696 C6W8SH 122483605 IC50 > 37000 nM T04696 CSOF59 122483606 IC50 = 16000 nM T04696 C4QH5Y 122483608 IC50 = 9300 nM T04696 C6FZQ4 122483609 IC50 = 16000 nM T04696 C7Q3LI 122483610 IC50 = 5200 nM T04696 C1WCV3 122483611 IC50 > 111000 nM T04696 C5UVQ3 122483612 IC50 = 3300 nM T04696 CN1W3U 122483613 IC50 > 111000 nM T04696 C2EX1V 122483614 IC50 = 4100 nM T04696 C4PG1R 122483615 IC50 = 4500 nM T04696 C52AQF 122483618 IC50 > 111000 nM T04696 CNO57Z 122483619 IC50 = 16000 nM T04696 CH95QN 122483620 IC50 = 36000 nM T04696 C9B0TV 122483622 IC50 = 42000 nM T04696 CV7H2F 122483623 IC50 > 111000 nM T04696 C5X8OF 122483624 IC50 = 3000 nM T04696 C8Q6ZY 122483625 IC50 = 4500 nM T04696 CSKF94 122483626 IC50 = 1900 nM T04696 CG6U2L 122483627 IC50 = 20000 nM T04696 CGB0R9 122483628 IC50 = 19000 nM T04696 C41LDF 122483629 IC50 = 21000 nM T04696 C8MC5T 122483630 IC50 = 25000 nM T04696 C8C9SW 122483631 IC50 = 5400 nM T04696 CW0KF2 122483633 IC50 = 14000 nM T04696 CAST90 122483634 IC50 = 23000 nM T04696 C0DBQ9 122483635 IC50 = 2700 nM T04696 CRDV43 122483636 IC50 = 50000 nM T04696 C2DEL7 122483637 IC50 = 11000 nM T04696 C3KDP2 122483638 IC50 = 11000 nM T04696 CGZ75H 122483639 IC50 = 11000 nM T04696 CP87QX 122483641 IC50 = 15000 nM T04696 C7BL9T 122484905 IC50 = 6300 nM T04696 C3FS6Y 122484906 IC50 = 8900 nM T04696 CT5OG6 127028881 IC50 = 5100 nM T04696 CPY24W 127029757 IC50 > 111000 nM T04696 C7YX4G 127030613 IC50 > 111000 nM T04696 CLT35C 127043728 IC50 > 111000 nM T04696 CJA2I1 127044083 IC50 = 37000 nM T04696 CBFS34 127044239 IC50 > 111000 nM T04696 CE15TB 127044402 IC50 > 111000 nM T04696 CF64IU 127044403 IC50 > 111000 nM T04696 C12IUQ 127044404 IC50 > 111000 nM T04696 CBE49O 127044405 IC50 > 111000 nM T04696 CM19WU 127044406 IC50 = 111000 nM T04696 CU15SD 127044408 IC50 = 111000 nM T04696 C0X5YU 127044409 IC50 = 111000 nM T04696 C3XO0J 127044411 IC50 > 111000 nM T04696 COX07F 127044412 IC50 > 111000 nM T04696 C5OQ3T 127044413 IC50 > 111000 nM T04696 C38YZG 127044414 IC50 > 111000 nM T04696 C0SP4E 127044557 IC50 > 111000 nM T04696 CPEU65 127044559 IC50 > 111000 nM T04696 C1W8YR 127044560 IC50 > 111000 nM T04696 CPWI81 127051466 IC50 = 12000 nM T04696 C9L1GO 129896914 IC50 = 12000 nM T04696 C5DA0Z 135163962 IC50 = 37000 nM T04696 C3OGL8 135438987 IC50 = 17700 nM T04696 C5K9YU 136236292 IC50 = 17000 nM T04696 CQZ79S 137633472 IC50 > 111000 nM T04696 CEMW84 137634763 IC50 = 1000 nM T04696 CY83RB 137635101 IC50 = 61600 nM T04696 CY4BH7 137635982 IC50 = 12000 nM T04696 CP8I0N 137635992 IC50 = 107000 nM T04696 CC1X7N 137637372 IC50 > 111000 nM T04696 CSKE17 137638583 IC50 > 111000 nM T04696 C7K5XB 137638718 IC50 > 111000 nM T04696 CY0G2M 137639745 IC50 = 32900 nM T04696 CE93VQ 137639878 IC50 = 108000 nM T04696 C7KVT8 137640123 IC50 = 37000 nM T04696 C7EHL1 137643195 IC50 > 111000 nM T04696 CQ89WF 137644721 IC50 > 111000 nM T04696 C7LY3U 137645346 IC50 > 111000 nM T04696 CT8A6V 137645479 IC50 = 37000 nM T04696 CTD0Q1 137645708 IC50 = 37000 nM T04696 C83FEH 137646143 IC50 > 111000 nM T04696 CR72BP 137646560 IC50 = 37000 nM T04696 CW24CA 137650951 IC50 > 111000 nM T04696 C2RVW9 137651075 IC50 > 111000 nM T04696 C7SUD6 137652086 IC50 = 104000 nM T04696 C9X2IG 137652438 IC50 > 111000 nM T04696 CY25WR 137653301 IC50 > 111000 nM T04696 CDQ41E 137656446 IC50 > 111000 nM T04696 CZ01OK 137658578 IC50 = 37000 nM T04696 CHXA46 137659333 IC50 = 37000 nM T04696 CB9GY3 137660083 IC50 > 111000 nM T04696 C09XQR 137661166 IC50 > 111000 nM T04696 CSB6M0 139368816 IC50 = 130 nM T04696 C84UBZ 139368818 IC50 = 65 nM T04696 CQ4G6B 139368820 IC50 = 70 nM T04696 C3F9GV 139368834 IC50 = 6.5 nM T04696 CWL01S 139368851 IC50 = 3800 nM T04696 CQ0F4V 139368854 IC50 = 320 nM T04696 CBM15W 139368874 IC50 = 20 nM T04696 CNI9A6 139368879 IC50 = 14 nM T04696 C5M1BA 139368887 IC50 = 880 nM T04696 CEH93B 139368894 IC50 = 33 nM T04696 CBM19D 139368902 IC50 = 7.3 nM T04696 CE9AK7 139368907 IC50 = 930 nM T04696 CQD73C 139368913 IC50 = 38 nM T04696 CS9UM7 139368918 IC50 = 200 nM T04696 CD9HM5 139368920 IC50 = 35 nM T04696 C2PUL4 139368923 IC50 = 300 nM T04696 CPDJ72 139368930 IC50 = 1100 nM T04696 C5G7JZ 139368935 IC50 = 6.1 nM T04696 C0AM4H 139368936 IC50 = 270 nM T04696 CVF8C5 139368940 IC50 > 10000 nM T04696 C8VH9F 139368954 IC50 = 190 nM T04696 CBI70J 139368955 IC50 = 150 nM T04696 CDW39J 139368964 IC50 = 33 nM T04696 C30ENM 139368966 IC50 = 960 nM T04696 CMP03R 139368970 IC50 = 1600 nM T04696 CT95OC 139368975 IC50 = 1500 nM T04696 C7EH0V 139368985 IC50 = 1000 nM T04696 C1LBE4 139368987 IC50 = 380 nM T04696 CC3QT9 139379823 IC50 = 990 nM T04696 C5Y2ZA 145949905 IC50 > 111000 nM T04696 CUL1I3 145950046 IC50 = 99000 nM T04696 CF6Y7J 145950454 IC50 > 111000 nM T04696 CDM0W7 145951675 IC50 = 28000 nM T04696 CEO83W 145952632 IC50 = 36000 nM T04696 C47WUP 145952847 IC50 > 111000 nM T04696 C74VYG 145953711 IC50 = 51000 nM T04696 CV35UN 145954864 IC50 = 24000 nM T04696 C0WC6Q 145955087 IC50 > 111000 nM T04696 CZ54YB 145955773 IC50 = 88000 nM T04696 C9IPA5 145956858 IC50 = 31000 nM T04696 C4UTW8 145957109 IC50 > 111000 nM T04696 CRA1K8 145957662 IC50 = 12000 nM T04696 C5X9ZY 145957721 IC50 = 38000 nM T04696 C1QE7V 145958498 IC50 = 29000 nM T04696 C3CHN5 145958644 IC50 = 28000 nM T04696 CUYA76 145959663 IC50 > 111000 nM T04696 C4NU9M 145960096 IC50 > 111000 nM T04696 C2X5SP 145972895 IC50 > 111000 nM T04696 C3DCY1 145973141 IC50 = 31000 nM T04696 C93HRO 148522856 IC50 = 1300 nM T04696 CUFI09 155511226 IC50 = 22000 nM T04696 C1OUY2 155511648 IC50 = 77300 nM T04696 CXY2T9 155513626 IC50 > 100000 nM T04696 CR06GW 155516031 IC50 > 100000 nM T04696 C82ZWB 155517851 IC50 = 80900 nM T04696 CSQ6J0 155520530 IC50 > 100000 nM T04696 C1UFN8 155520960 IC50 > 100000 nM T04696 C1F8SC 155521790 IC50 > 100000 nM T04696 CRQ5V4 155522028 IC50 > 100000 nM T04696 C2TAG8 155522368 IC50 > 100000 nM T04696 CYT67S 155522639 IC50 > 100000 nM T04696 CJ2YD3 155523314 IC50 = 80800 nM T04696 CKI09P 155527507 IC50 > 100000 nM T04696 C7GYW1 155527618 IC50 > 100000 nM T04696 CE1KY2 155527688 IC50 > 100000 nM T04696 CB4WA6 155527846 IC50 > 100000 nM T04696 CN4XT5 155528962 IC50 > 100000 nM T04696 CMS31Q 155529562 IC50 > 100000 nM T04696 C5CK8O 155530724 IC50 > 100000 nM T04696 CE6SN1 155532734 IC50 > 100000 nM T04696 C3FKI7 155533180 IC50 > 100000 nM T04696 C1BYP0 155534526 IC50 > 100000 nM T04696 CT81JB 155536721 IC50 > 100000 nM T04696 CTD2N5 155537102 IC50 = 43800 nM T04696 C9PV4T 155537144 IC50 = 85200 nM T04696 CU13XE 155539442 IC50 > 100000 nM T04696 C6V8HO 155541099 IC50 = 21000 nM T04696 CV1YX3 155546559 IC50 > 100000 nM T04696 C9J0VW 155547447 IC50 > 100000 nM T04696 C5BL8C 155547740 IC50 > 100000 nM T04696 C8OH9M 155548958 IC50 > 100000 nM T04696 C3DO8S 155550002 IC50 > 100000 nM T04696 CVM59F 155550044 IC50 > 100000 nM T04696 C01UYS 155553494 IC50 > 100000 nM T04696 C5ZR0U 155553817 IC50 > 100000 nM T04696 C4MT7Q 155561437 IC50 > 100000 nM T04696 C3A2VZ 155563144 IC50 = 94500 nM T04696 CI36HO 155563834 IC50 = 59000 nM T04696 CR0IP2 155564579 IC50 > 100000 nM T04696 CZ6R9X 155565688 IC50 > 100000 nM T04696 CXEY68 155566971 IC50 > 100000 nM T04696 C5EG2O 155567730 IC50 = 16600 nM T04696 CYHT71 155568211 IC50 > 100000 nM T04696 C0ST7X 155568568 IC50 > 100000 nM T04696 D0J1KH 262093 IC50 = 71000 nM T04696 D0P0CM 460747 EC50 = 1160 nM T16633 D0TV0C 9941444 Ki = 6.31 nM T16633 D06JFI 11251755 IC50 = 27 nM T16633 D0J8PI 158782 IC50 > 10000 nM T16633 D0L9QM 59568713 IC50 = 2630 nM T16633 D09JXL 5311430 Ki < 1000 nM T16633 C6XYL5 6918011 Ki = 501.19 nM T16633 CHM63P 6918026 Ki = 158.49 nM T16633 CR0U6E 9827283 Ki = 5382 nM T16633 CA8UQ7 9848232 Ki = 4264 nM T16633 CTRI07 9852911 Ki = 4000 nM T16633 C9BJ3Q 9854636 IC50 > 1000 nM T16633 CDU75Z 9857566 Ki = 5000 nM T16633 CMLP16 9918828 Ki = 630.96 nM T16633 C3Z5YJ 9963342 Ki = 3.981 nM T16633 CIT57N 9985523 Ki = 4100 nM T16633 C64LIB 10009650 Ki = 300 nM T16633 CL6G0Z 10094509 Ki = 2310 nM T16633 C9C7RK 10096510 Ki = 9700 nM T16633 CFZN71 10166743 Ki = 1730 nM T16633 CI21CK 10179247 Ki > 10000 nM T16633 C6DRE9 10210016 Ki = 1550 nM T16633 C4M9GN 10248767 Ki = 3400 nM T16633 C78LUH 10296743 Ki = 1400 nM T16633 CSY5K2 10325243 Ki = 2400 nM T16633 CL87OB 10411795 Ki = 2600 nM T16633 CS96ON 10534086 IC50 = 1000 nM T16633 CHZ9I8 10554930 Ki = 6800 nM T16633 CY3ZE9 10577746 IC50 = 501 nM T16633 C9C0HF 10580397 Ki = 2100 nM T16633 CU3DQ6 10630127 Ki = 1000 nM T16633 C45JIZ 10699714 Ki = 4400 nM T16633 CG2UX4 10701257 IC50 = 1000 nM T16633 CP0F7C 10724811 IC50 = 1000 nM T16633 C3TMY5 10724880 IC50 = 1580 nM T16633 CJM47E 10748701 IC50 = 2163 nM T16633 CWF2N5 10748831 IC50 = 1000 nM T16633 CLW4V6 10770814 Ki = 4000 nM T16633 CO56HI 10772403 IC50 = 1000 nM T16633 CGN0Z5 10772578 IC50 = 535 nM T16633 C3L4DH 10796238 IC50 = 4843 nM T16633 C15QGO 10819673 IC50 = 1000 nM T16633 CFL71O 10843862 IC50 = 1000 nM T16633 C2PJ1O 10876898 Ki = 10 nM T16633 C6TVQ8 10964197 Ki = 6.31 nM T16633 CXDG12 10996788 Ki = 1.585 nM T16633 C6AW0M 11112736 Ki > 10000 nM T16633 CK1RX4 11136828 Ki = 63.1 nM T16633 CR1JP9 11147505 Ki = 3.981 nM T16633 C1I9EX 11159133 IC50 = 757 nM T16633 C7REL4 11170698 IC50 = 117 nM T16633 CIEM12 11170867 IC50 > 10000 nM T16633 CW2JA8 11182381 IC50 = 410 nM T16633 CE3GC2 11205475 IC50 = 5.3 nM T16633 CXI32T 11205496 IC50 = 450 nM T16633 C2RNJ5 11205515 IC50 = 327 nM T16633 CUT8Z0 11240205 IC50 = 21 nM T16633 CK78SD 11240206 IC50 = 27 nM T16633 C67WXD 11274767 IC50 = 10.3 nM T16633 COK06N 11320738 IC50 > 1000 nM T16633 C5D6AM 11332138 IC50 > 1000 nM T16633 C5PAN4 11343811 IC50 > 1000 nM T16633 CLQ53A 11355270 IC50 = 410 nM T16633 CQ0UC7 11378229 IC50 = 607 nM T16633 CC09ZU 11378299 IC50 > 1000 nM T16633 CG7PT9 11389178 IC50 = 650 nM T16633 CFJD72 11423410 IC50 = 330 nM T16633 C4S2HG 11434734 IC50 = 49 nM T16633 C6XHC3 11457491 IC50 = 213 nM T16633 CJ5A9B 11457521 IC50 = 840 nM T16633 CMA8C7 11468709 IC50 > 10000 nM T16633 CG8A0J 11468887 IC50 = 6.5 nM T16633 CZ3N5J 11468916 IC50 = 55 nM T16633 CORY59 11480246 IC50 = 545 nM T16633 C63QMX 11535351 IC50 > 1000 nM T16633 CF6K7M 11563877 IC50 = 5100 nM T16633 CS68YA 11642413 IC50 = 9590 nM T16633 CZHN61 11678313 IC50 > 10000 nM T16633 CW65KY 11705763 Ki = 530 nM T16633 CN63YV 11787877 IC50 > 10000 nM T16633 CR6UF9 11788180 IC50 > 1000 nM T16633 CK4U8N 11804376 IC50 = 1000 nM T16633 C9XH7F 11815114 Ki = 1.585 nM T16633 CRA01O 11845058 IC50 > 1000 nM T16633 C8X3CL 11845059 IC50 > 1000 nM T16633 CO3HT9 11847587 IC50 > 1000 nM T16633 CMR10F 11848679 Ki = 1750 nM T16633 CBV2X0 11963995 Ki = 5100 nM T16633 CW7I8U 13690207 Ki = 224 nM T16633 C8OU7I 15429504 IC50 = 723 nM T16633 CEO3F0 15585102 IC50 > 1000 nM T16633 CC2YJ8 16062553 Ki > 10000 nM T16633 C3H1RT 16062555 Ki > 10000 nM T16633 C1LH5T 16062816 Ki = 4500 nM T16633 C1GKF8 16130982 Ki = 0.32 nM T16633 C2TRA5 16144717 IC50 = 1044 nM T16633 CW20OC 16144977 IC50 = 506 nM T16633 CS6A3Z 16145268 IC50 = 1000 nM T16633 CN3LS1 16145579 IC50 = 1000 nM T16633 C72MUC 16146425 IC50 = 1000 nM T16633 CD91IL 16148220 IC50 = 1000 nM T16633 C59OUC 16148481 Ki = 125.89 nM T16633 CJG1X9 16148596 Ki = 0.631 nM T16633 CNY09C 16148922 Ki = 1000 nM T16633 CP0DC8 16149640 Ki = 0.5012 nM T16633 CDPC19 16149975 Ki = 6.31 nM T16633 C0SE6V 16150676 Ki = 0.2512 nM T16633 CSP6A9 16150915 Ki = 0.1585 nM T16633 C6N7SR 16151159 Ki = 19.95 nM T16633 C2B9IL 16151570 IC50 = 189 nM T16633 CQM8J1 16151781 IC50 = 347 nM T16633 CM8UF7 16151826 IC50 = 3.3 nM T16633 CJ7UT6 16151923 IC50 > 1000 nM T16633 CIM03U 16152257 IC50 = 270 nM T16633 CU7X6V 16153077 IC50 = 88 nM T16633 CK4O1V 16153193 IC50 = 517 nM T16633 C16LMW 16153418 IC50 > 1000 nM T16633 CO0LG7 16154000 IC50 = 99 nM T16633 CX4RM8 16154096 IC50 = 13 nM T16633 COYU86 16156815 Ki = 1000 nM T16633 CI3FW1 16157160 IC50 = 1025 nM T16633 C7GN0S 16157479 Ki = 0.1995 nM T16633 CQL5O0 16181427 IC50 = 31 nM T16633 C2CUY9 16181428 EC50 = 33 nM T16633 CUH8D7 16737812 IC50 > 1000 nM T16633 C8QIT3 16737813 IC50 > 1000 nM T16633 CNP36U 16737814 IC50 = 233 nM T16633 C7Q6JL 16738359 IC50 = 89 nM T16633 C6F1RZ 24777672 IC50 = 961 nM T16633 C5GZO7 24858018 IC50 = 96 nM T16633 CV1U7H 24858920 IC50 = 14 nM T16633 C0UB7K 24859055 IC50 > 1000 nM T16633 CQCW58 24859056 IC50 = 22 nM T16633 CT6J2A 24859195 IC50 = 16 nM T16633 CUDV69 24859196 IC50 > 1000 nM T16633 C45NYA 24859341 IC50 > 1000 nM T16633 C4AB6I 24859342 IC50 = 416 nM T16633 CH50QU 24859494 IC50 = 79 nM T16633 C8L2KJ 24859495 IC50 > 1000 nM T16633 CDS6W5 24859645 IC50 = 358 nM T16633 CHF20D 24859646 IC50 > 1000 nM T16633 CKH2R4 24859787 IC50 = 540 nM T16633 CT1BM6 24859788 IC50 > 1000 nM T16633 C2IKX3 24859919 IC50 > 1000 nM T16633 C5OQ2X 24859920 IC50 > 1000 nM T16633 CSZ73L 24860057 IC50 > 1000 nM T16633 C36ZHQ 24860058 IC50 > 1000 nM T16633 CVL48C 24860201 IC50 = 302 nM T16633 C20ZFS 24860202 IC50 = 218 nM T16633 CHKC79 25187396 IC50 = 253 nM T16633 C4YXJ1 25187398 IC50 = 54 nM T16633 CO9PI7 25187400 IC50 = 27 nM T16633 C8C9PL 25187679 IC50 = 38 nM T16633 C9ECD8 25187681 IC50 > 1000 nM T16633 C43OES 25187683 IC50 = 247 nM T16633 CNTB73 25187685 IC50 = 89 nM T16633 C1IUQ2 25187953 IC50 = 837 nM T16633 CQ3F8L 25187955 IC50 = 379 nM T16633 CS2ZV1 25188218 IC50 = 630 nM T16633 CLI2U1 25188220 IC50 = 183 nM T16633 CNDU95 25188496 IC50 = 962 nM T16633 C7KF8N 25188776 IC50 > 1000 nM T16633 CCHN50 25188780 IC50 = 105 nM T16633 C3T8DA 25189052 IC50 = 76 nM T16633 CI21ED 25189054 IC50 = 372 nM T16633 C97LHK 25189325 IC50 = 75 nM T16633 CEG4J0 25189327 IC50 = 387 nM T16633 CSQH26 42637069 EC50 = 3.9 nM T16633 CJ1S9K 42637136 IC50 = 37 nM T16633 C3NYM8 42637137 IC50 = 97 nM T16633 CJ47CL 42637210 IC50 = 530 nM T16633 CR3A8Q 42637283 IC50 = 189 nM T16633 CENZ47 42637363 IC50 = 108 nM T16633 CX0JC7 42637503 IC50 = 0.19 nM T16633 C90LHS 42637563 IC50 = 4.7 nM T16633 C80WBK 42637632 IC50 = 8.2 nM T16633 CR49YE 42637984 IC50 > 1000 nM T16633 CEFO24 42638065 IC50 = 150 nM T16633 CF5JK4 42638066 IC50 = 14 nM T16633 CHY04A 44290718 IC50 > 1000 nM T16633 C16BKW 44290734 IC50 > 1000 nM T16633 CW76YB 44290735 IC50 > 1000 nM T16633 CA6IS7 44290766 IC50 > 1000 nM T16633 C6BZ1J 44298104 Ki = 348 nM T16633 CCXL10 44298113 Ki > 1000 nM T16633 CYW8O0 44298130 Ki = 1690 nM T16633 CB9JK1 44298131 Ki = 1030 nM T16633 CJ5WL8 44298155 Ki > 1000 nM T16633 CHL57J 44298156 Ki = 1200 nM T16633 CP61LB 44298165 Ki > 1000 nM T16633 CM0B6J 44298166 Ki > 1000 nM T16633 C8XZR7 44298169 Ki = 1060 nM T16633 C0DPX7 44298171 Ki = 413 nM T16633 C62OEU 44298177 Ki = 82 nM T16633 CS9JW8 44298178 Ki > 1000 nM T16633 C20MBI 44298179 Ki = 1950 nM T16633 C3QBP0 44298188 Ki = 525 nM T16633 C1R3QD 44298189 Ki = 575 nM T16633 C5RJ7U 44298195 Ki = 435 nM T16633 C8N3EJ 44298197 Ki = 443 nM T16633 CZU05A 44298214 Ki > 1000 nM T16633 CQUS98 44298218 Ki = 37 nM T16633 COTK07 44298219 Ki = 186 nM T16633 CAJO07 44298231 Ki = 415 nM T16633 C9S4IX 44298232 Ki = 845 nM T16633 CB1A3K 44298235 Ki = 174 nM T16633 C2TQ1V 44298248 Ki = 69 nM T16633 C3WFV5 44298250 Ki = 374 nM T16633 CVW19Y 44298328 Ki = 34 nM T16633 CT94HY 44298329 Ki = 568 nM T16633 CL4F1V 44298378 Ki = 238 nM T16633 CMO1Q9 44298441 Ki = 1400 nM T16633 C8Y9ZP 44298443 Ki > 1000 nM T16633 CUSR45 44298468 Ki > 1000 nM T16633 C8EN2H 44298469 Ki = 60 nM T16633 CWE7Q0 44298482 IC50 = 245 nM T16633 CF69PL 44298522 Ki = 484 nM T16633 CRQJ98 44308836 Ki = 537 nM T16633 CRFM02 44308969 Ki = 1.6 nM T16633 C40MJU 44308970 Ki = 0.38 nM T16633 C9KR7Q 44309052 Ki = 2430 nM T16633 C4YG1S 44311590 IC50 = 30.9 nM T16633 CY0OV9 44311591 IC50 = 309 nM T16633 C29GQB 44311601 IC50 = 1 nM T16633 CC8DS0 44311602 IC50 = 450 nM T16633 C5KST2 44311690 IC50 = 35 nM T16633 C6N4MH 44311691 IC50 = 530 nM T16633 CIR4G6 44311695 IC50 = 17.4 nM T16633 CTG6X5 44311696 IC50 = 2.5 nM T16633 C7Y8SF 44311697 IC50 = 8.1 nM T16633 CK52MY 44311702 IC50 = 15.1 nM T16633 CX39CV 44311703 IC50 = 187 nM T16633 C5RM2A 44311730 IC50 = 15 nM T16633 CBG70T 44311731 IC50 = 24 nM T16633 CQH20F 44311765 IC50 > 1000 nM T16633 CZG4K6 44311836 IC50 = 33 nM T16633 CWNP79 44311837 IC50 = 34.7 nM T16633 CWSF38 44311868 IC50 = 103 nM T16633 C2T0YP 44311869 IC50 = 101 nM T16633 C1ONB3 44311870 IC50 = 347 nM T16633 C1GY0F 44311912 IC50 = 3.6 nM T16633 C14DIH 44311913 IC50 > 1000 nM T16633 C1X4TI 44311914 IC50 = 27.3 nM T16633 C64WAE 44311958 IC50 = 130 nM T16633 CFT90E 44311959 IC50 > 1000 nM T16633 C3PQD0 44311960 IC50 = 720 nM T16633 CS7PB4 44312258 IC50 > 1000 nM T16633 C5PE1D 44325273 IC50 = 407 nM T16633 C1P0QV 44332931 Ki = 1800 nM T16633 CHP41F 44363816 Ki = 712 nM T16633 CH2DN4 44367916 IC50 > 10000 nM T16633 CM9YQ0 44367953 IC50 > 10000 nM T16633 C5W4YL 44368019 IC50 = 667 nM T16633 CO6ZJ9 44368020 IC50 > 1000 nM T16633 CQ5T1D 44368043 IC50 > 1000 nM T16633 C1SWO5 44368044 IC50 > 10000 nM T16633 C29EZK 44368080 IC50 = 778 nM T16633 C9ZW6U 44368093 IC50 > 1000 nM T16633 C71URM 44368094 IC50 > 1000 nM T16633 CC1ZP9 44368109 IC50 > 10000 nM T16633 CQ7OP1 44368112 IC50 > 1000 nM T16633 C0EW4I 44368117 IC50 > 1000 nM T16633 C6TNZ9 44368144 IC50 > 1000 nM T16633 C53IAG 44368153 IC50 = 545 nM T16633 CKU8J7 44368156 IC50 = 5.3 nM T16633 CR12GB 44368157 IC50 = 27 nM T16633 C50DMO 44368226 IC50 > 10000 nM T16633 CN31HS 44368398 IC50 > 1000 nM T16633 C2RC0P 44368406 IC50 = 45 nM T16633 CB1HC8 44368422 IC50 > 10000 nM T16633 C27DLY 44368489 IC50 > 10000 nM T16633 CWHK38 44377332 Ki > 10000 nM T16633 CVH1O7 44377366 Ki > 5000 nM T16633 CRC2N1 44377555 Ki = 2900 nM T16633 CS1WT5 44377591 Ki = 4000 nM T16633 C3LUY8 44377623 Ki > 10000 nM T16633 CQD0P4 44377645 Ki > 5000 nM T16633 CWNF42 44385504 Ki = 2570 nM T16633 CAFD79 44385508 Ki > 10000 nM T16633 CHY14B 44385591 Ki = 9100 nM T16633 CJQI19 44385652 Ki = 1520 nM T16633 CG12HD 44385712 Ki = 2840 nM T16633 C8MU5C 44385757 Ki = 1880 nM T16633 C0LRT9 44386389 Ki = 3430 nM T16633 C1EVK8 44387399 Ki = 1030 nM T16633 C6U9VC 44388027 IC50 = 14 nM T16633 C2IW5J 44388028 IC50 = 6.1 nM T16633 C27ANT 44388029 IC50 = 46 nM T16633 CHQK20 44388035 IC50 > 1000 nM T16633 CI9XS1 44388036 IC50 = 259 nM T16633 CD4BX6 44388037 IC50 = 620 nM T16633 CDS08Z 44388038 IC50 > 1000 nM T16633 CZA03Y 44388040 IC50 > 1000 nM T16633 C21WBR 44388043 IC50 > 1000 nM T16633 C7VK6B 44388052 IC50 > 1000 nM T16633 CT93BI 44388060 IC50 = 597 nM T16633 C4E5VS 44388061 IC50 > 1000 nM T16633 C7P5RO 44388066 IC50 > 1000 nM T16633 C7T8IY 44388069 IC50 = 208 nM T16633 C2TWO3 44388070 IC50 > 1000 nM T16633 CDBE87 44388075 IC50 = 5.2 nM T16633 C25GWK 44388078 IC50 > 1000 nM T16633 CT93LV 44388079 IC50 > 1000 nM T16633 CX54SC 44388083 IC50 = 53 nM T16633 C2C0RU 44388084 IC50 = 144 nM T16633 C5SMA2 44388085 IC50 = 255 nM T16633 C26OCG 44388086 IC50 = 30 nM T16633 C8SR2O 44388087 IC50 = 35 nM T16633 CHL5T1 44388088 IC50 > 1000 nM T16633 C4VNC2 44388089 IC50 > 1000 nM T16633 C1IH3T 44388090 IC50 > 1000 nM T16633 CNC91I 44388093 IC50 = 5.8 nM T16633 CN45OF 44388095 IC50 = 8.5 nM T16633 C82HJL 44388104 IC50 = 241 nM T16633 CV6T2H 44388105 IC50 = 554 nM T16633 CLC0N2 44388106 IC50 = 53 nM T16633 C0VO1K 44388107 IC50 = 94 nM T16633 CM5O3B 44388108 IC50 = 16 nM T16633 CAF02P 44388109 IC50 = 782 nM T16633 C23XBM 44388110 IC50 = 204 nM T16633 CPX74G 44388112 IC50 = 22 nM T16633 CG9SA3 44388114 IC50 = 43 nM T16633 C2C4MH 44388116 IC50 = 17 nM T16633 CW1EL5 44388118 IC50 > 1000 nM T16633 CN0K3V 44388119 IC50 = 74 nM T16633 CE8DH4 44388120 IC50 = 61 nM T16633 C1A0OY 44388121 IC50 = 3.3 nM T16633 CS53NP 44388122 IC50 > 1000 nM T16633 CX67WG 44388123 IC50 = 6.7 nM T16633 CB50EK 44388124 IC50 = 4.8 nM T16633 C9SN1X 44388132 IC50 = 64 nM T16633 C6W4YT 44388133 IC50 = 167 nM T16633 CMTN20 44388134 IC50 = 274 nM T16633 CAK42W 44388135 IC50 = 89 nM T16633 CTW48B 44388136 IC50 = 181 nM T16633 C4P1AS 44388137 IC50 = 18 nM T16633 CEAZ82 44388138 IC50 = 62 nM T16633 C1KMT8 44397389 Ki = 58 nM T16633 CN6Z8C 44397648 Ki = 180 nM T16633 CRW0M6 44397706 Ki = 130 nM T16633 CM1R8X 44400000 IC50 > 10000 nM T16633 CP89CS 44400135 IC50 > 10000 nM T16633 C1BY2P 44444935 IC50 > 1000 nM T16633 CH17TI 44560858 IC50 > 1000 nM T16633 C2AZY7 44560859 IC50 > 1000 nM T16633 C2I8NB 44560860 IC50 > 1000 nM T16633 C4XRT0 44560861 IC50 > 1000 nM T16633 C21TZI 44560862 IC50 > 1000 nM T16633 C2YM5N 44560863 IC50 > 1000 nM T16633 CS39FB 44560864 IC50 > 1000 nM T16633 CU3FD2 44560865 IC50 > 1000 nM T16633 C8IKU1 44560866 IC50 > 1000 nM T16633 CTQ83Z 44560867 IC50 > 1000 nM T16633 CQC29N 44560868 IC50 > 1000 nM T16633 C47MDA 44560869 IC50 > 1000 nM T16633 CHAJ41 44560870 IC50 > 1000 nM T16633 CT0A9U 44560871 IC50 > 1000 nM T16633 CM0T9R 44560872 IC50 > 1000 nM T16633 CO2J6R 44560873 IC50 > 1000 nM T16633 CKQD64 44560874 IC50 > 1000 nM T16633 CEK26Y 44560875 IC50 > 1000 nM T16633 CBL1P7 44560876 IC50 > 1000 nM T16633 CY47DM 44560877 IC50 > 1000 nM T16633 C5OZD1 44560878 IC50 > 1000 nM T16633 CFT47C 44560898 IC50 > 1000 nM T16633 CAO7R0 44560899 IC50 > 1000 nM T16633 C80ZCF 44560900 IC50 > 1000 nM T16633 CATH94 44560901 IC50 > 1000 nM T16633 C2AXG6 44560902 IC50 > 1000 nM T16633 COQ9W7 44560903 IC50 > 1000 nM T16633 CLZ23V 44560904 IC50 > 1000 nM T16633 C0OKG2 44560905 IC50 > 1000 nM T16633 CPIW17 44560906 IC50 > 1000 nM T16633 CFR3Y5 44560907 IC50 > 1000 nM T16633 CS85LR 44560908 IC50 > 1000 nM T16633 C6K1FI 44577218 IC50 > 1000 nM T16633 CAJ15T 44577219 IC50 > 1000 nM T16633 CQD56E 44577220 IC50 > 1000 nM T16633 CV18IC 44577221 IC50 = 763 nM T16633 CLJD09 45102042 IC50 > 10000 nM T16633 C63YJS 45139239 IC50 > 1000 nM T16633 C63XPN 45267999 IC50 > 1000 nM T16633 CF09UA 45268875 IC50 = 1 nM T16633 CU3MQ4 45268876 EC50 = 0.93 nM T16633 C2PNH4 45272264 IC50 = 17 nM T16633 CFL9K7 45273129 IC50 > 1000 nM T16633 C9Z4MR 45273130 IC50 > 1000 nM T16633 C4RGN0 45273131 IC50 = 20 nM T16633 C6KBJ2 46882133 Ki = 4950 nM T16633 CU1D6I 46902023 IC50 = 2800 nM T16633 CZ46AH 46911015 IC50 < 300 nM T16633 C84ZTC 49865341 IC50 > 1000 nM T16633 C3VZ4U 49865342 IC50 > 1000 nM T16633 CGYR09 49865343 IC50 = 25 nM T16633 C35WID 49865344 IC50 > 1000 nM T16633 C0RK7G 49865345 IC50 = 1000 nM T16633 C4YLM7 49865346 IC50 > 1000 nM T16633 CZ4RI1 49865347 IC50 = 57.5 nM T16633 C9SNL1 52941607 IC50 > 10000 nM T16633 C40ZRY 52948630 IC50 > 10000 nM T16633 CED3O6 53473658 IC50 = 138 nM T16633 CE7J0U 53473659 IC50 = 140 nM T16633 CY0G2K 53473744 IC50 = 2.7 nM T16633 CBQG96 53473824 IC50 = 4.1 nM T16633 CW53YV 53473917 IC50 > 1000 nM T16633 C87SME 53474004 IC50 > 1000 nM T16633 C7EO1Z 53474005 IC50 > 1000 nM T16633 CY3M2A 53474090 IC50 > 1000 nM T16633 C9JHI4 56664813 Ki = 2 nM T16633 C8ZW3O 56927659 IC50 = 2362 nM T16633 CHK8T1 56945132 Ki = 4750 nM T16633 C73XBL 57384077 IC50 > 1000 nM T16633 C3KC9Z 57398462 IC50 = 3.2 nM T16633 C0DEM2 68254010 IC50 = 6000 nM T16633 CTVI05 70683416 IC50 = 267 nM T16633 CV42WQ 70689221 IC50 > 10000 nM T16633 C3P0AN 70689413 IC50 > 1000 nM T16633 CP58HL 70689414 IC50 > 1000 nM T16633 CB14OW 70689415 IC50 > 1000 nM T16633 CNZC97 70689723 IC50 = 1.2 nM T16633 C2WQM9 70691295 IC50 > 1000 nM T16633 C5E8MY 70693613 IC50 > 1000 nM T16633 C3TZ9U 70695246 IC50 = 495 nM T16633 C34XGS 70695722 IC50 > 1000 nM T16633 CIPF50 70695723 IC50 > 1000 nM T16633 CF08XL 71458043 Ki = 4600 nM T16633 CU82HG 71460000 IC50 = 975 nM T16633 CPC69G 71461645 Ki = 3300 nM T16633 CLAV92 71461684 IC50 > 1000 nM T16633 C1NZU3 71461685 IC50 = 563 nM T16633 CFKH42 71717904 IC50 = 2003 nM T16633 CGDO59 72947672 Ki = 0.31 nM T16633 CIO28F 73345407 Ki = 1000 nM T16633 CMN6X8 73345525 IC50 > 10000 nM T16633 C70XZC 73345528 IC50 > 1000 nM T16633 CXGJ67 73345700 IC50 > 1000 nM T16633 CV23JS 73345701 IC50 > 1000 nM T16633 C81UME 73345740 Ki > 1000 nM T16633 CX5VM1 73346900 IC50 = 443 nM T16633 CA3MU5 73346903 IC50 = 5.4 nM T16633 C62NFY 73346927 Ki = 1000 nM T16633 CK64MX 73346930 Ki = 1000 nM T16633 C15CAN 73346972 Ki > 1000 nM T16633 CD09FU 73347225 Ki > 1000 nM T16633 CI4L6W 73347226 Ki = 736 nM T16633 CGM61R 73348311 Ki > 10000 nM T16633 CN1FD2 73348312 Ki = 4400 nM T16633 C01GIQ 73348427 Ki = 1000 nM T16633 C7Y9ZT 73348428 Ki = 1000 nM T16633 CFLT50 73348719 IC50 > 1000 nM T16633 C75NBQ 73348741 Ki > 1000 nM T16633 C5MNX3 73348742 Ki > 1000 nM T16633 CL94MY 73350006 Ki = 1000 nM T16633 C0N6XK 73350010 Ki = 1000 nM T16633 CTV30F 73350011 Ki = 1000 nM T16633 CF2AK4 73350012 Ki = 1000 nM T16633 CK9CS4 73351516 Ki = 1000 nM T16633 CNY13O 73351517 Ki = 1000 nM T16633 CUN6L1 73351622 IC50 = 607 nM T16633 CC98JE 73351624 IC50 > 1000 nM T16633 CWUH52 73351718 Ki = 1000 nM T16633 CS9I4W 73351829 Ki > 1000 nM T16633 CF70XH 73351873 IC50 = 104 nM T16633 CFB54J 73352985 Ki = 1395 nM T16633 CKFV85 73353009 Ki > 1000 nM T16633 CC45AV 73353272 IC50 > 10000 nM T16633 C41OCY 73353278 IC50 > 1000 nM T16633 CW54CU 73353340 IC50 > 1000 nM T16633 CL7DT2 73354494 Ki = 1000 nM T16633 CA48EL 73354535 Ki > 1000 nM T16633 CFK7Z3 73354633 IC50 > 10000 nM T16633 C1UYL2 73354783 IC50 > 1000 nM T16633 CG1CX0 73354798 IC50 > 1000 nM T16633 CIVZ67 73354818 Ki > 1000 nM T16633 CGCE64 73354819 Ki > 1000 nM T16633 C1Y0CI 73356066 Ki = 1000 nM T16633 C52JAS 73356068 Ki = 395 nM T16633 CN5LG8 73356069 Ki = 1000 nM T16633 C9GKV2 73356181 IC50 = 323 nM T16633 C7XFB6 73356331 IC50 > 1000 nM T16633 CI02SE 73356366 Ki > 1000 nM T16633 CW8L6C 76310862 IC50 > 1000 nM T16633 CHV6K7 76314485 IC50 = 18 nM T16633 C0PR3Y 76314486 IC50 > 1000 nM T16633 C94BWD 76314487 IC50 = 38 nM T16633 C25XKO 76314488 IC50 = 171 nM T16633 CS54IV 76321777 IC50 = 33 nM T16633 C94OAT 76321778 IC50 = 795 nM T16633 CU1IR8 76325402 IC50 = 14 nM T16633 CL09JQ 86279005 IC50 > 10000 nM T16633 C3JOS4 86292350 Ki > 9090 nM T16633 CVLE34 86293506 Ki = 848 nM T16633 C15VTO 86294248 Ki = 4535 nM T16633 C2BAV8 90644981 Ki = 656 nM T16633 CI58FM 90663867 IC50 > 1000 nM T16633 CK62FO 90663868 IC50 > 10000 nM T16633 C7AFD4 90663869 IC50 > 1000 nM T16633 C94XTF 90663872 IC50 > 10000 nM T16633 CA7W0U 90663873 IC50 > 10000 nM T16633 C4EG8T 90663874 IC50 > 10000 nM T16633 CW21UO 90663875 IC50 > 1000 nM T16633 C7Q4PD 90665458 Ki = 153000 nM T16633 CR43ZL 90665459 Ki = 102000 nM T16633 CLK7C3 90665460 Ki = 16000 nM T16633 CZ0UC6 90665461 Ki = 8200 nM T16633 C0IBJ6 90665462 Ki = 16000 nM T16633 CPX0C9 90665463 Ki = 12000 nM T16633 C3UVC8 91936728 IC50 > 10000 nM T16633 CT3UP7 91936729 IC50 > 10000 nM T16633 CD2E4L 101941290 IC50 = 1000 nM T16633 C9KB3W 117711399 Ki = 7360 nM T16633 CTH52C 118718416 Ki = 0.7943 nM T16633 CKQ4P6 118718462 IC50 = 945 nM T16633 C1Z7UJ 118718463 Ki < 1000 nM T16633 CPYA80 118718465 IC50 = 1000 nM T16633 CR61UD 118718466 IC50 = 1000 nM T16633 CW64XN 118718500 IC50 = 1000 nM T16633 CB4D5T 118718501 IC50 = 3219 nM T16633 CW5HG2 118718502 IC50 = 1000 nM T16633 CC36KP 118718503 IC50 = 1086 nM T16633 C7FIQ1 118718504 IC50 = 1008 nM T16633 CNBY57 118718505 IC50 = 1000 nM T16633 CPY4Q5 118718506 IC50 = 245 nM T16633 CO13JR 118718507 IC50 = 1000 nM T16633 CLFJ60 118718508 IC50 = 1439 nM T16633 C13YUH 118718509 IC50 = 588 nM T16633 CP2O7U 118718510 IC50 = 1000 nM T16633 CLDZ63 118718511 IC50 = 1000 nM T16633 CYQ7X2 118718854 IC50 > 1000 nM T16633 CA6C4T 118719101 IC50 = 397 nM T16633 CDZ3H4 118719196 IC50 > 1000 nM T16633 CQRO32 118719197 IC50 > 1000 nM T16633 CGXH91 118719198 IC50 > 1000 nM T16633 C1QJX7 118719199 IC50 > 1000 nM T16633 C0GLC8 118719200 IC50 > 10000 nM T16633 C40NGQ 118719201 IC50 > 10000 nM T16633 CK2W9T 118719202 IC50 > 1000 nM T16633 CW4AT0 118719275 IC50 > 10000 nM T16633 C5VWI1 118719303 IC50 = 1665 nM T16633 CS12JW 122179457 IC50 = 2300 nM T16633 CNGQ19 122179477 IC50 = 1330 nM T16633 CE79SV 138377584 IC50 > 10000 nM T16633 CE76TG 42637005 IC50 = 591 nM T16633 C6ELN4 42637006 IC50 = 356 nM T16633 CS73LG 42637433 IC50 = 449 nM T16633 C6C3YF 45270549 IC50 = 2.5 nM T16633 C9Y3BS 45270550 IC50 = 6.1 nM T16633 CQC51Z 45270552 IC50 > 1000 nM T16633 CXE30U 45271377 IC50 = 3.6 nM T16633 D01BWV 9802572 Ki = 3700 nM T16633 D01NID 44388055 IC50 = 71 nM T16633 D02CQW 11847438 IC50 > 1000 nM T16633 D02NJV 44388048 IC50 = 189 nM T16633 D02OJQ 44388115 IC50 = 10 nM T16633 D02WOX 44388129 IC50 = 33 nM T16633 D03DRL 44388045 IC50 = 176 nM T16633 D03SXC 44388041 IC50 = 325 nM T16633 D03VHX 44388111 IC50 = 25 nM T16633 D04EWA 44388034 IC50 = 535 nM T16633 D04FPW 44388024 IC50 = 720 nM T16633 D04ORV 44388047 IC50 = 5.3 nM T16633 D04QBM 5311374 IC50 > 1000 nM T16633 D05COQ 11847588 IC50 > 1000 nM T16633 D05XZA 44388071 IC50 = 14 nM T16633 D06JWT 44388073 IC50 = 75 nM T16633 D07DUF 44388130 IC50 = 248 nM T16633 D07OSF 44388044 IC50 = 583 nM T16633 D07WRP 15965425 Ki = 2392 nM T16633 D09DAC 44388046 IC50 = 59 nM T16633 D09LHN 44311674 IC50 = 15 nM T16633 D0A0DO 44388056 IC50 = 260 nM T16633 D0A1XX 44388113 IC50 = 45 nM T16633 D0BE3D 44388092 IC50 = 8 nM T16633 D0C5RH 44388125 IC50 = 112 nM T16633 D0CC1P 44388042 IC50 = 69 nM T16633 D0H0DC 44388051 IC50 > 1000 nM T16633 D0H4WH 44388128 IC50 = 0.98 nM T16633 D0I9ME 44388074 IC50 = 7.2 nM T16633 D0J5OY 44388022 IC50 = 79 nM T16633 D0M5LA 44388050 IC50 > 1000 nM T16633 D0N2MA 44388103 IC50 = 15 nM T16633 D0N4LH 44388065 IC50 = 151 nM T16633 D0O4GU 44403230 Ki > 1000 nM T16633 D0P6ZZ 10581102 IC50 > 1000 nM T16633 D0R0OX 44388102 IC50 = 16 nM T16633 D0R4IS 44388131 IC50 = 113 nM T16633 D0S7YR 44388059 IC50 = 14 nM T16633 D0T5RO 16129706 IC50 = 0.14 nM T16633 D0W0AF 44388072 IC50 = 10 nM T16633 D0WG0O 44388049 IC50 > 1000 nM T16633 D0Z0OF 44388094 IC50 = 2.5 nM T16633 D0Z1XY 44388064 IC50 = 23 nM T16633 D0Z3LZ 44388023 IC50 = 197 nM T65783 C2J1RE 351037 IC50 > 79000 nM T65783 CX9FV4 7217852 IC50 > 79000 nM T65783 CR1QE5 7217853 IC50 > 79000 nM T65783 C12BHY 7217856 IC50 > 79000 nM T65783 C86MDE 7217859 IC50 > 79000 nM T65783 C9UBG6 7217861 IC50 > 79000 nM T65783 C3XLA7 7217862 IC50 > 79000 nM T65783 C4Y6JF 7217867 IC50 > 79000 nM T65783 CB8NT2 7217870 IC50 > 79000 nM T65783 CT6F3C 7217876 IC50 > 79000 nM T65783 C8PK9D 7217878 IC50 > 79000 nM T65783 CYX8F6 7217879 IC50 > 79000 nM T65783 CH3I6U 7217884 IC50 > 79000 nM T65783 CI92NG 7217887 IC50 > 79000 nM T65783 C17GSL 7217891 IC50 > 79000 nM T65783 C1W3XE 7217912 IC50 > 79000 nM T65783 C8RWT6 7217913 IC50 > 79000 nM T65783 CFOJ16 7217916 IC50 > 59000 nM T65783 C5LZ0X 7217919 IC50 > 79000 nM T65783 CNG45O 7217921 IC50 = 54500 nM T65783 C2PQ8W 7217922 IC50 > 79000 nM T65783 CA7EW6 7217938 IC50 = 75700 nM T65783 CK9X8S 7217939 IC50 = 59200 nM T65783 CT89GV 7217942 IC50 = 3110 nM T65783 C07ZXA 7217944 IC50 = 72200 nM T65783 CUA9S4 7217946 IC50 = 7250 nM T65783 C7AMT6 7217947 IC50 = 4700 nM T65783 CCE5T6 7217950 IC50 = 29000 nM T65783 CW2AT7 7218011 IC50 > 79000 nM T65783 C9ZEC8 12005825 IC50 = 39900 nM T65783 C1D7HW 12005898 IC50 = 74100 nM T65783 C4K8HT 12005992 IC50 = 1750 nM T65783 CB78RO 16130452 EC50 = 1.9 nM T65783 C0A9WY 16194671 IC50 > 79000 nM T65783 C6J4NC 16805942 IC50 = 18200 nM T65783 C21UXH 16832372 IC50 > 79000 nM T65783 C9IP8D 18572334 IC50 > 79000 nM T65783 CK2L9R 18572335 IC50 = 58800 nM T65783 CO48HV 18572337 IC50 = 51000 nM T65783 CC70BA 18572338 IC50 = 6200 nM T65783 CMG17E 18572343 IC50 = 20600 nM T65783 CQ3ZV0 18572352 IC50 > 79000 nM T65783 CZ2FW0 18572378 IC50 > 79000 nM T65783 COP52X 18572379 IC50 > 79000 nM T65783 CAJH61 18572382 IC50 > 79000 nM T65783 CNKA87 18572395 IC50 > 79000 nM T65783 C27ZCA 25085173 EC50 = 0.0122 nM T65783 C8TX1U 42281625 IC50 > 79000 nM T65783 CB31ST 44726831 IC50 > 79000 nM T65783 CH41CI 46835118 IC50 > 79000 nM T65783 C5LJ0V 46835120 IC50 > 79000 nM T65783 CSBO37 46835124 IC50 > 79000 nM T65783 C6EFX7 46905014 IC50 > 79000 nM T65783 CCUA93 46905018 IC50 = 8510 nM T65783 C85DJM 46905020 IC50 > 79000 nM T65783 CBNT43 46905022 IC50 > 79000 nM T65783 CH20YA 46905025 IC50 > 79000 nM T65783 CWER26 46905028 IC50 = 9610 nM T65783 CD3CK1 46905029 IC50 = 6590 nM T65783 CU6D2Q 46905034 IC50 = 3210 nM T65783 CWY35N 46905037 IC50 > 79000 nM T65783 CP3M2F 46905038 IC50 > 79000 nM T65783 CQK7D4 49787115 IC50 > 79000 nM T65783 C86OIB 49787117 IC50 > 79000 nM T65783 CL3D2B 49787119 IC50 > 79000 nM T65783 CP5M7Y 49787120 IC50 > 79000 nM T65783 CW9G1R 49842899 IC50 = 24000 nM T65783 CVC2N3 49842902 IC50 = 4530 nM T65783 C9T3AM 49842903 IC50 = 8270 nM T65783 CQ6V4E 49842905 IC50 = 12800 nM T65783 C62CDL 49842908 IC50 > 79000 nM T65783 CCQK74 71456693 IC50 > 79000 nM T65783 CGM32X 71462076 IC50 > 79000 nM T65783 C0DO6L 90644396 EC50 > 30000 nM T65783 CWY43T 90644398 EC50 > 30000 nM T65783 CM1HI5 90656606 EC50 = 237 nM T65783 CEA07I 90656607 EC50 = 494 nM T65783 CKF15X 90656608 EC50 = 539 nM T65783 C6V8TM 90656609 EC50 = 637 nM T65783 CO51PF 90656610 EC50 = 691 nM T65783 C7QO0V 90656611 EC50 = 936 nM T65783 C2Q6JA 90656612 EC50 = 1383 nM T65783 C34OGA 90656613 EC50 = 2350 nM T65783 C7V8EM 90656614 EC50 > 3000 nM T65783 CXRO89 90656615 EC50 > 3000 nM T65783 CBAT91 90656616 EC50 > 3000 nM T65783 C8SH3Y 90656617 EC50 > 3000 nM T65783 C18FEA 90656618 EC50 > 3000 nM T65783 CSO54R 90656619 EC50 > 3000 nM T65783 CQ41HU 90656620 EC50 = 1.1 nM T65783 CU9WH0 90656621 EC50 = 1.7 nM T65783 CUP8F7 90656622 EC50 = 1.9 nM T65783 CDIT19 90656623 EC50 = 2.2 nM T65783 C8X2RV 90656624 EC50 = 3.2 nM T65783 C3ZYS4 90656625 EC50 = 4.4 nM T65783 C40WHE 90656626 EC50 = 4.7 nM T65783 CB3FP8 90656627 EC50 = 8.9 nM T65783 CS24BV 90656628 EC50 = 19 nM T65783 CB3GE1 90656629 EC50 = 20 nM T65783 CPM9T5 90656630 EC50 = 31 nM T65783 CF2K0U 90656631 EC50 = 33 nM T65783 C42XWN 90656632 EC50 = 44 nM T65783 CIG7P5 90656633 EC50 = 73 nM T65783 C4J2ZT 90656634 EC50 > 31622.78 nM T65783 C6A0XD 90656635 EC50 > 31622.78 nM T65783 C7CAH3 90656636 EC50 = 83.18 nM T65783 CH95OZ 118568543 EC50 > 30000 nM T65783 CW49MU 118568545 EC50 > 30000 nM T65783 CDN05V 118568560 EC50 > 30000 nM T65783 C1C2IW 118568561 EC50 > 30000 nM T65783 C9FZ8G 118568562 EC50 > 30000 nM T65783 C28JSA 118568565 EC50 > 30000 nM T65783 CMT3D1 118568636 EC50 > 30000 nM T65783 CI69JT 118568646 Ki = 600 nM T65783 C3XF1J 118568676 EC50 > 30000 nM T65783 C12TDY 118568780 EC50 > 30000 nM T65783 CL0J9I 118568782 EC50 > 30000 nM T65783 CJ5PN1 118568784 EC50 > 30000 nM T65783 C63ZXV 118568855 EC50 > 30000 nM T65783 C52VYU 118568856 EC50 > 30000 nM T65783 CR2Z9X 118568860 EC50 > 30000 nM T65783 C2M3GZ 118568863 EC50 > 30000 nM T65783 CUL40R 118568915 EC50 > 30000 nM T65783 C04CFZ 118568917 EC50 > 30000 nM T65783 CAGX81 118568919 EC50 > 30000 nM T65783 CMZ87V 118568922 EC50 > 30000 nM T65783 CS9PK1 118568930 EC50 > 30000 nM T65783 CUV5Y0 118715454 EC50 = 33.7 nM T65783 C6GV2L 118715455 EC50 > 30000 nM T65783 CQ1DR4 118715456 EC50 > 30000 nM T65783 C7BI9F 118715457 EC50 = 198.6 nM T65783 C7LC0E 118715458 EC50 = 41.3 nM T65783 CZHB45 118715459 EC50 > 30000 nM T65783 C3W1VQ 118715460 EC50 > 30000 nM T65783 CD89JW 118715461 EC50 > 30000 nM T65783 CAJ0T1 118715462 EC50 > 30000 nM T65783 C6VR9K 118715463 EC50 = 21.5 nM T65783 C9H6VU 118715464 EC50 = 95.7 nM T65783 CSJV63 118715465 EC50 > 30000 nM T65783 C80LTN 118715466 EC50 = 2.7 nM T65783 CJB6N8 118715467 EC50 > 30000 nM T65783 CS2V3H 118715468 EC50 > 30000 nM T65783 CML9P4 118715469 EC50 > 30000 nM T65783 C5WPH4 118715470 EC50 > 30000 nM T65783 C9OE3S 118715471 EC50 > 30000 nM T65783 CWX0L5 118715472 EC50 > 30000 nM T65783 C5N6XM 118715473 EC50 > 30000 nM T65783 CAJS62 118715474 EC50 > 30000 nM T65783 C9GU6K 118715475 EC50 > 30000 nM T65783 C0GEY6 118715476 EC50 > 30000 nM T65783 CXN6C1 118715477 EC50 = 225.5 nM T65783 CM5L8N 118715478 EC50 > 30000 nM T65783 CK4BT2 118715479 EC50 > 30000 nM T65783 CGRB51 118734703 EC50 = 0.53 nM T65783 C1LI8R 118734704 EC50 = 2.5 nM T65783 C8C5KO 118734767 EC50 = 1.3 nM T65783 C9ZWT7 118734768 EC50 = 2.7 nM T65783 C2H6BG 118734769 EC50 = 0.23 nM T65783 C63JPQ 118734770 EC50 = 0.17 nM T65783 C8H7JV 118734771 EC50 = 0.45 nM T65783 CSB8T7 118734772 Ki = 1.3 nM T65783 CT4AL0 118734773 EC50 = 3 nM T65783 C16IYO 118734774 EC50 = 2.7 nM T65783 CWG68D 118734775 EC50 = 0.24 nM T65783 CI8X3T 118734776 Ki = 0.016 nM T65783 C0S4AY 118734777 EC50 = 0.04 nM T65783 C87ZQV 118734778 EC50 = 0.63 nM T65783 C43YQF 118734779 EC50 = 6 nM T65783 CD8K0G 118734780 EC50 = 1.3 nM T65783 CBP0F2 118734781 EC50 = 0.07 nM T65783 C6FE7W 118734782 Ki = 0.69 nM T65783 CDS7I4 118734783 EC50 = 1.1 nM T65783 C4D3ZK 118734784 Ki = 46 nM T65783 CVD6R8 118734785 Ki > 10000 nM T65783 C3SVZ9 118734786 Ki > 10000 nM T65783 CZ93DF 118734787 Ki > 10000 nM T65783 CY4IS2 127043374 EC50 = 0.1175 nM T65783 CG0B6M 127044072 Ki = 11 nM T65783 CV98XE 127044698 Ki = 0.53 nM T65783 C0AQ2M 127045179 EC50 = 36 nM T65783 C1DOZ7 127045180 Ki = 3.4 nM T65783 C7PG9N 127045189 Ki = 8.4 nM T65783 CAYI14 127048431 EC50 > 30000 nM T65783 C3WSB4 127051011 Ki = 1400 nM T65783 CI1WH7 127051222 Ki = 3000 nM T65783 CNUA86 127051280 EC50 = 800 nM T65783 CR9PV6 127052214 EC50 > 30000 nM T65783 C45ZLA 134828250 EC50 = 0.2884 nM T65783 CM3L9F 137224964 EC50 > 30000 nM T65783 CB3N6E 137225067 EC50 > 30000 nM T65783 CD1OV6 137501999 EC50 = 0.093 nM T65783 C54VFS 137502080 EC50 = 0.083 nM T65783 CU62XA 137502125 EC50 = 1.4 nM T65783 CN5KB9 137502168 EC50 = 7.4 nM T65783 CKW9L0 137631382 Ki = 188 nM T65783 C3Z0OT 137632615 EC50 = 4.9 nM T65783 C48ZSL 137633995 Ki = 523 nM T65783 CB1WI7 137635080 Ki = 194 nM T65783 CI0BM8 137638986 Ki = 6074 nM T65783 C3TN2R 137639006 EC50 = 0.8 nM T65783 C0BFG1 137639727 Ki = 1.9 nM T65783 CG3IH1 137641320 Ki = 917 nM T65783 CJN34B 137643637 Ki = 14 nM T65783 CGXF65 137645721 Ki = 41 nM T65783 C6M1DB 137646730 Ki = 3 nM T65783 CIR0E2 137647010 Ki = 2.9 nM T65783 CNM5T3 137649041 Ki = 0.1 nM T65783 CB9TJ2 137649272 Ki = 5.7 nM T65783 CDC79S 137649320 EC50 = 0.4 nM T65783 CYN21T 137649702 Ki = 509 nM T65783 CYJ61K 137649936 Ki = 206 nM T65783 C1R2JM 137650169 EC50 = 2.1 nM T65783 C8UPE0 137650201 Ki = 310 nM T65783 C7E3TJ 137650464 Ki = 0.3 nM T65783 C2FNP8 137650548 Ki = 1.4 nM T65783 C78RKA 137650891 Ki = 445 nM T65783 C3OI7C 137650935 Ki = 1.1 nM T65783 C6PJB4 137651612 Ki = 489 nM T65783 C2EYV9 137652055 Ki > 10000 nM T65783 C9XIL8 137653279 Ki = 41 nM T65783 C64CAP 137654306 Ki = 268 nM T65783 C12MDR 137654459 EC50 = 2 nM T65783 C8E4TP 137654488 Ki = 0.15 nM T65783 CHS13O 137657220 Ki = 3.9 nM T65783 CZ2W4O 137657369 Ki > 10000 nM T65783 CH1TJ2 137658661 Ki = 9.1 nM T65783 CP93BF 137660518 Ki = 4.5 nM T65783 CZF97Q 137661816 EC50 = 4.1 nM T65783 C59HBK 145948593 Ki = 0.14 nM T65783 CZ2AO7 145948594 EC50 = 22 nM T65783 CA0RT3 145948599 Ki = 0.37 nM T65783 CZF6H8 145948600 Ki = 14 nM T65783 CJ2RY1 145948634 Ki = 0.93 nM T65783 CU2QW4 145948635 Ki = 0.19 nM T65783 C71CST 145948636 Ki = 0.14 nM T65783 C1QLU9 145948641 Ki = 6.8 nM T65783 C35JCH 145948642 Ki = 0.84 nM T65783 CE97TL 145948643 EC50 = 147 nM T65783 C8RW6H 145948663 Ki = 4 nM T65783 C8W0LA 145948664 EC50 = 19 nM T65783 CXY19O 145948665 Ki = 0.23 nM T65783 C27DKH 145948668 Ki = 48 nM T65783 C3CYU6 145948669 EC50 = 20 nM T65783 CG74BR 145948671 Ki = 0.34 nM T65783 CHZI56 145948672 Ki = 20 nM T65783 C81UGK 154603299 EC50 = 0.18 nM T65783 CXI28P 154603335 EC50 = 0.31 nM T65783 COES94 154603343 EC50 = 19 nM T65783 CYT83N 154603359 EC50 = 0.51 nM T65783 CKY36L 154603363 EC50 = 1.5 nM T65783 CE3Q6L 154603384 EC50 = 9 nM T65783 CCD21A 154603387 EC50 = 5.7 nM T65783 C9O1UP 154603393 EC50 = 5.7 nM T65783 CE17OJ 154603397 EC50 = 0.6 nM T65783 CLY4A3 154995949 EC50 = 0.062 nM T65783 CQ8LU1 155004167 EC50 = 51 nM T65783 CX7G0Z 155513131 EC50 = 50 nM T65783 C8D1MN 155514255 EC50 = 176 nM T65783 CNS13I 155514812 EC50 = 11.3 nM T65783 C2F4BN 155515730 EC50 = 29 nM T65783 C6PD7V 155516838 EC50 = 2.7 nM T65783 CSH8L0 155516953 EC50 = 0.19 nM T65783 CEF4W2 155529276 EC50 = 0.1 nM T65783 C1NCA3 155530998 EC50 = 6.3 nM T65783 CSO3T4 155536031 EC50 = 2.5 nM T65783 C5WY4V 155543212 EC50 = 4900 nM T65783 CO0PQ5 155550782 EC50 = 2.6 nM T65783 CRV3E4 155553677 EC50 = 59 nM T65783 CJ68GT 155557915 EC50 = 568 nM T65783 C8AWJ3 155558340 EC50 = 2100 nM T65783 C1PQR8 155566712 EC50 = 0.33 nM T65783 D00QYH 25078060 EC50 = 0.87 nM T65783 D05NXX 7217941 IC50 = 700 nM T65783 D0I8TR 46905036 EC50 = 3700 nM T98933 D0L5WM 2157 IC50 = 600 nM T98933 D0S6JG 5920 Ki = 0.08 nM T98933 D0Z4EI 55245 Ki > 2250 nM T98933 D01QXY 9862248 Ki = 0.32 nM T98933 D03MYO 15981237 EC50 = 210 nM T98933 D07ZTD 15942005 Ki = 600 nM T98933 D0J6XC 5803 IC50 = 0.048 nM T98933 D0V5FQ 166559 Ki = 2.17 nM T98933 D02WGY 10299876 Ki = 0.43 nM T98933 D07EGS 9874938 Ki = 0.47 nM T98933 CNJ29A 861 IC50 = 0.103 nM T98933 CLSK17 5804 IC50 = 0.019 nM T98933 C47GSU 79170 IC50 = 9100 nM T98933 C40JPQ 447271 Ki = 0.03 nM T98933 C57HCR 652088 IC50 = 69800 nM T98933 CB6HQ4 656928 IC50 = 0.6166 nM T98933 CG59SJ 2404806 IC50 = 23100 nM T98933 CJN3P5 4266779 IC50 = 16500 nM T98933 CU1I3O 4652254 IC50 > 100000 nM T98933 C3S6ZI 5184800 IC50 = 4100 nM T98933 C79ZDX 5287525 IC50 = 175 nM T98933 C6ZXJ7 6431911 IC50 = 0.1096 nM T98933 CRQ1O4 9819350 Ki = 0.5 nM T98933 C4PCB9 9825337 EC50 = 49 nM T98933 CZ4I9T 9828296 Ki = 0.46 nM T98933 CQR6U0 9838979 IC50 = 47 nM T98933 C3MZ1Y 9843007 Ki = 7.8 nM T98933 CJ6E2M 9847869 Ki = 0.63 nM T98933 CA27CJ 9862799 IC50 = 20.89 nM T98933 CZ82PF 9863447 Ki = 0.24 nM T98933 CC64MT 9869395 IC50 = 910 nM T98933 CZ1U7X 9932398 IC50 = 2.089 nM T98933 CY01RH 9933119 IC50 = 0.095 nM T98933 CHG6L7 9933993 IC50 = 18 nM T98933 CFS8T0 9944477 IC50 = 2620 nM T98933 C46NXU 9951790 Ki = 0.06 nM T98933 CFH9D2 9968513 IC50 = 1300 nM T98933 CN30MV 9980009 EC50 = 500 nM T98933 CX4MZ9 9980722 IC50 = 1.8 nM T98933 CZ96GN 10030727 IC50 = 12 nM T98933 CJ05DK 10049652 IC50 = 1.8 nM T98933 CP1R7A 10113366 IC50 = 120 nM T98933 CY8S9M 10133886 IC50 = 110 nM T98933 C72HTV 10135986 IC50 = 520 nM T98933 CMY69T 10137392 IC50 = 360 nM T98933 CGE9I7 10151760 Ki = 8.2 nM T98933 CUC0Y8 10172901 Ki = 59 nM T98933 C1Y3FJ 10174187 Ki = 6 nM T98933 CD4SX7 10202877 IC50 = 820 nM T98933 CNPD04 10216950 Ki = 1.19 nM T98933 CDY6F5 10238439 Ki = 3.7 nM T98933 C1DYU9 10269704 Ki = 10 nM T98933 CJB2E3 10274474 Ki = 0.4 nM T98933 C7UYX0 10276774 Ki = 0.5 nM T98933 CH5NX1 10279835 Ki = 2 nM T98933 CW26FQ 10287060 Ki = 2.59 nM T98933 CIB52S 10297431 IC50 = 141.25 nM T98933 CSC3T4 10299993 IC50 = 15.85 nM T98933 C81BSZ 10309431 Ki = 15.1 nM T98933 C09IJX 10310671 Ki = 57.6 nM T98933 CT13FC 10310672 Ki = 53.5 nM T98933 C0VMH3 10321482 IC50 = 680 nM T98933 C7TGL0 10322653 Ki = 0.51 nM T98933 CN3G5V 10390904 Ki = 0.07 nM T98933 CL81KF 10413582 EC50 = 380 nM T98933 CP8O0Q 10455127 IC50 = 13 nM T98933 C3UAD9 10456672 IC50 = 0.3 nM T98933 C5N7BD 10456830 IC50 = 0.025 nM T98933 C34MFS 10457976 IC50 = 22 nM T98933 C4T6ZH 10479778 IC50 = 0.3 nM T98933 CM4ED8 10479779 IC50 = 0.28 nM T98933 CU42IL 10897325 IC50 = 4000 nM T98933 CX2RY1 10904700 IC50 = 0.1514 nM T98933 CZ3SX1 10918755 IC50 = 480 nM T98933 CD9G7N 11164881 IC50 = 1819.7 nM T98933 C6OX1A 11209929 IC50 = 32000 nM T98933 CPY31C 11247142 IC50 = 120 nM T98933 CA8Z1T 11281247 IC50 = 810 nM T98933 CY0M1L 11395277 IC50 = 1800 nM T98933 C48UZO 11463526 IC50 = 700 nM T98933 C5CZ2Q 11998611 Ki = 14600 nM T98933 CRJ1N9 11999781 Ki = 2.5 nM T98933 C7N4HR 11999783 Ki = 1.51 nM T98933 CW01OG 12001110 EC50 = 40 nM T98933 C1AU0V 13958302 Ki = 238 nM T98933 CDB93J 15219550 IC50 = 17700 nM T98933 CDKZ56 15940421 Ki = 42.1 nM T98933 CM17XO 15941848 Ki = 2.17 nM T98933 C1QZ3U 15941849 Ki = 36 nM T98933 CRK5V2 15941850 Ki = 271 nM T98933 C7PV1O 15941997 Ki = 2.51 nM T98933 C7BD0S 15941998 Ki = 30.5 nM T98933 C93MUZ 15942131 Ki = 6.64 nM T98933 CNCW45 15942413 Ki = 9.1 nM T98933 CEQ1J5 15981204 EC50 = 7750 nM T98933 CZEJ29 15981205 EC50 = 7010 nM T98933 C47AYJ 15981206 EC50 = 460 nM T98933 CRF9T7 15981207 EC50 = 2380 nM T98933 C4XF0E 15981234 EC50 = 700 nM T98933 C7U4OQ 15981235 EC50 = 670 nM T98933 CT9N6B 15981236 EC50 = 120 nM T98933 CTI37Q 15981238 EC50 = 120 nM T98933 CIM62O 15981239 EC50 = 770 nM T98933 CB6UE5 15981240 EC50 = 220 nM T98933 CL0FG1 15981241 EC50 = 90 nM T98933 C4BU2G 15981272 EC50 = 2990 nM T98933 C5BO7H 15981273 EC50 = 600 nM T98933 CES0V2 15981274 EC50 = 2040 nM T98933 CCKG05 15981275 EC50 = 9170 nM T98933 C2SR1B 15981276 EC50 = 6980 nM T98933 CIB52A 15981279 EC50 = 140 nM T98933 CWK35C 16730429 IC50 = 60 nM T98933 C7G2AM 18415120 Ki = 15.5 nM T98933 CD0L4R 21110667 Ki = 12 nM T98933 C0AQU8 21110669 Ki = 30 nM T98933 CZI6V2 21110670 Ki = 41 nM T98933 C47HQO 21110672 Ki = 40 nM T98933 CV3FE0 21110673 Ki = 17 nM T98933 CCGP69 21110677 Ki = 53.6 nM T98933 CM0DL5 21110680 Ki = 81.3 nM T98933 CHN91T 21110689 Ki = 39.9 nM T98933 CHT5Y9 21110691 Ki = 19.7 nM T98933 C7TN9A 21110692 Ki = 40.2 nM T98933 CX5I2A 21636517 IC50 = 66000 nM T98933 C6TCO8 21992496 IC50 = 1320 nM T98933 C5EFH7 21992497 IC50 = 88 nM T98933 CO3X7S 21992575 IC50 = 48 nM T98933 COV0S9 21992584 IC50 = 121 nM T98933 CVD9T3 21992651 IC50 = 646 nM T98933 C0QS8C 21992678 IC50 = 78 nM T98933 C5N7DG 21992681 IC50 = 343 nM T98933 CSY41F 21992749 IC50 = 4000 nM T98933 CTF0Q7 21992824 IC50 = 877 nM T98933 C7KTU1 21992839 IC50 = 9290 nM T98933 C6QNL9 21992913 IC50 = 71 nM T98933 CNF16U 22339386 Ki = 0.1 nM T98933 CF2X6V 22339458 Ki = 0.04 nM T98933 CD08GC 22339531 Ki = 0.72 nM T98933 C3HMF6 22339537 Ki = 13 nM T98933 CF7ZI8 22339599 Ki = 0.64 nM T98933 CASB98 22339607 Ki = 1.9 nM T98933 CNLT41 22339633 Ki = 0.13 nM T98933 C89IYX 22339645 Ki = 0.02 nM T98933 CV57KF 22339648 Ki = 27 nM T98933 CY2HZ3 22339678 IC50 = 0.6457 nM T98933 CWV5B9 22339727 Ki = 0.4 nM T98933 CK0C8N 22339743 Ki = 0.46 nM T98933 CF2CQ7 22372339 IC50 = 61000 nM T98933 CR7DC6 23546124 IC50 = 104 nM T98933 CFV3P7 23635238 IC50 = 1500 nM T98933 CWE74Y 23635239 IC50 = 1600 nM T98933 CM6S4G 23635240 IC50 = 2000 nM T98933 CPR67K 23635363 IC50 = 3900 nM T98933 CI6D4Y 23635365 IC50 = 12100 nM T98933 CAHT12 23635366 IC50 = 12700 nM T98933 C1G2TO 23635477 IC50 = 23200 nM T98933 C17PKJ 23635478 IC50 > 100000 nM T98933 CC3VU5 23635479 IC50 > 100000 nM T98933 CGU3Z0 23635480 IC50 > 100000 nM T98933 C82WJG 23635600 IC50 = 55800 nM T98933 C18SZO 23635729 IC50 = 20300 nM T98933 C7BLC2 23635731 IC50 > 100000 nM T98933 CE6DP7 23635732 IC50 > 100000 nM T98933 CGL6T0 23635852 IC50 > 100000 nM T98933 CK4XI2 23635853 IC50 > 100000 nM T98933 CY80FR 23635854 IC50 > 100000 nM T98933 C7NAV1 23635855 IC50 = 35100 nM T98933 CU81CL 23635857 IC50 > 100000 nM T98933 C31FPX 23635859 IC50 > 100000 nM T98933 CQ2E7G 23642624 IC50 = 85900 nM T98933 CB38IZ 23644731 IC50 = 67.61 nM T98933 CT5QC3 23648079 IC50 = 0.11 nM T98933 CP7SV3 23648080 IC50 = 2.7 nM T98933 CYU20W 23648081 IC50 = 1.3 nM T98933 C3V1BH 23648082 IC50 = 5.9 nM T98933 C1JIZ5 23648083 IC50 = 0.27 nM T98933 C3QR1F 23648084 IC50 = 0.71 nM T98933 C0N2YD 23648085 IC50 = 0.78 nM T98933 C08JWQ 23648086 IC50 = 0.6 nM T98933 C5INJ3 23648087 IC50 = 290 nM T98933 CTJK20 23648089 IC50 = 1400 nM T98933 CE4R6V 23648090 IC50 = 2600 nM T98933 C84TAV 23648093 IC50 = 200 nM T98933 CB7OK8 23648094 IC50 = 160 nM T98933 C45JQX 23648095 IC50 = 190 nM T98933 C80CEB 23648096 IC50 = 87 nM T98933 CV20UI 23648101 IC50 = 0.1995 nM T98933 CIKD57 23648102 IC50 = 4.266 nM T98933 CV91YT 23648103 IC50 = 46.77 nM T98933 C5WKV2 23648104 IC50 = 44.67 nM T98933 C5V6OQ 23648105 IC50 = 2.884 nM T98933 C91FSP 23648106 IC50 = 3.236 nM T98933 CBD9J5 23648107 IC50 = 0.8511 nM T98933 C3R0GX 23648108 IC50 = 67.61 nM T98933 C1SXM0 23648109 IC50 = 3.981 nM T98933 C98FIL 23648110 IC50 = 20.89 nM T98933 C7R2XE 23648111 IC50 = 10.96 nM T98933 CR85SZ 23648112 IC50 = 0.7762 nM T98933 CN2YX0 23648113 IC50 = 3.388 nM T98933 CC69AB 23648114 IC50 = 50.12 nM T98933 COP12V 23648115 IC50 = 75.86 nM T98933 CN5T8D 23648116 IC50 = 87.1 nM T98933 C7ON2Q 23648118 IC50 = 40.74 nM T98933 CTR20F 23648121 IC50 = 7.762 nM T98933 CXTZ50 23648122 IC50 = 6.026 nM T98933 CZ8J0T 23648123 IC50 = 7.586 nM T98933 C12HDM 23648124 IC50 = 1.096 nM T98933 C0UJ6X 23648125 IC50 = 9.55 nM T98933 CFA1Y6 23648126 IC50 = 60.26 nM T98933 C35AZQ 23648127 IC50 = 83.18 nM T98933 CR1S4E 23648128 IC50 = 46.77 nM T98933 C0WY3I 23648129 IC50 = 6.026 nM T98933 CL60SF 23648130 IC50 = 34.67 nM T98933 C72TJZ 23648131 IC50 = 4.169 nM T98933 COL8Q7 23648132 IC50 = 6.761 nM T98933 CNWC43 23648133 IC50 = 18.2 nM T98933 C4SW8I 23648134 IC50 = 4.786 nM T98933 CQ7M3I 23648135 IC50 = 4.898 nM T98933 CQW43F 23648136 IC50 = 8.511 nM T98933 C62YFJ 23648137 IC50 = 37.15 nM T98933 CICP87 23648138 IC50 = 67.61 nM T98933 CWT25S 23648139 IC50 = 3.467 nM T98933 C5XD8Q 24830528 IC50 = 40 nM T98933 CR2A9H 24830680 EC50 = 220 nM T98933 CD6EI3 24830686 EC50 = 190 nM T98933 CKDP62 24830833 EC50 = 1300 nM T98933 CO9E2H 24894049 EC50 = 317 nM T98933 C5BS8M 25149230 Ki = 26 nM T98933 CJ6LC2 25149503 Ki = 9.72 nM T98933 CT0J6H 25149504 Ki = 106 nM T98933 CFW74J 25149505 Ki = 146 nM T98933 C5MFE8 25149592 Ki = 52.3 nM T98933 CLSD47 25149598 Ki = 25.4 nM T98933 CZP70F 25150124 Ki = 89.7 nM T98933 C4MT7I 25150127 Ki = 87 nM T98933 C7G5CL 25150225 Ki = 128 nM T98933 C57AUE 25150325 Ki = 0.84 nM T98933 CLZ86A 25150424 Ki = 0.97 nM T98933 CRW82I 44136896 IC50 = 430 nM T98933 C2Y6AG 44185845 IC50 = 1100 nM T98933 COT19A 44185854 IC50 = 600 nM T98933 CSQ1C0 44185855 IC50 = 1700 nM T98933 CTG0X6 44185856 IC50 = 1100 nM T98933 C1L8KQ 44185857 IC50 = 1100 nM T98933 C2VWY6 44185858 IC50 = 5300 nM T98933 CXF3N9 44185859 IC50 = 11200 nM T98933 C8GIP0 44185860 IC50 = 4000 nM T98933 CC4E7U 44185914 IC50 = 4200 nM T98933 CMS09A 44185915 IC50 = 600 nM T98933 C1GI8D 44185916 IC50 = 500 nM T98933 CQAT73 44186032 IC50 = 7100 nM T98933 CC0YN9 44186033 IC50 > 50000 nM T98933 C7VZI4 44186034 IC50 = 10100 nM T98933 CR1D9P 44186035 IC50 = 5300 nM T98933 CC32IS 44186097 IC50 = 7000 nM T98933 C2MG6T 44186098 IC50 = 25300 nM T98933 C4XV1B 44186099 IC50 = 5100 nM T98933 CFJ0P8 44186100 IC50 > 50000 nM T98933 C31NSX 44186101 IC50 = 4700 nM T98933 CBM5Z6 44186102 IC50 = 1800 nM T98933 CX10SK 44186103 IC50 = 2600 nM T98933 C8TU3K 44186104 IC50 = 2700 nM T98933 CWY0A2 44186168 IC50 = 8400 nM T98933 CO65HR 44186169 IC50 = 2700 nM T98933 C1TU5I 44186170 IC50 = 1900 nM T98933 CC49MP 44186171 IC50 = 5000 nM T98933 C3M4KR 44186172 IC50 = 1790 nM T98933 C4COU6 44186173 IC50 = 600 nM T98933 CPZ6T3 44186174 IC50 = 690 nM T98933 C40ENX 44186175 IC50 > 50000 nM T98933 CIL71S 44186232 IC50 > 50000 nM T98933 CP1A5G 44186233 IC50 > 50000 nM T98933 C4CMU9 44186234 IC50 > 50000 nM T98933 CM9V8Z 44186235 IC50 = 1700 nM T98933 CDI86U 44186236 IC50 = 1600 nM T98933 C2YL8N 44186237 IC50 = 18900 nM T98933 CYO36K 44186238 IC50 = 22000 nM T98933 CRHL62 44186239 IC50 = 3800 nM T98933 CS2N6F 44186298 IC50 > 50000 nM T98933 CES48R 44186299 IC50 > 50000 nM T98933 C6XEM3 44186300 IC50 > 50000 nM T98933 C35QER 44186301 IC50 > 50000 nM T98933 CREP27 44186302 IC50 > 50000 nM T98933 CPLW35 44186303 IC50 = 4900 nM T98933 C1PFT0 44186305 IC50 > 50000 nM T98933 C5A1HF 44186364 IC50 = 4600 nM T98933 C6PW0U 44186365 IC50 = 4800 nM T98933 CYE39G 44186366 IC50 = 1200 nM T98933 CS6MG3 44186367 IC50 = 5000 nM T98933 C7CP9D 44186368 IC50 = 1200 nM T98933 CC35ST 44186369 IC50 = 1200 nM T98933 CA62XQ 44186370 IC50 = 5000 nM T98933 C1O4YR 44186418 IC50 = 2000 nM T98933 CYH8U5 44186419 IC50 = 1700 nM T98933 C95GQS 44186420 IC50 = 800 nM T98933 CA1EV7 44186421 IC50 = 10400 nM T98933 CU64OD 44186422 IC50 = 5000 nM T98933 C9J0YD 44186423 IC50 = 4300 nM T98933 C25UOE 44186424 IC50 = 1400 nM T98933 CX9U3Q 44186425 IC50 = 2100 nM T98933 CTF94W 44186465 IC50 = 1500 nM T98933 C9G8JS 44186466 IC50 = 800 nM T98933 C7TFN6 44186467 IC50 = 2000 nM T98933 CD2UC4 44186468 IC50 = 1900 nM T98933 C0Z9OK 44186469 IC50 = 2400 nM T98933 CTJ1O5 44186470 IC50 = 3000 nM T98933 CN8QS2 44186471 IC50 = 700 nM T98933 C78TSP 44186472 IC50 = 1100 nM T98933 CL17KI 44186473 IC50 = 14100 nM T98933 COL0S6 44186474 IC50 = 4000 nM T98933 C75UOJ 44186475 IC50 > 50000 nM T98933 C1KVH2 44186476 IC50 > 50000 nM T98933 CK58UR 44186510 IC50 = 5400 nM T98933 CF1CU6 44186511 IC50 = 2000 nM T98933 CQB3X5 44186512 IC50 = 1700 nM T98933 C01ARC 44186513 IC50 = 1300 nM T98933 C7T3SZ 44186514 IC50 = 1300 nM T98933 CI27LX 44186515 IC50 = 900 nM T98933 C3DOF6 44186516 IC50 = 1200 nM T98933 C3SH2I 44186517 IC50 = 2300 nM T98933 C8X1EA 44186518 IC50 = 2700 nM T98933 CS7K3Y 44186519 IC50 = 5600 nM T98933 CHW5K6 44186520 IC50 > 50000 nM T98933 C58YWK 44186521 IC50 > 50000 nM T98933 CJPO14 44186523 IC50 = 5900 nM T98933 C3JN6A 44186555 IC50 = 4000 nM T98933 CUN70K 44186556 IC50 = 1000 nM T98933 C7CQN6 44186557 IC50 = 800 nM T98933 C9RI1Q 44186558 IC50 = 700 nM T98933 CP26OY 44186559 IC50 = 2400 nM T98933 C7FRJ9 44186560 IC50 = 1700 nM T98933 CB6C9M 44186561 IC50 = 1300 nM T98933 C2NPV9 44186562 IC50 = 12400 nM T98933 CYH38F 44186563 IC50 > 50000 nM T98933 C9G8SO 44186564 IC50 = 1800 nM T98933 C05IDW 44186565 IC50 = 2000 nM T98933 C73VSR 44186566 IC50 = 700 nM T98933 C3PH5N 44186567 IC50 = 600 nM T98933 C1F2WL 44186568 IC50 = 1400 nM T98933 CS6UN0 44186600 IC50 = 1600 nM T98933 CX5B3F 44186601 IC50 = 900 nM T98933 C9BJU8 44186602 IC50 = 3600 nM T98933 CE5MK1 44186603 IC50 = 2300 nM T98933 C1INA4 44186604 IC50 = 700 nM T98933 C60ECM 44186605 IC50 = 400 nM T98933 CM83FC 44186606 IC50 = 2900 nM T98933 CG2R8S 44186607 IC50 = 800 nM T98933 CM1UB2 44186608 IC50 = 4700 nM T98933 CWM3R1 44186609 IC50 = 600 nM T98933 CG2CH3 44186610 IC50 = 6500 nM T98933 CZQ2R1 44186611 IC50 = 18900 nM T98933 CFL30A 44186612 IC50 = 1500 nM T98933 C47SCQ 44186613 IC50 = 800 nM T98933 CZ7NW3 44186644 IC50 = 1500 nM T98933 CL52WN 44186645 IC50 = 700 nM T98933 CA5G8T 44186646 IC50 = 800 nM T98933 CEFM37 44186647 IC50 = 900 nM T98933 CK7N3X 44186648 IC50 = 1700 nM T98933 CE3JB8 44186649 IC50 = 600 nM T98933 CU7SG1 44186650 IC50 = 800 nM T98933 CI15SG 44186651 IC50 = 600 nM T98933 CY7VW4 44186652 IC50 = 3600 nM T98933 C0Q9AK 44186653 IC50 = 800 nM T98933 C0UL7Z 44186654 IC50 = 1200 nM T98933 C2ZF4S 44186655 IC50 = 1000 nM T98933 CKX1Q9 44186656 IC50 = 2100 nM T98933 C29QCE 44186657 IC50 = 900 nM T98933 CZQ7K2 44186691 IC50 = 800 nM T98933 CM80OW 44186692 IC50 = 700 nM T98933 C7OMH6 44186693 IC50 = 800 nM T98933 CQN2T6 44186694 IC50 = 3500 nM T98933 C0F2ZJ 44186695 IC50 = 5400 nM T98933 C63VSR 44186696 IC50 = 1500 nM T98933 C25FXN 44186698 IC50 = 800 nM T98933 CS0PI6 44186699 IC50 = 2100 nM T98933 C9PL4W 44186700 IC50 = 1000 nM T98933 C2ZEL5 44186701 IC50 = 1100 nM T98933 CO8R6C 44186702 IC50 = 900 nM T98933 CD0NW3 44186703 IC50 = 1200 nM T98933 C89HNC 44186704 IC50 = 700 nM T98933 C8UD7E 44299535 Ki = 2 nM T98933 CWH5G9 44345925 IC50 = 151 nM T98933 CQVW76 44346052 IC50 = 54 nM T98933 C87MEG 44346063 IC50 = 19500 nM T98933 C06YNJ 44349518 Ki = 0.16 nM T98933 CYAM86 44349526 Ki = 10000 nM T98933 CGXM40 44349576 Ki = 0.28 nM T98933 C1SM6H 44349600 Ki = 0.31 nM T98933 COFE32 44349601 Ki = 0.23 nM T98933 CB1P0S 44396251 Ki = 1900 nM T98933 CHY1C3 44396271 Ki > 2250 nM T98933 C29MBI 44396272 Ki > 2250 nM T98933 C4TQ6N 44396282 Ki = 1500 nM T98933 CH2Y3L 44396283 Ki > 2250 nM T98933 CWZB52 44396284 Ki > 2250 nM T98933 CD80LM 44396296 Ki > 2250 nM T98933 C6SI5L 44396297 Ki > 2250 nM T98933 CR4H1E 44396316 Ki > 2250 nM T98933 C45LRH 44396317 Ki > 2250 nM T98933 CA8V4G 44396331 Ki > 2250 nM T98933 CA8OB7 44400181 IC50 = 600 nM T98933 C4G9CF 44403605 IC50 = 2140 nM T98933 CW6EH8 44403606 IC50 = 9 nM T98933 C0L3WU 44403607 IC50 = 545 nM T98933 COU4B6 44403627 IC50 = 7.2 nM T98933 CVH75N 44403628 IC50 = 29 nM T98933 CTQ48J 44403634 IC50 = 0.3 nM T98933 C3SZ4I 44408427 IC50 = 15 nM T98933 CDE12F 44408544 EC50 = 4.3 nM T98933 C3TAU6 44408607 IC50 = 51 nM T98933 CM27EY 44417461 IC50 = 190 nM T98933 CC9BF0 44433089 IC50 = 26 nM T98933 C8QD9O 44434596 IC50 = 1.023 nM T98933 CLXF30 44434604 IC50 = 4.169 nM T98933 CP7C9J 44435761 IC50 = 100000 nM T98933 CWG53Q 44435778 IC50 = 33900 nM T98933 CH56GJ 44435779 IC50 = 43500 nM T98933 CB1UR7 44435786 IC50 = 69100 nM T98933 CL3FT4 44445692 IC50 = 3.467 nM T98933 C20LCQ 44445716 IC50 = 776.25 nM T98933 C1EGS9 44445719 IC50 = 190.55 nM T98933 CHT8I1 44445726 IC50 = 8.511 nM T98933 C9U7HY 44445727 IC50 = 870 nM T98933 C31JKD 44445730 IC50 = 9.55 nM T98933 C0NH4Z 44445731 IC50 = 239.88 nM T98933 CEX30A 44452442 EC50 = 58 nM T98933 CD38FN 44567764 EC50 = 70 nM T98933 CV1W9E 44589465 Ki = 31.3 nM T98933 C9K7HA 45270610 IC50 > 50000 nM T98933 CM7BY6 53385590 IC50 = 13000 nM T98933 C6Z7WI 60204885 EC50 = 550 nM T98933 C05ZRG 69428069 Ki = 14.1 nM T98933 CR2M8J 69844039 Ki = 31.7 nM T98933 C5SRF8 70681735 Ki = 20.3 nM T98933 C3A0DO 70682526 IC50 = 7400 nM T98933 CLJU20 70682537 IC50 = 2100 nM T98933 C2SVR8 70682538 IC50 = 2400 nM T98933 CBVQ29 70683842 Ki = 1.54 nM T98933 CVON79 70683843 Ki = 301 nM T98933 C9R0NB 70683844 Ki = 213 nM T98933 CG40IU 70684617 IC50 = 1700 nM T98933 CO1MQ8 70684618 IC50 = 2800 nM T98933 CU5VH3 70684619 IC50 = 8500 nM T98933 CARO49 70685018 Ki > 2250 nM T98933 CVK46F 70686763 IC50 = 8200 nM T98933 CWJ6U3 70686764 IC50 = 660 nM T98933 C70SIB 70688836 IC50 = 4200 nM T98933 CLF25D 70690926 IC50 = 5200 nM T98933 CB3ZC2 70690927 IC50 = 3400 nM T98933 C6FA0H 70690939 IC50 = 1400 nM T98933 C90XVL 70693065 IC50 = 1300 nM T98933 CC2EK8 70693080 IC50 = 1800 nM T98933 C2WC4V 70695111 IC50 = 7100 nM T98933 C92QMH 70695112 IC50 = 3300 nM T98933 CMNE57 70695113 IC50 = 310 nM T98933 CTQ37A 70697163 IC50 = 1600 nM T98933 CLU28H 71461159 EC50 = 0.47 nM T98933 CL8K9N 71523879 Ki = 1662 nM T98933 CQ0C5S 71523924 Ki = 441 nM T98933 C8DI5U 71523925 Ki = 124 nM T98933 CTU1K7 71523963 Ki = 223 nM T98933 CGHD73 71570928 IC50 = 16000 nM T98933 C49SBQ 71571065 IC50 = 5800 nM T98933 CE06XT 71571066 IC50 = 6600 nM T98933 CR92GT 71571067 IC50 = 3600 nM T98933 CTUC72 71571068 IC50 = 10600 nM T98933 C7UHM3 71571069 IC50 > 60000 nM T98933 C1P5HY 71571070 IC50 > 60000 nM T98933 C4CNP2 71571213 IC50 > 60000 nM T98933 CAV18D 71571215 IC50 > 60000 nM T98933 C97ISQ 71571216 IC50 = 20000 nM T98933 C5ZT9O 71716541 IC50 > 60000 nM T98933 C1TN8C 71716542 IC50 > 60000 nM T98933 CPJ4T2 71716543 IC50 > 60000 nM T98933 CP9B4C 71716544 IC50 > 60000 nM T98933 C4OE3H 71716545 IC50 > 60000 nM T98933 CIJ84X 71716546 IC50 = 59000 nM T98933 C4XL7Z 71716547 IC50 > 60000 nM T98933 C7BMG8 71716548 IC50 > 60000 nM T98933 C8O2NJ 71716549 IC50 > 60000 nM T98933 CA1Q0X 71716550 IC50 > 60000 nM T98933 CM6ZN5 71716551 IC50 > 60000 nM T98933 CX6RH7 71716552 IC50 > 60000 nM T98933 CTI7H2 71716553 IC50 > 60000 nM T98933 C8YEZ6 71716554 IC50 > 60000 nM T98933 CT3D1M 71717145 IC50 = 39000 nM T98933 CSHP85 71717146 IC50 > 60000 nM T98933 C5K3QG 71717147 IC50 > 60000 nM T98933 C6B5DO 71717148 IC50 > 60000 nM T98933 CK0ZQ9 71717149 IC50 > 60000 nM T98933 C96GSC 71717150 IC50 > 60000 nM T98933 C36SFW 71717155 IC50 > 60000 nM T98933 CLR58A 71717156 IC50 > 60000 nM T98933 CN4A9V 71717771 IC50 > 60000 nM T98933 CPLW58 71717772 IC50 > 60000 nM T98933 CIL03B 71717773 IC50 > 60000 nM T98933 C63QLG 71717774 IC50 = 38000 nM T98933 CV0I1H 71717775 IC50 > 60000 nM T98933 CUN4O0 71717776 IC50 > 60000 nM T98933 CSO2X5 71717777 IC50 > 60000 nM T98933 C52BZC 71717778 IC50 > 60000 nM T98933 CIE8V5 71717779 IC50 > 60000 nM T98933 C46ICD 71717780 IC50 > 60000 nM T98933 CPH02C 71718378 IC50 = 46000 nM T98933 COX71E 71718379 IC50 > 60000 nM T98933 CC94QZ 71718380 IC50 > 60000 nM T98933 CG2TH9 71718381 IC50 > 60000 nM T98933 C6G4BT 71718382 IC50 = 50000 nM T98933 CQ8AI1 71718383 IC50 > 60000 nM T98933 C4KOT9 71718386 IC50 > 60000 nM T98933 CH2TV1 71718387 IC50 > 60000 nM T98933 CXO1S7 71718388 IC50 > 60000 nM T98933 CI6AN0 71718985 IC50 = 24000 nM T98933 C5U7IR 71718986 IC50 > 60000 nM T98933 C0CJ8S 71718987 IC50 > 60000 nM T98933 C4KAZ7 71718988 IC50 > 60000 nM T98933 CIN3V1 71718992 IC50 > 60000 nM T98933 CZ3WG5 71718993 IC50 > 60000 nM T98933 CE6X2K 71718994 IC50 > 60000 nM T98933 C1IH2Q 71718995 IC50 > 60000 nM T98933 CN1RW4 71718996 IC50 > 60000 nM T98933 CKA36P 71718997 IC50 > 60000 nM T98933 C8LWP5 71719585 IC50 > 60000 nM T98933 CQ6BL0 71719586 IC50 > 60000 nM T98933 CFO1J2 71719587 IC50 > 60000 nM T98933 CT0DH9 71719588 IC50 > 60000 nM T98933 C3BT7V 71719589 IC50 > 60000 nM T98933 CBY36L 71719590 IC50 > 60000 nM T98933 C5SPB2 71719591 IC50 > 60000 nM T98933 CYNI30 71719592 IC50 > 60000 nM T98933 CJ5O6Q 71719593 IC50 > 60000 nM T98933 C7EKV1 71719594 IC50 > 60000 nM T98933 CB7O4D 71719597 IC50 > 60000 nM T98933 CD98PS 71719598 IC50 > 60000 nM T98933 CQ7U4O 71719599 IC50 > 60000 nM T98933 CXDE81 71719600 IC50 > 60000 nM T98933 CDM58X 71719601 IC50 > 60000 nM T98933 CCV8I1 71719602 IC50 > 60000 nM T98933 CH1EB5 71719603 IC50 > 60000 nM T98933 CX46KH 71719604 IC50 > 60000 nM T98933 C7KER0 71720182 IC50 > 60000 nM T98933 C0DYJ3 71720183 IC50 = 31000 nM T98933 CY4J2C 71720184 IC50 > 60000 nM T98933 C4Z0VS 71720185 IC50 > 60000 nM T98933 C5H0WP 71720186 IC50 > 60000 nM T98933 C9B4SP 71720187 IC50 > 60000 nM T98933 CHFZ51 71720188 IC50 > 60000 nM T98933 C2FM0U 71720189 IC50 > 60000 nM T98933 CUG52N 71720190 IC50 > 60000 nM T98933 CV1US9 71720192 IC50 > 60000 nM T98933 C7X8QB 71720193 IC50 > 60000 nM T98933 CB56IU 71720826 IC50 > 60000 nM T98933 CS5R7G 71720827 IC50 > 60000 nM T98933 CTF8D3 71720828 IC50 > 60000 nM T98933 CZ71PL 71720830 IC50 > 60000 nM T98933 C0Y9CT 71720831 IC50 > 60000 nM T98933 C5NU0T 71721539 IC50 > 100000 nM T98933 CP0G7O 73054742 EC50 = 150 nM T98933 CBJ8C9 73055020 EC50 = 37 nM T98933 CCO4X8 73055021 EC50 = 37 nM T98933 CZ8RJ5 73055022 EC50 = 62 nM T98933 C36LIJ 73055023 IC50 = 1100 nM T98933 C25DRF 73055024 IC50 = 1500 nM T98933 CANR79 76324858 IC50 = 24100 nM T98933 C4BA8W 90656430 IC50 > 69000 nM T98933 CO3KL0 118726602 Ki = 1.04 nM T98933 C45QSH 118726603 Ki = 1.12 nM T98933 CWQE31 118726604 Ki = 0.38 nM T98933 CZOI45 118726605 Ki = 0.26 nM T98933 C1QZ8J 118726606 Ki = 0.07 nM T98933 C0A9JB 118726607 Ki = 0.14 nM T98933 C94RVF 118726608 Ki = 0.04 nM T98933 C8IDF7 118726609 Ki = 0.18 nM T98933 C4KY2I 118726610 Ki = 0.09 nM T98933 CEW5K8 118726611 Ki = 0.3 nM T98933 CM2R8J 118726612 Ki = 0.54 nM T98933 CZM9O6 118726613 Ki = 0.64 nM T98933 CK8RB5 118726614 Ki = 1.11 nM T98933 CJA6K2 118726615 Ki = 3.14 nM T98933 C2J8PF 118726616 Ki = 8.04 nM T98933 CH1FA8 135528521 IC50 = 22 nM T98933 C0FWQ7 135559141 IC50 = 138.04 nM T98933 CU20KW 135559142 IC50 = 123.03 nM T98933 CW9R4B 135559143 IC50 = 28.18 nM T98933 CCF02H 145964530 IC50 = 7600 nM T98933 C56SHA 145964597 IC50 = 8800 nM T98933 C5H8EZ 145965425 IC50 = 970 nM T98933 C98CHS 145977976 IC50 = 9800 nM T98933 D01HAZ 23635364 IC50 = 4200 nM T98933 D01NTN 11350323 IC50 = 360 nM T98933 D01WVE 9872203 IC50 = 4100 nM T98933 D02CGG 44435789 IC50 = 8200 nM T98933 D03VOM 3092218 IC50 = 4300 nM T98933 D03XCG 23635367 IC50 = 15200 nM T98933 D05FRX 11153607 IC50 = 800 nM T98933 D05XMM 44186304 IC50 = 8100 nM T98933 D05ZJC 9925361 IC50 = 1905.46 nM T98933 D06IJW 23635362 IC50 = 2700 nM T98933 D07MAF 21653696 IC50 = 9600 nM T98933 D08BQI 11291923 IC50 = 5700 nM T98933 D09XOC 23635858 IC50 = 3000 nM T98933 D0A5XG 10027822 IC50 = 370 nM T98933 D0G7HF 23635860 IC50 = 19100 nM T98933 D0H6BV 24843916 IC50 = 4100 nM T98933 D0I2GK 71212 EC50 = 3.5 nM T98933 D0I7DH 23635476 IC50 = 7600 nM T98933 D0J0MD 23635730 IC50 = 17900 nM T98933 D0Q9ZN 23648092 IC50 = 230 nM T98933 D0U0GY 44435784 IC50 = 10500 nM T98933 D0U9JC 44435785 IC50 = 11400 nM T98933 D0YU9Z 14899645 IC50 = 18600 nM T98933 D0ZX0Y 23635856 IC50 = 6200 nM T39996 D02HFD 124886 IC50 > 100000 nM T39996 D07BDD 65359 IC50 > 100000 nM T39996 D0V0LB 6058 IC50 > 100000 nM T39996 D0X5SD 3117 IC50 = 1600 nM T39996 D0B1FE 3194 IC50 = 730 nM T39996 D09YFD 21928 IC50 = 1100 nM T39996 D0X2AU 23427 IC50 = 4900 nM T39996 CF3N7H 5941 IC50 > 100000 nM T39996 C8IWZ0 10236 IC50 > 100000 nM T39996 CGJ83B 15460 IC50 = 860 nM T39996 CX1LG8 65093 IC50 = 2700 nM T39996 C95WZA 123446 IC50 = 1500 nM T39996 CJ7FR6 533728 IC50 = 81000 nM T39996 C37UOC 590397 IC50 = 1000 nM T39996 CQE8T5 5462814 IC50 = 1700 nM T39996 C85NAQ 24858111 IC50 = 65000 nM T39996 C5N3LG 44251522 IC50 = 58 nM T39996 CCI45D 44604812 IC50 = 4 nM T39996 CFU9H7 44605025 IC50 = 12 nM T39996 CL76QF 44605026 IC50 = 13 nM T39996 CFQ17S 44605027 IC50 = 23 nM T39996 C6PY2V 44605028 IC50 = 11 nM T39996 CZF8V7 46174173 IC50 = 100 nM T39996 C70VHB 53315882 IC50 < 15 nM T39996 C7M0FJ 59457983 IC50 = 600000 nM T39996 CAVD69 70678415 IC50 = 25000 nM T39996 C52YJT 76310995 IC50 = 100000 nM T39996 CNQ86R 76314627 IC50 = 500000 nM T39996 CYB1U4 76318201 IC50 = 100000 nM T39996 CZ09ML 76321898 IC50 = 400000 nM T39996 C4XJ5N 78357767 IC50 > 100000 nM T39996 CCT09O 86288827 IC50 = 87000 nM T39996 C01DAP 86288828 IC50 = 1500 nM T39996 CA18TS 90655765 IC50 = 235000 nM T39996 C5NX4U 90655766 IC50 = 147000 nM T39996 C9BI8F 118607414 IC50 = 180 nM T39996 C7X2AQ 118613624 IC50 > 20000 nM T39996 C7TI9A 129012136 IC50 = 5 nM T39996 C6F2VK 129012137 IC50 = 4 nM T39996 CJI14M 129072680 IC50 > 20000 nM T39996 COL81P 129085358 IC50 > 20000 nM T39996 CTQE45 132471834 IC50 = 18 nM T39996 CBO31X 132471835 IC50 = 6 nM T39996 CL2ZI0 132609264 IC50 = 794300 nM T39996 CYJR92 132609265 IC50 = 21800 nM T39996 CBTH20 137348638 IC50 = 7 nM T39996 CR53YC 137631913 IC50 = 6 nM T39996 C8VT5L 137632046 IC50 = 203700 nM T39996 C8VO5D 137632076 IC50 = 44 nM T39996 C5AC6M 137632524 IC50 = 20 nM T39996 C46WLE 137633319 IC50 > 5000 nM T39996 CIB30Q 137633627 IC50 = 34 nM T39996 C8AM9L 137635489 IC50 = 808 nM T39996 CE60DR 137635748 IC50 = 12 nM T39996 CTU4G0 137636690 IC50 = 20 nM T39996 CI5Q3X 137636915 IC50 = 26 nM T39996 CK1WU6 137637870 IC50 = 28 nM T39996 C3TD2E 137638286 IC50 = 15 nM T39996 CO6JA8 137639333 IC50 > 5000 nM T39996 CO78IY 137639766 IC50 = 73 nM T39996 C0EYN9 137639969 IC50 = 20 nM T39996 CCSI40 137640754 IC50 = 17 nM T39996 C2P3JR 137640823 IC50 = 47700 nM T39996 C5TY4L 137640829 IC50 = 159 nM T39996 C7G9AB 137643064 IC50 = 46 nM T39996 CV4PI3 137643498 IC50 > 6000 nM T39996 C2DWX9 137643972 IC50 = 95100 nM T39996 CZM39K 137644029 IC50 = 1230 nM T39996 CS9RO5 137644870 IC50 = 11 nM T39996 C6NW5B 137645215 IC50 = 59 nM T39996 C6WLD1 137645686 IC50 = 11 nM T39996 CZTV84 137646234 IC50 = 18 nM T39996 C9EP0L 137647456 IC50 = 58 nM T39996 CN5UY2 137647689 IC50 > 1000 nM T39996 CD2JQ9 137648196 IC50 = 77 nM T39996 C7Y2RH 137648735 IC50 = 115000 nM T39996 CJO19V 137649514 IC50 = 135 nM T39996 CZD47A 137649599 IC50 = 35 nM T39996 CZR86C 137650174 IC50 = 24 nM T39996 CUM43J 137650973 IC50 = 145800 nM T39996 CSU4J8 137651295 IC50 = 97 nM T39996 CJ57XR 137652778 IC50 = 29 nM T39996 C8N2BU 137653025 IC50 = 12 nM T39996 C4JYZ0 137654123 IC50 = 341 nM T39996 CES2Y4 137654330 IC50 = 50 nM T39996 CF65YG 137654447 IC50 = 18 nM T39996 CX2RM3 137654889 IC50 = 43 nM T39996 C8MQ2I 137655652 IC50 = 24 nM T39996 C3BI4K 137655660 IC50 = 35 nM T39996 CHS71L 137656981 IC50 = 23 nM T39996 CYF6V9 137657228 IC50 = 27 nM T39996 C0R6QN 137658284 IC50 = 63 nM T39996 CR7GF2 137658708 IC50 = 16 nM T39996 CDQW60 137661215 IC50 > 5000 nM T39996 C19VQE 137661488 IC50 = 36 nM T39996 CD1K7J 137661663 IC50 = 28 nM T39996 C85XIG 137662224 IC50 = 30 nM T39996 C8LEV4 139267760 IC50 > 10000 nM T39996 CJT6G1 155511077 IC50 = 19 nM T39996 C4NS2X 155512777 IC50 = 18500 nM T39996 CO5P4T 155513225 IC50 = 41 nM T39996 CDWR24 155515450 IC50 = 10300 nM T39996 C04DFY 155516671 IC50 = 1460 nM T39996 CB9WP0 155517958 IC50 = 179 nM T39996 CFLK08 155520544 IC50 = 300 nM T39996 CYOD10 155522526 IC50 = 1080 nM T39996 CJOW75 155522891 IC50 = 19 nM T39996 CL4T2Q 155523641 IC50 = 280 nM T39996 CCI9U8 155524518 IC50 = 926 nM T39996 C4UXQ1 155526805 IC50 = 3090 nM T39996 CLQ18S 155527069 IC50 = 4090 nM T39996 CP60DZ 155527429 IC50 = 698 nM T39996 CG2EM1 155527465 IC50 = 53600 nM T39996 CH5X4E 155527661 IC50 = 16 nM T39996 CD8C5B 155528012 IC50 = 44 nM T39996 CKN4C6 155528155 IC50 = 9 nM T39996 C53YIH 155530887 IC50 = 12 nM T39996 CA9P6Y 155532307 IC50 = 9 nM T39996 C1J5TI 155532811 IC50 = 2860 nM T39996 CI0ML6 155534407 IC50 = 1350 nM T39996 C6FEP9 155535898 IC50 = 679 nM T39996 CU2XG3 155537180 IC50 = 953 nM T39996 C7Q9HD 155537279 IC50 = 47 nM T39996 C6R7JS 155537616 IC50 = 78 nM T39996 C78EAT 155538085 IC50 = 70 nM T39996 C5NH2I 155540357 IC50 = 1950 nM T39996 C9H4GL 155540760 IC50 = 205 nM T39996 C5OGN0 155542626 IC50 = 642 nM T39996 CHL9F7 155543202 IC50 = 1550 nM T39996 CT3M4J 155543558 IC50 = 1250 nM T39996 CQ20HW 155544061 IC50 = 3470 nM T39996 C0VJO4 155545582 IC50 = 2470 nM T39996 C2I8ES 155546390 IC50 = 529 nM T39996 CBLI45 155547053 IC50 = 2650 nM T39996 C51VKD 155547438 IC50 = 12 nM T39996 C8RD2L 155548665 IC50 = 4670 nM T39996 C8Q3GX 155550036 IC50 = 885 nM T39996 CSKE02 155550699 IC50 = 1310 nM T39996 C1QOP9 155550708 IC50 = 11 nM T39996 CS1TK5 155551475 IC50 = 2360 nM T39996 CJAT69 155553711 IC50 = 3990 nM T39996 CTIM98 155556005 IC50 = 27 nM T39996 CV9EZ2 155556376 IC50 = 2010 nM T39996 CVT50L 155557402 IC50 = 35 nM T39996 CYAP13 155557747 IC50 = 122 nM T39996 C5KZP1 155558337 IC50 = 19 nM T39996 CQ08KG 155559900 IC50 = 94 nM T39996 C2FIO6 155559947 IC50 = 2230 nM T39996 CD3HO4 155562561 IC50 = 7510 nM T39996 C0J6AT 155562781 IC50 = 152 nM T39996 C91BWQ 155564365 IC50 = 2380 nM T39996 C5VN8K 155564441 IC50 = 647 nM T39996 CVZ2C4 155565339 IC50 = 150 nM T39996 C84AKC 155566143 IC50 = 6 nM T39996 D00FLT 65482 IC50 = 100 nM T39996 D02UVS 5455 IC50 = 1100 nM T39996 D06PPL 25150857 IC50 = 700 nM T39996 D09CLP 439155 IC50 = 230 nM T39996 D0BI4T 53315878 IC50 < 2.5 nM T39996 D0C5EG 76285486 IC50 = 11 nM T39996 D0CX4W 46901937 IC50 = 15 nM T39996 D0DQ6Z 8530 IC50 = 14000 nM T39996 D0GK7A 46224516 IC50 = 19 nM T39996 D0L5LN 6780 IC50 > 100000 nM T39996 D0RO9T 73755260 IC50 = 1600 nM T54128 D00ENY 33032 IC50 = 613 nM T54128 D02VKC 3272524 Ki = 70 nM T54128 D0B0NQ 127894 IC50 = 1350 nM T54128 D02QZL 9903685 IC50 = 80 nM T54128 D06WHL 135484540 IC50 = 700 nM T54128 D0H1FV 68736 IC50 = 967 nM T54128 CO3XI2 125406 IC50 = 88000 nM T54128 C6RD3L 125407 IC50 = 12000 nM T54128 C32DCS 3018579 IC50 = 6700 nM T54128 C5OHM8 3481675 IC50 = 30 nM T54128 CRL5Z4 5353536 IC50 = 340 nM T54128 CS5V4U 5486548 Ki = 135 nM T54128 CB50FH 6604872 IC50 = 3000 nM T54128 C20IEF 9837860 IC50 = 5700 nM T54128 CW79HF 9909062 Ki = 215 nM T54128 C4SG1T 9927756 Ki = 600 nM T54128 CI7GM6 9937279 Ki = 7 nM T54128 CHIL12 9985663 Ki = 4 nM T54128 CPF74Y 10017901 IC50 = 153 nM T54128 CM5I3E 10036285 IC50 = 24000 nM T54128 C4LWR8 10037930 IC50 = 7000 nM T54128 CB8KW6 10048025 IC50 = 340 nM T54128 C76YSF 10051732 Ki = 15 nM T54128 C5G2WD 10084218 IC50 = 84500 nM T54128 C6XJD8 10244065 IC50 = 8000 nM T54128 C5NOI8 10244106 IC50 > 100000 nM T54128 C0AC4T 10247474 Ki = 180 nM T54128 C8THG7 10266209 IC50 = 166 nM T54128 C70WBQ 10401891 IC50 = 44000 nM T54128 CX1V3L 10437436 Ki = 5 nM T54128 C5M4IH 10538709 IC50 > 100000 nM T54128 CYX93H 10562939 IC50 = 94 nM T54128 C7WKJ2 10610792 IC50 > 100000 nM T54128 C6A1UE 10656900 IC50 > 100000 nM T54128 C0O6ZI 10658567 IC50 = 54000 nM T54128 C9BV5R 10729534 IC50 = 5800 nM T54128 CIW54Y 10752476 IC50 = 1500 nM T54128 C9H0TI 10800053 IC50 = 72000 nM T54128 C3B9HI 10823814 IC50 = 48000 nM T54128 C02QUD 10824747 IC50 = 700 nM T54128 CXLW54 11948707 Ki > 10000 nM T54128 CJZ6K9 15337998 Ki = 1500 nM T54128 CZ8BM3 15840183 Ki = 450 nM T54128 CT4ZO6 15840184 Ki = 54 nM T54128 C06MHR 15840185 Ki = 4 nM T54128 C3A5ES 15840186 Ki = 4 nM T54128 C1QA4W 15840187 Ki = 20 nM T54128 CT1I3Y 21710164 Ki = 10000 nM T54128 CB9E5R 21710166 Ki = 980 nM T54128 CL3UT2 22097086 Ki = 3000 nM T54128 CLRK62 22097088 Ki = 70 nM T54128 CJ52FG 22097105 Ki = 400 nM T54128 C4J3TO 22097119 Ki = 78 nM T54128 CD7H5E 22097148 Ki = 20000 nM T54128 C62FHX 22097151 Ki = 2000 nM T54128 CR5BZ4 22097158 Ki > 25000 nM T54128 CE20FP 22097165 Ki = 210 nM T54128 C3BKT5 22097178 Ki = 76 nM T54128 C72VRZ 22097186 Ki > 25000 nM T54128 CVD94P 22097194 Ki = 250 nM T54128 C9EO8L 22097211 Ki > 25000 nM T54128 C2H4CP 22100063 Ki = 95 nM T54128 C76PHV 22100072 Ki = 110 nM T54128 CM2H1L 22100104 Ki = 2000 nM T54128 CCMS36 22100119 Ki = 49 nM T54128 C1DMH8 22100133 Ki = 5 nM T54128 CJ8UB0 22100152 Ki = 840 nM T54128 CLX8S4 22100157 Ki = 71 nM T54128 CIG65E 22449297 Ki = 22 nM T54128 CM2AN8 44268202 Ki = 250 nM T54128 C5ES0F 44268209 Ki = 880 nM T54128 C9WG8T 44268224 Ki = 280 nM T54128 CG09WU 44268242 Ki = 500 nM T54128 CL0H9R 44268310 Ki = 3000 nM T54128 CJUL-93 44268318 Ki = 650 nM T54128 C49GIP 44268353 Ki = 140 nM T54128 C8V4DX 44268357 Ki = 890 nM T54128 CMC3B8 44268369 Ki > 25000 nM T54128 CRUJ15 44281577 IC50 = 1350 nM T54128 C4ZX5R 44281591 IC50 = 630 nM T54128 CT1X5A 44281631 IC50 = 580 nM T54128 C8GQ4A 44304811 IC50 = 1350 nM T54128 CWAX82 44317999 Ki = 60 nM T54128 C9J4ME 44348419 IC50 = 4300 nM T54128 C1JRT2 44377742 IC50 = 21000 nM T54128 C3YN8I 44377743 IC50 = 36000 nM T54128 C6PYE7 44379376 IC50 = 14000 nM T54128 CGX3P0 44460610 Ki = 66 nM T54128 CDI84E 71450922 IC50 > 10000 nM T54128 CDA4O8 135407136 IC50 = 2100 nM T54128 C0TK2B 135453826 IC50 = 1900 nM T54128 C4E0VH 135484474 IC50 = 150 nM T54128 C1ET2K 135535891 IC50 = 1800 nM T54128 CR45DZ 135976300 IC50 = 7200 nM T54128 CP9TR0 10324985 Ki > 10000 nM T54128 D03RGP 1221 IC50 = 23 nM T54128 D04DHB 1779 IC50 > 100000 nM T54128 D05KQC 3899541 IC50 = 200 nM T54128 D0J3EZ 4038142 IC50 = 2000 nM T54128 D0S6TW 1845 IC50 = 27000 nM T82739 D05PHH 3447 IC50 = 1350 nM T82739 D0I0RJ 16231 IC50 > 50000 nM T82739 D0ID3W 9911502 IC50 = 15800 nM T82739 D0PK7J 56599309 Ki = 2.4 nM T82739 D0D5RH 11641515 IC50 = 12000 nM T82739 D0N7WR 108040 Ki = 570 nM T82739 C1BHS3 193409 Ki = 22500 nM T82739 CR4KE5 445844 Ki = 800 nM T82739 C87OTC 447733 Ki = 7170 nM T82739 CF6D4B 447734 Ki = 2720 nM T82739 CHT05K 447735 Ki = 436 nM T82739 CCKZ79 668744 IC50 = 30100 nM T82739 C53FNM 674593 IC50 = 11900 nM T82739 C45NBS 674629 IC50 = 4400 nM T82739 C21HDC 674632 IC50 = 11300 nM T82739 CBX3U0 674652 IC50 = 6600 nM T82739 C98EGA 741761 IC50 > 50000 nM T82739 CFD4M6 747662 IC50 > 50000 nM T82739 C9D4IN 754821 IC50 > 50000 nM T82739 C0ER8S 767161 IC50 = 60500 nM T82739 CLR3H1 899247 IC50 = 42200 nM T82739 CQ2R0M 1011274 IC50 = 28100 nM T82739 C7P1UO 1201257 IC50 = 31700 nM T82739 C2PRY6 1269450 IC50 = 67400 nM T82739 CO4AB7 2264784 IC50 = 5500 nM T82739 CTE79D 3011892 Ki > 50000 nM T82739 CU43OY 3088969 Ki > 50000 nM T82739 C0K7TF 3123858 IC50 > 50000 nM T82739 C8KD9E 3162843 IC50 > 50000 nM T82739 CQY92E 3660962 IC50 = 7200 nM T82739 CQWL43 5039074 IC50 = 35400 nM T82739 CLD0C6 5348879 IC50 = 96200 nM T82739 C1B9GP 5400404 IC50 > 50000 nM T82739 CF1P5H 5430316 IC50 = 54200 nM T82739 CZ1XU5 5876194 IC50 = 13500 nM T82739 CG2A7X 7028541 IC50 = 120100 nM T82739 C6JDM9 9799627 Ki = 145 nM T82739 C2F5NS 9884570 Ki = 110 nM T82739 CKDP84 9895193 Ki = 7200 nM T82739 C0LKE7 9912771 Ki = 11000 nM T82739 CC0D5H 9915041 Ki = 58 nM T82739 CH8QJ4 9916876 IC50 = 14 nM T82739 CF9SD1 9917846 IC50 = 29 nM T82739 C8F5CW 9937921 Ki = 61 nM T82739 CNE34O 9939021 IC50 = 120 nM T82739 CX85LD 9954980 Ki > 16000 nM T82739 CM7IF6 9956559 Ki > 20000 nM T82739 CBC2K3 9959749 IC50 = 130 nM T82739 CA9S3O 9981709 IC50 = 41000 nM T82739 C7BD9S 10024676 IC50 = 19000 nM T82739 C7LZ2T 10050676 IC50 = 25000 nM T82739 CQP65H 10095093 Ki = 19000 nM T82739 C3OG5U 10095865 IC50 = 5010 nM T82739 C1VT4F 10117027 Ki = 3000 nM T82739 C31QAL 10143532 Ki > 2300 nM T82739 C5I0YH 10168444 Ki = 17000 nM T82739 CSVF04 10253001 IC50 = 28000 nM T82739 CQ9ZO1 10275412 Ki = 8900 nM T82739 CP64HV 10342843 Ki > 1000000 nM T82739 CK9J7X 10343728 IC50 = 25100 nM T82739 C6JF0P 10365153 IC50 = 35000 nM T82739 C10ISY 10367012 Ki = 5000 nM T82739 C57GFJ 10386993 IC50 = 16000 nM T82739 C6S4CO 10391715 Ki = 14000 nM T82739 CT75ZJ 10411941 IC50 = 16000 nM T82739 CBV6N7 10423722 IC50 > 50000 nM T82739 CJTH60 10432907 Ki = 3330 nM T82739 C6AZ8B 10435038 Ki = 8600 nM T82739 CISN08 10455169 IC50 = 54000 nM T82739 C6KJM2 10461790 Ki > 50000 nM T82739 CV0X6G 10480463 IC50 = 560 nM T82739 CEI65Z 10483775 Ki = 4.6 nM T82739 C5ED3G 10529121 Ki = 79000 nM T82739 CU8N3V 10578280 Ki = 7300 nM T82739 C8SUZ9 10624948 Ki = 12000 nM T82739 CEJ14F 10624997 Ki = 3300 nM T82739 CR5EX8 10648196 Ki = 7600 nM T82739 CPWH69 10648370 Ki = 35000 nM T82739 CJG9H6 10669349 Ki = 586000 nM T82739 C5VB1U 10695159 Ki = 18000 nM T82739 CP4QC5 10696511 Ki = 775000 nM T82739 CGYR23 10696955 Ki = 15000 nM T82739 CPGV87 10718240 Ki = 36000 nM T82739 CIKF89 10719580 Ki = 170000 nM T82739 CZ0Q8K 10742217 Ki = 816000 nM T82739 C7RWD8 10744643 Ki = 399000 nM T82739 CKOQ35 10767421 Ki = 29000 nM T82739 C3IN8W 10815545 Ki = 27000 nM T82739 CVQE76 10816339 Ki = 58000 nM T82739 CLB15C 10871563 Ki = 4800 nM T82739 C2TBO9 10959252 Ki = 600 nM T82739 CAD15G 11149953 Ki = 8000 nM T82739 C6LVG4 11186243 Ki = 2570 nM T82739 CTX9F3 11188793 Ki = 1350 nM T82739 CLA93S 11237163 Ki = 8458 nM T82739 CHLK70 11244460 Ki = 2430 nM T82739 C86DZB 11292119 Ki = 230 nM T82739 C6CDN3 11347670 Ki = 18100 nM T82739 CLY5G8 11350400 Ki = 849 nM T82739 CR8NW9 11351302 Ki > 10000 nM T82739 CTJ1Z2 11361949 Ki = 400 nM T82739 C63LIR 11473486 Ki = 1370 nM T82739 CK34OX 11509611 Ki = 330 nM T82739 CO68MA 11524737 Ki = 940 nM T82739 CJP9O1 11684611 Ki = 5 nM T82739 CQ5U8H 11739438 Ki = 112 nM T82739 C7WJP0 11754749 IC50 = 26000 nM T82739 C7JLR1 11774107 Ki = 4300 nM T82739 CNO67W 11798089 Ki = 14000 nM T82739 CYX74A 11824584 Ki = 1300 nM T82739 C2QO1B 15955412 Ki > 50000 nM T82739 C19ARJ 15984063 Ki = 43000 nM T82739 C53YRO 16098910 IC50 = 10 nM T82739 CN6CJ2 16220264 IC50 = 1340 nM T82739 CJSL38 18727836 IC50 = 300 nM T82739 CRX19I 23646295 Ki > 2300 nM T82739 CKH4O5 24180463 Ki > 6000 nM T82739 C7WTO3 24689997 IC50 = 8600 nM T82739 CTE3P4 24692287 IC50 = 20600 nM T82739 CJUE04 24860432 IC50 > 50000 nM T82739 C0UA9T 24860449 IC50 > 50000 nM T82739 C52CJA 24860451 IC50 > 50000 nM T82739 CZI85G 24984725 Ki = 0.1 nM T82739 CN0ZW3 24999867 Ki > 1000 nM T82739 CEM32W 25001205 Ki > 1000 nM T82739 C4Q9XM 25166807 Ki = 130 nM T82739 CX6A4M 25166808 Ki = 170 nM T82739 C2H4PJ 25166809 Ki = 122 nM T82739 CF1I6Q 25166810 Ki = 270 nM T82739 C9W0GO 25167018 Ki = 120 nM T82739 CHB21I 44265055 IC50 = 12000 nM T82739 CNK8W1 44310877 IC50 = 710 nM T82739 C8KOM9 44333945 Ki = 15500 nM T82739 CH32DA 44333955 Ki = 28 nM T82739 C75KOP 44333957 Ki = 500 nM T82739 C7A6KF 44333986 Ki = 4 nM T82739 CF1LQ4 44333999 Ki = 89 nM T82739 CZ7RK3 44334001 Ki = 5 nM T82739 CUO4N2 44334160 Ki = 2 nM T82739 CRT4G3 44335601 Ki = 22000 nM T82739 C7Z9WL 44335624 Ki = 97000 nM T82739 CAY34C 44347478 Ki > 1000000 nM T82739 CT0QN1 44347480 Ki = 476000 nM T82739 C1UN9I 44347534 Ki = 767000 nM T82739 C0V2FL 44347624 Ki = 1000000 nM T82739 CZ8XL6 44385679 IC50 = 210 nM T82739 CL5BA4 44385729 IC50 = 640 nM T82739 C3D2CL 44385935 IC50 = 500 nM T82739 CW08OY 44385998 IC50 = 790 nM T82739 CV6KG4 44386059 IC50 = 380 nM T82739 C5MR1F 44386934 IC50 = 500 nM T82739 C78QJO 44394249 Ki > 50000 nM T82739 CQRB69 44394250 Ki > 50000 nM T82739 CTS5W9 44404049 IC50 > 400000 nM T82739 C3BX5Y 44412781 Ki = 83000 nM T82739 CIP7E1 44415075 IC50 = 46200 nM T82739 C0THI1 44415189 IC50 = 75000 nM T82739 CVO5Q1 44432538 Ki > 10000 nM T82739 CR16BF 44434808 Ki > 10800 nM T82739 CQIX73 44434809 Ki > 6000 nM T82739 COG34X 44434818 Ki > 6000 nM T82739 C9T1DP 44434835 Ki > 10800 nM T82739 CB86HU 44453827 IC50 = 13 nM T82739 CVZW52 44537923 IC50 = 19000 nM T82739 COX6G5 52943174 IC50 = 1.7 nM T82739 CDH59M 52944043 IC50 = 2000 nM T82739 C8VI6M 52944358 IC50 = 39.1 nM T82739 CNA7U8 52946795 IC50 = 1500 nM T82739 C0T3CX 52948030 IC50 > 10000 nM T82739 CA6GQ5 53341037 Ki = 70 nM T82739 CIKQ81 53345652 Ki = 1.5 nM T82739 CXWS90 53345968 Ki = 0.3 nM T82739 C76GSI 53346181 Ki = 7.5 nM T82739 CV60BK 53488415 Ki = 6218 nM T82739 CI2ND0 54741583 Ki = 28 nM T82739 C17MSO 56640092 Ki = 136 nM T82739 CGP7Y6 56640160 Ki = 25.3 nM T82739 C30AJK 56640226 Ki = 19 nM T82739 CH1EI8 56954620 Ki = 25.4 nM T82739 C4EHU8 56954732 Ki = 868 nM T82739 C5C8XO 56954733 Ki = 493 nM T82739 CST4F0 56954834 Ki = 17.4 nM T82739 CRK92A 56954952 Ki = 10.1 nM T82739 CLY4C9 57390236 IC50 = 910000 nM T82739 CPBW48 57392333 Ki = 2000000 nM T82739 CEO1L3 57393799 IC50 = 380000 nM T82739 CL2JE5 57395841 Ki = 3300000 nM T82739 CXZ3D0 57400764 IC50 = 680000 nM T82739 CMG29L 57404341 IC50 = 1700 nM T82739 CXGW36 57404342 IC50 = 300 nM T82739 CTE30K 57842560 Ki > 6000 nM T82739 C0C6UB 57842624 Ki = 3600 nM T82739 C7XY5A 57842673 Ki > 6000 nM T82739 C41NSR 57842812 Ki = 50 nM T82739 C9XW1C 57842830 Ki > 10000 nM T82739 CWF0C3 57842850 Ki = 4600 nM T82739 C73CPB 57842913 Ki = 1700 nM T82739 C60HCV 57976401 Ki = 519 nM T82739 CHB27Y 57976410 Ki = 1850 nM T82739 CM8UJ7 57976444 Ki = 41 nM T82739 CQ71KE 57976446 Ki = 240 nM T82739 CSC0L5 59020200 Ki > 11000 nM T82739 CPW2H7 59315536 Ki > 10000 nM T82739 CL42XV 59401924 Ki = 350 nM T82739 CHJI56 59401943 Ki = 24 nM T82739 CA76HG 59401978 Ki = 340 nM T82739 CO38AC 59402011 Ki = 110 nM T82739 CVG75I 59402039 Ki = 23 nM T82739 CF26ZO 59402046 Ki > 6000 nM T82739 C7IWJ3 59402077 Ki = 20 nM T82739 CTW85S 59402125 Ki = 240 nM T82739 CKX9B7 59402220 Ki = 46 nM T82739 CZD0N4 59402226 Ki > 6000 nM T82739 CK7I1A 59402239 Ki = 210 nM T82739 C6JP8Q 60154989 Ki = 2 nM T82739 CE5A7B 60162406 Ki = 320 nM T82739 C3LT2W 66674079 Ki = 3820 nM T82739 CYH7X1 66674212 Ki = 3440 nM T82739 C3ND0L 66674351 Ki = 2217 nM T82739 C5N1GU 66674475 Ki = 4500 nM T82739 C23QOJ 66674821 Ki = 1924 nM T82739 CWOD93 66744646 Ki = 16 nM T82739 CKWQ82 67155200 Ki = 2900 nM T82739 C0SDB3 68020667 Ki = 392 nM T82739 C17JAZ 68284084 IC50 > 30000 nM T82739 C6AU1R 70252985 Ki = 268 nM T82739 CTO5I6 70253788 Ki = 1370 nM T82739 C8A7ZJ 70306716 Ki = 0.019 nM T82739 C1A2FN 70681010 IC50 = 13500 nM T82739 CHC3B5 70683145 IC50 = 12900 nM T82739 CM5BH2 70683146 IC50 = 3800 nM T82739 C4IFW3 70683249 Ki = 0.075 nM T82739 CN38UY 70687492 Ki = 9.4 nM T82739 C3Z7RM 70695744 IC50 = 7800 nM T82739 CC2Q7G 70695750 IC50 = 10600 nM T82739 CJPF90 71548883 Ki = 310 nM T82739 C30ZKJ 71561420 Ki = 1000 nM T82739 CH32TL 71561557 Ki = 187 nM T82739 C8RW7E 71562631 Ki = 3.2 nM T82739 C4UHB2 71562760 Ki = 118 nM T82739 C0EM6D 71562761 Ki = 24 nM T82739 CNS21T 71562882 Ki = 240 nM T82739 C3SBE2 71562883 Ki = 422 nM T82739 C2NY0B 71563006 Ki = 500 nM T82739 CG46AZ 71563007 Ki = 242 nM T82739 C2O4SB 71563124 Ki = 440 nM T82739 C4CT8O 71563125 Ki = 116 nM T82739 C78DJQ 71711730 IC50 < 10000 nM T82739 CS2CR9 71716063 IC50 = 20 nM T82739 C45APQ 71716064 IC50 = 30 nM T82739 C64YFO 71716065 IC50 = 50 nM T82739 CD53RA 71716975 Ki = 0.3 nM T82739 CSP5T2 71716976 Ki > 120000 nM T82739 CAR2J6 71717264 IC50 = 28.6 nM T82739 CWJ75U 71717265 IC50 = 30 nM T82739 C7JDE3 71719101 IC50 = 800 nM T82739 CQ3K2V 71719191 Ki = 12.9 nM T82739 C1Y0JV 71719710 IC50 = 21.2 nM T82739 C24UEO 71720319 IC50 = 1800 nM T82739 CVCM38 71818688 IC50 = 11200 nM T82739 CLI36U 72551247 Ki = 520 nM T82739 C01LOR 73051877 Ki = 3 nM T82739 C6M9ZP 73052197 Ki = 9 nM T82739 CXJ86Q 73052510 Ki = 1 nM T82739 CB14LR 73052831 Ki = 2.39 nM T82739 CU9C2F 73345352 IC50 = 7181 nM T82739 CDQP51 73347119 Ki > 50000 nM T82739 CM3PH8 73350210 Ki > 50000 nM T82739 C9ASZ2 86302628 IC50 > 1000000 nM T82739 CMD5V7 86583041 Ki = 24 nM T82739 CO6U9I 88582319 Ki > 6000 nM T82739 C9A7YX 90655485 IC50 > 1000000 nM T82739 C90UNY 90655486 IC50 = 740000 nM T82739 C75WHK 90655487 IC50 > 1000000 nM T82739 CZ1Q2P 90655488 IC50 > 1000000 nM T82739 CSG0L5 90655489 IC50 > 1000000 nM T82739 C8KX5F 90655490 IC50 > 1000000 nM T82739 C9W1CO 90655491 IC50 > 1000000 nM T82739 C5WIF7 90655492 IC50 > 1000000 nM T82739 C6FE2K 90655493 IC50 > 1000000 nM T82739 C2I7SQ 90655494 IC50 > 1000000 nM T82739 CXY0I6 90655495 IC50 > 1000000 nM T82739 CWL8U1 90655496 IC50 > 1000000 nM T82739 CRQ6I4 90655497 IC50 > 1000000 nM T82739 CL27GQ 90655498 IC50 > 1000000 nM T82739 CLG8M0 90655499 IC50 > 1000000 nM T82739 CBK7Y9 90655500 IC50 > 1000000 nM T82739 CD7WM6 90655501 IC50 > 1000000 nM T82739 CJ7B8Y 90655502 IC50 > 1000000 nM T82739 CW6VS9 90655503 IC50 > 1000000 nM T82739 CV1NM4 90655504 IC50 > 1000000 nM T82739 CKPN23 90655505 IC50 > 1000000 nM T82739 CZ8S4C 90655506 IC50 > 1000000 nM T82739 C65TLW 101862198 Ki > 1000000 nM T82739 CI4KC5 117986603 IC50 = 7.2 nM T82739 C3MVG0 118720988 Ki = 1360 nM T82739 C9M2IH 118720990 Ki = 1170 nM T82739 C1E6GW 118720991 Ki = 1470 nM T82739 C9BVI5 118720993 Ki = 5540 nM T82739 C1FQZ6 118720994 Ki = 60 nM T82739 C0WZA2 118720996 Ki = 220 nM T82739 CE89KB 118720997 Ki = 5270 nM T82739 CIAL50 118720998 Ki = 765 nM T82739 C4HLM3 118720999 Ki = 1310 nM T82739 CLD6I3 118721000 Ki = 910 nM T82739 C0XG7H 118721001 Ki = 920 nM T82739 CZC53M 118721002 Ki = 1902 nM T82739 C8FZ2L 118721003 Ki = 45 nM T82739 C0M4IQ 118721004 Ki = 20 nM T82739 CLRB29 118721005 Ki = 8 nM T82739 C9B1FX 118721007 Ki = 50 nM T82739 CRV5Y1 118721008 Ki = 5 nM T82739 CH6AQ9 118721009 Ki = 2 nM T82739 CHQ5P7 118987013 Ki = 42 nM T82739 C2V6PQ 122550396 IC50 = 8.5 nM T82739 C8NR0Y 122550417 IC50 = 0.7 nM T82739 C3W6DG 122551266 IC50 = 1.7 nM T82739 C5Y8IS 127025168 Ki = 7.5 nM T82739 CY03UC 127027302 Ki = 804 nM T82739 C18GDE 127027303 Ki = 317 nM T82739 CK0W2P 127027635 Ki = 59 nM T82739 CWJ0Y6 127027636 Ki = 55 nM T82739 C36DML 127029802 Ki = 150 nM T82739 CLJ40K 127029803 Ki = 120 nM T82739 CPC0M8 127031390 Ki = 550 nM T82739 C1BWV2 127035672 Ki = 22 nM T82739 CTMR64 127035685 Ki = 64 nM T82739 CVRY56 127036086 Ki = 8 nM T82739 C9B6LT 127037264 Ki = 9.93 nM T82739 C60HLK 127037469 Ki = 136 nM T82739 C85ROH 127041472 IC50 > 100000 nM T82739 CSB70O 129103433 IC50 = 4 nM T82739 C1QNA4 129103439 IC50 = 19 nM T82739 C82CEQ 129103576 IC50 = 900 nM T82739 CWXN62 129103630 IC50 = 9 nM T82739 CE2NT3 134130030 IC50 > 3000000 nM T82739 CT2RV6 134130781 IC50 = 2.4 nM T82739 CO13UB 134131040 IC50 = 1570 nM T82739 CWV3G6 134131077 IC50 = 153 nM T82739 CS8FV1 134131084 IC50 = 42.3 nM T82739 C1L3XV 134131107 IC50 = 8310 nM T82739 C92RTL 134131303 IC50 = 4.8 nM T82739 CSV13U 134131383 IC50 = 1210 nM T82739 CQOA40 134131498 IC50 = 53200 nM T82739 CL37SG 134131589 IC50 = 2 nM T82739 C6HTD5 135393470 IC50 = 11300 nM T82739 C7NA6E 135393474 IC50 > 50000 nM T82739 C4M5BF 135450980 Ki = 1300 nM T82739 CX62AU 135453491 Ki = 12 nM T82739 CYJ02B 135530536 Ki = 13 nM T82739 C8XC5J 135530568 Ki = 6 nM T82739 CBA90J 135532848 Ki = 4 nM T82739 CR6B1G 135532849 Ki = 6 nM T82739 CZHK63 135532851 Ki = 3 nM T82739 COA5Z0 135532896 Ki = 0.5 nM T82739 CW6DR2 135543006 Ki = 10 nM T82739 CTM4S0 135559104 Ki = 8 nM T82739 C3N1HW 135559111 Ki = 3 nM T82739 CYD5H1 135559116 Ki = 6 nM T82739 CD8XW3 135559124 Ki = 18 nM T82739 CZQ79E 135559125 Ki = 37 nM T82739 C90YUE 135559128 Ki = 65 nM T82739 C5DQ1E 135559129 Ki = 27 nM T82739 C4CMO6 136003658 Ki = 36 nM T82739 CM1LF3 136094796 Ki = 5 nM T82739 C1GPL0 136402490 Ki = 4820 nM T82739 CDQ62V 137637214 Ki = 3 nM T82739 C2K8JV 137639385 Ki = 0.25 nM T82739 C7EJ6B 137642984 Ki = 1.3 nM T82739 CG67RS 137643031 Ki = 0.06 nM T82739 CODW67 137644829 Ki = 45100 nM T82739 C83GDO 137646822 Ki = 0.44 nM T82739 C5SQZ6 137649699 Ki = 2.3 nM T82739 CCMQ19 137651042 Ki = 0.07 nM T82739 CN4ZT0 137651057 Ki = 0.39 nM T82739 C4M6NX 137651852 Ki = 0.21 nM T82739 CNX46H 137654508 Ki = 0.36 nM T82739 CMK09U 137655401 Ki = 0.15 nM T82739 CLQ5X7 137657674 Ki = 2.1 nM T82739 C8R7WM 137661862 Ki = 0.14 nM T82739 CUZ35A 138115400 IC50 = 6309.57 nM T82739 CO51HN 139030452 IC50 > 50000 nM T82739 CV86MX 145962597 IC50 = 1 nM T82739 C51YBM 145963085 IC50 = 1900 nM T82739 CE6C0A 145970642 Ki = 192 nM T82739 CZ1R3B 145982984 Ki = 0.02 nM T82739 C4HLX8 146029523 IC50 = 16700 nM T82739 CH59QO 155510375 Ki = 43190 nM T82739 CICU31 155511394 Ki = 277 nM T82739 CZR36C 155511554 IC50 = 79.43 nM T82739 CA81QV 155512709 Ki = 6380 nM T82739 C2VX3G 155512946 Ki = 6.3 nM T82739 C2CI8S 155513907 Ki = 2205 nM T82739 CYT20V 155514020 Ki > 50000 nM T82739 CAT98N 155514640 Ki > 10000 nM T82739 CG9H4N 155515624 Ki = 9090 nM T82739 C7ZM4R 155515728 Ki = 7405 nM T82739 CFRS54 155516565 Ki = 10390 nM T82739 C1ZSV0 155517054 Ki = 12550 nM T82739 CF96DM 155518671 Ki > 10000 nM T82739 C6NX4K 155519661 IC50 = 10 nM T82739 C4MS1B 155519676 IC50 = 794.33 nM T82739 C7DUX3 155520916 Ki > 10000 nM T82739 CH0N9A 155523885 Ki = 319 nM T82739 CYL8M0 155526377 Ki = 4640 nM T82739 CX7CO2 155527010 Ki = 600 nM T82739 CN3BH5 155527998 IC50 = 79.43 nM T82739 CHYW65 155528639 IC50 = 199.53 nM T82739 CI1FR2 155529536 Ki = 0.6 nM T82739 CD7O2G 155530095 IC50 = 794.33 nM T82739 C46AZL 155530642 Ki > 25000 nM T82739 C35QWO 155531023 IC50 = 398.11 nM T82739 CP8K2J 155531811 Ki = 10470 nM T82739 C0UR8Q 155531991 Ki = 12000 nM T82739 CIHM01 155535907 Ki > 100000 nM T82739 C12HON 155536142 IC50 = 199.53 nM T82739 C7JMK4 155538439 Ki = 800 nM T82739 C9QE5N 155538514 Ki = 3865 nM T82739 CRT3D4 155540148 Ki = 7245 nM T82739 CL90DN 155540666 Ki > 10000 nM T82739 CY6DK3 155540964 IC50 = 5.012 nM T82739 C4CHR9 155542229 Ki = 7920 nM T82739 C4P2GV 155543617 Ki > 25000 nM T82739 CU52QS 155545897 Ki > 10000 nM T82739 CH2S6R 155546346 Ki > 10000 nM T82739 C5MB9R 155547962 IC50 = 50.12 nM T82739 CLFB25 155548371 IC50 = 794.33 nM T82739 CSI5J1 155548907 Ki = 7270 nM T82739 CU9FL4 155551858 Ki > 50000 nM T82739 COM52R 155551892 IC50 = 79.43 nM T82739 CA5VG2 155552651 Ki = 24500 nM T82739 C5S6HO 155553129 Ki = 6950 nM T82739 CJ3FI5 155553630 IC50 = 1258.93 nM T82739 C5TV4J 155554082 Ki = 8246 nM T82739 CU8LR3 155555208 Ki > 25000 nM T82739 CSW48V 155557718 IC50 = 19.95 nM T82739 CXL5D4 155558368 Ki = 48690 nM T82739 CNZ1K5 155559920 Ki > 10000 nM T82739 C3SXY1 155561904 Ki = 64397 nM T82739 CX5O7K 155562968 Ki = 540 nM T82739 CM8XB1 155565537 IC50 = 100 nM T82739 CP4F1U 155567613 Ki = 32000 nM T82739 CEZ8B9 155568406 Ki > 50000 nM T82739 CK0EA2 155568484 Ki = 701 nM T82739 CL2S7B 90655701 Ki = 320000 nM T82739 D02AVL 18376720 Ki = 45 nM T82739 D02PAU 16731825 Ki = 1000 nM T82739 D02YIW 1794 IC50 > 50000 nM T82739 D05ZIP 674656 IC50 = 6200 nM T82739 D07ZRG 46899577 Ki = 8.3 nM T82739 D08KCA 72429 IC50 = 40000 nM T82739 D08OCS 699665 IC50 = 6100 nM T82739 D08WQJ 700133 IC50 = 18800 nM T82739 D0A8WP 447732 Ki = 2500 nM T82739 D0IU5E 716930 IC50 = 12300 nM T82739 D0J5VK 67145 IC50 = 67900 nM T82739 D0JU9N 6914623 Ki > 2800 nM T82739 D0K7YL 447476 Ki = 1.9 nM T82739 D0M4VZ 10456438 IC50 = 31 nM T82739 D0ON2Z 204102 Ki > 2300 nM T82739 D0R9CH 3400921 Ki = 37 nM T82739 D0X1OY 674628 IC50 = 5700 nM T82739 D0Y5IQ 44255320 IC50 = 10000 nM T45593 D05YBZ 7083 Ki = 69 nM T45593 D05TPI 72276 IC50 >= 200000 nM T45593 D07SDQ 969516 IC50 = 3500 nM T45593 D0U2BH 65064 IC50 = 1800 nM T45593 C2KJI7 3883 Ki = 2.5 nM T45593 C0VAW3 13735 IC50 = 69 nM T45593 CYX3S5 65043 IC50 = 69 nM T45593 C39BCE 68275 IC50 < 3000 nM T45593 CO41FC 964143 Ki = 789.8 nM T45593 CJ0O1B 1588443 IC50 = 380 nM T45593 CO1ZV8 2306524 Ki = 522.1 nM T45593 CY28LS 5293755 Ki = 617.6 nM T45593 C5ZS3K 5713403 Ki = 528.5 nM T45593 CZ9Q1O 5928757 Ki = 362.5 nM T45593 CQ3S8L 6450842 Ki = 261.5 nM T45593 CFXW58 11631766 Ki = 1410 nM T45593 C7EBU1 11776207 IC50 > 10000 nM T45593 CLV24A 14214498 IC50 = 1400 nM T45593 C62KEJ 14837578 IC50 = 710 nM T45593 CN0Y8F 15504852 IC50 = 13 nM T45593 CN9U3G 16049314 IC50 = 246 nM T45593 CWUS28 22361008 IC50 > 10000 nM T45593 CCL0P8 24858429 IC50 = 1635 nM T45593 CYDL23 24952085 IC50 = 440 nM T45593 C1RB4M 24966387 IC50 = 1200 nM T45593 C0BN8L 42643531 IC50 = 4 nM T45593 CD80XQ 54581735 IC50 = 80 nM T45593 C4FZ5A 56950118 Ki = 13 nM T45593 C90MUF 57176479 Ki = 599 nM T45593 C2K6JT 57379031 EC50 = 24 nM T45593 CTA24H 57578199 IC50 = 1700 nM T45593 CC8ZH7 58660303 IC50 > 10000 nM T45593 CU1D5F 58795397 Ki = 797.8 nM T45593 CQU9W0 66556402 Ki = 191.3 nM T45593 CJ4R7E 66571561 IC50 = 660 nM T45593 CAJ6B8 67973277 EC50 = 325 nM T45593 C2ZCF9 67973354 EC50 = 169 nM T45593 C9JMF7 68551830 IC50 = 910 nM T45593 CXS67Z 68552247 IC50 = 580 nM T45593 CWE58F 68553100 IC50 = 690 nM T45593 CH54DU 68553676 IC50 = 600 nM T45593 CY8HE3 68553756 IC50 = 420 nM T45593 C1LYJ4 68553873 IC50 > 10000 nM T45593 CAG5N8 68554590 IC50 = 2000 nM T45593 CSQ53N 68555084 IC50 = 520 nM T45593 CEI5O1 68555350 IC50 = 320 nM T45593 CNCS47 68556083 IC50 = 1400 nM T45593 CN2QL6 68556085 IC50 = 920 nM T45593 CR4VM9 70686684 Ki = 1428 nM T45593 CD1PU4 70688786 Ki = 17 nM T45593 C59PES 70694381 Ki = 0.48 nM T45593 CZ3QF7 70697093 Ki = 112 nM T45593 CW0ZX3 71452100 IC50 = 2 nM T45593 CUP70I 71453931 IC50 = 1251 nM T45593 C7EX1K 71457447 IC50 = 17 nM T45593 CM5E3R 71457448 IC50 = 2 nM T45593 C3GPE7 71457449 IC50 = 4707 nM T45593 C7XML1 71457851 IC50 = 5.1 nM T45593 C4AK0O 71459256 IC50 = 42 nM T45593 CQ0FG2 71459258 IC50 = 7469 nM T45593 CYN3M8 71461086 IC50 = 1591 nM T45593 CW1E7U 71462763 IC50 = 6 nM T45593 CM6R2W 71463212 IC50 = 1.41 nM T45593 CLVB69 73294880 IC50 = 13 nM T45593 CGZK85 73296378 IC50 = 2 nM T45593 C9L3VR 73296809 IC50 = 2 nM T45593 C2S9PZ 73296810 IC50 = 5 nM T45593 C4XR1C 73297137 IC50 = 1 nM T45593 CCPI94 73297139 IC50 = 3 nM T45593 CE9X5J 86713212 IC50 = 420 nM T45593 C45CME 89681657 IC50 > 10000 nM T45593 C3R4PD 89970609 IC50 = 330 nM T45593 C06FNJ 89970660 IC50 = 610 nM T45593 CE1IW4 89970765 IC50 = 700 nM T45593 CEF8J5 90040128 IC50 = 5 nM T45593 CD48HU 90277509 IC50 > 10000 nM T45593 CX28SL 90644922 IC50 = 2 nM T45593 CHD0Z7 90644923 IC50 = 79 nM T45593 CYPJ75 90644924 IC50 = 8 nM T45593 CTL20G 102196384 IC50 > 10000 nM T45593 C5PBW3 102398558 IC50 > 10000 nM T45593 C5W7PM 118713185 IC50 > 10000 nM T45593 CQ07AH 118713186 IC50 > 10000 nM T45593 C5OFH2 118713187 IC50 > 10000 nM T45593 C9ZGB4 118713188 IC50 > 10000 nM T45593 C7Z2GA 118713189 IC50 > 10000 nM T45593 C03URO 118713190 IC50 > 10000 nM T45593 CYK30H 118713191 IC50 > 10000 nM T45593 CK53ME 118713192 IC50 > 10000 nM T45593 C35IDH 118713193 IC50 < 290 nM T45593 CM7UC8 118713194 IC50 > 10000 nM T45593 C5C8LX 118713195 IC50 = 300 nM T45593 C1RH3Y 118713196 IC50 = 1600 nM T45593 CB03DR 122182244 Ki = 212.4 nM T45593 CI6WT0 122182245 Ki = 431.7 nM T45593 C3X5KJ 122182246 Ki = 364 nM T45593 CT5G1Q 122182247 Ki = 1116.2 nM T45593 CCT7H6 122182248 Ki = 858.8 nM T45593 CML3T5 122182249 Ki = 853.5 nM T45593 CMO1C3 122182250 Ki = 169 nM T45593 CIT52U 122182251 Ki = 53.7 nM T45593 C19GJH 122182252 Ki = 35.1 nM T45593 CUOB01 122182253 Ki = 48 nM T45593 CW2V5B 122182254 Ki = 682.4 nM T45593 C75OCP 122182255 Ki = 717.6 nM T45593 CVH2T0 122182256 Ki = 229.1 nM T45593 CKQF12 122182257 Ki = 374 nM T45593 C7AUF8 122182258 Ki = 239.7 nM T45593 C7BXY4 122182259 Ki = 90 nM T45593 CCEL74 122182260 Ki = 188 nM T45593 C32GEV 122182261 Ki = 263.2 nM T45593 CWIT38 122182262 Ki = 257 nM T45593 CMVS36 122182263 Ki = 204.3 nM T45593 CLW95X 122182264 Ki = 131.1 nM T45593 C4TNB1 122182265 Ki = 465.1 nM T45593 CQ4R0K 122182266 Ki = 38.3 nM T45593 C5C8FY 122182267 Ki = 1756.7 nM T45593 C7NV9G 122182268 Ki = 27.1 nM T45593 CU3NJ6 122182269 Ki = 208.7 nM T45593 CS84HC 122182270 Ki = 121.5 nM T45593 C8EYO3 122182271 Ki = 590.5 nM T45593 CFV32E 122182272 Ki = 72.4 nM T45593 C1LHQ2 122182273 Ki = 318.1 nM T45593 C24PHB 122182274 Ki = 228.6 nM T45593 C1U3FZ 122182275 Ki = 354.6 nM T45593 CX5NB4 122182276 Ki = 151.7 nM T45593 CAU9H6 122182277 Ki = 630.3 nM T45593 C2RB1F 122182278 Ki = 80.1 nM T45593 CTMV35 122182279 Ki = 455.7 nM T45593 CO54NG 134133007 IC50 = 230 nM T45593 C4G8CN 136259624 IC50 = 970 nM T45593 C0PX2K 145968691 IC50 = 12900 nM T45593 C4R3UA 145978145 IC50 = 27200 nM T45593 CYB0T8 155552280 Ki = 120 nM T45593 D05CCT 4139 EC50 = 130 nM T45593 D0O5FK 10171487 IC50 = 3255 nM T45593 D0T3PW 5281672 IC50 = 1200 nM T45593 D0Z7EL 5280647 IC50 < 3000 nM T62292 D07JVL 3016 Ki = 17 nM T62292 D0L9GG 2118 EC50 = 69 nM T62292 D0T1WN 5732 Ki = 400 nM T62292 D0CH7C 57336276 Ki = 489 nM T62292 D0HO2T 23581869 Ki = 1.3 nM T62292 D0Z9HW 23630026 Ki = 3.1 nM T62292 C4PAD5 5255267 Ki = 858 nM T62292 C1Z6YU 9821389 Ki = 12 nM T62292 CCX58U 9865233 Ki = 1.8 nM T62292 C7BA0Z 9908880 Ki = 0.7 nM T62292 C1VRB9 9951530 EC50 = 23 nM T62292 CPC3U1 9971547 Ki > 300 nM T62292 CUT5W8 9976743 EC50 = 33 nM T62292 CUSM85 10221761 Ki = 0.5 nM T62292 C15NXT 10926766 EC50 = 3826 nM T62292 CK1S7J 10927005 EC50 = 367 nM T62292 CWK02D 10936672 EC50 = 424 nM T62292 C09PCZ 10971225 EC50 = 500 nM T62292 C74SOK 11001453 EC50 = 935 nM T62292 CJB1V2 11035207 EC50 = 394 nM T62292 CBV36I 11047145 EC50 = 213 nM T62292 C8B7TF 11067772 EC50 = 116 nM T62292 CAU9O6 11142977 EC50 = 117 nM T62292 CWO70Q 11673720 Ki = 14 nM T62292 CX7G9K 11759134 EC50 = 344 nM T62292 CL4XD0 11783674 EC50 = 20 nM T62292 CYD2G3 11809547 EC50 = 71 nM T62292 C1ZXE0 15951053 Ki = 8545 nM T62292 C6HY4N 21065276 Ki = 272 nM T62292 C5R3SB 21930923 Ki = 96 nM T62292 CPM7G9 25093403 Ki = 2666 nM T62292 C8E3KW 25093404 Ki = 1864 nM T62292 CZK75V 44364548 EC50 = 425 nM T62292 C0FN6W 44364725 EC50 = 375 nM T62292 CE8F3Y 44364734 EC50 = 265 nM T62292 COH5G6 44364735 EC50 = 119 nM T62292 C2VHW7 44364747 EC50 = 148 nM T62292 CZL2P0 44364907 EC50 = 65 nM T62292 CCX08E 44364918 EC50 = 242 nM T62292 C6AO8S 44561476 Ki = 255 nM T62292 CLQZ42 44561477 Ki = 198 nM T62292 C27YZH 88286432 Ki = 1000 nM T62292 CQ91VU 118278442 Ki = 24 nM T62292 CH0D4J 130439777 Ki = 660 nM T62292 C56XBU 130439778 Ki = 63000 nM T62292 C9N8LW 130439889 Ki = 480 nM T62292 D06SOQ 6918451 Ki = 0.61 nM T62292 D09IHE 6918583 Ki = 0.77 nM T62292 D0D9RF 9927764 Ki = 18.7 nM T62292 D0E7PY 11624499 Ki = 80 nM T62292 D0GQ2G 5311418 Ki = 25.8 nM T62292 D0O9MG 5311203 Ki = 17 nM T21782 D06RGG 5819 IC50 > 50000 nM T21782 D0S6JG 5920 IC50 = 3600 nM T21782 D0J6XC 5803 IC50 = 25000 nM T21782 D0WM6E 160565 IC50 = 32000 nM T21782 CLSK17 5804 IC50 = 17000 nM T21782 CPR38J 92859 IC50 = 6300 nM T21782 C2VED9 107564 IC50 > 50000 nM T21782 CHM8L9 71185084 IC50 = 1200 nM T21782 CTN04E 71185155 IC50 = 9700 nM T21782 CU8KD9 71185156 IC50 = 1200 nM T21782 CB49TE 71185169 IC50 = 1000 nM T21782 CDLU47 71185374 IC50 = 1500 nM T21782 CB8R1S 71185474 IC50 = 6000 nM T21782 CP6Z7Y 71185477 IC50 = 1400 nM T21782 CNU60F 71185540 IC50 = 1000 nM T21782 CNR1C2 71487227 IC50 = 1900 nM T21782 CPM3Q9 71487297 IC50 = 2700 nM T21782 CD1T9B 71487299 IC50 = 2900 nM T21782 C2YMT4 71487301 IC50 = 3100 nM T21782 C06COQ 71487363 IC50 = 3700 nM T21782 CQV8L7 71487428 IC50 = 11000 nM T21782 CTB4V0 71583751 IC50 > 50000 nM T21782 C6UV0P 71583752 IC50 > 50000 nM T21782 C6E7DR 71583865 IC50 > 50000 nM T21782 C2CD7N 71583866 IC50 > 50000 nM T21782 CA2TH8 71583867 IC50 = 14000 nM T21782 CGX57L 71583868 IC50 = 8600 nM T21782 C76GXY 71583869 IC50 = 6500 nM T21782 CPI36K 71583870 IC50 = 2900 nM T21782 CH3J9Z 71583871 IC50 = 6000 nM T21782 CM4LY2 71583975 IC50 = 1300 nM T76369 D0E6YQ 1935 IC50 > 100000 nM T76369 D0NS6H 3152 IC50 > 100000 nM T76369 D0Y3KG 3121 Ki = 363000 nM T76369 D0B6IZ 137905 Ki = 2.1 nM T76369 D0W0VD 3885 Ki = 1220 nM T76369 D02UOE 160142 Ki = 2530 nM T76369 C13GAP 255 IC50 = 140 nM T76369 CXU4W0 650 Ki > 100000 nM T76369 C0RFA2 3102 Ki > 100000 nM T76369 C4IU5T 6889 Ki = 31700 nM T76369 C6B1HI 9905 IC50 = 4 nM T76369 C25CYL 10434 Ki > 100000 nM T76369 C47FYB 10662 Ki > 100000 nM T76369 CZP3G7 11100 Ki > 100000 nM T76369 COGY52 11321 Ki = 36000 nM T76369 C7U0TW 11747 Ki > 100000 nM T76369 C53FYO 11840 Ki > 100000 nM T76369 CKR3L9 12116 Ki > 100000 nM T76369 CU5KZ0 13005 Ki > 100000 nM T76369 CJ2GH1 13006 Ki > 100000 nM T76369 CG1LI5 14313 Ki > 100000 nM T76369 C4FW7E 18475 Ki > 100000 nM T76369 C7S3JO 26257 Ki = 3 nM T76369 C38JQX 31261 Ki > 100000 nM T76369 CN8A2G 38296 Ki > 100000 nM T76369 C7HE8W 38333 Ki > 100000 nM T76369 C0VK3I 39834 Ki > 100000 nM T76369 C8Z6TM 43402 Ki > 100000 nM T76369 CUNJ73 61209 Ki > 100000 nM T76369 C6U7FB 62539 Ki > 100000 nM T76369 CEKW96 68115 Ki = 125.89 nM T76369 CL5B7Z 68119 Ki = 1170 nM T76369 C27NHT 69147 Ki > 100000 nM T76369 CN0ID1 69282 Ki > 100000 nM T76369 CW54JA 69288 Ki > 100000 nM T76369 C6BEN0 70945 Ki > 100000 nM T76369 CV8R4B 76561 Ki > 100000 nM T76369 CVJ78Y 79690 Ki = 46.6 nM T76369 CAPG58 87502 Ki = 77.6 nM T76369 C0EH3Z 88695 Ki = 26900 nM T76369 C70KGR 92036 Ki = 3300 nM T76369 C13IQL 93772 Ki > 100000 nM T76369 C7JEN0 94320 IC50 = 49860 nM T76369 C8YU9Z 95415 Ki > 100000 nM T76369 CH91PI 95447 Ki > 100000 nM T76369 CO0QF3 97313 Ki = 942 nM T76369 C6L8SK 102135 IC50 = 22360 nM T76369 CR3E9L 103786 Ki > 100000 nM T76369 CFG6D1 111253 IC50 > 100000 nM T76369 C7KJ3B 114917 Ki = 26250 nM T76369 C20LIY 136371 Ki > 100000 nM T76369 CTU83D 137777 Ki = 22800 nM T76369 CHAN02 138508 Ki = 8060 nM T76369 CYX5V0 142278 Ki > 100000 nM T76369 C5X1YU 160254 Ki = 544 nM T76369 CXG41E 163959 Ki = 355000 nM T76369 C4IRY2 164676 Ki = 6890 nM T76369 CB9GM4 176443 IC50 = 2 nM T76369 CD35GB 181715 Ki = 707000 nM T76369 C6W8MB 219592 Ki > 100000 nM T76369 COQ09W 219605 Ki = 1550 nM T76369 C25BHS 222475 Ki > 100000 nM T76369 CN35KE 222570 Ki > 100000 nM T76369 C93DSW 222958 IC50 = 10 nM T76369 CP4W3S 229680 Ki = 3080 nM T76369 C2SQH9 232004 Ki > 100000 nM T76369 C0KV5M 236566 Ki > 100000 nM T76369 CE6U1D 237515 Ki = 4.8 nM T76369 C92OSL 241331 Ki = 53900 nM T76369 C1IW3D 261836 Ki > 100000 nM T76369 CHP1J7 262695 Ki > 100000 nM T76369 CDL3E1 262696 Ki > 100000 nM T76369 CPL6E4 272516 Ki = 32.1 nM T76369 CBV0N9 275005 Ki = 212 nM T76369 C18XWV 291540 Ki > 100000 nM T76369 CH52BM 306215 Ki > 100000 nM T76369 CKS3U9 366710 Ki = 34100 nM T76369 CKP61X 368568 Ki = 1054 nM T76369 CTWM69 586418 Ki > 100000 nM T76369 CH1E7N 590628 Ki > 100000 nM T76369 C4TE6S 597830 Ki > 100000 nM T76369 CCJQ96 599378 Ki = 170 nM T76369 COW64L 988563 Ki = 13700 nM T76369 C79KSZ 1009717 Ki > 100000 nM T76369 CAP82W 1103353 Ki > 100000 nM T76369 CB8I0Q 1133380 Ki > 100000 nM T76369 C21KSG 1137588 Ki > 100000 nM T76369 CF46TV 1167776 Ki > 100000 nM T76369 CN8BI5 1222869 Ki > 100000 nM T76369 CWTV42 1713189 Ki = 4350 nM T76369 C0EX9G 1755771 Ki = 66 nM T76369 CB0ZP3 1812008 Ki = 9800 nM T76369 C3FQD8 1906162 Ki > 100000 nM T76369 C3O6MN 1972026 Ki > 100000 nM T76369 CF37ZA 2147394 Ki = 610 nM T76369 CJD8B3 2305233 Ki = 2650 nM T76369 C0OZQ2 2731126 Ki > 100000 nM T76369 CNKV06 2731127 Ki = 1620 nM T76369 CEM2C8 2731732 Ki = 19500 nM T76369 C2HOC5 2731733 Ki = 1880 nM T76369 CVC36I 2731902 Ki = 1420 nM T76369 CG62CN 2731904 Ki = 36000 nM T76369 CVD82J 2734800 Ki = 1660 nM T76369 C9R5LQ 2749125 Ki = 2630 nM T76369 C84DSN 2749126 Ki = 107 nM T76369 C84VWR 2784639 Ki = 5380 nM T76369 CDCB42 2786143 Ki = 1540 nM T76369 C43YAR 2835143 Ki > 100000 nM T76369 C1AM0S 3114312 Ki = 1560 nM T76369 C61RSW 3126152 Ki > 100000 nM T76369 CCP07Y 3264931 Ki > 100000 nM T76369 CB21VL 3321360 Ki > 100000 nM T76369 CZV6G2 3329233 Ki > 100000 nM T76369 C6NH9P 3469206 Ki > 100000 nM T76369 C10GCK 3527426 Ki = 1690 nM T76369 C3T1CV 3531512 Ki > 100000 nM T76369 C5UM2D 3821945 Ki = 8 nM T76369 CU17BR 4088910 Ki > 100000 nM T76369 C8CFN7 4118889 Ki > 100000 nM T76369 CC1GF9 4338240 Ki = 580 nM T76369 C8KV7I 4350924 Ki > 100000 nM T76369 C0V6QI 4369935 Ki > 100000 nM T76369 C0GS5T 4381638 Ki > 100000 nM T76369 C42FGN 4384851 Ki = 7.5 nM T76369 CQ46SJ 4427802 Ki > 100000 nM T76369 CN9C3V 4513067 Ki = 55300 nM T76369 C5NJ3A 5004413 Ki > 100000 nM T76369 CNMY06 5038499 Ki > 100000 nM T76369 CWCG89 5080545 Ki > 100000 nM T76369 CK5XC9 5235003 Ki > 100000 nM T76369 CMJ30V 5353845 IC50 = 5000 nM T76369 CY6D5H 9821458 IC50 = 1000 nM T76369 CZ10UR 9905153 IC50 = 2000 nM T76369 CHT5U3 10044204 IC50 = 6000 nM T76369 CTZ42X 10337211 IC50 = 3470 nM T76369 CWE41Q 10655805 Ki = 6.65 nM T76369 CE64FC 10661387 Ki = 17.7 nM T76369 CF28NJ 10879668 Ki = 7.6 nM T76369 CH49NV 10899196 Ki = 102 nM T76369 CP93JE 10902085 Ki = 0.84 nM T76369 C7NZY9 11009341 Ki = 21000 nM T76369 C1P3HT 11226329 Ki > 100000 nM T76369 CC3D2X 11245953 Ki = 2.2 nM T76369 CYJ2M4 11278743 IC50 = 300 nM T76369 CSD58O 11280423 Ki = 7 nM T76369 C8GX1Y 11322015 Ki = 363.08 nM T76369 CI68UO 11393923 IC50 = 1000 nM T76369 C1JAC5 11425923 Ki = 398 nM T76369 CU94ZT 11484453 IC50 = 140 nM T76369 CG2B7X 11631387 IC50 = 30 nM T76369 C0QJ9O 11652690 IC50 = 30 nM T76369 C57KVO 11674428 IC50 = 10 nM T76369 CG7O5E 11695972 IC50 = 200 nM T76369 CV74JA 11696246 IC50 = 500 nM T76369 CAG6H2 11709766 IC50 = 250 nM T76369 CY58GA 11739291 IC50 = 200 nM T76369 CCQN45 11805526 Ki = 26 nM T76369 CMV1U9 11991810 IC50 = 7000 nM T76369 CVK4C5 11991896 IC50 = 200 nM T76369 CI9R2Y 11991988 IC50 = 100 nM T76369 CV2M3J 12057101 Ki = 0.302 nM T76369 CKG7A0 12222796 Ki > 100000 nM T76369 CJ65IL 12305517 IC50 = 10530 nM T76369 C8B5LO 13780062 Ki = 2.19 nM T76369 C3YOX2 13827082 Ki > 100000 nM T76369 C4CR1L 13827083 Ki > 100000 nM T76369 CH27JR 14609844 Ki = 0.328 nM T76369 CKX0P8 14610645 Ki = 1223 nM T76369 CA0E1T 14610646 Ki = 25.1 nM T76369 CI68WP 14707309 IC50 = 23610 nM T76369 CSI6M2 14828209 Ki = 131 nM T76369 CBA8U6 14856680 Ki = 23.8 nM T76369 CJ6H8G 14856681 Ki = 18.9 nM T76369 CL2C7Y 15044210 Ki = 870 nM T76369 C3UXC5 16084218 IC50 = 1960 nM T76369 C45MVX 16110641 IC50 > 100000 nM T76369 CC9N1G 16110651 IC50 = 500 nM T76369 CO94HF 16110652 IC50 = 400 nM T76369 CLC13N 16110653 IC50 = 200 nM T76369 COK20Z 16110654 IC50 = 600 nM T76369 C0H5RW 16110655 IC50 = 900 nM T76369 CS0VQ6 16110656 IC50 = 6000 nM T76369 COL87N 16110658 IC50 = 3000 nM T76369 C0KT5Q 16110666 IC50 = 30000 nM T76369 CVC17D 16110699 IC50 > 100000 nM T76369 C7O1KM 16110701 IC50 = 200 nM T76369 C97PDA 16110708 IC50 = 2000 nM T76369 C8P1JE 16110710 IC50 = 2000 nM T76369 CX3LI0 16110711 IC50 = 34000 nM T76369 C42XSZ 16110715 IC50 > 100000 nM T76369 CBH6F1 16110717 IC50 > 100000 nM T76369 CWV39U 16110722 IC50 = 8000 nM T76369 C5W1CT 16110723 IC50 = 30000 nM T76369 CPG32I 16307342 Ki > 100000 nM T76369 CXQO59 16324698 Ki > 100000 nM T76369 CX5UT9 16735161 IC50 = 200 nM T76369 C3KF9Y 16736226 IC50 = 2000 nM T76369 CR76ET 16737951 IC50 = 1200 nM T76369 C8G9AL 16756850 IC50 > 10000 nM T76369 CKX36J 17479504 Ki > 100000 nM T76369 CBG35K 17485200 Ki > 100000 nM T76369 C2OF8S 18471933 Ki > 100000 nM T76369 CG5DA4 22109309 Ki > 100000 nM T76369 C1IQ9L 22486206 IC50 = 5 nM T76369 CM3Y1I 22574246 Ki > 100000 nM T76369 CET65Y 22772978 Ki > 100000 nM T76369 C3F1EG 22772980 Ki > 100000 nM T76369 CKUJ63 22772981 Ki > 100000 nM T76369 C6WY3U 23669322 Ki > 100000 nM T76369 CX1G5Y 24319385 Ki > 100000 nM T76369 C0LP8T 24445964 Ki > 100000 nM T76369 CNF01W 24748349 IC50 = 70 nM T76369 CF9E1W 24748380 IC50 = 3000 nM T76369 COE7A6 24799115 IC50 > 100000 nM T76369 C3A6LN 24799306 IC50 = 7000 nM T76369 CMEC63 24799824 IC50 = 16 nM T76369 C59EGV 24799998 IC50 > 100000 nM T76369 C5V6OE 24800169 IC50 = 270 nM T76369 CU9Y3V 24800335 IC50 = 100 nM T76369 C5MK9H 24800509 IC50 = 17000 nM T76369 CSB1L8 24800681 IC50 > 100000 nM T76369 CLC63B 24800683 IC50 = 90000 nM T76369 CI67RX 24800861 IC50 = 2400 nM T76369 CT5C9E 24801041 IC50 = 37000 nM T76369 C0RT3I 24801044 IC50 = 26000 nM T76369 C8WGD9 24801560 IC50 = 26 nM T76369 CQNB75 24825630 Ki > 100000 nM T76369 C2EPR4 24948911 IC50 > 100000 nM T76369 C0MC4D 24948914 IC50 = 120 nM T76369 CSA71C 24949075 IC50 = 2000 nM T76369 CGK9I3 24949076 IC50 = 200 nM T76369 C79BEQ 24949227 IC50 = 12000 nM T76369 CGO7P4 24950363 IC50 > 100000 nM T76369 CS8H1V 24950364 IC50 = 8000 nM T76369 C90WNP 24950523 IC50 = 30000 nM T76369 C5O4JY 24950525 IC50 = 800 nM T76369 CO37IU 24950526 IC50 = 11000 nM T76369 CUH23T 24950528 IC50 > 100000 nM T76369 CY2NW6 24950843 IC50 = 40 nM T76369 C9BYQ6 24950844 IC50 = 40000 nM T76369 CLW02V 24951001 IC50 = 30 nM T76369 C4MXB8 24951004 IC50 = 150 nM T76369 CIF25O 24951005 IC50 = 40000 nM T76369 CFJW54 24951156 IC50 = 400 nM T76369 CDJ4N0 24951159 IC50 = 3000 nM T76369 C7O2MR 24951162 IC50 = 40000 nM T76369 C3GC9N 24951316 IC50 = 1500 nM T76369 C7NZ2X 24951318 IC50 > 100000 nM T76369 CUDP87 24951320 IC50 > 100000 nM T76369 CWID81 25325634 Ki > 100000 nM T76369 C8HQZ7 44157144 Ki > 100000 nM T76369 C4HL5B 44157145 Ki > 100000 nM T76369 CPM08L 44157218 Ki > 100000 nM T76369 CD5XW6 44157219 Ki > 100000 nM T76369 CU8EQ7 44157220 Ki > 100000 nM T76369 C2PZN0 44157221 Ki > 100000 nM T76369 CSW49B 44157293 Ki > 100000 nM T76369 CO30PI 44157294 Ki > 100000 nM T76369 C47BWL 44157295 Ki > 100000 nM T76369 CA80TE 44157296 Ki > 100000 nM T76369 CGZW85 44157297 Ki > 100000 nM T76369 C7GK9S 44157298 Ki > 100000 nM T76369 CUA79M 44157370 Ki > 100000 nM T76369 C8NK1F 44157371 Ki > 100000 nM T76369 CJXT82 44157372 Ki > 100000 nM T76369 C4UWK6 44157373 Ki > 100000 nM T76369 CZY1Q3 44157374 Ki > 100000 nM T76369 CWIH19 44157375 Ki > 100000 nM T76369 CLS06F 44157439 Ki > 100000 nM T76369 C4R5HG 44157440 Ki > 100000 nM T76369 C03DWN 44157441 Ki > 100000 nM T76369 C3U2AW 44157442 Ki > 100000 nM T76369 CR6DQ1 44157443 Ki > 100000 nM T76369 CKD82Y 44157512 Ki > 100000 nM T76369 CH4T2Z 44157513 Ki > 100000 nM T76369 C8RTA7 44389776 IC50 = 5 nM T76369 CS1JH5 44389963 IC50 = 20000 nM T76369 C84ISX 44389973 IC50 = 20000 nM T76369 CJ91NL 44391726 IC50 = 80 nM T76369 C0C2DX 44428836 Ki > 100000 nM T76369 CZS9U1 44428842 Ki > 100000 nM T76369 CWR3Y1 44428843 Ki > 100000 nM T76369 CUT0H7 44428844 Ki > 100000 nM T76369 C10PFH 44554611 IC50 = 10000 nM T76369 CL6C1X 44554613 IC50 = 700 nM T76369 C6KCQ1 44554787 IC50 = 60 nM T76369 C7M5YB 44569835 Ki = 0.3981 nM T76369 CS61ZR 44569836 Ki = 0.3981 nM T76369 CT3U4M 44569837 Ki = 0.5012 nM T76369 C6IEG1 44569871 Ki = 0.6026 nM T76369 C95PNJ 44569872 Ki = 0.6026 nM T76369 CZF6X0 44569873 Ki = 3.311 nM T76369 C6TQF9 44569874 Ki = 0.7079 nM T76369 C7KS9O 44569875 Ki = 1 nM T76369 C5KO9F 44569911 Ki = 6.457 nM T76369 CB78NA 44569912 Ki = 6.026 nM T76369 CXUP02 44583034 Ki > 100000 nM T76369 CEK3P8 44583159 Ki > 100000 nM T76369 C7IJ3C 49857726 Ki = 279 nM T76369 C04NYX 49857906 Ki > 100000 nM T76369 CDT4Y6 49857907 Ki = 437 nM T76369 C5XS3G 49857908 Ki = 1034 nM T76369 CHRB62 49857909 Ki = 1244 nM T76369 CV7J6X 49857910 Ki > 100000 nM T76369 CYU39N 49857911 Ki > 100000 nM T76369 C5WZL0 49857912 Ki = 756 nM T76369 CCG80U 49858100 Ki > 100000 nM T76369 CCN05H 49858101 Ki = 381 nM T76369 C6S0TB 52944501 IC50 = 26260 nM T76369 CY67HJ 52948155 IC50 = 10970 nM T76369 C5FE4Z 52948907 IC50 = 34 nM T76369 C4OF7Q 53483972 IC50 > 100000 nM T76369 C1QWH9 56931986 IC50 > 100000 nM T76369 CO29WI 71508729 Ki = 17.8 nM T76369 CM93WB 92131904 Ki = 468000 nM T76369 CS1GL7 96359892 Ki = 24800 nM T76369 CDBZ20 102189779 Ki = 0.417 nM T76369 C2CL6P 127030256 IC50 > 100000 nM T76369 CV6B4Z 127030257 IC50 = 12310 nM T76369 CZ0NI1 127030258 IC50 = 25090 nM T76369 C3DL4M 127031478 IC50 = 9130 nM T76369 C2YD1M 127031479 IC50 = 6990 nM T76369 CF0OI3 127034386 IC50 = 20410 nM T76369 C1ZP4G 130431469 IC50 > 10000 nM T76369 CMA35H 130431481 IC50 > 10000 nM T76369 CX59ME 133561407 Ki = 2.4 nM T76369 C8R0BI 137633433 Ki = 148 nM T76369 CFP68C 137635195 Ki = 45.3 nM T76369 CRO26U 137638968 Ki = 4.7 nM T76369 C56IMJ 137643802 Ki = 4.9 nM T76369 C0N3LP 137644595 Ki = 12.9 nM T76369 CBXV07 137652900 Ki = 16.1 nM T76369 CT9IF1 137657377 Ki = 15.6 nM T76369 C1UAZ3 137660095 Ki = 4.44 nM T76369 CEP6R2 137660441 Ki = 14.3 nM T76369 C7YDE3 145951659 IC50 > 100000 nM T76369 C0IS6K 145966157 Ki = 1871 nM T76369 C7HQ2O 145966235 Ki = 12.2 nM T76369 CH3W2Y 145966354 Ki = 102 nM T76369 C3TB2M 145966935 Ki = 25.9 nM T76369 CFT18Y 145969150 Ki = 2425 nM T76369 CQ9G1T 145972810 Ki = 31.9 nM T76369 C0V5WI 145974492 Ki = 48.7 nM T76369 CKD57H 145974917 Ki >= 10000 nM T76369 C6CQI9 145976186 Ki = 42.5 nM T76369 C60ICV 145976488 Ki = 4204 nM T76369 C6W2ZB 145976588 Ki = 14.4 nM T76369 CPL3T8 145977135 Ki = 42 nM T76369 C90CJY 145978164 Ki = 495 nM T76369 CVG8B2 145985484 Ki = 92.3 nM T76369 CQ61NL 145993296 Ki = 3.6 nM T76369 D00ANJ 1897797 Ki = 10 nM T76369 D00CKY 24951315 IC50 = 100 nM T76369 D00IAK 44455840 IC50 = 5.4 nM T76369 D00PLH 44428832 Ki = 230 nM T76369 D00ULT 10609180 IC50 = 10 nM T76369 D01HRG 12884 Ki = 23 nM T76369 D01HZN 44428835 Ki = 1000 nM T76369 D01NDE 11493344 Ki = 7.413 nM T76369 D01NWS 24801394 IC50 = 4.5 nM T76369 D01VAU 123493 Ki = 1540 nM T76369 D01VCS 44428837 Ki = 5650 nM T76369 D01XGP 123358 Ki = 5240 nM T76369 D02BDL 8433 Ki = 26000 nM T76369 D02ENI 10293363 IC50 = 10000 nM T76369 D02GJG 11043027 Ki = 185 nM T76369 D02HQS 19377173 Ki = 370 nM T76369 D02JVI 44387731 IC50 = 20 nM T76369 D02TLP 11363 Ki = 5270 nM T76369 D03HZT 89076 Ki = 1650 nM T76369 D03NTQ 24951319 IC50 = 5000 nM T76369 D03TPH 87203 Ki = 1220 nM T76369 D03WOU 3274712 Ki = 255 nM T76369 D03XIY 24951160 IC50 = 2000 nM T76369 D04AXR 96047 Ki = 8250 nM T76369 D04CDV 44428829 Ki = 190 nM T76369 D04EXR 251908 Ki = 890 nM T76369 D04PMA 15353606 IC50 = 70 nM T76369 D04UEN 44455866 IC50 = 5.5 nM T76369 D05AVX 60983 Ki = 16900 nM T76369 D05EMT 22574258 Ki = 260 nM T76369 D05EYA 18946 Ki = 1.6 nM T76369 D05LTW 22574224 Ki = 34.7 nM T76369 D05PNO 4135273 Ki = 130 nM T76369 D05VUC 19971657 Ki = 990 nM T76369 D05XRY 2752926 Ki = 2980 nM T76369 D05ZCX 44435802 Ki = 150 nM T76369 D06FFD 96430 Ki = 0.029 nM T76369 D06GYH 16745302 Ki = 260 nM T76369 D06MNW 44285344 IC50 = 9000 nM T76369 D06VGD 6724 Ki = 31 nM T76369 D06VSA 11991809 IC50 = 300 nM T76369 D07CFJ 589576 Ki = 17500 nM T76369 D07EDG 1901244 Ki = 31 nM T76369 D07GOA 11150976 IC50 = 3 nM T76369 D07MSJ 11441196 IC50 = 30000 nM T76369 D08AOG 90571 Ki = 15300 nM T76369 D08UOB 44428840 Ki = 140 nM T76369 D08YHD 9878121 IC50 = 0.5 nM T76369 D09GVB 10427006 IC50 = 600 nM T76369 D09LSR 11437501 Ki = 73.5 nM T76369 D0AW4P 10868634 Ki = 3130 nM T76369 D0B0KP 9977214 IC50 = 500 nM T76369 D0B1BQ 157730 IC50 = 4600 nM T76369 D0B1TQ 1810509 Ki = 5530 nM T76369 D0B8YX 75511 Ki = 125 nM T76369 D0BB2U 2385968 Ki = 524 nM T76369 D0C9AD 277990 Ki = 25 nM T76369 D0C9FO 11991892 IC50 = 2000 nM T76369 D0CH0K 11327355 IC50 = 50000 nM T76369 D0CN8Z 11392969 Ki = 371.54 nM T76369 D0D0BI 8371 Ki = 83.9 nM T76369 D0D2HH 44428834 Ki = 665 nM T76369 D0D7FN 283893 Ki = 213.8 nM T76369 D0D7HU 24950683 IC50 = 80 nM T76369 D0D9GS 24951006 IC50 = 10 nM T76369 D0DW9J 123072 Ki = 229.09 nM T76369 D0E0JC 11279040 IC50 = 700 nM T76369 D0E2IG 44428839 Ki = 320 nM T76369 D0E5CF 185195 Ki = 3.981 nM T76369 D0E5ZP 604575 Ki = 13100 nM T76369 D0EK7H 2734793 Ki = 590 nM T76369 D0F3RN 89801 Ki = 5.4 nM T76369 D0F5VY 94860 Ki = 15.9 nM T76369 D0FO4J 182197 Ki = 5.37 nM T76369 D0G2DQ 4669250 Ki > 100000 nM T76369 D0H5RS 11991808 IC50 = 20 nM T76369 D0I0MR 9840659 IC50 = 4800 nM T76369 D0I7FF 176445 Ki = 2.291 nM T76369 D0JH7C 72810 Ki = 5400 nM T76369 D0JI0H 3542734 Ki = 290 nM T76369 D0K6MH 25147546 IC50 = 30 nM T76369 D0K6OM 44428838 Ki = 300 nM T76369 D0K6PO 316765 Ki = 1.5 nM T76369 D0L1ST 2777298 Ki = 158.49 nM T76369 D0L4MF 44428833 Ki = 170 nM T76369 D0LJ2F 11806279 Ki = 5 nM T76369 D0M2EM 4650 Ki > 100000 nM T76369 D0M2ZD 44428831 Ki = 730 nM T76369 D0M5NR 3794313 Ki = 7690 nM T76369 D0M7SQ 9795477 IC50 = 5 nM T76369 D0M8AR 11154099 IC50 = 50000 nM T76369 D0N0HK 73252 Ki = 5440 nM T76369 D0N1CK 9813810 IC50 = 1 nM T76369 D0N8YZ 2427416 Ki = 18.8 nM T76369 D0N9ZR 1718647 Ki = 16500 nM T76369 D0NJ4G 80771 Ki = 3520 nM T76369 D0O0LU 264734 Ki = 1700 nM T76369 D0P1IK 44428841 Ki = 91.3 nM T76369 D0Q2CR 24950841 IC50 = 25 nM T76369 D0Q2YJ 6763 Ki = 2.5 nM T76369 D0Q3GH 146089 Ki = 4.169 nM T76369 D0S6TW 1845 Ki > 100000 nM T76369 D0SP2O 7054 Ki > 100000 nM T76369 D0T5XC 31494 Ki = 173.78 nM T76369 D0TN0A 10085812 IC50 = 1 nM T76369 D0TP1H 44554615 IC50 = 2500 nM T76369 D0U0BV 44428830 Ki = 1300 nM T76369 D0U3JD 16358 Ki = 5380 nM T76369 D0U8IF 10114 IC50 = 20970 nM T76369 D0U8YV 24951000 IC50 = 0.7 nM T76369 D0UK5A 76996 Ki = 532 nM T76369 D0UT1X 101375 Ki = 18100 nM T76369 D0UZ8R 71043 Ki = 3388.44 nM T76369 D0VQ3O 24799659 IC50 = 30 nM T76369 D0W7NY 11991895 IC50 = 20 nM T76369 D0W9VA 10667 Ki = 930 nM T76369 D0WX6R 3477013 Ki = 570 nM T76369 D0X0ER 344135 Ki = 11400 nM T76369 D0Y0XQ 2779383 Ki > 100000 nM T76369 D0Y6RZ 22574214 Ki = 100 nM T76369 D0Y7FX 8651 Ki = 6.9 nM T76369 D0Z1WQ 76915 Ki = 88.6 nM T76369 D0Z5KQ 8400 Ki = 7210 nM T76369 D0Z6CZ 5139980 Ki = 3020 nM T76369 D0Z7WK 10013998 Ki = 5.248 nM T76369 D0Z8HX 16786802 Ki = 9400 nM T76369 D0ZL6B 3772674 Ki = 16 nM T76369 D0ZR2T 2732752 Ki = 16500 nM T76369 D0ZT5C 44428828 Ki = 480 nM T91323 D05PZB 135398495 IC50 = 10 nM T91323 D07XOV 118598754 IC50 = 131 nM T91323 D0E3TC 44259 IC50 = 30.4 nM T91323 D0T3ME 156422 IC50 > 30000 nM T91323 CP04JC 11666231 IC50 = 12.8 nM T91323 CLS29B 46872626 IC50 > 10000 nM T91323 C8NA4L 53384644 IC50 > 30000 nM T91323 CV63UL 67240318 IC50 > 10000 nM T91323 C0EMZ1 71682213 IC50 = 2100 nM T91323 CQ53SW 71682214 IC50 = 2900 nM T91323 C5N1VZ 102581295 IC50 > 10000 nM T91323 C2B4SW 118714182 IC50 = 630 nM T91323 C4B6PX 118714183 IC50 = 4940 nM T91323 CH91ON 129245363 IC50 = 252 nM T91323 CCF8W2 129261617 IC50 = 25 nM T91323 C9C3XT 134163708 IC50 = 10 nM T91323 CGBZ13 134843302 IC50 = 9600 nM T91323 CJI0G1 135520135 IC50 = 32 nM T91323 CH64ID 136175114 IC50 = 51 nM T91323 C5S8CU 136175115 IC50 = 500 nM T91323 C6X4UA 136175116 IC50 = 780 nM T91323 CJKC57 136175117 IC50 = 250 nM T91323 CJ1NU2 136175118 IC50 = 3000 nM T91323 C3MI1P 136175119 IC50 = 360 nM T91323 CVBM76 136175120 IC50 = 110 nM T91323 C2WP5B 136175121 IC50 = 21 nM T91323 C1TS6F 136175122 IC50 = 120 nM T91323 CB5G4X 136175123 IC50 = 24 nM T91323 C3MK9W 136807986 IC50 > 10000 nM T91323 CSGM03 137210056 IC50 = 12 nM T91323 CW3A2B 137210057 IC50 = 700 nM T91323 C4ZGE1 137210058 IC50 = 1100 nM T91323 CX9RJ6 137210059 IC50 = 460 nM T91323 CBJV93 137210060 IC50 = 320 nM T91323 CPM62S 137210061 IC50 = 360 nM T91323 C6S3UF 137210062 IC50 = 1300 nM T91323 CM0AO9 137210063 IC50 = 24 nM T91323 C4DRX1 137643187 IC50 = 5810 nM T91323 CGW9I0 137656387 IC50 = 1410 nM T91323 C9ISH6 145925685 IC50 = 311 nM T91323 CJB1R5 155511461 IC50 = 15 nM T91323 C2MD1Q 155513187 IC50 > 10000 nM T91323 CHD09S 155543566 IC50 = 30 nM T91323 CO2I4P 155559898 IC50 = 4600 nM T91323 D0GN5Z 5281295 IC50 = 5850 nM T31391 D02EYG 10096344 IC50 = 0.1 nM T31391 D04AIT 5280445 IC50 = 120 nM T31391 D07MGA 72281 IC50 = 280 nM T31391 D0D7LA 4091 IC50 = 29000 nM T31391 D0K8KX 5280343 IC50 = 32730 nM T31391 D0K9MY 11243969 Ki = 0.6 nM T31391 D0L3DK 6918537 Ki = 3 nM T31391 D0N5HJ 5462501 IC50 > 100000 nM T31391 D0NI0C 21704 IC50 = 62 nM T31391 D0NJ5H 11450633 IC50 = 2.7 nM T31391 D0RA5Q 72172 IC50 > 100 ug.mL-1 T31391 D0T8XB 44513473 IC50 = 3.8 nM T31391 D0U2JP 4369359 IC50 = 3.5 nM T31391 D0Y7LD 222284 IC50 = 28840 nM T31391 D04XIO 11253490 IC50 = 23 nM T31391 D05LPW 25022354 IC50 = 0.9 nM T31391 D07EPV 11949652 IC50 = 0.37 nM T31391 D07HZG 11516136 IC50 = 11.3 nM T31391 D0FQ2U 6918572 Ki = 0.18 nM T31391 D0L4FS 5280961 IC50 = 480 nM T31391 D0M3XR 46209133 Ki = 0.8 nM T31391 D0N6SO 15983988 IC50 = 4 nM T31391 D0R9HL 11077541 IC50 = 3.5 nM T31391 D0R9YR 64971 IC50 = 55820 nM T31391 D0U2BH 65064 IC50 = 10210 nM T31391 D0U3EP 445154 IC50 = 0.6 nM T31391 D02LNB 22387295 IC50 = 12 nM T31391 D04MAZ 71731606 IC50 = 0.4 nM T31391 D05FMP 66561557 IC50 > 100000 nM T31391 D07JHU 71667377 IC50 > 100000 nM T31391 D0C6NX 73356493 IC50 > 100000 nM T31391 D0K2ZQ 57378228 IC50 = 0.42 nM T31391 D0QX2U 71667229 IC50 > 100000 nM T31391 D00FYF 9796290 IC50 = 22 nM T31391 D01XGX 178060 IC50 > 100000 nM T31391 D08PUW 64982 IC50 = 225000 nM T31391 D0A1NU 16049769 Ki = 1 nM T31391 D0F3TI 11673176 Ki = 1.8 nM T31391 D0Q4YP 11996845 IC50 = 5.3 nM T31391 D0T2IQ 443600 IC50 > 100 ug.mL-1 T31391 CR40US 18844 IC50 = 7 nM T31391 CT2EY7 56877 IC50 > 100000 nM T31391 CL1Y4H 68247 IC50 = 1410 nM T31391 CBP13T 69512 IC50 = 1410 nM T31391 C0V9WL 73324 IC50 > 100 ug.mL-1 T31391 CHAI28 83489 IC50 = 10360 nM T31391 C8EQ1Z 92855 IC50 = 35600 nM T31391 CP1JX4 124031 IC50 = 23.4 ug.mL-1 T31391 C15AMW 158341 IC50 = 14130 nM T31391 CB9Q1L 168182 IC50 = 65690 nM T31391 C6JM7L 182750 IC50 > 100 ug.mL-1 T31391 CV0J8H 182751 IC50 > 100 ug.mL-1 T31391 CGT6C5 276114 IC50 > 100 ug.mL-1 T31391 C7HME8 439246 IC50 = 240 nM T31391 CT2S6P 441667 IC50 = 420 nM T31391 CPKO72 448436 IC50 = 0.1 nM T31391 CP3EL4 454740 IC50 = 3350 nM T31391 C0GD3A 454742 IC50 = 890 nM T31391 C0TYO2 477693 IC50 = 19.8 ug.mL-1 T31391 C7G3CT 477696 IC50 > 100 ug.mL-1 T31391 C8P2LC 485077 IC50 = 56230 nM T31391 CG3C4U 489605 IC50 = 25000 nM T31391 CSJ38Y 679638 IC50 = 3900 nM T31391 CPEY84 688304 IC50 > 100000 nM T31391 C4TRL6 721814 IC50 > 337500 nM T31391 CO3KZ2 741570 IC50 > 100 ug.mL-1 T31391 C18XUS 978607 IC50 = 2800 nM T31391 C0L7TD 1235479 IC50 = 81 ug.mL-1 T31391 C2HQJ7 2302144 IC50 > 100 ug.mL-1 T31391 C30WIA 2750782 IC50 > 100000 nM T31391 CJW0G1 2854000 IC50 = 4000 nM T31391 CT2CQ8 3021908 IC50 = 21000 nM T31391 CX08LH 3081017 IC50 > 100000 nM T31391 CAZ25S 3318661 IC50 > 1000000 nM T31391 CQ0G4F 5281406 IC50 = 87100 nM T31391 C1DW0R 5316300 IC50 = 38430 nM T31391 CAU3O8 5317238 IC50 = 87720 nM T31391 CFB0N1 5318591 IC50 = 26920 nM T31391 CL6J0E 5320287 IC50 = 41690 nM T31391 CQP43H 5360349 IC50 = 5 nM T31391 CS5BG1 5494385 IC50 = 23 nM T31391 CDG53K 5494422 IC50 = 90 nM T31391 CT0E7G 6293081 IC50 = 33110 nM T31391 CE98OF 6451150 IC50 = 21.88 nM T31391 CPUF51 6918418 IC50 = 5700 nM T31391 C4RE5F 7020797 IC50 = 21000 nM T31391 C48BSO 7614279 IC50 = 26100 nM T31391 C37RIP 9655981 IC50 = 3440 nM T31391 C14VRG 9794073 IC50 = 3900 nM T31391 CQT36A 9794235 IC50 = 1700 nM T31391 CXEQ40 9795464 IC50 = 64 nM T31391 CMVO26 9795469 IC50 = 21 nM T31391 CBG8M2 9796291 IC50 = 1170 nM T31391 CSA6V9 9796352 Ki = 218 nM T31391 C7KR1T 9799867 IC50 = 4 nM T31391 CNJ0Z3 9800721 Ki = 2 nM T31391 C75RIB 9801978 IC50 = 7 nM T31391 C5F7DH 9815545 IC50 = 2 nM T31391 CUNB40 9817010 IC50 = 247000 nM T31391 C1I5JZ 9819537 IC50 = 298 nM T31391 CDP16K 9821063 IC50 = 17000 nM T31391 C8CR0Z 9821205 IC50 = 0.13 nM T31391 CKR9Y5 9823963 IC50 = 13 nM T31391 C8EK7G 9835053 IC50 = 3700 nM T31391 CW5EZ7 9835382 IC50 = 1600 nM T31391 CDY12G 9835472 IC50 = 3100 nM T31391 CV87XC 9835734 Ki = 154 nM T31391 CAHB35 9836210 IC50 = 922 nM T31391 CU2B0F 9838664 IC50 = 110 nM T31391 C62DNH 9843297 IC50 = 27 nM T31391 CUD46C 9855673 IC50 = 188000 nM T31391 CO2YQ4 9858442 IC50 = 69 nM T31391 C8XO1Z 9859008 Ki = 18 nM T31391 CNYI42 9859384 IC50 = 0.6 nM T31391 C2DMP6 9861924 IC50 > 100 ug.mL-1 T31391 CK0BS5 9864687 IC50 = 36 nM T31391 C5CZ6J 9865563 Ki = 53 nM T31391 CF3I8A 9865779 IC50 = 4.6 nM T31391 CR9AW7 9870934 IC50 = 23 nM T31391 CQN2L1 9882325 IC50 = 63 nM T31391 CZUQ34 9883487 IC50 = 460 nM T31391 C2TV9M 9884543 IC50 = 0.064 nM T31391 CBI2C9 9885607 IC50 = 82 nM T31391 CFMG63 9886974 IC50 = 12 ug.mL-1 T31391 CBW37X 9903629 IC50 = 466 nM T31391 C4T1CX 9904675 IC50 = 491 nM T31391 CU0I4K 9907074 IC50 = 270 nM T31391 CMGX12 9920733 IC50 = 23100 nM T31391 C4EC8A 9924995 IC50 = 610 nM T31391 C1S5VM 9927481 IC50 = 436 nM T31391 C6T0RU 9928326 IC50 = 360 nM T31391 C8Y5UK 9939534 IC50 = 23 nM T31391 CFH1V2 9942336 IC50 > 1000000 nM T31391 C28XTC 9942425 Ki = 2000 nM T31391 CZ1S9O 9942554 IC50 = 0.3 nM T31391 CZMT26 9947730 IC50 = 166 nM T31391 C2KW8I 9951445 IC50 = 1.8 nM T31391 CLR78W 9952894 IC50 = 88 nM T31391 CQ8J7T 9953181 IC50 = 59 nM T31391 C8OX9T 9964212 IC50 = 50400 nM T31391 C8THS1 9970277 IC50 = 64000 nM T31391 C1A3YN 9972358 IC50 = 2300 nM T31391 CH39FT 9973732 IC50 = 2000 nM T31391 C9EZ1X 9978478 IC50 = 2.2 nM T31391 CT6XQ2 9983092 IC50 = 1.4 nM T31391 C18ZXU 9990413 IC50 > 1000000 nM T31391 C1NB0Q 9992723 Ki = 79 nM T31391 C5Q6BJ 9995375 IC50 > 100 ug.mL-1 T31391 C17BCF 10003476 IC50 = 1 nM T31391 CN8XI3 10006926 IC50 = 1 nM T31391 CVG9I2 10012350 IC50 > 1000000 nM T31391 C7IB1W 10014222 Ki = 8 nM T31391 C4KT7I 10014539 IC50 > 1000000 nM T31391 CQ7G2R 10018887 IC50 = 1100 nM T31391 CV85MG 10019118 IC50 = 196000 nM T31391 CN0T5A 10019492 IC50 = 7400 nM T31391 C78NMY 10026124 IC50 = 234 nM T31391 CWQ21K 10038196 Ki = 96 nM T31391 CSZ75E 10046311 IC50 = 71 nM T31391 CRG1N0 10058240 IC50 >> 1000000 nM T31391 CYMG54 10058520 Ki = 210 nM T31391 C64ZDU 10059633 IC50 = 545000 nM T31391 CYH3C6 10061400 IC50 > 100 ug.mL-1 T31391 CV7SK8 10064801 IC50 = 57800 nM T31391 CI1Q6X 10081481 IC50 > 500000 nM T31391 CHC82B 10083376 IC50 > 1000000 nM T31391 CSHQ57 10084828 IC50 > 1000000 nM T31391 CB9J1F 10086451 IC50 = 16 nM T31391 C06KTL 10087724 IC50 > 1000000 nM T31391 C97FIB 10087948 IC50 = 245 nM T31391 C83ZDL 10096130 IC50 = 22 nM T31391 C8P3UC 10106636 Ki = 24 nM T31391 C5U0ON 10107122 IC50 = 3.3 nM T31391 C3K2MO 10109454 IC50 = 0.18 nM T31391 C7A3ZJ 10111068 Ki = 79 nM T31391 CKP5D7 10111288 IC50 = 7 nM T31391 CKY4R8 10112957 Ki = 281 nM T31391 CN5BD7 10114895 IC50 = 731 nM T31391 CIU12J 10116290 IC50 = 170 nM T31391 CM19YB 10125495 IC50 = 18000 nM T31391 CQT5Y2 10125644 IC50 = 1400 nM T31391 C10JOC 10125645 IC50 = 2500 nM T31391 CAOF95 10125896 IC50 = 200 nM T31391 C10BSW 10125952 IC50 = 1100 nM T31391 CD20SG 10125953 IC50 = 14000 nM T31391 CT6CG1 10126186 IC50 = 0.2 nM T31391 C0Q7BK 10127057 IC50 = 42 nM T31391 CNC5D4 10130367 Ki = 182 nM T31391 C9ERD7 10130575 IC50 = 22 nM T31391 CBL6T7 10132708 IC50 = 5 nM T31391 CLZF79 10133903 Ki = 12 nM T31391 C2RW5Z 10135822 Ki = 324 nM T31391 C4U3IC 10144962 IC50 = 139 nM T31391 C2H0UF 10149048 Ki = 0.03 nM T31391 C2YUP9 10149491 IC50 = 14000 nM T31391 CUE7K0 10156677 Ki = 112 nM T31391 C4CX1P 10157141 IC50 = 128 nM T31391 CUB1G7 10157334 Ki = 68 nM T31391 C6PZ1U 10160012 Ki = 316 nM T31391 C0L1KV 10162433 Ki = 428 nM T31391 C29RUO 10162817 Ki = 579 nM T31391 CQ3K8W 10164624 IC50 = 1900 nM T31391 C5X4NF 10171676 IC50 = 1000 nM T31391 C98FDL 10172375 IC50 = 0.9 nM T31391 C6SQ0P 10172376 IC50 = 90 nM T31391 CJ3MD2 10172601 IC50 = 100 nM T31391 C2SNQ8 10172681 IC50 = 240 nM T31391 C2KWM9 10172706 IC50 = 3 nM T31391 CXUC74 10173174 IC50 = 130 nM T31391 CKWE80 10176680 Ki = 2.2 nM T31391 C1UAG7 10176937 IC50 = 25 nM T31391 CEM94Y 10178009 IC50 = 539 nM T31391 C6S5OX 10179212 Ki = 29 nM T31391 CF7C3M 10180260 Ki = 45 nM T31391 C4FC2O 10183667 IC50 = 108 nM T31391 C7PWN9 10193213 IC50 = 31000 nM T31391 CWU9N2 10198228 Ki = 3 nM T31391 C05DXJ 10200731 Ki = 302 nM T31391 C6ISW4 10203198 Ki = 309 nM T31391 CD2U3A 10203599 Ki = 63 nM T31391 CQ8N1T 10209865 IC50 = 134 nM T31391 CFP27I 10214732 IC50 = 42000 nM T31391 C0CPY9 10215103 IC50 = 370 nM T31391 CL4T7Z 10215326 IC50 = 270 nM T31391 CLO81K 10215577 IC50 = 1750 nM T31391 C68WBI 10215628 IC50 = 47 nM T31391 CQ0V1C 10219838 IC50 = 39000 nM T31391 CZ9XN0 10220206 IC50 = 170 nM T31391 CBZ3P2 10221723 Ki = 56 nM T31391 CBC45I 10222923 Ki = 1278 nM T31391 CZ92XV 10225547 Ki = 76 nM T31391 CU9W8N 10233525 IC50 = 405 nM T31391 COD64C 10236556 IC50 = 47000 nM T31391 CYCJ68 10236557 IC50 = 1500 nM T31391 C9K3JS 10237877 IC50 = 180 nM T31391 C5P0AO 10238227 IC50 = 113 nM T31391 CTG4S9 10238900 IC50 = 1397 nM T31391 CCS75T 10242745 IC50 > 1000000 nM T31391 CW6PG0 10243173 Ki = 811 nM T31391 C07QCO 10243334 IC50 = 346 nM T31391 C6JS1Y 10245529 IC50 = 42 nM T31391 C0A9OY 10249393 IC50 = 30 nM T31391 CZ90LD 10250452 IC50 = 12 nM T31391 CU8C5K 10254918 IC50 = 5 nM T31391 C17HUN 10255762 IC50 = 8.4 nM T31391 C6ER9U 10269517 IC50 = 50 nM T31391 CQ07AR 10270647 Ki = 33 nM T31391 C9BPX2 10270831 IC50 = 280 nM T31391 CD0P5E 10271196 Ki = 530 nM T31391 CQ36IM 10272290 Ki = 24 nM T31391 C6M4SQ 10286219 IC50 = 1500 nM T31391 CAPB18 10286460 IC50 = 200 nM T31391 CZHS09 10286494 IC50 = 10000 nM T31391 CHWJ15 10286977 IC50 = 0.2 nM T31391 CT6FG8 10287141 IC50 = 340 nM T31391 C7AQS6 10287238 IC50 = 3 nM T31391 CHO8E7 10296151 Ki = 1 nM T31391 CC63ZN 10296260 IC50 = 864 nM T31391 CA7Q8J 10298482 Ki = 65 nM T31391 CY3LK8 10300368 Ki = 310 nM T31391 C9FZ2O 10304081 IC50 = 225 nM T31391 C8J3NA 10304145 IC50 = 44 nM T31391 C7US0V 10304855 IC50 = 114 nM T31391 CJDY62 10306170 IC50 = 14 nM T31391 C5AXF1 10308325 IC50 = 20000 nM T31391 CEGV15 10308355 IC50 = 40000 nM T31391 CNX7Q1 10308853 IC50 = 920 nM T31391 CTZN24 10309295 IC50 = 350 nM T31391 CQYE24 10309373 IC50 = 53 nM T31391 C3FB4T 10310021 IC50 = 91 nM T31391 CY6N9I 10318743 IC50 = 9.6 nM T31391 CF1S8U 10320144 IC50 = 4 nM T31391 C08UHI 10320529 IC50 = 117000 nM T31391 CC2TP8 10321088 IC50 = 5 nM T31391 CNV4R3 10324641 IC50 = 5.8 nM T31391 C0JD8Z 10333136 IC50 = 16 ug.mL-1 T31391 CIAV18 10333629 IC50 >> 1000000 nM T31391 CL72FC 10334538 IC50 > 1000000 nM T31391 C4UTO9 10336929 IC50 = 44 nM T31391 CM6Y1B 10339570 Ki = 5 nM T31391 CXP16T 10340933 IC50 = 15000 nM T31391 C1AEN6 10341846 IC50 > 125000 nM T31391 CEZ95L 10342016 IC50 = 58 nM T31391 CKZT43 10353699 IC50 = 518000 nM T31391 CU6LC2 10355512 IC50 = 104 nM T31391 CR0QC5 10367502 IC50 = 3 nM T31391 CP4M2R 10375745 IC50 = 80 nM T31391 CW70CV 10376453 IC50 >> 1000000 nM T31391 C7UO3L 10376704 Ki = 25 nM T31391 CK07VX 10376940 IC50 = 217000 nM T31391 CK8T4C 10381531 IC50 = 14.1 ug.mL-1 T31391 C79UAO 10381586 IC50 > 100 ug.mL-1 T31391 CQ7J2Z 10383508 IC50 = 15 nM T31391 C2GT0H 10384474 IC50 = 80 nM T31391 CY5M4R 10388027 IC50 = 26 nM T31391 CHZ85I 10393133 IC50 = 4800 nM T31391 CLI51Z 10398371 IC50 > 1000000 nM T31391 C29MEL 10399628 Ki = 22 nM T31391 C2EPA5 10401083 IC50 = 635 nM T31391 C6GWB8 10401570 IC50 > 100 ug.mL-1 T31391 C8NAX7 10403949 IC50 > 500000 nM T31391 CE0AS5 10405951 IC50 = 9 nM T31391 C7R6TZ 10406789 IC50 = 100 nM T31391 CVK1G5 10412922 IC50 = 13 nM T31391 CTK71I 10415171 IC50 = 400 nM T31391 C92DAJ 10415172 IC50 = 5600 nM T31391 C7F8SB 10420127 IC50 = 612 nM T31391 C7YIE3 10423532 Ki = 90 nM T31391 C1O2RY 10426457 IC50 = 11.5 nM T31391 C80ZBS 10429788 IC50 = 71 nM T31391 CUS9F6 10432611 IC50 = 13 nM T31391 C6GHF1 10433039 IC50 = 45 nM T31391 CWCA76 10439426 IC50 = 0.48 nM T31391 CAF71Y 10443207 IC50 = 247000 nM T31391 C4BKD9 10445283 Ki = 959 nM T31391 CO59EL 10450114 IC50 = 6.6 nM T31391 CCTY29 10451878 IC50 = 50 nM T31391 C4OC6P 10455620 IC50 = 175 nM T31391 C1WKE4 10455621 IC50 = 100 nM T31391 CHP37D 10456407 IC50 = 142000 nM T31391 C03IBO 10467163 Ki = 3800 nM T31391 CLV58Q 10468265 IC50 >> 1000000 nM T31391 CH1DG5 10478099 IC50 = 92 nM T31391 CL3H9I 10491923 IC50 > 100 ug.mL-1 T31391 CJ2RK6 10492044 IC50 > 100 ug.mL-1 T31391 CF46MR 10515590 IC50 = 70 nM T31391 C30TAX 10538170 IC50 = 95 nM T31391 CN4BI1 10564514 IC50 = 32 nM T31391 C8KLC3 10584166 IC50 = 11 nM T31391 CK3IW4 10584272 IC50 = 3500 nM T31391 C0KTQ5 10607253 IC50 = 50400 nM T31391 C38IDQ 10608000 IC50 = 250 nM T31391 C4PJ7H 10656779 Ki = 2150 nM T31391 C3YS4K 10659346 IC50 > 100 ug.mL-1 T31391 CN5KG9 10661540 IC50 = 12.8 ug.mL-1 T31391 CH6S5L 10704521 IC50 = 60 nM T31391 CXE71J 10750510 IC50 = 30000 nM T31391 CHA8X6 10751333 IC50 = 94000 nM T31391 CYLO09 10774283 IC50 = 52000 nM T31391 C1LSP2 10779050 IC50 > 100 ug.mL-1 T31391 CL26WQ 10780092 IC50 = 286000 nM T31391 C2KDY6 10798619 IC50 = 374000 nM T31391 C1WG0P 10798659 IC50 = 0.3 nM T31391 C1ZJ4I 10799226 IC50 = 107000 nM T31391 CJKX61 10821833 IC50 = 67000 nM T31391 C7BLJ1 10821834 IC50 > 1000000 nM T31391 CHC1X4 10824414 IC50 = 63 nM T31391 C3E8ID 10845163 IC50 = 15000 nM T31391 CK9SB4 10845727 IC50 = 93000 nM T31391 CCR8J7 10848386 IC50 = 17000 nM T31391 C04XQH 10850290 IC50 > 100 ug.mL-1 T31391 C1QL5M 10858831 IC50 > 1000000 nM T31391 C6QH7S 10860092 IC50 = 18600 nM T31391 C6WGA4 10861905 IC50 = 10 nM T31391 CJ39DG 10872395 IC50 > 500000 nM T31391 CS1LP6 10879478 IC50 = 24200 nM T31391 C3UGO0 10879937 IC50 = 53 nM T31391 C2QEW3 10883432 IC50 = 296 nM T31391 C4A5BM 10902702 IC50 = 598 nM T31391 C6ERS7 10904132 IC50 = 23 nM T31391 CVI2T1 10911918 IC50 = 103000 nM T31391 C42NLJ 10912330 IC50 = 7000 nM T31391 CV46YZ 10912691 IC50 = 33 nM T31391 CG9Q1Y 10923589 IC50 = 133 nM T31391 C9BL6G 10926029 IC50 = 70 nM T31391 CLA05J 10932707 Ki = 10 nM T31391 CPG58B 10943400 IC50 = 475 nM T31391 C6HNK4 10947008 IC50 = 7 nM T31391 CTWI82 10950467 IC50 = 149 nM T31391 CYP97B 10958030 IC50 = 17 nM T31391 CF60BW 10966961 IC50 = 26 nM T31391 CY9CW2 10969177 IC50 = 8 nM T31391 CW63DG 10980018 IC50 = 434000 nM T31391 C63VGB 10993665 IC50 = 64 nM T31391 CM5E1A 11000330 IC50 = 52600 nM T31391 CBFE09 11015514 IC50 = 183 nM T31391 CT9I8W 11020125 IC50 = 9610 nM T31391 CWR9G6 11023706 IC50 = 477000 nM T31391 CX1KF2 11024849 IC50 = 14 nM T31391 CA2OR9 11025044 IC50 = 228 nM T31391 CZ94WH 11025199 IC50 > 500000 nM T31391 C4MD5V 11037154 IC50 > 1000000 nM T31391 CH4TD3 11037548 IC50 = 326000 nM T31391 C0O8HF 11045633 IC50 = 29 nM T31391 CEPQ46 11053284 IC50 = 266 nM T31391 CTMK05 11056962 IC50 = 83 nM T31391 C42WCR 11065479 IC50 > 1000000 nM T31391 C9CYS1 11067211 IC50 = 931000 nM T31391 C9S8AG 11068388 IC50 = 16000 nM T31391 C0FWU4 11069462 IC50 = 22 nM T31391 CVJ81D 11075465 IC50 = 282 nM T31391 CNA61F 11076103 IC50 = 305 nM T31391 C60JXQ 11079321 IC50 > 1000000 nM T31391 C2N6MH 11084500 IC50 = 444 nM T31391 CX07LO 11085063 IC50 = 261 nM T31391 CSRO28 11089704 IC50 = 18 nM T31391 CS48RN 11098969 IC50 = 3000 nM T31391 COAR21 11101478 IC50 = 12000 nM T31391 CMO61N 11109983 IC50 = 338 nM T31391 C10CQP 11112644 IC50 = 62 nM T31391 CA4N0B 11117606 Ki = 11 nM T31391 C9GXD6 11117990 IC50 > 500000 nM T31391 C6QL3H 11122260 IC50 > 1000000 nM T31391 C1X8SI 11127914 IC50 = 398 nM T31391 CF41JX 11127915 IC50 = 105 nM T31391 CJB52P 11129932 IC50 = 3 nM T31391 CWDY68 11138020 IC50 = 192 nM T31391 C26ODF 11150893 IC50 > 500000 nM T31391 CXT8Y2 11151568 IC50 = 6 nM T31391 C4HBU9 11153488 IC50 = 30 nM T31391 CJ7E0N 11163434 IC50 = 0.13 nM T31391 CE94RO 11164254 IC50 = 9.3 nM T31391 C7HRW0 11164704 IC50 = 5 nM T31391 C82GSQ 11165177 IC50 = 77 nM T31391 CSB2T9 11166406 IC50 > 125000 nM T31391 CXR12G 11173505 Ki = 49 nM T31391 CX10UC 11173801 IC50 = 5.6 nM T31391 C5U1FY 11176598 IC50 = 830 nM T31391 CN3D5C 11180149 Ki = 0.59 nM T31391 CJS94B 11187292 IC50 = 5.6 nM T31391 C2ME1R 11187389 Ki = 8.9 nM T31391 CG49PR 11187940 Ki = 1.6 nM T31391 C9HKB7 11188314 IC50 = 23 nM T31391 C5E7VQ 11198004 IC50 = 20 nM T31391 CO9QM2 11198569 IC50 > 100000 nM T31391 CF1LD8 11199808 Ki = 0.4 nM T31391 C40SYQ 11200151 Ki = 8 nM T31391 C68XFD 11205761 IC50 > 1000000 nM T31391 C3BXS4 11206225 Ki = 14500 nM T31391 CMBT59 11207320 IC50 > 250000 nM T31391 CR60FN 11209195 IC50 = 17000 nM T31391 CW8FL2 11209569 IC50 = 301000 nM T31391 CJB87Z 11210511 IC50 = 9.7 nM T31391 C2PN1R 11211023 IC50 = 19 nM T31391 CH87RA 11211119 IC50 = 3.6 nM T31391 CHIZ26 11218348 IC50 = 6.3 nM T31391 C6VKT5 11219158 IC50 = 3700 nM T31391 CK5W4F 11220098 Ki = 143 nM T31391 CXAR72 11220471 IC50 = 250000 nM T31391 CSN6U7 11220682 IC50 = 18 nM T31391 CEUD41 11222126 IC50 = 2.6 nM T31391 CU3BG5 11222807 IC50 = 27 nM T31391 CJ2M8G 11222935 Ki = 1.4 nM T31391 C71YJO 11223701 Ki = 0.9 nM T31391 CK1UE7 11229192 IC50 = 188000 nM T31391 C35JSU 11229576 IC50 = 151000 nM T31391 C3X9SY 11229581 IC50 = 148000 nM T31391 CHX25W 11232123 IC50 = 345000 nM T31391 C0JD5Q 11232605 IC50 = 179000 nM T31391 CYL67P 11232890 Ki = 0.85 nM T31391 CR3PJ9 11233253 IC50 = 8 nM T31391 CVL7H4 11233695 IC50 = 30 nM T31391 C3UA7X 11234761 IC50 = 12 nM T31391 C32ZGY 11234800 IC50 = 3 nM T31391 CBES80 11235729 IC50 = 23 nM T31391 C5AB7G 11236208 IC50 = 1.49 nM T31391 C5CZH3 11242300 IC50 = 2130 nM T31391 CUS5G2 11243728 IC50 = 56000 nM T31391 CH82RJ 11244267 IC50 > 1000000 nM T31391 CDLT06 11245133 IC50 = 63 nM T31391 CQ6C5F 11246131 IC50 = 23 nM T31391 C4VQ0N 11246214 IC50 = 5 nM T31391 C67YUV 11253949 Ki = 3.9 nM T31391 CLJ7A1 11255193 IC50 = 417000 nM T31391 CR6N9B 11256457 IC50 = 430 nM T31391 C8M4XU 11256492 IC50 = 35 nM T31391 C2YS9G 11256520 IC50 = 5 nM T31391 C43HPD 11258527 IC50 = 990 nM T31391 C61KZW 11266019 IC50 = 496000 nM T31391 CN2O0L 11268786 IC50 = 4 nM T31391 CKL1A8 11268930 Ki = 0.93 nM T31391 CHO56W 11269281 IC50 = 570 nM T31391 CM0YI7 11269397 Ki = 0.96 nM T31391 C5IY0L 11269712 IC50 = 95000 nM T31391 CM1A5F 11270889 IC50 = 2.77 nM T31391 CR46GY 11277009 IC50 > 1000000 nM T31391 C17TLH 11277905 IC50 = 43 nM T31391 CXFV02 11278425 Ki = 3.5 nM T31391 CUB62P 11278798 IC50 = 4 nM T31391 CB5SD1 11280296 IC50 = 12 nM T31391 CUK58N 11281626 Ki = 0.4 nM T31391 CL5SH2 11281817 IC50 = 21 nM T31391 C0RWV3 11282205 IC50 = 7400 nM T31391 CWNT74 11283294 IC50 = 25 nM T31391 CUM48L 11288538 IC50 = 1.8 nM T31391 C0U2MV 11289193 IC50 = 205000 nM T31391 CO59DU 11289695 IC50 = 6.5 nM T31391 CTC0P9 11289792 IC50 = 148000 nM T31391 CM85DX 11291335 IC50 = 7800 nM T31391 C1YH5K 11291901 IC50 = 36 nM T31391 CCDX51 11292489 Ki = 3.8 nM T31391 CPD0L4 11292861 Ki = 0.35 nM T31391 CSH2N3 11294846 IC50 = 3 nM T31391 C51QAB 11300739 IC50 = 418000 nM T31391 CZV8P2 11300763 Ki = 10 nM T31391 CAL43D 11302841 IC50 = 13 nM T31391 C1TZY0 11302974 Ki = 42 nM T31391 CAW02M 11303089 IC50 = 14 nM T31391 CDZ79G 11304224 IC50 = 240 nM T31391 C2SOA8 11306467 IC50 = 71 nM T31391 CEJ32C 11306468 IC50 = 71 nM T31391 C06NLF 11309656 IC50 = 190000 nM T31391 C8I1QE 11310450 IC50 = 500000 nM T31391 C47GSV 11310499 IC50 = 23000 nM T31391 CP9LQ0 11312069 IC50 = 278000 nM T31391 CG8SA2 11312331 IC50 = 13 nM T31391 C4GUX3 11312733 IC50 > 500000 nM T31391 CMPH23 11313182 IC50 = 13 nM T31391 CEZ27P 11314348 Ki = 0.6 nM T31391 CM28RS 11314596 IC50 = 890 nM T31391 CL72NR 11314959 Ki = 0.45 nM T31391 CT6MF7 11316670 IC50 = 3 nM T31391 CTG12Q 11321743 IC50 = 23100 nM T31391 C9XYK1 11325183 IC50 = 6.2 nM T31391 CS8OH7 11326271 IC50 = 430 nM T31391 CK6G2V 11335782 Ki = 270 nM T31391 C43RXS 11337326 IC50 = 22 nM T31391 C38ADT 11346439 IC50 = 125000 nM T31391 C5SR4K 11346707 IC50 = 350 nM T31391 C9SJ0O 11347777 Ki = 607 nM T31391 CM4CT0 11348315 IC50 = 10 nM T31391 CM5E2A 11349317 IC50 = 57 nM T31391 C35GXU 11350142 Ki = 10 nM T31391 CNB7G8 11356095 IC50 = 39000 nM T31391 C24QLP 11356421 IC50 = 1000000 nM T31391 C1WOH9 11359214 IC50 > 500000 nM T31391 CK2T6J 11359671 IC50 = 17 nM T31391 CUH3S7 11360493 IC50 = 20 nM T31391 CQ9TJ5 11360810 IC50 = 3.7 nM T31391 CZ93VH 11361944 IC50 = 6 nM T31391 CKP0G9 11362130 IC50 = 34 nM T31391 CZ37IN 11372458 IC50 = 192000 nM T31391 CCNX41 11372959 IC50 = 540 nM T31391 CMZ1S9 11373129 IC50 = 6 nM T31391 CW3QZ7 11374531 IC50 = 19.4 nM T31391 C30JEU 11381416 IC50 = 69 nM T31391 C9FN7U 11381726 IC50 > 500000 nM T31391 CQ0MC7 11383372 IC50 = 200 nM T31391 CH74XT 11383468 IC50 > 500000 nM T31391 CE3O6K 11386357 IC50 = 14 nM T31391 CML13R 11389441 Ki = 7000 nM T31391 CH35IZ 11392716 IC50 = 14 nM T31391 CF01WK 11392988 Ki = 2.9 nM T31391 CL9HN3 11395030 Ki = 2 nM T31391 CD5A7Z 11395141 Ki = 10 nM T31391 CR9EB8 11396245 IC50 = 5 nM T31391 CEZS68 11403720 Ki = 28 nM T31391 CSR53F 11404106 IC50 = 186000 nM T31391 C0X6EK 11404881 Ki = 0.72 nM T31391 CI40EH 11405274 Ki = 57 nM T31391 C50PNA 11405365 Ki = 7.1 nM T31391 C3QZD5 11406220 Ki = 5.5 nM T31391 CTW02K 11406276 Ki = 0.67 nM T31391 CV1E7C 11406559 IC50 = 109 nM T31391 C3S8BD 11415118 IC50 = 5.6 nM T31391 C9AW7O 11416338 IC50 = 5 nM T31391 C0RIS4 11417008 IC50 = 15.1 nM T31391 CW8K3F 11417567 IC50 = 6.8 nM T31391 C2ZT0L 11418204 IC50 = 8 nM T31391 CRZ5F1 11418876 IC50 = 27 nM T31391 CFD62G 11419146 IC50 = 6 nM T31391 CPY7B2 11424308 Ki = 26 nM T31391 C3AZ7K 11426348 IC50 = 15 nM T31391 CB5C1T 11428334 Ki = 12 nM T31391 CY15PU 11429829 Ki = 0.83 nM T31391 CFTC85 11432169 IC50 = 29 nM T31391 C27ITV 11436930 IC50 = 250000 nM T31391 CLF89Y 11437087 IC50 > 1000000 nM T31391 CH39KX 11437726 IC50 = 188000 nM T31391 C82ENX 11439333 IC50 = 7 nM T31391 CRW3G4 11440163 IC50 = 10 nM T31391 CN9ZA8 11441300 IC50 = 68 nM T31391 CH09SE 11447824 IC50 > 1000000 nM T31391 CPNU92 11448828 IC50 = 4.9 nM T31391 CUG51Q 11449442 IC50 = 132000 nM T31391 C9RZC1 11450265 IC50 = 70000 nM T31391 CW27UK 11450266 IC50 = 500000 nM T31391 CZ68MT 11451290 IC50 = 8 nM T31391 CY0JG1 11451461 Ki = 1.6 nM T31391 C0DT1O 11451712 Ki = 7.4 nM T31391 CX5Y7J 11451739 Ki = 10 nM T31391 C6P2BR 11452943 Ki = 0.62 nM T31391 C6US2X 11461807 IC50 = 8 nM T31391 CV71FH 11464036 IC50 = 8 nM T31391 C1M9UX 11469862 Ki = 2.2 nM T31391 CWO06L 11471453 IC50 = 10 nM T31391 C7TOQ4 11472776 IC50 > 500000 nM T31391 CO7T4W 11473127 IC50 > 500000 nM T31391 C53RWU 11474019 IC50 = 266000 nM T31391 C6WT7P 11474308 Ki = 25 nM T31391 C5TQP7 11474372 Ki = 31 nM T31391 CE5A4M 11475797 IC50 = 34.3 nM T31391 C7JWD3 11476287 IC50 = 18 nM T31391 CS4H7X 11481506 Ki = 5.2 nM T31391 C6U9KB 11484559 IC50 = 4 nM T31391 C4G9AM 11484758 IC50 = 510 nM T31391 CPL64M 11486126 Ki = 21 nM T31391 CTD0S4 11486251 Ki = 0.98 nM T31391 CNMA97 11487118 IC50 = 128 nM T31391 CBV79P 11487883 Ki = 0.62 nM T31391 CEHI82 11493140 IC50 > 3000 nM T31391 C06RUA 11493219 IC50 = 64 nM T31391 C3MPY0 11493220 IC50 = 955 nM T31391 CDT16S 11493492 Ki = 28 nM T31391 CUTS18 11494449 IC50 = 2800 nM T31391 C50YHW 11494571 IC50 = 31300 nM T31391 C9PRY1 11494684 IC50 = 811 nM T31391 CJD30Y 11495704 IC50 = 2.3 nM T31391 CGA6Q4 11500119 IC50 = 4000 nM T31391 CAH5Z6 11500899 IC50 = 91 nM T31391 C2D9AT 11500939 Ki = 103 nM T31391 CKWZ03 11501743 IC50 = 80 nM T31391 CH7VS5 11505454 IC50 = 28 nM T31391 CBM01H 11507111 IC50 = 1600 nM T31391 CW38YC 11507527 IC50 = 89 nM T31391 C3XAT0 11507559 IC50 = 687 nM T31391 C62RBF 11507639 IC50 = 261 nM T31391 CF2S9Q 11507721 IC50 > 30000 nM T31391 C30JDP 11508177 IC50 = 1070 nM T31391 CLH62G 11508839 IC50 = 19 nM T31391 CM8QB3 11510166 Ki = 93 nM T31391 CQDM72 11514208 IC50 = 1000 nM T31391 C04OAE 11514331 IC50 = 1110 nM T31391 C7CLT9 11515196 IC50 = 118 nM T31391 CA3FS5 11515240 IC50 = 123 nM T31391 C15UQK 11515912 IC50 = 428 nM T31391 CO95FZ 11516000 IC50 = 1160 nM T31391 C0XVU3 11516085 IC50 = 7.6 nM T31391 C2S8BH 11516511 Ki = 14 nM T31391 CH5A7Q 11518007 IC50 = 2.5 nM T31391 C91OHR 11522044 IC50 > 3000 nM T31391 CJM1L9 11522376 IC50 = 62 nM T31391 C31ZBJ 11522467 IC50 = 689 nM T31391 C2TCM8 11523077 IC50 = 6.6 nM T31391 CY96CU 11523396 IC50 = 14800 nM T31391 CDCI64 11524392 IC50 = 14 nM T31391 C8KB4F 11524437 Ki = 612 nM T31391 CMYN65 11526865 IC50 = 150 nM T31391 C0O3XD 11527019 IC50 = 19 nM T31391 CWH3S0 11529375 IC50 = 52 nM T31391 CMN4Y5 11529427 IC50 = 1220 nM T31391 COL08I 11529539 IC50 = 97 nM T31391 CQ56DV 11529688 IC50 = 257 nM T31391 CXA53K 11529948 IC50 = 208 nM T31391 C10LHK 11531002 IC50 = 371 nM T31391 CV1N6Z 11531612 IC50 = 17 nM T31391 CZFI65 11531704 Ki = 30 nM T31391 C1B8JN 11532057 Ki > 10000 nM T31391 CZ35WN 11533932 IC50 = 13 nM T31391 C63DBH 11537823 Ki = 44 nM T31391 COXK41 11537890 Ki = 137 nM T31391 CKM89Z 11538673 IC50 = 22 nM T31391 CFXG35 11538686 IC50 = 13400 nM T31391 CMD6H8 11538715 IC50 = 5.8 nM T31391 CK36XC 11538961 Ki = 18 nM T31391 CG7I8Z 11538992 IC50 = 21 nM T31391 CPR71X 11540951 IC50 = 2.7 nM T31391 C98GDW 11541277 IC50 = 61 nM T31391 CBR9K8 11541314 IC50 = 7.5 nM T31391 CC5M2E 11544575 IC50 = 69 nM T31391 C1HV5Q 11544965 IC50 = 702 nM T31391 CVT52Y 11545508 IC50 = 30 nM T31391 C6KBN4 11546261 Ki = 2.2 nM T31391 CJIX61 11547698 IC50 = 9.9 nM T31391 C5AR6V 11550675 IC50 = 201 nM T31391 C9I5GV 11551088 IC50 = 26 nM T31391 C5NC3J 11551710 Ki = 21 nM T31391 CY3RK7 11551987 IC50 = 102 nM T31391 C6SA9R 11552616 IC50 = 25600 nM T31391 C2DJ6Y 11552953 Ki = 27 nM T31391 CA16WP 11554165 IC50 = 4.8 nM T31391 CCFP45 11558852 IC50 = 205 nM T31391 CV74GT 11559033 Ki = 143 nM T31391 C85EQW 11559371 IC50 = 50 nM T31391 CDK7I5 11559922 Ki = 0.4 nM T31391 CIZ52M 11561317 Ki = 11 nM T31391 CJF19H 11564906 IC50 = 663 nM T31391 CTE30Z 11565791 IC50 = 164 nM T31391 CL4D9A 11565911 IC50 = 66 nM T31391 CMN2K0 11566106 IC50 = 564 nM T31391 CI5W4Y 11566450 IC50 = 106 nM T31391 CLU15X 11566865 IC50 = 454 nM T31391 C4QG9W 11567318 Ki = 1310 nM T31391 CR37GC 11567606 Ki = 2.9 nM T31391 CAR0J5 11567905 IC50 = 24 nM T31391 CR4I1P 11568333 Ki = 4.4 nM T31391 CL41DG 11569450 Ki = 4.6 nM T31391 CY0A7J 11570138 IC50 = 4.3 nM T31391 CW4LO8 11572237 IC50 = 40000 nM T31391 CH76QT 11572962 IC50 = 8 nM T31391 C8G7UP 11573204 Ki = 49 nM T31391 CHL5Y0 11573374 IC50 = 875 nM T31391 C6F4OE 11573417 IC50 = 132 nM T31391 CAE39I 11573427 IC50 = 84 nM T31391 CCR9Q2 11574031 IC50 = 317 nM T31391 C25SEL 11574694 IC50 = 29 nM T31391 CE03TL 11574811 Ki = 28 nM T31391 CQU80H 11576569 IC50 = 55 nM T31391 C7P0NT 11576820 Ki = 54 nM T31391 CW94NS 11577331 IC50 = 8 nM T31391 CQ86GI 11577431 IC50 = 4.1 nM T31391 CJV39M 11579395 Ki = 377 nM T31391 CW31KG 11579932 IC50 = 61 nM T31391 C0T9NU 11580126 IC50 > 3000 nM T31391 C7BJK9 11580332 IC50 > 30000 nM T31391 C7EA6G 11580446 IC50 > 30000 nM T31391 CVG3B6 11580945 IC50 = 447 nM T31391 CCR0D7 11581247 IC50 = 83 nM T31391 CYT4Z1 11581458 IC50 = 49 nM T31391 CA4XU3 11581644 IC50 = 210 nM T31391 C9J1NO 11581694 IC50 = 24 nM T31391 CS6X0E 11581890 IC50 = 128 nM T31391 CAZL49 11584650 IC50 = 13 nM T31391 CUS2H6 11587911 IC50 > 3000 nM T31391 COH9V8 11589872 IC50 = 2.8 nM T31391 C5JYV7 11591936 IC50 = 8 nM T31391 CSCW37 11592154 IC50 = 2.6 nM T31391 CDE3P6 11594121 IC50 = 33 nM T31391 C3NT1E 11594414 IC50 = 160 nM T31391 CA51WQ 11595401 IC50 = 33 nM T31391 CI0E4X 11595565 Ki = 2.2 nM T31391 CO0QJ8 11596007 Ki = 1530 nM T31391 CE8M3K 11596123 Ki = 67 nM T31391 C9MXO0 11596219 IC50 = 116 nM T31391 CW48NY 11596451 Ki = 6.7 nM T31391 CMUV42 11596607 IC50 = 5.2 nM T31391 CSW3M9 11597271 IC50 = 6.9 nM T31391 C9SC1G 11602166 IC50 = 9400 nM T31391 CY4W0X 11602707 IC50 = 11 nM T31391 CHM2N0 11602713 Ki = 317 nM T31391 C9CM7N 11603627 IC50 = 18 nM T31391 CBE6K8 11603637 Ki = 22 nM T31391 CPXV24 11603996 IC50 = 17 nM T31391 C9N2EZ 11604004 Ki = 6.8 nM T31391 CGAF90 11604063 IC50 = 3059 nM T31391 CL4NM7 11604454 IC50 = 676 nM T31391 C0S2RQ 11605368 IC50 = 4.6 nM T31391 C15DLO 11608317 IC50 > 33000 nM T31391 C5V1XM 11608625 IC50 > 3000 nM T31391 C9JZM7 11608919 IC50 > 3000 nM T31391 C6I0XG 11609419 IC50 = 1500 nM T31391 COF62W 11611325 Ki = 9 nM T31391 CAOP57 11612570 IC50 = 715 nM T31391 CQL5S8 11613750 IC50 = 6.2 nM T31391 CZ91WO 11616288 IC50 = 630 nM T31391 C27JCR 11616775 IC50 = 13600 nM T31391 C6MO9K 11616857 IC50 = 651 nM T31391 CD3YU1 11616861 IC50 = 74 nM T31391 CEX4O6 11617338 IC50 = 54 nM T31391 C7KS2Q 11617492 IC50 = 600 nM T31391 C40ZJT 11619382 IC50 = 73 nM T31391 C2APG7 11623550 IC50 = 72 nM T31391 CR8XO2 11623606 IC50 = 59 nM T31391 C7QC6U 11623777 Ki = 1280 nM T31391 C17XSP 11623929 Ki = 8.3 nM T31391 CPSN73 11624012 Ki = 20 nM T31391 CH2JP9 11624034 IC50 > 30000 nM T31391 CDZ72J 11624893 IC50 = 1108 nM T31391 CRY2D5 11625412 Ki = 50 nM T31391 C7YKC0 11628195 IC50 = 22 nM T31391 C5AKH1 11630368 IC50 = 2000 nM T31391 CYR61O 11630666 IC50 = 320 nM T31391 CV17GF 11631125 IC50 = 66 nM T31391 CA1J8U 11631434 IC50 = 3300 nM T31391 CH3WM8 11632024 IC50 = 8400 nM T31391 CSO1D6 11632159 Ki = 43 nM T31391 CZT57X 11632256 IC50 = 52 nM T31391 C8Y3FM 11632315 IC50 = 29 nM T31391 CM1DR9 11632375 Ki = 22 nM T31391 C09KAV 11632502 IC50 = 17 nM T31391 C7SP9Y 11634778 Ki > 3000 nM T31391 CR6NM8 11638575 Ki = 33 nM T31391 CM6QE9 11638687 IC50 > 3000 nM T31391 CHLA97 11638762 Ki = 241 nM T31391 CRA0H5 11639131 Ki = 550 nM T31391 C0M1HR 11640120 IC50 = 4.8 nM T31391 C5P3NB 11644467 IC50 = 56 nM T31391 C3RZO9 11645337 IC50 = 452 nM T31391 CQO8U6 11648011 Ki > 10000 nM T31391 CXG1B4 11649741 IC50 = 6.3 nM T31391 CO2YH1 11652954 Ki = 764 nM T31391 C1Y2DC 11652956 Ki = 867 nM T31391 CZBD50 11653749 Ki = 96 nM T31391 C94OMG 11654093 Ki = 18 nM T31391 C8AU5P 11654528 Ki = 38 nM T31391 CUX2M0 11654810 Ki = 7.2 nM T31391 C52ION 11655271 Ki = 19 nM T31391 CT4W8K 11659101 IC50 = 790 nM T31391 C7M6ZY 11659120 IC50 = 45200 nM T31391 CR8Z6I 11659133 IC50 > 30000 nM T31391 CZFV81 11661472 IC50 = 260 nM T31391 CI8EF3 11666622 IC50 > 3000 nM T31391 CN3WA7 11668525 IC50 > 3000 nM T31391 CE91WR 11669357 IC50 = 20 nM T31391 C43OVS 11673852 IC50 = 96 nM T31391 CCBS09 11674180 Ki = 64 nM T31391 CH1KG5 11674534 IC50 = 57 nM T31391 CTNO72 11674721 IC50 = 4.6 nM T31391 C2G6RP 11675637 Ki = 75 nM T31391 CI1ED9 11676224 IC50 = 150 nM T31391 C3Y7EL 11678025 IC50 = 5.2 nM T31391 C1A7NS 11680394 IC50 = 98 nM T31391 C5BD4Q 11680960 Ki = 12 nM T31391 CV0XW8 11680991 IC50 = 298 nM T31391 CFX6Z9 11681207 IC50 = 32 nM T31391 CNF1M4 11681778 IC50 = 50 nM T31391 C2K9XG 11688776 IC50 = 10 nM T31391 C0IWC9 11689866 IC50 = 651 nM T31391 CA69TN 11690566 IC50 = 77 nM T31391 C8UYQ5 11690713 IC50 = 2500 nM T31391 CC9O1L 11692537 Ki = 0.27 nM T31391 CEAN27 11694995 Ki = 1610 nM T31391 CBW6A1 11695523 IC50 = 6300 nM T31391 C79ECL 11695535 IC50 = 3236 nM T31391 C45QIU 11695818 IC50 = 2800 nM T31391 C7DCV9 11696495 Ki = 438 nM T31391 C6JPE0 11696912 Ki = 495 nM T31391 CRU2Q1 11697286 Ki = 5.6 nM T31391 C2WK1Z 11697387 Ki = 20 nM T31391 C1KCR6 11702577 IC50 = 15000 nM T31391 C2F6BA 11702880 Ki = 15 nM T31391 C8SI4E 11702902 IC50 = 119 nM T31391 C0Q3IL 11703158 IC50 = 784 nM T31391 C8IQA2 11703413 IC50 = 90 nM T31391 CUJ07L 11703663 Ki = 720 nM T31391 CJP1U8 11703749 IC50 = 1.5 nM T31391 C2X5GC 11704411 Ki = 9 nM T31391 C6YHK3 11704412 Ki = 24 nM T31391 CFO63Q 11704578 IC50 = 527 nM T31391 C1MGA4 11705197 Ki = 2.7 nM T31391 C8LA3E 11705712 Ki = 76 nM T31391 CU8LZ4 11705859 IC50 = 1418 nM T31391 CUC0Z3 11708771 IC50 = 400 nM T31391 CZF5D9 11708829 IC50 = 63 nM T31391 CNG85M 11710587 Ki = 8.9 nM T31391 CK4I6J 11710700 Ki = 6 nM T31391 C0CG5R 11710963 IC50 = 42 nM T31391 C04OMI 11711314 Ki = 113 nM T31391 C8VC2D 11711413 Ki = 33 nM T31391 C8KD6N 11711414 Ki = 163 nM T31391 C0U7QC 11715518 IC50 = 105 nM T31391 C34BEP 11716483 Ki = 12 nM T31391 CMI90R 11716843 Ki = 3.4 nM T31391 CCR80L 11717090 IC50 = 116 nM T31391 CZS71R 11717268 IC50 = 369 nM T31391 C1XD5I 11718004 Ki = 113 nM T31391 C1M7PL 11718857 Ki = 30 nM T31391 CY1S3Q 11719625 IC50 = 2.8 nM T31391 C0UJ7G 11719823 IC50 = 910 nM T31391 CIEJ54 11720809 IC50 = 5.3 nM T31391 CHA7Z9 11722557 IC50 = 119 nM T31391 CIOY84 11723708 IC50 = 21.3 ug.mL-1 T31391 C6VG7O 11727562 IC50 = 989 nM T31391 CJ6XR8 11730284 IC50 > 125000 nM T31391 CX9U4G 11731880 IC50 = 503000 nM T31391 C96TGJ 11746838 IC50 = 988 nM T31391 CA2H1U 11747757 IC50 = 163 nM T31391 C3ZPG6 11772582 IC50 = 68 nM T31391 CX84PY 11772583 IC50 = 590 nM T31391 C1P9ZM 11776124 IC50 > 1000000 nM T31391 C6JY7V 11776638 Ki = 8 nM T31391 CS0WM6 11778955 IC50 = 320 nM T31391 C3MX2I 11781105 IC50 = 24 nM T31391 CO73AL 11784400 IC50 = 15000 nM T31391 CKTJ04 11791651 IC50 = 291 nM T31391 C67TXV 11791652 IC50 = 109000 nM T31391 C1P2AI 11809137 IC50 = 102 nM T31391 C6ET2R 11817181 IC50 = 43500 nM T31391 CK24XY 11819467 IC50 > 1000000 nM T31391 C19HAP 11825584 IC50 = 89000 nM T31391 CN79VL 11840913 Ki = 6.7 nM T31391 CSOC43 11840914 Ki = 0.82 nM T31391 CE6V2H 11840916 Ki = 3.8 nM T31391 C42BOS 11854299 IC50 = 56.9 nM T31391 C2FN7G 11854301 IC50 = 53.4 nM T31391 CQ0O5A 11952574 IC50 = 120 nM T31391 CQIB43 11957945 IC50 = 82 nM T31391 CTQI92 11974546 Ki = 45 nM T31391 C5BZW6 11998979 Ki = 140 nM T31391 CXHC16 11999086 Ki = 240 nM T31391 CU3HD8 11999088 Ki = 190 nM T31391 CLI17Z 11999090 Ki = 220 nM T31391 C8U5NY 11999093 Ki = 15 nM T31391 CBZ03A 11999206 Ki = 76 nM T31391 C2TAJ9 11999207 Ki = 200 nM T31391 C3E4ZB 11999208 Ki = 34 nM T31391 C6DK9R 11999211 Ki = 35 nM T31391 CQSP03 12043866 IC50 = 207000 nM T31391 C35DEQ 12043867 IC50 = 3400 nM T31391 C1P3MJ 12043868 IC50 = 18000 nM T31391 C7NRQ3 12043869 IC50 = 731000 nM T31391 CAI8E7 12043870 IC50 = 51400 nM T31391 C21PAF 12069363 IC50 = 0.6 nM T31391 CQY50P 12742483 IC50 = 250000 nM T31391 C9RA7N 13478499 Ki = 160000 nM T31391 CYV1F7 13784835 IC50 > 100 ug.mL-1 T31391 C1GF7B 13939278 IC50 = 750 nM T31391 C94FPE 14434173 IC50 > 100 ug.mL-1 T31391 CR8H4L 14978092 IC50 = 200 nM T31391 CJAE28 15036410 IC50 = 118000 nM T31391 C6BHJ9 15101668 IC50 > 1000000 nM T31391 C29IHT 15337406 IC50 = 16000 nM T31391 CNM5V2 15940321 IC50 = 32360 nM T31391 C2ZMH8 15948988 IC50 = 25.4 nM T31391 C13JIX 15949418 IC50 = 0.67 nM T31391 C49NUJ 15949507 IC50 = 5.3 nM T31391 CPD3V1 15949508 IC50 = 0.5 nM T31391 CU4P5X 15950383 Ki = 3 nM T31391 C16XRI 15950384 Ki = 51.5 nM T31391 CUMR27 15950385 Ki = 11 nM T31391 C69RAY 15950386 Ki = 9 nM T31391 CM63YP 15950387 Ki = 29 nM T31391 CH8F7W 15950388 Ki = 4 nM T31391 C0L4SH 15950456 Ki = 14 nM T31391 C8G7OJ 15950457 Ki = 12 nM T31391 C8FU1V 15950462 Ki = 29 nM T31391 C9KJ6D 15950538 Ki = 2.7 nM T31391 C3C6PM 15950539 Ki = 9 nM T31391 C4S7AB 15950540 Ki = 4 nM T31391 C2HGJ0 15950541 Ki = 16 nM T31391 C3U1VO 15950542 Ki = 9 nM T31391 CKX8M6 15950615 Ki = 4 nM T31391 CC0M2X 15951427 Ki = 8 nM T31391 CF3PX0 15951428 Ki = 30 nM T31391 CWTX01 15951429 Ki = 12 nM T31391 C3LQD9 15951431 Ki = 18 nM T31391 C8M0FT 15951543 IC50 = 27 nM T31391 CI3DB4 15951636 IC50 > 20000 nM T31391 C3SM4T 15951642 IC50 > 100000 nM T31391 C8QRV9 15951839 Ki = 38400 nM T31391 CMNT83 15951928 Ki = 608000 nM T31391 CL1E6O 15953860 IC50 = 17 nM T31391 CG2E3Z 15991577 IC50 = 84 nM T31391 CLG2Q1 16035093 IC50 = 24 nM T31391 CMUG74 16035094 IC50 = 25 nM T31391 CYPG43 16040279 Ki = 3.2 nM T31391 C13-MAR 16040457 IC50 > 100000 nM T31391 C0YQ9A 16046127 IC50 = 325000 nM T31391 C75ZNE 16058650 Ki = 4 nM T31391 C28IRJ 16064807 IC50 = 17 nM T31391 C4LJH3 16064808 IC50 = 24 nM T31391 CVIC15 16064809 IC50 = 11 nM T31391 CS7DQ3 16090844 Ki = 3 nM T31391 C8CVG9 16090856 Ki = 1.3 nM T31391 CB6WK0 16121107 Ki = 170000 nM T31391 CZQ8O9 16121199 Ki = 100000 nM T31391 C5Q9BH 16122596 IC50 = 16 nM T31391 CU3GB5 16126742 IC50 = 4.8 nM T31391 CUQT90 16202787 Ki = 12 nM T31391 CHUX72 16202788 Ki = 3.8 nM T31391 C8D2RM 16203032 Ki = 1400 nM T31391 CW0JF5 16203033 Ki = 17 nM T31391 C5F6DE 16203034 Ki = 590 nM T31391 C0LJA8 16203036 Ki = 105 nM T31391 CC20IT 16203037 Ki = 4 nM T31391 CW6AC3 16203151 Ki = 6 nM T31391 C5BE1I 16204461 Ki = 1600 nM T31391 CWY50B 16204462 Ki = 930 nM T31391 CAQ7S4 16204463 Ki = 440 nM T31391 CCW34I 16204464 Ki = 270 nM T31391 CCWF31 16204465 Ki = 83 nM T31391 C73HLC 16204466 Ki = 24 nM T31391 CA1PV5 16216352 IC50 > 33000 nM T31391 CD9MQ6 16223559 IC50 = 245 nM T31391 CQ7G8T 16223560 IC50 = 1.7 nM T31391 CN24YP 16223762 IC50 = 984 nM T31391 CF37TH 16226604 IC50 = 84 nM T31391 C6ANU2 16226605 IC50 = 109 nM T31391 CFW43X 16658022 IC50 = 5 nM T31391 C6H5VO 16658023 IC50 = 5 nM T31391 CC9W4S 16658024 IC50 = 15 nM T31391 CR51WX 16658101 IC50 = 13 nM T31391 CMLR19 16658102 IC50 = 5 nM T31391 CXN32U 16658103 IC50 = 8 nM T31391 C2XP7B 16658104 IC50 = 4 nM T31391 CD6L7Z 16658105 IC50 = 19 nM T31391 C63NWG 16658243 IC50 < 10 nM T31391 C82ZAL 16658881 IC50 = 460 nM T31391 C24NZK 16658917 Ki = 2.3 nM T31391 C28GEM 16662696 IC50 = 1.1 nM T31391 C53XZP 16721117 Ki = 2 nM T31391 CW62MC 16725327 IC50 = 1.3 nM T31391 C0EV4T 16725905 IC50 = 5 nM T31391 C56LTN 16739329 IC50 = 0.92 nM T31391 CT01PQ 16739331 IC50 = 70 nM T31391 C19UBP 16747699 IC50 = 13 nM T31391 C9JK5Q 16750059 Ki = 5.3 nM T31391 C61RFP 16755651 Ki = 13 nM T31391 C4RK2Q 17591662 IC50 = 94.82 nM T31391 CU05RG 17748274 IC50 = 16 nM T31391 C15TBF 17751406 IC50 = 15000 nM T31391 C5W3VY 17753031 IC50 = 76 nM T31391 CX5F2U 17763521 IC50 > 500000 nM T31391 CQG89Z 17853548 IC50 = 41400 nM T31391 C6L7MA 18391459 IC50 = 2.9 nM T31391 CV4Z6Q 18398587 IC50 = 134900 nM T31391 CP3S0V 18398588 IC50 = 247000 nM T31391 C7GDU9 20038035 IC50 > 100 ug.mL-1 T31391 CC8RN3 20198196 IC50 = 18100 nM T31391 CT42AI 20706081 IC50 = 330 nM T31391 CBZ1E6 21045424 IC50 = 765 nM T31391 C6ZMS8 21054400 Ki = 5 nM T31391 CWB93R 21054485 IC50 = 21 nM T31391 CBY6M2 21919450 IC50 = 142 nM T31391 CH7YL4 21919455 IC50 = 10000 nM T31391 C1PF7M 21919463 IC50 = 2200 nM T31391 C39STQ 21919469 IC50 = 1150 nM T31391 C2OXL1 21919478 IC50 = 13 nM T31391 CY8OJ7 21947630 IC50 = 26 nM T31391 CQ9LB5 21947637 IC50 = 89 nM T31391 CCFX26 21947643 IC50 = 7 nM T31391 C3SXF7 21947646 IC50 = 4 nM T31391 CPES59 21949259 IC50 = 190000 nM T31391 C2W4KV 21949272 IC50 = 67000 nM T31391 CZ9K4Q 22029435 IC50 = 580 nM T31391 C0X4SO 22029457 IC50 = 340 nM T31391 CLK4G6 22029894 IC50 = 1230 nM T31391 C6BME5 22175258 IC50 = 1100 nM T31391 CRA87P 22175262 IC50 = 360 nM T31391 C7E0NG 22175290 IC50 = 2400 nM T31391 C2SD9C 22175298 IC50 = 2400 nM T31391 CQ3EB8 22175361 IC50 = 47 nM T31391 C56RIP 22175474 IC50 = 1900 nM T31391 C28HMT 22175479 IC50 = 1100 nM T31391 CK4NR7 22175497 IC50 = 1200 nM T31391 C2ME4A 22175534 IC50 = 870 nM T31391 C2RM7H 22175568 IC50 = 980 nM T31391 C7X5DS 22175618 IC50 = 3800 nM T31391 CE3LM6 22175639 IC50 = 250 nM T31391 CLUH89 22175659 IC50 = 4000 nM T31391 C4AUK1 22175709 IC50 = 8300 nM T31391 C6KGB8 22175713 IC50 = 220 nM T31391 CBYP16 22175758 IC50 = 250 nM T31391 CB38EC 22176094 IC50 = 1500 nM T31391 CR23XQ 22176165 IC50 = 2400 nM T31391 C8QF7T 22176298 IC50 = 1900 nM T31391 CUND82 22176405 IC50 = 1600 nM T31391 CL68SA 22220623 IC50 = 80000 nM T31391 C2XAR9 22401333 IC50 > 100000 nM T31391 CED47V 22690988 IC50 = 24000 nM T31391 C9VGC8 22691359 IC50 > 100000 nM T31391 C43XCK 22691633 Ki = 5300 nM T31391 C1M2ZS 22691666 IC50 > 100000 nM T31391 CM4SH2 23595882 IC50 = 167000 nM T31391 CP1J3T 23596395 Ki = 14 nM T31391 C8JSI4 23628284 IC50 = 50 nM T31391 CC29GD 23633277 IC50 = 0.5 nM T31391 C1RV7P 23633348 IC50 = 17 nM T31391 CU1LK3 23633350 IC50 = 1.5 nM T31391 CKN67W 23633553 IC50 = 6 nM T31391 CG37EL 23633557 IC50 = 7 nM T31391 C5U3NL 23633697 IC50 = 9 nM T31391 CVC80Z 23633837 IC50 = 10 nM T31391 C8P9GL 23633839 IC50 = 400 nM T31391 C5UVZ9 23634061 IC50 = 60 nM T31391 C5ZF2X 23634210 IC50 = 25 nM T31391 C4KW2T 23634279 IC50 = 4 nM T31391 CVF78O 23634281 IC50 = 4 nM T31391 CA95UP 23634434 IC50 = 8.4 nM T31391 C7FSW5 23634528 IC50 > 36900 nM T31391 CAQ81M 23644660 IC50 = 455 nM T31391 CDPU25 23644665 IC50 = 7360 nM T31391 CCSU21 23645371 IC50 = 27 nM T31391 C5M6UX 23645373 Ki = 470 nM T31391 CFS6P4 23645374 Ki = 20 nM T31391 CAVN39 23645375 Ki = 26 nM T31391 CN0FR1 23645376 Ki = 3.1 nM T31391 CVQ39W 23645377 Ki = 5.3 nM T31391 CQPA42 23645378 Ki = 36 nM T31391 CQ5R2G 23645379 Ki = 360 nM T31391 C32KIA 23645380 Ki = 1160 nM T31391 C6TCN1 23645381 Ki > 12800 nM T31391 CL08ZV 23645382 Ki > 12800 nM T31391 C8P3OQ 23645383 Ki > 12800 nM T31391 C72KLP 23645384 Ki = 980 nM T31391 CNVP26 23645385 Ki = 360 nM T31391 C3OHM9 23645386 Ki = 310 nM T31391 C8TP3W 23645387 Ki = 166 nM T31391 CZXL64 23645388 Ki = 160 nM T31391 C7MAX0 23645389 Ki = 170 nM T31391 C7W6PC 23645390 Ki = 96 nM T31391 CX0VJ4 23645391 Ki = 8900 nM T31391 C4EM3K 23645392 Ki > 12800 nM T31391 CU76EP 23645393 Ki > 12800 nM T31391 CFV07G 23645410 IC50 = 231 nM T31391 CIMG82 23645411 IC50 = 68 nM T31391 C47OZL 23645510 IC50 = 520 nM T31391 C2Q5IK 23645581 IC50 = 48 nM T31391 C3VA0M 23645582 IC50 = 968 nM T31391 C1JAG6 23645622 IC50 = 110 nM T31391 CDL4G9 23645678 Ki = 2.1 nM T31391 CL1DC7 23645680 Ki = 1.8 nM T31391 C23BMA 23645681 IC50 = 170000 nM T31391 C4B9FM 23645685 Ki = 1 nM T31391 CP9GS5 23645686 IC50 = 19700 nM T31391 C6R2LP 23645687 IC50 = 1820 nM T31391 CN7FK3 23645688 IC50 = 12400 nM T31391 CSHX17 23645689 IC50 = 4790 nM T31391 CL8QV6 23645690 IC50 = 4820 nM T31391 C0AU9X 23645691 IC50 = 990 nM T31391 CRM3Y4 23645692 IC50 = 15600 nM T31391 CDM8A2 23645693 IC50 = 3820 nM T31391 CIR1F6 23645694 IC50 = 1790 nM T31391 CK5G6I 23645695 IC50 = 1610 nM T31391 CHS76O 23645696 IC50 = 330 nM T31391 CVP59D 23645697 IC50 = 190 nM T31391 CH13BW 23645698 IC50 = 122 nM T31391 CL0K1T 23645699 IC50 = 520 nM T31391 CB3Z7O 23645700 IC50 = 4590 nM T31391 CNO6Q1 23645702 IC50 = 160 nM T31391 CGMC54 23645703 IC50 = 830 nM T31391 C0V4WR 23645705 IC50 = 43 nM T31391 CY9XW5 23645721 IC50 = 40 nM T31391 C5MO2Q 23645882 Ki = 260 nM T31391 C1UR3L 23645883 Ki = 507 nM T31391 C5EQ1C 23645884 Ki > 10000 nM T31391 CO90SF 23645885 Ki = 212 nM T31391 C85TUY 23645886 Ki = 1311 nM T31391 CBNC76 23645887 Ki = 140 nM T31391 CE1H2R 23645888 Ki = 513 nM T31391 CR7C8Q 23645889 Ki > 10000 nM T31391 CSW5F3 23645890 Ki = 4422 nM T31391 C7E8AI 23645891 Ki > 10000 nM T31391 C8YGE5 23645892 Ki = 399 nM T31391 C31TSP 23645893 Ki > 10000 nM T31391 C87LMT 23645894 Ki > 10000 nM T31391 CX79LQ 23645895 Ki = 74 nM T31391 CON27H 23645896 Ki = 27 nM T31391 CAYT68 23645897 Ki = 673 nM T31391 C5SH6W 23645898 Ki = 37 nM T31391 CDFZ57 23645899 Ki = 188 nM T31391 C5XB6V 23645900 Ki > 10000 nM T31391 CS6WQ4 23645901 Ki = 18 nM T31391 C9AZD2 23645902 Ki = 3 nM T31391 C2O6ML 23645903 Ki = 23 nM T31391 CKM6Y8 23645917 IC50 = 250 nM T31391 C9Y2ZL 23645918 IC50 = 110 nM T31391 C4V6BX 23645919 IC50 = 130 nM T31391 C78PNU 23645920 IC50 = 150 nM T31391 C5YT6S 23645921 IC50 = 180 nM T31391 CELQ89 23645922 IC50 = 150 nM T31391 CGV92H 23645923 IC50 = 350 nM T31391 CJ60EH 23645924 IC50 = 160 nM T31391 CZG70A 23645925 IC50 = 160 nM T31391 CD6V7X 23645926 IC50 = 220 nM T31391 C1TD4J 23645927 IC50 = 300 nM T31391 C71PQU 23645928 IC50 = 270 nM T31391 C8EOB9 23645929 IC50 = 780 nM T31391 C0M1TH 23645930 IC50 = 150 nM T31391 CFHB36 23645931 IC50 = 130 nM T31391 CTG27F 23645932 IC50 = 39 nM T31391 CS2FT5 23645933 IC50 = 72 nM T31391 C98QGK 23645934 IC50 = 160 nM T31391 CS76DY 23645935 IC50 = 130 nM T31391 C91MYK 23645936 IC50 = 85 nM T31391 C3AQC0 23645937 IC50 = 590 nM T31391 C61GTC 23645938 IC50 = 480 nM T31391 C8XF6R 23645939 IC50 = 310 nM T31391 C7IX5B 23645940 IC50 = 360 nM T31391 CP6M3W 23645941 IC50 = 260 nM T31391 CQ75XK 23645942 IC50 = 380 nM T31391 C8T7GY 23645943 IC50 = 130 nM T31391 C25ZXC 23645944 IC50 = 290 nM T31391 C4A3NI 23645945 IC50 = 180 nM T31391 C9Y1BP 23646016 IC50 = 73 nM T31391 CL8DY2 23646017 IC50 = 73 nM T31391 CT6Q1R 23646018 IC50 = 72 nM T31391 C8VS1X 23646019 IC50 = 144 nM T31391 CL4BX5 23646020 IC50 = 4130 nM T31391 CZ24WC 23646021 IC50 = 1957 nM T31391 C98VYW 23646022 IC50 = 2587 nM T31391 CCL17M 23646023 IC50 = 228 nM T31391 CT16HE 23646024 IC50 = 129 nM T31391 CAL8T5 23646025 IC50 = 63 nM T31391 CVSH12 23646026 IC50 = 274 nM T31391 C15HJB 23646027 IC50 > 100000 nM T31391 CBUM54 23646029 IC50 > 100000 nM T31391 C32ZNH 23646030 IC50 = 31000 nM T31391 CE8L2I 23646031 Ki = 64 nM T31391 C8SIU2 23646032 IC50 > 100000 nM T31391 C7L6JR 23646033 IC50 > 100000 nM T31391 CJ9ZL3 23646080 IC50 > 1000000 nM T31391 C0S2UB 23646081 IC50 > 1000000 nM T31391 CQ3KF6 23646082 IC50 > 1000000 nM T31391 CZ9P0Q 23646083 IC50 > 1000000 nM T31391 CFPN10 23646084 IC50 > 1000000 nM T31391 C0NV1B 23646085 IC50 > 1000000 nM T31391 CSW9T1 23646086 IC50 > 250000 nM T31391 CH72RP 23646087 IC50 > 1000000 nM T31391 CH5Y2F 23646088 IC50 > 500000 nM T31391 CJ47OR 23646089 IC50 > 250000 nM T31391 CRT2B0 23646090 IC50 > 250000 nM T31391 C7JXN0 23646091 IC50 > 1000000 nM T31391 C4K1NE 23646092 IC50 > 250000 nM T31391 CJV2K1 23646093 IC50 > 250000 nM T31391 C51BSR 23646094 IC50 > 250000 nM T31391 C2WDG4 23646095 IC50 > 125000 nM T31391 CB2ZT7 23646096 IC50 > 1000000 nM T31391 COF57U 23646097 IC50 > 1000000 nM T31391 CU26YP 23646098 IC50 > 250000 nM T31391 CM37ZS 23646100 IC50 > 1000000 nM T31391 C4SV2J 23646101 IC50 > 1000000 nM T31391 CX68KV 23646102 IC50 > 1000000 nM T31391 CZ28UC 23646142 Ki = 62 nM T31391 CLA15H 23646143 Ki = 4 nM T31391 C0EK5I 23646441 IC50 = 7.2 nM T31391 CF1TP9 23646442 IC50 = 160 nM T31391 CZA78Q 23646443 IC50 = 89 nM T31391 C5VP2I 23646444 IC50 = 14 nM T31391 C9PW1E 23646445 IC50 = 150 nM T31391 CAI0B5 23646446 IC50 = 2300 nM T31391 C4XM2W 23646447 IC50 = 67000 nM T31391 CUZ0D8 23646448 IC50 = 142 nM T31391 C7PE0S 23646449 IC50 = 16 nM T31391 COT87G 23646450 IC50 = 0.91 nM T31391 CF2J9Q 23646451 IC50 = 0.49 nM T31391 CVHU93 23646508 Ki = 9 nM T31391 CJLP47 23646509 Ki = 10 nM T31391 C7P5TW 23646510 Ki = 22 nM T31391 C61FRE 23646511 Ki = 1200 nM T31391 C4EG5D 23646512 Ki = 11 nM T31391 CN47RA 23646513 Ki = 29 nM T31391 CDM3J0 23646514 Ki = 25 nM T31391 CW0J6X 23646515 Ki = 57 nM T31391 CS6L8X 23646516 Ki = 300 nM T31391 COPD36 23646517 Ki = 260 nM T31391 CWT7X1 23646518 Ki = 450 nM T31391 C5GQ7J 23646519 Ki = 11 nM T31391 C0E8SM 23647079 IC50 = 280 nM T31391 CA6X5F 23647080 IC50 = 39 nM T31391 CP2W3B 23647081 IC50 = 3800 nM T31391 CS8O6P 23647082 IC50 = 820 nM T31391 CA53BK 23647084 IC50 = 110 nM T31391 CK15XF 23647085 IC50 = 340 nM T31391 CFOA63 23647106 IC50 = 13 nM T31391 CRF32I 23647107 IC50 = 5 nM T31391 CFTW63 23647114 IC50 = 20.7 nM T31391 C0BQ2D 23647115 IC50 = 11.6 nM T31391 CLO1Y2 23647116 IC50 = 69.9 nM T31391 CSJ78F 23647117 IC50 = 9 nM T31391 CDE9L7 23647118 IC50 = 11.5 nM T31391 CZF25M 23647119 IC50 = 15.1 nM T31391 CW5U3C 23647120 IC50 = 10.5 nM T31391 CWO62C 23647121 IC50 = 19.2 nM T31391 C0X1CK 23647122 IC50 = 8 nM T31391 C7JOV9 23647123 IC50 = 33 nM T31391 C0UT7J 23647124 IC50 = 397 nM T31391 C8P2VJ 23647125 IC50 = 37.3 nM T31391 CQ85KB 23647126 IC50 = 60.3 nM T31391 CRFL12 23647127 IC50 = 24.6 nM T31391 CP3CF0 23647128 IC50 = 143 nM T31391 CJA3M7 23647129 IC50 = 142 nM T31391 C7L3RX 23647130 IC50 = 11 nM T31391 C8UWB7 23647132 IC50 = 29.6 nM T31391 C60MWC 23647133 IC50 = 126 nM T31391 C8TZD5 23647134 IC50 = 2 nM T31391 CBA8N1 23647136 IC50 = 21 nM T31391 CG0U2M 23647137 IC50 = 33 nM T31391 C3TSN4 23647138 IC50 = 37 nM T31391 C6QKM4 23647139 IC50 = 310 nM T31391 CQPN26 23647141 IC50 = 780 nM T31391 C4V5TC 23647142 IC50 = 995 nM T31391 C8TDA5 23647143 IC50 = 1247 nM T31391 CNRH86 23647144 IC50 = 1325 nM T31391 CY19JV 23647145 IC50 = 1460 nM T31391 C39DJX 23647146 IC50 = 1995 nM T31391 C4P2IJ 23647147 IC50 = 2209 nM T31391 CTB09J 23647311 IC50 = 13 nM T31391 CJ6XT7 23647314 IC50 = 18 nM T31391 CVI19F 23653088 IC50 = 3800 nM T31391 CO9GD8 23655077 IC50 = 22 nM T31391 CWVR37 23655298 IC50 > 500000 nM T31391 CPCX60 23655474 IC50 > 1000000 nM T31391 CB1E5P 23655476 IC50 > 500000 nM T31391 CWTD09 23655478 IC50 > 1000000 nM T31391 CLSE92 23655741 IC50 > 40200 nM T31391 CQ53MU 23655742 IC50 > 36900 nM T31391 C4DOR0 23655937 IC50 > 41300 nM T31391 CRA46X 23655938 IC50 > 39100 nM T31391 CW9UR3 23657402 IC50 > 250000 nM T31391 CU18EA 23657547 IC50 > 250000 nM T31391 CVF6E2 23661697 IC50 = 25 nM T31391 CM7C4W 23661708 IC50 = 26 nM T31391 CO6L9F 23661716 IC50 = 1.2 nM T31391 CHR14F 23661718 IC50 = 6 nM T31391 CG8TJ9 23824719 IC50 = 11000 nM T31391 CNP9T1 24180585 IC50 = 37 nM T31391 CO0ZA3 24692381 IC50 = 67000 nM T31391 CR7I3Y 24703639 IC50 > 1000000 nM T31391 CVA72K 24704198 IC50 = 374000 nM T31391 CKWZ51 24710701 IC50 = 360000 nM T31391 CKVQ51 24749924 IC50 = 1 nM T31391 CCW9N3 24749925 IC50 = 4 nM T31391 CXNY61 24749926 IC50 = 4 nM T31391 CZ4BH0 24749927 IC50 = 284 nM T31391 C9X8CK 24750044 IC50 = 5 nM T31391 CK7V6L 24750165 IC50 = 56 nM T31391 C7I4LK 24750278 IC50 = 3 nM T31391 CT21RV 24750279 IC50 = 2 nM T31391 CC6X1F 24750280 IC50 = 88 nM T31391 C5TIP2 24750281 IC50 = 9 nM T31391 C7QSH2 24752844 IC50 = 65 nM T31391 CI0W8A 24755210 IC50 = 1.3 nM T31391 CU7W4F 24768547 IC50 = 0.21 nM T31391 CX8DH1 24769723 IC50 = 1.4 nM T31391 C0H8OB 24776705 IC50 = 116 nM T31391 C24GLZ 24776939 IC50 = 0.18 nM T31391 C6LD2J 24777439 IC50 = 209 nM T31391 CK8EL5 24777568 IC50 = 12 nM T31391 CQ20PV 24777692 IC50 = 88 nM T31391 C1WF3I 24777804 IC50 = 4.3 nM T31391 C50SPA 24784161 IC50 = 123 nM T31391 C29SZR 24784416 IC50 = 90000 nM T31391 C0H8IZ 24784426 IC50 = 116 nM T31391 CO7L6R 24784427 IC50 = 73 nM T31391 C8FQT4 24784664 IC50 > 100000 nM T31391 C69QMZ 24784674 IC50 = 238 nM T31391 CW8LK2 24784675 IC50 = 47 nM T31391 CH1W5N 24784676 IC50 = 140 nM T31391 CJ0ZI7 24784677 IC50 = 251 nM T31391 CIZF59 24784915 IC50 = 72 nM T31391 CKFH56 24784916 IC50 = 195 nM T31391 C5HY0P 24784918 IC50 = 212 nM T31391 CS6HU2 24784925 IC50 = 182 nM T31391 CK6W8S 24784926 IC50 = 45 nM T31391 CUH32V 24785152 IC50 = 305 nM T31391 C2KL7G 24794725 IC50 = 63 nM T31391 CUM03S 24798754 IC50 = 0.12 nM T31391 CZ3ND1 24832041 IC50 = 32 nM T31391 CY9W8O 24860300 IC50 = 1 nM T31391 CKZ25G 24862861 IC50 = 7.5 nM T31391 CFNZ09 24893980 IC50 = 3670 nM T31391 CMK9B7 24894026 IC50 > 100000 nM T31391 CSIK84 24906298 IC50 = 500000 nM T31391 CYL69J 24951732 IC50 = 0.7 nM T31391 CNP3T1 24951733 IC50 = 3.7 nM T31391 CDCP18 24952087 IC50 = 7.3 nM T31391 CIM7S2 24952089 IC50 = 3.5 nM T31391 CX83WL 24963343 IC50 > 100000 nM T31391 CDU69X 24999325 IC50 = 50 nM T31391 CA94RD 24999327 IC50 = 9 nM T31391 CZJ2N6 24999330 IC50 = 24 nM T31391 C9ML5P 24999630 IC50 = 14 nM T31391 C3VU2K 24999632 IC50 = 69 nM T31391 CUO7Q4 24999636 IC50 = 120 nM T31391 CM6AW8 24999638 IC50 = 39 nM T31391 CY90LJ 25014552 IC50 = 2740 nM T31391 CA28YZ 25017799 IC50 = 2.28 nM T31391 C40ONC 25021195 IC50 = 223 nM T31391 C67ZQD 25054021 IC50 = 357 nM T31391 C3SW1V 25054553 IC50 = 64 nM T31391 CH9F2B 25054555 IC50 = 64 nM T31391 CHO68D 25054557 IC50 = 56 nM T31391 C3R9XM 25054809 IC50 = 50 nM T31391 C2D4LI 25054811 IC50 = 3 nM T31391 CHE83A 25054815 IC50 = 13 nM T31391 CXPO63 25054817 IC50 = 68 nM T31391 CA2EK8 25055067 IC50 = 328 nM T31391 C8J9ZG 25055304 IC50 = 80 nM T31391 C51KTQ 25055741 IC50 = 7.4 nM T31391 CI0K2T 25055743 IC50 = 4.3 nM T31391 C1Q6RS 25055745 IC50 = 2.2 nM T31391 CIA48J 25055828 IC50 = 204 nM T31391 CA3N5B 25055836 IC50 = 229 nM T31391 CEDP80 25055999 IC50 = 1.7 nM T31391 C5K3QM 25056001 IC50 = 11 nM T31391 CGX3K8 25056003 IC50 = 17 nM T31391 C6X9PG 25056005 IC50 = 5.2 nM T31391 C8P7VJ 25056091 IC50 = 601 nM T31391 CN83UK 25056093 IC50 = 77 nM T31391 C0LJF5 25056353 IC50 = 6 nM T31391 CS81DK 25056618 IC50 = 112 nM T31391 CQM3U1 25056620 IC50 = 192 nM T31391 C7WEY3 25056875 IC50 = 807 nM T31391 C62UCV 25056881 IC50 = 95 nM T31391 CK7B2E 25057130 IC50 = 102 nM T31391 CQCY54 25057136 IC50 = 25 nM T31391 CM3AU5 25057138 IC50 = 17 nM T31391 CR26DS 25057390 IC50 = 309 nM T31391 C8Q2GP 25057392 IC50 = 175 nM T31391 C9TQ7J 25057396 IC50 = 680 nM T31391 C6KHT4 25057400 IC50 = 1700 nM T31391 C6Q2CM 25057648 IC50 = 88 nM T31391 C1RN5F 25057650 IC50 = 101 nM T31391 CUF2P9 25057652 IC50 = 212 nM T31391 CQHM69 25110577 IC50 = 510 nM T31391 CTS7I5 25110685 IC50 = 3.6 nM T31391 CHTM74 25110898 IC50 = 2500 nM T31391 CBC24W 25110901 IC50 = 8500 nM T31391 CW3GZ6 25112031 IC50 = 710 nM T31391 C76RFD 25112033 IC50 = 2200 nM T31391 CYV1T4 25112035 IC50 = 1900 nM T31391 CW7UD1 25112037 IC50 = 1600 nM T31391 CX9NR5 25112039 IC50 = 3000 nM T31391 CN2MQ8 25112155 IC50 = 770 nM T31391 CO7UE8 25112157 IC50 = 3700 nM T31391 CUIW48 25112159 IC50 = 3100 nM T31391 C6B8CF 25112161 IC50 = 2000 nM T31391 CQ0GY8 25112163 IC50 = 1600 nM T31391 CI71VQ 25112265 IC50 = 8900 nM T31391 CR13HD 25112267 IC50 = 1900 nM T31391 CWE10R 25112269 IC50 = 3600 nM T31391 CK69WG 25112271 IC50 = 1400 nM T31391 C5W8KL 25112273 IC50 = 5900 nM T31391 CXM0N5 25112374 IC50 = 2800 nM T31391 CK16JS 25112376 IC50 = 4300 nM T31391 C9KF5T 25112378 IC50 = 2200 nM T31391 C5O9PU 25112380 IC50 = 2700 nM T31391 C19DPQ 25112382 IC50 = 1400 nM T31391 CYJ2B5 25112487 IC50 = 2700 nM T31391 CUA2K9 25112489 IC50 = 1600 nM T31391 C60EOS 25112491 IC50 = 5600 nM T31391 CV75BU 25112493 IC50 = 1600 nM T31391 CDL2S7 25112495 IC50 = 7400 nM T31391 CF97YP 25112497 IC50 = 1300 nM T31391 CDKE79 25112619 IC50 = 2100 nM T31391 C4TLZ7 25112621 IC50 = 9100 nM T31391 CI3KP5 25112623 IC50 = 690 nM T31391 CF9BO5 25112625 IC50 = 4800 nM T31391 C5QA1K 25112627 IC50 = 2600 nM T31391 C01GPL 25132159 Ki = 8.3 nM T31391 C7IDX9 25132160 IC50 = 0.89 nM T31391 C9VK8W 25132161 Ki = 17 nM T31391 CFZ4V2 25132162 Ki = 3300 nM T31391 CSU0B5 25189891 Ki = 14.4 nM T31391 CA98HO 25203967 IC50 = 2000 nM T31391 CPMN48 28787393 IC50 = 6.29 nM T31391 C9Q2OH 42601533 IC50 = 3850 nM T31391 C0BC9N 42601535 IC50 = 350 nM T31391 C7KN2U 42608447 IC50 = 0.38 nM T31391 C60SVD 42636924 IC50 = 15 nM T31391 C76NLT 42773972 IC50 > 250000 nM T31391 C6LQN3 43181622 IC50 > 1000000 nM T31391 C42OZD 43271345 IC50 = 377000 nM T31391 CK54OM 43650152 IC50 = 229000 nM T31391 CS40ML 44123747 IC50 = 1.1 nM T31391 CSX10M 44138030 IC50 = 4 nM T31391 CQF86D 44182505 IC50 = 13 nM T31391 C3I4TF 44201003 IC50 = 10 nM T31391 CE5B7H 44218404 IC50 = 13 nM T31391 CR8GT4 44218550 IC50 = 15 nM T31391 CBW7D4 44218551 IC50 = 39 nM T31391 CVH08B 44218552 IC50 = 18 nM T31391 CISE95 44218553 IC50 = 27 nM T31391 CLB72R 44218554 IC50 = 14 nM T31391 C2N9VR 44218555 IC50 = 63 nM T31391 CJ6L3S 44218693 IC50 = 29 nM T31391 C97IFE 44218695 IC50 = 32 nM T31391 C50EKW 44250174 IC50 = 9 nM T31391 CRZI12 44266022 IC50 = 14 nM T31391 C9YT6M 44270944 Ki = 1.1 nM T31391 C4MSN1 44285301 IC50 = 7900 nM T31391 CP9YN0 44285888 IC50 = 7000 nM T31391 CT3U1W 44286225 IC50 = 2400 nM T31391 C5UA6S 44286288 IC50 = 103000 nM T31391 CMG71F 44286291 IC50 = 52600 nM T31391 CQ5H8W 44286293 IC50 = 18000 nM T31391 CB6R9L 44286310 IC50 = 948000 nM T31391 C7ZHL3 44286477 IC50 = 277000 nM T31391 CF2H7C 44286480 IC50 = 746000 nM T31391 C7YU4C 44286501 IC50 = 6700 nM T31391 C0HZ5A 44286513 IC50 = 8400 nM T31391 C54LIM 44286562 IC50 = 170000 nM T31391 CH72YN 44286743 IC50 = 31800 nM T31391 C58LKI 44286823 IC50 = 14000 nM T31391 CVQ7K3 44286825 IC50 = 4700 nM T31391 CL3Q2J 44306072 IC50 = 4000 nM T31391 CMC8B9 44306777 IC50 = 44 nM T31391 CF2Q5V 44325514 Ki = 0.5 nM T31391 CE6G4X 44325523 Ki = 450 nM T31391 CI2YN1 44325525 Ki = 260 nM T31391 C29OIF 44325533 Ki = 0.8 nM T31391 CV4QM7 44325534 Ki = 6000 nM T31391 CLDY18 44325535 Ki = 4200 nM T31391 CN46PE 44325540 Ki = 21 nM T31391 CX94HW 44325697 Ki = 5 nM T31391 C1GRJ2 44325719 Ki = 0.41 nM T31391 CN45KP 44325734 Ki = 1.7 nM T31391 C4WTQ7 44326630 IC50 = 109000 nM T31391 C98LVO 44326651 IC50 = 372 nM T31391 C51EOL 44326652 IC50 = 218 nM T31391 C49PEQ 44326772 IC50 = 18700 nM T31391 C8NS4L 44326791 IC50 = 242 nM T31391 CYHE81 44327018 IC50 = 256 nM T31391 CNH8J3 44327071 IC50 = 16 nM T31391 CR3GE1 44327072 IC50 = 15 nM T31391 CSU32T 44327098 IC50 = 377 nM T31391 C0XFT4 44327160 IC50 = 13 nM T31391 CG7K1P 44327192 IC50 = 123 nM T31391 C2RC9I 44328126 IC50 = 14000 nM T31391 CTC40N 44328274 Ki = 47600 nM T31391 C8M0SH 44328300 Ki = 200 nM T31391 C6NZ9C 44328318 IC50 = 213000 nM T31391 C6OHV2 44328319 IC50 > 500000 nM T31391 CA53DN 44330624 IC50 = 13000 nM T31391 C7E1BJ 44330636 IC50 = 68000 nM T31391 C75JRD 44360575 IC50 = 24 nM T31391 CS72FI 44360697 IC50 = 7.5 nM T31391 CKSO92 44360724 IC50 = 26 nM T31391 CYED53 44360725 IC50 = 89 nM T31391 CXEC92 44360726 IC50 = 35 nM T31391 CL7WM8 44360734 IC50 = 64 nM T31391 CA0U8X 44360744 IC50 = 98 nM T31391 C50NME 44360749 IC50 = 94 nM T31391 CKI6W3 44360785 IC50 = 18 nM T31391 CRM9Y7 44360786 IC50 = 24 nM T31391 CXTP74 44360787 IC50 = 2.6 nM T31391 C5MB1D 44360809 IC50 = 46 nM T31391 C29DTA 44360810 IC50 = 190 nM T31391 CPTX82 44360812 IC50 = 2700 nM T31391 C3M8KF 44360910 IC50 = 38 nM T31391 CR7Q9N 44360911 IC50 = 53 nM T31391 CFY7P3 44360924 IC50 = 33 nM T31391 C62HNE 44360925 IC50 = 33 nM T31391 C1H5YG 44360938 IC50 = 21 nM T31391 C6IZ8L 44360955 IC50 = 15 nM T31391 CCJA09 44360967 IC50 = 29 nM T31391 CLMF32 44360976 IC50 = 20 nM T31391 CV1YL5 44360977 IC50 = 17 nM T31391 CY8A9K 44361010 IC50 = 10 nM T31391 C2KWI0 44361074 IC50 = 17 nM T31391 C1Z2FV 44361086 IC50 = 55 nM T31391 C8MJY5 44361216 IC50 = 9 nM T31391 CYK42S 44361230 IC50 = 25 nM T31391 CM3R2T 44364102 IC50 = 250000 nM T31391 CJ0VM6 44364126 IC50 = 3500 nM T31391 C83IUZ 44364133 IC50 = 217000 nM T31391 CJ8N0S 44364172 IC50 > 1000000 nM T31391 C7D2FW 44364210 IC50 = 93000 nM T31391 C8HO2F 44364211 IC50 = 500000 nM T31391 C9IQG4 44364212 IC50 > 1000000 nM T31391 C47NKP 44364213 IC50 = 52000 nM T31391 C6CYU9 44364227 IC50 > 500000 nM T31391 CHLV59 44364231 IC50 > 500000 nM T31391 CZF5N2 44364237 IC50 > 1000000 nM T31391 C7VR0N 44364252 IC50 > 1000000 nM T31391 CTS8U3 44364253 IC50 > 1000000 nM T31391 C0IW9L 44364296 IC50 = 289000 nM T31391 C6FBH7 44364297 IC50 = 81000 nM T31391 C79JMS 44364298 IC50 = 318000 nM T31391 CF2TA0 44364385 IC50 = 151000 nM T31391 C19DCN 44364405 IC50 = 51000 nM T31391 CX5AK7 44364446 IC50 > 500000 nM T31391 C4XIV2 44364456 IC50 > 1000000 nM T31391 C3XN5A 44364457 IC50 = 107000 nM T31391 CKA86J 44364458 IC50 = 500000 nM T31391 C4QON9 44368427 IC50 = 12.8 ug.mL-1 T31391 C8FB1S 44368725 IC50 = 64.4 ug.mL-1 T31391 CE83AK 44368726 IC50 > 100 ug.mL-1 T31391 CW9BG0 44368735 IC50 = 18.7 ug.mL-1 T31391 C37TIM 44368736 IC50 = 15.1 ug.mL-1 T31391 CX8I6C 44381633 IC50 = 550 nM T31391 CW9F3N 44381634 IC50 = 1200 nM T31391 CI39RJ 44381635 IC50 = 210 nM T31391 CLK90J 44381645 IC50 = 95 nM T31391 CT0EO4 44381646 IC50 = 240 nM T31391 CHX2T7 44381647 IC50 = 1100 nM T31391 C6Y4QW 44381687 IC50 = 110 nM T31391 CN96MI 44381721 IC50 = 420 nM T31391 CK4SP1 44381763 IC50 = 480 nM T31391 CI6RT5 44381811 IC50 = 4600 nM T31391 CG1CD7 44381826 IC50 = 110 nM T31391 CL51SX 44381845 IC50 = 660 nM T31391 CXBY42 44381846 IC50 = 230 nM T31391 C5SV9U 44381847 IC50 = 110 nM T31391 CRY5K1 44381848 IC50 = 3900 nM T31391 CRE8J7 44381849 IC50 = 280 nM T31391 CUX2Q9 44381861 IC50 = 220 nM T31391 C92CKY 44381862 IC50 = 130 nM T31391 CIX09S 44381884 IC50 = 46 nM T31391 C3GH0S 44381896 IC50 = 43 nM T31391 C0FQO1 44381899 IC50 = 47 nM T31391 CTRX81 44381910 IC50 = 420 nM T31391 C2XBA5 44381911 IC50 = 170 nM T31391 CBL60E 44381919 IC50 = 250 nM T31391 CARK25 44381928 IC50 = 94 nM T31391 C4LR3K 44381945 IC50 = 270 nM T31391 CQ4VZ3 44381966 IC50 = 440 nM T31391 CDCY49 44381967 IC50 = 670 nM T31391 CT9IN5 44381974 IC50 = 330 nM T31391 C0FQY4 44381979 IC50 = 180 nM T31391 CP7XG9 44382005 IC50 = 180 nM T31391 C6YFP9 44382006 IC50 = 870 nM T31391 CWJ3V5 44382013 IC50 = 1700 nM T31391 CI8O3F 44382065 IC50 = 150 nM T31391 CX2JS7 44382077 IC50 = 72 nM T31391 C38MSH 44382133 IC50 = 110 nM T31391 C8PD7J 44382134 IC50 = 83 nM T31391 C89LXF 44382393 IC50 = 840 nM T31391 CAJ50V 44382443 IC50 = 290 nM T31391 C8ZP1A 44382444 IC50 = 110 nM T31391 CKOD04 44382521 IC50 = 83 nM T31391 CY2C8J 44387751 IC50 > 1000000 nM T31391 CXSU53 44387755 IC50 > 1000000 nM T31391 CALG81 44387756 IC50 > 1000000 nM T31391 CL1M7V 44387758 IC50 > 125000 nM T31391 C6T2MW 44387765 IC50 > 1000000 nM T31391 CA7KI2 44390794 IC50 = 13000 nM T31391 CVD21W 44393563 IC50 = 39640 nM T31391 C24PMT 44393585 IC50 > 100000 nM T31391 CB9WA5 44393586 IC50 = 16480 nM T31391 C7N1GB 44393611 IC50 = 3000 nM T31391 CS51KL 44393656 IC50 = 33000 nM T31391 C7SB1I 44393657 IC50 = 44860 nM T31391 C9JT0N 44393695 IC50 = 46910 nM T31391 CPG38C 44393696 IC50 = 27470 nM T31391 CF6KR8 44393727 IC50 = 51000 nM T31391 C58KPC 44393728 IC50 = 5700 nM T31391 CDH6J1 44393857 IC50 = 200 nM T31391 C2PK9W 44393881 IC50 = 2620 nM T31391 CB6E5I 44393933 IC50 = 80 nM T31391 C08BMZ 44394001 IC50 = 51 nM T31391 C8RA0W 44394023 IC50 = 9400 nM T31391 C3KH1Q 44394024 IC50 = 589 nM T31391 C4QE5X 44394028 IC50 = 143 nM T31391 CPF49E 44394029 IC50 = 155 nM T31391 C8ZA9M 44394031 IC50 = 11000 nM T31391 CS35UP 44394072 IC50 = 2026 nM T31391 CW79MD 44394073 IC50 = 19 nM T31391 CW81MP 44394103 IC50 = 270 nM T31391 C7Y4LZ 44394104 IC50 = 8476 nM T31391 C25SDY 44394118 IC50 = 19000 nM T31391 CU85FA 44394119 IC50 = 30 nM T31391 CJ18AZ 44394135 IC50 = 35000 nM T31391 CTEP50 44394136 IC50 = 36000 nM T31391 C4BO3S 44394155 IC50 = 34 nM T31391 CALF89 44394157 IC50 = 0.1 nM T31391 C4B9OH 44394173 IC50 = 1100 nM T31391 CX75VF 44394180 IC50 = 14860 nM T31391 C85SEO 44394194 IC50 = 2519 nM T31391 CS1Z7X 44394195 IC50 = 2263 nM T31391 C39LZT 44394203 IC50 = 3028 nM T31391 CF6Y8L 44394209 IC50 = 10700 nM T31391 CQ09FB 44394210 IC50 = 1040 nM T31391 CXG8B6 44394238 IC50 = 931 nM T31391 CIJ95E 44394239 IC50 = 981 nM T31391 C3Q5WZ 44394241 IC50 = 3611 nM T31391 CL3EP4 44394242 IC50 = 690 nM T31391 C8U2ZQ 44394244 IC50 = 3279 nM T31391 CZA46H 44394270 IC50 = 2026 nM T31391 CUGH58 44394271 IC50 = 8951 nM T31391 CU7PY3 44394282 IC50 = 7688 nM T31391 C41ITO 44394305 IC50 = 1900 nM T31391 CG53YO 44394349 IC50 = 1552 nM T31391 C59NLA 44394350 IC50 = 1700 nM T31391 C0NSL3 44396153 IC50 = 4 nM T31391 C1VLP6 44399148 IC50 = 252 nM T31391 CIED90 44399244 IC50 = 87 nM T31391 C3PKV8 44399546 IC50 = 97 nM T31391 CEW52I 44400445 IC50 = 0.25 nM T31391 C8UDI1 44400447 IC50 = 0.33 nM T31391 CZ19WH 44400450 IC50 = 6.6 nM T31391 C0MEB2 44400462 IC50 = 1.5 nM T31391 C41SZA 44400473 IC50 = 0.28 nM T31391 C68USM 44400485 IC50 = 0.19 nM T31391 CZ6A8Q 44400504 IC50 = 3 nM T31391 CJD9B5 44400535 IC50 = 5.5 nM T31391 CU8CL1 44400547 IC50 = 6.7 nM T31391 CR87KM 44400555 IC50 = 1.9 nM T31391 CSJU72 44400574 IC50 = 4.6 nM T31391 C6VB2Q 44400588 IC50 = 9.7 nM T31391 C3RAW7 44400625 IC50 = 0.53 nM T31391 CUR51H 44402967 Ki = 504 nM T31391 CZO5J3 44402970 Ki = 1267 nM T31391 CIKW98 44402971 Ki = 61 nM T31391 CP72TO 44402972 Ki = 81 nM T31391 CA8K9B 44403068 Ki = 109 nM T31391 C32LIY 44403069 Ki = 117 nM T31391 CPX1M9 44403336 IC50 = 370 nM T31391 CSEN70 44403337 IC50 = 17000 nM T31391 C0NXE8 44403338 IC50 = 2000 nM T31391 CR53EK 44403354 IC50 = 1200 nM T31391 CRO16Q 44403360 IC50 = 4.5 nM T31391 C0FC7D 44403361 IC50 = 15 nM T31391 C3HFZ7 44403391 IC50 = 130 nM T31391 C3TOY4 44403392 IC50 = 75 nM T31391 CU39LX 44403393 IC50 = 25 nM T31391 CIA8Y3 44403397 IC50 = 27 nM T31391 C6P7NE 44403398 IC50 = 58 nM T31391 CP34SF 44403405 IC50 = 8 nM T31391 C60VBT 44403406 IC50 = 61 nM T31391 C50LWV 44403411 IC50 = 16000 nM T31391 CQ5T4Y 44403412 IC50 = 0.8 nM T31391 CMX9B1 44403416 IC50 = 12 nM T31391 CUKG07 44403417 IC50 = 560 nM T31391 CX29FU 44403421 IC50 = 1600 nM T31391 C2P4CQ 44403422 IC50 = 7.8 nM T31391 CCOA39 44403438 IC50 = 32000 nM T31391 CLYJ80 44403439 IC50 = 810 nM T31391 C4YAH3 44404393 IC50 = 25 nM T31391 C02SYC 44406179 Ki = 225 nM T31391 CU8B3S 44406189 Ki = 46 nM T31391 C1SBD5 44406234 Ki = 115 nM T31391 C5P1RX 44406284 Ki = 40 nM T31391 C0IQO3 44411572 IC50 = 771 nM T31391 C3HXA1 44411573 IC50 > 3000 nM T31391 CW73SO 44411579 IC50 > 3000 nM T31391 CB17FI 44411652 IC50 > 3000 nM T31391 C5WPL4 44411659 IC50 > 3000 nM T31391 C1HCZ6 44411660 IC50 > 3000 nM T31391 C29ZOU 44411665 IC50 > 3000 nM T31391 C9MH4X 44411669 IC50 > 3000 nM T31391 C54RFY 44411670 IC50 > 3000 nM T31391 CE86UP 44411700 IC50 = 237 nM T31391 CR7MX8 44411923 IC50 = 1860 nM T31391 CFP80H 44412105 Ki = 0.41 nM T31391 CZ15VN 44412163 Ki = 2.5 nM T31391 C0HA7I 44412169 Ki = 2900 nM T31391 CGJ17L 44415883 IC50 > 250000 nM T31391 CE0KW2 44415905 IC50 > 100000 nM T31391 CPR49A 44415906 IC50 > 125000 nM T31391 CQ5P2J 44415929 IC50 = 234000 nM T31391 CM2W5X 44415930 IC50 > 125000 nM T31391 COPZ87 44415944 IC50 > 125000 nM T31391 CGLB32 44417381 Ki = 49 nM T31391 C2TP5K 44417385 Ki = 97 nM T31391 CN2F6U 44417389 Ki > 30000 nM T31391 C12HGD 44417391 Ki > 30000 nM T31391 CSG4F8 44417393 Ki = 1 nM T31391 CE7UB0 44418114 IC50 = 0.29 nM T31391 CD9J3S 44418157 IC50 = 4 nM T31391 C70KAO 44418211 IC50 = 42 nM T31391 C8LC2A 44418213 IC50 = 127 nM T31391 CTM1Y8 44418214 IC50 = 269 nM T31391 C1EMA5 44418215 IC50 = 144 nM T31391 CWDH12 44418216 IC50 = 1300 nM T31391 C1FB4K 44418218 IC50 = 252 nM T31391 CVC3R4 44418219 IC50 = 236 nM T31391 CU1FG2 44418222 IC50 = 247 nM T31391 C8ZH5R 44418223 IC50 = 320 nM T31391 CA9YM3 44418225 IC50 = 232 nM T31391 CQE5Y0 44418229 IC50 = 181 nM T31391 CID62U 44418230 Ki = 4300 nM T31391 CI2H7Q 44418231 Ki = 9080 nM T31391 C2LXS7 44418232 IC50 = 118 nM T31391 CXCV19 44418233 Ki = 7391 nM T31391 CZW38C 44418239 Ki = 9500 nM T31391 C7KF0X 44418240 Ki = 4600 nM T31391 C8QJ7H 44418242 Ki = 19500 nM T31391 C60KPZ 44418243 Ki = 11300 nM T31391 CMKW39 44418246 Ki = 68 nM T31391 CEBQ24 44418249 Ki = 1430 nM T31391 C59HZQ 44418251 IC50 = 8000 nM T31391 CDX2Q5 44418253 Ki = 451000 nM T31391 C0RV8O 44418254 Ki = 182000 nM T31391 C37KEO 44418255 Ki = 6871 nM T31391 C2UR9X 44418256 IC50 = 239 nM T31391 CK20CA 44418257 IC50 = 190 nM T31391 CO3GL6 44418260 IC50 = 207 nM T31391 CY3O7C 44418261 IC50 = 197 nM T31391 C0ITV9 44418262 IC50 = 433 nM T31391 CGR3H7 44418263 IC50 = 21000 nM T31391 C68SHD 44418264 IC50 = 253 nM T31391 CDI98V 44418265 IC50 = 225 nM T31391 CHO5P1 44418266 IC50 = 911 nM T31391 C95XQC 44418268 IC50 = 174 nM T31391 CE3C4D 44420996 Ki = 140 nM T31391 CI2P6M 44420998 Ki = 6.1 nM T31391 C0FT8Q 44420999 Ki = 4 nM T31391 C7VU1I 44421000 Ki = 13 nM T31391 C38PJE 44421001 Ki = 2.3 nM T31391 CX4C3Y 44421002 Ki = 11 nM T31391 CF52AI 44421003 Ki = 23 nM T31391 C6NV0S 44421004 Ki = 1.6 nM T31391 C5W8VX 44421005 Ki = 2.3 nM T31391 C8KC3R 44421006 Ki = 3 nM T31391 C16YHQ 44422417 IC50 = 112 nM T31391 C9IRG5 44422418 IC50 = 11 nM T31391 C7XU0J 44422419 IC50 = 7.9 nM T31391 C58WCU 44422439 IC50 = 19.2 nM T31391 C2F9DG 44422440 IC50 = 51.5 nM T31391 CS63GZ 44422443 IC50 = 5.8 nM T31391 C9M5YC 44422444 IC50 = 7 nM T31391 C0J1UX 44422445 IC50 = 45.4 nM T31391 CKFM17 44422448 IC50 = 6.5 nM T31391 C6C3ZF 44422475 IC50 = 147 nM T31391 C9T1KM 44422476 IC50 = 25.2 nM T31391 CN5G6O 44422477 IC50 = 181 nM T31391 CNQC83 44422485 IC50 = 34 nM T31391 C5NK2E 44422486 IC50 > 300 nM T31391 CZ5UW9 44422487 IC50 = 37.2 nM T31391 C6TZM8 44422496 IC50 > 300 nM T31391 CX5M3Q 44422497 IC50 > 300 nM T31391 C86SXN 44422498 IC50 = 154 nM T31391 C4YP0T 44422507 IC50 = 85.9 nM T31391 C1IW2L 44422508 IC50 > 300 nM T31391 CRWM46 44422509 IC50 > 300 nM T31391 CJK1H2 44422513 IC50 = 9.6 nM T31391 C6C5PM 44422514 IC50 = 7.1 nM T31391 C4KSW0 44422518 IC50 = 9.1 nM T31391 CL40CD 44422519 IC50 = 6.4 nM T31391 CY4K6X 44422522 IC50 = 13.6 nM T31391 CZ8TO9 44422523 IC50 = 13.9 nM T31391 CCFT17 44422525 IC50 = 16.8 nM T31391 C0BXJ2 44422526 IC50 = 17 nM T31391 CGB32F 44422527 IC50 = 228 nM T31391 C1N4RA 44422528 IC50 = 26.4 nM T31391 C1D7ER 44425490 IC50 = 8 nM T31391 CZ2MB8 44426068 IC50 = 6.6 nM T31391 C8PKO5 44426070 IC50 = 139 nM T31391 CW7QD8 44429116 IC50 = 3.5 nM T31391 C1NF6D 44429117 IC50 = 3.4 nM T31391 CG67NO 44429119 IC50 = 5.7 nM T31391 CT54EH 44429120 IC50 = 2.9 nM T31391 C37SUV 44429122 IC50 = 2.4 nM T31391 C57GUJ 44429124 IC50 = 7.8 nM T31391 CW59YC 44429127 IC50 = 3.5 nM T31391 C0L9SG 44429129 IC50 = 6.1 nM T31391 CT2P8M 44429130 IC50 = 9.1 nM T31391 C4KRA5 44429131 IC50 = 3.9 nM T31391 CM2FK3 44429132 IC50 = 2.5 nM T31391 CEL8D9 44429133 IC50 = 3.3 nM T31391 CX48BO 44429134 IC50 = 8.3 nM T31391 CWF04T 44429135 IC50 = 23 nM T31391 CN68CG 44429136 IC50 = 8.9 nM T31391 C6J3CS 44429137 IC50 = 22 nM T31391 C6F1NE 44429138 IC50 = 4.9 nM T31391 CL2G7Z 44429139 IC50 = 7.1 nM T31391 CHT96Z 44429140 IC50 = 5.3 nM T31391 CVD9U0 44429602 IC50 = 3.8 nM T31391 C17MKX 44429603 IC50 = 16 nM T31391 C3SKR2 44429609 IC50 = 4.5 nM T31391 C0SU2X 44429610 IC50 = 2.4 nM T31391 CGQN20 44429612 IC50 = 7.7 nM T31391 CYGD28 44429613 IC50 = 3.5 nM T31391 CZ7LW9 44429614 IC50 = 4.4 nM T31391 CXJD74 44429616 IC50 = 5.7 nM T31391 C6R2IZ 44429619 IC50 = 6 nM T31391 C0A2CF 44429620 IC50 = 4 nM T31391 C4EH0L 44429622 IC50 = 4.9 nM T31391 CY4MF9 44429623 IC50 = 8.3 nM T31391 C02JQU 44429624 IC50 = 11 nM T31391 CG3C7E 44429625 IC50 = 4.3 nM T31391 CHNV25 44429626 IC50 = 4.8 nM T31391 C7IL3S 44431164 IC50 = 98 nM T31391 C0UOS8 44431165 IC50 = 135 nM T31391 CEG05S 44431166 IC50 = 272 nM T31391 CO8S3Z 44431170 IC50 = 805 nM T31391 C2K4RQ 44431176 IC50 = 151 nM T31391 CJZY21 44431177 IC50 = 87 nM T31391 CSJI40 44431185 IC50 = 1018 nM T31391 C36EJR 44431188 IC50 = 486 nM T31391 C2MCA1 44431191 IC50 = 366 nM T31391 C89XVB 44431197 IC50 = 511 nM T31391 CK76EP 44431199 IC50 = 145 nM T31391 C3FPT2 44431200 IC50 = 59 nM T31391 C4F8AG 44431201 IC50 = 264 nM T31391 CWX4I3 44431203 IC50 = 1580 nM T31391 CZ3N9E 44431204 IC50 = 23 nM T31391 C5NAS6 44431205 IC50 = 180 nM T31391 C37SGU 44431206 IC50 = 84 nM T31391 CYD62G 44431212 IC50 = 60 nM T31391 C72WTP 44431213 IC50 = 30 nM T31391 CC3T9G 44431214 IC50 = 65 nM T31391 CL4T3X 44431215 IC50 = 190 nM T31391 C4WVL8 44431216 IC50 = 69 nM T31391 CO08HZ 44431217 IC50 = 37 nM T31391 CCPZ23 44431218 IC50 = 30 nM T31391 C0J7WV 44431219 IC50 = 29 nM T31391 C16ZTV 44431220 IC50 = 219 nM T31391 CR0A1M 44431316 IC50 = 21 nM T31391 CV1R7A 44431317 IC50 = 140 nM T31391 CTB82G 44431744 IC50 = 520 nM T31391 C7O4GL 44431746 IC50 = 35700 nM T31391 CJOR92 44431752 IC50 = 2100 nM T31391 CETI27 44431756 IC50 = 5800 nM T31391 C2VY9T 44431757 IC50 = 142000 nM T31391 C09BFG 44431758 IC50 = 2600 nM T31391 CX3ZH1 44431759 IC50 = 4900 nM T31391 C5JYG0 44431760 IC50 = 26000 nM T31391 C1CRX9 44431761 IC50 = 2300 nM T31391 CB7SA0 44431762 IC50 = 18400 nM T31391 C4FT0P 44431764 IC50 = 8900 nM T31391 C7OJW0 44431765 IC50 = 220 nM T31391 CMU40B 44431766 IC50 = 990 nM T31391 CA9P1R 44431767 IC50 = 1520 nM T31391 CL0VB1 44431768 IC50 = 10590 nM T31391 CHG8I4 44431769 IC50 = 370 nM T31391 C7PLH0 44431770 IC50 = 9380 nM T31391 CC0J6A 44431771 IC50 = 3730 nM T31391 C4X1GA 44431772 IC50 = 5130 nM T31391 C4S8DE 44431773 IC50 = 650 nM T31391 CQX2S0 44431774 IC50 = 32 nM T31391 CL6B7S 44431775 IC50 = 4 nM T31391 C16CRQ 44431776 IC50 = 50 nM T31391 CY76AB 44432858 IC50 = 77 nM T31391 CS95EU 44432859 IC50 = 67 nM T31391 C1PX9V 44432860 IC50 = 223 nM T31391 C3AN4E 44432861 IC50 = 7939 nM T31391 CE4Q5X 44432862 IC50 = 35 nM T31391 CHN6E3 44432863 IC50 = 63 nM T31391 CF2AT6 44432881 IC50 = 15 nM T31391 CTD24F 44432889 IC50 = 95 nM T31391 CSC2E0 44432894 IC50 = 210 nM T31391 CU67PL 44432901 IC50 = 224 nM T31391 C35GZP 44432904 IC50 = 84 nM T31391 C21UQD 44432911 IC50 = 53 nM T31391 CU27DF 44432914 IC50 = 680 nM T31391 C9E1SZ 44432915 IC50 = 339 nM T31391 CZ47KB 44432929 IC50 = 20 nM T31391 CS5BT9 44432935 IC50 = 56 nM T31391 CI9M8R 44432936 IC50 = 17 nM T31391 C5LTR0 44432937 IC50 = 30 nM T31391 C6EJB0 44432938 IC50 = 10 nM T31391 CJ7YN0 44432940 IC50 = 255 nM T31391 CVZ3I2 44432942 IC50 = 47 nM T31391 CT29BC 44432944 IC50 = 25 nM T31391 CNOW68 44433160 IC50 = 140 nM T31391 CJUH82 44433161 IC50 = 2000 nM T31391 C8A1ZL 44433162 IC50 = 150 nM T31391 CJ61CN 44433163 IC50 > 3000 nM T31391 C20OBQ 44433164 IC50 > 3000 nM T31391 C1GBW2 44433165 IC50 > 3000 nM T31391 CEJC97 44433166 IC50 > 3000 nM T31391 CI1NU4 44433167 IC50 = 1000 nM T31391 C5NAI2 44433168 IC50 > 3000 nM T31391 C7TWF9 44433169 IC50 > 3000 nM T31391 C5YUC3 44433174 Ki = 1420 nM T31391 CI5UK4 44433203 IC50 = 790 nM T31391 CVL2Q7 44433204 IC50 = 1400 nM T31391 CR5X3V 44433205 IC50 = 2300 nM T31391 CGB9I5 44433206 IC50 = 2900 nM T31391 CZGM71 44433207 IC50 > 3000 nM T31391 C8PBJ4 44433208 IC50 > 3000 nM T31391 CQ71FG 44433209 IC50 > 3000 nM T31391 C3QOB8 44433210 IC50 > 3000 nM T31391 CO8WI2 44433212 IC50 > 3000 nM T31391 COC75P 44433213 IC50 > 3000 nM T31391 CIB5K2 44433214 IC50 > 3000 nM T31391 C7LI5A 44433215 IC50 > 3000 nM T31391 CCT2I4 44433216 IC50 = 260 nM T31391 CTA59M 44433217 IC50 = 93 nM T31391 CY73TI 44433218 IC50 = 230 nM T31391 C91CFD 44433219 IC50 = 57 nM T31391 CAN07M 44433220 IC50 = 180 nM T31391 C4UTL0 44433221 IC50 = 190 nM T31391 C8CWB2 44433222 IC50 = 37 nM T31391 C4O8SB 44433223 IC50 = 19 nM T31391 CQDS95 44433224 IC50 = 14 nM T31391 CNW1S2 44433225 IC50 = 47 nM T31391 CB04FG 44433226 IC50 = 470 nM T31391 C90GFZ 44433227 IC50 = 130 nM T31391 CSHA84 44433228 IC50 = 160 nM T31391 C6ZP3F 44433229 IC50 = 51 nM T31391 C7KR9C 44433230 IC50 = 120 nM T31391 CH96JN 44433231 IC50 = 71 nM T31391 CR7CQ3 44433232 IC50 = 1300 nM T31391 CWI98S 44433233 IC50 = 32 nM T31391 C23ZRQ 44433234 IC50 = 14 nM T31391 C43RDG 44433235 IC50 = 120 nM T31391 CU6O4S 44433236 IC50 = 70 nM T31391 C8U4QI 44433237 IC50 = 31 nM T31391 C9GIE3 44433617 IC50 = 16 nM T31391 C5B4HS 44433618 IC50 = 12 nM T31391 CU6XZ5 44433646 IC50 = 100 nM T31391 CM8E2D 44433661 IC50 = 38 nM T31391 C07PZD 44433929 Ki > 10000 nM T31391 CG8QR0 44433931 Ki = 3653 nM T31391 CMG6W7 44433932 Ki = 877 nM T31391 CMUR94 44433933 Ki > 10000 nM T31391 CU7AR9 44433934 Ki = 3007 nM T31391 C1ML6S 44433935 Ki > 10000 nM T31391 CM9V3B 44433936 Ki > 10000 nM T31391 C0PLN8 44433937 Ki > 10000 nM T31391 CE5F7Q 44433938 Ki > 10000 nM T31391 CCBR97 44433939 Ki > 10000 nM T31391 CCEO15 44433941 Ki > 10000 nM T31391 CL6V0G 44433942 Ki > 10000 nM T31391 CB70WG 44433943 Ki > 10000 nM T31391 CC02JQ 44433944 Ki > 10000 nM T31391 C9SO3Y 44433945 Ki = 3257 nM T31391 CU7WB6 44433946 Ki > 10000 nM T31391 CAD8G1 44433950 Ki = 1010 nM T31391 C1P2BE 44433951 Ki = 1065 nM T31391 CZA08G 44433952 Ki = 530 nM T31391 CIJF53 44433953 Ki = 731 nM T31391 CTF97G 44433954 Ki = 356 nM T31391 CQ9JD6 44433955 Ki > 10000 nM T31391 CP0M9W 44433956 Ki > 10000 nM T31391 CQ41OU 44433957 Ki = 112 nM T31391 CI15HN 44433958 Ki = 152 nM T31391 C1C9SZ 44433959 Ki = 1944 nM T31391 CA4VY1 44433960 Ki = 3311 nM T31391 CU69GM 44433961 Ki > 10000 nM T31391 CDF80C 44433962 Ki > 10000 nM T31391 CKN0C1 44433969 Ki = 3081 nM T31391 C53UEG 44434115 IC50 = 8 nM T31391 CE92DA 44435310 IC50 = 261000 nM T31391 C3SBK5 44435313 IC50 = 8000 nM T31391 CX7UN0 44435314 IC50 = 4200 nM T31391 CE7XI5 44435315 IC50 > 50000 nM T31391 CGAR49 44435316 IC50 > 250000 nM T31391 C17HRW 44439324 IC50 = 127 nM T31391 C1JQ8Y 44439325 IC50 = 47.6 nM T31391 CAOY46 44439326 IC50 = 13.9 nM T31391 C8XU3A 44439327 IC50 = 57.5 nM T31391 CI7SP9 44439328 IC50 = 10.9 nM T31391 CWG07L 44439329 IC50 = 30.5 nM T31391 CT9V8F 44439330 IC50 = 21 nM T31391 C74ANZ 44439331 IC50 = 13.5 nM T31391 C4B5DI 44439332 IC50 = 12.2 nM T31391 C7LEY1 44439333 IC50 = 8.7 nM T31391 CCJ8T1 44439334 IC50 = 4.1 nM T31391 CWU62R 44439335 IC50 = 10.8 nM T31391 CWG89M 44439336 IC50 = 8.2 nM T31391 CEL4H9 44439337 IC50 = 1.6 nM T31391 C4H3EF 44439338 IC50 = 4.3 nM T31391 C3MLU4 44439339 IC50 = 6.8 nM T31391 C8P1AX 44439340 IC50 = 3 nM T31391 C54TPV 44439341 IC50 = 1.3 nM T31391 CEP51V 44439342 IC50 = 5.6 nM T31391 C4YWH2 44439343 IC50 = 2.3 nM T31391 C1G5PI 44439344 IC50 = 2.4 nM T31391 C02LBF 44439345 IC50 = 2.7 nM T31391 CBE1D5 44439346 IC50 = 3.1 nM T31391 C5T7XF 44439347 IC50 = 2.5 nM T31391 CMC8H4 44439348 IC50 = 1.6 nM T31391 CX4MT0 44439350 IC50 = 1.5 nM T31391 C0OJ1T 44439353 IC50 = 1 nM T31391 C9T6FK 44439354 IC50 = 1.2 nM T31391 C69XIH 44439668 IC50 = 990 nM T31391 CDF76U 44439670 IC50 = 500 nM T31391 C6E8JI 44440627 Ki = 2700 nM T31391 CUQ7K0 44440629 Ki = 280 nM T31391 CSXH19 44440630 Ki = 610 nM T31391 CSI93Z 44440631 Ki = 490 nM T31391 COP6M3 44440633 Ki = 790 nM T31391 C5GKC8 44440634 Ki = 210 nM T31391 CTI8C4 44440635 Ki = 430 nM T31391 C2VAG9 44440645 Ki = 17 nM T31391 CTQR78 44440647 Ki = 20 nM T31391 C08ZST 44440659 Ki = 1 nM T31391 CA9WC3 44440660 Ki = 85 nM T31391 CXC50E 44440661 Ki = 7 nM T31391 CR3PM7 44440662 Ki = 1.7 nM T31391 CB4Q0H 44440663 Ki = 3.4 nM T31391 C6YEQ8 44440664 Ki = 9 nM T31391 CCSI57 44440665 Ki = 1.3 nM T31391 CR4B1M 44443293 IC50 = 30 nM T31391 CY16JP 44443294 IC50 = 38 nM T31391 CN24IJ 44443296 IC50 = 40 nM T31391 C8DSC1 44443297 IC50 = 42 nM T31391 C4F5JW 44443298 IC50 = 47 nM T31391 CJ0G3N 44443299 IC50 = 49 nM T31391 C9F7NQ 44443300 IC50 = 62 nM T31391 C7QCO2 44443301 IC50 = 79 nM T31391 CCQ82F 44443302 IC50 = 86 nM T31391 C1M5TF 44443309 IC50 = 27 nM T31391 CSAE59 44443313 IC50 = 50 nM T31391 CK5E8V 44443319 IC50 = 69 nM T31391 CD0NM4 44443335 IC50 = 78 nM T31391 CEF6H5 44443336 IC50 = 80 nM T31391 CTIM25 44443338 IC50 = 81 nM T31391 CE9Q7A 44443341 IC50 = 83 nM T31391 CI8Q5O 44443343 IC50 = 91 nM T31391 C0MOV3 44443346 IC50 = 2.4 nM T31391 C52VPZ 44443347 IC50 = 3.2 nM T31391 CJ8P7U 44443348 IC50 = 3.3 nM T31391 C8U1XN 44443349 IC50 = 3.6 nM T31391 CM5WU9 44443350 IC50 = 5.3 nM T31391 CB9IM0 44443351 IC50 = 5.4 nM T31391 C8WI4F 44443352 IC50 = 6.2 nM T31391 C3NI8P 44443353 IC50 = 6.7 nM T31391 C7M0HV 44443354 IC50 = 8.5 nM T31391 C0UG4R 44443355 IC50 = 10 nM T31391 C7B5HK 44443356 IC50 = 10 nM T31391 C2G1PX 44443357 IC50 = 3 nM T31391 C3AUF2 44443358 IC50 = 3.4 nM T31391 C0WO5B 44443359 IC50 = 3.5 nM T31391 CUG6X5 44443360 IC50 = 5.5 nM T31391 CARK80 44443361 IC50 = 5.3 nM T31391 CP7WL5 44443363 IC50 = 1.1 nM T31391 C4V0SN 44443364 IC50 = 4.7 nM T31391 CQL53Y 44443365 IC50 = 46 nM T31391 CD2L9G 44443366 IC50 = 3.8 nM T31391 CPN7J9 44443420 IC50 = 65 nM T31391 CI4VR8 44443421 IC50 > 3 nM T31391 CA0NZ7 44443707 IC50 = 140 nM T31391 C24ZHB 44443708 IC50 = 150 nM T31391 C8R4OD 44443709 IC50 = 130 nM T31391 CLDN63 44443710 IC50 = 180 nM T31391 C7LNP2 44443711 IC50 = 230 nM T31391 CJX2M7 44443712 IC50 = 220 nM T31391 C6RST0 44443713 IC50 = 260 nM T31391 C3YL9X 44443714 IC50 = 250 nM T31391 CRH8M1 44443715 IC50 = 250 nM T31391 CIB50E 44443717 IC50 = 130 nM T31391 CK6QF4 44443719 IC50 = 280 nM T31391 CX6O1P 44443720 IC50 = 65 nM T31391 C0YV2D 44443723 IC50 = 610 nM T31391 C1BUJ5 44443725 IC50 = 570 nM T31391 CXS34I 44443727 IC50 = 50 nM T31391 CCHS17 44443729 IC50 = 110 nM T31391 C39KZG 44443736 IC50 = 250 nM T31391 C5H8EJ 44443737 IC50 = 370 nM T31391 CS3Y1G 44444344 IC50 = 100 nM T31391 CL2U9C 44444352 IC50 = 68 nM T31391 C8VE5T 44444353 IC50 = 274 nM T31391 C8F5HC 44444371 IC50 = 4 nM T31391 CEW50M 44444373 IC50 = 4 nM T31391 CO0M7Y 44444375 IC50 = 7 nM T31391 CS93BI 44444377 IC50 = 12 nM T31391 C9J4FB 44444379 IC50 = 14 nM T31391 C3YA4K 44444383 IC50 = 18 nM T31391 C75OIP 44444386 IC50 = 2 nM T31391 C4J6ZG 44444390 IC50 = 4 nM T31391 C05EBU 44444391 IC50 = 2 nM T31391 CSN27E 44445042 IC50 = 5.7 nM T31391 CGN61Q 44445047 IC50 = 1.5 nM T31391 CYW8E3 44445051 IC50 = 2.8 nM T31391 CRG64M 44445053 IC50 = 0.66 nM T31391 C6ZID3 44445055 IC50 = 0.43 nM T31391 C72KOR 44445057 IC50 = 438 nM T31391 C0RTA6 44445060 IC50 = 0.46 nM T31391 CIK8G3 44445063 IC50 = 0.32 nM T31391 CN05VX 44445065 IC50 = 6.3 nM T31391 COA90R 44445067 IC50 = 132 nM T31391 CHRX61 44445075 IC50 > 36900 nM T31391 C6C5IN 44448853 IC50 = 559 nM T31391 CB7MS5 44448857 IC50 = 582 nM T31391 C4IXY7 44448987 IC50 = 2 nM T31391 COP51N 44448988 IC50 = 1 nM T31391 C8KW2A 44448989 IC50 = 99 nM T31391 C9ZRP1 44449015 IC50 = 19 nM T31391 C7E4ZI 44449016 IC50 = 107 nM T31391 CKM5H1 44449017 IC50 = 52 nM T31391 CJ2WY0 44449038 IC50 = 4 nM T31391 C8F2SQ 44449064 IC50 = 2 nM T31391 C7PBF3 44449092 IC50 = 15 nM T31391 CUM32L 44449149 IC50 = 1 nM T31391 CK5M4R 44451509 IC50 = 56 nM T31391 CWI3J9 44451511 IC50 = 41 nM T31391 CEFD93 44451512 IC50 = 600 nM T31391 CKCF72 44451863 IC50 = 51 nM T31391 CR51UD 44451910 IC50 = 60 nM T31391 C76NDG 44451911 IC50 = 16 nM T31391 C20LHD 44452002 IC50 = 13000 nM T31391 CODZ87 44452030 IC50 = 110 nM T31391 CV0Z4T 44452035 IC50 = 70 nM T31391 C7RI2V 44452075 IC50 = 16 nM T31391 CUC93Q 44452076 IC50 = 1100 nM T31391 CK5DW6 44453458 IC50 = 30 nM T31391 C3X8BJ 44453460 IC50 = 42 nM T31391 CDF8R2 44453520 IC50 = 50000 nM T31391 CVO9F2 44453648 IC50 = 57 nM T31391 C91FSI 44453672 IC50 = 90 nM T31391 C5UET4 44453690 IC50 = 645 nM T31391 C2JE8C 44453692 IC50 = 1165 nM T31391 C6EC4J 44453922 IC50 = 12 nM T31391 C4C6NK 44453968 IC50 = 93 nM T31391 CDS52W 44453970 IC50 = 3.2 nM T31391 C9V2HU 44454016 IC50 = 50 nM T31391 CW4H0F 44455959 IC50 = 52 nM T31391 C0S2TV 44455961 IC50 = 21 nM T31391 CH04ND 44455993 IC50 = 37 nM T31391 C50MTS 44456000 IC50 = 604 nM T31391 CQF6O5 44456002 IC50 = 620 nM T31391 CFZB21 44456030 IC50 = 1900 nM T31391 CI0K1D 44456032 IC50 = 340 nM T31391 CYN5Z3 44456147 IC50 = 310 nM T31391 C1WBL5 44456148 IC50 = 350 nM T31391 C3HE5Z 44456310 IC50 = 670 nM T31391 CHKT64 44458509 IC50 = 830 nM T31391 CXWQ16 44458510 IC50 = 360 nM T31391 CBSZ02 44458521 IC50 = 88 nM T31391 CIA6J1 44458523 IC50 = 56 nM T31391 C6LKZ7 44458534 IC50 = 27 nM T31391 CR41OX 44458540 IC50 = 870 nM T31391 CNK09O 44458542 IC50 = 70 nM T31391 CM65HC 44458548 IC50 = 23 nM T31391 CKM0F5 44458549 IC50 = 75 nM T31391 CR4CP3 44458554 IC50 = 21 nM T31391 CU68KW 44458566 IC50 = 270 nM T31391 CC7I6Y 44458573 IC50 = 110 nM T31391 CCI52U 44458574 IC50 = 250 nM T31391 C0K7EZ 44458575 IC50 = 210 nM T31391 CNK64C 44458581 IC50 = 250 nM T31391 CF7I9V 44458586 IC50 = 67 nM T31391 CW7QX0 44458587 IC50 = 55 nM T31391 CJ7Y6A 44458592 IC50 = 35 nM T31391 C9QMB2 44458594 Ki = 56 nM T31391 CPJW14 44458603 Ki = 128 nM T31391 C0K2SV 44458617 Ki = 28 nM T31391 CSIL15 44458629 IC50 = 54 nM T31391 C3EZ1V 44458770 IC50 = 89 nM T31391 COHJ95 44560137 IC50 = 252 nM T31391 CAY0V7 44560138 IC50 = 7.3 nM T31391 C8LNP1 44560139 IC50 = 6.2 nM T31391 CUJR76 44560140 IC50 = 22 nM T31391 C0V4UW 44560141 IC50 = 8.6 nM T31391 CFX7Y2 44560154 IC50 = 12 nM T31391 CGW57E 44560155 IC50 = 88 nM T31391 C0Z5AB 44560156 IC50 = 16 nM T31391 C9JL5Y 44560157 IC50 = 27 nM T31391 C4NC6K 44560158 IC50 = 2.9 nM T31391 CHJ2I3 44560159 IC50 = 7.8 nM T31391 CR4AD0 44560160 IC50 = 8.7 nM T31391 CO9I7S 44560169 IC50 = 13 nM T31391 CD6H2S 44560170 IC50 > 316 nM T31391 C9QC1W 44560171 IC50 = 33 nM T31391 CNF05Y 44560172 IC50 = 3.1 nM T31391 CB73HS 44560173 IC50 = 2.6 nM T31391 CC9B5Y 44560174 IC50 = 3.3 nM T31391 C41LTG 44560184 IC50 = 4.1 nM T31391 C7E1TG 44560185 IC50 = 3.1 nM T31391 C8Z2AR 44560186 IC50 = 3.1 nM T31391 CX3EK8 44560187 IC50 = 8.3 nM T31391 C1BX6I 44560188 IC50 = 5.3 nM T31391 CY78ZH 44560250 IC50 = 2.8 nM T31391 CR69YS 44560251 IC50 = 2.7 nM T31391 C60VSL 44560252 IC50 = 2.4 nM T31391 C70CYA 44560253 IC50 = 8.2 nM T31391 C8CED7 44560254 IC50 = 4.5 nM T31391 CC09EL 44560255 IC50 = 5.4 nM T31391 C5MN2V 44560265 IC50 = 2.9 nM T31391 C75KOL 44560266 IC50 = 5.7 nM T31391 CED9I6 44560267 IC50 = 5.8 nM T31391 C9DLI3 44560268 IC50 = 13 nM T31391 CU65ER 44560279 IC50 = 109 nM T31391 C17LFS 44560280 IC50 = 75 nM T31391 CTD6U0 44560281 IC50 = 31 nM T31391 CB7V0P 44560282 IC50 > 316 nM T31391 CJ4EN1 44560283 IC50 = 39 nM T31391 C91DWY 44560396 IC50 > 100000 nM T31391 CZ9WJ0 44560397 IC50 > 100000 nM T31391 C0FLU7 44560398 IC50 = 80100 nM T31391 CZ43JR 44560454 IC50 > 100000 nM T31391 CY38QP 44560549 IC50 > 100000 nM T31391 C7IL3K 44560550 IC50 > 100000 nM T31391 CF9J7Z 44560551 IC50 > 100000 nM T31391 C1QAI4 44560552 IC50 > 100000 nM T31391 CK25CG 44560553 IC50 > 50000 nM T31391 C4C9NG 44560554 IC50 > 100000 nM T31391 CKIH45 44560555 IC50 > 100000 nM T31391 C2LW3C 44560595 IC50 > 100000 nM T31391 C47WCK 44560596 IC50 > 100000 nM T31391 CL8AE5 44560597 IC50 > 100000 nM T31391 C1YJ8C 44560648 IC50 > 50000 nM T31391 CY6GU1 44560649 IC50 > 62500 nM T31391 C12EYZ 44560650 IC50 = 178000 nM T31391 C7LY9V 44560651 IC50 > 31250 nM T31391 CG5CB2 44560698 IC50 > 250000 nM T31391 CR56BA 44560699 IC50 = 4970 nM T31391 CAK3U5 44560701 IC50 > 100000 nM T31391 C5OW2C 44560747 IC50 > 500000 nM T31391 CM2GN5 44560748 IC50 > 1000000 nM T31391 C5FSB4 44560749 IC50 > 500000 nM T31391 C5WEG1 44560750 IC50 > 250000 nM T31391 CN0KO4 44560770 IC50 = 22 nM T31391 CZSO82 44560823 Ki = 4900 nM T31391 C4IVD9 44560824 IC50 = 37000 nM T31391 C4L3VZ 44560825 IC50 = 15600 nM T31391 CHV7S1 44560826 IC50 = 9700 nM T31391 CE3NF4 44560849 IC50 = 12700 nM T31391 CT6P5E 44560850 IC50 = 16800 nM T31391 CTH9P2 44560851 Ki = 1200 nM T31391 CGZ48C 44560928 IC50 = 51000 nM T31391 C9EK8A 44560929 IC50 > 1000000 nM T31391 CM68VD 44560930 IC50 = 3700 nM T31391 C4SMJ1 44560961 IC50 = 35 nM T31391 C2I3TR 44560962 IC50 = 340 nM T31391 CGV49L 44560963 IC50 = 290 nM T31391 CY0L1G 44560964 IC50 = 2200 nM T31391 C7FST1 44560988 IC50 = 530 nM T31391 CGOM86 44560989 IC50 = 52000 nM T31391 C74ZNK 44560990 IC50 = 2500 nM T31391 C95AUS 44560991 IC50 = 560 nM T31391 CTJ23N 44561008 IC50 = 1300 nM T31391 CR2A0E 44561009 IC50 = 253 nM T31391 C4LQY2 44561010 IC50 = 107 nM T31391 C28XDF 44561011 IC50 = 71 nM T31391 CQ04BE 44561046 IC50 = 9800 nM T31391 C8IF7B 44561117 IC50 = 9200 nM T31391 C29VDX 44561118 IC50 = 200 nM T31391 CB4JA7 44561119 IC50 = 8800 nM T31391 C5K9CX 44561120 IC50 = 55 nM T31391 CQ8DN4 44561152 IC50 = 4400 nM T31391 C4DBU1 44561153 IC50 = 615 nM T31391 C73WBR 44561154 IC50 = 600 nM T31391 CJ91UC 44561155 IC50 = 46 nM T31391 CMO6S2 44561191 IC50 = 20 nM T31391 CF9SB3 44561192 IC50 = 40 nM T31391 C5X1VJ 44561193 IC50 = 120 nM T31391 C31GMV 44561194 IC50 = 85 nM T31391 C1U4YQ 44565237 IC50 = 27 nM T31391 CRK69O 44565238 IC50 = 19 nM T31391 C6M2WD 44565239 IC50 = 21 nM T31391 CTZ9L0 44565254 IC50 = 22 nM T31391 CEMV93 44565274 IC50 = 26 nM T31391 C5E6PQ 44565275 IC50 = 17 nM T31391 CI93OK 44565276 IC50 = 20 nM T31391 C2HRF1 44565277 IC50 = 26 nM T31391 CFEC28 44565466 IC50 = 85 nM T31391 C5MON6 44565467 IC50 = 54 nM T31391 CGA4U6 44565488 IC50 = 64 nM T31391 C1BZ3I 44565489 IC50 = 84 nM T31391 CP3C5F 44565490 IC50 = 75 nM T31391 CRU86T 44565491 IC50 = 62 nM T31391 C3C2DL 44565492 IC50 = 85 nM T31391 CJ2W1P 44565512 IC50 = 60 nM T31391 C5Z9GW 44565513 IC50 = 73 nM T31391 C3I0MO 44565514 IC50 = 86 nM T31391 CI3J6Y 44565535 IC50 = 68 nM T31391 CB90XZ 44565536 IC50 = 101 nM T31391 C01SLH 44565537 IC50 = 24 nM T31391 C8Y2LX 44565538 IC50 = 10 nM T31391 CXD19F 44565539 IC50 = 56 nM T31391 C5BIY6 44565582 IC50 = 309 nM T31391 CFK92H 44565583 IC50 = 25 nM T31391 CE3UT4 44565584 IC50 = 309 nM T31391 CA0O7F 44565585 IC50 = 41 nM T31391 C7LPW8 44565586 IC50 = 134 nM T31391 C39RGP 44565611 IC50 = 338 nM T31391 CPZ7J3 44565844 IC50 = 8.7 nM T31391 C9BGR3 44565845 IC50 = 8.2 nM T31391 CR83QA 44565869 IC50 = 7.4 nM T31391 C6K2WL 44565870 IC50 = 5.6 nM T31391 C3UL2E 44565871 IC50 = 5.2 nM T31391 C9SL5D 44565872 IC50 = 4.8 nM T31391 CZBX95 44565889 IC50 = 31 nM T31391 C1TLY0 44565890 IC50 = 51 nM T31391 CEO20N 44565891 IC50 = 31 nM T31391 COA7X5 44565892 IC50 = 13 nM T31391 CRO3D2 44567651 IC50 = 186 nM T31391 CM95OD 44567652 IC50 = 221 nM T31391 CX6WL5 44567653 IC50 = 27 nM T31391 C4MP9D 44567654 IC50 = 49 nM T31391 CV23FP 44567668 IC50 = 85 nM T31391 CD4C7Y 44567710 IC50 = 123 nM T31391 C4CUJ6 44567711 IC50 = 147 nM T31391 CK1C7W 44567712 IC50 = 78 nM T31391 CTK1I9 44567713 IC50 = 91 nM T31391 C9LQ7N 44567714 IC50 = 1300 nM T31391 CM50CU 44567747 IC50 = 93 nM T31391 C9IF5L 44567748 IC50 > 10000 nM T31391 CMGJ56 44567749 Ki = 5 nM T31391 CR43EI 44567750 Ki = 12 nM T31391 CZ3G4I 44567783 Ki = 31 nM T31391 CNA0I9 44567918 IC50 = 165 nM T31391 C6BXT0 44567919 IC50 = 153 nM T31391 CJ85MG 44567920 IC50 = 110 nM T31391 CUJD19 44567976 IC50 = 38 nM T31391 C5YB6E 44567977 IC50 = 95 nM T31391 CNF09E 44567978 IC50 = 152 nM T31391 C70WEI 44567979 IC50 = 59 nM T31391 CJ0YL5 44568015 IC50 = 2540 nM T31391 CW7NB6 44568016 IC50 = 109 nM T31391 CY8Z3F 44568017 IC50 = 229 nM T31391 CRM76D 44568018 IC50 = 95 nM T31391 C7D4EP 44568055 IC50 = 3430 nM T31391 C3E2UC 44568056 IC50 = 3740 nM T31391 CCG83U 44568057 IC50 = 51 nM T31391 C8XW9A 44568058 IC50 = 31 nM T31391 CMQ7D5 44568097 IC50 = 42 nM T31391 C1F9OL 44568098 IC50 = 63 nM T31391 CUYK75 44568099 IC50 = 92 nM T31391 CZ81XF 44568100 IC50 = 141 nM T31391 C6GT0A 44568134 IC50 = 422 nM T31391 C6IW5D 44568135 IC50 = 630 nM T31391 C3PWD8 44568136 IC50 = 118 nM T31391 C3JBY7 44568137 IC50 = 1715 nM T31391 C4NCA7 44568169 IC50 = 84 nM T31391 C8TXH9 44568170 IC50 = 181 nM T31391 C17PZX 44568171 IC50 = 146 nM T31391 C7SCJ1 44568172 IC50 = 186 nM T31391 CT10GB 44571684 IC50 = 1440 nM T31391 CAT7M0 44571686 IC50 = 510 nM T31391 CSU97M 44571688 IC50 = 3400 nM T31391 C8UGS0 44571690 IC50 = 490 nM T31391 C2WC7S 44571735 IC50 = 410 nM T31391 C0BX2S 44571737 IC50 = 490 nM T31391 C7KYX8 44571739 IC50 = 1392 nM T31391 C2ZYC9 44571741 IC50 = 1500 nM T31391 C68DZI 44571781 IC50 = 350 nM T31391 C1HSU7 44571783 IC50 = 3100 nM T31391 C5WDE4 44571785 IC50 = 405 nM T31391 CB20PW 44571787 IC50 = 387 nM T31391 C8NB2X 44571851 IC50 = 6400 nM T31391 C40YLT 44571853 IC50 = 597 nM T31391 CV9BW0 44571855 IC50 = 423 nM T31391 C0LMD8 44571898 IC50 = 239 nM T31391 CLFG01 44571900 IC50 = 788 nM T31391 C1U5MS 44571902 IC50 = 180 nM T31391 C8DAK4 44571945 IC50 = 288 nM T31391 CM9DP7 44571947 IC50 = 150 nM T31391 CZCU54 44571949 IC50 = 50 nM T31391 CJ96CO 44571951 IC50 = 67 nM T31391 CQW5N2 44571996 IC50 = 260 nM T31391 C7E6IB 44572718 IC50 = 298 nM T31391 CUH81Y 44572719 IC50 = 2 nM T31391 CJHR19 44572720 IC50 = 10 nM T31391 CG71OU 44572782 IC50 = 1600 nM T31391 CG86WR 44580460 IC50 = 13000 nM T31391 C7NP1S 44580497 IC50 = 12000 nM T31391 CQU6S5 44580498 IC50 = 50000 nM T31391 C9JY0C 44580499 IC50 = 180000 nM T31391 CT1N3H 44580500 IC50 = 390000 nM T31391 CYO50L 44580540 IC50 = 11 nM T31391 CSX3I9 44580589 IC50 = 25 nM T31391 CGB0H3 44580664 IC50 = 21 nM T31391 CPR2S7 44589876 IC50 = 7800 nM T31391 C3H0AD 44589877 IC50 = 1000 nM T31391 CY5TC1 44589878 IC50 = 2200 nM T31391 CKM0Z1 44589879 IC50 = 870 nM T31391 CPU4J0 44589931 IC50 = 2500 nM T31391 C4X9GH 44589932 IC50 = 3300 nM T31391 C2DQ0C 44589933 IC50 = 570 nM T31391 C27TUB 44589934 IC50 = 470 nM T31391 CUZ3P0 44589935 IC50 = 190 nM T31391 CM18AD 44589985 IC50 = 64 nM T31391 C4LEZ6 44589986 IC50 = 13 nM T31391 CW2T9J 44589987 IC50 = 12 nM T31391 C1SK7V 44590037 IC50 = 2.7 nM T31391 C6NE1Y 44590038 IC50 = 3.3 nM T31391 CGV2A7 44590039 IC50 = 270 nM T31391 C1KC3N 44590040 IC50 = 35 nM T31391 CZGQ12 44590126 IC50 = 130 nM T31391 CV7RD4 44590127 IC50 = 70 nM T31391 CIE7S0 44590128 IC50 = 350 nM T31391 CCK2S8 44590129 IC50 = 1 nM T31391 C39MKI 44590183 IC50 = 0.64 nM T31391 C82PIC 44590184 IC50 = 1.9 nM T31391 C85SFW 44590185 IC50 = 0.79 nM T31391 C48MPJ 44590596 IC50 = 251 nM T31391 CYE25R 44590598 Ki = 3.6 nM T31391 CI98LA 44590648 IC50 = 22 nM T31391 CBAH06 44590649 IC50 = 6.2 nM T31391 C5R9NI 44590650 IC50 = 0.13 nM T31391 C0W2FC 44590651 IC50 = 0.15 nM T31391 CRN4U5 44590696 IC50 = 4.3 nM T31391 CTC24F 44590734 IC50 = 8 nM T31391 C8CRO4 44590736 IC50 = 18 nM T31391 C91FTW 44591848 IC50 = 18 nM T31391 CY78PR 44591849 IC50 = 22 nM T31391 CE2LW5 44591850 IC50 = 27 nM T31391 CZW0V4 44592369 IC50 > 30000 nM T31391 C3WJ6O 44592370 IC50 = 1930 nM T31391 C07LHO 44592439 IC50 = 3580 nM T31391 CTC4G9 44592440 IC50 > 30000 nM T31391 CIVD36 44592441 IC50 = 25900 nM T31391 C65OXJ 44592442 IC50 > 30000 nM T31391 C8Z0CX 44592443 IC50 = 3250 nM T31391 C9PL5R 44592444 IC50 = 1420 nM T31391 C7L8UN 44592445 IC50 > 30000 nM T31391 CQG62W 44592506 IC50 = 1970 nM T31391 CQHL54 44592507 IC50 = 272 nM T31391 CV42SK 44592508 IC50 = 270 nM T31391 C82YQS 44592509 IC50 = 35 nM T31391 CWJ2U0 44592510 IC50 = 26 nM T31391 CQI40A 44592511 IC50 = 19 nM T31391 CY8R3Q 44593399 IC50 = 115000 nM T31391 CP8YC3 44593408 IC50 = 161000 nM T31391 C4L6NS 44593409 IC50 = 245000 nM T31391 CI0FT1 44593463 IC50 = 47 nM T31391 CAWO01 44593726 IC50 = 6030 nM T31391 CY7Q8W 44629524 IC50 = 22 nM T31391 C65KPR 45101722 IC50 = 6.3 nM T31391 CXYT36 45101723 IC50 = 3 nM T31391 C2RNP7 45102670 IC50 = 16 nM T31391 CQ85WF 45263621 Ki = 6 nM T31391 CGZD98 45265711 IC50 = 103 nM T31391 CW09DZ 45265891 Ki = 3.2 nM T31391 CCO76A 45266134 IC50 = 1700 nM T31391 CU4C5P 45266135 IC50 = 20 nM T31391 CLVM20 45266136 IC50 = 19 nM T31391 CIS3Z8 45267371 IC50 = 92 nM T31391 C8H9GV 45267527 IC50 = 3.2 nM T31391 CP9B0W 45267530 IC50 = 15 nM T31391 C3GJK0 45267531 IC50 = 5.4 nM T31391 CD67HE 45268222 IC50 = 47 nM T31391 CN38QU 45268229 IC50 = 12 nM T31391 CEQ16V 45268233 IC50 = 8 nM T31391 CT93EB 45268323 IC50 = 27 nM T31391 C0QB1V 45268417 IC50 = 2 nM T31391 C2S9ZT 45268436 IC50 = 27 nM T31391 C60MVX 45269112 IC50 = 66 nM T31391 CV7IL1 45269122 IC50 = 24 nM T31391 CX8WC0 45269123 IC50 = 30 nM T31391 C9HR0K 45269274 IC50 = 7.8 nM T31391 CZ1N2O 45269275 IC50 = 12 nM T31391 CIE21V 45269276 IC50 = 5.6 nM T31391 C2W6MT 45269961 IC50 = 87 nM T31391 CWT60M 45269971 IC50 = 14 nM T31391 C4CG2K 45269976 IC50 = 27 nM T31391 CK5P9W 45269994 IC50 = 152 nM T31391 C2A8WO 45269995 IC50 > 16000 nM T31391 C8QJ7X 45270108 IC50 = 7.1 nM T31391 CYWK62 45270115 IC50 = 10 nM T31391 C6E7PR 45270793 IC50 = 92 nM T31391 C6B0CO 45270800 IC50 = 20 nM T31391 CS89DP 45270806 IC50 = 53 nM T31391 CZI9A4 45270821 IC50 > 1600 nM T31391 CQM4X3 45270889 IC50 = 49 nM T31391 CGF7Z6 45270958 IC50 = 2.7 nM T31391 CH5S8Y 45270959 IC50 = 2.2 nM T31391 CM80NZ 45271662 IC50 > 1600 nM T31391 C5NH6Q 45271791 IC50 = 4 nM T31391 C8Z3DK 45271794 IC50 = 3.9 nM T31391 CX62YA 45271796 IC50 = 1.3 nM T31391 CZ8EO2 45271803 IC50 = 3.5 nM T31391 CJ7Q9E 45271813 IC50 = 6.8 nM T31391 CLSJ45 45272523 IC50 = 77 nM T31391 C75XKZ 45272524 IC50 = 27 nM T31391 CSC67Y 45272544 IC50 > 16000 nM T31391 CJI2R6 45272664 IC50 = 2.3 nM T31391 C49BKQ 45272672 IC50 = 5.9 nM T31391 CP36CT 45272682 IC50 = 1.5 nM T31391 C8NL4U 45272683 IC50 = 2.7 nM T31391 CI5AU6 45273390 IC50 = 94 nM T31391 C6S0OC 45273404 IC50 = 8 nM T31391 C2EK3O 45273409 IC50 = 53 nM T31391 C1ZX6U 45273413 IC50 > 1600 nM T31391 CYMR87 45273573 IC50 = 3.5 nM T31391 CFL87A 45273581 IC50 = 6.3 nM T31391 C2XB0P 45273589 IC50 = 6.1 nM T31391 C28PRV 45273594 IC50 = 4.8 nM T31391 CSX2T9 45273602 IC50 = 3.7 nM T31391 CMP59Q 45273603 IC50 = 1.1 nM T31391 C2R3QM 45481268 IC50 = 9 nM T31391 C31XRV 45482320 IC50 = 14130 nM T31391 C28ZXW 45487888 IC50 = 2 nM T31391 C74SVC 45487893 IC50 = 31 nM T31391 C2N3IZ 45487894 IC50 = 3 nM T31391 CP62TC 45487898 IC50 = 4 nM T31391 CPBA81 45487901 IC50 = 90 nM T31391 C0SQW3 45487902 IC50 = 62 nM T31391 CWQ1R9 45487903 IC50 = 2 nM T31391 C8H1KY 45487904 IC50 = 4 nM T31391 C1LJR6 45487907 IC50 = 120 nM T31391 C6X7WJ 45487908 IC50 = 4 nM T31391 CZDS09 45487910 IC50 = 76 nM T31391 CNVU49 45487911 IC50 = 180 nM T31391 C5OXM9 45487915 IC50 = 17 nM T31391 CPJ19X 45487917 IC50 = 2 nM T31391 C16DIR 45487918 IC50 = 28 nM T31391 CV2R7M 45487920 IC50 = 1 nM T31391 C57JRG 45487921 IC50 = 11 nM T31391 C4JD1P 45487922 IC50 = 32 nM T31391 CH30BL 45487925 IC50 = 130 nM T31391 CPB85R 45487926 IC50 = 17 nM T31391 CTY16E 45487930 IC50 = 7 nM T31391 C4QTL9 45487931 IC50 = 5 nM T31391 CG9V0L 45487940 IC50 = 22 nM T31391 C5XTV1 45487945 IC50 = 10 nM T31391 C3VK4G 45487946 IC50 = 2 nM T31391 C0SNL2 46209134 IC50 = 1.6 nM T31391 CE9M5C 46209244 IC50 = 1.6 nM T31391 CW60IG 46209246 IC50 = 1.6 nM T31391 CV65TL 46216691 IC50 = 11 nM T31391 C4QO6X 46216692 IC50 = 0.5 nM T31391 C4GPM1 46229765 IC50 = 61 nM T31391 CCO56J 46229809 IC50 = 38 nM T31391 C0CQM4 46229810 IC50 = 5500 nM T31391 CQ5S8A 46229811 IC50 = 0.5 nM T31391 C6K1YR 46229812 IC50 = 1.7 nM T31391 CU4GE7 46230652 IC50 = 53000 nM T31391 CI4A3C 46230653 IC50 = 19 nM T31391 CEPY06 46231493 IC50 = 1.2 nM T31391 CIEK51 46842529 IC50 = 2810 nM T31391 CDP7Q4 46870369 IC50 = 17 nM T31391 CPH7B4 46871723 IC50 = 8 nM T31391 CDBC45 46890720 IC50 = 180 nM T31391 CLK47C 46890721 IC50 = 23 nM T31391 CS6HL3 46890722 IC50 = 50 nM T31391 C2JY6P 46890723 IC50 = 24 nM T31391 CP7C1L 46890780 IC50 = 26 nM T31391 CED80Z 46890852 IC50 = 93 nM T31391 CA3PE4 46890853 IC50 = 160 nM T31391 CY9T8W 46890854 IC50 = 66 nM T31391 C3TJ0H 46890912 IC50 = 27 nM T31391 CT9HQ6 46890913 IC50 = 24 nM T31391 C9IP7B 46890914 IC50 = 18 nM T31391 CSZE87 46891193 IC50 = 12 nM T31391 C18UES 46891235 IC50 = 59 nM T31391 C23LCY 46891237 IC50 = 65 nM T31391 C57UXS 46891239 IC50 = 80 nM T31391 CIM3K6 46891241 IC50 = 204 nM T31391 C4AUV2 46891291 IC50 = 326 nM T31391 C0UKG7 46891293 IC50 = 121 nM T31391 CJ4G6X 46891342 IC50 = 32 nM T31391 CAL9K6 46891534 IC50 = 15 nM T31391 CPN5T2 46891535 IC50 = 71 nM T31391 C4XTW7 46893990 IC50 > 100000 nM T31391 C8O5VR 46899592 Ki = 8.7 nM T31391 CTY0M5 46899593 Ki = 1 nM T31391 CK9TH1 46899594 Ki = 3.1 nM T31391 C8XD0Q 46899595 Ki = 0.2 nM T31391 CZ84ST 46899596 Ki = 0.5 nM T31391 CPZ70E 46899597 Ki = 0.3 nM T31391 CD3IJ8 46899752 Ki = 0.9 nM T31391 CRK59N 46899753 Ki = 6.6 nM T31391 C6LXU5 46899754 Ki = 2 nM T31391 C52JZL 46899755 Ki = 0.6 nM T31391 C4RC1S 46899756 Ki = 1.8 nM T31391 CP84HR 46899757 Ki = 3.8 nM T31391 CBV4W0 46899937 Ki = 2.6 nM T31391 C5QEJ4 46899938 Ki = 1.1 nM T31391 CHR6V9 46899939 Ki = 2 nM T31391 CQ3A8F 46899940 Ki = 3.2 nM T31391 CX2P8Z 46899941 Ki = 0.7 nM T31391 CC2X1J 46899942 Ki = 2.6 nM T31391 C5QA9M 46900103 Ki = 4 nM T31391 CBI0Q2 46900104 Ki = 0.9 nM T31391 C4IU2E 46900105 Ki = 5 nM T31391 CZEB71 46900106 Ki = 4.7 nM T31391 C2TJW5 46900108 Ki = 1.5 nM T31391 C54ATK 46900259 Ki = 1.3 nM T31391 CI3P6J 46900261 Ki = 2.4 nM T31391 C6DP2G 46900418 Ki = 3.1 nM T31391 CP50DR 46900420 Ki = 5 nM T31391 CF3BL8 46905362 IC50 = 1500 nM T31391 C9JKO5 46905992 IC50 = 21 nM T31391 C8DSG7 46916343 IC50 > 100000 nM T31391 C3RO8F 46916345 IC50 > 100000 nM T31391 CX07LJ 46916346 IC50 > 100000 nM T31391 CF94MW 46916347 IC50 > 100000 nM T31391 CH3F7O 46916384 IC50 > 100000 nM T31391 CM8W6E 46916385 IC50 > 100000 nM T31391 C6FA9Q 46916386 IC50 > 100000 nM T31391 CAW86J 46916387 IC50 > 100000 nM T31391 C63HBE 46916388 IC50 > 100000 nM T31391 CD1CZ7 46916389 IC50 > 100000 nM T31391 CH80LK 46916433 IC50 > 100000 nM T31391 CN4A3P 46916435 IC50 > 100000 nM T31391 CUQ86M 46917047 IC50 > 100000 nM T31391 CS5X9L 46917048 IC50 > 100000 nM T31391 CZP24U 46917049 IC50 = 570 nM T31391 COY5T4 46937042 IC50 = 19 nM T31391 CGMJ52 46938499 IC50 > 100000 nM T31391 C5RAS7 46938602 IC50 > 100000 nM T31391 C3B1LX 46938704 IC50 > 100000 nM T31391 C5TU1F 46938705 IC50 > 100000 nM T31391 CAGP83 46938706 IC50 > 100000 nM T31391 CP9V8Q 46938799 IC50 > 100000 nM T31391 CAB2H9 46938802 IC50 > 100000 nM T31391 C80RAT 47370344 IC50 > 100000 nM T31391 CR5X3K 49785099 IC50 = 0.33 nM T31391 C2HU0V 49785100 IC50 = 1.72 nM T31391 CX7M2K 49785101 IC50 = 0.87 nM T31391 C3XCV4 49785102 IC50 = 1.32 nM T31391 CC8Z5M 49795916 IC50 = 500 nM T31391 CI6U4M 49795917 IC50 = 700 nM T31391 C7HV2K 49795919 IC50 = 2300 nM T31391 CHE51J 49795928 IC50 = 5000 nM T31391 CI6QC3 49795929 IC50 = 800 nM T31391 C8GIY2 49795930 IC50 = 9100000 nM T31391 C2Y5FT 49795931 IC50 = 36 nM T31391 CS1TY7 49795932 IC50 = 23 nM T31391 CUW13V 49795933 IC50 = 47000 nM T31391 CZNL37 49795934 IC50 = 1800000 nM T31391 CGQC72 49795935 IC50 = 31000 nM T31391 CK72BR 49795936 IC50 = 22000 nM T31391 CNB64H 49795937 IC50 = 30 nM T31391 CE2P1Y 49795938 IC50 = 190000 nM T31391 C2TY4D 49795939 IC50 > 10000 nM T31391 COHI43 49795940 IC50 = 400 nM T31391 CDI04P 49795942 IC50 = 1400 nM T31391 CKF3D9 49795943 IC50 = 5000 nM T31391 C95AGZ 49795944 IC50 = 600 nM T31391 CT3XF0 49795948 IC50 = 16 nM T31391 C5RP2S 49796932 IC50 = 510 nM T31391 CZ7A9E 49796933 IC50 = 87 nM T31391 C8D7IG 49796934 IC50 = 539 nM T31391 CBX38D 49796935 IC50 = 1200 nM T31391 CC74RX 49796936 IC50 = 161 nM T31391 CLBU64 49796937 IC50 = 54 nM T31391 C5RF0Y 49796938 IC50 = 7200 nM T31391 CE0C3Y 49796939 IC50 = 75 nM T31391 CI4ZE6 49796940 IC50 = 37 nM T31391 CA54TF 49796941 IC50 = 0.3 nM T31391 CBD8K2 49796942 IC50 = 39 nM T31391 CD21SQ 49796943 IC50 = 170 nM T31391 CODZ18 49796944 IC50 = 118 nM T31391 CI25XP 49796945 IC50 = 721 nM T31391 CF65YQ 49796946 IC50 = 1640 nM T31391 C32MAO 49796947 IC50 = 10 nM T31391 CHJ76U 49796948 IC50 = 3.7 nM T31391 CU25OB 49796949 IC50 = 5.1 nM T31391 C1ZJS7 49796950 IC50 = 4200 nM T31391 C8GWI5 49796951 IC50 = 1.8 nM T31391 CH2W5L 49796952 IC50 = 18 nM T31391 C8WYA5 49796953 IC50 = 0.48 nM T31391 C0P6JR 49796954 IC50 = 1.6 nM T31391 CQH86V 49796955 IC50 = 8.2 nM T31391 C08NMS 49796956 IC50 = 0.83 nM T31391 CR63MS 49796957 IC50 = 18 nM T31391 CJ5FR6 49796958 IC50 = 7.1 nM T31391 C7IBX0 49796959 IC50 = 3300 nM T31391 CU83MS 49796960 IC50 = 12 nM T31391 CQ5YV7 49796961 IC50 = 13 nM T31391 C1T9ON 49796962 IC50 = 3600 nM T31391 C1ZVH6 49796963 IC50 = 82 nM T31391 CB26OQ 49796964 IC50 = 1200 nM T31391 C0NO8F 49796965 IC50 = 9.5 nM T31391 C69JQC 49796966 IC50 = 33 nM T31391 C01RDX 49796967 IC50 = 1.7 nM T31391 C2SXO4 49796968 IC50 = 1.6 nM T31391 C7SH5C 49796969 IC50 = 12 nM T31391 C7K3HC 49796970 IC50 = 295 nM T31391 CBMV50 49796972 IC50 = 64 nM T31391 C8IL0K 49796973 IC50 = 980 nM T31391 CA90LB 49796974 IC50 = 1600 nM T31391 C07DHG 49796977 IC50 = 3500 nM T31391 CAS2P4 49796982 IC50 = 220 nM T31391 CG79KT 49796985 IC50 = 390 nM T31391 C4D8RE 49796990 IC50 = 6.6 nM T31391 CUKB68 49796994 IC50 = 550 nM T31391 CUR9B0 49796995 IC50 = 9.2 nM T31391 CWHO58 49796998 IC50 = 45 nM T31391 CX74RG 49796999 IC50 = 12 nM T31391 C20MAQ 49797000 IC50 = 13 nM T31391 CD67OX 49797001 IC50 = 192 nM T31391 C9LEF5 49797002 IC50 = 9.1 nM T31391 CO2AX9 49797003 IC50 = 3.3 nM T31391 CEM61W 49797006 IC50 = 520 nM T31391 C7Y0JL 49797007 IC50 = 59 nM T31391 CW45IK 49797008 IC50 = 37 nM T31391 C79JUI 49797011 IC50 = 67 nM T31391 CVAK94 49797012 IC50 = 29 nM T31391 CUK5J1 49797013 IC50 = 43 nM T31391 C4ZK5C 49797014 IC50 = 2.2 nM T31391 C1PV8J 49797015 IC50 = 30 nM T31391 C9YEU6 49797016 IC50 = 17 nM T31391 CZD4S2 49797017 IC50 = 99 nM T31391 CKY80F 49797018 IC50 = 11 nM T31391 CS0D8Q 49797021 IC50 = 27 nM T31391 C3GF4M 49797022 IC50 = 100 nM T31391 C8XZT9 49797023 IC50 = 71 nM T31391 C5H2AS 49797024 IC50 = 94 nM T31391 C4P0VW 49797025 IC50 = 20 nM T31391 CVY8M1 49797028 IC50 = 110 nM T31391 CM59HB 49797029 IC50 = 230 nM T31391 CH7Y1J 49797030 IC50 = 44 nM T31391 CX18HI 49797031 IC50 = 21 nM T31391 CUM28Z 49797035 IC50 = 110 nM T31391 COS23G 49797036 IC50 = 7.5 nM T31391 C2TSG6 49797038 IC50 = 56 nM T31391 C7BI3W 49797039 IC50 = 21 nM T31391 C71THK 49797040 IC50 = 1100 nM T31391 C0SG5O 49797041 IC50 = 7900 nM T31391 CM37VB 49797042 IC50 = 170 nM T31391 C51NUG 49797043 IC50 = 480 nM T31391 C65WXC 49797044 IC50 = 600 nM T31391 CHTO37 49797045 IC50 = 2000 nM T31391 CA8R5K 49797046 IC50 = 3700 nM T31391 CLAR35 49797047 IC50 = 250 nM T31391 C9OCZ3 49797048 IC50 = 54000 nM T31391 C49RUW 49797049 IC50 = 1100 nM T31391 C4EHT7 49797050 IC50 = 3700 nM T31391 CW6G5R 49797051 IC50 = 2800 nM T31391 CUK6G0 49797052 IC50 = 120 nM T31391 CJ1FE2 49797053 IC50 = 280 nM T31391 CKJO08 49797054 IC50 = 4200 nM T31391 C70KVU 49797055 IC50 = 3600 nM T31391 CP59BI 49797056 IC50 = 360 nM T31391 CEDL61 49797057 IC50 = 770 nM T31391 C5J2LV 49797058 IC50 = 1400 nM T31391 CEI20Q 49797059 IC50 = 1100 nM T31391 C7B5DY 49797060 IC50 = 6 nM T31391 C5B1RM 49797061 IC50 = 100 nM T31391 C40HJC 49797062 IC50 = 240 nM T31391 CL3P4H 49797063 IC50 = 98 nM T31391 CPC76U 49797064 IC50 = 140 nM T31391 C5F4JN 49797065 IC50 = 580 nM T31391 C86HND 49797066 IC50 = 130 nM T31391 C8E4XD 49797067 IC50 = 1500 nM T31391 CHO1U0 49797068 IC50 = 100 nM T31391 CO1TW7 49797069 IC50 = 69 nM T31391 CAD6W1 49797071 IC50 = 110 nM T31391 CQYU80 49797072 IC50 = 110 nM T31391 CEZ38H 49797073 IC50 = 110 nM T31391 C0CEU7 49797074 IC50 = 140 nM T31391 C72JXY 49797075 IC50 = 27 nM T31391 COA41Q 49797076 IC50 = 510 nM T31391 CPQ3Z2 49797077 IC50 = 140 nM T31391 C1WI0D 49797078 IC50 = 60 nM T31391 C4D8XP 49797079 IC50 = 390 nM T31391 CQG4J6 49797080 IC50 = 130 nM T31391 CKM9S4 49797081 IC50 = 75 nM T31391 C3JRW0 49797082 IC50 = 370 nM T31391 C27IEB 49797083 IC50 = 150 nM T31391 C0JUL3 49797084 IC50 = 110 nM T31391 C85DOL 49797085 IC50 = 110 nM T31391 CEGO30 49797086 IC50 = 150 nM T31391 C2TC3I 49797087 IC50 = 440 nM T31391 C04JWY 49797088 IC50 = 240 nM T31391 CA2U4Y 49797089 IC50 = 56 nM T31391 CFT46J 49797090 IC50 = 37 nM T31391 C35TFW 49797091 IC50 = 86 nM T31391 CRL7Z5 49797092 IC50 = 710 nM T31391 CYU74X 49797093 IC50 = 420 nM T31391 C2O3SG 49797094 IC50 = 150 nM T31391 CFL3O2 49797106 IC50 = 48 nM T31391 CF4NR7 49797107 IC50 = 26 nM T31391 CV9QW6 49797108 IC50 = 31 nM T31391 CJZA65 49797109 IC50 = 1100 nM T31391 CBS36X 49797110 IC50 = 38 nM T31391 C0STP5 49797111 IC50 = 29 nM T31391 C7KV5R 49797112 IC50 = 320 nM T31391 CJPX53 49797113 IC50 = 570 nM T31391 C2OI0Y 49797114 IC50 = 25 nM T31391 CW20FJ 49797115 IC50 = 34 nM T31391 C9P6VU 49797116 IC50 = 49 nM T31391 C67SIA 49797117 IC50 = 74 nM T31391 CCI8Y0 49797118 IC50 = 67 nM T31391 CE10UF 49797119 IC50 = 37 nM T31391 CLH0V3 49797120 IC50 = 120 nM T31391 C2N8WX 49797121 IC50 = 26 nM T31391 CNCE06 49797122 IC50 = 90 nM T31391 C76UAB 49797123 IC50 = 69 nM T31391 CHWT89 49797124 IC50 = 92 nM T31391 C1Z6NE 49797125 IC50 = 61 nM T31391 C25MQG 49797126 IC50 = 229 nM T31391 COL54B 49797127 IC50 = 117 nM T31391 C5OUQ3 49797128 IC50 = 52 nM T31391 C3NMI8 49797173 Ki = 12 nM T31391 C1E3YB 49797174 Ki = 6 nM T31391 CVD0I1 49797175 Ki = 3.6 nM T31391 CH02OC 49797176 Ki = 4.7 nM T31391 CY1OJ5 49797177 Ki = 1.3 nM T31391 CL8TW4 49797178 Ki < 140 nM T31391 C25ZSD 49797191 IC50 = 203 nM T31391 C0OJX9 49797192 IC50 = 8 nM T31391 C7GZ4B 49797193 IC50 = 19 nM T31391 CVT2E5 49797194 IC50 = 40 nM T31391 C75MGE 49797195 IC50 = 13 nM T31391 CVS70C 49797196 IC50 = 13 nM T31391 C42QPW 49797197 IC50 = 70 nM T31391 C6ZGL5 49797198 IC50 = 52 nM T31391 C1B5NH 49797199 IC50 = 31 nM T31391 CGQN24 49797200 IC50 = 560 nM T31391 CS2AI5 49797201 IC50 = 1210 nM T31391 CM7RE3 49797202 IC50 = 1830 nM T31391 CGM9E7 49797203 IC50 = 3050 nM T31391 COU0I6 49797204 IC50 = 19 nM T31391 C3XML2 49797205 IC50 = 19 nM T31391 CP0O2F 49797223 IC50 = 210 nM T31391 CTH7I8 49797224 IC50 = 58 nM T31391 CG9P7O 49797225 IC50 = 144 nM T31391 C3A2QK 49797226 IC50 = 125 nM T31391 C4NOK2 49797227 IC50 = 111 nM T31391 CB13PO 49797228 IC50 = 67 nM T31391 C47VOG 49797229 IC50 = 463 nM T31391 CD2CL1 49797230 IC50 = 650 nM T31391 C0LK6B 49797231 IC50 = 14 nM T31391 CON0A6 49797232 IC50 = 37 nM T31391 C4AVU3 49797233 IC50 = 90 nM T31391 CQ93MI 49797234 IC50 = 82 nM T31391 CO2JV8 49797235 IC50 = 63 nM T31391 C27LDC 49797236 IC50 = 54 nM T31391 CA5GM6 49797237 IC50 = 3700 nM T31391 CT8PW1 49797238 IC50 = 7 nM T31391 CJQ38S 49797239 IC50 = 12 nM T31391 CT65MR 49797240 IC50 = 130 nM T31391 C08IFZ 49797241 IC50 = 43 nM T31391 CA4E8M 49797242 IC50 = 13 nM T31391 CN8FR2 49797243 IC50 = 22 nM T31391 C37MDP 49797244 IC50 = 5 nM T31391 CM41RN 49797245 IC50 = 2 nM T31391 C59JEK 49797246 IC50 = 8 nM T31391 CUMH43 49797248 IC50 = 8 nM T31391 CM59PE 49797249 IC50 = 5 nM T31391 CN5K1S 49797250 IC50 = 31 nM T31391 CT5HY0 49797251 IC50 = 6 nM T31391 C0E5PY 49797252 IC50 = 9 nM T31391 C3E5JB 49797253 IC50 = 16 nM T31391 CA8P5N 49797344 IC50 = 870 nM T31391 CJL2B8 49797345 IC50 = 430 nM T31391 CT79YI 49797346 IC50 = 25 nM T31391 C93VJO 49797347 IC50 = 160 nM T31391 CDI52A 49797348 IC50 = 300 nM T31391 C7ATK9 49797349 IC50 = 160 nM T31391 C2Y3DS 49797350 IC50 = 600 nM T31391 CA4CE3 49797351 IC50 = 150 nM T31391 C3A8YT 49797352 IC50 = 210 nM T31391 C1Z8HB 49797353 IC50 = 48 nM T31391 CC0T8H 49797354 IC50 = 330 nM T31391 C92QND 49797355 IC50 = 1490 nM T31391 C2HPE8 49797356 IC50 = 1280 nM T31391 C9UXH2 49797357 IC50 = 440 nM T31391 CTYO37 49797358 IC50 = 24 nM T31391 C1K4FR 49797359 IC50 = 22 nM T31391 CJ2D0P 49797360 IC50 = 74 nM T31391 CA3Q2W 49797361 IC50 = 29 nM T31391 CNMF62 49797362 IC50 = 21 nM T31391 C3HU6X 49797446 IC50 = 1490 nM T31391 C3U1KQ 49797450 IC50 = 525 nM T31391 C76KMB 49797451 IC50 = 17 nM T31391 C02MPV 49797452 IC50 = 122 nM T31391 CLVF17 49797501 IC50 = 9 nM T31391 CR0AK2 49797502 IC50 = 6 nM T31391 CM1Y7K 49797503 IC50 = 7 nM T31391 CUSI73 49797504 IC50 = 10 nM T31391 CJ0DX6 49797505 IC50 = 22 nM T31391 C2A7LE 49797506 IC50 = 7 nM T31391 CU4M3T 49797507 IC50 = 15 nM T31391 C8GCS5 49797508 IC50 = 17 nM T31391 CTP9L2 49797509 IC50 = 31 nM T31391 CT76PM 49797510 IC50 = 8 nM T31391 C4K0QT 49797511 IC50 = 19 nM T31391 CLHB50 49797512 IC50 = 37 nM T31391 CC56FE 49797513 IC50 = 11 nM T31391 C4T6AB 49797514 IC50 = 8 nM T31391 C41VHF 49797515 IC50 = 31 nM T31391 CBD9H2 49797516 IC50 = 12 nM T31391 CAOC90 49797517 IC50 = 31 nM T31391 C0F5QX 49797518 IC50 = 12 nM T31391 C7T5XW 49797519 IC50 = 16 nM T31391 CM6SF5 49797520 IC50 = 25 nM T31391 CQZN45 49797521 IC50 = 14 nM T31391 CG64BU 49797522 IC50 = 13 nM T31391 C5G3MA 49797524 IC50 = 5 nM T31391 CO42DE 49797525 IC50 = 35 nM T31391 C5L1EP 49797526 IC50 = 40 nM T31391 CTWR80 49797527 IC50 = 6 nM T31391 CPIC42 49797528 IC50 = 7 nM T31391 C5N1ZB 49797529 IC50 = 5 nM T31391 CU72EZ 49797596 IC50 = 17 nM T31391 C6AZ2C 49797599 IC50 = 52 nM T31391 CR86PO 49797604 IC50 = 22 nM T31391 C6DJX7 49797605 IC50 = 4.2 nM T31391 CK3ZI1 49797607 IC50 = 7.1 nM T31391 C7AD0C 49797610 IC50 = 53 nM T31391 C4XHO5 49797612 IC50 = 8 nM T31391 C7VL5U 49797614 IC50 = 28 nM T31391 CY09JE 49797615 IC50 = 47 nM T31391 C1ZLF0 49797616 IC50 = 13 nM T31391 CN48OE 49797627 IC50 = 77 nM T31391 CV6I0O 49797630 IC50 = 14 nM T31391 CAG1U7 49797631 IC50 = 56 nM T31391 C8JNU1 49797636 IC50 = 68 nM T31391 C0DN5G 49797642 IC50 = 47 nM T31391 CJVS96 49797644 IC50 = 18 nM T31391 CBRT78 49797650 IC50 = 8.6 nM T31391 CZW93Y 49797653 IC50 = 30 nM T31391 COM5Q7 49836030 IC50 = 27 nM T31391 CKZJ30 49837952 IC50 = 16 nM T31391 CXR05H 49837954 IC50 = 11 nM T31391 C4QSP1 49837961 IC50 = 10 nM T31391 C1WSF0 49843627 IC50 = 300 nM T31391 C31PHS 49843629 IC50 = 101 nM T31391 CDAK59 49843631 IC50 = 124 nM T31391 CSWR53 49845007 IC50 = 2300 nM T31391 C02RWO 49845009 IC50 = 1060 nM T31391 CG5O9N 49845011 IC50 = 1240 nM T31391 C9ST1E 49845161 IC50 = 460 nM T31391 C64NVQ 49845166 IC50 = 1236 nM T31391 C3CVF2 49845349 IC50 = 360 nM T31391 CTDR85 49862539 Ki = 73 nM T31391 CT8Q9N 49862713 Ki = 73 nM T31391 C0OB8C 49862714 Ki = 50 nM T31391 CJ58AG 49862715 Ki = 50 nM T31391 C42TSR 49862716 Ki = 31 nM T31391 CPU7F6 49862790 Ki = 29 nM T31391 C4FZY2 49862791 Ki = 442 nM T31391 CF40YM 49862792 Ki = 106 nM T31391 CK0GC5 49864113 Ki = 5.4 nM T31391 CK1CD3 50925423 IC50 = 23 nM T31391 C8XA7H 50942035 IC50 = 13 nM T31391 CFT4L5 50970490 IC50 = 93 nM T31391 C7T6PI 50994092 IC50 = 1.1 nM T31391 C67CTP 51032641 IC50 = 88.82 nM T31391 C1ECS9 51050448 IC50 = 66 nM T31391 CL4S9Y 51050450 IC50 = 39 nM T31391 CWZ76P 51050544 IC50 = 23 nM T31391 CT3D7J 51050546 IC50 = 8.7 nM T31391 C5O1PJ 51050548 IC50 = 9.6 nM T31391 CR6ZG8 51050550 IC50 = 6.6 nM T31391 CY3W8O 51051127 IC50 = 57 nM T31391 C2GNK6 51051129 IC50 = 58 nM T31391 CLU39H 51051131 IC50 = 18 nM T31391 C5PRF8 51051132 IC50 = 18 nM T31391 CYF04M 51051134 IC50 = 5.7 nM T31391 CPCY75 51051136 IC50 = 4.4 nM T31391 C7JM3I 51051236 IC50 = 19 nM T31391 CZ5HJ0 51051238 IC50 = 4.6 nM T31391 C1OUG5 51051240 IC50 = 2.5 nM T31391 C6GAP9 51051329 IC50 = 20 nM T31391 C9KPJ6 51051331 IC50 = 10 nM T31391 C85CEJ 51346970 IC50 = 55 nM T31391 C4PFT3 51346971 IC50 = 94 nM T31391 CLG9I5 51355035 IC50 = 89.5 nM T31391 CLND76 51356956 IC50 = 44 nM T31391 CH92AI 51356957 IC50 = 80 nM T31391 CH89VX 51356958 IC50 = 686 nM T31391 C5D4HV 51356959 IC50 = 674 nM T31391 C03ROM 51356960 IC50 < 50000 nM T31391 C8WOG2 51356962 IC50 = 674 nM T31391 CJ0Q4A 52918281 IC50 = 50.66 nM T31391 C4VC2U 52942435 IC50 = 87 nM T31391 C2B6EX 52943488 Ki = 11 nM T31391 CGOM96 52943515 IC50 = 114 nM T31391 C56CXU 52943631 IC50 = 151 nM T31391 CHD7O6 52943758 IC50 = 13 nM T31391 C4I6ML 52944843 IC50 = 23 nM T31391 C57XSM 52944845 IC50 = 122 nM T31391 CT6SQ3 52944941 IC50 = 28 nM T31391 C7RJM9 52945660 IC50 = 10 nM T31391 C9OAF1 52946149 IC50 = 1.8 nM T31391 CBVC96 52946447 IC50 = 10 nM T31391 CC56BV 52946866 IC50 > 100000 nM T31391 CC7N8S 52948914 IC50 = 36 nM T31391 C4LVO6 52948971 IC50 = 12 nM T31391 CTU0J1 52949742 IC50 = 103 nM T31391 CD4HQ1 53233695 IC50 = 3100 nM T31391 C89KWN 53233798 IC50 = 4000 nM T31391 CEFX05 53311069 IC50 = 1100 nM T31391 CQL50R 53311070 IC50 > 100000 nM T31391 C1Q4WK 53311071 IC50 = 20000 nM T31391 C67LHZ 53311072 IC50 = 530 nM T31391 CQ0ZJ2 53311073 IC50 = 5200 nM T31391 C7PMY1 53311074 IC50 = 38000 nM T31391 CWN9H7 53311140 IC50 = 100 nM T31391 CAL51C 53311141 IC50 = 16000 nM T31391 C2SXV0 53311142 IC50 = 88000 nM T31391 C7AEF8 53311143 IC50 > 100000 nM T31391 C5IOZ6 53311144 IC50 = 3400 nM T31391 CVR4H3 53311222 IC50 = 430 nM T31391 CNX08H 53311223 IC50 = 110 nM T31391 CET6W5 53311225 IC50 = 2500 nM T31391 C3RZS4 53311226 IC50 = 480 nM T31391 CHR17Y 53311227 IC50 = 13 nM T31391 C3HGW8 53312238 IC50 > 100000 nM T31391 CM03UX 53312239 IC50 > 100000 nM T31391 C9K4CZ 53312243 IC50 > 100000 nM T31391 CU4BS2 53312323 IC50 = 23000 nM T31391 CF5I6O 53312326 IC50 = 22 nM T31391 C6PSL2 53312327 IC50 > 100000 nM T31391 C0WYS5 53312328 IC50 = 45 nM T31391 CI0Z2A 53317343 IC50 > 50000 nM T31391 CLZ1M4 53317345 IC50 > 50000 nM T31391 CO3SY5 53317346 IC50 > 50000 nM T31391 C4M7TX 53317347 IC50 > 50000 nM T31391 C37HQG 53317348 IC50 > 50000 nM T31391 CYC69Q 53317564 IC50 = 85 nM T31391 C0QOV9 53317565 IC50 = 180 nM T31391 CURC70 53317566 IC50 = 400 nM T31391 C3ZK1W 53317575 IC50 = 120 nM T31391 CBQ0J7 53317579 IC50 = 280 nM T31391 CIY9F7 53317580 IC50 = 57 nM T31391 C5DMS9 53317581 IC50 = 450 nM T31391 C1XD9W 53317582 IC50 = 82 nM T31391 CR0O8T 53317583 IC50 = 18 nM T31391 CHW98L 53317619 IC50 = 13 nM T31391 C9AB1E 53317627 IC50 = 488 nM T31391 C0XQ2B 53318462 IC50 = 22.53 nM T31391 CJO28A 53318492 IC50 = 29.92 nM T31391 C45YDV 53318494 IC50 = 52.34 nM T31391 C6H4ZL 53318496 IC50 = 30.03 nM T31391 CYBP96 53318498 IC50 = 36.43 nM T31391 C9GLH7 53318841 IC50 = 84 nM T31391 C06TDE 53318842 IC50 = 150 nM T31391 C73TER 53318856 IC50 = 110 nM T31391 CC56NE 53318863 IC50 = 110 nM T31391 C4UJI8 53318864 IC50 = 310 nM T31391 C8CZ2A 53318865 IC50 = 110 nM T31391 CLVY47 53318866 IC50 = 51 nM T31391 CQC8N4 53318918 IC50 = 80 nM T31391 C7P2UE 53318921 IC50 = 1400 nM T31391 CP67YM 53318983 IC50 > 50000 nM T31391 C6SJ4Z 53318987 IC50 = 74 nM T31391 CM7S5W 53319067 IC50 = 110 nM T31391 C85NSB 53319824 IC50 = 37.54 nM T31391 CTW2R8 53319826 IC50 = 46.89 nM T31391 CW83TR 53319828 IC50 = 15.8 nM T31391 CC59LI 53319949 IC50 > 50000 nM T31391 CNW4K5 53319950 IC50 > 50000 nM T31391 CQK53D 53319951 IC50 > 50000 nM T31391 CD9LA8 53320113 IC50 > 50000 nM T31391 C1X3NE 53320178 IC50 = 120 nM T31391 C1P8BK 53320179 IC50 = 110 nM T31391 C50UBZ 53320180 IC50 = 140 nM T31391 C2JTR7 53320181 IC50 = 260 nM T31391 C0TYJ5 53320182 IC50 = 77 nM T31391 C7RSX2 53320183 IC50 = 72 nM T31391 CJU34O 53320232 IC50 = 19 nM T31391 C8ML9Y 53321113 IC50 = 45.2 nM T31391 CF0B3T 53321115 IC50 = 46.61 nM T31391 CEO6M2 53321117 IC50 = 22.76 nM T31391 CFPY75 53321119 IC50 = 17.83 nM T31391 CXZ47P 53321201 IC50 < 50000 nM T31391 CJ2V8E 53321202 IC50 = 937 nM T31391 CGVE79 53321203 IC50 < 50000 nM T31391 CP12HY 53321204 IC50 < 50000 nM T31391 C0XLS2 53321252 IC50 < 50000 nM T31391 CNT89R 53321253 IC50 > 50000 nM T31391 CO58YD 53321254 IC50 > 50000 nM T31391 C9XGE4 53321472 IC50 = 140 nM T31391 CY0ZV9 53321485 IC50 = 170 nM T31391 CK0OB2 53321486 IC50 = 38 nM T31391 CNK34J 53321487 IC50 = 260 nM T31391 C7EO3D 53321495 IC50 = 140 nM T31391 C3M7PQ 53321496 IC50 = 850 nM T31391 C0NUQ7 53321497 IC50 = 330 nM T31391 C31DSJ 53321498 IC50 = 450 nM T31391 C2ZKV9 53321499 IC50 = 71 nM T31391 CGA05O 53321545 IC50 = 216 nM T31391 CAU2F0 53321549 IC50 = 12 nM T31391 CB76JK 53321550 IC50 = 59 nM T31391 C50RJL 53321566 IC50 = 13 nM T31391 C3QT0R 53321621 IC50 = 140 nM T31391 CF2GQ1 53321670 IC50 = 22 nM T31391 C4UA2C 53322441 IC50 = 12.4 nM T31391 CF5M0P 53322443 IC50 = 33.17 nM T31391 CQK38R 53322445 IC50 = 33.25 nM T31391 C3OTG6 53322447 IC50 = 47.27 nM T31391 CKT3E2 53322456 IC50 = 77.06 nM T31391 CR9TY2 53322529 IC50 > 50000 nM T31391 C56URQ 53322530 IC50 < 50000 nM T31391 C1ZIS9 53322575 IC50 > 50000 nM T31391 C2MA6T 53322742 IC50 > 50000 nM T31391 CXIS21 53322758 IC50 = 730 nM T31391 CY71QL 53322814 IC50 = 130 nM T31391 CLU96Y 53322820 IC50 = 270 nM T31391 C8YVF1 53322821 IC50 = 290 nM T31391 C4QS6V 53322822 IC50 = 220 nM T31391 C62JTB 53322823 IC50 = 710 nM T31391 CT14FU 53322824 IC50 = 690 nM T31391 CXJ1F8 53322825 IC50 = 670 nM T31391 C3K1VY 53322826 IC50 = 21 nM T31391 CC09IP 53322885 IC50 = 41 nM T31391 C9N6HK 53322952 IC50 = 70 nM T31391 C7NUF3 53323807 IC50 = 28.6 nM T31391 C3QGT8 53323865 IC50 < 50000 nM T31391 C0FOV2 53323866 IC50 < 50000 nM T31391 CZ4I5J 53323915 IC50 < 50000 nM T31391 C4E8OK 53323916 IC50 > 50000 nM T31391 CB7HG9 53323917 IC50 > 50000 nM T31391 C9LU8M 53324129 IC50 = 99 nM T31391 CCY7M0 53324130 IC50 = 130 nM T31391 C4F1QK 53324142 IC50 = 500 nM T31391 CZN71C 53324143 IC50 = 670 nM T31391 CG83JZ 53324144 IC50 = 140 nM T31391 CE8J1D 53324145 IC50 = 140 nM T31391 C0Y3AC 53324153 IC50 = 120 nM T31391 C9O1IW 53324154 IC50 = 910 nM T31391 CTW5G0 53324155 IC50 = 130 nM T31391 C2DPZ0 53324156 IC50 = 54 nM T31391 C9A4JG 53324203 IC50 = 28 nM T31391 CPCE78 53324209 IC50 = 47 nM T31391 C6CJ0H 53324210 IC50 = 1.6 nM T31391 CL5Z8N 53324211 IC50 = 39 nM T31391 CV7UM8 53324212 IC50 = 37 nM T31391 C98EJV 53324213 IC50 = 13 nM T31391 CSN28M 53324293 IC50 = 2400 nM T31391 C2FRA0 53324311 IC50 > 50000 nM T31391 CDW31Y 53325018 IC50 < 50000 nM T31391 C76TDZ 53325194 IC50 < 50000 nM T31391 CJWL87 53325195 IC50 > 50000 nM T31391 CBT0Z8 53325196 IC50 > 50000 nM T31391 C2N5BX 53325197 IC50 > 50000 nM T31391 CF65NE 53325325 IC50 = 77 nM T31391 C25OJW 53325399 IC50 = 430 nM T31391 CXW5O9 53325446 IC50 = 280 nM T31391 C1SO0C 53325447 IC50 = 570 nM T31391 C1S3WB 53325453 IC50 = 200 nM T31391 C2KFW6 53325454 IC50 = 75 nM T31391 C4ZFR5 53325455 IC50 = 78 nM T31391 CPS51R 53325503 IC50 = 153 nM T31391 CW8TM9 53325504 IC50 = 26 nM T31391 CCOQ72 53325553 IC50 = 26.17 nM T31391 C5UB1G 53325568 IC50 < 50000 nM T31391 C1Z4RT 53326344 IC50 = 15.09 nM T31391 CX6Q3E 53326370 IC50 = 75.35 nM T31391 C30OEU 53326372 IC50 = 26.64 nM T31391 CL7T1U 53326374 IC50 = 33.78 nM T31391 CJP5V7 53326443 IC50 < 50000 nM T31391 C65JNF 53326490 IC50 > 50000 nM T31391 CYIA49 53326515 IC50 = 2.8 nM T31391 CV0H8P 53326691 IC50 = 110 nM T31391 C3ZWN6 53326704 IC50 = 100 nM T31391 C73SKG 53326705 IC50 = 1300 nM T31391 CG9V4W 53326706 IC50 = 110 nM T31391 C5K8CP 53326713 IC50 = 100 nM T31391 CHCE65 53326766 IC50 = 51 nM T31391 C4LCU1 53326767 IC50 = 1.2 nM T31391 C9UBW8 53326841 IC50 > 50000 nM T31391 C1HYV2 53326876 IC50 > 50000 nM T31391 CN12AO 53353383 IC50 = 255 nM T31391 C51GUC 53354365 IC50 = 67 nM T31391 CRJ5P9 53354369 IC50 = 102 nM T31391 C4G2HT 53354470 IC50 = 57 nM T31391 CUC1N3 53356519 Ki = 0.37 nM T31391 CSD1Q4 53357353 IC50 = 1.1 nM T31391 C5P9VZ 53465973 IC50 > 100000 nM T31391 C7OBF2 53465974 IC50 > 100000 nM T31391 CF5YJ8 53465975 IC50 > 100000 nM T31391 C5XER7 53466046 IC50 > 100000 nM T31391 CJ9T8M 53466047 IC50 > 50000 nM T31391 CP1CL8 53466049 IC50 > 100000 nM T31391 CPSQ16 53466050 IC50 > 100000 nM T31391 C4UC1P 53466119 IC50 > 100000 nM T31391 C59SML 53466121 IC50 > 100000 nM T31391 C7JPY2 53466122 IC50 > 100000 nM T31391 CYZK63 53466123 IC50 > 50000 nM T31391 CVJ0D5 53466193 IC50 > 100000 nM T31391 C2XE8Y 53466195 IC50 > 100000 nM T31391 C0P2YE 53466196 IC50 > 100000 nM T31391 CPA0K4 53466271 IC50 > 100000 nM T31391 CYG36O 53466361 IC50 = 17700 nM T31391 C5J9EB 53770701 IC50 = 510 nM T31391 CEK45S 54294055 IC50 = 87000 nM T31391 CRL42P 54573912 IC50 = 400 nM T31391 CUZS62 54580221 IC50 = 19 nM T31391 CG3S0X 54580222 IC50 = 0.7 nM T31391 CAQ8U7 54580310 IC50 = 21300 nM T31391 CX6K2C 54580311 IC50 = 26200 nM T31391 CS21IF 54580575 IC50 = 44.8 nM T31391 COZ98J 54580576 IC50 = 116 nM T31391 C2TSH1 54580577 IC50 = 54.1 nM T31391 CZL0N3 54580578 IC50 = 30.8 nM T31391 CNAQ35 54580579 IC50 = 7.4 nM T31391 CT24DU 54581222 IC50 = 7 nM T31391 CABF19 54581317 IC50 = 32700 nM T31391 C9JBG4 54581584 IC50 = 26.7 nM T31391 CJZ4S8 54582330 IC50 = 29100 nM T31391 C4L9SF 54582574 IC50 = 38.5 nM T31391 C0LQ9Z 54582575 IC50 = 13.7 nM T31391 CG84BL 54582898 IC50 = 12 nM T31391 CE5X6H 54583545 IC50 = 33.9 nM T31391 CB52YA 54583546 IC50 = 12 nM T31391 CST5M7 54584528 IC50 = 311 nM T31391 CV10YB 54585462 IC50 = 42.7 nM T31391 CG6M8J 54585463 IC50 = 38.9 nM T31391 CLCU50 54585464 IC50 = 1.3 nM T31391 CPWB63 54586434 IC50 = 50.7 nM T31391 C4G2PK 54586435 IC50 = 29 nM T31391 C71GKO 54586787 IC50 = 3 nM T31391 C4B2EW 54587461 IC50 = 92.6 nM T31391 C7VL9M 54587462 IC50 = 48.9 nM T31391 C04FAR 54587463 IC50 = 33.8 nM T31391 CQH56N 54698732 IC50 = 730 nM T31391 CY0ZH5 54698792 IC50 = 2950 nM T31391 C5UW0D 56652661 IC50 = 45 nM T31391 CMT0J9 56656630 IC50 = 133.6 nM T31391 C1QX0O 56657809 IC50 = 2 nM T31391 CU74VH 56658024 IC50 > 100000 nM T31391 CF6PV5 56658026 IC50 > 100000 nM T31391 C2KI8Y 56658028 IC50 > 100000 nM T31391 CY4E6U 56658138 IC50 > 100000 nM T31391 C5OT6W 56658248 IC50 = 26 nM T31391 C07KTW 56658249 IC50 > 1000 nM T31391 C1UDJ5 56659853 IC50 = 34 nM T31391 CX31TJ 56661748 IC50 = 0.34 nM T31391 COI5B0 56663604 IC50 = 65.1 nM T31391 C3VIA8 56663606 IC50 = 68.1 nM T31391 CD31AI 56663612 IC50 = 29.3 nM T31391 C52TBZ 56664349 IC50 = 20.4 nM T31391 C1PI4L 56664962 IC50 > 100000 nM T31391 C8GPO1 56665883 IC50 = 190 nM T31391 CA0BO6 56666264 IC50 > 100000 nM T31391 C8F5QV 56666543 IC50 = 4.2 nM T31391 C76MXW 56666747 IC50 = 49 nM T31391 C8DB0L 56670173 IC50 = 57 nM T31391 CJ9Q3V 56670497 IC50 = 47.8 nM T31391 CNL7D4 56671283 IC50 = 68.6 nM T31391 CXH5W7 56671896 IC50 > 100000 nM T31391 CMW3T8 56673186 IC50 > 100000 nM T31391 C1Q4XU 56673980 IC50 = 165.6 nM T31391 CP87EK 56674589 IC50 = 60.1 nM T31391 C2B6PY 56674700 IC50 = 34.8 nM T31391 C3OHT5 56675121 IC50 = 82.4 nM T31391 CBK31U 56675279 IC50 > 100000 nM T31391 CW8KU6 56675536 IC50 > 50000 nM T31391 C7WCK5 56676440 IC50 = 790 nM T31391 CH13RF 56676769 IC50 = 26 nM T31391 CX92YZ 56676772 IC50 = 2.7 nM T31391 CAO6M3 56677318 IC50 = 53.5 nM T31391 CPT94R 56678428 IC50 = 44.5 nM T31391 CN9S8A 56679836 IC50 > 100000 nM T31391 CF08YD 56680615 IC50 = 25.8 nM T31391 CZ1P7K 56851484 IC50 = 72 nM T31391 CU61OI 56851486 IC50 = 94 nM T31391 C9OL5C 56962798 IC50 = 10 nM T31391 CQX8J0 57385070 IC50 = 13.78 nM T31391 CPS89B 57385071 IC50 = 2.64 nM T31391 CNU9C0 57385072 IC50 = 2.34 nM T31391 CG5MT6 57385073 IC50 = 1.4 nM T31391 CQZ09L 57390626 IC50 = 80 nM T31391 CWR4E5 57390923 Ki = 0.55 nM T31391 C0RAD8 57390924 Ki = 0.3 nM T31391 C2AR3V 57391609 IC50 = 5.5 nM T31391 CKPB03 57391802 IC50 = 4 nM T31391 C8SW9E 57391803 IC50 = 10 nM T31391 C5UWC6 57391804 IC50 = 1 nM T31391 C78QEY 57391805 IC50 = 25 nM T31391 CYAQ83 57391806 IC50 = 20 nM T31391 COL58X 57391831 IC50 = 1 nM T31391 C5U6RF 57392407 IC50 = 13 nM T31391 CD0OT2 57392409 IC50 = 15 nM T31391 C4QYJ6 57392724 Ki = 0.27 nM T31391 CKS3X9 57393534 IC50 = 4 nM T31391 CM2EH0 57393535 IC50 = 250 nM T31391 CNP60T 57393564 IC50 = 10 nM T31391 CWDY79 57394441 Ki = 1.5 nM T31391 C5USX7 57395248 IC50 = 0.5 nM T31391 CJ80BU 57395249 IC50 = 1 nM T31391 C27MRL 57395273 IC50 = 20 nM T31391 CX5MG4 57395274 IC50 = 5 nM T31391 C40WGY 57395275 IC50 = 45 nM T31391 CZ23RJ 57395915 IC50 = 32 nM T31391 C8KMS2 57396206 Ki = 0.4 nM T31391 C0P8KM 57397016 IC50 = 2 nM T31391 CE85SV 57397017 IC50 = 2 nM T31391 C0J9MO 57397044 IC50 = 1 nM T31391 CCZ61A 57397045 IC50 = 8 nM T31391 CZJ1P7 57397046 IC50 = 9 nM T31391 C2QL6K 57397702 IC50 = 1.8 nM T31391 CBQ85O 57397704 IC50 = 11 nM T31391 C2ZE3R 57397706 IC50 = 28 nM T31391 CW97SN 57398006 Ki = 0.67 nM T31391 CSU2O9 57398779 IC50 = 2 nM T31391 C01KCU 57399665 Ki = 0.31 nM T31391 CDQ57A 57400458 IC50 = 3 nM T31391 CED9C4 57400459 IC50 = 2 nM T31391 CSEK63 57400487 IC50 = 4 nM T31391 CH6YT2 57400488 IC50 = 3 nM T31391 CX0N7O 57400489 IC50 = 60 nM T31391 C65ZFW 57401128 IC50 = 110 nM T31391 CYX43T 57401419 Ki = 0.29 nM T31391 CV2ME6 57402260 IC50 = 9 nM T31391 CQ1A8P 57402261 IC50 = 2 nM T31391 CW94QA 57402262 IC50 = 10 nM T31391 CMJA69 57402263 IC50 = 5 nM T31391 CV2CF5 57402294 IC50 = 23 nM T31391 C1T0AD 57403169 Ki = 0.43 nM T31391 C12QCM 57403170 Ki = 0.46 nM T31391 CX94UQ 57403171 Ki = 0.26 nM T31391 CX31VN 57403989 IC50 = 7.5 nM T31391 C4E7UI 57404016 IC50 = 2100 nM T31391 C5FHR8 57404017 IC50 = 15 nM T31391 C1L8YD 57404359 IC50 = 1650 nM T31391 C8SX7A 57404360 IC50 = 1100 nM T31391 C0Q1OZ 57404374 IC50 = 350 nM T31391 CXRS60 57406622 IC50 = 10 nM T31391 CNOX18 57406623 IC50 = 43.5 nM T31391 CZS03L 57406803 IC50 = 1.28 nM T31391 C80RBH 57406804 IC50 = 38.6 nM T31391 CMH17V 57406805 IC50 = 1.61 nM T31391 C2EX0S 57406806 IC50 = 19.3 nM T31391 CR6QP4 57406990 IC50 = 32 nM T31391 CFML71 57406991 IC50 = 8.15 nM T31391 C2PX9N 57406992 IC50 = 44.3 nM T31391 CHV47A 57406994 IC50 = 539 nM T31391 C0COE1 57407188 IC50 = 11.2 nM T31391 C5G3KT 57407189 IC50 = 9.31 nM T31391 C8MJK5 57407191 IC50 = 14.1 nM T31391 CVS34M 57407192 IC50 = 29.2 nM T31391 C7AZB3 57407370 IC50 = 82.2 nM T31391 CL0UA1 57525787 IC50 = 0.37 nM T31391 C75MLI 58874215 IC50 = 5.8 nM T31391 C9ZE7J 58874273 IC50 = 0.48 nM T31391 C3TSN9 58874353 IC50 = 14 nM T31391 C4KDJ8 58874386 IC50 = 0.55 nM T31391 COIQ05 58874405 IC50 = 418 nM T31391 C2I4JY 58874420 IC50 = 3.4 nM T31391 C0F5MP 58874435 IC50 = 4.8 nM T31391 CMW4N9 58874436 IC50 = 103 nM T31391 CZ4VD5 60032916 IC50 = 2.3 nM T31391 CI87CZ 61148520 Ki = 880 nM T31391 CAQ1O3 61148706 IC50 = 3.4 nM T31391 C68SUW 61174564 IC50 = 6.93 nM T31391 CXG48F 66545741 IC50 = 5.6 nM T31391 C2YPI7 66559296 IC50 = 0.61 nM T31391 CO2H1S 66559297 IC50 = 1.6 nM T31391 CRI16X 66559298 IC50 = 0.8 nM T31391 C5CX6V 66559299 IC50 = 0.59 nM T31391 CT15QA 66559300 IC50 = 0.39 nM T31391 CX48AY 66559301 IC50 = 1.2 nM T31391 CO0JP1 66559376 IC50 = 0.5 nM T31391 C2W0LI 66559377 IC50 = 0.55 nM T31391 C0NT6U 66559378 IC50 = 0.42 nM T31391 CG6EY9 66560524 IC50 = 0.61 nM T31391 CQMO80 66560608 IC50 = 0.73 nM T31391 CN4RL2 66560609 IC50 = 0.51 nM T31391 CS30FN 66560610 IC50 = 2.2 nM T31391 CZ4OU2 66560611 IC50 = 0.95 nM T31391 C02XCY 66560612 IC50 = 0.56 nM T31391 CW64RD 66561555 IC50 > 100000 nM T31391 C9GTI7 66561556 IC50 > 100000 nM T31391 CC85DI 66561873 IC50 = 2.3 nM T31391 C0QCA2 66561874 IC50 = 3.8 nM T31391 C5F6NR 66896083 Ki = 4 nM T31391 COIA16 66953432 IC50 = 645 nM T31391 C8CMU1 66953714 IC50 = 9 nM T31391 CUR3E1 66954220 IC50 = 1.6 nM T31391 CFW13I 66954232 IC50 = 100 nM T31391 CJY9L6 66962050 IC50 > 5000 nM T31391 CVOH80 66963065 IC50 = 290 nM T31391 CX7Z8R 67506840 IC50 = 4.5 nM T31391 C7Y1PN 67507142 IC50 = 4.3 nM T31391 CUIB42 67507176 IC50 = 0.2 nM T31391 CF92IB 67507913 IC50 = 0.26 nM T31391 C9SND1 68305755 IC50 > 100000 nM T31391 CP3E2X 68416066 IC50 = 0.3 nM T31391 CX34PR 68417107 IC50 = 0.94 nM T31391 CCS6K9 68417211 IC50 = 0.63 nM T31391 CUKP32 68417894 IC50 = 15 nM T31391 C54VZI 68417897 IC50 = 5 nM T31391 C69VWN 68418230 IC50 = 0.85 nM T31391 C6K0XY 68418986 IC50 = 3.4 nM T31391 C6U9SP 68419033 IC50 = 12 nM T31391 CFNU91 68419172 IC50 = 2.9 nM T31391 CZ7QX8 68419268 IC50 = 4 nM T31391 CEF87L 68419860 IC50 = 0.62 nM T31391 CH3Z7F 68658979 IC50 = 0.14 nM T31391 C31XFM 68828690 IC50 = 140 nM T31391 C7X2WD 68828739 IC50 = 100 nM T31391 C4C3BL 68828935 IC50 = 9.2 nM T31391 CR27HN 68829000 IC50 = 7.5 nM T31391 CVGE51 68829025 IC50 = 28 nM T31391 CU4K6C 68829197 IC50 = 55 nM T31391 CP1NA4 68829414 IC50 = 4.6 nM T31391 C45ICV 68829529 IC50 = 250 nM T31391 C06ZLV 68829605 IC50 = 720 nM T31391 C2K3PM 68829714 IC50 = 13 nM T31391 CZOG14 68829854 IC50 = 510 nM T31391 C6R7ZV 68829908 IC50 = 540 nM T31391 C5I4BK 68829917 IC50 = 620 nM T31391 CCE26Z 68830038 IC50 = 52 nM T31391 C1HR3S 68830304 IC50 = 17 nM T31391 C47PHV 68830457 IC50 = 170 nM T31391 CYV1A0 68830878 IC50 = 6.8 nM T31391 C62LNY 68830888 IC50 = 0.38 nM T31391 CL1VS3 68832119 IC50 = 630 nM T31391 C6HRX1 68845950 IC50 = 56 nM T31391 CDJI62 68914093 IC50 = 8.2 nM T31391 C2TOQ7 69089363 IC50 = 60000 nM T31391 CO95AZ 69442708 IC50 = 23 nM T31391 CY98ML 69445181 IC50 = 1.1 nM T31391 C6BR4W 69445419 IC50 = 30 nM T31391 CD42CX 69446073 IC50 = 29 nM T31391 CS85UC 69446132 IC50 = 470 nM T31391 CZ49VQ 69446166 IC50 = 3.7 nM T31391 CFL92T 69446285 IC50 = 80 nM T31391 CXM07R 69446326 IC50 = 87 nM T31391 CWTN63 69446993 IC50 = 17 nM T31391 CBQJ90 69447448 IC50 = 19 nM T31391 C67CPF 69576646 IC50 = 45.3 nM T31391 CW4O2C 69689410 Ki = 34 nM T31391 CQ2DM1 69890803 Ki = 910 nM T31391 C0C8JW 70293564 IC50 = 200 nM T31391 CK26FY 70295607 IC50 = 4 nM T31391 CV4X5S 70295927 IC50 = 7 nM T31391 CXSV41 70296244 IC50 = 3 nM T31391 C3SB1V 70296823 IC50 = 40 nM T31391 CL64SQ 70297489 IC50 = 19900 nM T31391 CXD5V6 70297609 IC50 = 2 nM T31391 CEG1L5 70330884 IC50 = 23 nM T31391 C5W6LY 70681316 IC50 = 14 nM T31391 CLO96S 70681357 IC50 > 100000 nM T31391 CWP41T 70681469 IC50 > 100000 nM T31391 C7Z2KY 70681470 IC50 > 100000 nM T31391 C97JFS 70682267 IC50 = 17 nM T31391 CE1FU2 70682268 IC50 = 17 nM T31391 CI8EQ5 70682492 IC50 = 45.3 nM T31391 C03SDB 70682493 IC50 = 67.7 nM T31391 CF0U3A 70682494 IC50 = 57.6 nM T31391 C8Z2UQ 70682495 IC50 = 57.4 nM T31391 C14AWU 70682667 IC50 = 31 nM T31391 C71BSM 70682668 IC50 = 723 nM T31391 C49RIG 70682669 IC50 = 14.3 nM T31391 C19XIQ 70683454 IC50 > 100000 nM T31391 C07ADL 70683455 IC50 > 100000 nM T31391 C4YW5T 70684349 IC50 = 200 nM T31391 C6W1CT 70684350 IC50 = 18000 nM T31391 C1GF3E 70684351 IC50 = 53 nM T31391 C2GUS0 70684568 IC50 = 212 nM T31391 CU1I5S 70684569 IC50 = 39 nM T31391 CM96VS 70684570 IC50 = 47.7 nM T31391 C1NHS4 70684571 IC50 = 42.2 nM T31391 C7HF3B 70684748 IC50 = 298 nM T31391 C74WUS 70684749 IC50 = 879 nM T31391 CL8OZ4 70684750 IC50 = 10.3 nM T31391 CV5T8O 70684751 IC50 = 13.2 nM T31391 CO2NK6 70685557 IC50 > 100000 nM T31391 CK0WX8 70685558 IC50 > 100000 nM T31391 CLF84U 70685559 IC50 > 100000 nM T31391 C0K7PS 70685560 IC50 > 100000 nM T31391 C2T0NS 70685696 IC50 > 100000 nM T31391 C1Q3ZO 70686506 IC50 = 6.2 nM T31391 CM90BQ 70686720 IC50 = 264 nM T31391 CNQ50W 70686721 IC50 = 569 nM T31391 CRA4G1 70686722 IC50 = 64.6 nM T31391 C5I9BL 70686723 IC50 = 24.9 nM T31391 CT2LK4 70686905 IC50 = 104 nM T31391 CVD76F 70687705 IC50 > 100000 nM T31391 C28GVW 70687706 IC50 > 100000 nM T31391 CLQC52 70688610 IC50 = 29 nM T31391 C6MZ4N 70688809 IC50 = 101 nM T31391 C3GY6A 70688810 IC50 = 103 nM T31391 CGQV87 70688811 IC50 = 31.2 nM T31391 CHL1T9 70688964 IC50 = 320 nM T31391 C76SEY 70688965 IC50 = 28 nM T31391 CDVF75 70688966 IC50 = 715 nM T31391 CK2UC9 70688967 IC50 = 869 nM T31391 CI0VF5 70688968 IC50 = 843 nM T31391 C8K4WF 70688969 IC50 = 74 nM T31391 CVYH31 70689717 IC50 = 23 nM T31391 CUY81P 70689750 IC50 > 100000 nM T31391 CX2O0Z 70689751 IC50 > 100000 nM T31391 C17YKW 70689752 IC50 > 100000 nM T31391 CYO5X6 70690674 IC50 = 59 nM T31391 C2J7FS 70690675 IC50 = 15 nM T31391 CL6KR9 70690676 IC50 = 0.3 nM T31391 CXE41O 70690893 IC50 = 30.5 nM T31391 C4QCP6 70691068 IC50 = 863 nM T31391 C7ROY0 70691069 IC50 = 100 nM T31391 CC0D7S 70691070 IC50 = 34 nM T31391 C87LMG 70691901 IC50 > 100000 nM T31391 CL5EG7 70691902 IC50 > 100000 nM T31391 CGND49 70691903 IC50 > 100000 nM T31391 CGT57B 70691904 IC50 > 100000 nM T31391 CT89CW 70691905 IC50 > 100000 nM T31391 C5WI6V 70691906 IC50 > 100000 nM T31391 C19FJC 70692822 IC50 = 48 nM T31391 C8JZ3Q 70692823 IC50 = 16 nM T31391 C7FIR6 70693034 IC50 = 85.7 nM T31391 CM3L1E 70693035 IC50 = 50.4 nM T31391 C3DV6C 70693036 IC50 = 56.4 nM T31391 C3MF7C 70693037 IC50 = 91.5 nM T31391 C5YQ9B 70693038 IC50 = 33.9 nM T31391 CEQ4N8 70693039 IC50 = 76.2 nM T31391 CYQO06 70693040 IC50 = 36.7 nM T31391 C0S9LO 70693199 IC50 = 890 nM T31391 CY7M8K 70693200 IC50 = 19 nM T31391 C4P5TC 70693201 IC50 = 863 nM T31391 CEB6L2 70693202 IC50 = 116 nM T31391 CQMV53 70693949 IC50 > 100000 nM T31391 CBP8U7 70693950 IC50 > 100000 nM T31391 C0I2CV 70693951 IC50 > 100000 nM T31391 CCB64G 70693952 IC50 > 100000 nM T31391 C3ZUK2 70693953 IC50 > 100000 nM T31391 CS76EN 70693954 IC50 > 100000 nM T31391 C27PFC 70693955 IC50 > 100000 nM T31391 CVY48R 70693956 IC50 > 100000 nM T31391 CIX3F9 70694853 IC50 = 6.5 nM T31391 CQJD92 70694854 IC50 = 20 nM T31391 C8JRC5 70695073 IC50 = 99.7 nM T31391 CA0W8R 70695074 IC50 = 65.4 nM T31391 CYB1P3 70695075 IC50 = 74.4 nM T31391 C4ETL9 70695076 IC50 = 113.9 nM T31391 C5ZN7P 70695277 IC50 = 107 nM T31391 C3S5EX 70695278 IC50 = 26 nM T31391 CC6B7L 70695279 IC50 = 694 nM T31391 CXG5O4 70695280 IC50 = 311 nM T31391 CA01KO 70696068 IC50 > 100000 nM T31391 CSW43K 70696069 IC50 = 13100 nM T31391 C1NGL5 70696903 IC50 = 2.1 nM T31391 CR6FY8 70697121 IC50 = 194 nM T31391 C2B5UF 70697122 IC50 = 291 nM T31391 CV38GW 70697123 IC50 = 52.6 nM T31391 CJ4M0N 70697124 IC50 = 50.6 nM T31391 C4GIH1 70697292 IC50 = 31 nM T31391 CALB67 70697293 IC50 = 11.6 nM T31391 C19ZWC 70789754 IC50 > 100000 nM T31391 C31UTS 71184301 IC50 = 250 nM T31391 C8LY1U 71184352 IC50 = 9 nM T31391 C9IRW7 71184590 IC50 = 40 nM T31391 C8BK4O 71184607 IC50 = 4200 nM T31391 CS29MW 71184623 IC50 = 15700 nM T31391 C08NDK 71184749 IC50 = 20 nM T31391 CP91OE 71203742 IC50 = 625 nM T31391 CP6G5W 71203746 IC50 = 11.2 nM T31391 C32UMV 71203748 IC50 = 1.7 nM T31391 C04XQY 71203752 IC50 = 27.4 nM T31391 CE2I0K 71203758 IC50 = 123 nM T31391 CIQ7O2 71203767 IC50 = 13.5 nM T31391 C5GEJ9 71203769 IC50 = 156.1 nM T31391 C7LKV0 71203783 IC50 = 10.6 nM T31391 CBK26E 71449262 IC50 = 160 nM T31391 CW8JE0 71449264 IC50 = 150 nM T31391 CD9C3R 71449266 IC50 = 6900 nM T31391 CBX46U 71449270 IC50 = 54 nM T31391 CT35BK 71449272 IC50 = 64 nM T31391 C6D0WY 71449276 IC50 = 22 nM T31391 C46QSR 71449278 IC50 = 660 nM T31391 CKR1E6 71449280 IC50 = 72 nM T31391 CAJ8F0 71449608 IC50 = 20 nM T31391 CM5DB6 71450086 IC50 > 100000 nM T31391 CQU0Z1 71450087 IC50 > 100000 nM T31391 C65BCE 71450089 IC50 > 100000 nM T31391 CP9K2W 71450603 IC50 = 12 nM T31391 C8GBF1 71450604 IC50 = 670 nM T31391 CA3LP4 71450605 IC50 = 94 nM T31391 CD80JE 71451064 IC50 = 90 nM T31391 CH83NV 71451066 IC50 = 13 nM T31391 CM86TF 71451071 IC50 = 400 nM T31391 C9BK1J 71451073 IC50 = 17 nM T31391 CLC2N8 71451900 IC50 > 100000 nM T31391 CMU63C 71451901 IC50 > 100000 nM T31391 CT5WU4 71451902 IC50 > 100000 nM T31391 CL0X3F 71451939 IC50 > 100000 nM T31391 C7ZN6W 71452445 IC50 = 41 nM T31391 CKVA72 71452446 IC50 = 250 nM T31391 CP5NS6 71452447 IC50 = 110 nM T31391 C61LNR 71452448 IC50 = 83 nM T31391 C2J3GF 71452890 IC50 > 10000 nM T31391 C4GQ5B 71452892 IC50 = 90 nM T31391 CEM2O9 71453723 IC50 > 100000 nM T31391 CB1EX7 71453762 IC50 > 100000 nM T31391 CN4FE7 71454208 IC50 = 24 nM T31391 CD4IE2 71454659 IC50 = 3500 nM T31391 C2GO8L 71454668 IC50 = 12 nM T31391 CT9YS3 71454883 IC50 = 16 nM T31391 CBOK64 71455456 IC50 > 100000 nM T31391 CD32GT 71455458 IC50 > 100000 nM T31391 CQA9L7 71455494 IC50 > 100000 nM T31391 C1LRH5 71455960 IC50 = 84 nM T31391 CGH7R6 71455961 IC50 = 55 nM T31391 CGKJ82 71456385 IC50 = 38 nM T31391 CCY8P7 71456387 IC50 = 8900 nM T31391 CIC59O 71456389 IC50 = 3.8 nM T31391 CNGO29 71456391 IC50 = 60 nM T31391 C7AU4I 71456393 IC50 = 17 nM T31391 CVIF92 71456398 IC50 > 10000 nM T31391 C0CHQ9 71456400 IC50 = 66 nM T31391 C4T7CO 71457236 IC50 > 100000 nM T31391 C3GAO1 71457237 IC50 > 100000 nM T31391 CE3MP2 71457238 IC50 > 100000 nM T31391 C42BSO 71457239 IC50 > 100000 nM T31391 C8VI9L 71457240 IC50 > 50000 nM T31391 CK0O9D 71457760 IC50 = 490 nM T31391 C59TGZ 71457761 IC50 = 16 nM T31391 C8O6HJ 71457762 IC50 = 59 nM T31391 CBKA19 71457763 IC50 = 190 nM T31391 CI15BH 71457764 IC50 = 160 nM T31391 C5T6QP 71457765 IC50 = 72 nM T31391 C87VPZ 71458224 IC50 = 51 nM T31391 C89DPI 71458226 IC50 = 10 nM T31391 CK6S7X 71458227 IC50 = 6.3 nM T31391 CB67AV 71458229 IC50 = 3.5 nM T31391 CLRE92 71458241 IC50 = 66 nM T31391 CW76HL 71458243 IC50 = 16 nM T31391 CIO50T 71459090 IC50 > 100000 nM T31391 CXIM97 71459091 IC50 > 100000 nM T31391 CJ6N1C 71459092 IC50 > 100000 nM T31391 CUB4V8 71459679 IC50 = 7.8 nM T31391 C10JPO 71459680 IC50 = 330 nM T31391 CWQ59G 71460084 IC50 = 25 nM T31391 CZ7E1K 71460086 IC50 = 56 nM T31391 CS89OV 71460088 IC50 = 21 nM T31391 C6Z8RT 71460094 IC50 = 271 nM T31391 CKXG80 71460143 IC50 = 0.32 nM T31391 CEY13Z 71460148 IC50 = 6.3 nM T31391 CEU0B1 71460149 IC50 > 1000 nM T31391 CSC3I7 71460901 IC50 > 100000 nM T31391 CG7VX2 71460902 IC50 > 100000 nM T31391 C5K3WJ 71460903 IC50 > 100000 nM T31391 C3UF9P 71460904 IC50 > 100000 nM T31391 CUJT52 71461398 IC50 = 1100 nM T31391 CQ6GA0 71461399 IC50 = 50 nM T31391 CJ07GY 71461805 IC50 = 110 nM T31391 C8LB7A 71461808 IC50 = 11 nM T31391 C79EIW 71461811 IC50 = 1.6 nM T31391 CPAN79 71461821 IC50 = 3400 nM T31391 C02ALK 71461822 IC50 = 340 nM T31391 C7TS9F 71462596 IC50 > 100000 nM T31391 C63SUR 71462597 IC50 > 100000 nM T31391 CZT3S0 71462641 IC50 > 100000 nM T31391 CY2W5V 71463119 IC50 = 390 nM T31391 C16PTB 71463120 IC50 = 280 nM T31391 CKZ17B 71463121 IC50 = 60 nM T31391 C4VKM3 71463122 IC50 = 100 nM T31391 CY4W8D 71520057 IC50 = 660 nM T31391 C0JUM4 71520123 IC50 = 1320 nM T31391 CZ0UG8 71520163 IC50 = 720 nM T31391 CQO90M 71550930 IC50 = 1.55 nM T31391 C57JVN 71566829 Ki = 4 nM T31391 CMX9E3 71566830 Ki = 18 nM T31391 CDJ2T7 71566831 Ki = 14 nM T31391 C2SB3J 71566832 Ki = 18 nM T31391 C3J4DA 71566833 Ki = 11 nM T31391 CGVS23 71566834 Ki = 18 nM T31391 C5EQ8X 71566966 Ki = 13 nM T31391 C1VG2P 71566967 Ki = 30 nM T31391 C8FH4K 71566968 Ki = 8 nM T31391 C6AQ8P 71566969 Ki = 5 nM T31391 CM3NB6 71566970 Ki = 4 nM T31391 C92TKQ 71566971 Ki = 2 nM T31391 CZN30Q 71567105 Ki = 35 nM T31391 CL0BY5 71567106 Ki = 38 nM T31391 C63UAJ 71567107 Ki = 15 nM T31391 CPLH40 71567235 Ki = 10 nM T31391 CNM83T 71568676 Ki = 98 nM T31391 CEGB81 71568801 Ki = 75 nM T31391 C1G5WV 71568802 Ki = 25 nM T31391 CGXB93 71568803 Ki = 23 nM T31391 C0XK9O 71568804 Ki = 18 nM T31391 CL57TN 71568805 Ki = 14 nM T31391 CGJQ86 71568806 Ki = 18 nM T31391 CY3ZG6 71582959 IC50 = 211.9 nM T31391 C97MES 71583061 IC50 = 44 nM T31391 CB1YX0 71583062 IC50 = 44.1 nM T31391 CX43IU 71583063 IC50 = 27.6 nM T31391 C3KW9P 71583064 IC50 = 48.2 nM T31391 CEK26O 71583065 IC50 = 7.05 nM T31391 C53UMG 71583066 IC50 = 139.2 nM T31391 C9IRB0 71583175 IC50 = 60.1 nM T31391 CY87XJ 71583176 IC50 = 14.5 nM T31391 CD5O8F 71583177 IC50 = 52.6 nM T31391 C85BGF 71583178 IC50 = 11.4 nM T31391 CA67NL 71583179 IC50 = 4.67 nM T31391 C17-APR 71583292 IC50 = 5.93 nM T31391 CUH48W 71583293 IC50 = 15.5 nM T31391 C9AKS7 71594483 IC50 = 22390 nM T31391 C7B8AO 71621488 IC50 > 100000 nM T31391 C8T2PW 71655265 IC50 = 2800 nM T31391 CVB75Q 71655394 IC50 = 1800 nM T31391 CH4ZS0 71655395 IC50 > 100000 nM T31391 CC93KJ 71655554 IC50 > 100000 nM T31391 CN90KH 71655555 IC50 > 100000 nM T31391 CUT37D 71655556 IC50 > 100000 nM T31391 C71OFQ 71655557 IC50 > 100000 nM T31391 C7R6HU 71655622 IC50 > 100000 nM T31391 C2NA1M 71655623 IC50 > 100000 nM T31391 CDF08H 71655624 IC50 > 100000 nM T31391 CBEX27 71655625 IC50 > 100000 nM T31391 CT6XB5 71655626 IC50 > 100000 nM T31391 C1ND2P 71655627 IC50 > 100000 nM T31391 CXZ8N4 71667081 IC50 > 100000 nM T31391 CJ9QU7 71667226 IC50 > 100000 nM T31391 CE0Z8G 71667227 IC50 > 100000 nM T31391 CL7CS3 71667230 IC50 > 100000 nM T31391 CB6SI5 71667231 IC50 > 100000 nM T31391 C75UWV 71667375 IC50 > 100000 nM T31391 C19CTI 71667376 IC50 > 100000 nM T31391 C69CJB 71667378 IC50 > 100000 nM T31391 C07HNK 71667379 IC50 > 100000 nM T31391 CK74SP 71667380 IC50 > 100000 nM T31391 CMYZ68 71667381 IC50 > 100000 nM T31391 CDI39U 71667510 IC50 > 100000 nM T31391 CT49CO 71674688 IC50 = 34650 nM T31391 C8YTW3 71716406 Ki = 109 nM T31391 CQR5A1 71718946 IC50 = 460 nM T31391 CXKP89 71719452 Ki = 695 nM T31391 C0V3ZW 71720156 IC50 = 860 nM T31391 C0SC3Q 71720681 Ki = 1201 nM T31391 C7BD2R 71720854 IC50 = 2 nM T31391 CW3JG7 71731241 IC50 > 10000 nM T31391 C3D4HJ 71731243 IC50 = 31.3 nM T31391 CU6BC5 71731355 IC50 = 22 nM T31391 C5TS9Y 71731356 IC50 = 3.1 nM T31391 C5RTY9 71731357 IC50 = 3.4 nM T31391 CD9F5X 71731476 IC50 = 10.8 nM T31391 C3IO9H 71731477 IC50 = 6.6 nM T31391 CVAD62 71731478 IC50 = 2 nM T31391 C1ON0X 71731479 IC50 = 9.1 nM T31391 CZYQ05 71731604 IC50 = 1.9 nM T31391 C40YRO 71731605 IC50 = 0.7 nM T31391 C9Q8MO 72164809 IC50 = 9.39 nM T31391 CL5X1Z 72164811 IC50 = 25.5 nM T31391 C7N8WB 72164813 IC50 = 17.61 nM T31391 C2R0NV 72164815 IC50 = 8.28 nM T31391 C4JLM5 72164817 IC50 = 19.54 nM T31391 C6RQ9A 72164819 IC50 = 7.56 nM T31391 C38GWP 72164942 IC50 = 3.79 nM T31391 C4T0MY 72164944 IC50 = 15.24 nM T31391 C0T4UW 72164946 IC50 = 10.45 nM T31391 CLV02R 72164948 IC50 = 6.05 nM T31391 CHPN10 72164950 IC50 = 20.84 nM T31391 CI78FQ 72165082 IC50 = 7.5 nM T31391 CN0VU2 72165084 IC50 = 4.35 nM T31391 C84SYX 72165086 IC50 = 8.57 nM T31391 C1RQA3 72165088 IC50 = 10.02 nM T31391 CH51ZR 72165090 IC50 = 15.7 nM T31391 C1HL2A 72188903 IC50 = 13100 nM T31391 CLS1A0 72188904 IC50 > 100000 nM T31391 CO15AV 72188905 IC50 = 0.66 nM T31391 CPDC28 72188906 IC50 = 140 nM T31391 CL7P3D 72193502 IC50 = 24400 nM T31391 C4AXB8 72193503 IC50 = 38000 nM T31391 CQC28P 72193504 IC50 = 2800 nM T31391 CV87PE 72193505 IC50 = 26600 nM T31391 C65DFP 72697059 IC50 = 18 nM T31391 CX07OC 72697060 IC50 = 248 nM T31391 CZ56DO 72697061 IC50 = 11 nM T31391 C1A2KX 72697062 IC50 = 17 nM T31391 CS5U1F 72697063 IC50 = 29 nM T31391 CA3HI1 72697064 IC50 = 75 nM T31391 CCZJ47 72697206 IC50 = 20 nM T31391 CWNZ91 72697207 IC50 = 21 nM T31391 C6BWI4 72697208 IC50 = 31 nM T31391 C9JA1Q 72697209 IC50 = 4 nM T31391 CF6A8N 72697210 IC50 = 4 nM T31391 CTMR03 72697211 IC50 = 42 nM T31391 CP9NV5 72697212 IC50 = 27 nM T31391 C1P8HS 72697352 IC50 = 46 nM T31391 CC7G3M 72697353 IC50 = 63 nM T31391 CXYO73 72697354 IC50 = 209 nM T31391 CAXV78 72697355 IC50 = 17 nM T31391 CGV09W 72697356 IC50 = 3 nM T31391 CIF9D7 72697357 IC50 = 4 nM T31391 CC8RA6 72697358 IC50 = 15 nM T31391 C1EC7S 72697359 IC50 = 292 nM T31391 C8CRO6 72697494 IC50 = 5 nM T31391 C03NKY 72697495 IC50 = 6 nM T31391 CP0MU3 72697496 IC50 = 125 nM T31391 CI60AK 72697497 IC50 = 94 nM T31391 CO19YK 72697498 IC50 = 22 nM T31391 C47IGZ 72697499 IC50 = 20 nM T31391 C65OPG 72697500 IC50 = 6 nM T31391 C3ZP7N 72697501 IC50 = 23 nM T31391 C7EF8C 72697646 IC50 = 60 nM T31391 C08IGP 72699737 IC50 = 1.98 nM T31391 CMT61I 72707535 IC50 = 198 nM T31391 CAEF04 72707536 IC50 = 2177.5 nM T31391 C7ARW4 72707537 IC50 = 1.2 nM T31391 C8D5PB 72725804 IC50 = 11900 nM T31391 CC10AZ 73345857 IC50 > 100000 nM T31391 CSZR98 73346173 IC50 = 48 nM T31391 C1L4RX 73346174 IC50 = 1 nM T31391 CX4F0Y 73347359 IC50 > 100000 nM T31391 C3XFM5 73347360 IC50 > 100000 nM T31391 CGNL10 73347698 IC50 = 720 nM T31391 CR09PJ 73348871 IC50 > 10000 nM T31391 CA79DR 73349143 IC50 = 265 nM T31391 CO5TB8 73349220 IC50 = 37 nM T31391 C06WRM 73350448 IC50 > 100000 nM T31391 C1T7LK 73350449 IC50 > 100000 nM T31391 CCIZ12 73350450 IC50 > 100000 nM T31391 CNC6B8 73350798 IC50 = 125 nM T31391 CDBV29 73350799 IC50 = 27 nM T31391 CYG04J 73352283 IC50 = 12600 nM T31391 CFV5U3 73353424 IC50 > 100000 nM T31391 CRS4O0 73353425 IC50 > 100000 nM T31391 C7X9ZG 73353601 IC50 > 1000 nM T31391 CV6BA3 73353756 IC50 = 37 nM T31391 C51QGP 73353757 IC50 = 27 nM T31391 CBK37N 73353758 IC50 = 64 nM T31391 CLYP23 73354936 IC50 > 100000 nM T31391 CLO76J 73355285 IC50 = 11 nM T31391 CCVT96 73355286 IC50 = 1.6 nM T31391 CH9W2R 73356494 IC50 > 100000 nM T31391 CKD46T 73356495 IC50 > 100000 nM T31391 CI0N6E 73356496 IC50 > 10000 nM T31391 C7R3ZT 76309823 Ki = 142000 nM T31391 CY0N9K 76311138 IC50 = 170 nM T31391 CWK7M6 76311139 IC50 = 50 nM T31391 CF5S9X 76313540 Ki = 61000 nM T31391 CIP4R0 76314754 IC50 = 40 nM T31391 C3HRA1 76314755 IC50 = 50 nM T31391 C1ZAC3 76317994 IC50 = 113760 nM T31391 C68JOX 76318341 IC50 = 30 nM T31391 CET31O 76318342 Ki = 3.5 nM T31391 CP0H8I 76320760 Ki = 4500 nM T31391 C9UGA3 76325642 IC50 = 113600 nM T31391 CNIP02 76325643 IC50 = 5 nM T31391 C08DYM 76325644 IC50 = 120 nM T31391 C3C7HE 76325645 Ki = 9 nM T31391 CWBL62 76327979 Ki = 6300 nM T31391 CW4M6E 76329221 IC50 = 390 nM T31391 C3LPR2 76331631 Ki = 5000 nM T31391 C7S6EY 76332265 IC50 = 4364 nM T31391 CH95ZJ 76336484 IC50 = 520 nM T31391 C4W7RE 77461184 IC50 = 8.5 nM T31391 CRG30N 86267497 IC50 = 148 nM T31391 C7JRH1 86267498 IC50 = 89.6 nM T31391 CTXI04 86267501 IC50 = 3 nM T31391 CO78UK 86267502 IC50 = 3.4 nM T31391 C7K2NA 86267708 IC50 = 3.8 nM T31391 CPS4U2 86268135 IC50 = 2290 nM T31391 C9GA1T 86268138 IC50 = 299 nM T31391 CBJ6N8 86268336 IC50 = 19.2 nM T31391 CA3L2Q 86268337 IC50 = 15.4 nM T31391 C6HCF9 86268525 IC50 = 18.6 nM T31391 CLG83C 86268944 IC50 = 4.9 nM T31391 C31OGJ 86279928 IC50 = 10.8 nM T31391 CB60OP 89488720 IC50 = 2.6 nM T31391 CIV7Y8 89668929 IC50 > 100000 nM T31391 C87GJT 89704940 IC50 > 100000 nM T31391 CHI7U9 89704942 IC50 > 100000 nM T31391 CSLI09 89704955 IC50 > 100000 nM T31391 CA3K7R 89704970 IC50 > 100000 nM T31391 CF89OD 89705045 IC50 > 100000 nM T31391 CK3Z8J 89705076 IC50 > 100000 nM T31391 CH6P0S 89705081 IC50 > 100000 nM T31391 C63DGS 89705096 IC50 > 100000 nM T31391 CND56S 89705098 IC50 > 100000 nM T31391 C0CKQ7 89705100 IC50 > 100000 nM T31391 C0CPD1 89705103 IC50 > 100000 nM T31391 C1IL7N 89705109 IC50 > 50000 nM T31391 CA48MR 89705136 IC50 > 100000 nM T31391 C5F9OA 89705152 IC50 > 100000 nM T31391 C1VSG5 89705179 IC50 > 100000 nM T31391 CHAS49 89705195 IC50 > 100000 nM T31391 C0RP1J 89705223 IC50 > 100000 nM T31391 CQO0I6 89705242 IC50 > 100000 nM T31391 C7DF1P 89705244 IC50 > 100000 nM T31391 C03OGJ 89705273 IC50 > 100000 nM T31391 CGX4I7 89705275 IC50 = 19000 nM T31391 CX9BC3 89712515 IC50 > 100000 nM T31391 CM5N8H 90654714 IC50 = 1436 nM T31391 CFY63H 90654715 IC50 = 378 nM T31391 CC6VX3 90654716 IC50 = 382 nM T31391 CA0SL5 90654717 IC50 = 342 nM T31391 CAM68Q 90654718 IC50 = 217 nM T31391 CQ93MA 90654719 IC50 = 193 nM T31391 CNDG24 90654720 IC50 = 1388 nM T31391 CC46WF 90654721 IC50 = 452 nM T31391 CCX20I 90654722 IC50 = 443 nM T31391 COV32D 90654723 IC50 = 404 nM T31391 CZ7KU8 90654724 IC50 = 885 nM T31391 CUH0W7 90654725 IC50 = 910 nM T31391 CCX14G 90654726 IC50 = 1034 nM T31391 CXUY06 90654727 IC50 = 1023 nM T31391 CKC94W 90654728 IC50 = 997 nM T31391 C8VBP2 90654729 IC50 = 119 nM T31391 C2UN8K 90654730 IC50 = 84 nM T31391 C1GSQ3 90654731 IC50 = 77.6 nM T31391 C47YVG 90654732 IC50 = 122 nM T31391 C20CDE 90654733 IC50 = 79 nM T31391 C9B2MJ 90654734 IC50 = 74 nM T31391 C30OWT 90654735 IC50 = 157 nM T31391 C3XP8C 90654736 IC50 = 119 nM T31391 CQD53I 90654737 IC50 = 125 nM T31391 C10TVX 90654738 IC50 = 111 nM T31391 C17RCY 90654739 IC50 = 19 nM T31391 CLT2X9 90654740 IC50 = 197 nM T31391 CDO0J4 90654741 IC50 = 148 nM T31391 CS62OC 90654742 IC50 = 134 nM T31391 C4B8KC 90654743 IC50 = 137 nM T31391 CKU5M8 90654744 IC50 = 43 nM T31391 C6TGZ5 90655538 IC50 > 100000 nM T31391 C9P3HJ 90655539 IC50 > 100000 nM T31391 CT98OM 90655540 IC50 > 100000 nM T31391 CVQ8M4 90655541 IC50 > 100000 nM T31391 CT6Q2L 90655542 IC50 > 100000 nM T31391 C7Z4GV 90655543 IC50 > 100000 nM T31391 CE3HC2 90655544 IC50 > 100000 nM T31391 CU2I3V 90655545 IC50 > 100000 nM T31391 C2NZ7X 90655546 IC50 > 100000 nM T31391 C0E5UP 90655547 IC50 > 100000 nM T31391 CF23RI 90655548 IC50 > 100000 nM T31391 CW3QG7 90655549 IC50 > 100000 nM T31391 CHG4E2 90655550 IC50 > 100000 nM T31391 CTA78W 90655551 IC50 > 100000 nM T31391 CA6S4W 90655552 IC50 > 100000 nM T31391 C3LT0S 90655553 IC50 > 100000 nM T31391 CEW45X 90655554 IC50 > 100000 nM T31391 CRX52D 90655555 IC50 > 100000 nM T31391 C9KG1U 90655556 IC50 > 100000 nM T31391 CXYE76 90655557 IC50 > 100000 nM T31391 CES85Q 90655558 IC50 > 100000 nM T31391 CK7IB9 90655559 IC50 >= 100000 nM T31391 CAG5X4 90655560 IC50 > 100000 nM T31391 C3IJA0 90655561 IC50 > 100000 nM T31391 C4V0ZY 90655562 IC50 > 100000 nM T31391 CY9G8Q 90655563 IC50 > 100000 nM T31391 CPIN84 90664318 IC50 = 53 nM T31391 CY76CR 90664436 IC50 = 1.8 nM T31391 C8YPL7 90664437 IC50 = 11 nM T31391 CU9LB2 90664438 IC50 > 100000 nM T31391 CQ20XA 90664578 IC50 > 100000 nM T31391 CV87ZH 90664579 IC50 > 100000 nM T31391 C9OC4Q 90664688 IC50 = 8.1 nM T31391 CJVF52 90664689 IC50 = 19 nM T31391 CDEN13 90664693 IC50 > 100000 nM T31391 CFG21I 90664805 IC50 = 2.9 nM T31391 C37YWE 90664828 IC50 = 84 nM T31391 CP60NA 90664941 IC50 = 7.8 nM T31391 CJ04US 90664942 IC50 = 69 nM T31391 CCH31U 90665060 IC50 = 23 nM T31391 C4LB2V 90665061 IC50 = 17 nM T31391 C0C1VT 90665186 IC50 = 12 nM T31391 CJ81VK 90665187 IC50 = 73 nM T31391 CHB2D6 90666864 IC50 = 16580 nM T31391 CFH71J 91937923 IC50 = 3730 nM T31391 COA7Z6 92131131 IC50 = 14 nM T31391 CBQ38C 101879512 IC50 = 170 nM T31391 CM7E4V 101887269 IC50 > 50000 nM T31391 C8EH0J 101887270 IC50 = 5.8 nM T31391 CDT67J 101887271 IC50 = 25 nM T31391 C4F2CS 101887272 IC50 > 100000 nM T31391 C58XWA 101887273 IC50 = 18100 nM T31391 C3Y9ET 101887274 IC50 > 100000 nM T31391 C1AF8C 101887275 IC50 = 1440 nM T31391 CH7QC5 101887276 IC50 > 50000 nM T31391 CO4FR2 101887277 IC50 = 29 nM T31391 C9JEH0 101887278 IC50 = 13900 nM T31391 C52GIO 101887279 IC50 > 100000 nM T31391 CO95EZ 118705501 IC50 = 570 nM T31391 CH8VO2 118705502 IC50 = 30 nM T31391 CZ1G3O 118712516 IC50 > 100000 nM T31391 C8X4JA 118712517 IC50 > 100000 nM T31391 CC29AB 118712518 IC50 > 100000 nM T31391 CB09PD 118712519 IC50 > 100000 nM T31391 CD4U1X 118712520 IC50 > 100000 nM T31391 CU0V5J 118712521 IC50 > 100000 nM T31391 C03OUP 118712522 IC50 > 100000 nM T31391 CT2MZ8 118712764 IC50 = 450 nM T31391 C3W5RU 118712765 IC50 = 220 nM T31391 CKA1N5 118712766 IC50 = 160 nM T31391 C8M6ZW 118712767 IC50 = 220 nM T31391 CV5C6D 118712768 IC50 = 320 nM T31391 C2NSC7 118712769 IC50 = 430 nM T31391 CV8JY3 118712770 IC50 = 640 nM T31391 C4KCZ1 118712771 IC50 = 770 nM T31391 CAR4W5 118712772 IC50 = 40 nM T31391 CRWT85 118712773 IC50 = 530 nM T31391 C36YUB 118712774 IC50 = 1580 nM T31391 C4T2FY 118712775 IC50 = 50 nM T31391 C0MYA1 118712776 IC50 = 1940 nM T31391 C8IF4E 118712777 IC50 = 440 nM T31391 CJ8EL0 118712778 IC50 = 70 nM T31391 C07UOL 118712779 IC50 = 360 nM T31391 C25HYG 118712780 IC50 = 130 nM T31391 CD0HQ4 118712781 IC50 = 270 nM T31391 C5D9RH 118712782 IC50 = 8800 nM T31391 CB7NX6 118712783 IC50 = 1980 nM T31391 C46TMQ 118712785 IC50 = 70 nM T31391 CA1I4M 118712786 IC50 = 47440 nM T31391 CUN79Q 118712787 IC50 = 9650 nM T31391 C5M3BX 118712788 IC50 = 10 nM T31391 CV3AK9 118717414 IC50 = 2390 nM T31391 C1NAQ9 118717415 IC50 > 100000 nM T31391 CKES65 118717416 IC50 > 100000 nM T31391 CYP07B 118719171 Ki = 6000 nM T31391 CD3L8W 118719172 Ki = 520 nM T31391 C8WJL2 118719173 Ki = 900 nM T31391 C5HU8M 118719174 Ki = 2700 nM T31391 C36XYR 118722404 IC50 = 5810 nM T31391 CX6J2E 118722405 IC50 = 340 nM T31391 C7BD8K 118722406 IC50 = 380 nM T31391 C0K6YG 118722407 IC50 = 760 nM T31391 CK7HN4 118722408 IC50 = 70 nM T31391 CFV6N4 118722409 IC50 = 3660 nM T31391 CK71WT 118722410 IC50 = 70 nM T31391 CI74ZM 118722411 IC50 = 80 nM T31391 CH1P7Y 118722412 IC50 = 70 nM T31391 CL8TY5 118722413 IC50 = 180 nM T31391 CGK98I 118722414 IC50 = 320 nM T31391 CBK91L 118722415 IC50 = 510 nM T31391 C8KUP0 118722416 IC50 = 290 nM T31391 C76DBO 118722417 IC50 = 540 nM T31391 CW6L5X 118722418 IC50 = 330 nM T31391 CM6Y5I 118722419 IC50 = 430 nM T31391 C37BGF 118722420 IC50 = 610 nM T31391 COG4V6 118722421 IC50 = 140 nM T31391 CIQ5Z7 118722422 IC50 = 430 nM T31391 CH6GX2 118728164 IC50 = 6 nM T31391 CFCI13 118728166 IC50 = 4.7 nM T31391 CS08AG 118728168 IC50 = 1.4 nM T31391 C0AG2Q 118728920 IC50 = 500 nM T31391 CE1ZS2 118728922 IC50 = 230 nM T31391 CVG84E 118728927 IC50 = 640 nM T31391 CBI68Y 118728931 IC50 = 36 nM T31391 CI0E1U 118736611 IC50 = 695 nM T31391 C2NX7C 118736612 IC50 = 2801 nM T31391 CP71VU 118736613 IC50 = 27.54 nM T31391 CL40TU 118736614 IC50 = 145 nM T31391 CJI2B8 118736615 IC50 = 85 nM T31391 C15XMK 118736616 IC50 = 108 nM T31391 C1IGJ6 118736617 IC50 = 67 nM T31391 C4BI2T 118736618 IC50 = 258 nM T31391 CED50R 118736620 IC50 = 100 nM T31391 C3DT9O 118736622 IC50 = 94 nM T31391 C6TYS7 122172854 IC50 = 4376 nM T31391 C2U5PE 122178432 IC50 = 20 nM T31391 C7TEY3 122178433 IC50 = 19.8 nM T31391 C8OLP9 122178434 IC50 = 346 nM T31391 C9GP3L 122178435 IC50 = 2.9 nM T31391 C8P2DB 122178436 IC50 = 6.4 nM T31391 CGFU89 122178437 IC50 = 3.4 nM T31391 CN78TQ 122189864 IC50 = 650 nM T31391 CNM82F 122189865 IC50 > 100000 nM T31391 C19GHJ 122189866 IC50 = 12200 nM T31391 C3U9KC 122189867 IC50 > 100000 nM T31391 CW5V3U 122189868 IC50 = 180 nM T31391 CCG05R 122189869 IC50 = 1800 nM T31391 CI01PT 122189870 IC50 = 180 nM T31391 C80EWF 122189871 IC50 = 220 nM T31391 C3N7JC 122189872 IC50 > 100000 nM T31391 CG8O1J 122189873 IC50 > 100000 nM T31391 CK0US2 122189874 IC50 = 980 nM T31391 C5V6NI 122189875 IC50 > 100000 nM T31391 CV7A9Y 122189876 IC50 > 100000 nM T31391 CN86VR 122189878 IC50 > 100000 nM T31391 C24OVE 122190735 IC50 = 1320 nM T31391 CSN6E0 122190738 IC50 = 24000 nM T31391 CD4EF9 122190739 IC50 = 1060 nM T31391 CVU5G7 122190835 IC50 = 2230 nM T31391 CB5X2Q 122190838 IC50 = 100000 nM T31391 CG69FQ 122190841 IC50 = 1250 nM T31391 CJ7X2U 122194794 IC50 = 1.5 nM T31391 C8XVB4 122194795 IC50 = 290 nM T31391 CL43TO 122194796 IC50 = 0.8 nM T31391 CAPX63 126456388 IC50 = 2.06 nM T31391 C0DUI4 126842756 IC50 = 1.33 nM T31391 CZXV13 126842761 IC50 = 0.76 nM T31391 CF7KI9 126842762 IC50 = 1.62 nM T31391 CG93JS 126842771 IC50 = 1.22 nM T31391 C6PLX9 127035081 IC50 = 4.9 nM T31391 CJ0KS7 127035239 IC50 = 2.3 nM T31391 CKSZ13 127035240 IC50 = 1.8 nM T31391 C6T1IM 127035241 IC50 = 5.7 nM T31391 CJRL72 127035242 IC50 = 0.7 nM T31391 CVKI59 127035243 IC50 = 1.9 nM T31391 CWJX95 127035244 IC50 = 2.3 nM T31391 C0XMS7 127035375 IC50 = 1.9 nM T31391 CMK5Q9 127035376 IC50 = 1.4 nM T31391 C4N7QB 127035377 IC50 = 1.6 nM T31391 CGN49F 127035378 IC50 = 4.3 nM T31391 C36UHW 127035569 IC50 = 0.3 nM T31391 CTKS36 127035740 IC50 = 3.7 nM T31391 CAXT02 127035741 IC50 = 3.2 nM T31391 CZB0L6 127035742 IC50 = 1.1 nM T31391 C4QWL5 127035743 IC50 = 1.3 nM T31391 CPGF39 127035744 IC50 = 1.8 nM T31391 CXTD34 127035745 IC50 = 1.8 nM T31391 CM98XR 127035752 IC50 = 1.7 nM T31391 C87MVA 127035753 IC50 = 1.7 nM T31391 CDW25O 127035754 IC50 = 0.4 nM T31391 CN08IS 127045827 IC50 > 100000 nM T31391 CAK85G 127046590 IC50 > 50000 nM T31391 CP3U8J 127046622 IC50 > 100000 nM T31391 CFAI71 127046624 IC50 = 56000 nM T31391 CB6PA7 127046626 IC50 > 100000 nM T31391 C76IGF 127046628 IC50 > 100000 nM T31391 CHL49F 127046630 IC50 = 790 nM T31391 CH0D2Z 127046632 IC50 = 4000 nM T31391 CK4SO7 127047730 IC50 = 2600 nM T31391 CSO9L3 127047731 IC50 = 19400 nM T31391 C4KIA9 127047732 IC50 = 16200 nM T31391 CHX41E 127047733 IC50 = 680 nM T31391 C6I7HW 127047734 IC50 = 34000 nM T31391 C2CP4F 127047761 IC50 > 100000 nM T31391 CYR1X2 127047762 IC50 > 100000 nM T31391 CIV4C2 127047839 IC50 > 100000 nM T31391 CDYA70 127047985 IC50 > 100000 nM T31391 C0FS5E 127048116 IC50 > 100000 nM T31391 C6NIM5 127048874 IC50 = 8.6 nM T31391 CXD69M 127048875 IC50 = 289 nM T31391 C65MAC 127048876 IC50 = 44 nM T31391 C23BWQ 127049179 IC50 = 1.4 nM T31391 CNCB06 127049180 IC50 = 1.9 nM T31391 CJ8SG3 127049204 IC50 = 1.5 nM T31391 CRM04V 127049507 IC50 = 0.5 nM T31391 C76VPA 127049823 IC50 = 54 nM T31391 CH0X6Q 127050132 IC50 = 0.5 nM T31391 CIGA32 127050759 IC50 = 1.1 nM T31391 CNY90B 127050760 IC50 = 1.5 nM T31391 C80WCY 127050761 IC50 = 0.6 nM T31391 CUVQ34 127050762 IC50 = 2.9 nM T31391 CJMS57 127051032 IC50 = 1.1 nM T31391 C9V4EG 127051045 IC50 = 0.7 nM T31391 C7W8JR 127051639 IC50 = 699 nM T31391 C36SXH 127052286 IC50 = 1.1 nM T31391 CBR1F8 127052287 IC50 = 26 nM T31391 CHZX75 127052288 IC50 = 0.6 nM T31391 CB34GQ 127052289 IC50 = 0.7 nM T31391 CLG0Q3 127052290 IC50 = 16 nM T31391 CL2S0F 127052581 IC50 = 1.7 nM T31391 C1W5AL 127052582 IC50 = 155 nM T31391 C4TI8H 127052590 IC50 = 1170 nM T31391 CNV0A8 127052636 IC50 = 0.56 nM T31391 CS2Z9R 127052637 IC50 = 0.23 nM T31391 C75EAL 127052638 IC50 = 0.24 nM T31391 CRP1K2 130385241 IC50 = 5.8 nM T31391 CTIO26 130385242 IC50 = 5.17 nM T31391 C30ERZ 130385243 IC50 = 1.9 nM T31391 C09MJL 130385246 IC50 = 205.2 nM T31391 CZ29WO 130385251 IC50 = 19.64 nM T31391 CED01R 130385253 IC50 = 14.95 nM T31391 C83CDX 130385258 IC50 = 8.42 nM T31391 CB37AX 130385267 IC50 = 216.2 nM T31391 C5DWM6 130391940 IC50 = 70.42 nM T31391 C41QVU 130391961 IC50 = 6.13 nM T31391 C6PMX7 130391978 IC50 = 17.65 nM T31391 CD7B2H 130392003 IC50 = 8.91 nM T31391 C15BEV 130392042 IC50 = 563.9 nM T31391 CD6C4U 130392043 IC50 = 13070 nM T31391 CH9E4W 132055397 IC50 = 110.1 nM T31391 C6CV5J 132069286 IC50 = 154.67 nM T31391 CALB73 134131859 IC50 = 5400 nM T31391 CA5Y0V 134132454 IC50 = 250 nM T31391 CMY0V5 134132485 IC50 = 5000 nM T31391 CTZU69 134132901 IC50 = 14.6 nM T31391 CH1G3A 134133219 IC50 = 260 nM T31391 CS9K7A 134133834 IC50 = 360 nM T31391 C2BA5L 134134276 IC50 = 890 nM T31391 CVE96U 134134571 IC50 = 300 nM T31391 CB59UX 134135207 IC50 = 73 nM T31391 CIXJ53 134135875 IC50 = 250 nM T31391 C4Q2GB 134136466 IC50 = 121.56 nM T31391 C5OS4T 134136634 IC50 = 39.2 nM T31391 C14XET 134137196 IC50 = 140 nM T31391 CMB8T7 134137851 IC50 = 32.64 nM T31391 CTP9X4 134138048 IC50 = 21520 nM T31391 C58KIQ 134138807 IC50 = 500 nM T31391 C2OWQ1 134138838 IC50 = 760 nM T31391 CPLI26 134139792 IC50 = 400 nM T31391 CDV6U9 134140856 IC50 = 49.73 nM T31391 C5TS2J 134141415 IC50 = 2600 nM T31391 CB8QD9 134142015 IC50 = 770 nM T31391 CY2CJ4 134142362 IC50 = 510 nM T31391 CK27IY 134143858 IC50 = 2930 nM T31391 CKP0Z5 134144315 IC50 = 78.33 nM T31391 COT7P4 134144691 IC50 = 206.71 nM T31391 CD0XT6 134145610 IC50 = 800 nM T31391 C8B3CU 134150931 IC50 = 280 nM T31391 CEC9Y2 134151020 IC50 = 50860 nM T31391 C0G5PV 134151859 IC50 = 220 nM T31391 C3NF8J 134151937 IC50 = 140 nM T31391 CQRM94 134152842 IC50 = 360 nM T31391 C6TL9Z 134153173 IC50 = 950 nM T31391 CBN6Z7 134153444 IC50 = 610 nM T31391 CZX9V0 134154214 IC50 = 337.8 nM T31391 C4ZWS1 134157002 IC50 = 120 nM T31391 CNO0R1 135411740 IC50 = 2120 nM T31391 CRM4Q8 135518358 IC50 = 3 nM T31391 CMI5A6 135964368 IC50 = 95 nM T31391 CC4L2F 136060652 IC50 > 3000 nM T31391 CP7BS2 136098501 IC50 = 6113 nM T31391 CO04QA 136177302 IC50 = 7 nM T31391 C1GYM8 136411530 IC50 = 11 nM T31391 CR4VI2 137225025 IC50 = 0.6 nM T31391 CAN18C 137631813 IC50 = 2.1 nM T31391 C95BML 137632265 IC50 = 70 nM T31391 C5H2EA 137637131 IC50 = 27.54 nM T31391 C2FA1T 137637208 IC50 = 7.2 nM T31391 CS2L6B 137637588 IC50 = 43.4 nM T31391 CO9BH6 137638100 IC50 = 50.2 nM T31391 C6IJ3A 137642352 IC50 = 8.5 nM T31391 CY0R4C 137644720 IC50 = 60 nM T31391 CI8FG2 137644837 IC50 = 1200 nM T31391 C1MBC4 137646578 IC50 = 31.8 nM T31391 C67NZA 137650009 IC50 = 123.3 nM T31391 C8BH1R 137650030 IC50 = 537 nM T31391 CG8HS3 137652269 IC50 = 29 nM T31391 C9SX0Q 137653253 IC50 = 139 nM T31391 CH4MT1 137655300 IC50 = 8.7 nM T31391 CV5A3F 137657117 IC50 = 470 nM T31391 CKF03W 137659671 IC50 = 5.5 nM T31391 C2MV9K 137661375 IC50 = 151.7 nM T31391 CJT56Y 137662038 IC50 = 2.6 nM T31391 CO6JA3 141514759 IC50 = 188.7 nM T31391 C1SQ2R 141514762 IC50 = 64.47 nM T31391 CHI84B 141514764 IC50 = 65.36 nM T31391 C3SKH4 145948172 IC50 = 97 nM T31391 C8S7FY 145949528 IC50 = 1.45 nM T31391 CR2UP9 145950777 IC50 > 100 nM T31391 C7IZU2 145950786 IC50 = 1.61 nM T31391 C7SMW4 145951086 IC50 = 0.72 nM T31391 CR5AJ7 145952072 IC50 = 26.6 nM T31391 C2MWR4 145952134 IC50 = 15.3 nM T31391 CV30OD 145952476 IC50 = 0.77 nM T31391 CBFR49 145953292 IC50 = 1.69 nM T31391 CYF24S 145953544 IC50 = 0.76 nM T31391 C38IOE 145953726 IC50 = 0.61 nM T31391 C4JQT5 145953757 IC50 > 100 nM T31391 C0C4KJ 145954860 IC50 = 0.79 nM T31391 C48AXH 145955793 IC50 = 2.4 nM T31391 C6QY1K 145957483 IC50 = 1.58 nM T31391 CMO0J1 145957949 IC50 = 1.67 nM T31391 C35FNU 145957994 IC50 = 18 nM T31391 CR9S6F 145958227 IC50 = 2.3 nM T31391 CB72HG 145958828 IC50 = 1.25 nM T31391 C60WXK 145959997 IC50 = 0.77 nM T31391 C8V5PA 145962482 IC50 = 0.54 nM T31391 CBL76R 145964231 IC50 = 2500 nM T31391 CF53NA 145964407 IC50 = 400 nM T31391 CNMT16 145965136 IC50 = 1200 nM T31391 CQW63D 145965301 IC50 = 11500 nM T31391 C6D0VY 145967130 IC50 = 21500 nM T31391 CI82EJ 145973071 IC50 = 10400 nM T31391 C1Y5FP 145973406 IC50 = 6.8 nM T31391 CP8EN1 145973616 IC50 = 0.54 nM T31391 CP7VT2 145973710 IC50 = 1300 nM T31391 C2C1ZR 145974002 IC50 = 17200 nM T31391 C9C4WU 145975568 IC50 = 80 nM T31391 CRNK53 145977284 IC50 = 46500 nM T31391 CWF4Y7 145977953 IC50 = 2000 nM T31391 CB3K0Q 145978529 IC50 = 59900 nM T31391 CR3I9D 145978547 IC50 = 49 nM T31391 CNG4Z2 145983347 IC50 = 1.12 nM T31391 CH6P8Q 145983352 IC50 = 1270 nM T31391 C02BLT 145983464 IC50 = 7580 nM T31391 CN1V6D 145984069 IC50 = 28050 nM T31391 C3QT0G 145984247 IC50 = 1780 nM T31391 CMWH26 145984429 IC50 = 15780 nM T31391 CL6D3F 145984547 IC50 = 19.6 nM T31391 CIX4P5 145985997 IC50 = 232.8 nM T31391 CM6L4K 155510749 IC50 = 190 nM T31391 C5ZQ7W 155511281 IC50 = 2.91 nM T31391 CP4SH8 155511399 IC50 > 100000 nM T31391 CEL39X 155511987 IC50 = 74.6 nM T31391 CQA73O 155512586 IC50 = 197 nM T31391 C57QZJ 155512836 IC50 = 7.6 nM T31391 CX3U8Z 155515016 IC50 = 10.21 nM T31391 C7FOS5 155516136 IC50 = 538 nM T31391 CTE94M 155516800 IC50 > 10000 nM T31391 C19ZCJ 155518265 IC50 = 395 nM T31391 C8UOJ4 155518381 IC50 = 1.7 nM T31391 C8U9ON 155518908 Ki = 217.9 nM T31391 CW0NI8 155519444 IC50 = 0.1 nM T31391 C7O2UF 155519988 IC50 > 100000 nM T31391 C3I8AW 155520161 IC50 = 60 nM T31391 C1Z2NP 155522069 Ki = 152.8 nM T31391 C4AZ9V 155523785 IC50 = 93.2 nM T31391 CG18KV 155524302 IC50 = 0.75 nM T31391 C0RAC6 155524362 IC50 = 3900 nM T31391 CTSA30 155526359 IC50 = 5.61 nM T31391 CVD89H 155526728 IC50 = 208 nM T31391 C5C4UV 155526759 IC50 = 5.99 nM T31391 CAT3J0 155526949 IC50 = 3.9 nM T31391 C7J4VQ 155527859 IC50 = 1.75 nM T31391 CLE9I0 155528648 IC50 = 0.22 nM T31391 C3LT9C 155529752 IC50 > 100000 nM T31391 C8FHJ2 155529886 IC50 = 2.43 nM T31391 CCX9H6 155530472 IC50 = 226 nM T31391 C7YP3B 155530585 IC50 = 4.41 nM T31391 C2YWG1 155530817 IC50 = 790 nM T31391 CB6N4S 155531120 IC50 = 0.18 nM T31391 CGV6C1 155531169 IC50 = 22.09 nM T31391 CEOQ32 155531330 IC50 = 50.9 nM T31391 CMY59I 155531892 IC50 > 100000 nM T31391 C0ZCE3 155533243 IC50 = 89.8 nM T31391 CN04KW 155533304 IC50 = 74.43 nM T31391 C95ZUT 155534726 Ki = 180.8 nM T31391 CW8Z1X 155535213 IC50 > 100000 nM T31391 CA9Z6Q 155538747 IC50 = 121300 nM T31391 CG3RS6 155540249 IC50 = 223 nM T31391 CJ67GL 155540375 IC50 = 3.5 nM T31391 CM1FA9 155544265 Ki = 380.1 nM T31391 CY25EZ 155544299 IC50 = 4.6 nM T31391 C8H3MJ 155544665 IC50 = 20.48 nM T31391 CU17DA 155544967 IC50 = 2.35 nM T31391 CY2V6P 155545256 IC50 = 2.25 nM T31391 C62YMT 155545522 IC50 = 85.48 nM T31391 CMS63L 155545906 IC50 = 56.6 nM T31391 CGZ08R 155547532 IC50 = 3830000 nM T31391 CDGW26 155547608 IC50 = 76170 nM T31391 CNA9X4 155548276 IC50 = 217 nM T31391 CWF0L6 155548277 IC50 = 483 nM T31391 CM9K4B 155548792 IC50 = 0.72 nM T31391 CB1AF4 155549522 IC50 = 7.5 nM T31391 CL9R1Y 155549582 IC50 > 100000 nM T31391 C3MW1B 155550953 IC50 > 10000 nM T31391 CX9Y4B 155552378 IC50 = 1.05 nM T31391 C8XSI3 155553379 IC50 = 2 nM T31391 C6QKL9 155553392 Ki = 412.2 nM T31391 C1D5QZ 155554658 IC50 = 2.5 nM T31391 CR8AU9 155555628 IC50 = 68510 nM T31391 C1GD0E 155555672 Ki = 941.2 nM T31391 CHV85S 155556058 IC50 > 100000 nM T31391 C6N4WH 155557237 IC50 > 100000 nM T31391 CSCD34 155559193 IC50 > 100000 nM T31391 C7KVR5 155559306 IC50 = 3.9 nM T31391 CRL47X 155559391 IC50 = 28.7 nM T31391 C1NE4T 155560255 IC50 > 100000 nM T31391 C68CRH 155561682 IC50 = 4 nM T31391 CQ7JL5 155562412 IC50 = 55870 nM T31391 C90QLF 155563643 Ki = 103.7 nM T31391 C48ETF 155565121 IC50 = 170 nM T31391 CUL27B 155565517 Ki = 341.6 nM T31391 CE5SI7 155566076 IC50 > 100000 nM T31391 CI5C6P 155568161 IC50 = 0.44 nM T31391 CUQL05 155568269 IC50 = 5.06 nM T31391 CDB0S2 155568427 IC50 = 421 nM T31391 D00HSG 44408767 IC50 = 3300 nM T31391 D00KMP 44431763 IC50 = 5300 nM T31391 D00RIX 5280443 IC50 = 140 nM T31391 D00YEV 5281605 IC50 > 200000 nM T31391 D02RDY 11375559 IC50 > 100000 nM T31391 D02RIE 44440628 Ki = 13000 nM T31391 D02WBC 3847395 IC50 = 33000 nM T31391 D03DNV 71655266 IC50 > 100000 nM T31391 D04CAR 10607286 Ki = 0.4 nM T31391 D05LYC 11403745 IC50 = 140 nM T31391 D05UUA 16049437 Ki = 820 nM T31391 D05XWX 10130510 Ki = 3.8 nM T31391 D06AUB 44440618 Ki = 3400 nM T31391 D06NRU 1393052 IC50 = 2300 nM T31391 D06UKY 44440632 Ki = 2800 nM T31391 D07ALM 11232124 Ki = 0.082 nM T31391 D07HWI 6931234 IC50 = 75000 nM T31391 D07IJU 13578534 Ki = 2100 nM T31391 D08NMS 46900258 Ki = 1.4 nM T31391 D09ALJ 5280805 IC50 = 145000 nM T31391 D09BYA 44431745 IC50 = 3500 nM T31391 D09MVE 263366 IC50 = 30000 nM T31391 D0AU0M 637542 IC50 = 83180 nM T31391 D0CP1J 56658139 IC50 > 50000 nM T31391 D0G3TK 5280863 IC50 = 132000 nM T31391 D0JI3S 11674875 IC50 = 18600 nM T31391 D0JL2T 5393152 IC50 > 200000 nM T31391 D0L5RI 44328273 Ki = 7880 nM T31391 D0L9XR 447256 Ki = 470 nM T31391 D0N1FU 6918465 Ki = 126 nM T31391 D0N1QQ 94701 Ki = 2200 nM T31391 D0N5CI 11615508 IC50 = 12000 nM T31391 D0O9RD 44403067 Ki = 3350 nM T31391 D0P5OE 2724998 IC50 = 45000 nM T31391 D0PB2M 23645372 Ki = 34 nM T31391 D0R5OE 44422449 IC50 = 538 nM T31391 D0S0RK 10680 IC50 = 170 nM T31391 D0T2EW 11075394 Ki = 1.4 nM T31391 D0T3PW 5281672 IC50 = 37150 nM T31391 D0U4HG 23634523 IC50 > 36900 nM T31391 D0V9EN 689043 IC50 = 3370 nM T31391 D0W4GM 205131 IC50 = 40000 nM T31391 D0X0IF 23655936 IC50 > 39100 nM T31391 D0X2JG 2777206 IC50 = 37000 nM T31391 D0Y3TZ 370 IC50 = 4650 nM T31391 D0Y5IQ 44255320 IC50 = 10000 nM T02439 CJ6R1L 18445508 IC50 = 199.53 nM T02439 C3HVM7 18445520 IC50 = 31.62 nM T02439 C8OR0L 18445737 IC50 = 3162.28 nM T02439 CM28GF 18445739 IC50 = 63.1 nM T02439 C0TC2X 18445833 IC50 = 630.96 nM T02439 C3VRO9 44557921 IC50 > 10000 nM T02439 CL0OC7 45375855 IC50 = 2511.89 nM T02439 CZXJ98 45483394 IC50 = 125.89 nM T02439 C25NVM 45483417 IC50 = 316.23 nM T02439 C0I2MB 45483418 IC50 = 251.19 nM T02439 C6CJ2N 45483436 IC50 = 794.33 nM T02439 CZOK17 45483447 IC50 = 1000 nM T02439 C1W0AX 45483460 IC50 = 1000 nM T02439 CICD40 45483461 IC50 = 2511.89 nM T02439 CXK2H9 45483468 IC50 = 1584.89 nM T02439 C7MQI8 45483469 IC50 > 10000 nM T02439 CED7U8 45483470 IC50 = 50.12 nM T02439 CBV30W 45483507 IC50 = 501.19 nM T02439 CAL8P6 45483508 IC50 = 794.33 nM T02439 C2UPW3 45483509 IC50 = 1258.93 nM T02439 CA23TC 45483510 IC50 = 7.943 nM T02439 CZC96T 45483513 IC50 = 19.95 nM T02439 C2ABD6 45483530 IC50 = 251.19 nM T02439 C4EZO3 45483716 IC50 = 63.1 nM T02439 CB3N6J 45483717 IC50 = 501.19 nM T02439 CH1S9G 45483725 IC50 = 79.43 nM T02439 CE6K8L 45483734 IC50 > 10000 nM T02439 C4DG0Z 45483735 IC50 > 10000 nM T02439 CXB94H 53466728 IC50 = 17020 nM T02439 CYQ41S 53466951 IC50 = 1863 nM T02439 CX0R1K 53469059 IC50 = 460 nM T02439 CV7C0D 53469060 IC50 = 37 nM T02439 CCKD45 53469061 IC50 = 61 nM T02439 C91STB 53469449 IC50 = 214 nM T02439 CZ1CI3 53469824 IC50 = 12080 nM T02439 CX4H6I 86583042 IC50 > 10000 nM T02439 C4TXF2 118730409 IC50 > 10000 nM T02439 CXC69T 137321158 IC50 = 26 nM T02439 C2MD1Q 155513187 IC50 > 10000 nM T02439 D02LIR 45375987 IC50 = 6.31 nM T02439 D0N4LR 53469448 IC50 = 420 nM T15023 C31FHD 156080 IC50 = 25000 nM T15023 CC7OA9 9854089 IC50 = 84100 nM T15023 CHKV76 15984054 IC50 = 2000 nM T15023 C0VBC2 22779253 IC50 = 9300 nM T15023 COB8R4 24765913 IC50 = 13000 nM T15023 CS5O8W 24815567 IC50 = 14000 nM T15023 C6UM9C 24815571 IC50 = 52000 nM T15023 CX0BK1 24815653 IC50 = 18000 nM T15023 CCPS98 24815654 IC50 = 9000 nM T15023 C3V9CG 24815655 IC50 = 17000 nM T15023 CT86UJ 24815656 IC50 = 33000 nM T15023 CPZQ89 44415045 IC50 = 80000 nM T15023 CI8GD1 44415050 IC50 = 3000 nM T15023 CFK0E3 44415051 IC50 = 3000 nM T15023 CJ5O9B 44415067 IC50 = 62000 nM T15023 CGIB09 44415068 IC50 = 60000 nM T15023 CQ0P6M 44415069 IC50 = 3000 nM T15023 CJ51WK 44415070 IC50 = 3000 nM T15023 C09FPC 44415084 IC50 = 47000 nM T15023 C2X0IH 44415085 IC50 = 43000 nM T15023 CUK58S 44415107 IC50 = 19000 nM T15023 CCO95R 44415108 IC50 = 13000 nM T15023 CALV50 44415122 IC50 = 9000 nM T15023 C8DT5W 44415123 IC50 = 4000 nM T15023 C8DA3X 44415134 IC50 = 4000 nM T15023 C4E6OP 44415135 IC50 = 3000 nM T15023 C7K9YM 44415146 IC50 = 2000 nM T15023 C4CRI6 44415160 IC50 = 95000 nM T15023 C7H6QP 44415168 IC50 = 22000 nM T15023 C95GPD 44415171 IC50 = 14000 nM T15023 CXUY04 44415198 IC50 = 13000 nM T15023 C7MAV1 44415199 IC50 = 13000 nM T15023 CD3X5N 44415203 IC50 = 10000 nM T15023 CQ4Y6E 44415204 IC50 = 10000 nM T15023 CUBP89 44415228 IC50 = 29000 nM T15023 C2FL1O 44415229 IC50 = 9000 nM T15023 CEJH97 44415230 IC50 = 6000 nM T15023 CSGQ74 44415243 IC50 = 6000 nM T15023 CN5F8H 44415244 IC50 = 6000 nM T15023 C3RB4Q 44415264 IC50 = 5000 nM T15023 CGU69B 44415265 IC50 = 5000 nM T15023 CWJ86B 44415284 IC50 = 79000 nM T15023 CG4O3L 44415285 IC50 = 42000 nM T15023 C1TGL7 44415286 IC50 = 5000 nM T15023 C5QZO0 44415287 IC50 = 4000 nM T15023 C7PXM4 44415303 IC50 = 4000 nM T15023 CL5SJ9 44415321 IC50 = 3000 nM T15023 CW2V1K 44415322 IC50 = 2000 nM T15023 CF2B9J 44415323 IC50 = 2000 nM T15023 CMXN47 44415328 IC50 = 2000 nM T15023 C4CO0Q 44415329 IC50 = 2000 nM T15023 CXNB21 44631827 IC50 = 3000 nM T15023 CFS01Z 45139618 IC50 = 17000 nM T15023 C3FIO4 45139619 IC50 = 12000 nM T15023 CYV65U 45139620 IC50 = 6000 nM T15023 C6F4MD 46881769 IC50 = 30000 nM T15023 CD53IC 46888232 IC50 = 92000 nM T15023 CSZN86 73345690 IC50 = 18000 nM T15023 C1V4YX 117919744 IC50 = 8900 nM T15023 CN3XO8 133081972 IC50 = 1600 nM T15023 CH63VL 145979165 IC50 = 800 nM T15023 CLP5J8 155510478 IC50 = 10715.19 nM T15023 C8BHO5 155519379 IC50 = 120000 nM T15023 CM7XI4 155521636 IC50 = 26000 nM T15023 C89PUV 155535868 IC50 = 187000 nM T15023 C62ATN 155538638 IC50 = 2951.21 nM T15023 CC39XR 155539536 IC50 = 50100 nM T15023 CV7JH9 155541491 IC50 = 20900 nM T15023 CKF02B 155541869 IC50 = 181000 nM T15023 CDP3A5 155542006 IC50 = 2884.03 nM T15023 C4LT0D 155542021 IC50 = 16000 nM T15023 CKR03L 155542693 IC50 = 18100 nM T15023 CUX2Z1 155543565 IC50 = 7700 nM T15023 CN2GQ1 155544385 IC50 = 16100 nM T15023 CF79TY 155545026 IC50 = 23400 nM T15023 CRA0T4 155545299 IC50 = 15848.93 nM T15023 C6TJV0 155545675 IC50 = 9200 nM T15023 C3U9ID 155545743 IC50 = 2300 nM T15023 C5C0LF 155548104 IC50 = 21300 nM T15023 CUS5A3 155549314 IC50 = 88000 nM T15023 CZGJ90 155549636 IC50 = 39000 nM T15023 C73BNV 155550340 IC50 > 100000 nM T15023 C06ERO 155552650 IC50 = 48600 nM T15023 CY9T5X 155554019 IC50 = 69000 nM T15023 CVIM57 155555240 IC50 = 14000 nM T15023 C2ROS0 155556517 IC50 = 80500 nM T15023 C2HMC4 155557562 IC50 = 21300 nM T15023 C84LDU 155560254 IC50 > 100000 nM T15023 CP6GZ9 155560763 IC50 = 134000 nM T15023 CCN1U7 155566104 IC50 = 21300 nM T15023 CQ4E5Y 155566947 IC50 = 5370.32 nM T15023 CBE1X8 155569690 IC50 = 7200 nM T15023 D0GD5G 15858500 IC50 = 4600 nM T00563 D09JEJ 24748573 IC50 = 11 nM T00563 D0E3TC 44259 IC50 = 844 nM T00563 D02GEJ 5326976 Ki = 112 nM T00563 CJH12X 537952 IC50 = 32200 nM T00563 CR9EJ0 11352337 Ki = 35 nM T00563 C8V7ZF 11352967 Ki = 37 nM T00563 CV78IN 16224258 IC50 = 190 nM T00563 CY8X0J 24811794 IC50 = 701 nM T00563 C4HY6I 44263430 Ki = 21 nM T00563 CYX19V 44263445 Ki = 78 nM T00563 C0RK5W 44263447 Ki = 62 nM T00563 CNZ19H 44263451 Ki = 342 nM T00563 C3VRO9 44557921 IC50 > 10000 nM T00563 CDK93W 56946894 IC50 < 3000 nM T00563 CE2DU7 56968171 Ki = 188 nM T00563 C4RIA1 56968172 Ki = 93 nM T00563 CYIO69 56968174 Ki = 31 nM T00563 CT1ZJ3 56968175 Ki = 55 nM T00563 C73NVJ 56968176 Ki = 44 nM T00563 C0MS9N 56968177 Ki = 83 nM T00563 C8WDK1 57342036 IC50 = 11 nM T00563 C0I6SZ 57342039 IC50 = 32000 nM T00563 CA7BS4 57342210 IC50 = 63 nM T00563 CVBF89 57342215 IC50 = 25000 nM T00563 C8P1ZB 57342375 IC50 = 5300 nM T00563 CH6RV3 57342376 IC50 = 3300 nM T00563 C65NOS 57342377 IC50 = 1700 nM T00563 C8TFC7 57342378 IC50 = 1200 nM T00563 CZ0R4K 57342379 IC50 = 5800 nM T00563 C8U4MB 57342380 IC50 = 1800 nM T00563 CJSO14 57342381 IC50 = 2800 nM T00563 CW3P9K 57342382 IC50 = 4300 nM T00563 CFX60S 57342541 IC50 = 1600 nM T00563 CF9BZ1 57342542 IC50 = 2900 nM T00563 C2C4XB 57342543 IC50 = 4300 nM T00563 C9XPF2 57342544 IC50 = 2700 nM T00563 C9MA4U 57342545 IC50 = 3000 nM T00563 CWZY51 57342546 IC50 = 8200 nM T00563 CK9IC1 57342547 IC50 = 3100 nM T00563 CO14NX 57342548 IC50 = 5700 nM T00563 CTNX36 57342718 IC50 = 2400 nM T00563 C8G6RK 57342719 IC50 = 2100 nM T00563 CJ9OF3 57400663 Ki = 24 nM T00563 CV63UL 67240318 IC50 > 10000 nM T00563 CDE3Y9 76321032 IC50 < 4000 nM T00563 C4T7YB 127025199 IC50 = 4.6 nM T00563 CP02TW 127025200 IC50 = 10 nM T00563 C57ECS 127025201 IC50 = 280 nM T00563 CP31UE 127025202 IC50 = 10 nM T00563 CHP6R9 127025499 IC50 = 12 nM T00563 CY37QE 127025500 IC50 = 12 nM T00563 CR59LY 127026094 IC50 = 11 nM T00563 CWIG59 127026095 IC50 = 9.8 nM T00563 C45BZG 127026096 IC50 = 160 nM T00563 C0HLT9 127026097 IC50 = 19 nM T00563 CW5JB1 127026098 IC50 = 14 nM T00563 CL4CG5 127026727 IC50 = 13 nM T00563 CO6X5B 127026728 IC50 = 11 nM T00563 CA5XG8 127026729 IC50 = 9.5 nM T00563 C6EIR3 127027657 IC50 = 9.6 nM T00563 C1MF5T 127029513 IC50 = 8.8 nM T00563 C86HPW 155518524 IC50 = 99000 nM T00563 D0CP3M 5149739 Ki = 270 nM T00563 D0K6BI 46943415 Ki = 21 nM T00563 D0US9O 45275255 IC50 = 2.7 nM T44351 D0P1FO 16078 Ki = 41 nM T44351 D0YZ8I 4273754 Ki = 164 nM T44351 D0J7RW 5311501 Ki = 24 nM T44351 CRM5P4 9845561 Ki = 0.46 nM T44351 C7SW3C 10360860 Ki = 9.5 nM T44351 C2FK8Z 13645595 Ki > 10000 nM T44351 C52FSE 24096428 Ki = 0.77 nM T44351 C3MZ0J 44327221 Ki = 0.81 nM T44351 CIBP20 44327403 Ki = 0.6 nM T44351 CX03ZD 44327404 Ki = 0.84 nM T44351 CG59OH 44327429 Ki = 0.46 nM T44351 CLH31M 44368310 Ki = 22 nM T44351 C52UYW 44368361 Ki = 1250 nM T44351 CETG63 44368362 Ki = 46 nM T44351 CIZ10X 44368367 Ki > 10000 nM T44351 CG92UC 44368388 Ki = 48 nM T44351 CLK34Y 44368424 Ki = 81 nM T44351 C52RNY 44368441 Ki = 72 nM T44351 CTKI30 44368442 Ki = 33 nM T44351 C83XUB 44368703 Ki > 10000 nM T44351 CO0RU5 44371487 Ki = 800 nM T44351 CY92LZ 53310757 Ki > 1000 nM T44351 D04GDY 638026 Ki = 44 nM T44351 D0D6OH 104895 Ki = 0.924 nM T44351 D0F4BX 9821569 Ki = 0.73 nM T01138 D01GBY 124087 IC50 = 172000 nM T01138 D06ABF 3957 IC50 = 4000 nM T01138 D0S1CQ 133017 IC50 > 40000 nM T01138 D0C2HI 60680 IC50 = 54800 nM T01138 C0TSD5 31843 IC50 > 80000 nM T01138 CA95CK 4161540 IC50 = 18300 nM T01138 CL4VY5 10137458 IC50 = 16100 nM T01138 CQWE69 10363386 IC50 = 4600 nM T01138 CF97IO 14554122 IC50 = 26400 nM T01138 CZQM08 14554127 IC50 = 4900 nM T01138 CSXR86 14554128 IC50 = 5300 nM T01138 CJU02M 14554129 IC50 = 36000 nM T01138 C80GMR 18337326 IC50 > 80000 nM T01138 C8RD9C 18337327 IC50 > 80000 nM T01138 CI2W9S 18337331 IC50 = 7800 nM T01138 C71YDN 18337336 IC50 = 19600 nM T01138 C9RWZ3 18382725 IC50 = 4500 nM T01138 C74WSR 20659961 IC50 = 5700 nM T01138 COP68C 22914796 IC50 = 22900 nM T01138 C29SNE 29918864 IC50 = 17600 nM T01138 CFGH46 29976517 IC50 > 80000 nM T01138 C5F8WR 29976521 IC50 > 80000 nM T01138 C5GW8F 29981724 IC50 > 80000 nM T01138 C9MZ5R 29983056 IC50 = 12400 nM T01138 CLK4Y7 59047051 IC50 = 14800 nM T01138 CS2N1P 118721922 IC50 = 35000 nM T01138 C5CV9A 118721923 IC50 > 80000 nM T01138 CB3L9V 118721924 IC50 = 16800 nM T01138 CGE6B0 118721925 IC50 > 80000 nM T01138 CZF1A9 118721926 IC50 = 4900 nM T01138 CVI2B6 118721927 IC50 = 41500 nM T01138 C2K6ML 118721928 IC50 = 5000 nM T01138 C6YF0A 118721929 IC50 = 10800 nM T01138 CK03VE 118721930 IC50 = 3400 nM T01138 CD0O2N 118721931 IC50 = 5200 nM T01138 C7JP0Z 118721932 IC50 = 18700 nM T01138 CI56NQ 118721933 IC50 = 39100 nM T01138 CBM7V0 118721934 IC50 = 7700 nM T03634 D07SDQ 969516 IC50 = 25000 nM T03634 D0PH9I 118693659 Ki = 6309.57 nM T03634 D0U2BH 65064 IC50 = 50000 nM T03634 D0ZW4W 46907787 IC50 = 9600 nM T03634 CZI4N9 13387 IC50 = 2300000 nM T03634 C5XSG3 19868 IC50 = 32000 nM T03634 C76RDA 43000 IC50 > 50000 nM T03634 CFAL50 43001 IC50 > 50000 nM T03634 CZX1K3 223771 IC50 > 200000 nM T03634 CJ6X2Y 572983 IC50 = 10000 nM T03634 CAT79Z 589098 IC50 = 99000 nM T03634 CG5O0H 638578 IC50 = 11800 nM T03634 CM1EX8 735746 IC50 > 2000000 nM T03634 COP70H 735747 IC50 = 27000 nM T03634 CGR7Y5 755980 IC50 > 50000 nM T03634 CBG2A0 1078352 IC50 = 230 nM T03634 CVF47X 1238761 IC50 > 50000 nM T03634 CML94F 1415890 IC50 = 30000 nM T03634 C2M0SE 1511198 IC50 = 1584.89 nM T03634 CJK1F0 1511199 IC50 = 1258.93 nM T03634 CJWR09 1561807 IC50 = 41000 nM T03634 CS05BM 1600566 IC50 = 115700 nM T03634 C6XQA3 1797300 IC50 = 3200 nM T03634 CE17KZ 1821586 IC50 = 9110 nM T03634 CH01FB 2054569 IC50 = 41360 nM T03634 COZK67 2728636 IC50 = 7000 nM T03634 CV8A1O 2763642 IC50 = 1900000 nM T03634 C3GU6L 2766364 IC50 = 40000 nM T03634 CXD3U8 3152392 IC50 > 200000 nM T03634 C9GO8K 3326945 IC50 > 50000 nM T03634 C2P6IC 3846558 IC50 = 29400 nM T03634 CJ73FZ 4247469 IC50 = 440 nM T03634 CR3SF5 4907545 IC50 = 15848.93 nM T03634 CWG19Q 4908238 IC50 = 6309.57 nM T03634 CUGH30 5157255 IC50 > 50000 nM T03634 CO1H6V 5304236 IC50 = 1440 nM T03634 C8BZ9Y 5325760 IC50 > 200000 nM T03634 CQCH54 6210261 IC50 = 60000 nM T03634 CV67KR 6490661 IC50 = 16730 nM T03634 CH41UK 9992116 IC50 = 2500 nM T03634 CV47EZ 10081070 IC50 = 500000 nM T03634 CUD8X4 10355367 IC50 = 5280 nM T03634 C93EDN 10442296 IC50 > 100000 nM T03634 CK8O6Q 11238147 IC50 = 3000 nM T03634 CT53WA 12206142 IC50 > 200000 nM T03634 C75UZW 12564532 IC50 = 455000 nM T03634 C34GWI 12622087 IC50 = 12000 nM T03634 CE24BV 12689741 IC50 > 50000 nM T03634 C7U9KW 13099766 IC50 = 1950 nM T03634 CCSB13 16662818 IC50 = 1670 nM T03634 C49GBY 27604952 IC50 = 3000 nM T03634 C3UFS6 39791103 IC50 = 3400 nM T03634 C1OEL5 40889550 IC50 = 23000 nM T03634 C2P0IW 44243549 IC50 = 55700 nM T03634 C8XFC2 45494549 IC50 = 13620 nM T03634 CEK9S5 45917950 IC50 > 50000 nM T03634 CV92LK 46786182 IC50 > 50000 nM T03634 CHFE80 51081283 IC50 > 100000 nM T03634 C35MQH 51371083 IC50 = 270 nM T03634 CFX06I 51721279 IC50 = 6800 nM T03634 CG3PR6 52912222 IC50 = 31622.78 nM T03634 C4XCJ0 53257845 IC50 = 2850 nM T03634 CQEF28 53308655 IC50 = 32200 nM T03634 CEK3X6 54757749 IC50 = 86900 nM T03634 C1D3WH 54757750 IC50 = 45400 nM T03634 C1DZ7Y 54757751 IC50 = 49400 nM T03634 C6W5OZ 54757752 IC50 = 12900 nM T03634 CBOE48 56669892 IC50 = 1270 nM T03634 CT76FH 56877138 IC50 = 55000 nM T03634 CCGW97 60149330 IC50 = 758 nM T03634 C6KWC8 69236418 IC50 = 130000 nM T03634 C9L0KD 70699440 IC50 = 1100 nM T03634 CV7OR2 70699441 IC50 = 771 nM T03634 C4MJ0T 71624784 IC50 = 4100 nM T03634 CIX91F 71624785 IC50 = 6300 nM T03634 C1D8GF 71624786 IC50 = 8600 nM T03634 C3R9WA 71624787 IC50 = 8500 nM T03634 CLQ1X8 71624896 IC50 = 10800 nM T03634 CODK30 71624901 IC50 = 3960 nM T03634 CI15JC 71624902 IC50 = 2070 nM T03634 CLZ7C8 71624903 IC50 = 2810 nM T03634 CIPN50 71760902 IC50 = 1000 nM T03634 CA81BL 72201025 IC50 = 240 nM T03634 CQ78NK 76310219 IC50 = 199.53 nM T03634 CM4J8Q 76317442 IC50 = 630.96 nM T03634 CM7TH3 76328466 IC50 = 794.33 nM T03634 C0T5NK 76335637 IC50 = 630.96 nM T03634 C5TB9S 77843982 IC50 = 1000 nM T03634 CL3R7M 81689862 IC50 = 1000 nM T03634 CB9AL4 86287631 IC50 = 3700 nM T03634 CYQ91J 90667397 IC50 = 3980 nM T03634 CS3W6O 90667751 IC50 = 40900 nM T03634 CZBD29 90667752 IC50 = 28400 nM T03634 CF4W8Q 90667754 IC50 = 35900 nM T03634 C2B4NA 90667755 IC50 = 38500 nM T03634 C32KSA 91808023 IC50 = 8700 nM T03634 CTA46H 91826273 IC50 = 1100 nM T03634 C0N1GO 91826363 IC50 = 630 nM T03634 C8XL0I 91826394 IC50 = 1400 nM T03634 CD0W7N 91971372 IC50 = 210 nM T03634 C9WB3G 95828281 IC50 = 740 nM T03634 CJ4MO9 95991007 IC50 = 18000 nM T03634 CB19IE 102358573 IC50 = 323 nM T03634 C89GTS 113207960 IC50 = 25370 nM T03634 C7ZLK4 113207965 IC50 = 3390 nM T03634 CGUK73 117098446 IC50 = 39550 nM T03634 CPB3K7 118626392 IC50 = 1000 nM T03634 CZ07JN 118626421 IC50 = 64000 nM T03634 CTF52P 118626429 IC50 = 5000 nM T03634 C9OD6I 118626439 IC50 = 15000 nM T03634 CBQI47 118626440 IC50 = 7400 nM T03634 CA3Q1L 118626445 IC50 = 2000 nM T03634 CD1L7R 118626450 IC50 = 3000 nM T03634 C4H3GM 118633152 IC50 = 7500 nM T03634 CT31MB 118633154 IC50 = 3000 nM T03634 CU95AV 118740117 IC50 = 32000 nM T03634 CFMJ96 119081417 IC50 = 130 nM T03634 C8AZ4C 119081691 IC50 > 20000 nM T03634 CUWX94 119081692 IC50 = 560 nM T03634 C4JN5Q 121237855 IC50 = 120 nM T03634 C4AU0X 121237856 IC50 = 10600 nM T03634 C7A2UY 121237857 IC50 = 650 nM T03634 CBN53Q 121271705 IC50 = 4100 nM T03634 CGBI67 121271742 EC50 = 1900 nM T03634 CPU76D 121271756 IC50 = 250 nM T03634 CN4X9G 121271781 IC50 = 33 nM T03634 CB83MK 121271792 EC50 = 300 nM T03634 C0F6MH 121277645 IC50 = 120000 nM T03634 C0FA3C 121277864 EC50 = 3400 nM T03634 CP1NH2 121277975 IC50 = 3.4 nM T03634 C0XVY8 121277987 EC50 = 1200 nM T03634 CHO97R 121277993 IC50 = 130 nM T03634 COW87E 121278062 IC50 = 110 nM T03634 C1PGY8 121278155 IC50 = 240 nM T03634 C3GD2W 121335190 IC50 > 20000 nM T03634 CECP26 121335281 IC50 > 20000 nM T03634 C8YE5F 121365519 IC50 = 1.5 nM T03634 C4UHQ1 121372691 IC50 = 150 nM T03634 C46MHD 121372830 IC50 = 2 nM T03634 C34YHN 121372887 IC50 = 410 nM T03634 CL67ME 121372914 IC50 = 120 nM T03634 CQ8ZL9 121372939 IC50 = 320 nM T03634 C3I8SV 121372947 IC50 = 1 nM T03634 CVO7B2 121373072 IC50 = 4.7 nM T03634 C57GXL 121373316 IC50 = 1 nM T03634 C04UKS 121373365 IC50 = 1.2 nM T03634 CDH8M4 121373418 IC50 = 1.1 nM T03634 C1TK3U 121373476 IC50 = 1800 nM T03634 C2V6AX 121373769 IC50 = 3.1 nM T03634 C47QXT 121376807 IC50 = 20 nM T03634 C9XWC0 121376818 IC50 = 31 nM T03634 C0QKG5 121376850 IC50 = 4.3 nM T03634 CP6R5B 121382912 IC50 = 46 nM T03634 CVY6B3 122191330 IC50 = 5370 nM T03634 C1EGJ9 122664496 IC50 = 51000 nM T03634 CWJD15 122705990 IC50 = 1710 nM T03634 C5Z9EY 127025709 IC50 > 100000 nM T03634 CNX2L1 127026318 IC50 > 100000 nM T03634 CDA04U 127026319 IC50 > 100000 nM T03634 CP52CH 127027538 IC50 > 10000 nM T03634 C0E7IG 127029904 IC50 > 10000 nM T03634 CT19QO 127029905 IC50 = 1500 nM T03634 C3IJM2 127032947 IC50 = 500000 nM T03634 CT5H3K 127034116 IC50 = 5000 nM T03634 CS56IU 127035170 IC50 = 500000 nM T03634 C6BT3U 127048317 IC50 = 620 nM T03634 C9DY4Z 127048318 IC50 = 670 nM T03634 CEN16G 127049286 IC50 = 900 nM T03634 C9C0MB 127049631 IC50 = 1900 nM T03634 C8MXQ7 127049932 IC50 = 6500 nM T03634 C12KXI 127051477 IC50 = 3400 nM T03634 C5EYK2 127053005 IC50 = 530 nM T03634 CG6AY7 127053006 IC50 = 5000 nM T03634 CY6ZE0 131955089 IC50 = 15 nM T03634 CN62BM 131955090 IC50 = 59 nM T03634 CGNQ49 132168874 IC50 = 170 nM T03634 CHC6A0 132168907 IC50 = 58 nM T03634 CRV1I6 132168917 IC50 = 2.4 nM T03634 CB4X0G 132169005 IC50 = 69 nM T03634 CX9U1Y 132169030 IC50 = 120 nM T03634 CO7QW0 132169133 IC50 = 24 nM T03634 CD8SE7 132169397 IC50 = 69 nM T03634 CG4X6Z 132169416 IC50 = 42 nM T03634 CV8F3O 132169466 IC50 = 90 nM T03634 C7EHB4 132169581 IC50 = 13 nM T03634 CI3HC8 132169624 IC50 = 9.5 nM T03634 CF7H3C 132169928 IC50 = 450 nM T03634 C6HQ0I 132181409 IC50 = 34 nM T03634 C2S4IT 132181414 IC50 = 3.6 nM T03634 C3MV7Y 132181499 IC50 = 5 nM T03634 CM2K6Z 132181651 IC50 = 69 nM T03634 CZW36J 132181706 IC50 = 47 nM T03634 CVZ87Y 132181707 IC50 = 20 nM T03634 CXVW94 132181717 IC50 = 38 nM T03634 CG13LT 132186451 IC50 = 38 nM T03634 CGC84J 132186467 IC50 = 65 nM T03634 CB23YA 132186468 IC50 = 31 nM T03634 C06KYU 132186469 IC50 = 1.2 nM T03634 CI56DE 132186470 IC50 = 81 nM T03634 COK17B 132186514 IC50 = 130 nM T03634 CE3H2T 132186523 IC50 = 1.2 nM T03634 CG5SN9 132186583 IC50 = 120 nM T03634 CN90OX 132186586 IC50 = 30 nM T03634 CAR2X5 132186700 IC50 = 3.3 nM T03634 C5A3QS 132186701 IC50 = 2.8 nM T03634 CKY07I 132186706 IC50 = 79 nM T03634 C4DOU1 132186760 IC50 = 90 nM T03634 CFB2X6 132186767 IC50 = 23 nM T03634 CM6K0J 132186772 IC50 = 13 nM T03634 CL29US 132186773 IC50 = 27 nM T03634 CC6PW8 132186817 IC50 = 31 nM T03634 CUH7W8 132186890 IC50 = 3.3 nM T03634 C31EOG 132275014 IC50 = 19 nM T03634 CGDN94 132275066 IC50 = 0.94 nM T03634 CL1FY9 132451787 IC50 = 1.4 nM T03634 COR87Y 134812725 IC50 = 140 nM T03634 CBF35S 134812726 IC50 = 2200 nM T03634 C3J8KX 134812727 IC50 = 146 nM T03634 C8IDE3 134812728 IC50 = 40 nM T03634 CS7WX6 134821995 IC50 > 20000 nM T03634 CI2AM1 134828588 IC50 = 2450 nM T03634 CV4X7R 135566898 Ki = 7150 nM T03634 CU2F1G 135566900 Ki = 5120 nM T03634 CW94QO 136226511 Ki = 5590 nM T03634 C60DNA 137250528 IC50 = 43 nM T03634 CO71RI 137285009 IC50 > 10000 nM T03634 CS9MR6 137285011 IC50 > 10000 nM T03634 CI1WA0 137319664 IC50 = 130 nM T03634 C53KAO 137631500 IC50 = 300 nM T03634 CA2VS4 137631629 IC50 = 500 nM T03634 C0Y3UF 137631784 IC50 = 740 nM T03634 CUE7F1 137631875 IC50 = 76 nM T03634 C25OZB 137632559 IC50 = 1400 nM T03634 C9XVL1 137635109 IC50 = 260 nM T03634 CM9P2A 137635443 IC50 = 2.2 nM T03634 C0D1LR 137635790 IC50 = 61 nM T03634 CQT3A9 137636309 IC50 > 100000 nM T03634 CYZJ80 137636683 IC50 = 160 nM T03634 C7NZ4E 137637179 IC50 = 330 nM T03634 CT2D8X 137638314 IC50 = 580 nM T03634 CRN21V 137638824 IC50 = 650 nM T03634 CJG6R8 137640750 IC50 = 90 nM T03634 C0SYB2 137640929 IC50 = 170 nM T03634 COK20S 137641504 IC50 = 200 nM T03634 C01BVT 137642411 IC50 = 450 nM T03634 COY3A6 137642659 IC50 = 920 nM T03634 C0R3FG 137646519 IC50 = 39 nM T03634 CWJ7N5 137647079 IC50 = 690 nM T03634 CJ9UI7 137647118 IC50 = 31 nM T03634 CXD50J 137647775 IC50 = 2500 nM T03634 C89VWP 137649346 IC50 = 310 nM T03634 C85QNS 137649815 IC50 = 470 nM T03634 CKN60B 137649822 IC50 = 500 nM T03634 CO7K6Y 137649906 IC50 = 360 nM T03634 C4Y8HV 137650663 IC50 = 310 nM T03634 CE42GP 137650954 IC50 = 400 nM T03634 CSV15U 137650957 IC50 = 540 nM T03634 CV9F6J 137651164 IC50 = 1500 nM T03634 CHN7A8 137652035 IC50 = 200 nM T03634 CCZD32 137652808 IC50 = 140 nM T03634 CHU2W4 137653154 IC50 > 30000 nM T03634 C7Y6IH 137653562 IC50 = 210 nM T03634 CL1V9T 137654008 IC50 = 240 nM T03634 C3OX9R 137655043 IC50 = 2400 nM T03634 CM7Y4D 137655923 IC50 = 980 nM T03634 C5B7LO 137656022 IC50 = 780 nM T03634 CX35DY 137656164 IC50 = 240 nM T03634 C8BP5R 137656667 IC50 = 310 nM T03634 CW9C8L 137657087 IC50 = 400 nM T03634 C5TEY3 137657620 IC50 = 1300 nM T03634 CE3CQ5 137659158 IC50 = 130 nM T03634 CQ6XB7 139030526 IC50 > 100000 nM T03634 CYQ79A 139382567 IC50 = 81 nM T03634 C9IDO1 141736322 IC50 = 1860 nM T03634 CWM80Y 141736350 IC50 = 33850 nM T03634 C7YR4W 141736357 IC50 = 690 nM T03634 C8ZQ2U 141736359 IC50 = 140 nM T03634 CV7G1U 141736363 IC50 = 19840 nM T03634 C5VNM4 141736367 IC50 = 37 nM T03634 C1P3TL 141736369 IC50 = 2070 nM T03634 C5O6SU 141736374 IC50 = 1000 nM T03634 C4SCT9 141736375 IC50 = 2800 nM T03634 CB68VY 141736376 IC50 = 3520 nM T03634 C4NHG5 141736379 IC50 = 4050 nM T03634 C1V4ND 141736380 IC50 = 1440 nM T03634 CM6ZO2 141736388 IC50 = 32640 nM T03634 C7SQ8T 141736403 IC50 = 6360 nM T03634 C0TB5Z 141736419 IC50 = 26190 nM T03634 C0RV7I 141736434 IC50 = 170 nM T03634 C5UAO0 145949218 IC50 = 2330 nM T03634 COT05Q 145949275 IC50 = 1670 nM T03634 C4IXO6 145950180 IC50 = 290 nM T03634 CIA1W6 145950654 IC50 = 1890 nM T03634 C96NCH 145950955 IC50 = 770 nM T03634 C03SNP 145951746 IC50 = 3890 nM T03634 CYS60Q 145951844 IC50 = 2990 nM T03634 C3ZV1O 145952497 IC50 = 1690 nM T03634 C6LO5F 145953516 IC50 = 2740 nM T03634 C2YR6U 145953602 IC50 = 1690 nM T03634 CSR9N7 145953663 IC50 = 2560 nM T03634 CTE74G 145954441 IC50 = 1000 nM T03634 CR6OX1 145954766 IC50 = 2650 nM T03634 C2Y3ZT 145955733 IC50 = 2330 nM T03634 CNQD23 145956474 IC50 = 4700 nM T03634 CCNU52 145956492 IC50 = 2470 nM T03634 C1NSW8 145956646 IC50 > 50000 nM T03634 C4AI2J 145957252 IC50 = 6560 nM T03634 CN5YO3 145957310 IC50 = 160 nM T03634 CN7G8J 145957486 IC50 = 2480 nM T03634 C7C5WL 145958595 IC50 = 650 nM T03634 C2TH1N 145959035 IC50 = 4840 nM T03634 CE5FW8 145959058 IC50 = 8500 nM T03634 CW6O3D 145959144 IC50 > 50000 nM T03634 CCP03T 145959259 IC50 = 2810 nM T03634 CDNG83 145959505 IC50 = 2060 nM T03634 C4Y0PN 145967100 IC50 = 280 nM T03634 C3BSE8 145971523 IC50 = 1560 nM T03634 C5CXR4 145971749 IC50 = 1960 nM T03634 CIU53N 145972433 IC50 = 7090 nM T03634 CEY8P5 145972450 IC50 = 3390 nM T03634 CNU4O9 145972623 IC50 = 0.9 nM T03634 CC8LU2 145972824 IC50 = 240 nM T03634 CD4A3Y 145973334 IC50 = 650 nM T03634 CR3E9H 145973362 IC50 = 21580 nM T03634 C37UVN 145973834 IC50 = 4110 nM T03634 CP49HN 145974181 IC50 = 180 nM T03634 CA85TK 145975493 IC50 = 190 nM T03634 CZV20H 145976144 IC50 = 7700 nM T03634 CQN6G3 155532286 IC50 > 20000 nM T03634 C0QV9U 155534567 IC50 > 20000 nM T03634 C95OQP 155536635 IC50 = 1200 nM T03634 C62EMT 155540785 IC50 > 20000 nM T03634 C7VRN8 155541456 IC50 > 20000 nM T03634 C5NU8A 155564453 IC50 > 20000 nM T03634 D00DXI 135566302 IC50 = 5000 nM T03634 D03XXT 72201027 IC50 = 30 nM T03634 D09HBR 135566899 Ki = 2180 nM T03634 D0H3TC 54669868 IC50 = 28100 nM T03634 D0J3JI 90488984 IC50 = 440 nM T03634 D0O2RX 71624782 IC50 = 2480 nM T03634 D0YL8Z 1285940 IC50 = 2.6 nM T66237 D03KZM 216237 Ki = 0.43 nM T66237 D08FJL 16681432 EC50 = 170 nM T66237 D09GOS 2812 IC50 = 15848.93 nM T66237 D0D8XY 5311010 Ki = 330 nM T66237 D0F4NS 119369 Ki = 9.42 nM T66237 D0K8KX 5280343 IC50 = 15200 nM T66237 D0M3FJ 439302 EC50 = 7.3 nM T66237 D0N4OW 644077 EC50 = 0.05 nM T66237 D0U7SH 5311065 EC50 = 0.2 nM T66237 D0VU2X 151171 Ki = 0.36 nM T66237 D04QZI 11340891 Ki = 950 nM T66237 D06VWL 10298385 EC50 = 24 nM T66237 D07EEN 172997 IC50 = 1 nM T66237 D09WYL 11634973 Ki = 3981.07 nM T66237 D0L6XQ 11157078 IC50 = 34 nM T66237 D0LI1C 44469321 IC50 > 30000 nM T66237 D0S3YN 53330936 EC50 = 2630.27 nM T66237 D0SY9B 9895468 Ki = 290 nM T66237 D02RDE 9939929 IC50 = 20 nM T66237 D03RYS 5311500 EC50 = 0.7 nM T66237 D08ORO 114904 Ki > 10000 nM T66237 D08PAC 6918320 Ki = 37000 nM T66237 D0A1KU 11683187 IC50 = 1530 nM T66237 D0AV0O 3038506 Ki = 91.9 nM T66237 D0I8ZZ 60943 Ki = 178 nM T66237 D0Q8RX 9872389 Ki = 590 nM T66237 CY4WG9 3793 IC50 = 6000 nM T66237 C0R7SI 449224 EC50 = 3.5 nM T66237 C5F1ST 1103817 Ki = 2500 nM T66237 C7AD6Y 5034737 Ki = 2460 nM T66237 CQB93O 5306925 Ki = 507 nM T66237 COSN76 6918573 EC50 = 58 nM T66237 C93WRU 9690136 Ki > 10000 nM T66237 C5E3XU 9799174 IC50 = 390 nM T66237 C4PY7Z 9801970 IC50 = 390 nM T66237 CC07MW 9807249 Ki = 0.9 nM T66237 CC24MQ 9807250 Ki = 15 nM T66237 CO3SD6 9811830 EC50 = 154.88 nM T66237 CML46C 9824954 EC50 = 1.67 nM T66237 C57WZH 9826033 IC50 = 20 nM T66237 CS8Q6R 9826254 IC50 = 3.2 nM T66237 CW8ZA7 9828129 IC50 = 8 nM T66237 C6OV5R 9829108 IC50 > 1000 nM T66237 CK4UY8 9848300 IC50 = 8 nM T66237 CQYU70 9849525 Ki = 5 nM T66237 CZ3M1F 9850567 IC50 = 13 nM T66237 C0K2IJ 9851013 IC50 = 5.2 nM T66237 CU1W4L 9868852 IC50 = 296 nM T66237 C17GIC 9869993 IC50 = 11 nM T66237 CA7RO2 9871426 IC50 = 7 nM T66237 CGTK84 9874047 IC50 = 2.6 nM T66237 C6D0OX 9887157 IC50 = 933 nM T66237 CA2J5M 9888109 IC50 = 91.5 nM T66237 C8LR0K 9889904 IC50 = 413 nM T66237 CT4S6Q 9910527 IC50 = 475 nM T66237 CDFI62 9915472 IC50 = 4 nM T66237 CRM93H 9931699 IC50 = 183 nM T66237 CPBC63 9935694 IC50 = 210 nM T66237 C9DAQ2 9935969 IC50 = 44 nM T66237 C1C6HA 9937535 IC50 = 341 nM T66237 COUA25 9938406 Ki = 130 nM T66237 C4V2XT 9939024 IC50 = 2 nM T66237 CH2K5E 9954641 EC50 = 47 nM T66237 CNJ81W 9959174 EC50 = 1.8 nM T66237 CD4B6A 9959838 IC50 = 7.5 nM T66237 CW9U3E 9961036 IC50 = 11.5 nM T66237 CK97LP 9974701 IC50 = 18 nM T66237 CIE8X5 9981665 Ki = 5600 nM T66237 C9J4MZ 10003306 IC50 = 1.5 nM T66237 CFO98G 10043741 IC50 = 9 nM T66237 CBI6W4 10098338 IC50 = 1.7 nM T66237 CT7SZ8 10119966 Ki = 21 nM T66237 C1C4SX 10142915 Ki = 2470 nM T66237 C98HVI 10144208 Ki = 8520 nM T66237 C68ZRW 10156521 IC50 = 2000 nM T66237 CRQW02 10162731 EC50 = 2.3 nM T66237 CL71MC 10164478 Ki = 1780 nM T66237 C2NEU9 10165683 Ki = 8890 nM T66237 C7VW8K 10187283 Ki = 585 nM T66237 CZPR64 10187625 EC50 = 890 nM T66237 C91QFB 10206789 EC50 = 4.7 nM T66237 CV7A0N 10206901 Ki = 6930 nM T66237 CPE3F8 10208389 Ki = 14400 nM T66237 CP7N1H 10231366 IC50 = 4 nM T66237 CV2Z3J 10278394 Ki = 4850 nM T66237 CH2XI7 10279928 IC50 = 6 nM T66237 C8UK7I 10281429 EC50 = 10 nM T66237 C72BJX 10282736 EC50 = 1100 nM T66237 C4LU8J 10303620 Ki = 979 nM T66237 C52SOK 10304617 Ki = 1920 nM T66237 CF6A5Y 10322392 IC50 = 67 nM T66237 CW50TU 10345610 EC50 = 215 nM T66237 CPA89S 10390899 IC50 = 6.8 nM T66237 C06SVZ 10392505 IC50 = 7 nM T66237 CTWG68 10411308 Ki = 0.57 nM T66237 CKD75B 10414302 Ki = 3.2 nM T66237 C1OIW6 10416272 Ki > 3000 nM T66237 C8DWH6 10456892 EC50 = 13 nM T66237 C5JSO3 10459252 IC50 = 2.7 nM T66237 C1Z3WY 10461417 IC50 = 11 nM T66237 CR6VX2 10483105 Ki = 181 nM T66237 C9H8WU 10495509 IC50 = 4.1 nM T66237 C8WK5N 10498917 IC50 = 13 nM T66237 CY58RQ 10503858 IC50 = 2.1 nM T66237 C6WXS4 10519373 IC50 = 35 nM T66237 C6PS5H 10569977 IC50 = 8.8 nM T66237 C79NZO 10570880 IC50 = 13 nM T66237 CM7Q1K 10578000 IC50 = 80 nM T66237 CFP17Y 10578460 IC50 = 60 nM T66237 C2Z7RB 10587836 IC50 = 180 nM T66237 CS39QY 10591515 IC50 = 320 nM T66237 CQEP07 10595255 IC50 = 120 nM T66237 CR01ZV 10603742 IC50 > 10000 nM T66237 CSP1C3 10626339 IC50 = 80 nM T66237 CD9ZU1 10642447 IC50 = 5 nM T66237 C5NIU8 10648029 IC50 = 0.5 nM T66237 CLXT94 10672170 IC50 = 1.9 nM T66237 C8VB3L 10673295 IC50 = 2 nM T66237 CZKU73 10673699 IC50 = 8.3 nM T66237 C4RAN8 10691737 IC50 = 16 nM T66237 CYE0I7 10696913 IC50 = 1.9 nM T66237 CRAC01 10710850 IC50 = 1000 nM T66237 C96EYF 10711405 IC50 = 18 nM T66237 CCU35N 10715974 Ki = 7.56 nM T66237 CH84ZE 10719289 IC50 = 4 nM T66237 CEC70P 10737018 IC50 = 22 nM T66237 C6FW1B 10737785 IC50 = 51 nM T66237 CR8QV4 10742418 IC50 = 1 nM T66237 CL1N4A 10743786 IC50 = 0.7 nM T66237 CODM17 10758700 IC50 = 34 nM T66237 CU4EL3 10766720 IC50 = 2 nM T66237 CCHY18 10784361 IC50 = 210 nM T66237 C4GTY9 10814200 IC50 = 4.2 nM T66237 C5GB4F 10831068 IC50 = 5.9 nM T66237 CA9C1V 10831734 IC50 = 7.5 nM T66237 C2TL5U 10837633 IC50 = 4 nM T66237 C58XOT 10840974 IC50 = 50 nM T66237 C3U6QA 10863737 Ki = 11100 nM T66237 CQJ52W 10873853 Ki = 8170 nM T66237 C1WD7P 10907482 Ki = 6650 nM T66237 CI8AQ1 10929819 Ki = 14300 nM T66237 CMZ2W9 10984131 IC50 = 14 nM T66237 CBOS05 11016093 Ki = 4430 nM T66237 C9GX3E 11070458 IC50 = 980 nM T66237 CFL2P5 11092056 Ki = 10200 nM T66237 CDF9W0 11144861 Ki = 7370 nM T66237 C4C8QJ 11158261 IC50 = 9 nM T66237 CZWJ61 11167861 IC50 = 30 nM T66237 C4JKH8 11190868 IC50 = 30 nM T66237 C0FJM7 11194023 Ki = 568 nM T66237 C6D3UR 11237434 EC50 = 265 nM T66237 C2PE4M 11238362 IC50 = 71 nM T66237 CB43VY 11239468 IC50 = 30 nM T66237 CO3A5Z 11240155 Ki = 36.8 nM T66237 CC0KT1 11251777 Ki = 621 nM T66237 CUED54 11257380 Ki > 10000 nM T66237 CU1E4A 11261339 IC50 = 120 nM T66237 C9Q7RV 11262100 IC50 = 80 nM T66237 CE0DX4 11269308 IC50 > 10000 nM T66237 CZ0JW9 11270497 IC50 > 10000 nM T66237 C89CZT 11272841 IC50 = 200 nM T66237 C5OTG4 11274745 Ki = 1090 nM T66237 C9T8BV 11286254 Ki = 80 nM T66237 CB6TF8 11297732 Ki = 1067 nM T66237 CTP85J 11317662 IC50 < 10 nM T66237 CFU2E1 11351397 IC50 = 60 nM T66237 CN2YM9 11365307 IC50 = 50 nM T66237 CYJ23D 11384094 Ki = 103 nM T66237 CON43W 11386922 IC50 = 20 nM T66237 CPND10 11389106 Ki = 24.7 nM T66237 CHRT50 11397211 IC50 < 10 nM T66237 CEM1X7 11400547 Ki = 1386 nM T66237 C93VQG 11418441 IC50 > 10000 nM T66237 CPG63Z 11422294 IC50 = 8 nM T66237 CG0Q5O 11432362 IC50 = 53 nM T66237 CR4N5I 11465834 Ki = 39.81 nM T66237 CM83DS 11468862 Ki = 11170 nM T66237 C37TNB 11475469 Ki > 10000 nM T66237 CN14VO 11476070 IC50 > 10000 nM T66237 C9SY7Q 11486351 Ki = 6400 nM T66237 COC7Q9 11488952 Ki = 5011.87 nM T66237 CIS2N6 11490514 IC50 = 1 nM T66237 CZ3PM4 11490613 IC50 = 6 nM T66237 CR5SH4 11502419 Ki > 10000 nM T66237 C5PU0J 11538526 Ki > 10000 nM T66237 CQ96XZ 11569194 Ki = 1258.93 nM T66237 C60DKW 11569672 Ki > 79432.82 nM T66237 CM15EB 11574636 Ki > 10000 nM T66237 CG7CL9 11578939 EC50 = 281.84 nM T66237 CU9F1K 11618185 Ki > 10000 nM T66237 CFPR21 11625088 Ki > 10000 nM T66237 CQ4SX5 11667812 Ki > 10000 nM T66237 CY0HE4 11677610 IC50 > 100000 nM T66237 CIC93G 11740743 Ki = 2.68 nM T66237 CVWH18 11757222 IC50 = 15 nM T66237 COJ27D 11763684 IC50 = 10 nM T66237 CJ7BP8 11792631 IC50 = 19 nM T66237 C6XGN2 11793558 IC50 = 31 nM T66237 C91CIO 11815584 Ki = 50 nM T66237 C8GC2P 11854507 IC50 > 100000 nM T66237 CEX2I5 14182908 Ki = 400000 nM T66237 C4CTD2 14257660 EC50 = 0.4467 nM T66237 C1E4BW 15298022 IC50 = 510 nM T66237 CEI74X 15307998 IC50 = 9 nM T66237 CIDT94 15307999 IC50 = 19 nM T66237 CMP0I2 15308000 IC50 = 0.7 nM T66237 C06DHE 15416417 Ki = 4.87 nM T66237 CU3M1I 15416418 Ki = 8.3 nM T66237 C9HNQ6 15896091 EC50 = 140 nM T66237 C0WNE9 15896092 EC50 = 180 nM T66237 CA3B4L 15896094 EC50 = 37 nM T66237 CTEW91 15951937 Ki > 27000 nM T66237 C1SKJ3 15953022 Ki = 9308 nM T66237 CHU5E4 16051933 Ki = 5 nM T66237 C3TX0W 18759802 EC50 = 210 nM T66237 CUX27F 18759808 EC50 = 150 nM T66237 C2U0JN 18759812 EC50 = 140 nM T66237 C0OT2Q 18759822 EC50 = 120 nM T66237 CFOU06 18759824 EC50 = 100 nM T66237 C8CY9A 19607875 Ki = 870 nM T66237 CGDY68 19608069 Ki = 21 nM T66237 CJ8MC9 19699060 IC50 = 140 nM T66237 CGC20J 19699093 IC50 = 130 nM T66237 C65CTX 19699097 IC50 = 71 nM T66237 CY89CI 19699133 IC50 = 150 nM T66237 C6TKQ8 20825285 IC50 = 30 nM T66237 C84GPV 21083206 EC50 = 140 nM T66237 CX5H6M 21083210 EC50 = 180 nM T66237 C8R5PD 21083212 EC50 = 82 nM T66237 C7D8XH 21467167 IC50 = 5 nM T66237 C59LDI 22405322 IC50 = 58 nM T66237 CUD2I8 22405325 IC50 = 15000 nM T66237 CGD49J 22405327 IC50 = 96 nM T66237 CW7O1M 22405331 IC50 = 2500 nM T66237 C10PQM 23505561 IC50 = 170 nM T66237 CE4Z6R 23598556 IC50 = 550 nM T66237 CEOZ91 23598560 IC50 = 29 nM T66237 C71XOU 23598595 IC50 = 14 nM T66237 CBRI52 23598597 IC50 = 110 nM T66237 CJ8Z6N 23598598 IC50 = 8 nM T66237 CM1F7K 23598600 IC50 = 39 nM T66237 CP8GK0 23598619 IC50 > 10000 nM T66237 CPZE93 23598641 IC50 = 18 nM T66237 CP64WA 23598642 IC50 = 44 nM T66237 CG20SB 25132666 IC50 = 40 nM T66237 C7C1TG 25132999 IC50 = 1050 nM T66237 CWSF74 25133000 IC50 = 11 nM T66237 C3Q0AD 25133001 IC50 = 730 nM T66237 CM2CP4 25178587 EC50 = 110 nM T66237 C5PHN1 25178591 EC50 = 130 nM T66237 C3WBD7 25178592 EC50 = 820 nM T66237 CS81BP 25178784 EC50 = 270 nM T66237 C65RXN 25178785 EC50 = 100 nM T66237 CG96CK 25178786 EC50 = 390 nM T66237 C8BE6A 25178787 EC50 = 380 nM T66237 C0FH5N 25178959 EC50 = 46 nM T66237 CHA97X 25178960 EC50 = 27 nM T66237 C1E2JZ 25178961 EC50 = 230 nM T66237 C5MV7R 25178962 EC50 = 1700 nM T66237 CWD3Q1 25178963 EC50 = 120 nM T66237 CLD0E7 25180311 EC50 = 30 nM T66237 C1ACZ3 25180507 EC50 = 730 nM T66237 C27WJL 25180508 EC50 = 680 nM T66237 CHV48R 25180509 EC50 = 950 nM T66237 CA9B6P 25180695 EC50 = 350 nM T66237 C5EGS7 25180696 EC50 = 3.2 nM T66237 COJ3F2 25180697 EC50 = 4.3 nM T66237 C5HPT0 25180884 EC50 = 220 nM T66237 CU1OE3 25180885 EC50 = 1000 nM T66237 CM9D7O 25180886 EC50 = 84 nM T66237 CVF12W 25180887 EC50 = 140 nM T66237 C4FLY0 25181104 EC50 = 40 nM T66237 CM1QA7 25181105 EC50 = 10 nM T66237 COC73W 25212177 Ki = 12589.25 nM T66237 CCX14Y 26434734 Ki = 468 nM T66237 CY67HA 42611262 Ki = 251.19 nM T66237 CS04KE 42629368 EC50 = 4.2 nM T66237 CYGN52 42629369 EC50 = 6.3 nM T66237 CMS6P8 44214518 IC50 = 4 nM T66237 CB82ZC 44232512 EC50 = 160 nM T66237 CBV47F 44243143 Ki = 500 nM T66237 CDI2Q4 44247566 IC50 > 31622.78 nM T66237 CVI6Q3 44275104 Ki = 137 nM T66237 CW7JM3 44275447 Ki = 282 nM T66237 CDQ3A6 44294573 Ki = 3.3 nM T66237 C2J8GK 44316235 Ki = 13.7 nM T66237 CIE6Y1 44316236 Ki = 554 nM T66237 C24NQS 44316241 Ki = 245 nM T66237 CS2ZN9 44321415 Ki = 10200 nM T66237 CK2JA7 44325332 Ki = 3.7 nM T66237 CHW9O4 44325345 Ki = 2.8 nM T66237 CS4UM7 44325362 Ki = 1.9 nM T66237 C4STM0 44325363 Ki = 4.2 nM T66237 CXU9H7 44325377 Ki = 17 nM T66237 C1H6JQ 44325505 Ki = 11 nM T66237 CAUJ69 44325531 Ki = 9 nM T66237 CAG0C8 44325538 Ki = 4.2 nM T66237 CK5TS8 44325543 Ki = 10 nM T66237 CE8F7A 44325545 Ki = 18 nM T66237 CH1P8N 44325558 Ki = 5 nM T66237 CP4FH8 44325579 Ki = 3.2 nM T66237 C6OV2D 44325607 Ki = 2.8 nM T66237 CZ0BD9 44325689 Ki = 11 nM T66237 C91EAF 44325691 Ki = 3.7 nM T66237 CO3ZL8 44325695 Ki = 2 nM T66237 CQ6MC5 44325703 Ki = 1.4 nM T66237 C1BA7W 44325704 Ki = 13 nM T66237 CO9Y1C 44325731 Ki = 10 nM T66237 CW23ZH 44325732 Ki = 10 nM T66237 CR4TV5 44325733 Ki = 15 nM T66237 C19AEH 44325766 Ki = 3.7 nM T66237 CD86NE 44325804 Ki = 8 nM T66237 CG8P5Z 44325895 Ki = 25 nM T66237 CM94YJ 44325896 Ki = 40 nM T66237 CV54FN 44325905 Ki = 37 nM T66237 C08ETV 44325915 Ki = 60 nM T66237 C95HKU 44332168 IC50 = 390 nM T66237 CSF89I 44332181 IC50 > 1000 nM T66237 C6NW1Z 44332207 IC50 = 274 nM T66237 CF3QT6 44332208 IC50 = 159 nM T66237 CPF97V 44332209 IC50 = 180 nM T66237 CRL53G 44332212 IC50 > 1000 nM T66237 C5N1TG 44332226 IC50 > 1000 nM T66237 C4UD2C 44332237 IC50 > 1000 nM T66237 CB2VP5 44332238 IC50 > 1000 nM T66237 C98OKM 44332239 IC50 = 0.2 nM T66237 CLJN56 44332261 IC50 > 1000 nM T66237 CA1OL4 44332269 IC50 > 1000 nM T66237 C8L7KE 44332272 IC50 = 380 nM T66237 C0S9TC 44332273 IC50 = 70 nM T66237 CGT2A0 44335241 IC50 = 72 nM T66237 C6HO3T 44335329 IC50 = 5 nM T66237 CO0EQ9 44335343 IC50 = 13 nM T66237 CZ75ET 44335345 IC50 = 10 nM T66237 C23MCR 44335356 IC50 = 28 nM T66237 CONI47 44335357 IC50 = 19 nM T66237 C8VWX6 44335386 IC50 = 26 nM T66237 C92YST 44336379 IC50 = 23 nM T66237 C7X3QZ 44336402 IC50 > 1000 nM T66237 CDTJ17 44336403 IC50 > 1000 nM T66237 CENA29 44336404 IC50 = 20 nM T66237 CM61WN 44336418 IC50 = 10 nM T66237 C7ML9D 44336636 IC50 = 11 nM T66237 CZYV25 44336768 IC50 = 18 nM T66237 CD62CM 44336784 IC50 = 16 nM T66237 C7AU5H 44336791 IC50 > 1000 nM T66237 C2IJS5 44336799 IC50 > 1000 nM T66237 C1TEP7 44351278 Ki = 6.6 nM T66237 CL2R8E 44351441 Ki = 3.7 nM T66237 COE18X 44351500 Ki = 1.5 nM T66237 CJR5B7 44352302 IC50 = 430 nM T66237 CZ60LX 44352757 IC50 = 7 nM T66237 CM4ZJ0 44352767 IC50 = 100 nM T66237 C9UBG4 44352768 IC50 = 16 nM T66237 C2X8GD 44352776 IC50 = 20 nM T66237 CTNY07 44352777 IC50 = 12 nM T66237 CT3Z9C 44352783 IC50 = 8 nM T66237 CVK34U 44352796 IC50 = 85 nM T66237 CLA4U8 44352804 IC50 = 15 nM T66237 CH41KQ 44357890 IC50 = 0.95 nM T66237 COUJ27 44374802 IC50 = 3.4 nM T66237 CVR8H4 44374839 IC50 = 220 nM T66237 CY4TC0 44375638 Ki = 1 nM T66237 CMI9C7 44377521 IC50 = 550 nM T66237 CQ50CE 44377836 IC50 = 50 nM T66237 CVU70Y 44377837 IC50 = 190 nM T66237 C9WO6P 44377894 IC50 = 180 nM T66237 CXG0R3 44377903 IC50 = 15 nM T66237 C5HWR0 44377961 IC50 = 12 nM T66237 CV1BR7 44378675 IC50 = 8.8 nM T66237 CU6CL9 44378702 IC50 = 2 nM T66237 CPWO06 44378703 IC50 = 2.1 nM T66237 C6TX2Q 44378719 IC50 = 1.3 nM T66237 C6OTD5 44378885 IC50 = 7 nM T66237 C1NA5W 44378886 IC50 = 14.8 nM T66237 CYBX91 44382370 Ki = 1.1 nM T66237 CH47GO 44382498 Ki = 0.99 nM T66237 CKL2S9 44382499 Ki = 1 nM T66237 CJBV97 44386548 IC50 < 10 nM T66237 C9E5JO 44393911 EC50 = 200 nM T66237 CDK52W 44393912 EC50 = 100 nM T66237 CZ4UB9 44393941 EC50 = 570 nM T66237 C9JBI3 44393965 EC50 = 1300 nM T66237 CGW9Z6 44393998 EC50 = 1800 nM T66237 CUS19Z 44394044 EC50 = 230 nM T66237 C05DOG 44394045 EC50 = 1200 nM T66237 CZ4B0C 44394063 EC50 = 1800 nM T66237 C9BH3V 44404614 IC50 = 300 nM T66237 CF80BP 44433360 IC50 = 1214 nM T66237 CS8M2O 44433363 IC50 = 11 nM T66237 CLBA10 44433367 IC50 = 34 nM T66237 CCI04H 44433372 IC50 = 1000 nM T66237 C9BDH6 44433375 IC50 = 1000 nM T66237 CF2U3N 44444760 IC50 = 76 nM T66237 CR8OX5 44444761 IC50 > 10000 nM T66237 C1YR6A 44444762 IC50 = 36 nM T66237 CLE7W0 44466239 IC50 > 31622.78 nM T66237 CKA3S0 44467347 IC50 > 31622.78 nM T66237 C2N8FY 44520848 EC50 = 2.4 nM T66237 C91HXT 44520849 EC50 = 0.99 nM T66237 C3HP9Y 44520850 EC50 = 1 nM T66237 CZ5E2V 44520851 EC50 = 0.98 nM T66237 CMGE92 44520852 EC50 = 1 nM T66237 CVA7R2 44520853 Ki = 20 nM T66237 C1U0RY 44520854 Ki = 19 nM T66237 CHE1Y6 44520855 Ki = 5.6 nM T66237 CCW48G 44520856 Ki = 16 nM T66237 CK7O1L 44520857 Ki = 10 nM T66237 C6TOE7 44520858 Ki = 11 nM T66237 CQF23X 44520859 Ki = 7.4 nM T66237 CFD98V 44520860 Ki = 14 nM T66237 CJCB39 44520861 Ki = 3.4 nM T66237 CTVS34 44520862 Ki = 11 nM T66237 CT5A0C 44520863 Ki = 11 nM T66237 CPR8F2 44520864 Ki = 11 nM T66237 CR7Y8G 44520865 Ki = 12 nM T66237 CUN6S2 44520866 Ki = 27 nM T66237 CY61JM 44520867 Ki = 33 nM T66237 CW9RI7 44520868 Ki = 18 nM T66237 CRIF68 44520869 Ki = 53 nM T66237 C1JN3D 44520870 Ki = 22 nM T66237 C8X5FQ 44520871 Ki = 11 nM T66237 C2SDC4 44563370 EC50 = 50 nM T66237 CZF2R4 44563371 EC50 = 20 nM T66237 CPI04M 44563579 EC50 = 2.1 nM T66237 CMG70R 44577936 Ki = 500 nM T66237 CZD7E3 44577937 Ki = 160 nM T66237 C0HXR2 44577938 Ki > 10000 nM T66237 COP3Q0 44577939 Ki > 10000 nM T66237 C10ZLO 44577981 Ki > 10000 nM T66237 CED75W 44577983 Ki > 10000 nM T66237 C1E6GX 44577984 Ki > 10000 nM T66237 C6R0AW 44578010 Ki > 10000 nM T66237 CLCK14 44579399 Ki > 10000 nM T66237 C6OK3X 44579400 Ki > 10000 nM T66237 C0IHE7 44579401 Ki > 10000 nM T66237 CU31MF 44579402 Ki > 10000 nM T66237 CXOJ34 44579441 Ki > 10000 nM T66237 CMW6Q7 44579442 Ki = 1000 nM T66237 CM7HN8 44581240 Ki = 501.19 nM T66237 CG68XT 44581241 Ki = 1258.93 nM T66237 CC5AT2 44581242 Ki = 251.19 nM T66237 C4FZQ9 44581266 Ki = 63.1 nM T66237 CZ9KU4 44589838 EC50 = 1.8 nM T66237 C8R7ZF 44589839 Ki = 9.2 nM T66237 C8YJ1I 44589840 Ki = 21 nM T66237 C6MRI9 44589841 Ki = 18 nM T66237 C58BYM 44589842 Ki = 11 nM T66237 CR32JK 44589843 Ki = 9.1 nM T66237 CF5LG2 44589844 Ki = 6 nM T66237 CD64HU 44589892 Ki = 20 nM T66237 C4OT3X 44589893 EC50 = 3.13 nM T66237 C4CX0I 44589894 EC50 = 1.25 nM T66237 C7DT5U 44589895 Ki = 16 nM T66237 C91MTZ 44589946 Ki = 14 nM T66237 C6J3KX 44589947 Ki = 11 nM T66237 C49UZD 44589948 Ki = 200 nM T66237 CTA89E 44589949 Ki = 170 nM T66237 CSZ70I 45103785 Ki = 3400 nM T66237 CK4XM7 45103786 Ki > 5000 nM T66237 C6LX7B 46225023 Ki > 10000 nM T66237 C48JOB 46225048 Ki > 10000 nM T66237 CX2S6L 46225049 Ki > 10000 nM T66237 C70FCZ 46225050 Ki > 10000 nM T66237 CIM9Y4 46225051 Ki > 10000 nM T66237 CZ36XD 46225079 Ki > 10000 nM T66237 CA6DS1 46225080 Ki > 10000 nM T66237 COT65W 46225081 Ki > 10000 nM T66237 C53ZIX 46225082 Ki > 10000 nM T66237 CFLW87 46225083 Ki > 10000 nM T66237 C7A8DU 46225116 Ki > 10000 nM T66237 C4E8NX 46225117 Ki > 10000 nM T66237 C3W6VI 46225118 Ki = 2770 nM T66237 CT8LO5 46225153 Ki = 1190 nM T66237 C98EDC 46233065 Ki > 1000 nM T66237 C4K7AV 46830094 Ki = 2400 nM T66237 CH4F6K 46830095 Ki = 2300 nM T66237 CNU72P 46830096 Ki = 2830 nM T66237 C0EMW2 46884414 Ki > 10000 nM T66237 C3FUB6 46884437 Ki > 10000 nM T66237 CM0RI1 46884438 Ki > 10000 nM T66237 C4DP6I 46884439 Ki > 10000 nM T66237 CXTE54 46884441 Ki > 10000 nM T66237 C27WFG 46884478 Ki > 10000 nM T66237 C3U2WD 46884479 Ki > 10000 nM T66237 CB8WK2 46884480 Ki = 343000 nM T66237 CIS28Y 46890052 Ki = 63 nM T66237 CWH0O5 46890053 Ki = 2380 nM T66237 CG35DC 46890054 Ki = 2090 nM T66237 CQPV07 46890055 Ki = 2470 nM T66237 CMBS14 46890099 Ki = 1890 nM T66237 CLFP63 46890100 Ki = 770 nM T66237 CRP96J 46890101 Ki = 130 nM T66237 CNJB38 46890102 Ki > 2500 nM T66237 CE84XQ 46890151 Ki > 2500 nM T66237 C8Y6ET 46890152 Ki = 124 nM T66237 C8CXM4 46890153 Ki = 233 nM T66237 CZWV30 46890154 Ki = 171 nM T66237 CY3P8V 46890184 Ki = 36.5 nM T66237 C60CEY 46890185 Ki = 21 nM T66237 CO4CU1 46890186 Ki = 60.6 nM T66237 CJD1S7 46890187 Ki = 133 nM T66237 CLON70 46890214 Ki = 176 nM T66237 CN76SA 46890215 Ki = 39.2 nM T66237 C0AZT4 46890216 Ki > 2550 nM T66237 CJ0AM6 46890217 Ki > 2550 nM T66237 C1DG3H 46890258 Ki > 2550 nM T66237 CJ2L6D 46890259 Ki > 2550 nM T66237 CM70JW 46890260 Ki > 2550 nM T66237 CQWM92 46890261 Ki = 9.2 nM T66237 CC85GR 46890262 Ki = 82 nM T66237 CIC2E8 46890288 Ki = 40 nM T66237 CC75DR 46890289 Ki = 43.4 nM T66237 CW38OV 46890290 Ki = 420 nM T66237 CHFR58 46890438 Ki = 204 nM T66237 CVD95O 46890439 Ki = 3345 nM T66237 COE5S9 46890440 Ki = 54 nM T66237 C0N1MO 46890484 Ki = 1032 nM T66237 CR84PB 46890485 Ki = 478 nM T66237 CA7BO2 46890486 Ki = 1057 nM T66237 CAR94C 46890487 Ki = 82 nM T66237 CEM4L1 46890528 Ki = 107 nM T66237 C2PYH3 46890529 Ki = 1205 nM T66237 CCI0R6 46890530 Ki > 2500 nM T66237 CF83TS 46890531 Ki = 846 nM T66237 C0T5MG 46890569 Ki = 189 nM T66237 C1JSF8 46890570 Ki > 2500 nM T66237 C9QJ5V 46890571 Ki = 713 nM T66237 C83LYU 46890572 Ki = 1170 nM T66237 C1VNK6 46890612 Ki = 30 nM T66237 C2XDO1 46890613 Ki > 2500 nM T66237 CC9E4R 46890614 Ki = 1810 nM T66237 CCM29N 46890615 Ki = 291 nM T66237 C39HAX 46890654 Ki = 556 nM T66237 CQUA46 46890655 Ki > 2500 nM T66237 CLJ2O5 46890656 Ki = 675 nM T66237 CEH20W 46890657 Ki > 2500 nM T66237 CC7Y0V 46890706 Ki > 2500 nM T66237 CIP1L7 46890707 Ki = 15 nM T66237 CKQ1Y0 46890708 Ki > 2500 nM T66237 C02IDZ 46890709 Ki = 600 nM T66237 CUWG39 46934434 IC50 > 100000 nM T66237 CI9J7N 47177173 Ki = 160 nM T66237 CO9JL6 47177176 Ki = 713 nM T66237 CMPE57 52941704 Ki > 10000 nM T66237 CBDS48 52949017 Ki > 10000 nM T66237 C01HUJ 53349364 Ki = 640 nM T66237 CK2Y5W 53349471 Ki = 98 nM T66237 C4TEY2 53358902 Ki > 10000 nM T66237 C63IVJ 53362154 EC50 = 3000 nM T66237 C21HMW 53362155 EC50 = 1698.24 nM T66237 CF60LM 53362156 EC50 = 1200 nM T66237 CGMY47 53362202 EC50 = 165.96 nM T66237 C9V8RI 53362203 EC50 > 10000 nM T66237 CAL1Y3 53362204 EC50 > 10000 nM T66237 C6N5EX 53362257 EC50 > 10000 nM T66237 CS40QD 53362258 EC50 > 10000 nM T66237 CFWL28 53362259 EC50 = 2600 nM T66237 CNDR76 53362310 EC50 > 10000 nM T66237 COUH09 53362311 EC50 > 10000 nM T66237 C1MU4B 53362312 EC50 > 10000 nM T66237 CLRT87 53362368 EC50 > 10000 nM T66237 CG8J6H 53362369 EC50 > 10000 nM T66237 CD1N3U 53362370 EC50 = 1600 nM T66237 CRY95P 53362428 EC50 = 720 nM T66237 C3TFA8 53362429 EC50 = 130 nM T66237 C4U1PT 53362430 EC50 = 138.04 nM T66237 C09KLV 53362488 EC50 = 257.04 nM T66237 CRX54F 53362489 EC50 = 186.21 nM T66237 C3KCI9 53362490 EC50 = 1100 nM T66237 CW32MV 53362546 EC50 > 10000 nM T66237 C5EG6T 53362547 EC50 = 5248.07 nM T66237 CUD9F0 53362548 EC50 = 1600 nM T66237 CVJ9U2 53362603 EC50 = 3700 nM T66237 CMY7V4 53362604 EC50 > 10000 nM T66237 CK9V1G 53362605 EC50 > 10000 nM T66237 CCRZ83 53362670 EC50 > 10000 nM T66237 CYK9B3 53362671 EC50 = 950 nM T66237 CCK0P6 53362672 EC50 > 10000 nM T66237 CYG85M 53362729 EC50 = 72.44 nM T66237 C1IBT7 53362730 EC50 > 10000 nM T66237 CI0F3Y 53362731 EC50 > 10000 nM T66237 C3XW1F 53362732 EC50 > 10000 nM T66237 CYTJ92 53362793 EC50 > 10000 nM T66237 CQ9CD8 53362794 EC50 > 10000 nM T66237 CAN2C1 53362795 EC50 > 10000 nM T66237 CO4UA0 53362796 EC50 = 389.05 nM T66237 C0NSZ5 53362797 EC50 > 10000 nM T66237 CFJO73 53362798 EC50 > 10000 nM T66237 C2RSW6 53362849 EC50 = 2500 nM T66237 C5K9YV 53362850 EC50 = 114.82 nM T66237 CB3AR7 53362851 EC50 = 200 nM T66237 C42SJF 53362852 EC50 > 10000 nM T66237 C8U6LX 53362853 EC50 > 10000 nM T66237 CH93SM 53362854 EC50 > 10000 nM T66237 C7RYJ0 53362909 EC50 = 330 nM T66237 CKV9D6 53362910 EC50 > 10000 nM T66237 CX9YM6 53362911 EC50 = 467.74 nM T66237 C76TQB 53362913 EC50 > 10000 nM T66237 C5XCD8 53362914 EC50 > 10000 nM T66237 C8N0TX 53362915 EC50 > 10000 nM T66237 CU9X3P 53362962 EC50 = 1200 nM T66237 C61CNE 53362963 EC50 = 1174.9 nM T66237 CF30CI 53362964 EC50 = 758.58 nM T66237 C6SB7W 53362965 EC50 = 970 nM T66237 C32FZM 53362966 EC50 > 10000 nM T66237 CJ06TA 53362967 EC50 > 10000 nM T66237 C6AN7Y 53363015 EC50 = 380 nM T66237 C52IOF 53363016 EC50 = 208.93 nM T66237 C1SHU3 53363017 EC50 = 2600 nM T66237 CNA2L1 53364234 Ki > 10000 nM T66237 C3L7RP 54580516 Ki > 1000 nM T66237 CX1H3Z 54580518 Ki > 1000 nM T66237 C7X4LI 54581307 Ki = 5200 nM T66237 CB5R2M 54581528 Ki > 1000 nM T66237 CR7GD2 54581529 Ki > 1000 nM T66237 CUW8C7 54581530 Ki > 1000 nM T66237 CD21EL 54581533 Ki > 1000 nM T66237 C0ZNY9 54582318 Ki = 31100 nM T66237 CQ7Z8U 54582526 Ki > 1000 nM T66237 C8UN6Y 54582950 IC50 = 8 nM T66237 C7MP0S 54584254 Ki >= 10000 nM T66237 C73IGF 54584265 Ki = 6714 nM T66237 CX5T1G 54584266 Ki = 4918 nM T66237 CIGN05 54584267 Ki = 22010 nM T66237 CC49GD 54584268 Ki = 45000 nM T66237 C9N2QH 54584476 Ki = 618 nM T66237 CD1A0H 54584477 Ki > 1000 nM T66237 CXPY04 54584478 Ki > 1000 nM T66237 CHR91Z 54585227 Ki = 1558 nM T66237 C8YD0H 54585429 Ki = 636 nM T66237 C5N7VS 54585431 Ki > 1000 nM T66237 C3MLH7 54586172 Ki >= 10000 nM T66237 CL79ME 54586390 Ki > 1000 nM T66237 C1N7LU 54586391 Ki > 1000 nM T66237 C60DIQ 54586392 Ki > 1000 nM T66237 CJ76VF 56657866 Ki > 10000 nM T66237 CQG9J6 56657868 Ki > 1000 nM T66237 C31CRV 56658409 EC50 = 1.4 nM T66237 C6T3VC 56658416 EC50 = 4.074 nM T66237 CJ5FQ4 56664848 Ki > 10000 nM T66237 C5V3ME 56664849 Ki > 10000 nM T66237 C3SYC9 56665377 EC50 = 9.12 nM T66237 CQN0G9 56668257 Ki > 10000 nM T66237 CU9DK4 56671721 Ki > 10000 nM T66237 CSL0C7 56671723 Ki > 10000 nM T66237 CK9L4C 56672570 EC50 = 31 nM T66237 C8GLI4 56675151 Ki > 10000 nM T66237 C05JPT 56678446 Ki = 930 nM T66237 CNZU65 56682530 Ki = 9.9 nM T66237 CAG71L 57391220 Ki > 10000 nM T66237 C26OTQ 57394727 Ki > 10000 nM T66237 CFM91W 57399933 Ki > 1000 nM T66237 CHG37B 57519947 Ki = 580 nM T66237 C0DB5C 57519948 Ki = 1800 nM T66237 C15NPY 57520031 Ki = 3700 nM T66237 CBTU57 67839485 Ki = 78 nM T66237 CD1IQ4 70685417 Ki = 1400 nM T66237 CCTZ13 70685423 Ki > 1000 nM T66237 CJM18X 71449932 Ki = 7.6 nM T66237 CUD97X 71451749 Ki = 26.1 nM T66237 C7BCA6 71451750 Ki = 187.7 nM T66237 CJGO63 71451752 Ki = 54.3 nM T66237 C8KO3M 71453576 Ki = 14.05 nM T66237 CG03VC 71455302 Ki = 1.93 nM T66237 C1WME0 71455306 Ki = 16.8 nM T66237 C0IZ5N 71457081 Ki = 5.69 nM T66237 CDU2C8 71460752 Ki = 25.3 nM T66237 CT8C1G 71460754 Ki = 12.7 nM T66237 CE2AI3 71462477 Ki = 0.83 nM T66237 C1Q6RX 71462479 Ki = 4 nM T66237 C8GV2J 71552165 IC50 = 10200 nM T66237 CR14LV 71552166 IC50 = 2000 nM T66237 CZG2O3 71720517 IC50 = 398.11 nM T66237 CPB34Y 73345487 Ki = 7.6 nM T66237 C8N1IS 73347164 Ki = 500000 nM T66237 C2Y4UX 73348432 Ki = 1.5 nM T66237 CKAC48 73348509 Ki = 4.8 nM T66237 COP37N 73348674 Ki = 1100000 nM T66237 C7GDP3 73350017 Ki = 24.1 nM T66237 CLC49J 73350187 Ki = 0.7 nM T66237 C8BRM6 73350188 Ki = 0.5 nM T66237 CS3GK0 73350258 Ki = 1000000 nM T66237 C8GQK9 73350823 Ki = 8700 nM T66237 CQ8UO2 73351518 Ki = 2.1 nM T66237 CY4IW8 73351519 Ki = 117 nM T66237 CG8AD1 73354500 Ki = 4416 nM T66237 CI8Z1B 73354581 Ki = 4.2 nM T66237 C5CDG2 73354746 Ki = 1500000 nM T66237 CQV35P 73356145 Ki = 3.6 nM T66237 CLMY01 76073634 EC50 = 330 nM T66237 C1YLV9 90468623 EC50 = 0.29 nM T66237 CGZ9F1 90469608 EC50 = 0.08 nM T66237 CLXN70 90469674 EC50 = 0.07 nM T66237 CRO49T 90469675 EC50 = 0.1 nM T66237 CSKZ30 90469676 EC50 = 0.39 nM T66237 C3FE9W 118476329 EC50 = 0.22 nM T66237 CGKN68 118476331 EC50 = 0.23 nM T66237 C2TGY7 118476332 EC50 = 0.35 nM T66237 C4HGR0 118476333 EC50 = 0.45 nM T66237 CL2UK1 118476335 EC50 = 0.22 nM T66237 C2G3FX 118476336 EC50 = 0.19 nM T66237 CR3O9G 118476337 EC50 = 0.1 nM T66237 C76ONJ 118476338 EC50 = 0.1 nM T66237 CC2UJ0 118476339 EC50 = 0.38 nM T66237 CTV5Z6 118476341 EC50 = 0.27 nM T66237 C81BRW 118476342 EC50 = 0.29 nM T66237 CRG4T1 118476343 EC50 = 0.12 nM T66237 C3YZ5M 118476344 EC50 = 0.32 nM T66237 C24TBU 118476346 EC50 = 0.26 nM T66237 CEP13D 118476347 EC50 = 0.22 nM T66237 C2RE7I 118476348 EC50 = 0.31 nM T66237 C5E0HL 118476355 EC50 = 0.25 nM T66237 CUMW51 118476356 EC50 = 0.21 nM T66237 C21GNB 118476357 EC50 = 0.1 nM T66237 C6KZH9 118476358 EC50 = 0.23 nM T66237 C69TMC 118476359 EC50 = 0.29 nM T66237 C5Z9SC 118476360 EC50 = 0.14 nM T66237 C36WLI 118476361 EC50 = 0.11 nM T66237 CX9YV2 118476362 EC50 = 0.21 nM T66237 C94FHB 118476365 EC50 = 0.19 nM T66237 CI1E7V 118476366 EC50 = 0.26 nM T66237 CY4WD9 118476367 EC50 = 0.33 nM T66237 CS7DP0 118476369 EC50 = 0.19 nM T66237 C7DAO4 118476383 EC50 = 0.31 nM T66237 C1KUY3 118476384 EC50 = 0.1 nM T66237 C5IFR0 118476385 EC50 = 0.27 nM T66237 C50MTE 118705579 Ki > 100000 nM T66237 C9HX7Z 118705580 Ki > 100000 nM T66237 CR3TZ0 118719818 EC50 = 4.2 nM T66237 CFG2V7 118719819 EC50 = 9.9 nM T66237 C4J6ZO 118719820 EC50 = 35 nM T66237 C9B2WS 118719821 EC50 = 1.8 nM T66237 CAFX95 118719822 EC50 = 690 nM T66237 CH74ZW 118719823 EC50 = 670 nM T66237 C7QI5K 118719824 EC50 = 40 nM T66237 CAP85S 118719825 EC50 = 450 nM T66237 CDR70N 118719826 EC50 = 450 nM T66237 CH0WU8 118719827 EC50 = 77 nM T66237 C1OMZ4 118719828 EC50 = 11 nM T66237 C72LOG 118719829 EC50 = 100 nM T66237 CD0P3Q 118719830 EC50 = 57 nM T66237 CAKC58 118719831 EC50 = 80 nM T66237 CIK48G 118719832 EC50 = 100 nM T66237 CDSK02 118719833 EC50 = 34 nM T66237 C9GSF2 118719834 EC50 = 68 nM T66237 CS89AW 118719835 EC50 = 30 nM T66237 CTWG46 118719836 EC50 = 84 nM T66237 COQ71F 118719837 EC50 = 82 nM T66237 CT3LR1 118719838 EC50 = 78 nM T66237 CX3R0J 118719839 EC50 = 180 nM T66237 CT3O7P 118719840 EC50 = 170 nM T66237 CW2F8P 118719841 EC50 = 380 nM T66237 CC9ZH4 118719842 EC50 = 66 nM T66237 C0LIH8 118719843 EC50 = 180 nM T66237 CYWM79 118719844 EC50 = 47 nM T66237 CGJ05D 118719845 EC50 = 57 nM T66237 CH3DE8 118720259 EC50 = 62 nM T66237 C3DLZ2 118720260 EC50 = 86 nM T66237 COD37S 118720261 EC50 = 230 nM T66237 CPNB13 118720262 EC50 = 1400 nM T66237 CW4Q3B 118720263 EC50 = 1400 nM T66237 CI1SA4 118720264 EC50 = 70 nM T66237 CX2K6O 118720265 EC50 = 52 nM T66237 COHG04 118720266 EC50 = 1100 nM T66237 CL2WY9 118720267 EC50 = 1300 nM T66237 C53KXO 118720268 EC50 = 500 nM T66237 CH2T3S 118720269 EC50 = 150 nM T66237 C7KCE4 118720270 EC50 = 2600 nM T66237 CEK5A6 118720271 EC50 = 73 nM T66237 C4OSR7 118720272 EC50 = 18 nM T66237 C2Z8IG 118720273 EC50 = 2000 nM T66237 C3SD1R 118720274 EC50 = 1200 nM T66237 CXGF75 118720275 EC50 = 110 nM T66237 CZ96MR 118720276 EC50 = 2100 nM T66237 CM1V0E 118720277 EC50 = 1000 nM T66237 CJB1T7 118720278 EC50 = 140 nM T66237 C4KHJ3 118720279 EC50 = 36 nM T66237 C85IJS 118720280 EC50 = 720 nM T66237 CMK0A4 118720281 EC50 = 210 nM T66237 C1KPF5 118720282 EC50 = 55 nM T66237 C9XE0M 118720283 EC50 = 1600 nM T66237 CXV09J 118720284 EC50 = 140 nM T66237 C2VF6Q 118720285 EC50 = 1400 nM T66237 CLE5W1 118720286 EC50 = 100 nM T66237 C8QYZ7 118720287 EC50 = 3000 nM T66237 CMC18U 118720288 EC50 = 250 nM T66237 CF1RM4 118720289 EC50 = 30 nM T66237 CTS3Q9 118720290 EC50 = 760 nM T66237 C3AOC2 118734334 Ki = 184 nM T66237 CT9D1K 118734335 Ki = 880 nM T66237 CBR9L6 118734336 Ki = 820 nM T66237 C7CNM8 132095331 EC50 = 0.2 nM T66237 C3NMS8 132822145 Ki = 170 nM T66237 CGI81M 132822146 Ki = 160 nM T66237 CC09BD 135192928 IC50 = 25665 nM T66237 CWQ30S 135192932 IC50 = 7320 nM T66237 CSQ0Y2 135192979 IC50 = 23047 nM T66237 CQI48P 135192983 IC50 = 32604 nM T66237 CS8A2H 135192997 IC50 = 21450 nM T66237 C86LKI 135413563 EC50 = 850 nM T66237 CM26GP 135506374 Ki >= 58.4 nM T66237 CT0A1P 135916059 Ki = 6.4 nM T66237 CHJ03T 135916060 Ki > 1000 nM T66237 CO6G5W 135916061 Ki > 1000 nM T66237 CAN9M3 135916069 Ki = 913 nM T66237 CH2L4N 135916070 Ki = 29 nM T66237 CO03UG 136961690 Ki = 913 nM T66237 C8R7MZ 137637867 Ki = 140 nM T66237 CW8AC7 137642420 Ki = 54 nM T66237 C8F4QJ 137648906 Ki = 1790 nM T66237 CO2S9U 137652605 Ki = 46 nM T66237 C7XTV3 145711714 EC50 = 41 nM T66237 C63UNT 145960494 EC50 = 3669 nM T66237 CIG1P6 145961670 Ki > 6000 nM T66237 C53JQB 145962220 EC50 = 3900 nM T66237 CRXH51 145963213 Ki > 6000 nM T66237 CY0FL4 145964296 Ki = 334 nM T66237 CS40EH 145965644 Ki < 10 nM T66237 CYSP85 145965794 Ki > 1000 nM T66237 CAHB80 145966126 Ki = 331 nM T66237 CYIE13 145970269 Ki > 1000 nM T66237 C3H7SY 145970757 Ki = 52 nM T66237 C43AQD 145971417 Ki > 1000 nM T66237 CJF16G 145972114 Ki > 1000 nM T66237 CPY61F 145972843 Ki > 1000 nM T66237 CI9G0B 145974527 Ki > 1000 nM T66237 CFQ05K 145974615 Ki < 10 nM T66237 CNF1J3 145974638 Ki = 1148 nM T66237 CVE64Z 145975166 Ki = 233 nM T66237 CJT06P 145976546 Ki = 100 nM T66237 CQ2IG7 145976595 EC50 = 4 nM T66237 CF14DJ 145976648 Ki = 121 nM T66237 CS5CD6 145977918 Ki > 1000 nM T66237 CT1PI4 145978570 Ki = 282 nM T66237 CTYI46 145978612 Ki > 1000 nM T66237 CC65HB 155513872 EC50 = 0.3 nM T66237 C8BKV3 155523986 EC50 = 0.08 nM T66237 C2IZ6F 155535667 EC50 = 0.17 nM T66237 CA6DC4 155542670 EC50 = 0.35 nM T66237 C7N8YM 155548766 EC50 = 1800 nM T66237 CP9TR0 10324985 Ki > 10000 nM T66237 D00NIT 9810140 Ki = 1.19 nM T66237 D00SGZ 9917025 Ki = 381 nM T66237 D01WHI 135413562 Ki = 0.67 nM T66237 D09RIE 44419028 Ki = 750 nM T66237 D0K5NV 44428109 Ki > 1000 nM T66237 D0L0RP 44428107 Ki > 1000 nM T66237 D0NC8V 6918854 Ki = 630.96 nM T66237 D0Q0OR 10461270 Ki > 1000 nM T66237 D0R7QC 44419039 Ki = 131 nM T66237 D0T4ML 5311202 Ki = 28000 nM T66237 D0W3IQ 44419025 Ki = 1.2 nM T66237 D0Y0SO 44419026 EC50 = 0.05 nM T66237 D0ZD0W 11366713 Ki = 1125 nM T22655 CZYM47 44287934 IC50 = 276000 nM T22655 CYW1J0 44318263 IC50 = 298000 nM T22655 C0X4WJ 44375633 IC50 = 219000 nM T22655 CB1I4O 44375924 IC50 > 500000 nM T22655 CD0X2A 44375925 IC50 = 126000 nM T33124 D07ACT 5479530 IC50 = 10000 nM T33124 D07MOX 439260 IC50 > 10000000 nM T33124 D0N0ES 938 IC50 = 1125000 nM T33124 D0X9RY 243 Ki = 2000 nM T33124 D01LAC 6437850 IC50 > 10000 nM T33124 CD5JX0 6097 IC50 > 100000 nM T33124 CFR5J9 6918 IC50 = 4400 nM T33124 CLE87P 7419 IC50 = 392000 nM T33124 CAZ4Q3 7436 IC50 > 1000000 nM T33124 CBHG51 9822 IC50 = 910 nM T33124 C18YBO 10009 IC50 > 10000000 nM T33124 CXD8L9 10700 IC50 = 7800 nM T33124 C5JS6C 11985 IC50 > 100000 nM T33124 CC4Q8S 12473 IC50 > 5000 nM T33124 C8S5IX 12476 IC50 = 3929000 nM T33124 C3MK6N 13401 IC50 = 2478000 nM T33124 CL70CJ 13650 Ki = 13 nM T33124 CG1LI5 14313 IC50 = 13140 nM T33124 C61YWO 16976 IC50 > 2500000 nM T33124 C1VBO0 18496 IC50 > 2500000 nM T33124 C03POM 28115 IC50 = 1150 nM T33124 CC2IU7 34037 IC50 > 10000000 nM T33124 CK4HU2 67658 IC50 = 1045000 nM T33124 CL89PK 72899 IC50 = 745 nM T33124 C9WSN7 72930 IC50 > 1000000 nM T33124 CU50OJ 73836 IC50 > 1000000 nM T33124 CA1EO9 74713 IC50 = 4600 nM T33124 CVI0R4 90269 IC50 > 100000 nM T33124 C1B3QA 94960 IC50 > 10000000 nM T33124 CS6Z8K 95048 IC50 = 720 nM T33124 CNOH14 97629 IC50 = 930 nM T33124 C2N7BJ 209069 IC50 = 220 nM T33124 CI98OR 210830 IC50 = 418 nM T33124 CDE95F 219248 IC50 = 10100 nM T33124 CXQ68R 225438 IC50 = 27000 nM T33124 C31RYP 234556 IC50 > 100000 nM T33124 C87CMX 235702 IC50 > 100000 nM T33124 CC24UA 278396 IC50 > 100000 nM T33124 CGOC06 279630 IC50 > 10000000 nM T33124 C2WQ9Y 305687 IC50 = 90 nM T33124 CI1KB2 319979 IC50 > 100000 nM T33124 C2ULI9 343030 IC50 > 5000 nM T33124 CFB6G2 349115 IC50 = 1300 nM T33124 CJR18X 351036 IC50 = 200 nM T33124 C2J1RE 351037 IC50 = 300 nM T33124 CU0EP6 351652 IC50 > 100000 nM T33124 CJ49VP 352208 IC50 = 253000 nM T33124 C0V8FN 354316 IC50 > 2500000 nM T33124 C49KEP 447315 IC50 > 10000000 nM T33124 CA92XL 458349 IC50 > 100000 nM T33124 C5K3ZJ 459531 IC50 > 5000000 nM T33124 CKXO12 568654 IC50 > 500000 nM T33124 CGZ01B 588192 IC50 > 100000 nM T33124 CK97ZC 637090 IC50 = 357000 nM T33124 CP58OT 637541 IC50 = 6269000 nM T33124 C0L9OX 735156 IC50 > 10000000 nM T33124 C79CFS 770980 Ki = 4590 nM T33124 COT5M0 773806 IC50 > 100000 nM T33124 CN5E4T 818159 IC50 = 4 nM T33124 CK19RN 818882 IC50 > 100000 nM T33124 CH0FY8 819049 IC50 = 36 nM T33124 CH7W9X 819050 IC50 > 100000 nM T33124 C10HYM 819556 IC50 > 100000 nM T33124 CV2OD0 820270 IC50 > 26200 nM T33124 CC6G4J 833670 IC50 = 199000 nM T33124 C6YKO9 2049051 IC50 = 21000 nM T33124 C0R1SD 2050103 IC50 > 10000000 nM T33124 CXL02M 2050132 IC50 > 100000 nM T33124 CRKD94 2062168 IC50 > 2500000 nM T33124 C9VNH4 2063443 IC50 = 900000 nM T33124 C0GJ3Y 2113906 IC50 = 7905000 nM T33124 CO1V8G 2512481 IC50 = 1104000 nM T33124 CJ70WI 2734324 IC50 > 100000 nM T33124 CU4Q0T 2769634 IC50 = 7300 nM T33124 C2J9ML 2781852 IC50 = 17.2 nM T33124 C9T1JS 2794584 IC50 = 1300 nM T33124 CPU87E 3264479 IC50 = 1200 nM T33124 C73BKE 3561548 IC50 = 38000 nM T33124 C51QOE 3686650 IC50 = 1832000 nM T33124 CC0LA2 4179726 IC50 > 10000000 nM T33124 C16EGI 4961254 Ki = 3.5 nM T33124 CW3T0B 5183334 IC50 > 100000 nM T33124 CU68IK 7141881 Ki = 31.7 nM T33124 CVSU04 9817917 IC50 > 100000 nM T33124 CN50HC 10261088 IC50 = 140 nM T33124 C7X8OB 10344711 IC50 > 100000 nM T33124 C5MV2C 10531257 IC50 > 100000 nM T33124 C9YA8W 10531300 IC50 = 50000 nM T33124 CRV54N 11171714 Ki = 1.7 nM T33124 COT47F 11299678 Ki = 7.2 nM T33124 CEK10J 11622394 IC50 = 269 nM T33124 C8WCD5 11804901 IC50 = 1400 nM T33124 CZ2H9W 12205754 IC50 = 600 nM T33124 C58UTM 12501973 IC50 = 200 nM T33124 C8GJ3Q 12527112 IC50 > 5000 nM T33124 CN43EO 12605957 IC50 = 360 nM T33124 C72TKZ 12703605 IC50 = 55000 nM T33124 CM34ZV 13271054 IC50 = 33 nM T33124 CY6CM5 13711789 IC50 > 100000 nM T33124 C39KXP 15187160 IC50 = 3260 nM T33124 CBC9U1 15219883 IC50 = 150 nM T33124 C1WTA4 15933663 IC50 > 5000 nM T33124 CPGJ74 16225169 IC50 = 1426 nM T33124 CX1V8D 18938079 IC50 > 100000 nM T33124 CJE9H3 18938081 IC50 = 8800 nM T33124 CJ92GZ 20317991 IC50 = 8 nM T33124 C7UE9X 20431233 IC50 = 155 nM T33124 C8XM6E 21194199 IC50 = 1340 nM T33124 CV96GA 21622350 IC50 = 16 nM T33124 CD4CO9 21625970 IC50 = 1130 nM T33124 CK0N1C 21626163 IC50 > 100000 nM T33124 COW47N 21661241 IC50 = 900 nM T33124 C5NC3Z 21931591 IC50 = 1440000 nM T33124 CXG78T 22556501 IC50 > 5000 nM T33124 CK36HZ 22556514 IC50 > 5000 nM T33124 C1E6MC 23354375 IC50 = 9 nM T33124 C40MNJ 23423218 IC50 = 343 nM T33124 CWP84K 24728218 IC50 = 120 nM T33124 CB0G4A 24815611 IC50 = 516 nM T33124 CMK53H 24815612 IC50 > 5000 nM T33124 CI35UR 24815613 IC50 = 4204 nM T33124 CSRP35 24972975 IC50 = 2750 nM T33124 C8IDU3 24978023 IC50 > 100000 nM T33124 CJ29DL 39733327 IC50 > 5000 nM T33124 C8TX1U 42281625 IC50 = 4000 nM T33124 CFYI84 42601491 IC50 > 30000 nM T33124 C8EK3R 42623200 IC50 = 2460 nM T33124 CJ4MD2 42623269 IC50 = 26130 nM T33124 CCAW14 42623272 IC50 = 74070 nM T33124 CV6X3I 44128604 IC50 = 3 nM T33124 C6UOJ1 44157408 IC50 = 4 nM T33124 CTZ25D 44157409 IC50 = 197 nM T33124 C53UPY 44157410 IC50 = 8 nM T33124 C9WI1U 44157412 IC50 = 32 nM T33124 C9XZV5 44157495 IC50 = 3 nM T33124 C67KDR 44157496 IC50 = 10 nM T33124 C0VG5Y 44157497 IC50 = 8 nM T33124 C15TSZ 44157498 IC50 = 38 nM T33124 C1KQA4 44157568 IC50 = 22600 nM T33124 CY3WA8 44157569 IC50 = 14400 nM T33124 CAS7T0 44157572 IC50 = 5 nM T33124 C3XUV4 44176138 IC50 = 100 nM T33124 CYO2V3 44176139 IC50 = 17300 nM T33124 CL6IU7 44576687 IC50 > 5000 nM T33124 C32UWQ 44576688 IC50 = 1153 nM T33124 CF20IT 44576689 IC50 > 5000 nM T33124 C60UWG 44576721 IC50 > 5000 nM T33124 CI1XM7 44576722 IC50 > 5000 nM T33124 CF46RK 44576723 IC50 > 5000 nM T33124 C9DRE2 44623061 Ki = 190 nM T33124 CB31ST 44726831 IC50 = 200 nM T33124 CC8U0N 45792205 IC50 = 347000 nM T33124 C1RGC0 49875138 IC50 > 100000 nM T33124 C4M2KG 59223400 IC50 = 20000 nM T33124 CI34QL 60143296 IC50 = 1.5 nM T33124 C0T4LE 71187181 IC50 = 3.9 nM T33124 CP0AZ1 71270044 IC50 = 1.4 nM T33124 CU2KV9 71270093 IC50 = 2.4 nM T33124 CQS64G 71270196 IC50 = 2.7 nM T33124 C1W2RE 71270198 IC50 = 3.8 nM T33124 CL6W3K 71270282 IC50 = 3.1 nM T33124 CI61AC 71270376 IC50 = 8.4 nM T33124 C7IU4W 71270397 IC50 = 2 nM T33124 C6XR9F 71270399 IC50 = 4.7 nM T33124 C4N5JH 71270479 IC50 = 4.9 nM T33124 CWV4I2 71270546 IC50 = 12 nM T33124 C0IS5L 71449458 IC50 = 20000 nM T33124 C8AZ1U 71449459 IC50 = 2000 nM T33124 C7XG8C 71449460 IC50 = 30000 nM T33124 CA6FM9 71449461 IC50 = 8000 nM T33124 C6SK0A 71449462 IC50 > 100000 nM T33124 C9YI1X 71451262 IC50 = 30000 nM T33124 CL2XW7 71451263 IC50 = 10000 nM T33124 CEQ5F1 71451264 IC50 = 50000 nM T33124 CMTJ62 71451276 IC50 = 3000 nM T33124 CACF59 71451277 IC50 = 40000 nM T33124 CPEM98 71453078 IC50 > 100000 nM T33124 CB8Y6P 71453079 IC50 = 30000 nM T33124 C8WE1K 71453080 IC50 = 9000 nM T33124 C38GXB 71454820 IC50 = 800 nM T33124 C38PBS 71454821 IC50 = 900 nM T33124 CNUJ38 71454822 IC50 = 70000 nM T33124 CL53DU 71456592 IC50 = 1000 nM T33124 C2YNK3 71456593 IC50 = 100 nM T33124 C3H6WR 71456594 IC50 = 20000 nM T33124 CG0X1K 71456595 IC50 = 4000 nM T33124 CMO34X 71456607 IC50 > 100000 nM T33124 CLXK57 71458455 IC50 = 100 nM T33124 CD7J0T 71458456 IC50 = 20000 nM T33124 C6QJ4A 71460302 IC50 = 70000 nM T33124 CBZ94K 71460303 IC50 = 80000 nM T33124 CUS05W 71460304 IC50 = 70 nM T33124 CU54RF 71460305 IC50 = 20000 nM T33124 C9LK8Q 71460306 IC50 = 80 nM T33124 CR30CZ 71462001 IC50 = 400 nM T33124 CCXS16 71505692 IC50 = 63 nM T33124 CVS4A1 71655533 IC50 = 13 nM T33124 CL03AI 71655534 IC50 = 120 nM T33124 C3TWJ4 71655535 IC50 = 300 nM T33124 C4KT0Z 71655536 IC50 = 670 nM T33124 CNT97G 71655604 IC50 = 2.2 nM T33124 CZ2Q4W 71655605 IC50 = 2.1 nM T33124 CP7SX0 71655670 IC50 = 13 nM T33124 CC04YH 71655735 IC50 = 10 nM T33124 CE34DT 71681571 IC50 = 500 nM T33124 COSM37 71681572 IC50 > 100000 nM T33124 C39ZSJ 71681730 IC50 = 800 nM T33124 C9CPV2 71681731 IC50 = 700 nM T33124 CZT49J 71681732 IC50 = 500 nM T33124 CL2EX8 71681733 IC50 = 3000 nM T33124 C7LA5I 71681734 IC50 = 900 nM T33124 CZ3SG0 71681735 IC50 = 800 nM T33124 C4OIY3 71681895 IC50 = 100 nM T33124 CA1QD2 71719322 IC50 > 1000000 nM T33124 CE9DN5 72793909 IC50 = 50 nM T33124 C0V8XQ 73295540 IC50 = 270 nM T33124 CKG17U 73295541 IC50 = 5100 nM T33124 CAS13P 73295701 IC50 = 40000 nM T33124 C0QM8G 73295702 IC50 = 1700 nM T33124 CR87BW 73295704 IC50 = 260 nM T33124 CA16QM 73295707 IC50 = 50 nM T33124 CR0OC5 73295872 IC50 = 80 nM T33124 C2FL4S 73295873 IC50 = 70 nM T33124 C1E7QX 73295874 IC50 = 90 nM T33124 CKQ3Z1 73295875 IC50 = 100 nM T33124 CPFB91 73295876 IC50 = 60 nM T33124 C5M3LR 73295877 IC50 = 40 nM T33124 CQT56C 73295878 IC50 = 80 nM T33124 CGD8X7 73295879 IC50 = 60 nM T33124 CQF14U 73295880 IC50 = 50 nM T33124 CXY98I 73296039 IC50 = 70 nM T33124 CC3OY6 73296040 IC50 = 120 nM T33124 C6JO4N 73296041 IC50 = 90 nM T33124 C9SP8Z 73296042 IC50 = 120 nM T33124 CGT0V3 73296043 IC50 = 160 nM T33124 CM49EJ 73296045 IC50 = 110 nM T33124 CDA1H9 73296046 IC50 = 220 nM T33124 CRWJ56 73296203 IC50 = 240 nM T33124 CO59BH 73296206 IC50 = 400 nM T33124 CJPM21 73296209 IC50 = 330 nM T33124 C42PEI 73296357 IC50 = 310 nM T33124 C9A4OJ 73296358 IC50 = 440 nM T33124 CUJ0M3 73296362 IC50 = 760 nM T33124 CRO37J 73296643 IC50 = 50 nM T33124 C28GVC 73296644 IC50 = 850 nM T33124 C5SY7R 73296645 IC50 = 470 nM T33124 CM67HU 90036033 IC50 = 2800 nM T33124 C0N6DR 90036293 IC50 = 100 nM T33124 C7BL0V 90036412 IC50 = 80 nM T33124 C3VZO0 90036575 IC50 = 100 nM T33124 CIV3X7 90036814 IC50 = 80 nM T33124 CRD5C3 110172411 IC50 > 100000 nM T33124 C9AGD1 119086959 IC50 = 230 nM T33124 C37OUM 119086960 IC50 = 210 nM T33124 CY7XA0 122189434 IC50 = 3300 nM T33124 CGC64V 122189435 IC50 = 80 nM T33124 C0GM6P 127048506 IC50 = 1380 nM T33124 CE48SG 127049189 IC50 = 340 nM T33124 C84UJE 130302628 IC50 > 10000 nM T33124 C6EO4Y 132091077 IC50 = 1300 nM T33124 CKG6Z5 135418577 IC50 > 5000000 nM T33124 CJN8Y5 135610212 IC50 > 500000 nM T33124 CN2Z8I 135894470 IC50 = 128 nM T33124 CZB3C9 135894471 IC50 = 784 nM T33124 C1QOJ9 135930270 IC50 > 50000 nM T33124 CJN0O2 135976840 IC50 > 5000 nM T33124 CV6TY5 137006778 IC50 = 60 nM T33124 CO25FI 137175021 IC50 = 30 nM T33124 CT16VM 137175066 IC50 = 30 nM T33124 CP7F4O 137175067 IC50 = 600 nM T33124 CWYD74 137175089 IC50 = 40000 nM T33124 CZ2R4V 137175100 IC50 = 100 nM T33124 CN02WV 137175101 IC50 = 90 nM T33124 C6IL7F 137175103 IC50 = 300 nM T33124 CEK6Q4 137175104 IC50 = 50 nM T33124 CL64XB 137175105 IC50 = 50 nM T33124 C20YPI 137175123 IC50 = 700 nM T33124 CAB72Q 137175141 IC50 = 70 nM T33124 CND13F 137175185 IC50 = 4000 nM T33124 CC2XQ7 137175265 IC50 = 200 nM T33124 CRMU97 137175266 IC50 = 60 nM T33124 C9P4YE 137459864 IC50 = 3981.07 nM T33124 CE9G2I 145967877 IC50 = 390 nM T33124 C8AO1L 145969548 IC50 = 490 nM T33124 CNG10S 145970871 IC50 = 5200 nM T33124 C8B6GK 145971079 IC50 = 6700 nM T33124 C1I6NU 145971095 IC50 = 8800 nM T33124 C93VJH 145991239 IC50 = 39000 nM T33124 CCN0P3 155545992 IC50 = 316.23 nM T33124 CM5YS3 155551104 Ki = 1000000 nM T33124 CA35OS 155560404 IC50 = 316.23 nM T33124 D05FMD 9447 IC50 = 3671000 nM T33124 D08JNG 867 IC50 > 10000000 nM T33124 D0ET2F 256208 IC50 = 1499000 nM T33124 D0F3CO 3840 IC50 = 2000 nM T33124 D0X0ER 344135 IC50 = 7870 nM T70490 D05UFG 10184653 IC50 > 10000 nM T70490 D0O8GK 71496458 IC50 = 32900 nM T70490 D0J6AU 10152654 IC50 > 10 nM T70490 D0YB3W 156414 IC50 = 2700 nM T70490 D0HM5J 118253852 IC50 = 3.981 nM T70490 C0XQP7 6917747 IC50 > 100000 nM T70490 CD54AH 6993099 Ki = 6200000 nM T70490 CBS6P7 8022437 IC50 = 11000 nM T70490 CXE30M 11334066 IC50 = 822 nM T70490 C9D6XI 11736400 IC50 = 172 nM T70490 C8D7BS 11771234 IC50 = 13 nM T70490 CN4IM8 11817961 IC50 = 96 nM T70490 C31MCN 13186896 IC50 > 100000 nM T70490 C6XPN4 16664855 IC50 = 18 nM T70490 CZ8DI1 23643986 IC50 = 70 nM T70490 CZPF48 23648277 IC50 > 10000 nM T70490 C31XJH 23648296 IC50 > 10000 nM T70490 CN0VA7 24822701 IC50 = 14 nM T70490 CQU38W 24900755 IC50 = 1727 nM T70490 C2S8VB 24901099 IC50 = 29 nM T70490 CIN28B 24901100 IC50 = 403 nM T70490 CD2EH0 24901101 IC50 = 191 nM T70490 CS7B3F 24901102 IC50 > 10000 nM T70490 CGI0U2 25023791 Ki = 10000 nM T70490 C3C8YJ 25174148 IC50 = 1.995 nM T70490 C5M1BT 25195691 IC50 = 158.49 nM T70490 CJ63ZU 42641779 IC50 = 158.49 nM T70490 CZM36T 42641892 IC50 = 39.81 nM T70490 CRYH80 42642459 IC50 = 1 nM T70490 C25ELB 44143088 IC50 = 34.67 nM T70490 CL0M7R 44143089 IC50 = 6918.31 nM T70490 C9QDC0 44143091 IC50 = 588.84 nM T70490 CDVC01 44268431 Ki = 180000 nM T70490 CK8EB3 44268436 Ki = 220000 nM T70490 CAPM01 44413250 IC50 = 6296 nM T70490 C7EKG5 44413251 IC50 = 9637 nM T70490 CCG5S4 44413390 IC50 = 137 nM T70490 CS6X7V 44426055 IC50 = 606 nM T70490 C8IB2W 44426056 IC50 > 100000 nM T70490 C9TFJ8 44464926 IC50 = 10 nM T70490 CYO0T1 44465454 IC50 = 7.943 nM T70490 CE83YL 44465721 IC50 < 0.3981 nM T70490 C6OC4Z 44607530 IC50 = 2100 nM T70490 CWMN69 46882864 IC50 = 2545 nM T70490 CQT8N7 46882865 IC50 = 271 nM T70490 CP47RN 46882866 IC50 = 8.2 nM T70490 C75BEM 46882867 IC50 = 1.7 nM T70490 C2PKZ9 46882868 IC50 = 880 nM T70490 CLV43E 46882869 IC50 = 336 nM T70490 CY2MQ1 46882870 IC50 = 2193 nM T70490 C0M4PL 46882914 IC50 = 250 nM T70490 CC94XY 46882915 IC50 = 67 nM T70490 C5X4SE 46883366 IC50 = 1230 nM T70490 CO5PD8 46883367 IC50 = 29 nM T70490 C9J4KG 46883368 IC50 = 5.8 nM T70490 CNA0W6 46883391 IC50 = 200 nM T70490 CW1RB0 46883392 IC50 = 630 nM T70490 CEB8W0 46883393 IC50 = 1580 nM T70490 CXST57 46883394 IC50 = 330 nM T70490 C7I6OU 46883395 IC50 = 17 nM T70490 CA6BD2 46883396 IC50 = 215 nM T70490 CP0V2B 46883425 IC50 = 3.8 nM T70490 C4WNV1 46883426 IC50 = 5.1 nM T70490 C16KZC 46883427 IC50 = 0.9 nM T70490 CQX57K 46883428 IC50 = 11 nM T70490 CQN34G 46883429 IC50 = 1 nM T70490 C0ZH2Y 46883430 IC50 = 0.7 nM T70490 C56QYZ 46883464 IC50 = 0.3 nM T70490 CEZ54V 46883465 IC50 > 3000 nM T70490 C2QM7R 46883466 IC50 = 12 nM T70490 CE80HK 46883467 IC50 = 1419 nM T70490 CHA61U 46883468 IC50 = 1832 nM T70490 CI2FX9 46883469 IC50 = 63 nM T70490 CM4O6Q 46883470 IC50 = 17 nM T70490 C68XTP 46883502 IC50 = 2502 nM T70490 CYN9C1 46883503 IC50 = 1081 nM T70490 C6FI5J 46883504 IC50 = 495 nM T70490 C7IOX5 46883505 IC50 = 133 nM T70490 C3I0FZ 46883506 IC50 > 10000 nM T70490 CUI91D 46905615 IC50 > 220 nM T70490 C9PAR7 46905616 IC50 = 790 nM T70490 CAFW31 49783666 IC50 = 0.7943 nM T70490 CN0B1V 49783830 IC50 = 0.2512 nM T70490 CNI1P6 49783903 IC50 = 0.7943 nM T70490 CGF65B 49783985 IC50 = 5.012 nM T70490 CI59MV 49797572 IC50 > 30000 nM T70490 C96CKU 49797573 IC50 = 14 nM T70490 C56OCA 53317528 IC50 = 1995.26 nM T70490 C7I9AO 53317529 IC50 > 25118.86 nM T70490 CM60RJ 53317530 IC50 > 25118.86 nM T70490 C5A6IH 53317737 IC50 = 1000 nM T70490 C6FEH9 53318816 IC50 > 25118.86 nM T70490 CJAX07 53318817 IC50 = 15848.93 nM T70490 CG5AP6 53318818 IC50 = 125.89 nM T70490 C0QV5D 53322753 IC50 = 2511.89 nM T70490 CHB96K 53324300 IC50 = 316.23 nM T70490 CR1L4Y 53325394 IC50 > 25118.86 nM T70490 CVU0J1 53326656 IC50 = 316.23 nM T70490 CFC91M 54769914 IC50 = 2.512 nM T70490 CF3XA9 57999656 IC50 = 158.49 nM T70490 CLA3R9 66645269 IC50 = 1.995 nM T70490 C62SML 90655967 IC50 = 25.12 nM T70490 CJ7LT3 90655968 IC50 = 12.59 nM T70490 CB61WC 90655969 IC50 = 3.981 nM T70490 CK5X2M 91826235 IC50 = 2.512 nM T70490 CGFK60 101201806 IC50 = 51 nM T70490 C8E4WS 102323332 IC50 = 1 nM T70490 CI9L7M 118253811 IC50 = 15.85 nM T70490 C3BAX2 118253818 IC50 = 6309.57 nM T70490 CL5C4K 118253824 IC50 = 7.943 nM T70490 CO53KU 118253851 IC50 = 12.59 nM T70490 C7YFQ0 118253855 IC50 = 15.85 nM T70490 CCH97D 118253857 IC50 = 31.62 nM T70490 C24IWU 118253859 IC50 = 39.81 nM T70490 CM63RL 118253870 IC50 = 12.59 nM T70490 CPBD92 118253877 IC50 = 63.1 nM T70490 CCG7Y6 118253883 IC50 = 5.012 nM T70490 CA72QZ 118253888 IC50 = 6.31 nM T70490 C63BSU 118260121 IC50 = 63.1 nM T70490 CTE34I 118720232 IC50 > 100000 nM T70490 CSD62B 118720233 IC50 > 100000 nM T70490 C9WF7Q 118720234 IC50 = 66000 nM T70490 C76HIO 118720235 IC50 = 18000 nM T70490 CAT1R6 118720236 IC50 > 100000 nM T70490 CGAF42 118720237 IC50 > 100000 nM T70490 CJ28KZ 118720238 IC50 > 100000 nM T70490 CPH2V9 118720239 IC50 > 100000 nM T70490 CQA83T 134131850 IC50 = 199.53 nM T70490 C7UNJ4 134132070 IC50 > 10000 nM T70490 CVAH73 134134180 IC50 = 398.11 nM T70490 CD6H8U 134134303 IC50 > 10000 nM T70490 C1RWN0 134134473 IC50 = 1000 nM T70490 CB93JM 134134976 IC50 = 1258.93 nM T70490 CZL0G9 134138927 IC50 = 158.49 nM T70490 C1W7EY 134140481 IC50 = 501.19 nM T70490 C6B5RW 134141023 IC50 = 39.81 nM T70490 CO9E0J 134145021 IC50 = 25.12 nM T70490 CI6FZ3 134147640 IC50 > 10000 nM T70490 C3DCQ9 134148503 IC50 = 501.19 nM T70490 C9OLA1 134148630 IC50 > 10000 nM T70490 C8SH1L 134154191 IC50 = 31.62 nM T70490 CTQY96 136117851 IC50 = 450 nM T70490 C3YHN7 146685679 IC50 = 32.3 nM T70490 C7TI5V 147202641 IC50 > 10000 nM T70490 CIK2C0 147243243 IC50 = 2150 nM T70490 C0JL2F 147323358 IC50 = 4 nM T70490 CUAY08 148018738 IC50 = 12.3 nM T70490 CH0NR2 148192765 IC50 > 10000 nM T70490 CT25HK 148412521 IC50 = 2.7 nM T70490 CWD7A1 148809433 IC50 = 2051 nM T70490 C0SW6H 148967294 IC50 = 6.5 nM T70490 CQK39B 149491764 IC50 = 3.9 nM T70490 C1ZX5D 149494192 IC50 = 1.9 nM T70490 CCU10W 149589615 IC50 = 505 nM T70490 CN6G2P 149839762 IC50 = 307.1 nM T70490 C4GCQ2 149933110 IC50 > 10000 nM T70490 C08LSG 150088178 IC50 = 154 nM T70490 CJZ3L2 150363449 IC50 = 783 nM T70490 C26MXO 150396261 IC50 = 1520 nM T70490 C3IPK7 150631495 IC50 = 271 nM T70490 CJ6A9B 150967523 IC50 = 221 nM T70490 CFXO59 151118910 IC50 = 499 nM T70490 CO6QT1 151217326 IC50 = 2.8 nM T70490 CMX4K7 151268438 IC50 = 4.9 nM T70490 CG6CN4 151286177 IC50 = 1605 nM T70490 C7RZO2 151821865 IC50 = 785 nM T70490 CDL4W5 151971947 IC50 = 1 nM T70490 CYN8L2 152157601 IC50 = 537 nM T70490 CJ2KV5 152225461 IC50 = 135.4 nM T70490 CKZ6H9 152242423 IC50 = 21.3 nM T70490 COE18M 152296790 IC50 = 175 nM T70490 CR0EQ1 152335936 IC50 = 835 nM T70490 C0IO7L 152457310 IC50 = 391.5 nM T70490 CZG2D5 152823047 IC50 = 2.3 nM T70490 CPF6I5 155518852 IC50 = 483 nM T70490 CQF3W2 155521718 IC50 > 10000 nM T70490 CXC8Q2 155522247 IC50 = 79.43 nM T70490 CMJO87 155528739 IC50 = 630.96 nM T70490 CY2HC7 155538869 IC50 = 6.31 nM T70490 CVGT48 155543410 IC50 = 0.3981 nM T70490 C2J5NY 155559747 IC50 = 50.12 nM T70490 CU67FS 155561515 IC50 = 50.12 nM T70490 CA8WQ7 155565392 IC50 = 1.585 nM T70490 D00FGA 73737 IC50 > 25118.86 nM T70490 D09FGQ 123985 IC50 = 770 nM T70490 D0IV5D 11241135 Ki = 2700 nM T70490 D0L9VP 5287864 IC50 = 2600 nM T70490 D0U4TA 44413276 IC50 = 4787 nM T70490 D0Y5IQ 44255320 IC50 = 10000 nM T73694 D09KTS 24821094 IC50 = 18 nM T73694 D0E6XR 3062316 IC50 = 5.3 nM T73694 D03HUX 49792852 IC50 > 10000 nM T73694 D0E3TC 44259 IC50 = 247 nM T73694 D0G5XV 135565884 IC50 = 33 nM T73694 D0O0LS 25141092 IC50 = 195 nM T73694 D03BNU 59604787 IC50 > 10000 nM T73694 D0T3ME 156422 IC50 > 30000 nM T73694 CJ2SQ9 683690 IC50 > 10000 nM T73694 C3PL7H 961174 IC50 > 10000 nM T73694 C9U7NK 1128774 IC50 = 520 nM T73694 C9RQC1 1521040 IC50 = 5600 nM T73694 CVZ37I 2351464 IC50 = 1900 nM T73694 CLH1T0 4376831 IC50 > 10000 nM T73694 CM5VN6 4600415 IC50 = 120 nM T73694 C9YK6Q 4603900 IC50 > 10000 nM T73694 C3LN1Y 5240683 IC50 = 5830 nM T73694 CY2UO9 5329275 IC50 = 2320 nM T73694 C9JT4S 11847343 IC50 > 10000 nM T73694 CA3I4T 24753787 IC50 > 50000 nM T73694 C7YG1N 24759534 IC50 = 1700 nM T73694 CQN3Z7 24825710 IC50 = 310 nM T73694 C1RP0I 25094211 IC50 = 500 nM T73694 CGT1W6 25144294 IC50 = 13 nM T73694 CNG96H 25210579 IC50 > 10000 nM T73694 C3VRO9 44557921 IC50 > 10000 nM T73694 CU3RF1 45139989 IC50 > 10000 nM T73694 CQGZ06 45139991 IC50 > 10000 nM T73694 CYT37A 46232443 IC50 > 50000 nM T73694 C48ZVW 46232555 IC50 = 32000 nM T73694 CS9B1U 46232556 IC50 > 50000 nM T73694 C7ON5A 46233287 IC50 > 10000 nM T73694 CF91RS 49843531 IC50 > 10000 nM T73694 CV8X0G 50924500 IC50 = 5.65 nM T73694 C2Y6QS 50938552 IC50 > 10000 nM T73694 C9NYP4 51036677 IC50 > 10000 nM T73694 C4WRY3 51037112 IC50 > 10000 nM T73694 CRI28Z 51037948 IC50 > 10000 nM T73694 C8NA4L 53384644 IC50 > 30000 nM T73694 CXA92G 53484170 IC50 = 10 nM T73694 C7UK2N 53484181 IC50 = 7 nM T73694 CKD9H6 53484182 IC50 = 9 nM T73694 CH05EO 53484183 IC50 = 7 nM T73694 CAR45T 53484184 IC50 = 6 nM T73694 CE1ZK6 54759168 IC50 > 10000 nM T73694 COM26L 56658690 IC50 = 177 nM T73694 C8DWL7 56658691 IC50 = 477 nM T73694 C8GJ9S 56658692 IC50 = 10 nM T73694 CK3A4Z 56658700 IC50 = 19 nM T73694 CRE75Z 56658839 IC50 = 75 nM T73694 C0JK4L 56658840 IC50 = 495 nM T73694 C1JD6Z 56658841 IC50 = 15 nM T73694 C98WRJ 56658842 IC50 = 38 nM T73694 C9R5IT 56658843 IC50 = 8 nM T73694 C2Z9YO 56662177 IC50 = 42 nM T73694 CR50XZ 56662178 IC50 = 11 nM T73694 C8NGC7 56662179 IC50 = 14 nM T73694 C3H0VQ 56662180 IC50 = 13 nM T73694 CWM35E 56662181 IC50 = 64 nM T73694 CB0VE5 56662182 IC50 = 38 nM T73694 CVBK03 56662332 IC50 = 16 nM T73694 CFW3I1 56665626 IC50 > 10000 nM T73694 C5XW3F 56665627 IC50 > 10000 nM T73694 CO96CB 56665628 IC50 = 51 nM T73694 CO51RL 56665629 IC50 = 97 nM T73694 CEI39Q 56665634 IC50 = 5 nM T73694 CG5K2Q 56665635 IC50 = 17 nM T73694 CVEM27 56665636 IC50 = 63 nM T73694 CDT3K4 56665637 IC50 = 156 nM T73694 CCD3U6 56665765 IC50 = 32 nM T73694 CVBF37 56665766 IC50 = 379 nM T73694 C9OB2T 56665767 IC50 = 72 nM T73694 CXO10E 56669082 IC50 = 1524 nM T73694 CF7K6A 56669083 IC50 = 319 nM T73694 CLE86K 56669084 IC50 = 391 nM T73694 C7JCP2 56669085 IC50 = 104 nM T73694 C9ZTL3 56669088 IC50 = 70 nM T73694 CC8F0R 56669218 IC50 = 254 nM T73694 CXW95K 56669219 IC50 = 23 nM T73694 C2GB4J 56672541 IC50 = 256 nM T73694 C5VS7B 56672542 IC50 = 12 nM T73694 C8R9TW 56672548 IC50 = 47 nM T73694 C0ROQ7 56672549 IC50 = 124 nM T73694 CI6K1R 56672550 IC50 = 156 nM T73694 CC5NQ4 56672551 IC50 = 7 nM T73694 CY0PA7 56672679 IC50 = 35 nM T73694 CP6AE8 56672680 IC50 = 68 nM T73694 C0GUO4 56672681 IC50 = 34 nM T73694 C25WIJ 56675923 IC50 = 355 nM T73694 CJA2N4 56675924 IC50 = 6 nM T73694 CWY32H 56676047 IC50 = 22 nM T73694 CR0CJ1 56679234 IC50 > 10000 nM T73694 CHB5T1 56679235 IC50 = 2643 nM T73694 CF3TD1 56679236 IC50 = 799 nM T73694 CF5YP1 56679374 IC50 = 10 nM T73694 C8QR1J 56679375 IC50 = 93 nM T73694 CLKP65 56682548 IC50 = 10 nM T73694 CW2YZ7 56682555 IC50 = 19 nM T73694 C1JWN7 56682556 IC50 = 7 nM T73694 CS9YF2 56682557 IC50 = 52 nM T73694 COM56E 56682674 IC50 = 109 nM T73694 C03OTV 56682675 IC50 = 3 nM T73694 CG2A4M 56682676 IC50 = 137 nM T73694 CPHX64 57325478 IC50 > 50000 nM T73694 CQ9BW4 57325479 IC50 > 50000 nM T73694 CVK0G4 58056356 IC50 > 50000 nM T73694 CXJ63M 59603829 IC50 > 100000 nM T73694 CQEU96 59603842 IC50 = 390 nM T73694 CV63UL 67240318 IC50 > 10000 nM T73694 C5DGR9 69036886 IC50 = 10000 nM T73694 COU73Y 71226944 IC50 = 60 nM T73694 C40JOZ 71235465 IC50 = 77 nM T73694 CCN01X 71547862 IC50 > 10000 nM T73694 CP5C7Y 76311266 IC50 = 5.7 nM T73694 C4GD6X 76311267 IC50 = 4.8 nM T73694 C9XZ0C 76311268 IC50 > 1000000 nM T73694 C29NOJ 76314857 IC50 = 9.2 nM T73694 CQT97B 76314858 IC50 > 1000000 nM T73694 CIV6B3 76318467 IC50 = 410 nM T73694 C4PRL2 76318468 IC50 = 55 nM T73694 CFTP19 76318469 IC50 = 26 nM T73694 CQ01AS 76318470 IC50 = 186 nM T73694 CV0C8D 76322137 IC50 = 13 nM T73694 C3QMZ9 76325759 IC50 = 21 nM T73694 C65WFX 76325760 IC50 = 4.7 nM T73694 CWG41I 76325761 IC50 = 479 nM T73694 CV9H0X 76329340 IC50 = 13 nM T73694 CJKG82 76329341 IC50 = 4.1 nM T73694 CCP9B2 76329342 IC50 > 1000000 nM T73694 CX8Q2U 76329343 IC50 > 1000000 nM T73694 CY1N5G 76332981 IC50 > 1000000 nM T73694 CXBD37 76332982 IC50 = 7.6 nM T73694 CJ2T9E 76332983 IC50 = 3.2 nM T73694 CL0UZ2 76332984 IC50 > 1000000 nM T73694 C9I2BO 76335834 IC50 = 5300 nM T73694 CPG3A5 86302574 IC50 > 30000 nM T73694 C1HW4B 89735655 IC50 > 100000 nM T73694 CY0UC4 90645194 IC50 > 10000 nM T73694 CTE8D6 90654489 IC50 = 4.41 nM T73694 C7OT8X 90654490 IC50 = 40.7 nM T73694 CTL9V6 90654491 IC50 = 43.5 nM T73694 CP8XL9 90654492 IC50 = 53.4 nM T73694 C34VGE 90654493 IC50 = 59.4 nM T73694 CA1KD0 90654494 IC50 = 64.5 nM T73694 C8T5IA 90654495 IC50 = 69.5 nM T73694 C5M3YN 90654496 IC50 = 75.6 nM T73694 CW4MA2 90654497 IC50 = 154 nM T73694 CYW6C8 90654498 IC50 = 155 nM T73694 C0IE3P 90654499 IC50 = 190 nM T73694 CY7BI2 118706214 IC50 > 10000 nM T73694 C1KQ4A 118714325 IC50 > 10000 nM T73694 C8VP5J 118714336 IC50 > 10000 nM T73694 CF80US 135406083 IC50 = 1680 nM T73694 CZFA70 135611366 IC50 = 933 nM T73694 CHA4N2 136013680 IC50 > 10 nM T73694 CSON28 136044162 IC50 = 58100 nM T73694 CQ8GK2 136044163 IC50 = 2540 nM T73694 C1XYU3 136044164 IC50 = 130 nM T73694 CIOP32 136044165 IC50 = 1290 nM T73694 C5PF2R 136044166 IC50 = 11750 nM T73694 CPMJ51 136044167 IC50 = 3900 nM T73694 CKQM03 136044169 IC50 = 1350 nM T73694 CV78CR 136044170 IC50 > 10000 nM T73694 C78HUT 136044171 IC50 = 1990 nM T73694 C1YUD0 136219394 IC50 > 10 nM T73694 CIU8W3 136254389 IC50 > 10 nM T73694 C2QV3C 136998781 IC50 = 360 nM T73694 C0NM9J 136998782 IC50 = 1300 nM T73694 CFE05J 136998783 IC50 = 200 nM T73694 CV53AZ 136998784 IC50 = 270 nM T73694 CXC69T 137321158 IC50 = 111 nM T73694 CZOD53 137633880 IC50 = 350 nM T73694 C7BJY5 137636807 IC50 = 113 nM T73694 CO89DX 137649100 IC50 = 48 nM T73694 CINE03 137652514 IC50 = 173 nM T73694 C28QUP 137652864 IC50 = 220.2 nM T73694 CF27EG 155511610 IC50 = 956 nM T73694 C0AN1O 155512752 IC50 = 626 nM T73694 C2MD1Q 155513187 IC50 > 10000 nM T73694 D08HFG 24809764 IC50 > 10000 nM T73694 D09HVH 135566652 IC50 > 10 nM T73694 D09PTP 57325421 IC50 = 73 nM T73694 D0IZ8M 56675928 IC50 = 2 nM T73694 D0N4LR 53469448 IC50 = 412 nM T39698 D03BNU 59604787 IC50 > 10000 nM T39698 CV63UL 67240318 IC50 > 10000 nM T39698 C2MD1Q 155513187 IC50 > 10000 nM T39698 D0C1DQ 6490494 IC50 = 7280 nM T84634 D0N0RU 82146 IC50 = 13500 nM T84634 D08UGX 60652 IC50 = 540 nM T84634 D0AA6Z 9799888 IC50 = 5.1 nM T84634 D09YUQ 127019 IC50 = 7800 nM T84634 C9LCD8 3823 IC50 = 12000 nM T84634 C3NS4E 132775 IC50 = 1300 nM T84634 CXQ40P 5862285 IC50 = 20000 nM T84634 C62RUG 9821132 IC50 = 10 nM T84634 CO39KV 9838239 IC50 = 39000 nM T84634 CI6V2U 9870337 IC50 = 10 nM T84634 C9VEF0 9949645 IC50 > 25000 nM T84634 CDLS47 10021552 IC50 = 4700 nM T84634 CKPQ58 11154980 IC50 = 25 nM T84634 C4GO0T 11231328 IC50 = 20000 nM T84634 CVO5A3 11235737 IC50 = 3.5 nM T84634 C3TF0M 11236452 IC50 = 24 nM T84634 CB7YS1 11315814 IC50 = 1.3 nM T84634 C9W0QH 11373414 IC50 = 5.2 nM T84634 C5VC8J 11406760 IC50 = 47 nM T84634 C5KMI6 11427427 IC50 = 10000 nM T84634 C0PWX2 11441615 IC50 = 35 nM T84634 C2KXN4 11475327 IC50 = 54 nM T84634 CYH36X 11493096 IC50 = 25000 nM T84634 C39PJT 11495962 IC50 = 16 nM T84634 CS0J3Q 11499978 IC50 = 25000 nM T84634 CEV5B3 11501485 IC50 = 73 nM T84634 CRV87M 11510548 IC50 = 7 nM T84634 CW51VQ 11523005 IC50 = 9000 nM T84634 C3QH2T 11558212 IC50 = 7000 nM T84634 CG24YV 11565407 IC50 = 5000 nM T84634 CVO62B 11582136 IC50 = 50000 nM T84634 CKW1Z2 11582790 IC50 = 77 nM T84634 C2H7WN 11590652 IC50 = 34 nM T84634 C1ZO5J 11595033 IC50 = 50000 nM T84634 C7S3EY 11618244 IC50 = 50000 nM T84634 C1MS3D 11623142 IC50 = 20000 nM T84634 C7OF9S 11633939 IC50 = 100 nM T84634 CMF5L2 11645016 IC50 = 50000 nM T84634 CFLM39 11652817 IC50 = 20000 nM T84634 CX4A9P 11659007 IC50 = 9000 nM T84634 CE4KR7 11688435 IC50 = 20000 nM T84634 C9UL1Q 11688471 IC50 = 10000 nM T84634 CM8R9J 11690073 IC50 = 6 nM T84634 CL5S9K 11719046 IC50 = 4.2 nM T84634 CI1P7M 11750760 IC50 = 12 nM T84634 C6TS4D 11773824 IC50 = 46 nM T84634 C98WNZ 14795724 IC50 = 2800 nM T84634 CYZ8E7 15950260 IC50 = 4500 nM T84634 CS8QM5 16039690 IC50 = 900 nM T84634 C1RV2O 23442837 IC50 = 4000 nM T84634 CVG5R8 25141344 IC50 = 500 nM T84634 CAWG69 44390123 IC50 = 37 nM T84634 CDZH20 44390134 IC50 = 50 nM T84634 CIOY83 44390142 IC50 = 14.4 nM T84634 CDQ90V 44390161 IC50 = 19 nM T84634 CS5NY3 44390206 IC50 = 48 nM T84634 CT5DF2 44390231 IC50 = 8 nM T84634 CH1QM4 44390265 IC50 = 335 nM T84634 C8V7OA 44410763 IC50 = 125 nM T84634 C0SXD3 44410799 IC50 = 20 nM T84634 C3PYC4 44410807 IC50 = 37 nM T84634 CB6H1M 44410808 IC50 = 34.7 nM T84634 CXM15V 44410812 IC50 = 583 nM T84634 CM4Z0T 44410814 IC50 = 1.6 nM T84634 CR4HX5 44410840 IC50 = 7.3 nM T84634 C73OZJ 44410841 IC50 = 11.2 nM T84634 C3NED2 44410860 IC50 = 46.7 nM T84634 C1EA6U 44410861 IC50 = 9 nM T84634 CU5E6C 44410862 IC50 = 5 nM T84634 CR5Y0N 44410871 IC50 = 3 nM T84634 C8IV5K 44410881 IC50 = 40 nM T84634 CBS59K 44411032 IC50 = 60 nM T84634 CRU1S5 44411036 IC50 = 34 nM T84634 C9J8MS 44411109 IC50 = 1.4 nM T84634 CFA64M 44411110 IC50 = 403 nM T84634 CD53XR 44411116 IC50 = 26 nM T84634 CINM87 44421467 IC50 = 800 nM T84634 CS9W1C 44421568 IC50 = 43000 nM T84634 CX2D7Y 44421596 IC50 = 4 nM T84634 C3J4IK 44445028 IC50 = 2200 nM T84634 CER28I 44547030 IC50 = 140 nM T84634 CCP59J 44547031 IC50 = 50 nM T84634 CYA5V4 44547032 IC50 > 1000 nM T84634 CECD12 44547033 IC50 = 0.3 nM T84634 C8V0RF 44547182 IC50 = 300 nM T84634 CGHQ08 44547183 IC50 = 0.35 nM T84634 C4OH1Q 44547184 IC50 = 290 nM T84634 C6K0OT 44547185 IC50 = 200 nM T84634 CZT18X 44547186 IC50 = 120 nM T84634 CYVB48 44547187 IC50 = 50 nM T84634 C0NPS7 44547331 IC50 = 12 nM T84634 C1O9MY 44547332 IC50 = 75 nM T84634 CB9NJ4 44547333 IC50 = 8 nM T84634 C02MSK 44547334 IC50 = 3 nM T84634 C8K2VD 44547335 IC50 = 40 nM T84634 CY6RM7 44547336 IC50 = 6 nM T84634 C4YST2 44547474 IC50 = 125 nM T84634 CJS5M2 44547475 IC50 = 400 nM T84634 CQZM23 44547476 IC50 = 140 nM T84634 CZ3YF8 44569168 IC50 > 50000 nM T84634 CTU37D 44569169 IC50 = 5000 nM T84634 COQ93E 44569170 IC50 = 35000 nM T84634 CQ4R9W 44569193 IC50 = 5000 nM T84634 CCW9S3 44569194 IC50 = 15000 nM T84634 CQ9V3E 44569195 IC50 = 1000 nM T84634 C5L3BW 44569196 IC50 = 2500 nM T84634 CHR3B7 44569222 IC50 = 1500 nM T84634 CQ6L0D 44569244 IC50 = 7000 nM T84634 C4X7SL 52951448 IC50 = 10 nM T84634 CG9N3R 52951561 IC50 = 8 nM T84634 CXKQ83 52951562 IC50 = 250 nM T84634 CWT95A 52951563 IC50 = 10 nM T84634 C2LB4Z 52951564 IC50 = 100 nM T84634 CY61IQ 52951683 IC50 = 40 nM T84634 CTH5P9 52951684 IC50 = 26 nM T84634 C2QIY0 52951823 IC50 > 1000 nM T84634 C2XV8F 54581365 IC50 = 3 nM T84634 C9PC5O 54758311 IC50 > 1000 nM T84634 C1MT9P 54758312 IC50 = 350 nM T84634 CK6E8U 71450543 IC50 > 1000 nM T84634 C0J7GV 71452887 IC50 = 450 nM T84634 CME8C6 71452888 IC50 = 9.4 nM T84634 C9RQK0 71452893 IC50 = 90 nM T84634 C6M4HK 71454655 IC50 = 100 nM T84634 C5F6TC 71454656 IC50 = 45 nM T84634 C7KL6A 71454657 IC50 = 5.7 nM T84634 CDJ7S2 71456381 IC50 = 16 nM T84634 CF8SN4 71457688 IC50 = 95 nM T84634 CO6VP9 71457689 IC50 = 200 nM T84634 C3C8IE 71458230 IC50 > 10 nM T84634 C7H3KI 71459597 IC50 = 85 nM T84634 CT83JM 71459598 IC50 = 250 nM T84634 C8WRL9 71459599 IC50 = 1000 nM T84634 C5RW7V 71460077 IC50 = 250 nM T84634 C1F5PV 71460078 IC50 = 700 nM T84634 CP4JI3 71460079 IC50 > 1000 nM T84634 C0PQ4J 71461338 IC50 = 1000 nM T84634 CH9E1A 71461802 IC50 = 14 nM T84634 CM4QL3 71461812 IC50 = 500 nM T84634 CH80VJ 71461813 IC50 = 6.7 nM T84634 CD81EJ 71463058 IC50 = 13 nM T84634 COJC78 71463059 IC50 > 1000 nM T84634 CEVW85 90659735 IC50 > 10000 nM T84634 CPW37E 117911702 IC50 > 5000 nM T84634 CH3L7C 117911715 IC50 > 5000 nM T84634 C87YKP 118727453 IC50 = 3040 nM T84634 C14EWO 118727454 IC50 = 3260 nM T84634 CYX1B9 118727455 IC50 = 2620 nM T84634 CU34VL 118727456 IC50 = 2810 nM T84634 CCI1P2 118727457 IC50 = 3020 nM T84634 CDV98T 118727458 IC50 = 5070 nM T84634 CSDL81 118727459 IC50 = 2830 nM T84634 CGQB23 118727460 IC50 = 3090 nM T84634 C05CPH 118727461 IC50 = 2730 nM T84634 C30IXV 118727462 IC50 = 4020 nM T84634 C2TV4J 118727463 IC50 = 3140 nM T84634 CUH6X7 118727464 IC50 = 2340 nM T84634 C89AOJ 118727465 IC50 = 3130 nM T84634 C9Y4FQ 118727466 IC50 = 5190 nM T84634 C06KVH 118727467 IC50 = 3350 nM T84634 C9YJ4H 118727468 IC50 = 3480 nM T84634 CMN01I 118727469 IC50 = 2070 nM T84634 C1PBO9 118727470 IC50 = 1360 nM T84634 C3X5GN 118727471 IC50 = 3220 nM T84634 C6G3NA 118727472 IC50 = 1870 nM T84634 CARH21 118727473 IC50 = 3210 nM T84634 CWI1Z8 121472067 IC50 = 270 nM T84634 CZP07X 121472068 IC50 = 10600 nM T84634 C4AD2S 121472069 IC50 > 5000 nM T84634 CT7YX5 121472072 IC50 = 240 nM T84634 CVX1Q8 121472075 IC50 = 340 nM T84634 CGK83X 121472076 IC50 = 1660 nM T84634 C9JBV4 121472081 IC50 > 5000 nM T84634 CJD30N 121472085 IC50 > 5000 nM T84634 CXAD12 121474361 IC50 = 110 nM T84634 C9JA6W 122190692 IC50 = 370 nM T84634 CCE2I8 122190693 IC50 = 650 nM T84634 CK2AJ7 122190694 IC50 = 790 nM T84634 CJQ2X5 122190695 IC50 = 540 nM T84634 C4SHV9 122190696 IC50 = 970 nM T84634 CCD9E8 122190697 IC50 = 220 nM T84634 C4WUJ1 122190698 IC50 = 600 nM T84634 C0Q7FL 122190699 IC50 = 620 nM T84634 CF0KD5 122190700 IC50 = 460 nM T84634 C09BCZ 122190701 IC50 = 1020 nM T84634 CI0MK6 122190702 IC50 = 410 nM T84634 CQ9L8H 122190703 IC50 = 740 nM T84634 CM82GH 122190704 IC50 = 840 nM T84634 CV9L3K 122190705 IC50 = 630 nM T84634 C0XY8O 122190706 IC50 = 1110 nM T84634 CWOC89 127031597 IC50 = 3500 nM T84634 D06RAM 10389639 IC50 = 60 nM T84634 D07VYX 10786043 IC50 = 200 nM T84634 D0F8JO 9951075 IC50 = 2.4 nM T84634 D0O6QU 2605 IC50 = 1630 nM T38875 D06ACW 6083 EC50 = 1519 nM T38875 D08UUL 46700756 IC50 = 101.62 nM T38875 CL7KB0 265479 EC50 = 1800 nM T38875 CKJP46 1825716 EC50 = 550 nM T38875 C1SVD2 2132479 IC50 = 2500 nM T38875 C18HKQ 9885748 IC50 = 46000 nM T38875 CVZ5X1 13042082 EC50 = 30000 nM T38875 CKV4G1 16079040 IC50 = 1500 nM T38875 C7YG1N 24759534 IC50 < 10 nM T38875 C4IY8M 45256689 EC50 = 8 nM T38875 C1R7WB 45256693 EC50 = 3 nM T38875 CEF64I 45273893 EC50 = 0.6 nM T38875 C2JHA7 45375932 EC50 = 13 nM T38875 C6EU8K 45375934 EC50 = 58 nM T38875 CHM6E5 45378798 EC50 = 300 nM T38875 C74OZB 46190967 EC50 = 97 nM T38875 CC17KH 46194961 EC50 = 1.2 nM T38875 CF38CI 51034107 EC50 = 1240 nM T38875 C4R8VQ 51034984 EC50 = 660 nM T38875 CMS4C2 53372240 EC50 = 4 nM T38875 C4W9XL 53372379 EC50 = 17 nM T38875 C1OGK6 54708532 EC50 = 800 nM T38875 CJ37NF 56591699 EC50 = 1490 nM T38875 C0PLM2 56591796 EC50 = 1240 nM T38875 CX93PS 56592835 EC50 = 1240 nM T38875 CT4E8R 56832546 IC50 = 26000 nM T38875 CXJ63M 59603829 IC50 = 26 nM T38875 CQEU96 59603842 IC50 = 4.6 nM T38875 CPD80M 60171744 EC50 = 1 nM T38875 C1Z3YP 60194103 EC50 = 630.96 nM T38875 CK6WO0 66552478 IC50 < 10000 nM T38875 CZ0V9E 67232851 EC50 = 870 nM T38875 C5DGR9 69036886 IC50 = 98 nM T38875 CXSI14 71718330 IC50 = 10000 nM T38875 C1TM3P 71720141 IC50 = 10000 nM T38875 COWG10 71748255 EC50 = 1.9 nM T38875 C95VYQ 71765798 EC50 = 57 nM T38875 CZ2NS1 71765801 EC50 = 80 nM T38875 C25TYS 71765951 EC50 = 43 nM T38875 C7Q5IH 71765955 EC50 = 1.3 nM T38875 CMZ4X2 71766100 EC50 = 47 nM T38875 C6PZY8 71767831 EC50 = 52 nM T38875 C19TPH 71767833 EC50 = 35 nM T38875 C6KQP7 71767991 EC50 = 7 nM T38875 C8Y2FX 86698571 EC50 = 53 nM T38875 CF0IS4 86698599 EC50 = 100 nM T38875 CWQA67 86698790 EC50 = 323 nM T38875 C6F3IK 86698802 EC50 = 8.3 nM T38875 C1HW4B 89735655 IC50 = 53 nM T38875 COSC89 89837093 EC50 = 24 nM T38875 CBY6J2 118053829 EC50 = 1 nM T38875 C24RMQ 118640135 EC50 = 11 nM T38875 C63DSU 118725336 EC50 = 1.1 nM T38875 CXG30B 118725337 EC50 = 184 nM T38875 CK1IS9 118725338 EC50 = 1840 nM T38875 CW1EO2 121396404 EC50 = 8 nM T38875 C9IMB0 121396405 EC50 = 59 nM T38875 CQMS08 121396411 EC50 = 38.1 nM T38875 CKCR81 121396412 EC50 = 76 nM T38875 C0U7DQ 134149170 EC50 = 3391 nM T38875 C3RWH7 134149412 EC50 = 3 nM T38875 C1S3NP 134150934 EC50 = 4 nM T38875 CUKT54 135398518 EC50 = 300 nM T38875 CJ1I5T 136183528 EC50 = 39.81 nM T38875 CY9G0L 137637206 EC50 = 62 nM T38875 CB1EZ5 137644835 EC50 = 1200 nM T38875 CVIM80 137651306 EC50 = 1600 nM T38875 CM5ZV6 137660838 EC50 = 270 nM T38875 CITW61 142771124 EC50 = 25118.86 nM T38875 CE0S8V 155532038 EC50 = 338.84 nM T38875 CG09DP 155548590 EC50 = 440 nM T38875 CZQM57 155554194 IC50 = 107.5 nM T59082 CTR94V 439281 Ki = 11000000 nM T59082 C68JEM 71623467 IC50 = 420000 nM T59082 CQ7H4I 76310828 IC50 = 40000 nM T59082 C4KA5F 76310829 IC50 = 7160000 nM T59082 CK7GZ9 76310830 IC50 = 5730000 nM T59082 C5UW2S 76310831 IC50 > 500000 nM T59082 CPNL61 76314448 IC50 = 4370000 nM T59082 C5XJR9 76314449 IC50 = 5150000 nM T59082 CWG83I 76318036 IC50 = 8790000 nM T59082 C5FNJ0 76318037 IC50 = 6490000 nM T59082 C7U3FD 76318038 IC50 > 500000 nM T59082 CNBD52 76318039 IC50 = 1010000 nM T59082 CWN58O 76321750 IC50 = 1020000 nM T59082 C6GCM4 76321751 IC50 = 13250000 nM T59082 CGE2N3 76321752 IC50 = 8640000 nM T59082 C06FQB 76325364 IC50 = 1340000 nM T59082 CNL49F 76325365 IC50 = 2410000 nM T59082 CUS61H 76325366 IC50 = 50000 nM T59082 CCY93X 76325367 IC50 > 500000 nM T59082 C5V3ZB 76325368 IC50 = 395000 nM T59082 CK6RA9 76332597 IC50 = 3890000 nM T59082 C7XGH3 76332598 IC50 = 14940000 nM T59082 C51OKC 86573947 IC50 = 310 nM T59082 CK5TZ1 122182803 IC50 = 34000 nM T59082 CRY0J4 122182804 IC50 = 1010000 nM T59082 CO4I6D 137631793 IC50 = 776000 nM T59082 CUH4X7 137638019 IC50 = 776000 nM T59082 CG9OE2 137653829 IC50 = 720000 nM T59082 C9B7YT 145979496 IC50 = 3200000 nM T59082 C2WPC9 145979996 IC50 = 100000 nM T59082 CRVW17 145981767 IC50 = 1400000 nM T59082 C4WM7S 145993839 IC50 = 450000 nM T59082 CAZ65D 155545302 IC50 = 481000 nM T59082 CU81IK 155569069 IC50 = 254000 nM T59082 D07LUR 185698 IC50 = 6400000 nM T59082 D0G6XS 17106 IC50 = 2950000 nM T59082 D0GS9E 18950 Ki = 13100000 nM T28132 C3G7VB 1234292 IC50 < 1000 nM T28132 CA2JU7 46911115 IC50 = 3981 nM T28132 C73VYX 46911116 IC50 = 200 nM T28132 CVD43F 56659471 IC50 = 79 nM T28132 C8SR2X 56659475 IC50 = 22 nM T28132 CNM68T 56662903 IC50 = 1071 nM T28132 CP2LW0 56662936 IC50 = 631 nM T28132 CX9FB0 56662937 IC50 = 6310 nM T28132 C8PQ0U 56666408 IC50 = 85 nM T28132 C7BQD3 56669824 IC50 = 126 nM T28132 CHAK86 56669827 IC50 = 1000 nM T28132 CU0KW5 56673309 IC50 = 398 nM T28132 CDX09S 56673310 IC50 = 1585 nM T28132 CK8U1S 56673311 IC50 = 1995 nM T28132 C0OYQ1 56676613 IC50 = 1000 nM T28132 C04IVB 56676641 IC50 = 316 nM T28132 CW37HG 56676642 IC50 = 631 nM T28132 CLF76V 56676643 IC50 = 794 nM T28132 C4QCS7 56676649 IC50 = 59 nM T28132 CZ98WA 56676650 IC50 = 537 nM T28132 C8QO3N 56679972 IC50 = 398 nM T28132 C4CY2J 56679973 IC50 = 1995 nM T28132 C7TR6Q 56679975 IC50 = 2131 nM T28132 CMWY31 56683305 IC50 = 10 nM T28132 CY5S9E 56683306 IC50 = 794 nM T28132 C3J2FI 56683309 IC50 = 158 nM T25847 D02EEJ 6479267 IC50 = 10.3 nM T25847 D0G7UX 5284373 IC50 = 8.78 nM T25847 C8RA6C 6476061 IC50 = 12.7 nM T25847 C31GDL 24814873 IC50 = 97.1 nM T25847 CWI47U 50899161 IC50 = 19.8 nM T25847 CHN71J 52940634 IC50 = 26.1 nM T25847 CQ83LE 52940669 IC50 = 25.2 nM T25847 C2H0IK 52940670 IC50 = 59.5 nM T25847 CPKZ45 52940671 IC50 = 28.9 nM T25847 C7MA9P 52941831 IC50 = 9.45 nM T25847 CH9QA8 52941859 IC50 = 17.2 nM T25847 C97YWD 52945243 IC50 = 30.5 nM T25847 CE05IO 52945473 IC50 = 151 nM T25847 C43LWJ 52945496 IC50 = 158 nM T25847 C3BCG7 52946681 IC50 = 66.8 nM T25847 CR63JF 52946682 IC50 = 20.6 nM T25847 CH8TZ9 52946683 IC50 = 79.7 nM T25847 C7KW3U 52947912 IC50 = 24.2 nM T25847 C4KAU1 52947949 IC50 = 1583 nM T25847 CGX04A 52947950 IC50 = 55.9 nM T25847 CDF54U 73333515 Ki = 35.2 nM T13057 D03DXN 66435 IC50 = 19900 nM T13057 D03SRY 259331 IC50 > 300000 nM T13057 D08QMX 5757 IC50 > 300000 nM T13057 D00MFW 92577 IC50 = 318 nM T13057 D0I2AN 86298439 IC50 = 200 nM T13057 CQ7GE6 20834 IC50 = 12640 nM T13057 CW68ZS 61672 IC50 = 24.1 ug.mL-1 T13057 CD6SZ4 69748 IC50 > 500000 nM T13057 CN2GL3 92576 IC50 = 300 nM T13057 C7KJ3B 114917 IC50 = 2570 nM T13057 C5X1YU 160254 IC50 = 22500 nM T13057 C4IRY2 164676 IC50 = 2590 nM T13057 CCEG90 259329 IC50 = 17100 nM T13057 CA8WX9 314313 IC50 = 39130 nM T13057 CM0IQ3 446665 IC50 = 91000 nM T13057 CELG48 998012 IC50 = 52070 nM T13057 CJ90PO 1159989 IC50 = 176000 nM T13057 CE3S9R 1820399 IC50 > 50000 nM T13057 CIV1E3 2775086 IC50 > 500000 nM T13057 CB7OS1 2964738 IC50 = 181000 nM T13057 CCHX35 3096032 IC50 = 42390 nM T13057 C2C5UW 3109390 Ki = 700 nM T13057 C3NL9W 3246406 IC50 = 4990 nM T13057 C9G0CA 3653077 IC50 = 29000 nM T13057 CGA0N7 3734796 IC50 > 60000 nM T13057 CTCI08 3784946 IC50 > 60000 nM T13057 CI7F3L 5098884 IC50 = 161 nM T13057 CSU5J3 5098885 IC50 = 97 nM T13057 CAW37X 5240714 IC50 > 60000 nM T13057 CPM09B 5327156 IC50 > 500000 nM T13057 C6XCJ8 6420094 IC50 = 1800 nM T13057 CH03PR 9866186 IC50 = 2100 nM T13057 C1ECT8 9867205 IC50 = 5000 nM T13057 CA75NG 9985013 IC50 = 60000 nM T13057 CYV93G 10172292 IC50 = 9000 nM T13057 CUV6M1 10198815 IC50 = 14000 nM T13057 C3A8JL 10256983 IC50 = 16000 nM T13057 CH45KB 10258785 IC50 = 10000 nM T13057 C9R7GJ 10260791 IC50 = 22000 nM T13057 C0D9QX 10372989 Ki > 30000 nM T13057 CT4H0O 11006141 IC50 = 32000 nM T13057 C2WP1J 11343454 IC50 = 2600 nM T13057 C1JAC5 11425923 IC50 = 3940 nM T13057 COIR53 11456678 IC50 = 1800 nM T13057 CM1XL8 11844603 IC50 > 100000 nM T13057 C75UVA 11844604 IC50 > 100000 nM T13057 C96HKI 11886168 IC50 = 2500 nM T13057 CPV08O 12658768 IC50 > 20000 nM T13057 CE8Y4G 13779016 IC50 = 201800 nM T13057 CWU92E 20866464 IC50 > 50000 nM T13057 CJKO23 20866499 IC50 > 50000 nM T13057 C12GAZ 21145366 Ki > 30000 nM T13057 C54IUM 21778115 IC50 > 50000 nM T13057 CWJ2N6 23577107 IC50 = 5370 nM T13057 CV07UA 23577108 IC50 = 19900 nM T13057 CS91QU 23577109 IC50 = 450 nM T13057 CJ7UP5 23577110 IC50 = 2270 nM T13057 CE9B6H 25014222 IC50 > 20000 nM T13057 CW69GS 25023777 IC50 = 4550 nM T13057 CSN1R4 25023778 IC50 = 1830 nM T13057 CW2H8L 25023779 IC50 = 2110 nM T13057 CR0E7L 25023780 IC50 = 500000 nM T13057 CZ4R5U 25023781 IC50 = 3910 nM T13057 C7KPR6 25023782 IC50 = 6400 nM T13057 CL41YO 25023783 IC50 = 10200 nM T13057 C40QFI 25147702 IC50 > 100000 nM T13057 C09KZA 25262525 IC50 = 36000 nM T13057 C4WM9S 25262527 Ki = 5200 nM T13057 C6ND7U 25640845 IC50 > 100000 nM T13057 C3P8XN 42644186 IC50 > 40000 nM T13057 C98IOF 42644187 IC50 > 40000 nM T13057 CL04IU 44156271 IC50 = 14000 nM T13057 C92TBJ 44324648 IC50 > 100000 nM T13057 CF3R6Y 44336593 Ki > 30000 nM T13057 CQ31LB 44356471 IC50 = 1540 nM T13057 CJUM36 44415112 IC50 > 100000 nM T13057 C46QTA 44423905 IC50 = 2200 nM T13057 C01HDT 44562085 IC50 = 2470 nM T13057 CT6WJ3 45271336 IC50 = 2900 nM T13057 CSA7P5 45378656 IC50 = 212000 nM T13057 C10PAG 45378788 IC50 = 7800 nM T13057 CY4FW6 45378789 IC50 = 10400 nM T13057 CPZW76 45378927 IC50 = 9100 nM T13057 CZW2K9 45378928 IC50 = 8000 nM T13057 CN3SI9 45378929 IC50 = 86000 nM T13057 CPY85V 45378930 IC50 = 9300 nM T13057 CY9O0P 45378931 IC50 = 12000 nM T13057 CYRC54 45482878 IC50 > 40000 nM T13057 CK98JB 45482885 IC50 > 40000 nM T13057 CQ5U3C 45482886 IC50 > 40000 nM T13057 C8Z7HX 45482894 IC50 > 40000 nM T13057 CCKE09 45482895 IC50 > 40000 nM T13057 CLGB06 46830252 IC50 > 10000000 nM T13057 C81CPM 46861833 IC50 = 15200 nM T13057 C0A9LD 46861834 IC50 = 12200 nM T13057 C83GCS 46882340 IC50 > 44000 nM T13057 CPEG29 46888174 IC50 = 9590 nM T13057 C2IU1Z 49796692 IC50 = 152000 nM T13057 C2NJ3B 51003508 IC50 = 14000 nM T13057 CMDB84 53316640 IC50 > 50000 nM T13057 C9GVU5 53317937 IC50 > 50000 nM T13057 CV4QD5 53317938 IC50 = 15700 nM T13057 CWT10N 53319270 IC50 > 50000 nM T13057 CRE6Y5 53319872 IC50 > 300000 nM T13057 CRC82E 53320578 IC50 > 50000 nM T13057 C8Y4KW 53320579 IC50 = 20600 nM T13057 CF35GK 53320580 IC50 = 17400 nM T13057 C04CYS 53320581 IC50 > 50000 nM T13057 CBI29Z 53321875 IC50 = 33300 nM T13057 C94WKB 53324565 IC50 > 50000 nM T13057 CNZY43 56589511 IC50 > 10000000 nM T13057 C53XYO 56589513 IC50 > 10000000 nM T13057 CHM5V3 56660070 IC50 > 120000 nM T13057 CHOF39 56670422 IC50 > 120000 nM T13057 CI9R8M 56670423 IC50 > 120000 nM T13057 CL3N0K 56673907 IC50 > 120000 nM T13057 CAL96I 56673908 IC50 > 120000 nM T13057 CEK3S2 56680547 IC50 > 120000 nM T13057 C72JTU 56681854 IC50 = 54300 nM T13057 CJ50EL 56681855 IC50 = 34500 nM T13057 CN3EW7 56683882 IC50 > 120000 nM T13057 C5CQY2 56683883 IC50 > 120000 nM T13057 CV4PW2 56683884 IC50 = 47600 nM T13057 CZP28F 57327772 IC50 = 20910 nM T13057 CG71TE 57380427 IC50 > 10000000 nM T13057 C4QJD7 57380429 IC50 > 10000000 nM T13057 CLTX25 57380431 IC50 > 10000000 nM T13057 CU94DW 57380433 IC50 = 191000 nM T13057 CCY75L 57380662 IC50 > 10000000 nM T13057 CE24LJ 57380664 IC50 = 210000 nM T13057 CWZ9E2 57380666 IC50 > 10000000 nM T13057 C9H7GI 57380668 IC50 > 10000000 nM T13057 CXW05S 57390693 IC50 > 10000000 nM T13057 CE57HQ 57395972 IC50 > 10000000 nM T13057 CGC16T 57397768 IC50 > 10000000 nM T13057 C18FTX 57397769 IC50 > 10000000 nM T13057 CQNG21 57397770 IC50 > 10000000 nM T13057 CX3A5R 57399431 IC50 > 10000000 nM T13057 CU5ND3 57514697 Ki = 6600 nM T13057 C4ZE0T 60142018 IC50 = 6900 nM T13057 COH1S4 60142154 IC50 = 7800 nM T13057 C49OYN 60142155 IC50 = 8000 nM T13057 CJ7AP3 67762287 IC50 > 20000 nM T13057 C2BT9H 70673568 IC50 = 2500 nM T13057 CUS3F6 70691280 IC50 > 100000 nM T13057 C3AJ7H 70981706 IC50 = 1800 nM T13057 CP4H6L 70981726 IC50 = 2200 nM T13057 C2KS7Y 70982811 IC50 = 1800 nM T13057 C7VES4 71449486 IC50 = 16670 nM T13057 CXI0F3 71561559 IC50 > 100000 nM T13057 CE0Y3O 71561685 IC50 = 4000 nM T13057 C3M4CF 71561686 IC50 = 3600 nM T13057 C82KCZ 71561687 IC50 = 2300 nM T13057 CDA8P2 71561688 IC50 = 38000 nM T13057 C87EXF 71561689 IC50 = 2830 nM T13057 CP9HX5 71561815 IC50 = 600 nM T13057 C9H5YS 71561816 IC50 = 5000 nM T13057 C61MWP 71561817 IC50 = 4500 nM T13057 C9GO5M 71561818 IC50 = 10900 nM T13057 CWA30F 71561819 IC50 = 4500 nM T13057 CBC4G0 71561820 IC50 = 5200 nM T13057 CPV8Y3 71561944 IC50 = 3600 nM T13057 CPWU40 71597177 IC50 = 31000 nM T13057 CT4MK9 71717989 IC50 = 30000 nM T13057 CCY15D 71734765 IC50 = 560 nM T13057 C6F1TD 72163289 IC50 = 13360 nM T13057 C0FWS2 72163422 IC50 = 13810 nM T13057 C2RNH4 72163424 IC50 = 21450 nM T13057 CNLB62 72163425 IC50 = 22290 nM T13057 CMC9L2 72190151 IC50 = 3400 nM T13057 CM1W6X 73352369 IC50 = 9200 nM T13057 C1DWU4 73353952 IC50 = 5300 nM T13057 C9UP3V 73353954 IC50 = 9890 nM T13057 CS5O4J 73355491 IC50 = 11660 nM T13057 CMDC47 73357035 IC50 = 6790 nM T13057 CY0K7L 73357036 IC50 = 10150 nM T13057 CH3V7I 76966642 IC50 = 12000 nM T13057 CERG27 86763337 IC50 = 4660 nM T13057 CGMI50 86763338 IC50 = 5420 nM T13057 CF05WT 86763339 IC50 = 220 nM T13057 CCFJ28 86763340 IC50 = 310 nM T13057 CD5W1T 86763452 IC50 = 420 nM T13057 CQE36J 86763453 IC50 = 630 nM T13057 CUX1G9 86764668 IC50 = 620 nM T13057 C2S3RG 86764669 IC50 = 660 nM T13057 C1W0XL 86764771 IC50 = 760 nM T13057 CW4A9E 86764772 IC50 = 770 nM T13057 CG5MU6 86764773 IC50 = 860 nM T13057 CNV49T 86764774 IC50 = 1050 nM T13057 CHD8N6 86764775 IC50 = 1200 nM T13057 CNW67M 86764883 IC50 = 1250 nM T13057 C0F7ES 86764884 IC50 = 1460 nM T13057 CWG7N1 86764885 IC50 = 1350 nM T13057 CGKE84 86764886 IC50 = 1490 nM T13057 C34KEY 86764887 IC50 = 1760 nM T13057 C6KM9C 86764996 IC50 = 1790 nM T13057 CP50RV 86764997 IC50 = 1840 nM T13057 C9KMS4 86764998 IC50 = 2310 nM T13057 CCR5O1 86764999 IC50 = 2390 nM T13057 CRU5W9 86765000 IC50 = 2730 nM T13057 CL4IN3 86766306 IC50 = 19740 nM T13057 CI8XJ4 90663933 IC50 > 5 nM T13057 CBK96X 90666455 IC50 > 20000 nM T13057 C61PBQ 90666456 IC50 > 20000 nM T13057 C40WCO 90666457 IC50 > 20000 nM T13057 C2ZGE9 90666458 IC50 > 20000 nM T13057 CG5TY1 90666459 IC50 > 20000 nM T13057 CWQN87 90666460 IC50 > 20000 nM T13057 CLU52N 90666461 IC50 = 19140 nM T13057 C0DW7A 90666462 IC50 > 20000 nM T13057 CXMC74 90666463 IC50 > 20000 nM T13057 CG36RV 91667928 IC50 = 14000 nM T13057 C19JKD 101884098 IC50 = 50000 nM T13057 CYW80L 102307785 IC50 = 2730 nM T13057 CL96MC 102532094 IC50 = 12500 nM T13057 C2BAM5 117803691 IC50 = 380 nM T13057 C6QM2W 118238298 IC50 = 70 nM T13057 CBEN51 118239663 IC50 = 300 nM T13057 C01WAG 118239984 IC50 = 1980 nM T13057 CPL19A 118247966 IC50 = 5700 nM T13057 CS41QV 118709487 IC50 = 14400 nM T13057 CL4IR5 118709488 IC50 = 370 nM T13057 CL8AK6 118709489 IC50 = 56000 nM T13057 CPDG83 118709490 IC50 = 2300 nM T13057 C8QWA7 118709491 IC50 = 3600 nM T13057 C8ISV6 118709492 IC50 = 5000 nM T13057 C6VAX0 118709493 IC50 = 4500 nM T13057 CLA0N9 118709494 IC50 = 5300 nM T13057 CR53LW 118709495 IC50 = 7200 nM T13057 C92GFL 118709496 IC50 = 8600 nM T13057 CP2V7L 118709497 IC50 = 10700 nM T13057 CIE91Q 118709498 IC50 > 20000 nM T13057 C3QK4Y 118709499 IC50 = 26000 nM T13057 CX2A8G 118722143 IC50 > 120000 nM T13057 CV5F0I 118722144 IC50 > 120000 nM T13057 C32ODE 118729111 IC50 = 6640 nM T13057 CTV62N 118729112 IC50 = 34620 nM T13057 CP9E4Q 118729113 IC50 = 18330 nM T13057 CS2XI7 118729114 IC50 = 10450 nM T13057 C3LN4T 118729115 IC50 = 8910 nM T13057 CF9KD7 118729116 IC50 = 9410 nM T13057 C27YKT 118729117 IC50 = 11460 nM T13057 C5FXC0 118729118 IC50 = 22250 nM T13057 C90UMX 118729119 IC50 = 24580 nM T13057 C0YGL1 118729120 IC50 = 13220 nM T13057 C4XZ2J 118729123 IC50 = 10870 nM T13057 C5GM1D 118729125 IC50 = 9690 nM T13057 CHF7U0 118729126 IC50 = 8250 nM T13057 C0M3VK 118729722 IC50 = 36800 nM T13057 CP4D5Q 118729725 IC50 = 33200 nM T13057 CWU09Y 118729729 IC50 = 31900 nM T13057 C0IJ2X 118737463 IC50 = 5400 nM T13057 C12OHP 122187565 Ki = 510 nM T13057 CXHR32 122187566 IC50 = 1400 nM T13057 C59OUG 122187567 IC50 = 2300 nM T13057 C2PVC5 122196288 IC50 = 11640 nM T13057 CUO46T 124140941 IC50 = 67 nM T13057 C04VCS 124140943 IC50 = 30 nM T13057 C0UAQ6 124147818 IC50 = 32 nM T13057 C8QAD1 124147824 IC50 = 37 nM T13057 C9SO3J 124147915 IC50 = 34 nM T13057 CS43YV 124147927 IC50 = 8 nM T13057 CZEC76 124147932 IC50 = 36 nM T13057 C5B4UL 124147957 IC50 = 50 nM T13057 C1KFO8 124147973 IC50 = 22 nM T13057 C70DOJ 124147979 IC50 = 27 nM T13057 C2VE5C 124148108 IC50 = 39 nM T13057 C3ER2Z 124148120 IC50 = 12 nM T13057 CH7OZ3 124148123 IC50 = 28 nM T13057 CFR2G7 124148125 IC50 = 260 nM T13057 CON3T6 124150358 IC50 = 105 nM T13057 CD5RM3 124150360 IC50 = 181 nM T13057 C25IJY 124150428 IC50 = 5 nM T13057 CHC02A 124150434 IC50 = 177 nM T13057 C04FYJ 124150499 IC50 = 23 nM T13057 C5H2QB 124150512 IC50 = 5 nM T13057 CD52ZW 124150523 IC50 = 429 nM T13057 CLJ36I 124150528 IC50 = 4 nM T13057 CE2W0X 124150540 IC50 = 31 nM T13057 C8N5JR 124150544 IC50 = 26 nM T13057 C9TB6E 124150550 IC50 = 28 nM T13057 C58EUN 124150620 IC50 = 10 nM T13057 C94XQA 124150663 IC50 = 12 nM T13057 C46PST 127024952 IC50 > 120000 nM T13057 CF05SB 127025572 IC50 > 120000 nM T13057 C0KDZ2 127025573 IC50 > 120000 nM T13057 CI0NR9 127025574 IC50 > 120000 nM T13057 C6RI3J 127025575 IC50 > 120000 nM T13057 C5Z4PH 127025576 IC50 > 120000 nM T13057 C94EIF 127025577 IC50 > 120000 nM T13057 CR87HW 127025578 IC50 > 120000 nM T13057 CM9CP5 127027398 IC50 > 120000 nM T13057 C2A4GS 127027399 IC50 > 120000 nM T13057 CYOQ30 127027703 IC50 > 120000 nM T13057 CX52UN 127027704 IC50 > 120000 nM T13057 C6TIJ1 127027705 IC50 > 120000 nM T13057 C6H9SE 127027706 IC50 > 120000 nM T13057 C2X4JK 127027707 IC50 > 120000 nM T13057 C6UR4C 127027724 IC50 > 120000 nM T13057 C0RQ1U 127027725 IC50 > 120000 nM T13057 C0K2UI 127028022 IC50 > 120000 nM T13057 C1WA5T 127028346 IC50 > 120000 nM T13057 CC8HW0 127028347 IC50 > 120000 nM T13057 C6T0DY 127028683 IC50 > 120000 nM T13057 CL6QV7 127028684 IC50 > 120000 nM T13057 CG68NT 127028685 IC50 > 120000 nM T13057 C3MCH5 127028686 IC50 > 120000 nM T13057 CIAX67 127050086 IC50 = 2160 nM T13057 CO8V1Q 134130829 IC50 > 20000 nM T13057 C9BH3S 134131790 IC50 = 114800 nM T13057 C3Q6HX 134132029 IC50 > 20000 nM T13057 COG29Y 134132248 IC50 = 6900 nM T13057 CXM14Y 134132344 IC50 > 20000 nM T13057 CY4N3A 134132971 IC50 = 12800 nM T13057 CJV5H9 134133280 IC50 = 8500 nM T13057 CQV2R8 134133435 IC50 = 9000 nM T13057 CIM15P 134134309 IC50 > 500000 nM T13057 CK1ED4 134137535 IC50 > 20000 nM T13057 CO69VN 134138834 IC50 = 392200 nM T13057 C9WV1I 134139428 IC50 > 20000 nM T13057 CCS63E 134140312 IC50 = 3500 nM T13057 CFVU60 134141414 IC50 = 20300 nM T13057 C4E0TR 134148396 IC50 > 20000 nM T13057 C9NU1K 134148434 IC50 = 136000 nM T13057 CRG1A0 134150611 IC50 > 20000 nM T13057 CR72FZ 134152023 IC50 = 19500 nM T13057 C1FGJ5 134152452 IC50 = 6700 nM T13057 CO24SI 134154614 IC50 = 19000 nM T13057 C5CU3J 134157618 IC50 > 20000 nM T13057 CN23HD 134157879 IC50 = 3200 nM T13057 CBD40I 135445085 Ki = 54500 nM T13057 CU29KR 135556239 IC50 = 1300 nM T13057 C72YQR 135647237 IC50 > 60000 nM T13057 CM40ZF 135656202 IC50 = 8658 nM T13057 CZLK13 135783298 Ki = 25600 nM T13057 CJC62N 135783299 Ki = 473600 nM T13057 CW61GO 135783300 Ki = 32300 nM T13057 C5OLC0 135783301 Ki = 388000 nM T13057 CI0ZD2 135783302 Ki = 11700 nM T13057 C7JY1E 135783303 Ki = 547500 nM T13057 CF1W0U 135783304 Ki = 1088200 nM T13057 CZC42X 135924009 IC50 = 4500 nM T13057 C5BL1Z 135924010 IC50 = 11900 nM T13057 C9UA3N 135924011 IC50 = 5000 nM T13057 C1V8JE 135924012 IC50 = 1300 nM T13057 C8HP1O 135924013 IC50 = 1400 nM T13057 CHUD85 135924014 IC50 = 5900 nM T13057 CTZ5K1 135924015 IC50 = 5500 nM T13057 CAF8B6 135924016 IC50 = 22900 nM T13057 CK4X8S 135924017 IC50 = 6300 nM T13057 CE1FB0 135924018 IC50 = 4800 nM T13057 C39EPD 135924019 IC50 = 8300 nM T13057 CEH2M5 135924020 IC50 = 10600 nM T13057 CN6I5O 135924021 IC50 = 15800 nM T13057 CKW8X5 135924023 IC50 = 22300 nM T13057 CO3EX1 135924024 IC50 = 4500 nM T13057 CBJ7F8 135924025 IC50 = 4400 nM T13057 C81SHP 135924026 IC50 = 3800 nM T13057 CI62JU 135924027 IC50 = 7400 nM T13057 CAL83P 135924028 IC50 = 1000 nM T13057 CJ14VX 135924029 IC50 = 5200 nM T13057 C5C4EP 135924030 IC50 = 800 nM T13057 C3OU8V 135924155 Ki = 18100 nM T13057 CE9O5C 135924156 Ki = 12900 nM T13057 CKMV15 135924157 Ki = 28700 nM T13057 CL32WR 135924158 Ki = 90800 nM T13057 CNF1P0 135924159 Ki = 103200 nM T13057 C0T8UJ 135924160 Ki = 11700 nM T13057 C76NSI 135924161 Ki = 16200 nM T13057 CZ0NP3 135924162 Ki = 22800 nM T13057 CQJ65M 135929084 Ki = 12300 nM T13057 C5QIK7 137174949 IC50 > 120000 nM T13057 CUF76K 137331590 IC50 = 46000 nM T13057 C9O8DG 137632552 IC50 = 4530 nM T13057 CPD4V1 137633197 IC50 = 1050 nM T13057 CA0G1S 137638114 IC50 = 14980 nM T13057 C7D4SW 137644380 IC50 = 940 nM T13057 CN1X0J 137651804 IC50 = 1700 nM T13057 CFV26J 137652273 IC50 = 180 nM T13057 CXQ40F 137653094 IC50 = 920 nM T13057 CQ7T4S 137653723 IC50 = 4700 nM T13057 CL4Z1R 137657281 IC50 = 1100 nM T13057 C4CY9T 137661102 IC50 = 15860 nM T13057 CRU6Z7 137796282 IC50 = 7670 nM T13057 C0WMZ4 139593950 IC50 > 36800 nM T13057 CTOP13 142357867 IC50 = 949 nM T13057 C6NQ9I 145720956 IC50 = 14000 nM T13057 C4DWG8 145950748 IC50 = 7760 nM T13057 CT6I5O 145961409 IC50 = 910 nM T13057 CX54KW 145965216 IC50 = 30620 nM T13057 C0UT4Z 145966104 IC50 = 15530 nM T13057 C5H4PZ 145966112 IC50 = 25800 nM T13057 C9ICD0 145966982 IC50 = 23920 nM T13057 C58OBV 145971193 IC50 = 1590 nM T13057 CUE85W 145971302 IC50 = 2110 nM T13057 C73LAX 145972390 IC50 = 26510 nM T13057 C4IKH8 145973652 IC50 = 29950 nM T13057 COKV83 145974730 IC50 = 10000 nM T13057 C82EIW 145976484 IC50 = 5810 nM T13057 C2OZ8G 145976572 IC50 = 13980 nM T13057 CC2YO9 155516358 IC50 = 4870 nM T13057 C3PVL6 155517759 IC50 = 7830 nM T13057 CGUP05 155517773 IC50 = 4260 nM T13057 C7L3BR 155518108 IC50 = 3290 nM T13057 C2LYI7 155518870 IC50 = 985 nM T13057 CDYT42 155519082 IC50 = 2280 nM T13057 CZ75SL 155521073 IC50 = 6930 nM T13057 C9SD1X 155522483 IC50 = 6544 nM T13057 C4IA1T 155522941 IC50 = 1300 nM T13057 CL3I5G 155526321 IC50 = 1573 nM T13057 CG5YL4 155527104 IC50 = 54000 nM T13057 CTB6J8 155531587 IC50 = 2180 nM T13057 C38HEA 155532611 IC50 = 3280 nM T13057 C3NIE0 155532810 IC50 = 277 nM T13057 CZ94EY 155534761 IC50 = 7743 nM T13057 CLZ31N 155536741 IC50 = 2670 nM T13057 CEPN70 155536960 IC50 = 7552 nM T13057 C8YO9Q 155537362 IC50 = 6 nM T13057 CQ63GA 155537698 IC50 = 3800 nM T13057 CRU6F2 155538623 IC50 = 5810 nM T13057 C3Y6ZF 155538861 IC50 > 38900 nM T13057 CLF25Z 155545436 IC50 = 1950 nM T13057 CL78UG 155545756 IC50 = 4600 nM T13057 CARH78 155548168 IC50 = 23500 nM T13057 C1N8YP 155548589 IC50 = 5650 nM T13057 CRH8J5 155548680 IC50 = 8110 nM T13057 C50TQN 155550512 IC50 = 3700 nM T13057 C3GD5P 155550890 IC50 = 1230 nM T13057 CN6G0X 155556117 IC50 = 55200 nM T13057 CA75HC 155556730 IC50 = 2940 nM T13057 CG3I4L 155557442 IC50 > 100000 nM T13057 C0XU6Z 155559063 IC50 = 22000 nM T13057 CJI90K 155559808 IC50 = 4110 nM T13057 C5E0GW 155560770 IC50 = 500 nM T13057 CD4E5F 155560948 IC50 = 99000 nM T13057 CR03FB 155562299 IC50 = 6500 nM T13057 CE74XH 155564341 IC50 = 3100 nM T13057 CL1S9J 155565716 IC50 = 7780 nM T13057 C7W5HT 155566457 IC50 > 37700 nM T13057 D01BZE 73659 IC50 > 40000 nM T13057 D0SJ2Q 10494 IC50 = 11620 nM T13057 D0U8IF 10114 IC50 = 9600 nM T18904 D00SUC 74766595 IC50 = 99 nM T18904 D03TPE 97394 IC50 = 1700 nM T18904 D05PXW 6451399 IC50 = 15300 nM T18904 D09NCT 53392492 IC50 = 3300 nM T18904 D0C8CI 45376513 IC50 = 14000 nM T18904 D0JQ9Z 575125 IC50 = 3300 nM T18904 D0WC4Z 45376646 IC50 = 13000 nM T18904 C25LHT 125134 IC50 = 72000 nM T18904 C76AMR 439391 IC50 = 24000 nM T18904 CT0H6S 439939 IC50 = 26000 nM T18904 C5K3ZJ 459531 IC50 = 501.19 nM T18904 C4C0EB 2816189 Ki = 3020 nM T18904 CW2JY7 5715254 Ki = 520 nM T18904 C2JW1I 6288112 Ki = 5500 nM T18904 CCYF63 9942424 IC50 = 1258.93 nM T18904 CW01ZQ 22581416 IC50 = 16700 nM T18904 CP65KR 22581444 IC50 = 13200 nM T18904 C75LNS 22581449 IC50 = 10900 nM T18904 CCAM68 22959876 IC50 = 14000 nM T18904 C9J8TY 25721068 IC50 = 25000 nM T18904 C7X3WA 28330466 IC50 > 100000 nM T18904 CB2H6R 44820611 IC50 = 33000 nM T18904 CP59WA 45376516 IC50 = 12000 nM T18904 C1WL2X 45376644 IC50 = 20000 nM T18904 C62OQG 45376778 IC50 = 10000 nM T18904 CGF78A 45376782 IC50 = 13000 nM T18904 C32PQB 45376911 IC50 = 17000 nM T18904 C7OJ5E 46899602 IC50 = 8700 nM T18904 CUMF70 46899605 IC50 = 6000 nM T18904 C2DBN5 46899607 IC50 = 800 nM T18904 C3G4QK 46899609 IC50 = 5500 nM T18904 C24GUR 46899759 IC50 = 11000 nM T18904 C6ZR3Y 46899761 IC50 = 22000 nM T18904 CLK96Z 46899763 IC50 = 8100 nM T18904 CBOM64 46899765 IC50 = 3200 nM T18904 C9ENX8 46899767 IC50 = 2000 nM T18904 CF2QL4 46899769 IC50 = 4400 nM T18904 CW10BJ 46901089 IC50 = 17000 nM T18904 C6Z1NU 46901246 IC50 = 120000 nM T18904 CC23YW 49847498 IC50 > 25000 nM T18904 CWP7L0 49848519 IC50 > 25000 nM T18904 CU8AX0 55281807 Ki = 1940 nM T18904 CVK29R 57386523 IC50 = 4690 nM T18904 C8VM6P 67283460 IC50 > 25000 nM T18904 CY21XA 70702122 IC50 = 34000 nM T18904 C5XA3R 71733941 IC50 = 23500 nM T18904 C4PW1L 71734037 IC50 = 2400 nM T18904 C14GIV 71735687 IC50 > 120000 nM T18904 CM02VN 71735839 IC50 = 100000 nM T18904 C4WS1H 71735840 IC50 = 65000 nM T18904 CT4YO5 71735841 IC50 > 120000 nM T18904 C2ZFM8 71735842 IC50 = 99000 nM T18904 CI5W0K 71735843 IC50 > 120000 nM T18904 CYF8O7 71767874 IC50 = 125.89 nM T18904 CFY18G 73333510 IC50 > 120000 nM T18904 CN5B4O 73352277 IC50 = 92000 nM T18904 CX23ZP 78426670 IC50 > 2500 nM T18904 CKXW73 78427224 IC50 > 2500 nM T18904 C63ATV 81750201 IC50 = 100 nM T18904 CS4Q1F 86268882 IC50 < 100 nM T18904 CRQ51Z 86346639 IC50 < 100 nM T18904 CW9F0K 89564218 IC50 < 1000 nM T18904 C83TUW 89825693 IC50 = 100 nM T18904 CFX8E0 90407594 IC50 > 10000 nM T18904 C2NA5I 91801131 IC50 = 3162.28 nM T18904 CP3DK0 96607511 IC50 = 200 nM T18904 C85UGZ 96608360 IC50 = 16500 nM T18904 CCZ4Q9 96617507 IC50 = 900 nM T18904 C10RDJ 101882871 IC50 = 15848.93 nM T18904 CY87WL 112499933 IC50 = 104200 nM T18904 C4FPD3 112726150 IC50 > 100000 nM T18904 C6YT2Q 118598059 IC50 = 104 nM T18904 C75JVN 122191451 IC50 = 19952.62 nM T18904 C59KNQ 122191457 IC50 = 79432.82 nM T18904 CM5X8J 122191459 IC50 = 63095.73 nM T18904 C7ASR0 122191460 IC50 > 100000 nM T18904 CRI6J4 122191461 IC50 > 100000 nM T18904 C75NJO 122191464 IC50 = 50118.72 nM T18904 C50VYK 122191465 IC50 = 39810.72 nM T18904 CSKY20 122191466 IC50 = 79432.82 nM T18904 CS3L8H 122191467 IC50 = 2511.89 nM T18904 CZ2NV1 122191468 IC50 = 5011.87 nM T18904 CYTW93 122191469 IC50 = 5011.87 nM T18904 CZV45H 122191470 IC50 > 100000 nM T18904 CZU02B 122191472 IC50 = 6309.57 nM T18904 CQ04FW 122191477 IC50 = 39810.72 nM T18904 CT6HG3 122191480 IC50 = 63095.73 nM T18904 C2OVF5 122196456 IC50 = 2800 nM T18904 C8ADX6 122196457 IC50 > 100000 nM T18904 C0BEV2 122196458 IC50 > 100000 nM T18904 C6TP8J 122196459 IC50 = 3700 nM T18904 CWJL93 122196460 IC50 > 100000 nM T18904 C6MN0G 122196461 IC50 > 100000 nM T18904 CO4Y6T 122196462 IC50 > 100000 nM T18904 C2QGM6 122196463 IC50 > 100000 nM T18904 C83MKU 122196464 IC50 > 100000 nM T18904 CY7E0F 122196465 IC50 > 100000 nM T18904 C5OS8R 122196466 IC50 > 100000 nM T18904 C17TXO 122196467 IC50 > 100000 nM T18904 CNO5H7 122196468 IC50 > 100000 nM T18904 CW7U8M 122196469 IC50 > 100000 nM T18904 CT9R8C 122196470 IC50 > 100000 nM T18904 CGB05N 122196471 IC50 = 19000 nM T18904 CJG7O8 122196472 IC50 = 6200 nM T18904 CGO9Q2 122196473 IC50 = 24000 nM T18904 CEVG21 122196474 IC50 = 1800 nM T18904 CP4T8R 122196475 IC50 = 82000 nM T18904 CFI31P 122196476 IC50 = 1600 nM T18904 CJF70B 122196477 IC50 = 5100 nM T18904 CL89QK 122196478 IC50 = 50000 nM T18904 C6H2YQ 122383780 EC50 = 9000 nM T18904 CT2UZ4 125377518 EC50 = 3800 nM T18904 CF7KD3 127030402 Ki = 420 nM T18904 C63NWD 127030711 IC50 < 1000 nM T18904 CXF0U5 127030712 IC50 < 1000 nM T18904 CN16WB 127030937 IC50 = 1000 nM T18904 C2FPM6 127031758 IC50 = 30600 nM T18904 C7W8TS 127031759 IC50 = 300 nM T18904 CMJE83 127031760 IC50 = 950 nM T18904 CDC17F 127032730 IC50 = 100 nM T18904 CL38FP 127033048 IC50 = 100 nM T18904 CEV3A1 133053816 IC50 = 230000 nM T18904 C2Z6CV 135567105 IC50 = 11500 nM T18904 CIW61V 135567106 IC50 = 1700 nM T18904 CNZ8K9 135567107 IC50 = 8000 nM T18904 CL9ZD4 135567108 IC50 = 900 nM T18904 CJM4Z2 135567109 IC50 = 4100 nM T18904 CDY98J 135567110 IC50 = 138 nM T18904 C1VAI3 135567112 IC50 = 126 nM T18904 CWI0N7 135567114 IC50 = 16700 nM T18904 C8LFY7 135567115 IC50 = 80 nM T18904 C5E0ZN 135567116 IC50 = 15600 nM T18904 CO1F4A 135567128 IC50 = 630.96 nM T18904 CWCY64 136048725 IC50 = 21800 nM T18904 CE1SW8 136053677 IC50 = 630.96 nM T18904 CMW30T 136053680 IC50 = 794.33 nM T18904 C6IJ5M 136053683 IC50 = 1584.89 nM T18904 CNY5T7 136053684 IC50 = 398.11 nM T18904 C2V6MX 136644692 IC50 > 100000 nM T18904 CF5XJ1 137146154 IC50 = 6900 nM T18904 CK8DR7 137174994 IC50 = 1400 nM T18904 CA6DH2 137174995 IC50 = 1800 nM T18904 CLDH80 137174999 IC50 = 390 nM T18904 CR37AY 137175000 IC50 = 660 nM T18904 C1J3YB 137175001 IC50 = 600 nM T18904 CGAS95 137175002 IC50 = 880 nM T18904 CS5C6F 137175084 IC50 = 42800 nM T18904 C7PZ2T 137175085 IC50 = 6100 nM T18904 C1B5CK 137175086 IC50 = 13100 nM T18904 CWV4Y6 137175087 IC50 > 100000 nM T18904 C9XOV5 137175088 IC50 = 58600 nM T18904 C34LUV 137175094 Ki = 3 nM T18904 CSWN28 137175120 IC50 = 138 nM T18904 C23GYQ 137175121 IC50 = 110 nM T18904 C8Y2PR 137175122 IC50 = 128 nM T18904 C7GUC3 137175140 IC50 = 136 nM T18904 CBD1Q8 137175175 IC50 = 600 nM T18904 CEL6B1 137175176 IC50 = 770 nM T18904 C7SC6T 137175177 IC50 = 175 nM T18904 CPU73A 137175178 IC50 = 123 nM T18904 CFJ76N 137175179 IC50 = 411 nM T18904 CA89LW 137175180 IC50 = 456 nM T18904 C5GV3Q 137175209 IC50 = 145 nM T18904 C93YUK 137175210 IC50 = 143 nM T18904 CB2XV7 137175225 IC50 > 100000 nM T18904 C0XN8Y 137175239 IC50 = 9800 nM T18904 CI4D3P 137175249 IC50 = 181 nM T18904 CTVD83 137175250 IC50 = 147 nM T18904 C80LCT 137175251 IC50 = 158 nM T18904 CKQ1I2 137175252 IC50 = 144 nM T18904 C1YGB9 137175253 IC50 = 540 nM T18904 C5OZR6 137175260 IC50 = 109 nM T18904 CIKW02 137175261 IC50 = 118 nM T18904 C91JZQ 137321153 IC50 = 5300 nM T18904 C0D7SY 137349487 IC50 = 290000 nM T18904 C7J1RC 138393333 IC50 = 2060 nM T18904 CYG29R 138393334 Ki = 4 nM T18904 CNG82D 138393336 Ki = 4 nM T18904 CPFZ83 138393339 IC50 = 613 nM T18904 CC6SU2 138393341 Ki = 5 nM T18904 CXV31U 138753208 IC50 = 131 nM T18904 C41KVR 138753209 IC50 = 77 nM T18904 CIQJ26 138753211 Ki = 2 nM T18904 CARJ34 138753212 Ki = 26 nM T18904 C6LWR4 145963760 IC50 = 81 nM T18904 C0RPS4 145964567 IC50 = 41 nM T18904 CONJ19 145965089 EC50 = 105000 nM T18904 C3U8OD 145966600 IC50 = 615 nM T18904 CM9X8H 145967298 IC50 = 11 nM T18904 C9U5TQ 145967792 IC50 = 23 nM T18904 CB97SG 145968018 IC50 = 34 nM T18904 CT5MO6 145971004 IC50 = 82 nM T18904 CK9V5O 145972063 IC50 = 17 nM T18904 CX4W7P 145975124 EC50 = 1216000 nM T18904 CC8KI6 145976146 IC50 = 31 nM T18904 CKU0D3 145976400 IC50 = 208 nM T18904 CQ4E0O 145977225 IC50 = 269 nM T18904 CIQ6Y7 145977327 IC50 = 6 nM T18904 C5TBS2 145977546 IC50 = 41 nM T18904 CL2FR4 145978064 IC50 = 43 nM T18904 C8OL2Q 145978411 IC50 = 373 nM T18904 CA8UD0 145978535 IC50 = 15 nM T18904 C0GX1R 145985174 IC50 = 4200 nM T18904 C0UEA8 145992575 IC50 = 2200 nM T18904 CEQD63 155510449 IC50 = 246 nM T18904 CCB54Y 155510907 IC50 = 143 nM T18904 CAMR98 155512849 IC50 = 68 nM T18904 C9TWS3 155514456 IC50 = 59 nM T18904 C7XNM9 155518054 IC50 = 1060 nM T18904 C4M1EO 155519111 Ki = 4 nM T18904 CRT5Z2 155525082 IC50 = 848 nM T18904 CMB9N3 155530704 IC50 = 184 nM T18904 C2HN9G 155536799 IC50 = 282 nM T18904 C7VX3Y 155538517 IC50 = 178 nM T18904 C6YJ5R 155539215 IC50 > 25000 nM T18904 CP8K5E 155540290 IC50 = 71 nM T18904 C7LFH3 155540572 IC50 = 2410 nM T18904 COL30E 155540589 IC50 > 25000 nM T18904 CTF1K9 155542268 IC50 = 141 nM T18904 C7EG9J 155543678 IC50 = 188 nM T18904 C3M0TR 155546359 IC50 = 756 nM T18904 CTU53I 155547264 IC50 = 42 nM T18904 C5MFJ8 155548449 IC50 = 12350 nM T18904 CIM7D4 155548682 IC50 = 25000 nM T18904 C1CNK5 155549007 IC50 = 212 nM T18904 CX9OP1 155550806 IC50 = 259 nM T18904 CN7H9B 155554391 IC50 > 25000 nM T18904 C48ANL 155557731 IC50 = 88 nM T18904 C4MU5J 155558505 IC50 = 693 nM T18904 CTDM51 155558717 IC50 = 136 nM T18904 C0GU8Y 155559177 IC50 > 25000 nM T18904 CPOM30 155560356 Ki = 3 nM T18904 CGU0A2 155563031 IC50 > 25000 nM T18904 CA9T8I 155563296 IC50 = 218 nM T18904 C32NYC 155565735 IC50 > 25000 nM T18904 CGCN43 155567831 IC50 = 103 nM T18904 C3SQ4A 155569285 IC50 = 83 nM T18904 D07IOY 10365 IC50 = 4200 nM T18904 D08IZY 3080614 IC50 = 250000 nM T18904 D0B2WZ 15331 IC50 > 3300000 nM T18904 D0P7MU 4119262 IC50 = 20900 nM T18904 D0S3DD 56963315 IC50 = 400000 nM T18904 D0X5US 459617 IC50 = 1700 nM T22717 CU7X3G 2384714 IC50 > 5000 nM T22717 CRCA04 13590499 IC50 = 1700 nM T22717 CJ8YF2 13590558 IC50 > 5000 nM T22717 C1KN9T 24938152 IC50 = 310 nM T22717 C9EZ0X 25016113 IC50 = 830 nM T22717 C1WNJ5 25016370 IC50 = 520 nM T22717 CW7ZY1 25016377 IC50 = 720 nM T22717 CO7TN0 25016625 IC50 = 330 nM T22717 C1Q7XM 25016626 IC50 = 400 nM T22717 C4RA5E 25016628 IC50 = 150 nM T22717 C8VWT2 25016629 IC50 > 5000 nM T22717 CHC32Q 25016630 IC50 = 560 nM T22717 C6MOR1 25016631 IC50 = 1760 nM T22717 C0KR6F 25016883 IC50 = 260 nM T22717 C1G2EV 25016886 IC50 = 270 nM T22717 C87SMQ 25016887 IC50 = 210 nM T22717 CM19XI 25016888 IC50 > 5000 nM T22717 CL8S6A 25016889 IC50 = 2770 nM T22717 C4ML3F 25095022 IC50 = 660 nM T22717 C6M2FV 25095025 IC50 > 5000 nM T22717 CXGU79 25096820 IC50 = 150 nM T22717 CD7V1J 25097072 IC50 = 320 nM T22717 C3KGR7 25097315 IC50 = 2190 nM T22717 CAC4H7 25097316 IC50 = 430 nM T22717 CH8DY0 25097317 IC50 = 520 nM T22717 C95MYB 25097319 IC50 = 1040 nM T22717 C4GFB3 25097320 IC50 = 390 nM T22717 CJA2M5 25097322 IC50 > 5000 nM T22717 C37PQX 25097579 IC50 = 2820 nM T22717 C7N0JG 25097580 IC50 > 5000 nM T22717 CML61T 25097581 IC50 = 360 nM T22717 C1MQ5P 25097582 IC50 = 910 nM T22717 CFQY57 25097583 IC50 = 770 nM T22717 C9NKV4 25098135 IC50 = 640 nM T22717 C04ZFM 25098136 IC50 = 1220 nM T22717 CF01QP 25098137 IC50 = 710 nM T22717 CA0BL7 25098138 IC50 = 1000 nM T22717 CO32GA 25098140 IC50 = 410 nM T22717 CVF1L2 25098141 IC50 = 690 nM T22717 C75IZF 25098410 IC50 = 170 nM T22717 CT53KC 25098411 IC50 = 200 nM T22717 CY8WB9 25098412 IC50 = 290 nM T22717 CP03DL 57391543 IC50 = 60 nM T22717 CU48OP 57398520 IC50 > 5000 nM T22717 CB2DV7 57401984 IC50 > 5000 nM T22717 CL42OS 57402116 IC50 = 260 nM T22717 CBO25P 135412019 IC50 = 2570 nM T90070 D09BHB 5509 IC50 = 90 nM T90070 D0R1RS 3715 IC50 = 50 nM T90070 D0TG1H 3033 IC50 = 8 nM T90070 D0ZL4F 180540 IC50 = 20 nM T90070 CCZ3K9 15250 IC50 > 1000 nM T90070 C4PG1B 30931 IC50 > 1000 nM T90070 CNB6V7 114864 IC50 = 50 nM T90070 C7AKH8 141222 IC50 > 1000 nM T90070 C6EVL8 854057 IC50 > 1000 nM T90070 CNRE12 13309832 IC50 > 1000 nM T90070 CRB2H6 14762946 IC50 = 500 nM T90070 CNJ72V 18546323 IC50 > 1000 nM T90070 C5FD2Z 22218600 IC50 > 1000 nM T90070 CM3NT2 44298341 Ki = 13000 nM T90070 CX79VC 45268160 IC50 > 1000 nM T90070 C95IAE 45269044 IC50 = 600 nM T90070 CS2JM1 45269050 IC50 = 12 nM T90070 CEGP42 45269893 IC50 = 50 nM T90070 C5TE3O 45269894 IC50 = 13 nM T90070 C4O9EY 45269895 IC50 = 650 nM T90070 C34QNT 45269905 IC50 = 10 nM T90070 CGVT73 45270722 IC50 = 20 nM T90070 C4KH1C 45272452 IC50 = 25 nM T90070 C03KDJ 78224453 Ki = 7000 nM T90070 C0M8ZV 134130686 Ki = 106000 nM T90070 C1AS4F 134130687 Ki = 4000 nM T90070 CG0QB1 134130688 Ki = 12000 nM T90070 CFZG03 134130848 Ki = 10000 nM T90070 CGH9T1 134130849 Ki = 13000 nM T90070 CGW47R 134130850 Ki = 14000 nM T90070 C1NY6S 134130851 Ki = 6000 nM T90070 C2B3KN 134130852 Ki = 31000 nM T90070 CA0X3S 134130853 Ki = 4000 nM T90070 C42SCP 134130854 Ki = 383000 nM T90070 CD1TK0 134130855 Ki = 9300 nM T90070 CG35UE 134130856 Ki = 2300 nM T90070 D05EMX 14076674 IC50 = 25 nM T90070 D08GOT 13752584 IC50 = 400 nM T90070 D0I8YN 18546352 IC50 = 9 nM T90070 D0Q8ZV 15581854 IC50 = 500 nM T90070 D0T8RL 13409348 IC50 = 13 nM T39716 D00PEH 135449332 IC50 = 316227.77 nM T39716 D00STL 644241 IC50 = 1000000 nM T39716 D01AXB 60835 IC50 = 7943.28 nM T39716 D01AZG 5073 IC50 = 102000 nM T39716 D01FGR 3100 IC50 = 41000 nM T39716 D01UTL 2995 IC50 = 1520 nM T39716 D03DAP 3356 IC50 = 6500 nM T39716 D03FLC 3878 IC50 = 39810.72 nM T39716 D03HFG 5324346 IC50 = 39400 nM T39716 D03IGH 213039 IC50 = 39810.72 nM T39716 D03QWT 73303 IC50 = 1584893.19 nM T39716 D04FVU 6337614 IC50 = 19952.62 nM T39716 D04JEE 4946 IC50 = 2100 nM T39716 D05MQK 110635 IC50 = 125892.54 nM T39716 D05OFX 219078 IC50 = 501187.23 nM T39716 D08CDI 208908 IC50 = 3162277.66 nM T39716 D08HQK 5411 IC50 = 530 nM T39716 D09MWJ 2092 IC50 = 199526.23 nM T39716 D0B3UJ 115237 IC50 = 158489.32 nM T39716 D0BP9C 193962 IC50 = 501187.23 nM T39716 D0BZ7W 443879 IC50 = 6309.57 nM T39716 D0C7ET 11174599 IC50 > 30 nM T39716 D0C9SY 135400189 IC50 = 2511886.43 nM T39716 D0CL9S 159269 IC50 = 3162277.66 nM T39716 D0CS2F 3955 IC50 = 239 nM T39716 D0D7KC 5488548 IC50 = 251188.64 nM T39716 D0E4DW 1775 IC50 = 49000 nM T39716 D0E6XR 3062316 IC50 = 398107.17 nM T39716 D0H7KF 5002 IC50 = 16900 nM T39716 D0I1FQ 54671008 IC50 = 316227.77 nM T39716 D0J2KV 4932 IC50 = 1190 nM T39716 D0K3QS 6442177 IC50 = 199526.23 nM T39716 D0L4YD 154059 IC50 = 6309.57 nM T39716 D0NR6S 3002977 IC50 = 630957.34 nM T39716 D0NW3X 71329 IC50 > 300000 nM T39716 D0O3FG 125017 IC50 = 199526.23 nM T39716 D0Q5UQ 214348 IC50 = 79432.82 nM T39716 D0R0FE 2520 IC50 = 41500 nM T39716 D0R0MW 5329102 IC50 = 39810.72 nM T39716 D0U0VU 5312125 IC50 = 63095.73 nM T39716 D0U1OE 5452 IC50 = 1830 nM T39716 D0U2JP 4369359 IC50 = 630957.34 nM T39716 D0X0RI 4178 IC50 = 58000 nM T39716 D0X4RN 3676 IC50 = 108000 nM T39716 D0X5ZI 6918493 IC50 = 1000000 nM T39716 D0Y4JJ 2351 IC50 = 3700 nM T39716 D0Y5AM 444031 IC50 = 1584.89 nM T39716 D0Y5UG 2160 IC50 = 1600 nM T39716 D0Z1UA 71301 IC50 = 7943.28 nM T39716 D0Z7ZM 135398744 IC50 = 501187.23 nM T39716 D02AIN 122678117 IC50 > 33000 nM T39716 D04JZH 11659955 IC50 = 9000 nM T39716 D04PER 49836093 IC50 = 84 nM T39716 D06ENM 66553195 IC50 = 4700 nM T39716 D06TQR 76287260 IC50 > 100000 nM T39716 D0DH5X 44472635 IC50 > 30000 nM T39716 D0K9IF 71666749 IC50 > 30000 nM T39716 D0L9QM 59568713 IC50 > 30000 nM T39716 D0M3XR 46209133 IC50 > 30000 nM T39716 D0O7QA 46840946 IC50 = 11 nM T39716 D0OX9F 16046068 IC50 = 84000 nM T39716 D0P5CM 56945146 IC50 = 12589.25 nM T39716 D0S5IR 86294073 IC50 > 30000 nM T39716 D0W8XT 60663 IC50 = 500 nM T39716 D08IMD 16755780 IC50 = 14000 nM T39716 D0E2FZ 10149311 IC50 > 30000 nM T39716 D0HG2S 86294663 IC50 > 30000 nM T39716 D08SOF 5405 IC50 = 971 nM T39716 CZUI83 2769 IC50 = 14700 nM T39716 CP1QC0 9801 IC50 = 2520 nM T39716 C3H6AQ 21467 IC50 = 7800 nM T39716 CP8F7B 64143 IC50 = 501187.23 nM T39716 CLD6J9 441074 IC50 = 6900 nM T39716 CZN6S9 743974 IC50 > 100000 nM T39716 CPN25U 998021 IC50 = 9200 nM T39716 CTZ4R5 2730286 IC50 = 200 nM T39716 CORX94 2804997 IC50 = 5495.41 nM T39716 CMV0O1 3035569 IC50 = 30000 nM T39716 CM8IR4 4879545 IC50 = 980 nM T39716 C9ZT3K 9799052 IC50 = 2100 nM T39716 C5Z2KM 9805944 IC50 = 483 nM T39716 CY30OZ 9819588 IC50 = 2850 nM T39716 CS6FN7 9883254 IC50 = 8520 nM T39716 C4CH5D 9927877 IC50 = 4000 nM T39716 CREZ06 9928808 IC50 = 9000 nM T39716 CGY63T 10004877 IC50 > 100000 nM T39716 C5WLU0 10039502 IC50 = 5780 nM T39716 C1N5LX 10065677 IC50 = 13000 nM T39716 CF7OC8 10073954 IC50 = 30000 nM T39716 C97OQC 10088458 IC50 = 25000 nM T39716 C71ZGK 10316911 IC50 = 560 nM T39716 CT6Y9I 10365686 IC50 = 126000 nM T39716 C2KO8V 10388264 IC50 > 30000 nM T39716 CP7CH6 10389946 IC50 > 100000 nM T39716 CZN82G 10406083 IC50 = 15000 nM T39716 CBR9K8 11541314 IC50 = 60000 nM T39716 CS1V0J 11566989 IC50 = 2560 nM T39716 CKI9D5 11599973 IC50 > 31600 nM T39716 CQL5S8 11613750 IC50 > 100000 nM T39716 CXG1B4 11649741 IC50 > 100000 nM T39716 CH8K2V 11780892 IC50 > 100000 nM T39716 CD34SB 15982534 IC50 > 100000 nM T39716 CPCZ62 16040329 IC50 = 4700 nM T39716 CBF18D 21558498 IC50 = 455 nM T39716 CL73HJ 21589240 IC50 = 0.28 nM T39716 C5V2PF 22149197 IC50 = 14200 nM T39716 CAL57W 22149198 IC50 = 1510 nM T39716 CNM8X9 22149200 IC50 = 5250 nM T39716 C13HDG 22149207 IC50 = 5600 nM T39716 CYU64Q 22149216 IC50 = 8500 nM T39716 CUI6D7 22149230 IC50 = 8850 nM T39716 CNT32Z 22149267 IC50 = 2350 nM T39716 CH76LZ 22149271 IC50 = 1750 nM T39716 C2LUF7 22149278 IC50 = 7890 nM T39716 CL14RW 22149294 IC50 = 1100 nM T39716 CGBU69 22149297 IC50 = 4100 nM T39716 CMRN02 22149337 IC50 = 10800 nM T39716 CCY65J 22149344 IC50 = 3600 nM T39716 C6X0LN 22149356 IC50 = 3600 nM T39716 CFYW59 22149360 IC50 = 5400 nM T39716 CPXW92 22149373 IC50 = 2710 nM T39716 CUGR26 24757965 IC50 = 12000 nM T39716 CX79CS 24757966 IC50 > 30000 nM T39716 CDF15M 24759558 IC50 = 9000 nM T39716 CTG41H 24778289 IC50 > 2000 nM T39716 CM2DL3 24795066 IC50 > 30000 nM T39716 CF75YB 24857856 IC50 = 100 nM T39716 C3UNC4 24864147 IC50 = 14000 nM T39716 C6CK5U 24883321 IC50 = 4780 nM T39716 C5WOA3 24883322 IC50 = 7430 nM T39716 C5KA0N 24893979 IC50 = 84000 nM T39716 C21VCQ 25001553 IC50 = 7000 nM T39716 C6H4YL 25001554 IC50 = 25000 nM T39716 CUMH07 25001555 IC50 > 30000 nM T39716 CJR70I 25001557 IC50 = 26000 nM T39716 CIWR78 25001850 IC50 = 6000 nM T39716 C91QFN 25019282 IC50 > 30000 nM T39716 C0Z2SQ 25056787 IC50 = 2511.89 nM T39716 CPAZ91 25056788 IC50 = 5011.87 nM T39716 CP03LT 25113806 IC50 = 3981.07 nM T39716 CY5A6Q 25113809 IC50 = 3162.28 nM T39716 CK3JN1 25138309 IC50 = 7244.36 nM T39716 CWF5Z3 25143506 IC50 > 30000 nM T39716 CP72MB 25159060 IC50 = 12000 nM T39716 CBK27L 25196164 IC50 > 30000 nM T39716 CXKB13 25204469 IC50 = 8709.64 nM T39716 CAW05V 25204470 IC50 = 2630.27 nM T39716 C38CAX 25204471 IC50 > 25703.96 nM T39716 CUZ1Y2 25204472 IC50 = 8709.64 nM T39716 C1GO8L 25204473 IC50 = 1348.96 nM T39716 C9ZTJ3 25204533 IC50 > 15848.93 nM T39716 C2O6LT 25204534 IC50 > 33113.11 nM T39716 CBG48F 25204535 IC50 > 28840.32 nM T39716 C3JN6D 25204536 IC50 > 28183.83 nM T39716 C76UDL 25204600 IC50 = 8511.38 nM T39716 CXOZ41 25204603 IC50 = 5888.44 nM T39716 C08BDN 25204604 IC50 = 7762.47 nM T39716 C4IUB3 25204605 IC50 > 10471.29 nM T39716 CBH9O2 25204669 IC50 = 19952.62 nM T39716 C92WAR 25204670 IC50 > 33113.11 nM T39716 CYIV75 25204736 IC50 > 33113.11 nM T39716 CZY68S 25204738 IC50 > 33113.11 nM T39716 C1IW5M 25261456 IC50 > 10000 nM T39716 CY4LG8 42622934 IC50 > 30000 nM T39716 C96FIN 42644084 IC50 > 10000 nM T39716 C8BI5F 42644088 IC50 > 10000 nM T39716 CREJ31 42646199 IC50 > 10000 nM T39716 CKZ76R 42646202 IC50 < 10000 nM T39716 C81NVM 42646450 IC50 < 10000 nM T39716 CVBO78 42647178 IC50 < 10000 nM T39716 CX4YL8 44232522 IC50 > 10000 nM T39716 C7UY5F 44235863 IC50 > 10000 nM T39716 CX2W8Y 44236320 IC50 > 10000 nM T39716 C8LN0U 44236321 IC50 > 10000 nM T39716 CK4S5Y 44236322 IC50 > 10000 nM T39716 C62NRA 44337110 IC50 = 1760 nM T39716 C4K5MJ 44337198 IC50 = 15500 nM T39716 CP92BO 44337462 IC50 = 3920 nM T39716 CSMF57 44337512 IC50 = 10500 nM T39716 C85VGK 44337552 IC50 = 7900 nM T39716 C2QK4J 44472590 IC50 > 30000 nM T39716 CQ8C3F 44472591 IC50 > 30000 nM T39716 CC2TA5 44472592 IC50 > 30000 nM T39716 CWN95E 44472610 IC50 > 30000 nM T39716 C1H2ZT 44472612 IC50 > 30000 nM T39716 C9G5ID 44472613 IC50 > 30000 nM T39716 C5N4KE 44472633 IC50 > 30000 nM T39716 C5RNK0 44476261 IC50 = 4000 nM T39716 C6AK3W 44476911 IC50 > 30000 nM T39716 CLDQ43 44476913 IC50 > 30000 nM T39716 CG3R4T 44477000 IC50 = 27000 nM T39716 C1FTA7 44481065 IC50 > 30000 nM T39716 C01UWF 44540282 IC50 > 33000 nM T39716 CWP9Q3 44540283 IC50 > 33000 nM T39716 CKCG52 44540374 IC50 = 4400 nM T39716 CPFO82 44540469 IC50 = 18000 nM T39716 C46HBA 44540470 IC50 = 12000 nM T39716 C5NFE6 44540656 IC50 = 2900 nM T39716 C2MF7Z 44540754 IC50 = 4500 nM T39716 C5O4TM 44540839 IC50 = 19000 nM T39716 CYM71J 44543780 IC50 = 940 nM T39716 CD4LN9 44543781 IC50 = 2800 nM T39716 CE0K5T 44543783 IC50 = 12000 nM T39716 CS10AL 44543784 IC50 = 8700 nM T39716 C17LUC 44543889 IC50 = 4400 nM T39716 C9X2SL 44543890 IC50 > 26000 nM T39716 CE6HW8 44543891 IC50 = 6100 nM T39716 CB83EJ 44544123 IC50 > 31000 nM T39716 CN64WQ 44544347 IC50 = 730 nM T39716 CQ79RB 44544349 IC50 = 1600 nM T39716 CSV3F9 44544441 IC50 = 12000 nM T39716 C0RI5Z 44544444 IC50 = 3700 nM T39716 CK8T7U 44544546 IC50 = 8900 nM T39716 C7B0LF 44544548 IC50 = 8500 nM T39716 COJ7H6 44544644 IC50 = 6100 nM T39716 CYJB15 44544645 IC50 = 2600 nM T39716 CIO82A 44544649 IC50 > 23000 nM T39716 C8RAF0 44544851 IC50 = 19000 nM T39716 CWKZ36 44544853 IC50 > 8300 nM T39716 C6AX2C 44544950 IC50 = 4300 nM T39716 CGB50M 44545053 IC50 = 1900 nM T39716 C6VF4T 44545055 IC50 = 7900 nM T39716 CU16DA 44545166 IC50 = 16000 nM T39716 C9V7OF 44545167 IC50 > 33000 nM T39716 CW78UO 44545168 IC50 = 13000 nM T39716 CNZ12F 44545169 IC50 = 4700 nM T39716 CCD1V2 44545286 IC50 > 25000 nM T39716 C5KZ2M 44545289 IC50 = 1900 nM T39716 C9JK4V 44545402 IC50 = 17000 nM T39716 C6L8QO 44545403 IC50 = 810 nM T39716 CGLQ31 44552634 IC50 > 33000 nM T39716 CC2IO4 44552811 IC50 > 33000 nM T39716 CTX13C 44555196 IC50 > 33000 nM T39716 C5EX1K 44555473 IC50 > 10000 nM T39716 CXHT91 44571305 IC50 > 30000 nM T39716 CR32XZ 44571307 IC50 > 30000 nM T39716 C0IP7C 44583234 IC50 > 10000 nM T39716 C6HTC1 44583235 IC50 > 10000 nM T39716 CZJU04 44583236 IC50 < 10000 nM T39716 C3TYW0 44583237 IC50 < 10000 nM T39716 CCL9R0 44583238 IC50 > 10000 nM T39716 COX7F1 44583287 IC50 > 10000 nM T39716 C5SI9Q 44583288 IC50 > 10000 nM T39716 CFT74N 44583289 IC50 > 10000 nM T39716 CC19TZ 44583290 IC50 > 10000 nM T39716 C90RAV 44583349 IC50 > 10000 nM T39716 CK81NJ 44583350 IC50 > 10000 nM T39716 C20VTN 44583351 IC50 > 10000 nM T39716 CD5U3A 44583352 IC50 > 10000 nM T39716 C9G7VT 44583353 IC50 > 10000 nM T39716 C6QF4O 44583354 IC50 > 10000 nM T39716 C48AQR 44583355 IC50 > 10000 nM T39716 CG5X0M 44583356 IC50 < 10000 nM T39716 CUG9Y0 44583357 IC50 = 1000 nM T39716 CER76K 44585595 IC50 = 2300 nM T39716 C64ZKC 44593664 IC50 > 10000 nM T39716 C01BFQ 44593665 IC50 > 10000 nM T39716 C40BIM 45139151 IC50 = 15800 nM T39716 CUT2B4 45267348 IC50 > 10000 nM T39716 CJH3A2 45268206 IC50 > 10000 nM T39716 C4WR0V 45269087 IC50 > 10000 nM T39716 CRPS25 45269096 IC50 > 10000 nM T39716 C7BNY6 45269104 IC50 < 10000 nM T39716 CS1Q2X 45269947 IC50 > 10000 nM T39716 C1BE5U 45269948 IC50 > 10000 nM T39716 CG1H9N 45269950 IC50 = 10000 nM T39716 C1NT2M 45270771 IC50 > 10000 nM T39716 CA05IG 45270778 IC50 > 10000 nM T39716 CZ7MK9 45270788 IC50 < 10000 nM T39716 C9TM2P 45271593 IC50 > 10000 nM T39716 C06YAD 45271599 IC50 > 10000 nM T39716 CG0I8P 45271610 IC50 > 10000 nM T39716 C6FBH0 45271618 IC50 < 10000 nM T39716 C71VIG 45272510 IC50 > 10000 nM T39716 C05EDY 45272511 IC50 > 10000 nM T39716 CD62AH 45273373 IC50 > 10000 nM T39716 CMN39U 45273380 IC50 > 10000 nM T39716 C9L4KT 46205341 IC50 > 333000 nM T39716 CL41FE 46206000 IC50 > 333000 nM T39716 C1L0GS 46840949 IC50 = 17060 nM T39716 C4C0ED 46840950 IC50 > 10000 nM T39716 CI1YK3 46841216 IC50 = 35118 nM T39716 CD8M3F 46841499 IC50 = 29291 nM T39716 CO76ID 46841501 IC50 > 10000 nM T39716 CS5EJ1 46841648 IC50 > 30000 nM T39716 CRE97F 46841787 IC50 > 30000 nM T39716 COV0Q3 46841788 IC50 = 14413 nM T39716 C2OWF8 46841789 IC50 = 10549 nM T39716 CRU1P2 46882874 IC50 > 10000 nM T39716 C0FM2D 46882917 IC50 > 10000 nM T39716 CC1VO9 46882918 IC50 > 10000 nM T39716 C27RIV 46882919 IC50 > 10000 nM T39716 CE3O7D 46882949 IC50 > 10000 nM T39716 CHS1X0 46882950 IC50 > 10000 nM T39716 C3A1ZF 46882969 IC50 > 10000 nM T39716 CD7XA2 46882972 IC50 > 10000 nM T39716 CY5CW2 46882973 IC50 > 10000 nM T39716 C3ZPY7 46882986 IC50 > 10000 nM T39716 CKX8N2 46882987 IC50 > 10000 nM T39716 CG81CZ 46882988 IC50 > 10000 nM T39716 CP87CA 46883032 IC50 > 10000 nM T39716 CWU4T2 46883033 IC50 > 10000 nM T39716 C41RYD 46883034 IC50 > 10000 nM T39716 C3SQ2Z 46883035 IC50 > 10000 nM T39716 CS51UC 46883473 IC50 > 10000 nM T39716 CL0S4B 46883474 IC50 < 10000 nM T39716 C0K5ZJ 46883508 IC50 > 1000 nM T39716 CMNJ24 46883509 IC50 = 10000 nM T39716 CF4VC1 46883510 IC50 > 10000 nM T39716 C8Z0VS 49831248 IC50 = 351 nM T39716 C5LE0P 49850210 IC50 = 182 nM T39716 CLJ89W 49869305 IC50 = 1034 nM T39716 C9YM1Q 49869306 IC50 = 2938 nM T39716 CQ9PZ5 49869459 IC50 = 4577 nM T39716 C2N0XV 49869747 IC50 = 13770 nM T39716 C90UKY 50899643 IC50 > 30000 nM T39716 C94NCJ 50905973 IC50 = 223 nM T39716 CENW12 50925404 IC50 = 1320 nM T39716 C06OXV 52920492 IC50 = 69000 nM T39716 C6RFU2 53025800 IC50 = 4384 nM T39716 CPD0F2 53025889 IC50 = 7601 nM T39716 C0GF1R 53025891 IC50 = 4418 nM T39716 CMU7X8 53025901 IC50 = 7172 nM T39716 C08VWL 53025902 IC50 = 6943 nM T39716 CY74FO 53025906 IC50 = 8033 nM T39716 C5PB6K 53025909 IC50 = 4891 nM T39716 CY3R7J 53058099 IC50 = 4325 nM T39716 C8BG5J 53058100 IC50 = 3949 nM T39716 C02VSJ 53058119 IC50 = 8144 nM T39716 CK59VP 53058205 IC50 = 8092 nM T39716 CMS2F7 53239561 IC50 = 920 nM T39716 CRB6N5 53307604 IC50 > 33113.11 nM T39716 CJ83EB 53311393 IC50 > 10000 nM T39716 C23WVS 53361524 IC50 = 1100 nM T39716 C54YUZ 53362500 IC50 = 6800 nM T39716 CBAC86 53362558 IC50 = 500 nM T39716 CYX87Q 53362559 IC50 = 300 nM T39716 C8B1ZY 53362973 IC50 = 5400 nM T39716 CWA14L 53802926 IC50 > 6309.57 nM T39716 C28RDF 54746913 IC50 > 30000 nM T39716 CXEH21 56595883 IC50 = 1330 nM T39716 CSO3U5 56595888 IC50 = 541000 nM T39716 CY91VM 56595933 IC50 = 3300 nM T39716 CQ2J8B 56596030 IC50 = 2500 nM T39716 CY87LA 56596233 IC50 = 134000 nM T39716 CZ0K2U 56596475 IC50 = 215000 nM T39716 CXI5V1 56643481 IC50 > 5000 nM T39716 CH3BN6 56643486 IC50 > 5000 nM T39716 C6PUX9 56645570 IC50 > 30000 nM T39716 C6XI4W 56647652 IC50 > 5000 nM T39716 CG5T6R 56659661 IC50 > 33113.11 nM T39716 CUGJ21 56666584 IC50 > 33113.11 nM T39716 C39VWM 56676812 IC50 = 12022.64 nM T39716 C2LD6Y 56680137 IC50 = 4677.35 nM T39716 C5I4WJ 56680138 IC50 > 33113.11 nM T39716 CN5SE7 56683480 IC50 > 33113.11 nM T39716 C1IY0P 56944164 IC50 > 20000 nM T39716 CQT5I3 57328465 IC50 = 1260 nM T39716 CS1XE6 57328466 IC50 = 160 nM T39716 C4E1NK 57331209 IC50 > 30000 nM T39716 COUZ63 57494822 IC50 = 11102 nM T39716 C3N4MF 57520842 IC50 > 30000 nM T39716 CEL56T 57520942 IC50 > 30000 nM T39716 CR34CL 57582353 IC50 = 37000 nM T39716 C35GXV 57720515 EC50 = 29000 nM T39716 C09FAM 58044314 IC50 = 4000 nM T39716 CE3H1Q 58044315 IC50 > 10000 nM T39716 CZ28IJ 58044318 IC50 = 2500 nM T39716 CK0UY9 58044383 IC50 = 740000 nM T39716 CT4N2G 58044433 IC50 = 1903000 nM T39716 C2TRY9 58044589 IC50 = 1900 nM T39716 C0NFE7 58044606 IC50 = 981000 nM T39716 CF7PR9 58044619 IC50 = 3500 nM T39716 C9JCL7 58080768 IC50 = 10300 nM T39716 CRW9A3 58118918 IC50 = 102 nM T39716 C4FH0W 58118983 IC50 = 333 nM T39716 CCQM76 59153288 IC50 > 30000 nM T39716 CYF3R7 60167367 IC50 > 30000 nM T39716 C2D3HQ 60168069 IC50 > 100000 nM T39716 CSA3I9 60200914 IC50 = 1200 nM T39716 CK76WB 60200915 IC50 > 33000 nM T39716 CI40XK 60201083 IC50 = 19000 nM T39716 CNR41U 60201084 IC50 > 33000 nM T39716 CO5HD0 60201085 IC50 = 1200 nM T39716 CA57OQ 60201086 IC50 = 9700 nM T39716 C5UKQ8 60201087 IC50 = 25000 nM T39716 CA7NI3 60201088 IC50 > 16000 nM T39716 C56KOS 60201255 IC50 = 17000 nM T39716 C1YQ8J 60201256 IC50 > 25000 nM T39716 CVW28G 60201257 IC50 > 10000 nM T39716 CC82DM 65459349 IC50 = 27000 nM T39716 C6EJ3F 66551245 IC50 = 31622.78 nM T39716 C2LBW7 66551925 IC50 > 30000 nM T39716 CV7ZG3 66632452 IC50 = 3000 nM T39716 COTD35 66667669 IC50 = 11000 nM T39716 CD2HV3 66813354 IC50 > 31622.78 nM T39716 C78XLS 66813470 IC50 = 6309.57 nM T39716 CAOB97 66813557 IC50 = 3162.28 nM T39716 C89WUE 66813671 IC50 = 3981.07 nM T39716 CSY3F6 66813695 IC50 > 31622.78 nM T39716 CPK67V 66813703 IC50 > 31622.78 nM T39716 C7DX6Z 66813839 IC50 = 3981.07 nM T39716 CH2D5F 66813859 IC50 = 3162.28 nM T39716 C90OSR 66813870 IC50 = 7943.28 nM T39716 COZ0U9 66813914 IC50 = 6309.57 nM T39716 C5OTD2 66813927 IC50 = 5011.87 nM T39716 C39PEZ 66814019 IC50 = 3981.07 nM T39716 CG80RS 66814110 IC50 = 10000 nM T39716 C6QT5C 66849358 IC50 = 2221 nM T39716 CB2W9O 66849404 IC50 = 941 nM T39716 C7LOU6 66849415 IC50 = 8935 nM T39716 C4NZ5B 66849520 IC50 = 59 nM T39716 C6YC4U 66849571 IC50 = 887 nM T39716 CV9OX3 66849729 IC50 = 351 nM T39716 CWV2Z9 66849946 IC50 = 7541 nM T39716 CBQ5O1 67523614 IC50 = 1452 nM T39716 CM7AT3 67523656 IC50 = 1653 nM T39716 CB05ID 67972431 IC50 > 30000 nM T39716 CA7UZ6 68434755 IC50 > 30000 nM T39716 CBH6T3 69003776 IC50 = 14000 nM T39716 CXF5P9 69213151 IC50 = 1995.26 nM T39716 CP8XS4 70681040 IC50 = 360 nM T39716 CF85AB 70681063 IC50 = 120 nM T39716 C9LW7K 70681064 IC50 = 50 nM T39716 CX6UZ8 70681066 IC50 = 580 nM T39716 CS8V7G 70681068 IC50 = 150 nM T39716 CL28PN 70682458 IC50 = 10000 nM T39716 CJV64I 70683156 IC50 = 11800 nM T39716 C9BR3A 70683161 IC50 = 720 nM T39716 C36DYJ 70683164 IC50 = 2270 nM T39716 CN79ZX 70683165 IC50 = 780 nM T39716 CRXZ90 70683167 IC50 = 3000 nM T39716 C94GTH 70683168 IC50 = 460 nM T39716 C3ZY6F 70683178 IC50 = 50 nM T39716 C7NAV4 70683180 IC50 = 350 nM T39716 CN17AS 70683181 IC50 = 250 nM T39716 CA8VC6 70683182 IC50 = 130 nM T39716 C6QC5J 70683184 IC50 = 40 nM T39716 CK6JM8 70683187 IC50 = 60 nM T39716 CWK3H8 70683188 IC50 = 90 nM T39716 C1ARO8 70684544 IC50 = 6309.57 nM T39716 C3T1WM 70684545 IC50 > 31622.78 nM T39716 CIV4S6 70685239 IC50 = 1400 nM T39716 CLW68N 70685259 IC50 = 30 nM T39716 C65PTC 70685263 IC50 = 930 nM T39716 C2IDQ6 70685264 IC50 = 20 nM T39716 C02FWG 70685265 IC50 = 110 nM T39716 CO1ZR5 70685266 IC50 = 190 nM T39716 CRP7Z1 70685269 IC50 = 550 nM T39716 CRDJ83 70686683 IC50 = 19952.62 nM T39716 CEAK85 70687392 IC50 = 3700 nM T39716 CC32TO 70687393 IC50 = 1800 nM T39716 C0A3VH 70687418 IC50 = 40 nM T39716 CD2EW1 70688785 IC50 > 25118.86 nM T39716 C6YJL1 70689452 IC50 = 470 nM T39716 CO89VX 70689473 IC50 = 740 nM T39716 C56TAW 70689474 IC50 = 2700 nM T39716 CM3PD8 70689475 IC50 = 40 nM T39716 CV82BX 70690866 IC50 = 5011.87 nM T39716 C8R0SZ 70691558 IC50 = 590 nM T39716 CRXG05 70691559 IC50 = 1200 nM T39716 CYJ3F6 70691560 IC50 = 240 nM T39716 CK6I2V 70691577 IC50 = 80 nM T39716 C7ET5J 70691581 IC50 = 1570 nM T39716 CJ85NC 70691582 IC50 = 60 nM T39716 C27IPY 70691584 IC50 = 110 nM T39716 C8OKQ0 70693647 IC50 = 1700 nM T39716 CLN9F4 70693648 IC50 < 1000 nM T39716 CM3LU4 70693649 IC50 = 410 nM T39716 C3GVN0 70693667 IC50 = 200 nM T39716 CKP02Q 70693669 IC50 = 300 nM T39716 C6N3DT 70693670 IC50 = 2200 nM T39716 CEI84H 70693672 IC50 = 80 nM T39716 C6GCU1 70693673 IC50 = 30 nM T39716 CHUE45 70693674 IC50 = 80 nM T39716 CCQ49A 70695045 IC50 = 5011.87 nM T39716 CBCD89 70695046 IC50 = 5011.87 nM T39716 C63MTE 70695047 IC50 > 3162.28 nM T39716 CEK60M 70695761 IC50 = 500 nM T39716 CX6L3G 70695764 IC50 = 2000 nM T39716 CF4HZ3 70695774 IC50 = 120 nM T39716 CBHD70 70695780 IC50 = 140 nM T39716 CZL9G2 70695782 IC50 = 70 nM T39716 CKCE67 70695783 IC50 = 440 nM T39716 CUL37Y 70695784 IC50 = 90 nM T39716 C26OHM 70695785 IC50 = 20 nM T39716 CD1V2W 70695786 IC50 = 190 nM T39716 CBDL19 70792359 IC50 > 30000 nM T39716 CE9W1Z 70814180 IC50 = 6882 nM T39716 C7Z6HJ 70814238 IC50 = 8289 nM T39716 C7JD8A 70814244 IC50 = 9174 nM T39716 C1ST3M 70814308 IC50 = 4871 nM T39716 C5OT1G 70814333 IC50 = 9291 nM T39716 CLIH32 71226367 IC50 > 30000 nM T39716 C2FNI6 71259239 IC50 > 10000 nM T39716 CG0L7O 71259621 IC50 > 30000 nM T39716 C6BE5X 71271461 IC50 > 30000 nM T39716 CR4L9T 71449282 IC50 = 12589.25 nM T39716 CHF08N 71449283 IC50 = 6309.57 nM T39716 CMB7U1 71449284 IC50 = 6309.57 nM T39716 CVY54C 71449294 IC50 = 7943.28 nM T39716 C7L6QZ 71449295 IC50 > 31622.78 nM T39716 CIFE14 71451076 IC50 = 5011.87 nM T39716 CLSQ82 71451077 IC50 > 31622.78 nM T39716 C0RL3C 71451078 IC50 = 6309.57 nM T39716 CGJ7K0 71451084 IC50 = 19952.62 nM T39716 CI0B8V 71451085 IC50 = 1584.89 nM T39716 CXT57R 71452899 IC50 = 6309.57 nM T39716 CG21NF 71452900 IC50 > 31622.78 nM T39716 C7D9SN 71452907 IC50 > 31622.78 nM T39716 C5WU8L 71454670 IC50 = 5011.87 nM T39716 C7XQZ4 71454678 IC50 = 1000 nM T39716 CVU2O8 71454679 IC50 > 31622.78 nM T39716 C1X6TY 71456401 IC50 = 6309.57 nM T39716 C7AL1C 71456402 IC50 > 12589.25 nM T39716 CORH12 71456403 IC50 = 6309.57 nM T39716 C9FX5O 71456404 IC50 > 31622.78 nM T39716 CR4ZO3 71456412 IC50 = 794.33 nM T39716 CC3Q9J 71456413 IC50 = 2511.89 nM T39716 C7OW1B 71458245 IC50 > 31622.78 nM T39716 C6K4BO 71460096 IC50 > 31622.78 nM T39716 C9A7HP 71460097 IC50 > 31622.78 nM T39716 CYBR37 71460098 IC50 = 3162.28 nM T39716 CQW3L4 71460099 IC50 = 19952.62 nM T39716 CSB76D 71460108 IC50 = 1584.89 nM T39716 CQ30OU 71461829 IC50 > 31622.78 nM T39716 CV7ML5 71461830 IC50 = 10000 nM T39716 CA07TC 71517197 IC50 > 33000 nM T39716 CE60RK 71521279 IC50 = 4800 nM T39716 C5IK7D 71521280 IC50 = 5900 nM T39716 C2MC6B 71522734 IC50 > 10000 nM T39716 CM1B0W 71523649 IC50 = 36000 nM T39716 CHAU76 71555980 IC50 > 30000 nM T39716 C3EC1H 71557026 IC50 > 10000 nM T39716 CL85YK 71557177 IC50 > 10000 nM T39716 CY59CA 71557630 IC50 = 5200 nM T39716 CTI52S 71557789 IC50 > 10000 nM T39716 CO09GI 71558118 IC50 > 10000 nM T39716 CMKH30 71558122 IC50 > 10000 nM T39716 C48RIB 71558271 IC50 > 10000 nM T39716 CK2HF0 71558274 IC50 > 10000 nM T39716 CUI6M5 71558468 IC50 > 10000 nM T39716 C0DO9Y 71558578 IC50 > 10000 nM T39716 C2ZN4G 71558725 IC50 > 10000 nM T39716 CIDS01 71558883 IC50 > 10000 nM T39716 CY6Z1T 71558917 IC50 = 230 nM T39716 CHRO29 71558920 IC50 > 10000 nM T39716 C9WGA1 71559034 IC50 > 10000 nM T39716 C20ELR 71559363 IC50 > 10000 nM T39716 CJXK67 71559365 IC50 > 1000 nM T39716 CLAZ62 71585735 IC50 > 30000 nM T39716 CRC01X 71585929 IC50 = 5100 nM T39716 CXA29H 71585930 IC50 = 12000 nM T39716 CPI61F 71586033 IC50 > 30000 nM T39716 C4U3GM 71586128 IC50 > 30000 nM T39716 CNY52I 71586326 IC50 = 27000 nM T39716 C9J0EH 71603917 IC50 > 30000 nM T39716 C5LM0G 71711363 IC50 = 610 nM T39716 C1VC7P 71711696 IC50 = 4600 nM T39716 C8D7FJ 71711834 IC50 > 10000 nM T39716 CD4Z0Y 71711979 IC50 = 320 nM T39716 CK0L1B 71712241 IC50 > 10000 nM T39716 CZ5PL8 71716262 IC50 > 10000 nM T39716 C31BYG 71716276 IC50 > 30000 nM T39716 CC4A3K 71716821 IC50 = 43699 nM T39716 C7EG3T 71716825 IC50 = 25448 nM T39716 C9MUK3 71716856 IC50 = 15060 nM T39716 CUG2V3 71716866 IC50 > 30000 nM T39716 CIZ40M 71716873 IC50 > 10000 nM T39716 C4XYN9 71717494 IC50 = 22451 nM T39716 C0TK9Q 71718072 IC50 > 10000 nM T39716 C89GSF 71718127 IC50 > 30000 nM T39716 C7TM8H 71718630 IC50 > 10000 nM T39716 CW38FM 71718726 IC50 = 22210 nM T39716 CY6D2J 71719903 IC50 = 25786 nM T39716 CL0O5N 71719912 IC50 = 25231 nM T39716 CYQH30 71719914 IC50 > 30000 nM T39716 CMDI34 71720470 IC50 = 25578 nM T39716 C7B8UH 71720543 IC50 > 10000 nM T39716 C30NBJ 71722055 IC50 > 30000 nM T39716 C2QT3H 71812413 IC50 > 30000 nM T39716 CZPJ89 71812414 IC50 > 30000 nM T39716 CU1KS7 71812606 IC50 = 4000 nM T39716 CRAB14 71812607 IC50 = 11000 nM T39716 CQD1F2 71812796 IC50 = 24000 nM T39716 C2UOA5 71812797 IC50 = 28000 nM T39716 C9NK1C 71812798 IC50 > 30000 nM T39716 C3RE7M 71812799 IC50 > 30000 nM T39716 CW20HQ 71818431 IC50 = 50000 nM T39716 C2L7TX 71818575 IC50 = 3300 nM T39716 CYMS42 72545669 IC50 = 1070 nM T39716 C29YGC 72712370 IC50 = 9000 nM T39716 CCEX08 72949434 IC50 = 7200 nM T39716 C2E7QW 75201901 IC50 = 1100 nM T39716 C7OE1X 76309796 IC50 > 30000 nM T39716 CBH4N7 76309797 IC50 = 21000 nM T39716 C10UTF 76310404 IC50 > 30000 nM T39716 C6T1NV 76310406 IC50 > 30000 nM T39716 CC4BK5 76310408 IC50 = 20000 nM T39716 C8M7RN 76310409 IC50 > 30000 nM T39716 CHFC49 76313502 IC50 > 30000 nM T39716 C1PM7H 76314065 IC50 = 20000 nM T39716 CBK0T8 76314067 IC50 > 30000 nM T39716 C20ILA 76314069 IC50 > 30000 nM T39716 C8OQT1 76314070 IC50 = 27000 nM T39716 CNM4K0 76317019 IC50 > 30000 nM T39716 C32OSF 76317020 IC50 > 30000 nM T39716 CKG5A9 76317629 IC50 > 30000 nM T39716 CQ7JK4 76317631 IC50 > 30000 nM T39716 CT2R5J 76320732 IC50 > 30000 nM T39716 CVP8U9 76320733 IC50 > 30000 nM T39716 C2RJW0 76320734 IC50 > 30000 nM T39716 CY8NT4 76321352 IC50 > 30000 nM T39716 CRU30A 76321353 IC50 > 30000 nM T39716 CNY2D6 76321910 EC50 = 30000 nM T39716 CR05PL 76322043 IC50 > 30000 nM T39716 CQ3CW1 76322044 IC50 > 30000 nM T39716 C46MFT 76324385 IC50 > 30000 nM T39716 C4W1NV 76324386 IC50 = 20000 nM T39716 CJF20G 76324950 IC50 > 30000 nM T39716 CP3UI7 76327945 IC50 > 30000 nM T39716 CNY5X1 76328517 IC50 > 30000 nM T39716 CX54MA 76328518 IC50 > 30000 nM T39716 CINA95 76331591 IC50 > 30000 nM T39716 CCXK29 76332197 IC50 > 30000 nM T39716 CH4K7Q 76332198 IC50 > 30000 nM T39716 C4WO6Y 76332199 IC50 > 30000 nM T39716 CK47NO 76332200 IC50 > 30000 nM T39716 CANB89 76332201 IC50 > 30000 nM T39716 CO2N7R 76335221 IC50 > 30000 nM T39716 C05RSQ 76335223 IC50 > 30000 nM T39716 C8ND6L 76335224 IC50 = 21000 nM T39716 CUO84S 76335833 IC50 > 30000 nM T39716 C92WBQ 76336500 IC50 = 5600 nM T39716 C34TAM 77845572 IC50 > 30000 nM T39716 C2NCH9 78318214 IC50 > 30000 nM T39716 C2GET7 78318815 IC50 > 30000 nM T39716 C15BSO 86270136 IC50 = 265 nM T39716 CZL23E 86271138 IC50 > 30000 nM T39716 C7J9FE 86687346 IC50 = 21000 nM T39716 C0OTF5 86687356 IC50 = 21000 nM T39716 C50EDA 86687482 IC50 > 30000 nM T39716 CEQ0C1 86687530 IC50 > 30000 nM T39716 CTG76E 86687532 IC50 = 16000 nM T39716 CQN21C 86687557 IC50 > 30000 nM T39716 CFT89Y 86687602 IC50 = 1500 nM T39716 CY8JW3 86687604 IC50 > 10000 nM T39716 C7OXV8 86687606 IC50 > 10000 nM T39716 C63MCA 86687768 IC50 = 4750 nM T39716 CRJ9F2 86699098 IC50 > 10000 nM T39716 C4ZPG9 87178530 IC50 = 123 nM T39716 CHU2Z5 87178553 IC50 = 1647 nM T39716 CJ2OI4 87178572 IC50 = 211 nM T39716 CRHC58 87178657 IC50 = 281 nM T39716 CEH51J 87178674 IC50 = 166 nM T39716 C4FJ5M 87206909 IC50 = 397 nM T39716 CJC29A 89544489 IC50 > 10000 nM T39716 COK7U5 89545491 IC50 > 10000 nM T39716 CAM65C 89545507 IC50 > 10000 nM T39716 CMZ8P5 89545670 IC50 = 2600 nM T39716 C74SBC 89555961 IC50 > 10000 nM T39716 C01NKB 89555963 IC50 > 10000 nM T39716 C29LHS 89556026 IC50 > 10000 nM T39716 CXHC49 89556028 IC50 > 10000 nM T39716 CJRK20 89556063 IC50 > 10000 nM T39716 CH6AT7 89556066 IC50 = 5900 nM T39716 C9AMI1 89556077 IC50 > 10000 nM T39716 C72BSC 89556129 IC50 > 10000 nM T39716 CP8X3E 89573118 IC50 > 10000 nM T39716 C47HED 89583208 IC50 > 10000 nM T39716 CM6SL8 89613863 IC50 > 30000 nM T39716 CK8O4U 89614559 IC50 = 23000 nM T39716 C90UQK 89614650 IC50 > 30000 nM T39716 CQK1S9 89614770 IC50 > 30000 nM T39716 CV7UN4 89761281 IC50 = 1500 nM T39716 C7PT4Z 89761284 IC50 = 14000 nM T39716 CAO3I6 89761608 IC50 = 650 nM T39716 C29BFD 89761642 IC50 > 30000 nM T39716 CGI6O0 89761704 IC50 = 2100 nM T39716 C8IJ0Y 89761742 IC50 = 1500 nM T39716 C4BQC6 89761777 IC50 > 30000 nM T39716 COU52N 89761779 IC50 = 2000 nM T39716 C95IFK 89761981 IC50 > 30000 nM T39716 C48RCZ 90021555 IC50 = 1200 nM T39716 C1BIF8 90026208 IC50 = 50 nM T39716 C26LKW 90341025 IC50 > 30000 nM T39716 COYC71 90700276 IC50 = 1186 nM T39716 CN07GH 90846203 IC50 = 217 nM T39716 CX85KF 91134217 IC50 = 17810 nM T39716 C26BZK 91666633 IC50 = 110 nM T39716 C9ETC1 91666645 IC50 > 30000 nM T39716 C0S3JN 91799666 IC50 = 7200 nM T39716 C7NLE8 91809347 IC50 = 49 nM T39716 CTS64R 91809389 IC50 = 22000 nM T39716 CXN69G 100657083 IC50 = 1300 nM T39716 CQ9PN8 102593934 IC50 > 100000 nM T39716 CNFW42 117608566 IC50 = 1313 nM T39716 CC5N9I 117737142 IC50 > 14000 nM T39716 C4NH6M 117740584 IC50 > 10000 nM T39716 CC1A0T 117741702 IC50 > 10000 nM T39716 C3C2YG 117741784 IC50 > 10000 nM T39716 C4ZO0A 117741876 IC50 > 10000 nM T39716 C10BKY 117749324 IC50 > 30000 nM T39716 COVX65 117753917 IC50 > 10000 nM T39716 CS5X4R 117753922 IC50 = 140 nM T39716 CQK1U5 117753939 IC50 = 820 nM T39716 CW8RS3 117760464 IC50 > 30000 nM T39716 C3P1LN 117789501 IC50 = 419 nM T39716 CK0RV9 117993874 IC50 = 18000 nM T39716 CL4O0J 117993881 IC50 = 18800 nM T39716 CB8I3S 117993884 IC50 = 11000 nM T39716 C92RVJ 117993886 IC50 = 6000 nM T39716 CM2H5Q 117993976 IC50 = 2350 nM T39716 C9KV7L 117993993 IC50 = 6900 nM T39716 CNV24M 117993998 IC50 > 30000 nM T39716 C8DSV0 117994021 IC50 = 21000 nM T39716 C57PMF 118002063 IC50 = 32000 nM T39716 CT8C0X 118109014 IC50 = 5700 nM T39716 COH9J3 118109161 IC50 > 30000 nM T39716 CG3M4J 118109168 IC50 = 19000 nM T39716 CO6KX7 118109201 IC50 > 30000 nM T39716 CAU5T9 118109234 IC50 > 30000 nM T39716 CT4ZN7 118109256 IC50 > 30000 nM T39716 CG8FJ5 118109302 IC50 > 30000 nM T39716 C8OAL5 118109304 IC50 > 30000 nM T39716 C3N0KS 118109319 IC50 = 24200 nM T39716 CU85FO 118109356 IC50 = 1900 nM T39716 CWJ7T6 118109371 IC50 = 17600 nM T39716 CS0B7V 118112295 IC50 > 30000 nM T39716 CWR6I1 118112300 IC50 = 2.2 nM T39716 CXY23I 118121135 IC50 > 30000 nM T39716 CB4I7H 118121139 IC50 = 22500 nM T39716 C7AYV5 118540795 IC50 = 2000 nM T39716 CKA2F8 118554582 IC50 > 3000 nM T39716 C2O7GE 118707553 IC50 > 33000 nM T39716 C8S9VW 118707562 IC50 > 33000 nM T39716 CR8TX9 118708662 IC50 = 79 nM T39716 CMDN36 118710321 IC50 = 9716 nM T39716 CPL32R 118710322 IC50 = 12875 nM T39716 CA79ZM 118710323 IC50 > 30000 nM T39716 CLS68B 118710324 IC50 = 947 nM T39716 CL2PK9 118710325 IC50 = 7240 nM T39716 CDO95Z 118710326 IC50 = 572 nM T39716 CG7X9J 118710327 IC50 = 934 nM T39716 C83LIE 118710328 IC50 = 1329 nM T39716 CH29DT 118711022 IC50 = 24700 nM T39716 C3BQM2 118714771 IC50 = 181 nM T39716 CPVC71 118714772 IC50 = 340 nM T39716 CEB6T7 118714773 IC50 = 2216 nM T39716 C65NKL 118714774 IC50 = 358 nM T39716 C39NSR 118714775 IC50 = 3261 nM T39716 CJ8E7U 118714776 IC50 = 519 nM T39716 C84KNW 118714777 IC50 = 30000 nM T39716 CHS5K3 118714778 IC50 = 3069 nM T39716 C58YHZ 118714779 IC50 = 2450 nM T39716 CF2YQ4 118714780 IC50 = 30000 nM T39716 C40SOZ 118714781 IC50 = 1138 nM T39716 C67FSV 118714782 IC50 = 118 nM T39716 CREM47 118714783 IC50 = 1732 nM T39716 CX4I5Q 118714784 IC50 = 2811 nM T39716 CC56DO 118718808 IC50 > 30000 nM T39716 C69PLO 118734433 IC50 > 5000 nM T39716 C2NAE8 118734434 IC50 > 5000 nM T39716 CD4B5E 118734435 IC50 > 5000 nM T39716 C91PCO 118734436 IC50 > 5000 nM T39716 CM2Y6W 118734437 IC50 = 27000 nM T39716 CFL60J 118734438 IC50 > 5000 nM T39716 CQ0R3E 118734439 IC50 > 5000 nM T39716 CY8A1T 118734440 IC50 > 5000 nM T39716 CFRZ45 118734441 IC50 > 5000 nM T39716 C3ZJ0K 118734442 IC50 > 5000 nM T39716 CI30YK 118734443 IC50 > 5000 nM T39716 CUAQ60 118734444 IC50 > 5000 nM T39716 CFNR84 118734445 IC50 > 5000 nM T39716 CK12TX 118734446 IC50 > 20000 nM T39716 C09BDT 118734447 IC50 > 20000 nM T39716 C6F9BI 118734448 IC50 > 5000 nM T39716 C8ZLX9 118734449 IC50 > 20000 nM T39716 C01BNE 118734450 IC50 > 5000 nM T39716 CI0FE2 118734451 IC50 > 4700 nM T39716 C1CED0 118734452 IC50 > 5000 nM T39716 C8NBL5 118734453 IC50 > 5000 nM T39716 C0CY2K 118734454 IC50 > 5000 nM T39716 CTR7O8 118734455 IC50 > 5000 nM T39716 CZQD84 118734456 IC50 > 5000 nM T39716 CGBF25 118734457 IC50 > 5000 nM T39716 C6I8HF 118734458 IC50 > 5000 nM T39716 C5G7DQ 118734459 IC50 > 5000 nM T39716 CVW15D 118734460 IC50 > 5000 nM T39716 CSE60C 118734461 IC50 > 5000 nM T39716 CO4U1R 118734462 IC50 > 10000 nM T39716 CA95IF 118734463 IC50 > 10000 nM T39716 C14ILF 118734464 IC50 > 10000 nM T39716 C3TOV9 118734465 IC50 > 10000 nM T39716 C2RO8T 118734466 IC50 > 10000 nM T39716 CSP25D 118734467 IC50 > 10000 nM T39716 CJD80C 118734468 IC50 > 10000 nM T39716 C06TAI 118734469 IC50 > 10000 nM T39716 CBY5M0 118734470 IC50 > 10000 nM T39716 CHO8I3 118734471 IC50 = 3500 nM T39716 C38BCH 118734472 IC50 > 10000 nM T39716 CV7UH5 118734473 IC50 > 10000 nM T39716 C6SEA7 118734474 IC50 > 10000 nM T39716 CO7DP2 118734475 IC50 = 2100 nM T39716 CX2R0E 118734476 IC50 = 1100 nM T39716 C16AEK 118734477 IC50 > 10000 nM T39716 CO1UF9 118734478 IC50 = 2800 nM T39716 C16AUM 118734479 IC50 = 3000 nM T39716 CI2P1V 118734480 IC50 > 10000 nM T39716 C1Z8AN 118734481 IC50 = 3400 nM T39716 CYD8N6 118734482 IC50 = 400 nM T39716 CW05LY 118734483 IC50 > 10000 nM T39716 CN01US 118734484 IC50 > 10000 nM T39716 C3E7GP 118734485 IC50 > 10000 nM T39716 CCA41Z 118734486 IC50 > 10000 nM T39716 CM2QS5 118734487 IC50 = 3600 nM T39716 C3T1QC 118734488 IC50 = 4600 nM T39716 CM6Y8X 118734489 IC50 = 500 nM T39716 C93LMC 118734490 IC50 > 10000 nM T39716 C8LHA3 118734491 IC50 = 4500 nM T39716 C26ADB 118734547 IC50 = 8800 nM T39716 C82UBF 118734548 IC50 > 10000 nM T39716 CO4KD2 118734549 IC50 > 10000 nM T39716 CX6L4C 118734550 IC50 > 10000 nM T39716 C5JNX2 118734551 IC50 > 10000 nM T39716 C0UJ8Q 118734552 IC50 > 10000 nM T39716 CJDP52 118734553 IC50 > 10000 nM T39716 CM59EQ 118917669 IC50 > 100000 nM T39716 C6J8YF 118917671 IC50 > 30000 nM T39716 C0RFQ5 118937646 IC50 = 14200 nM T39716 CTR37C 118937656 IC50 > 33000 nM T39716 CTC20B 118937664 IC50 = 19000 nM T39716 CR9Y6M 118937702 IC50 = 3100 nM T39716 C1Y7MU 118937716 IC50 = 23000 nM T39716 C9JL4Y 118937760 IC50 > 33000 nM T39716 CXI1F9 118937849 IC50 > 33000 nM T39716 CWL1S3 118937903 IC50 > 33000 nM T39716 CXZ43S 118937913 IC50 = 5000 nM T39716 CMQB61 118937925 IC50 = 15000 nM T39716 CU4CW1 121313969 IC50 > 30000 nM T39716 C9H0BR 121333853 IC50 > 10000 nM T39716 CGH4B7 121333855 IC50 > 10000 nM T39716 CZ3X9J 121333858 IC50 > 10000 nM T39716 CT4FA9 121333871 IC50 > 10000 nM T39716 CIQ8C0 121333899 IC50 > 10000 nM T39716 C83STC 121333902 IC50 > 10000 nM T39716 CMA2O3 121333930 IC50 > 10000 nM T39716 C9Q2ND 121333973 IC50 = 12000 nM T39716 CO9SQ6 121454909 IC50 > 30000 nM T39716 CH0X4Z 121454982 IC50 > 30000 nM T39716 CT0KS4 121455652 IC50 > 30000 nM T39716 CW35TI 121455794 IC50 > 30000 nM T39716 CHD26A 121596332 IC50 > 33300 nM T39716 CNGQ19 122179477 IC50 > 30000 nM T39716 C1XKA8 122191834 IC50 > 30000 nM T39716 CHPL50 122194669 IC50 = 4400 nM T39716 CWSA14 122194670 IC50 = 2800 nM T39716 C05AUF 122194671 IC50 = 5600 nM T39716 CY2B6W 122194672 IC50 = 3000 nM T39716 CP38IW 122194673 IC50 = 6100 nM T39716 CWGY65 122194675 IC50 = 1100 nM T39716 C1MH8Y 122194676 IC50 = 3400 nM T39716 CP4L5A 122194677 IC50 = 16000 nM T39716 CW3D9H 122196008 IC50 = 20000 nM T39716 C5G9FH 122196009 IC50 = 7000 nM T39716 C2RBF4 122196010 IC50 = 17000 nM T39716 C0R8OS 122196011 IC50 = 18000 nM T39716 C61QNK 122196012 IC50 > 33000 nM T39716 CZ2HR6 122196013 IC50 = 5200 nM T39716 C6W5IA 122196014 IC50 = 3400 nM T39716 CKEH54 122196015 IC50 = 33000 nM T39716 C38XFL 122196016 IC50 = 24000 nM T39716 CLQ8O5 122196017 IC50 = 4900 nM T39716 C82UNL 122196018 IC50 = 1900 nM T39716 C0KG7Z 122196019 IC50 = 3700 nM T39716 CS0W4O 122196020 IC50 = 1200 nM T39716 CK8FH3 122196021 IC50 = 38000 nM T39716 C9N1CF 122196022 IC50 = 77000 nM T39716 CR4JT9 122196023 IC50 = 10000 nM T39716 C80OZQ 122196024 IC50 = 13000 nM T39716 CT9N7O 122196025 IC50 = 7100 nM T39716 C3B0RY 122422350 IC50 = 2500 nM T39716 C81EPB 122422402 IC50 = 23700 nM T39716 CC2TE4 122422536 IC50 = 16100 nM T39716 CEGS87 122513481 IC50 = 16400 nM T39716 C9K5RV 122513516 IC50 > 33000 nM T39716 CC1J0T 122591381 IC50 > 30000 nM T39716 C1YK2E 122678192 IC50 > 33000 nM T39716 C4D9QY 127026491 IC50 > 30000 nM T39716 C7L1DB 127037832 IC50 > 30000 nM T39716 CB98DL 127044262 IC50 = 7915 nM T39716 CZF2X5 127044562 IC50 = 5052 nM T39716 C4WEA5 127044563 IC50 = 425 nM T39716 C5J3AM 127044564 IC50 = 417 nM T39716 CE7MG6 127044736 IC50 > 10000 nM T39716 CMF6K2 127044897 IC50 = 353 nM T39716 CJC30T 127044898 IC50 = 3345 nM T39716 CXEZ15 127044899 IC50 = 1512 nM T39716 CYVO30 127045496 IC50 = 901 nM T39716 C7JT8V 127045799 IC50 > 5000 nM T39716 CH2Z3S 127045806 IC50 > 5000 nM T39716 CSJD60 127045808 IC50 > 4800 nM T39716 COWD91 127045811 IC50 > 10000 nM T39716 C90JPN 127045813 IC50 > 5000 nM T39716 C21JCE 127045825 IC50 > 5000 nM T39716 CNF0G1 127045829 IC50 > 5000 nM T39716 CC9TY3 127045830 IC50 > 5000 nM T39716 CDC0M9 127046018 IC50 > 5000 nM T39716 C74SHI 127046022 IC50 > 5000 nM T39716 CH0CD1 127046023 IC50 > 5000 nM T39716 CPX1F0 127046025 IC50 > 5000 nM T39716 CAVD37 127046026 IC50 > 5000 nM T39716 C8UW6X 127046032 IC50 = 900 nM T39716 CMPZ51 127046033 IC50 > 5000 nM T39716 CY5J0R 127046039 IC50 > 5000 nM T39716 CBQ47D 127046045 IC50 > 5000 nM T39716 C6NVQ1 127046047 IC50 > 5000 nM T39716 C4MU2J 127046230 IC50 > 5000 nM T39716 CGYE23 127046231 IC50 > 5000 nM T39716 C69GBJ 127046239 IC50 > 5000 nM T39716 CM1IH3 127046241 IC50 > 5000 nM T39716 C4L1VA 127046242 IC50 > 5000 nM T39716 CWN2J7 127046243 IC50 > 5000 nM T39716 CI1VA2 127046252 IC50 = 15900 nM T39716 CE67AD 127046253 IC50 = 1000 nM T39716 C53RIX 127046257 IC50 > 5000 nM T39716 COK9Z3 127046259 IC50 > 5000 nM T39716 CL5VY9 127046359 IC50 = 1800 nM T39716 C3M6YT 127046415 IC50 > 5000 nM T39716 C90HYR 127046420 IC50 > 5000 nM T39716 C8BES0 127046422 IC50 > 10000 nM T39716 C2EI4Q 127046423 IC50 = 37900 nM T39716 CM2HB0 127046424 IC50 > 5000 nM T39716 CM5D6J 127046425 IC50 > 5000 nM T39716 C9LH4U 127046428 IC50 > 5000 nM T39716 C20KGH 127046429 IC50 > 5000 nM T39716 CH27MP 127046433 IC50 > 5000 nM T39716 CWH7Y0 127046434 IC50 > 5000 nM T39716 C1CV8E 127046436 IC50 > 5000 nM T39716 C87YLU 127046583 IC50 > 5000 nM T39716 C74ELB 127046587 IC50 > 5000 nM T39716 CI9XY7 127046589 IC50 > 5000 nM T39716 CQ3EV4 127046592 IC50 > 5000 nM T39716 C8PO4C 127046597 IC50 = 22700 nM T39716 C31XHN 127046598 IC50 > 5000 nM T39716 CFSH84 127046606 IC50 > 5000 nM T39716 CP8T2D 127046764 IC50 > 5000 nM T39716 C0A7SK 127046767 IC50 > 5000 nM T39716 CC2Y1J 127046770 IC50 > 5000 nM T39716 C1XON9 127046774 IC50 > 5000 nM T39716 C80RLU 127046781 IC50 > 5000 nM T39716 C34GAN 127046799 IC50 = 2000 nM T39716 CCXR80 127046802 IC50 = 3400 nM T39716 CSKX63 127046908 IC50 > 5000 nM T39716 CVUW94 127046909 IC50 = 3200 nM T39716 C02HPV 127046912 IC50 > 2700 nM T39716 C8CK6P 127046914 IC50 > 5000 nM T39716 C3CSI0 127046916 IC50 = 4500 nM T39716 C4X2OU 127046919 IC50 > 5000 nM T39716 CL9W8T 127046920 IC50 > 5000 nM T39716 CLH51Y 127046923 IC50 > 5000 nM T39716 CXMC23 127046930 IC50 > 5000 nM T39716 CB9EF5 127046932 IC50 > 4800 nM T39716 CZ7G6T 127047057 IC50 > 5000 nM T39716 CND20E 127047062 IC50 > 5000 nM T39716 CNSZ83 127047063 IC50 > 5000 nM T39716 C1R4VN 127047068 IC50 > 5000 nM T39716 C5VU7H 127047069 IC50 > 5000 nM T39716 CFG94A 127047073 IC50 > 5000 nM T39716 CF5D0S 127047074 IC50 > 5000 nM T39716 C0XS7B 127047075 IC50 > 5000 nM T39716 CI60KD 127047206 IC50 > 10000 nM T39716 CA7YG4 127047208 IC50 > 5000 nM T39716 CXT5Y0 127047216 IC50 > 5000 nM T39716 CY8RH9 127047220 IC50 > 5000 nM T39716 CV4OB1 127047223 IC50 > 5000 nM T39716 C1RD6X 127047251 IC50 = 4400 nM T39716 CZLT12 127047252 IC50 = 2500 nM T39716 CFPJ73 127047320 IC50 > 5000 nM T39716 C3JK6P 127047322 IC50 > 5000 nM T39716 C1T5PC 127047323 IC50 > 5000 nM T39716 C28REX 127047327 IC50 > 5000 nM T39716 CVSF19 127047330 IC50 > 5000 nM T39716 C0IO2K 127047331 IC50 > 5000 nM T39716 C9SIK3 127047333 IC50 > 5000 nM T39716 CKD78E 127047346 IC50 = 3600 nM T39716 C5DO7I 127047347 IC50 > 5000 nM T39716 CM5TX2 127047468 IC50 > 5000 nM T39716 C54TRJ 127047469 IC50 > 5000 nM T39716 C3K5YI 127047471 IC50 > 5000 nM T39716 C2M5JH 127047472 IC50 > 5000 nM T39716 C3SLJ4 127047473 IC50 > 5000 nM T39716 CCA51M 127047474 IC50 = 7800 nM T39716 C6EM0G 127047476 IC50 > 5000 nM T39716 C5RKB7 127047479 IC50 > 4700 nM T39716 C96VDX 127047480 IC50 > 5000 nM T39716 CJ7IQ4 127047485 IC50 > 4000 nM T39716 CZKB91 127047487 IC50 > 5000 nM T39716 C7OTX3 127047488 IC50 > 5000 nM T39716 CVR95B 127047489 IC50 > 5000 nM T39716 CW8P5Y 127047613 IC50 > 5000 nM T39716 C0WXP3 127047615 IC50 > 5000 nM T39716 C1RK5C 127047619 IC50 > 5000 nM T39716 C9QZH7 127047622 IC50 > 5000 nM T39716 CJ31BC 127047628 IC50 > 5000 nM T39716 C9MXK5 127047633 IC50 > 5000 nM T39716 CB16MW 127047643 IC50 = 1000 nM T39716 C09QIY 127047645 IC50 = 2800 nM T39716 C5S1AI 127047646 IC50 = 5100 nM T39716 C1ULZ3 127047735 IC50 > 5000 nM T39716 C4T5WS 127047736 IC50 > 5000 nM T39716 CQ45AO 127047757 IC50 > 5000 nM T39716 CG5X0Y 127047758 IC50 = 5000 nM T39716 CTRE63 127047854 IC50 > 5000 nM T39716 CDGS14 127047866 IC50 > 5000 nM T39716 C16NUB 127047867 IC50 > 5000 nM T39716 CG52RP 127047873 IC50 > 5000 nM T39716 C8PWL6 127047983 IC50 > 5000 nM T39716 CGW63M 127047988 IC50 > 5000 nM T39716 CR6AB0 127047989 IC50 > 5000 nM T39716 CK9ZO8 127047990 IC50 > 5000 nM T39716 CQ2SO8 127047999 IC50 > 10000 nM T39716 C2D9LN 127048108 IC50 > 10000 nM T39716 C25GJD 127048113 IC50 = 3400 nM T39716 C4VID9 127048115 IC50 > 5000 nM T39716 CCI81A 127048120 IC50 > 5000 nM T39716 CE1Z4W 127048121 IC50 = 3400 nM T39716 CI0P1M 127048127 IC50 > 5000 nM T39716 C4CUP9 127048128 IC50 > 5000 nM T39716 C7HGD0 127048130 IC50 > 5000 nM T39716 C4LK6A 127048137 IC50 > 5000 nM T39716 CNA30T 127048138 IC50 > 5000 nM T39716 C38WDU 129012089 IC50 = 13000 nM T39716 C4Z5MQ 131839619 IC50 > 30000 nM T39716 C4A2JF 132020399 IC50 = 15105 nM T39716 C9C5PT 132020406 IC50 > 30000 nM T39716 COH0K2 132020407 IC50 = 18000 nM T39716 CX6WL3 132020408 IC50 > 30000 nM T39716 CABH81 132020419 IC50 > 30000 nM T39716 C79BLN 132020421 IC50 = 6300 nM T39716 CZ5H2B 132020452 IC50 = 18347 nM T39716 CNK15D 132020464 IC50 = 16000 nM T39716 CMD5X6 132020466 IC50 = 14000 nM T39716 C4FPR1 132020468 IC50 > 30000 nM T39716 CTRG94 132020475 IC50 > 30000 nM T39716 C76RHU 132020480 IC50 = 8600 nM T39716 C6ME9R 132020486 IC50 = 24000 nM T39716 C69ELN 132020488 IC50 = 1700 nM T39716 CIM31O 132020491 IC50 = 5700 nM T39716 CB74IC 132020507 IC50 = 12000 nM T39716 C4JP3T 132020512 IC50 > 30000 nM T39716 CDL95F 132020518 IC50 = 20000 nM T39716 CUZ03K 132020526 IC50 = 9666 nM T39716 CD4HS0 132020533 IC50 = 3900 nM T39716 C5LYQ6 132020541 IC50 = 30000 nM T39716 C5G1PQ 132020544 IC50 = 8400 nM T39716 CAZI64 132020570 IC50 = 3697 nM T39716 CTC7E3 132020571 IC50 = 6508 nM T39716 CP8A1Q 132020575 IC50 = 16000 nM T39716 C7ZIP5 132020580 IC50 = 7500 nM T39716 CLV79P 132020582 IC50 = 5100 nM T39716 CF2QM1 132020584 IC50 = 7200 nM T39716 CM42HK 132020589 IC50 > 30000 nM T39716 C21QHW 132051336 IC50 = 18000 nM T39716 C9RBP0 132051461 IC50 > 30000 nM T39716 CVFK13 132051462 IC50 > 30000 nM T39716 CNZA27 132051626 IC50 > 30000 nM T39716 CHL97M 132051650 IC50 = 11000 nM T39716 C83UBM 132051677 IC50 = 3800 nM T39716 CG1S2M 132519335 IC50 = 13000 nM T39716 CO2SH1 132519336 IC50 = 13000 nM T39716 CO1RW6 134132142 IC50 = 9134 nM T39716 CF2M4S 134132899 IC50 = 21000 nM T39716 C1M8ZR 134133921 IC50 > 30000 nM T39716 CJOQ95 134134229 IC50 > 30000 nM T39716 CC7OQ2 134135307 IC50 > 30000 nM T39716 CE5TV4 134135453 IC50 = 21000 nM T39716 CN7RI4 134146511 IC50 > 30000 nM T39716 CA5B2J 134150245 IC50 = 17430 nM T39716 COPA84 134151189 IC50 > 30000 nM T39716 CA49BH 134156727 IC50 = 27000 nM T39716 CFR87X 134477051 IC50 = 74 nM T39716 CFYC29 134477061 IC50 > 30000 nM T39716 C20QBE 134477062 IC50 = 1900 nM T39716 CT58HM 134477070 IC50 > 30000 nM T39716 C8W9YN 134477076 IC50 = 108 nM T39716 CX5MS3 134477080 IC50 = 50 nM T39716 CSO3Q9 134477081 IC50 = 37 nM T39716 CAED75 134477093 IC50 > 30000 nM T39716 CO15IT 134477094 IC50 > 30000 nM T39716 C0Q1MD 134477108 IC50 > 30000 nM T39716 CX64SG 134477133 IC50 > 30000 nM T39716 CT7J4U 134477136 IC50 > 30000 nM T39716 C51SKX 134477137 IC50 = 120 nM T39716 CCVX65 134477139 IC50 = 156 nM T39716 C03SFG 134477143 IC50 > 30000 nM T39716 C70XMC 134477147 IC50 > 30000 nM T39716 C7JM1E 134477177 IC50 = 5100 nM T39716 C4LS2A 134477178 IC50 = 2600 nM T39716 CNU8M6 134477183 IC50 = 133 nM T39716 CK9SR3 134477213 IC50 = 127 nM T39716 C9WN3E 134477214 IC50 = 4900 nM T39716 C9IB8P 134477217 IC50 > 30000 nM T39716 C1AB5Q 134477222 IC50 = 189 nM T39716 CN37XZ 134477224 IC50 > 30000 nM T39716 CR39TS 134477260 IC50 > 30000 nM T39716 C9O5FS 134477264 IC50 = 237 nM T39716 CS5ME8 134477268 IC50 = 150 nM T39716 CC0OF9 134477275 IC50 = 188 nM T39716 C1R9DV 134477283 IC50 > 30000 nM T39716 CMH4G1 135412290 IC50 = 1200 nM T39716 CB1VD9 135426471 IC50 = 300 nM T39716 CZ6WT3 135469086 IC50 = 19700 nM T39716 CY4MV6 135566354 IC50 > 30000 nM T39716 CMC7Q6 135568488 IC50 = 4500 nM T39716 C3YB0A 135568523 IC50 = 24350 nM T39716 CL43OY 135568535 IC50 = 5750 nM T39716 C4OVP2 136416802 IC50 > 30000 nM T39716 C7ZCT8 136416815 IC50 > 30000 nM T39716 C6B5US 137628648 IC50 > 10000 nM T39716 C2QCA5 137631487 IC50 > 30000 nM T39716 C8JA9G 137631733 IC50 > 30000 nM T39716 CB4A0Y 137632255 IC50 = 3200 nM T39716 C2XI8Y 137632393 IC50 > 30000 nM T39716 CES7L0 137632608 IC50 = 874 nM T39716 C28PMQ 137634084 IC50 = 6500 nM T39716 C8HPN4 137634334 IC50 > 30000 nM T39716 CLG25H 137634494 IC50 > 30000 nM T39716 C7S8YV 137636062 IC50 = 444 nM T39716 C08DOT 137636231 IC50 = 480 nM T39716 CM51CG 137636524 IC50 = 156 nM T39716 CNA56O 137636856 IC50 = 336 nM T39716 CO3QJ8 137637393 IC50 = 1200 nM T39716 CJH2V9 137637559 IC50 = 18200 nM T39716 CH3M0S 137637752 IC50 = 260 nM T39716 CFK9D8 137638117 IC50 = 169 nM T39716 C8EZ4N 137638256 IC50 = 6400 nM T39716 CW95QX 137638418 IC50 = 3900 nM T39716 CEP37F 137638536 IC50 > 30000 nM T39716 CLEF51 137638686 IC50 = 12800 nM T39716 C0ZS9N 137638993 IC50 = 76 nM T39716 C5KEW7 137639838 IC50 = 931 nM T39716 CK1C5F 137640087 IC50 > 10000 nM T39716 C53ENH 137640507 IC50 = 1300 nM T39716 CN1RV9 137640762 IC50 = 162 nM T39716 CU0BS2 137641410 IC50 = 916 nM T39716 C70XZQ 137643636 IC50 > 30000 nM T39716 C2FOK7 137644816 IC50 = 1500 nM T39716 C5UL6D 137645197 IC50 = 1900 nM T39716 CNB72K 137645644 IC50 = 415 nM T39716 CH0TP2 137645931 IC50 = 3400 nM T39716 CMG27C 137645959 IC50 = 1600 nM T39716 CDCH19 137646766 IC50 = 242 nM T39716 CFKR53 137646837 IC50 > 30000 nM T39716 C4XVD2 137647076 IC50 = 660 nM T39716 CE57QM 137647529 IC50 = 281 nM T39716 C9L8CZ 137647771 IC50 = 1900 nM T39716 CD2WA1 137647899 IC50 = 2700 nM T39716 CTD69B 137647980 IC50 = 40000 nM T39716 CL06NY 137648464 IC50 > 30000 nM T39716 C3VO8H 137648536 IC50 = 6800 nM T39716 CP32AR 137648836 IC50 = 266 nM T39716 CQ93EC 137649075 IC50 = 400 nM T39716 COLY80 137649218 IC50 > 30000 nM T39716 CUFO39 137649223 IC50 > 30000 nM T39716 CV03MT 137649269 IC50 = 520 nM T39716 CJ59RF 137649283 IC50 = 820 nM T39716 CYU2J5 137649494 IC50 = 221 nM T39716 C04JSE 137649716 IC50 > 10000 nM T39716 C6PL9C 137651460 IC50 = 430 nM T39716 CE1OC6 137651969 IC50 = 18 nM T39716 CV4AP0 137652684 IC50 = 3200 nM T39716 C65XKJ 137653127 IC50 > 30000 nM T39716 CM1CP2 137653473 IC50 = 13000 nM T39716 CMJ0X9 137654527 IC50 = 24200 nM T39716 C8BDX5 137655281 IC50 > 30000 nM T39716 C9PJC3 137655604 IC50 > 10000 nM T39716 C3LG7W 137655838 IC50 > 30000 nM T39716 CJ7D8K 137655914 IC50 = 151 nM T39716 CTW5P4 137656265 IC50 = 328 nM T39716 CN2UE9 137656598 IC50 > 30000 nM T39716 CU28CY 137657424 IC50 = 52 nM T39716 C2ME3D 137657693 IC50 > 10000 nM T39716 CA72YP 137658615 IC50 = 220 nM T39716 CDO4F5 137658625 IC50 = 1100 nM T39716 C9VOB4 137658779 IC50 = 348 nM T39716 CZ2G4H 137659479 IC50 > 30000 nM T39716 C8UK1W 137659739 IC50 = 2400 nM T39716 CH4M3X 137659806 IC50 = 94 nM T39716 C2KX3V 137661020 IC50 = 17300 nM T39716 CF8HN9 137661762 IC50 = 1400 nM T39716 C0XCS4 137661956 IC50 = 77 nM T39716 CFC3L4 137662114 IC50 = 796 nM T39716 CC9K8L 137796790 IC50 = 22000 nM T39716 C7TAV3 138319685 IC50 > 300000 nM T39716 CE79SV 138377584 IC50 > 15000 nM T39716 C81ILP 138471783 IC50 > 30000 nM T39716 CJ68PM 138558077 IC50 > 30000 nM T39716 CF78ZM 138571094 IC50 = 19000 nM T39716 CR23HX 145948497 IC50 = 25000 nM T39716 CNSU46 145948687 IC50 > 5000 nM T39716 CRH94T 145948711 IC50 > 5000 nM T39716 CDZK19 145948712 IC50 > 5000 nM T39716 C8KW9F 145948730 IC50 = 2700 nM T39716 CQPL31 145948977 IC50 > 5000 nM T39716 CF6L8Q 145955101 IC50 = 260 nM T39716 CWJ0K6 145955642 IC50 > 100000 nM T39716 CCTB54 145958837 IC50 = 6640 nM T39716 C38DYW 145959291 IC50 = 3072 nM T39716 C3PA1D 145960602 IC50 = 4000 nM T39716 CZ8W1F 145960626 IC50 > 30000 nM T39716 CX3VH5 145960676 IC50 = 27000 nM T39716 CJ1O5H 145961103 IC50 > 30000 nM T39716 CBHA12 145961383 IC50 = 1100 nM T39716 CTVR05 145961491 IC50 = 18000 nM T39716 CSAR89 145961545 IC50 = 5300 nM T39716 C90GVK 145961619 IC50 = 13000 nM T39716 CRYN14 145961777 IC50 > 30000 nM T39716 CKM9A7 145961840 IC50 > 100000 nM T39716 CIM9O6 145961922 IC50 > 100000 nM T39716 CRQ9Z2 145962160 IC50 = 10000 nM T39716 C5HE2I 145962668 IC50 = 12000 nM T39716 CWL65X 145962677 IC50 = 2600 nM T39716 C52VFR 145962752 IC50 = 1300 nM T39716 C5E3RJ 145962891 IC50 > 100000 nM T39716 C6VNH3 145962956 IC50 > 100000 nM T39716 CS86IX 145963060 IC50 = 29000 nM T39716 C8CQX3 145963143 IC50 > 100000 nM T39716 CC1T5Z 145963172 IC50 > 100000 nM T39716 CP9TU4 145963182 IC50 = 7300 nM T39716 CWS86L 145963466 IC50 = 29000 nM T39716 CF7K5G 145963483 IC50 > 30000 nM T39716 C3UZX8 145963617 IC50 = 1800 nM T39716 CB9S3T 145963706 IC50 > 100000 nM T39716 CQT0L8 145963819 IC50 = 4800 nM T39716 C91CMS 145964520 IC50 = 4400 nM T39716 CW21LJ 145964527 IC50 > 30000 nM T39716 C5MJ1S 145964650 IC50 > 30000 nM T39716 CONK20 145964797 IC50 > 30000 nM T39716 CSK8Y1 145965486 IC50 = 4020 nM T39716 C3RYM4 145965521 IC50 > 30000 nM T39716 CR1U5T 145965937 IC50 > 30000 nM T39716 CL0UK1 145966092 IC50 > 30000 nM T39716 CYB3D7 145967129 IC50 = 1700 nM T39716 CHF13C 145967515 IC50 > 30000 nM T39716 CK7PN3 145969142 IC50 = 6000 nM T39716 C05NCW 145969596 IC50 > 30000 nM T39716 C4O5HA 145972742 IC50 > 30000 nM T39716 C8RFM3 145973261 IC50 > 33000 nM T39716 C1EH5C 145975024 IC50 > 30000 nM T39716 CT6Q3V 145975287 IC50 > 30000 nM T39716 CC49BG 145975892 IC50 = 1000 nM T39716 C59HVM 145977053 IC50 > 30000 nM T39716 CC1EP9 145977316 IC50 = 5000 nM T39716 CN9Q2I 145977501 IC50 = 5600 nM T39716 CUV49K 145977796 IC50 > 10000 nM T39716 C07URC 145978291 IC50 > 30000 nM T39716 C4O0KS 145978491 IC50 > 30000 nM T39716 C3QB6J 145978986 IC50 = 2400 nM T39716 CUXB52 145979881 IC50 = 6500 nM T39716 C87TKG 145980518 IC50 = 3000 nM T39716 C7XK3P 145981121 IC50 = 10000 nM T39716 CY8IF4 145981627 IC50 > 10000 nM T39716 C8RA5D 145981858 IC50 = 27000 nM T39716 C1YW4D 145982684 IC50 = 950 nM T39716 CBK7Z6 145986895 IC50 = 7900 nM T39716 C4GA2N 145987154 IC50 = 9100 nM T39716 CNL1W0 145987554 IC50 = 4200 nM T39716 C8Q2EG 145988110 IC50 = 4870 nM T39716 CP21ZQ 145988400 IC50 = 14000 nM T39716 CP45ZX 145988718 IC50 > 42000 nM T39716 C6U7LS 145990658 IC50 = 9500 nM T39716 C42YMJ 145990677 IC50 = 9600 nM T39716 CHZB80 145990751 IC50 = 710 nM T39716 CU0K2Y 145990810 IC50 > 10000 nM T39716 CGP61R 145991617 IC50 = 140 nM T39716 C0E2AZ 145991842 IC50 = 500 nM T39716 CMP27V 145992366 IC50 = 400 nM T39716 CQY2K6 145992782 IC50 = 42000 nM T39716 CDG51F 145993858 IC50 = 11000 nM T39716 CN86HU 145994027 IC50 = 6700 nM T39716 CW3B0G 145994131 IC50 = 3100 nM T39716 CBLA80 146683623 IC50 = 4600 nM T39716 C6Q2PL 155511032 IC50 = 13000 nM T39716 CNJ74U 155511848 IC50 > 30000 nM T39716 C3LFE7 155512957 IC50 > 30000 nM T39716 CXAL69 155513487 IC50 > 30000 nM T39716 C30OPH 155516574 IC50 = 6700 nM T39716 C8DA2L 155516676 IC50 = 23000 nM T39716 C4W6SR 155517129 IC50 = 9500 nM T39716 CY5UE9 155517299 IC50 > 42000 nM T39716 C03QEN 155519060 IC50 = 8400 nM T39716 CM96HX 155520010 IC50 = 6400 nM T39716 CAG7J0 155521246 IC50 > 30000 nM T39716 C76JKY 155521282 IC50 > 30000 nM T39716 C3A1YG 155522007 IC50 > 30000 nM T39716 C26JPN 155523322 IC50 = 12000 nM T39716 COZ54G 155523716 IC50 > 10000 nM T39716 C65NKP 155524061 IC50 > 30000 nM T39716 CTM01D 155525057 IC50 > 30000 nM T39716 C9RQ1Z 155526268 IC50 = 2400 nM T39716 CZX19C 155526353 IC50 = 3100 nM T39716 CF12TX 155527767 IC50 = 11000 nM T39716 CRE0O6 155528016 IC50 = 18000 nM T39716 C5P0YG 155529298 IC50 > 30000 nM T39716 C9U8FN 155529326 IC50 = 8700 nM T39716 C4PR0S 155530319 IC50 > 30000 nM T39716 CQ15KS 155530714 IC50 = 460 nM T39716 CGO81N 155532622 IC50 = 24000 nM T39716 CZ3F2O 155533245 IC50 > 30000 nM T39716 CQE8Y5 155534372 IC50 = 5200 nM T39716 CIKQ03 155534824 IC50 = 24000 nM T39716 CXA95Z 155535618 IC50 > 30000 nM T39716 C87RFO 155536189 IC50 > 30000 nM T39716 CO71LS 155536843 IC50 > 30000 nM T39716 CG8I5F 155538033 IC50 = 19000 nM T39716 CSDO95 155538523 IC50 > 30000 nM T39716 C64QKD 155538732 IC50 > 10000 nM T39716 CW1D7Y 155538889 IC50 = 5400 nM T39716 CRQW26 155539819 IC50 > 30000 nM T39716 CH63BD 155540878 IC50 > 42000 nM T39716 CQO68V 155541113 IC50 > 30000 nM T39716 C5T9KE 155542416 IC50 > 30000 nM T39716 CEL05R 155543885 IC50 > 25000 nM T39716 CQ7W0S 155544240 IC50 > 30000 nM T39716 C9H1RS 155545131 IC50 = 16000 nM T39716 CZ47YD 155545889 IC50 = 8900 nM T39716 CPD1B3 155547824 IC50 > 30000 nM T39716 CI94QY 155550095 IC50 = 3700 nM T39716 C1WTQ7 155553777 IC50 > 30000 nM T39716 CAV3Q9 155553847 IC50 > 30000 nM T39716 C8Q2FG 155555556 IC50 = 12290 nM T39716 CGE76T 155555738 IC50 > 30000 nM T39716 C3WT2Q 155556441 IC50 > 30000 nM T39716 CJX1Q7 155557620 IC50 = 9300 nM T39716 C0T6WM 155558045 IC50 > 42000 nM T39716 CKZT21 155559364 IC50 > 33000 nM T39716 CZ0VL5 155559622 IC50 > 30000 nM T39716 CY06UB 155561401 IC50 = 21000 nM T39716 CL96XW 155562578 IC50 > 30000 nM T39716 CPL2D9 155562982 IC50 = 11600 nM T39716 CSDR68 155563772 IC50 = 4100 nM T39716 CC5FE7 155564581 IC50 > 30000 nM T39716 CJL8Y5 155565696 IC50 = 14400 nM T39716 C2EKM7 155566527 IC50 = 5900 nM T39716 CZ9OW6 155567417 IC50 > 30000 nM T39716 CE3H4Z 155567528 IC50 = 800 nM T39716 CG97KZ 155568180 IC50 = 17800 nM T39716 D00TGC 56951318 IC50 = 200 nM T39716 D01AGR 24857857 IC50 = 4600 nM T39716 D06GQO 10955473 IC50 = 9000 nM T39716 D0FF6S 16038374 IC50 = 7340 nM T39716 D0N2KU 44517677 IC50 > 26000 nM T39716 D0O2RN 22149251 IC50 = 5650 nM T39716 D0P8TL 56947150 IC50 = 210 nM T05090 D00SQN 12136798 IC50 = 265 nM T05090 D07POC 176870 IC50 > 32000 nM T05090 D08CDI 208908 IC50 > 10000 nM T05090 D09DHY 6167 IC50 > 20 ug.mL-1 T05090 D0E3SH 6918837 Ki = 1.1 nM T05090 D0E7PQ 5311 IC50 = 1.4 nM T05090 D0L7LC 5352062 Ki = 0.15 nM T05090 D0Y3KG 3121 IC50 = 161000 nM T05090 D00FHR 9865515 Ki = 265 nM T05090 D05KED 53340666 IC50 = 51 nM T05090 D06TKI 49857317 IC50 = 7 nM T05090 D07FPY 6918877 Ki = 12 nM T05090 D09XIZ 11538455 Ki = 2.1 nM T05090 D0B3FV 6445533 IC50 = 0.4 nM T05090 D0B7CH 4775 IC50 = 260000 nM T05090 D0E6UZ 54575456 IC50 = 1.8 nM T05090 D0GE5B 56654642 IC50 = 60 nM T05090 D0GH3Q 9804992 Ki = 3 nM T05090 D0L2UQ 49855250 Ki = 19 nM T05090 D0M8FD 4261 IC50 < 300 nM T05090 D0V0SL 11749858 Ki = 8.2 nM T05090 D0XT6W 6918638 Ki = 1.5 nM T05090 D0Z4RC 24756910 IC50 = 9.1 nM T05090 D03SZR 5353484 IC50 = 70 nM T05090 D0J8OC 5186 Ki = 4.1 nM T05090 D0CH8Q 56965342 IC50 = 16 nM T05090 D0N2DK 72710871 IC50 = 2 nM T05090 D0QX3G 71532921 IC50 = 1700 nM T05090 D0N3SH 4996 Ki = 8 nM T05090 D0W9NH 2746 IC50 = 46 nM T05090 CBIR94 10313 IC50 = 7830 nM T05090 CL25FN 76175 IC50 > 30000 nM T05090 C1N2KZ 88129 IC50 = 340000 nM T05090 CH1JD3 419176 IC50 = 10000 nM T05090 CU3HS2 1108280 IC50 > 100000 nM T05090 C18ENP 6918846 Ki = 11 nM T05090 C1RD7E 6918878 IC50 = 398 nM T05090 CE9LP2 9543539 IC50 = 69 nM T05090 CJ07ZA 9800555 IC50 = 67 nM T05090 CC0EU7 9828788 IC50 = 4.8 nM T05090 C81EYJ 9923508 IC50 = 4.9 nM T05090 CQG4V8 9924543 IC50 = 2.8 nM T05090 CZL7C8 10017099 IC50 = 10 nM T05090 CL4C9H 10154438 Ki = 2.7 nM T05090 C7RC1E 10309899 IC50 = 9 nM T05090 C8G5WP 11210533 IC50 = 6900 nM T05090 CYJ60V 11244651 IC50 = 80100 nM T05090 CY34EQ 11393847 IC50 > 20000 nM T05090 CRZ7H2 11556677 IC50 = 12 nM T05090 C24SBP 11657529 IC50 = 250 nM T05090 CQ32FV 11664499 IC50 = 1.6 nM T05090 CG9OC4 11682502 IC50 = 30 nM T05090 CYB26W 11688197 IC50 = 187 nM T05090 CC3GQ0 11700059 IC50 = 48 nM T05090 C9G1BN 11993595 IC50 = 440 nM T05090 CH5JS7 11993694 IC50 = 23 nM T05090 C1BVY9 12325934 IC50 > 30000 nM T05090 C06UTF 13507024 IC50 = 10 nM T05090 C4XJ8M 13889849 Ki = 1350 nM T05090 C1KR4L 14113324 IC50 > 50000 nM T05090 C15MQN 14113325 IC50 > 50000 nM T05090 C2D1KP 15983982 Ki = 20 nM T05090 CA2YF9 15984018 IC50 = 230 nM T05090 CB81VC 15985904 IC50 = 130 nM T05090 CHB82E 15986417 IC50 = 55600 nM T05090 C52EVH 15986418 IC50 = 4570 nM T05090 CS1QO9 15986509 IC50 = 84500 nM T05090 C5T1WF 16006672 IC50 = 697 nM T05090 CQGC05 16036765 IC50 = 14 nM T05090 CM3T2E 16049824 IC50 = 17 nM T05090 C30UFT 16066811 IC50 = 939 nM T05090 CFK8J5 16068056 Ki = 20 nM T05090 CMQP70 16068495 Ki = 27 nM T05090 CT84XO 16068594 Ki = 15 nM T05090 CF3ZG5 16068595 Ki = 13 nM T05090 CL60CA 16068912 Ki = 10 nM T05090 CVT0E7 16070046 IC50 = 276 nM T05090 C5CIB4 16663079 IC50 > 50000 nM T05090 CWO7V0 16733295 IC50 = 1560 nM T05090 CV54SY 16733414 IC50 = 1320 nM T05090 CB4IN2 16773791 IC50 = 289 nM T05090 CKM7F9 17747371 IC50 > 1000 nM T05090 CF7JR0 17756401 IC50 = 50 nM T05090 C3FN8M 17756403 IC50 = 79 nM T05090 CE2W3M 21630365 IC50 = 988 nM T05090 CS5R0U 22836624 Ki = 14500 nM T05090 CEF8W4 23625604 IC50 = 3162.28 nM T05090 CB8A5Q 23648260 IC50 = 27710 nM T05090 C36NKL 23648268 IC50 > 20000 nM T05090 C4UV3T 24726843 IC50 = 3500 nM T05090 C8RC9P 24744325 IC50 = 7000 nM T05090 CMI5E4 24746277 IC50 = 16480 nM T05090 CVB7J3 24746434 IC50 = 1260000 nM T05090 C8EYH1 24746435 IC50 = 340000 nM T05090 C28AWJ 24746436 IC50 = 1270000 nM T05090 C17GDO 24779722 IC50 = 131 nM T05090 CIO7Q6 24853792 IC50 = 1000 nM T05090 CBN0J5 24853793 IC50 = 120 nM T05090 CI3B6L 24857909 IC50 = 670 nM T05090 C5GCM1 24881328 IC50 = 13.7 nM T05090 C8QVB1 24881329 IC50 = 25.3 nM T05090 CU0AM3 24881330 IC50 = 7.9 nM T05090 CQM51L 24881331 IC50 = 7.2 nM T05090 C4KH8F 24881332 IC50 = 16.4 nM T05090 C1KA3V 24881333 IC50 = 15.1 nM T05090 C47APB 24881402 IC50 = 4.5 nM T05090 CSN8W1 24881403 IC50 = 7.7 nM T05090 C1UQ3K 24881404 IC50 = 8 nM T05090 C51TMH 24881405 IC50 = 4 nM T05090 C9EZI7 24881406 IC50 = 2.7 nM T05090 C6P3HS 24881407 IC50 = 9.7 nM T05090 CZ3TU1 24881464 IC50 = 12 nM T05090 CDI49N 24881465 IC50 = 5.8 nM T05090 CQGP87 24881466 IC50 = 4.2 nM T05090 CS1MH8 24888322 IC50 = 22000 nM T05090 CC0R9O 24938735 IC50 = 0.7 nM T05090 CF03HD 24948905 IC50 = 115 nM T05090 CHP8O6 24948906 IC50 = 4.04 nM T05090 C1KRT8 24948907 IC50 = 144 nM T05090 CKY2P8 24948908 IC50 = 10.2 nM T05090 C25CFI 24948909 IC50 = 65.8 nM T05090 CWQ04Z 24948910 IC50 = 18 nM T05090 CM9I3X 24951310 IC50 = 12.9 nM T05090 CX1YF8 24951311 IC50 = 158 nM T05090 CV10XU 24951312 IC50 < 0.002 nM T05090 CD6KV0 24951313 IC50 = 83.6 nM T05090 CQY9Z0 24951314 IC50 = 190 nM T05090 C5B0IJ 25023793 IC50 = 120 nM T05090 CLG23N 25023794 IC50 = 10 nM T05090 CHE82I 25023795 IC50 > 10000 nM T05090 CX8G3W 25023796 IC50 = 1700 nM T05090 CVRS37 25023797 IC50 = 560 nM T05090 C7GO3U 25023798 IC50 = 9400 nM T05090 C3G2AU 25023799 IC50 = 120 nM T05090 CAS18V 25023800 IC50 = 3100 nM T05090 CX7D5B 25023801 IC50 = 1400 nM T05090 CZG50I 25023802 IC50 > 5000 nM T05090 CP4T7J 25023806 IC50 = 2900 nM T05090 CVS1M4 25023811 IC50 = 4600 nM T05090 CJG8C5 25023818 IC50 = 7300 nM T05090 CLA50V 25023819 IC50 = 7600 nM T05090 CV8EF6 25032862 IC50 = 22450 nM T05090 CX69SY 25066355 IC50 = 369 nM T05090 CF8VP4 25066356 IC50 = 176 nM T05090 CS9XH7 25066547 IC50 = 240 nM T05090 C46AGN 25066548 IC50 = 39.6 nM T05090 CJF2M7 25066549 IC50 = 246 nM T05090 CPTI96 25110599 IC50 = 12 nM T05090 C7ZN2W 25118059 IC50 = 3.4 nM T05090 C4I1CJ 25155417 IC50 = 6180 nM T05090 CB4E2J 25155956 IC50 > 50000 nM T05090 CKG24O 25157972 IC50 = 6390 nM T05090 C19JIO 25157973 IC50 = 5384 nM T05090 CFS5O4 25168576 IC50 = 7100 nM T05090 C0R5OK 25168856 IC50 > 1000 nM T05090 CO14XG 25195084 IC50 = 320 nM T05090 C6BDX3 25207860 IC50 = 104000 nM T05090 C5COM1 25218554 IC50 = 6928 nM T05090 CN6XA4 25218555 IC50 = 9617 nM T05090 CL8K9U 25218556 IC50 = 8706 nM T05090 C9WA4B 25218557 IC50 = 17390 nM T05090 CRG29Y 25218558 IC50 = 5727 nM T05090 CEH71M 25218560 IC50 = 4330 nM T05090 CIZD97 25218561 IC50 > 50000 nM T05090 C7I5EL 25218562 IC50 = 3202 nM T05090 C15YDI 25218563 IC50 = 5102 nM T05090 CCD5M7 25227504 IC50 = 55.7 nM T05090 CK0D5S 25227505 IC50 = 89 nM T05090 CN97JP 25227508 IC50 = 93.6 nM T05090 CW8R1B 25227513 IC50 = 94.5 nM T05090 CPNQ02 25257992 IC50 = 85 nM T05090 CE0NV4 25257993 IC50 = 3.07 nM T05090 C43BHY 25269097 IC50 = 25 nM T05090 CU53WB 42596953 IC50 = 66 nM T05090 C2LES7 42599455 IC50 = 5.3 nM T05090 C2KO0F 42599456 IC50 = 6.7 nM T05090 C1UAO7 42601485 IC50 = 12000 nM T05090 COI7Y3 42611300 IC50 = 143 nM T05090 CU23PG 42611301 IC50 = 8 nM T05090 CW1G2R 42611390 IC50 = 280 nM T05090 CQ37HN 42612743 IC50 = 2.59 nM T05090 CX1UT9 42612744 IC50 = 1151 nM T05090 CLH2Q7 42612852 IC50 = 608 nM T05090 CXK4C1 42618298 IC50 = 1.2 nM T05090 CDT65Y 42631047 IC50 > 100000 nM T05090 CO57GS 44138033 IC50 = 659 nM T05090 C7RCY4 44178890 IC50 = 9 nM T05090 CQ2VD5 44219634 IC50 = 25 nM T05090 C0JY2Q 44249789 IC50 = 1300 nM T05090 CU7SL0 44249820 IC50 = 2200 nM T05090 CY0QB9 44253226 IC50 = 65 nM T05090 CZ8R1N 44253780 IC50 = 87 nM T05090 C5YRC9 44431499 IC50 = 91000 nM T05090 CV7P0C 44447120 IC50 = 2810 nM T05090 CNC51G 44447194 IC50 > 50000 nM T05090 C8WKU9 44453790 IC50 = 42 nM T05090 C5VP4D 44454144 IC50 = 11000 nM T05090 C8A1ZD 44456564 IC50 = 3.7 nM T05090 CJ0L4C 44456965 IC50 = 14 nM T05090 C74LTB 44506448 IC50 = 61 nM T05090 C4FKU6 44541235 IC50 > 1000 nM T05090 C7F8YJ 44543715 Ki = 250 nM T05090 CQ2TU3 44550557 Ki = 740 nM T05090 CW4KH2 44551271 IC50 = 16800 nM T05090 CDW54Z 44562605 IC50 > 1000 nM T05090 C9MB4K 44562607 IC50 = 500 nM T05090 CH2NP3 44562608 IC50 > 1000 nM T05090 CBYZ26 44562609 IC50 > 1000 nM T05090 C3QSI4 44562762 IC50 > 1000 nM T05090 CRJS52 44562763 IC50 > 1000 nM T05090 CJ5US8 44562765 IC50 > 1000 nM T05090 CQ5RJ3 44562799 IC50 = 630 nM T05090 CDY0E1 44562801 IC50 > 1000 nM T05090 CEM91G 44562802 IC50 = 380 nM T05090 CEA9D0 44562840 IC50 > 1000 nM T05090 C3DMN0 44563197 IC50 = 520 nM T05090 CGF8R5 44563236 IC50 > 1000 nM T05090 CT63QG 44563237 IC50 = 500 nM T05090 CIO34V 44564642 Ki = 11 nM T05090 COM65J 44572384 IC50 = 620 nM T05090 CMA3R6 44574139 IC50 = 30 nM T05090 C5KLR7 44574177 IC50 > 30000 nM T05090 CFS49I 44574178 IC50 = 10600 nM T05090 CJ32DK 44574179 IC50 > 30000 nM T05090 CQOS28 44574180 IC50 = 102 nM T05090 CN96ZV 44574181 IC50 = 7410 nM T05090 C46XHW 44574207 IC50 > 30000 nM T05090 C3RY9V 44574208 IC50 = 1920 nM T05090 CS4JP5 44589733 IC50 > 10000 nM T05090 CEPG12 44589734 IC50 = 840 nM T05090 CZVO54 44589735 IC50 = 1500 nM T05090 CPB1G7 44589736 IC50 = 2800 nM T05090 CZ7VE6 44589745 IC50 = 27 nM T05090 CDH14U 44589746 IC50 = 180 nM T05090 C3C6WU 44589911 IC50 = 5340000 nM T05090 CVA4I9 44589912 IC50 = 5500000 nM T05090 CVQ83W 44589913 IC50 > 30000000 nM T05090 C16-FEB 44591258 IC50 = 19320 nM T05090 C1OCI9 44591315 IC50 = 4803 nM T05090 CA6Q9Y 44592060 IC50 = 3140 nM T05090 CH2J8R 44598238 IC50 = 1670 nM T05090 CE5W3U 44598288 IC50 = 690 nM T05090 C68BJH 44598289 IC50 = 2990 nM T05090 C9K2WV 44598290 IC50 = 970 nM T05090 C16ZEP 44598291 IC50 = 54 nM T05090 C28GHB 44598344 IC50 = 260 nM T05090 CU65LR 44598345 IC50 = 262 nM T05090 C41VTN 44598346 IC50 = 1090 nM T05090 CHQ86X 44598347 IC50 = 694 nM T05090 CCVA51 44598385 IC50 = 1040 nM T05090 C29NXL 44598386 IC50 = 3630 nM T05090 C5WM7H 44598387 IC50 > 10000 nM T05090 CK8V9I 44598388 IC50 = 164 nM T05090 CJ54OH 44598429 IC50 = 31 nM T05090 C1TYW6 44598430 IC50 = 240 nM T05090 C3TOK2 44598431 IC50 = 190 nM T05090 CPZ65Q 44598479 IC50 > 10000 nM T05090 CGT51H 44598480 IC50 = 62 nM T05090 CZ62IW 44598481 IC50 > 10000 nM T05090 C0OT6I 44598482 IC50 = 7080 nM T05090 CX8U6S 44598483 IC50 > 10000 nM T05090 CO5YJ8 44598535 IC50 = 990 nM T05090 C5H8RA 44598536 IC50 = 32 nM T05090 CC2QV9 44623002 IC50 > 50000 nM T05090 CVJ51M 44623152 IC50 > 50000 nM T05090 C6TJ2G 44623153 IC50 > 50000 nM T05090 COZ25S 45268021 IC50 = 69300 nM T05090 CS9DW4 45268025 IC50 = 3400 nM T05090 C0BQF9 45268900 IC50 = 46900 nM T05090 CH08UF 45268906 IC50 = 5600 nM T05090 C27VLQ 45269750 IC50 = 4300 nM T05090 CK1AP8 45269751 IC50 = 27200 nM T05090 CSM1O6 45271073 IC50 = 260 nM T05090 C02LVF 45485792 IC50 = 32 nM T05090 C7EAV5 45485820 IC50 = 54 nM T05090 CIO0T2 46179730 IC50 = 3.39 nM T05090 C2M4GV 46179732 IC50 = 3.7 nM T05090 CS75CD 46179779 IC50 = 2.8 nM T05090 C39YKM 46179780 IC50 = 5.3 nM T05090 C0CKE5 46180624 IC50 = 120 nM T05090 C7GYH0 46180758 IC50 = 18.1 nM T05090 C27IKH 46180759 IC50 = 3 nM T05090 CSC1Y9 46180760 IC50 = 3.4 nM T05090 C4XHL5 46180761 IC50 = 1.4 nM T05090 C70FSJ 46180763 IC50 = 3.3 nM T05090 CD57RJ 46197798 IC50 = 9 nM T05090 CR04HA 46197799 IC50 = 21 nM T05090 CB2G1W 46881144 IC50 = 1.66 nM T05090 C85RDN 46881213 IC50 = 1.55 nM T05090 CQTI31 46881225 IC50 = 122 nM T05090 C48QWG 46884058 IC50 = 2263 nM T05090 CVU0D3 46884059 IC50 = 35 nM T05090 C5UMJ3 46884060 IC50 = 240 nM T05090 CQ76JG 46884061 IC50 = 1750 nM T05090 C9HMN4 46884114 IC50 = 1100 nM T05090 C8V3HK 46884115 IC50 = 1346 nM T05090 C8CI2D 46884116 IC50 = 4989 nM T05090 C35OPR 46884117 IC50 = 56 nM T05090 CI0W9C 46884118 IC50 = 30 nM T05090 C25DSY 46887918 IC50 = 24.7 nM T05090 C93CLK 46887919 IC50 = 22000 nM T05090 CPSI47 46890583 Ki = 8 nM T05090 C90NYX 46896338 IC50 = 230 nM T05090 CU7L5W 46906597 IC50 = 470000 nM T05090 CG46KJ 46906641 IC50 = 605000 nM T05090 CAT34L 46906643 IC50 = 36000 nM T05090 C4V7PG 46907052 IC50 = 13300 nM T05090 CSNU34 46907053 IC50 = 3200 nM T05090 CMQ3R0 46907054 IC50 = 14500 nM T05090 C05KTS 46907124 IC50 = 460000 nM T05090 C2PC1Z 46907160 IC50 = 32300 nM T05090 C72BEW 46907196 IC50 = 730000 nM T05090 C4V3ZK 46907197 IC50 = 718000 nM T05090 C6TRS7 46907198 IC50 = 695000 nM T05090 C0K4DL 46907280 IC50 = 725000 nM T05090 C3NE0Q 46907281 IC50 = 508000 nM T05090 C1HV6U 46907409 IC50 > 20000 nM T05090 C6GY9I 46934544 IC50 = 26700 nM T05090 C3OD2Y 46934546 IC50 = 28100 nM T05090 CL7PS1 49831258 IC50 = 46000 nM T05090 CC7Y9U 49850262 IC50 = 155 nM T05090 C50PXU 49855444 IC50 > 50000 nM T05090 CE7D2J 49855568 IC50 = 6300 nM T05090 CFD9P3 49855569 IC50 > 32000 nM T05090 C1AU5N 49855758 IC50 > 32000 nM T05090 CIFK93 49855759 IC50 > 32000 nM T05090 CK48OJ 49855760 IC50 > 32000 nM T05090 CZI3M1 49855761 IC50 > 32000 nM T05090 CRPZ58 49855949 IC50 > 32000 nM T05090 CTU0K3 49855950 IC50 > 32000 nM T05090 CF85NL 49855951 IC50 > 32000 nM T05090 CF7YS9 49855952 IC50 > 32000 nM T05090 CJU38G 49855953 IC50 = 560 nM T05090 C6POK9 49856931 IC50 = 10 nM T05090 C52ABG 50942502 IC50 = 460 nM T05090 CPQ0F7 50991199 IC50 = 2 nM T05090 COA5W3 51051073 IC50 = 28 nM T05090 C5LZ4R 51351536 IC50 > 30000 nM T05090 CV76KB 51357270 IC50 = 30 nM T05090 C8SUQ5 53317424 IC50 > 30000 nM T05090 C7MO2J 53325871 IC50 = 2.1 nM T05090 CG84JS 53325976 IC50 = 1000 nM T05090 CVM4Q3 53357987 IC50 = 20000 nM T05090 C78GKN 53361474 Ki = 64 nM T05090 CNB63X 53361475 Ki = 23 nM T05090 CQ43VH 53363518 Ki = 16 nM T05090 C6Y2EV 53374826 IC50 = 5370 nM T05090 CC5K2U 53380601 IC50 = 760 nM T05090 CN17BX 53380699 IC50 = 1520 nM T05090 CYQV72 54030066 IC50 = 39000 nM T05090 C5A7MU 54613496 IC50 = 6.4 nM T05090 CVP16C 54753629 IC50 = 97000 nM T05090 CIO96M 56659403 IC50 > 100000 nM T05090 CT4ZY0 56661203 IC50 = 6 nM T05090 C7R9TZ 56663191 IC50 = 0.7 nM T05090 CL18NI 56666337 IC50 > 100000 nM T05090 C9LC5Y 56673234 IC50 > 100000 nM T05090 CWH5N4 56673261 IC50 > 100000 nM T05090 C2ML5S 56837168 IC50 = 9.77 nM T05090 CCW89V 56932477 IC50 = 0.669 nM T05090 CZ25SN 56935695 IC50 > 30000 nM T05090 CP4EL2 57328394 IC50 = 14000 nM T05090 C5CRJ1 57412107 IC50 = 90 nM T05090 COG4Q8 57412108 IC50 = 130 nM T05090 C4LI0D 57521296 IC50 = 4700 nM T05090 CA5Q6O 58147189 IC50 > 50000 nM T05090 C4DYC0 58147224 IC50 > 50000 nM T05090 CMP04X 58147302 IC50 > 50000 nM T05090 C4V7FY 58191950 IC50 = 840 nM T05090 CPCA29 58191961 IC50 = 15 nM T05090 C7HF1L 58191965 IC50 = 550 nM T05090 CR4BX0 58191982 IC50 = 440 nM T05090 C8V1NK 58191988 IC50 = 920 nM T05090 C8LWY9 58191997 IC50 = 510 nM T05090 C3IQ9B 58191999 IC50 = 770 nM T05090 CQB69R 58192003 IC50 = 610 nM T05090 CLD40J 58465708 IC50 = 8500 nM T05090 C1MB4Q 59323957 IC50 > 30000 nM T05090 CK6LX0 59454220 IC50 = 230 nM T05090 C2SDN1 59454252 IC50 = 200 nM T05090 CPZ5Q3 60148646 IC50 = 25000 nM T05090 CP2HK9 60148667 IC50 = 18000 nM T05090 C8ZL3J 60148690 IC50 = 16000 nM T05090 CK5N4E 60148693 IC50 = 12000 nM T05090 C27DKW 60148711 IC50 = 9400 nM T05090 CS2E6C 60148712 IC50 = 26000 nM T05090 CPF50R 60148997 IC50 = 33000 nM T05090 CB7X2E 60151224 IC50 = 7.67 nM T05090 CY05OU 60151225 IC50 = 73 nM T05090 CWO8H0 60152596 IC50 = 1680 nM T05090 CBN3L0 69950064 Ki > 43000 nM T05090 C6RFQ8 70676597 IC50 = 3000 nM T05090 CM4XB8 70681905 IC50 = 5090 nM T05090 CW5MP0 70681906 IC50 = 4890 nM T05090 CGYX13 70681907 IC50 = 5700 nM T05090 CPMZ01 70681908 IC50 = 2190 nM T05090 CM62BN 70682297 IC50 = 1440 nM T05090 C3PR4C 70684025 IC50 = 34120 nM T05090 C8R9XE 70684026 IC50 = 4800 nM T05090 CT64UC 70686159 IC50 = 16070 nM T05090 C94YFZ 70686160 IC50 = 26390 nM T05090 CBZ8W0 70688300 IC50 = 13480 nM T05090 C0CQP5 70690303 IC50 = 6620 nM T05090 C8T1FV 70690304 IC50 = 1940 nM T05090 C7VF1B 70692849 IC50 = 800 nM T05090 C28UMB 70693708 IC50 = 62 nM T05090 CGSM24 70694519 IC50 = 2660 nM T05090 CX23AC 70696578 IC50 = 9380 nM T05090 CW6F1J 70696579 IC50 = 19200 nM T05090 CQY1I6 70789579 Ki > 43000 nM T05090 C76SGF 71457594 IC50 = 5400 nM T05090 C72DJO 71465631 IC50 = 1090 nM T05090 CQ7VL0 71467493 IC50 = 60 nM T05090 C5BR1D 71467494 IC50 = 110 nM T05090 CS74UB 71467495 IC50 = 2830 nM T05090 CX3U9M 71467628 IC50 = 3560 nM T05090 C3PIK2 71467958 IC50 = 110 nM T05090 CTNS49 71467959 IC50 = 620 nM T05090 CQ6B2I 71467960 IC50 = 260 nM T05090 C0YXF2 71467961 IC50 = 360 nM T05090 C1MH5Z 71467962 IC50 = 100 nM T05090 C7ESZ2 71467963 IC50 = 190 nM T05090 C45FCJ 71468055 IC50 = 380 nM T05090 C3H0CR 71468158 IC50 = 140 nM T05090 CQ26IW 71468159 IC50 = 110 nM T05090 C6ZPJ4 71468160 IC50 = 2590 nM T05090 CJU64Z 71468161 IC50 = 73.91 nM T05090 CD8O7W 71468162 IC50 = 330 nM T05090 CSDO79 71468163 IC50 = 280 nM T05090 CN97RG 71468164 IC50 = 380 nM T05090 C5I0TX 71468273 IC50 = 310 nM T05090 CJKU04 71468274 IC50 = 450 nM T05090 CZJ84E 71468275 IC50 = 590 nM T05090 C6L0RV 71468277 IC50 = 200 nM T05090 CAH65F 71468278 IC50 = 80 nM T05090 CVP26X 71468393 IC50 = 160 nM T05090 CFW2I5 71468672 IC50 = 27.51 nM T05090 CIS73X 71468801 IC50 = 1640 nM T05090 CS86BK 71468803 IC50 = 3170 nM T05090 CJD46S 71468805 IC50 = 2220 nM T05090 CU9FQ3 71468924 IC50 = 1580 nM T05090 C01IKD 71468927 IC50 = 270 nM T05090 CNXK19 71468928 IC50 = 150 nM T05090 C7GY8U 71495390 IC50 = 69 nM T05090 CBE46I 71495482 IC50 = 81 nM T05090 CQ5FC3 71495575 IC50 = 188 nM T05090 CIQ3E7 71495576 IC50 = 155 nM T05090 CAL79Y 71495577 IC50 = 49 nM T05090 C1SXH7 71495578 IC50 = 9.6 nM T05090 C1Q8LP 71495673 IC50 = 69 nM T05090 CF72JS 71495674 IC50 = 217 nM T05090 C3T7UP 71495675 IC50 = 53 nM T05090 CSW12I 71502605 IC50 = 230 nM T05090 C89SWX 71527724 IC50 = 15000 nM T05090 C6S5JQ 71527847 IC50 = 7.5 nM T05090 C6KBD4 71534512 IC50 = 72 nM T05090 CT51EW 71534810 IC50 = 3 nM T05090 C7QN3O 71534812 IC50 = 1 nM T05090 C8M3HU 71537640 IC50 = 55 nM T05090 C2QML7 71537641 IC50 = 2 nM T05090 CZJX53 71537927 IC50 = 6330 nM T05090 CU0ZE6 71537928 IC50 = 5 nM T05090 CH9FS7 71537929 IC50 = 122 nM T05090 CTW95A 71537931 IC50 = 5 nM T05090 CW3BT5 71537932 IC50 = 17100 nM T05090 C3C0RO 71538475 IC50 = 7 nM T05090 CIA28E 71538746 IC50 = 10 nM T05090 CFCV26 71538748 IC50 = 495 nM T05090 CY2T1Q 71538749 IC50 = 475 nM T05090 C4A6VJ 71538750 IC50 = 8 nM T05090 CG72NC 71538751 IC50 = 9 nM T05090 C7RUE6 71540743 IC50 = 14000 nM T05090 C9LA4F 71540744 IC50 = 885 nM T05090 C0EK5J 71540745 IC50 = 3990 nM T05090 C80HZX 71540746 IC50 = 31 nM T05090 C5UZQ0 71540747 IC50 = 10400 nM T05090 C4G5US 71540862 IC50 = 649 nM T05090 CKR6U8 71583101 IC50 = 23000 nM T05090 CBZ5S9 71583103 IC50 = 29000 nM T05090 C3PSJ9 71583105 IC50 = 26000 nM T05090 C21GHR 71624738 IC50 = 1600 nM T05090 C7HG0K 71655802 IC50 = 694 nM T05090 CV73YD 71660259 IC50 = 1360 nM T05090 CQ5UR0 71660260 IC50 = 8360 nM T05090 CQ5P0T 71660261 IC50 = 830 nM T05090 C8EIX0 71660262 IC50 = 1030 nM T05090 CPJ4V7 71680913 IC50 = 23000 nM T05090 CI9G3B 71681069 IC50 = 18000 nM T05090 CIR56T 71721558 IC50 = 260 nM T05090 CCD18W 71721946 IC50 = 240 nM T05090 CI9H6L 72164895 IC50 = 19 nM T05090 CS5UL7 72195322 IC50 = 68 nM T05090 CAC5Q7 72375561 IC50 = 550 nM T05090 C3WQV2 72375562 IC50 = 7.2 nM T05090 CC1W6J 72375670 IC50 = 1900 nM T05090 CY8R0O 72696205 IC50 = 11620 nM T05090 CM3KS6 72696333 IC50 = 1690 nM T05090 CI2EH8 72696334 IC50 = 520 nM T05090 C0CM8Q 72696335 IC50 = 230 nM T05090 CG31RX 72696336 IC50 = 2110 nM T05090 CJ3EH7 72696464 IC50 = 590 nM T05090 C1OA0T 72696465 IC50 = 130 nM T05090 C1I9TZ 72696466 IC50 = 193 nM T05090 CFU3V5 72696467 IC50 = 242 nM T05090 CTR52Z 72696598 IC50 = 767 nM T05090 C4O2ZT 72696599 IC50 = 111 nM T05090 C5N9BQ 72696600 IC50 = 1444 nM T05090 CE87BF 72696601 IC50 = 899 nM T05090 C73XOU 72734382 IC50 = 64 nM T05090 CQA16N 72946833 IC50 = 62 nM T05090 CHQ39Y 72947043 IC50 = 88 nM T05090 CCST90 72947044 IC50 = 11 nM T05090 CX3W1T 73333311 IC50 = 4500 nM T05090 C68LBO 73349131 IC50 = 2 nM T05090 CUD02X 73355098 IC50 = 102 nM T05090 CD6L5K 73707349 IC50 = 2 nM T05090 C26KZD 73707535 IC50 = 1.4 nM T05090 CM1H3U 73707536 IC50 = 5.4 nM T05090 CH97TE 73707543 IC50 = 1.8 nM T05090 C2PWQ3 73707544 IC50 = 2.4 nM T05090 CEM5B6 73707545 IC50 = 1.6 nM T05090 CPQ43R 73707550 IC50 = 0.8 nM T05090 CJ1DA8 73774764 IC50 = 403.2 nM T05090 CQ3K6G 73776326 IC50 = 14.1 nM T05090 CC4L0G 73776327 IC50 = 143 nM T05090 CZB6G7 73776472 IC50 = 3.9 nM T05090 CSRE84 73776614 IC50 = 5.5 nM T05090 C01FVX 73776616 IC50 = 3.2 nM T05090 C3UC9H 73891099 IC50 = 12400 nM T05090 CMU19S 74221664 IC50 = 330 nM T05090 CM6H9C 76324878 IC50 = 8900 nM T05090 CKI74A 76853213 IC50 > 20000 nM T05090 CCR7L2 76853289 IC50 = 12000 nM T05090 CJ6Z0X 78324068 IC50 > 20000 nM T05090 CG5ZD9 86291495 IC50 = 15 nM T05090 C3EM7H 86581004 IC50 = 85 nM T05090 C7UK3Y 86581005 IC50 = 69 nM T05090 CY64UM 86581152 IC50 = 91 nM T05090 CY5V7C 86581153 IC50 = 89 nM T05090 C1HE8I 86581432 IC50 = 210 nM T05090 CZM07I 86581434 IC50 = 65 nM T05090 C8ZQG9 86581435 IC50 = 87 nM T05090 CS5I4Y 87261507 IC50 = 80 nM T05090 C5JIT0 87618609 IC50 = 320 nM T05090 CRQO37 88005144 IC50 = 500 nM T05090 CP1NA9 89183138 IC50 > 33330 nM T05090 CQS6C0 89183185 IC50 = 1490 nM T05090 CB47VC 89464167 IC50 = 35800 nM T05090 CD7J6C 90644927 IC50 = 200 nM T05090 C62GSL 90654859 IC50 = 47 nM T05090 CYW51P 90654946 IC50 = 340000 nM T05090 CJH1S6 90654947 IC50 > 100000 nM T05090 CSDO81 90664458 Ki = 19 nM T05090 CAQL21 91667420 IC50 = 42.5 nM T05090 C5M9AK 91667421 IC50 = 14.59 nM T05090 CJO6T1 91810840 IC50 = 2100 nM T05090 CYJ12Q 91884636 IC50 = 5 nM T05090 C0FCU9 91938063 IC50 = 25.84 nM T05090 C34WIG 92045024 IC50 > 100000 nM T05090 CYO9J5 101879983 IC50 = 3.56 nM T05090 C9OC0F 101882265 IC50 = 6590 nM T05090 CVE07R 101882857 IC50 = 394 nM T05090 C63EWT 101882858 IC50 = 2.42 nM T05090 C8KZB4 101883993 Ki = 800 nM T05090 C7Q6ID 101884982 IC50 = 13 nM T05090 CR46PQ 101884983 IC50 = 6 nM T05090 CRZ83C 101884989 IC50 = 138 nM T05090 CS2UL0 117829456 IC50 = 28 nM T05090 C7L4OT 117829461 IC50 = 28 nM T05090 C50VUN 117829462 IC50 = 98 nM T05090 CH27PR 118613747 IC50 = 7.8 nM T05090 C0OX4M 118613748 IC50 = 1.1 nM T05090 CNF09H 118613750 IC50 = 100 nM T05090 C3ETI2 118613751 IC50 = 4.2 nM T05090 C9KZQ0 118613755 IC50 = 1.1 nM T05090 C30OPU 118613756 IC50 = 6 nM T05090 C46TFD 118613757 IC50 = 1.8 nM T05090 C1J5AG 118613783 IC50 = 0.68 nM T05090 C9T0ML 118613821 IC50 = 0.38 nM T05090 CSU52M 118656852 IC50 = 24000 nM T05090 C45UYG 118709095 IC50 = 12000 nM T05090 C7QHE4 118712502 IC50 = 0.3 nM T05090 C8KSD6 118712503 IC50 = 0.6 nM T05090 C1JFZ7 118714371 IC50 = 367 nM T05090 CXF0U3 118714375 IC50 = 246 nM T05090 C2M5OR 118714376 IC50 = 13 nM T05090 CY4GN9 118714377 IC50 = 30 nM T05090 C7P3KH 118715726 IC50 = 126.56 nM T05090 CK6UM0 118715727 IC50 = 37.67 nM T05090 CW85VZ 118715728 IC50 = 17.91 nM T05090 C39EXL 118715729 IC50 = 607.03 nM T05090 CYGT73 118715730 IC50 = 48.26 nM T05090 CCAM49 118715731 IC50 = 23.53 nM T05090 C37NXA 118715732 IC50 = 16.85 nM T05090 CEN1J3 118715733 IC50 = 14.47 nM T05090 CFD2B8 118715734 IC50 = 11.88 nM T05090 CO8TJ6 118715735 IC50 = 13.52 nM T05090 C90TIX 118715736 IC50 = 14.63 nM T05090 C14KQU 118715737 IC50 = 6.46 nM T05090 CMK8B7 118715738 IC50 = 20.77 nM T05090 CQ6V9M 118715739 IC50 = 3.47 nM T05090 CWM04T 118715740 IC50 = 9.33 nM T05090 CLYS39 118715741 IC50 = 2.92 nM T05090 C04XZU 118715742 IC50 = 14.74 nM T05090 CJ4FS3 118715743 IC50 = 39.72 nM T05090 C3BH1K 118715744 IC50 = 3.52 nM T05090 CA12OP 118715745 IC50 = 3.22 nM T05090 C51RTI 118715746 IC50 = 3.58 nM T05090 CFX16A 118715747 IC50 = 8.19 nM T05090 C5OWL1 118715748 IC50 = 14.05 nM T05090 C8AW9X 118715749 IC50 = 14.1 nM T05090 C2Y7ZC 118715750 IC50 = 26.53 nM T05090 CM5QT7 118719376 Ki = 1400 nM T05090 CPB7C3 118719377 Ki = 500 nM T05090 C09OGH 118719378 Ki = 600 nM T05090 CR5VC1 118719379 Ki = 700 nM T05090 C32LCM 118719380 Ki = 200 nM T05090 C8U6YR 118719381 Ki = 500 nM T05090 C9Y0HV 118719382 Ki = 300 nM T05090 CY0J4D 118719383 Ki = 500 nM T05090 CCYU59 118719817 IC50 = 11 nM T05090 CSC47W 118720522 IC50 = 223.6 nM T05090 CUI51W 118720529 IC50 = 28.7 nM T05090 CMV2W9 118721625 IC50 = 3 nM T05090 CF5TO3 118721859 IC50 = 49 nM T05090 CK97TZ 118721860 IC50 = 4 nM T05090 CYV30O 118721861 IC50 = 3 nM T05090 C5WYI1 118721862 IC50 = 5 nM T05090 CSMW25 118721863 IC50 = 897 nM T05090 C5B1KM 118721864 IC50 = 98 nM T05090 CG8LZ0 118721865 IC50 = 2710 nM T05090 CPCN23 118721866 IC50 = 2950 nM T05090 CM0A9U 118721867 IC50 = 2600 nM T05090 C8IAG9 118734664 IC50 = 12100 nM T05090 CJ6KL7 118734665 IC50 = 1970 nM T05090 C2VQ5P 118734666 IC50 = 10780 nM T05090 CYF71E 118734667 IC50 = 1490 nM T05090 CQC7H0 118734668 IC50 = 11230 nM T05090 CP27CN 118734669 IC50 = 1470 nM T05090 CBIY72 118734670 IC50 > 20 ug.mL-1 T05090 C9C7UX 118734705 IC50 = 19680 nM T05090 CI8G4X 118737400 IC50 = 80 nM T05090 C2F8TQ 118737455 IC50 = 532 nM T05090 CZ61KV 118753026 IC50 = 180 nM T05090 CFI23Y 118753027 IC50 = 930 nM T05090 C75LTK 118753189 IC50 = 3300 nM T05090 CB84TO 121278998 IC50 > 50000 nM T05090 C9S5OK 121279020 IC50 > 50000 nM T05090 CIA40K 121472983 IC50 > 10000 nM T05090 CL3M2F 121499152 IC50 = 2280 nM T05090 C93JAV 122177622 IC50 = 149 nM T05090 C5HJ0C 122177623 IC50 > 10000 nM T05090 CW4K2U 122181880 IC50 = 332.1 nM T05090 CK63UH 122181881 IC50 = 319.5 nM T05090 C0H9WU 122181882 IC50 = 2.31 nM T05090 CR3TU6 122181883 IC50 = 332.4 nM T05090 C57VRL 122181884 IC50 = 846.5 nM T05090 C81QDF 122182040 IC50 = 25.01 nM T05090 C2VO8E 122184845 IC50 = 16.65 nM T05090 CGSF80 122184846 IC50 = 21.62 nM T05090 CN4H8Q 122184847 IC50 = 4 nM T05090 CT94PN 122184848 IC50 = 5.42 nM T05090 CI2X8M 122184849 IC50 = 39.67 nM T05090 C5HOK3 122184850 IC50 = 21.2 nM T05090 CZC3Q4 122184851 IC50 = 17.63 nM T05090 CQW6T3 122184852 IC50 = 18.88 nM T05090 CE4M7C 122184853 IC50 = 192 nM T05090 C7MT9U 122184854 IC50 = 40.78 nM T05090 C4AQ5H 122184855 IC50 = 36 nM T05090 C07UQJ 122184856 IC50 = 13.95 nM T05090 CST56N 122184857 IC50 = 92.03 nM T05090 C6K1HJ 122184858 IC50 = 74.42 nM T05090 CG19IO 122185146 IC50 = 69.19 nM T05090 CI4U2H 122185147 IC50 = 107.7 nM T05090 CU47DI 122185148 IC50 = 275.74 nM T05090 C9XMU5 122185149 IC50 = 263.98 nM T05090 C5QCF0 122185150 IC50 = 176.48 nM T05090 CSA1H8 122185151 IC50 = 474.74 nM T05090 CZG70W 122185152 IC50 = 632.54 nM T05090 C28JVO 122192004 IC50 = 9.77 nM T05090 CF2D8U 122192005 IC50 = 3150 nM T05090 C5W8OZ 122376192 IC50 = 2.65 nM T05090 C3V5ND 122550211 IC50 = 439 nM T05090 CW03VD 126582837 IC50 = 65.08 nM T05090 C5UV6J 126582839 IC50 = 26.76 nM T05090 CR9AC4 126582841 IC50 = 113.45 nM T05090 C1HS3A 126582843 IC50 = 20.79 nM T05090 CFI58L 126582907 IC50 = 151.45 nM T05090 CMT02Y 126582908 IC50 > 10000 nM T05090 CE4CI8 127025178 IC50 = 29 nM T05090 CM38EU 127025541 IC50 = 68 nM T05090 C68TYH 127027490 IC50 = 470 nM T05090 CA14VM 127027506 IC50 = 3248.71 nM T05090 CB9PL5 127027507 IC50 > 10000 nM T05090 CBOJ07 127027508 IC50 > 10000 nM T05090 CT18SH 127027509 IC50 = 8861.76 nM T05090 CG7Q3V 127027808 IC50 = 13700 nM T05090 C6JUF9 127027813 IC50 > 30000 nM T05090 CG8NU7 127027995 IC50 = 11 nM T05090 CV07OM 127028943 IC50 = 23 nM T05090 CC6FD8 127034721 IC50 = 960 nM T05090 C4EH3T 127034722 IC50 = 3180 nM T05090 C2YXR7 127034902 IC50 > 5000 nM T05090 C9ZF0D 127035369 IC50 = 1550 nM T05090 C4GI0F 127037614 IC50 = 113 nM T05090 CZ8A1F 127041696 IC50 > 100000 nM T05090 C5D2OJ 127044292 IC50 = 5950 nM T05090 C58KRZ 127044343 IC50 = 19800 nM T05090 C1TYS6 127044344 IC50 = 25900 nM T05090 C3G0SM 127044498 IC50 = 5730 nM T05090 C5CP9M 127045259 IC50 = 6260 nM T05090 CB8HR2 129104138 IC50 > 50000 nM T05090 CCH65A 129104183 IC50 > 50000 nM T05090 CFH8Q4 129104227 IC50 > 50000 nM T05090 C6HM5P 129104349 IC50 > 50000 nM T05090 CZTF90 129104374 IC50 > 50000 nM T05090 CUJ2P5 129104402 IC50 > 50000 nM T05090 CY3I6X 129104426 IC50 > 50000 nM T05090 C2N5JD 132279660 IC50 > 10000 nM T05090 C4L6UZ 132547258 IC50 = 338 nM T05090 CGBR54 132547259 IC50 = 424 nM T05090 CW4MP2 132547260 IC50 = 356 nM T05090 C1YO2Z 132547261 IC50 = 35 nM T05090 CU63DV 132569672 IC50 = 311 nM T05090 C4KE3N 132938351 IC50 = 368 nM T05090 C4UAN3 134129876 IC50 = 333 nM T05090 C25EVA 134129883 IC50 = 59 nM T05090 CWRH43 134129994 IC50 = 191 nM T05090 CK2TM6 134130010 IC50 = 1020 nM T05090 CYW6H1 134130165 IC50 = 33 nM T05090 C8CY7S 134131006 IC50 = 283 nM T05090 CQ7SN8 134131102 IC50 = 256 nM T05090 CYCS54 134131113 IC50 = 722 nM T05090 CQO23I 134131456 IC50 = 181 nM T05090 CHZ8A3 134131564 IC50 = 224 nM T05090 CN9DL4 134132030 IC50 > 10000 nM T05090 CX93QK 134135812 IC50 > 100000 nM T05090 CN8L9J 134136160 IC50 = 530000 nM T05090 C53UTO 134137062 IC50 = 2000 nM T05090 CSX58U 134139437 IC50 > 10000 nM T05090 C75NRQ 134141877 IC50 > 100000 nM T05090 C62SVR 134142119 IC50 > 100000 nM T05090 CLI48U 134143743 IC50 = 5400 nM T05090 CUA26W 134143927 IC50 = 43000 nM T05090 CWRJ15 134147087 IC50 = 20200 nM T05090 C8K0XJ 134147090 IC50 = 280 nM T05090 CQ61SB 134150479 IC50 = 49200 nM T05090 CDX75O 134152551 IC50 = 10700 nM T05090 C2JV5X 134153768 IC50 > 100000 nM T05090 C38DIF 134156853 IC50 = 98000 nM T05090 C4FLQ5 134157355 IC50 > 100000 nM T05090 C1UP3S 134157845 IC50 = 1830 nM T05090 CZV43J 134283792 IC50 = 23000 nM T05090 C62WXO 134283796 IC50 = 37000 nM T05090 CO7K3N 134283799 IC50 = 6000 nM T05090 CBQ17L 134283800 IC50 = 27000 nM T05090 C1Y4TA 134283810 IC50 = 30000 nM T05090 CV2YF7 134283813 IC50 = 42000 nM T05090 C05FVT 134492522 IC50 > 10000 nM T05090 CS1V6A 135367138 IC50 > 50000 nM T05090 CVO59N 135367789 IC50 > 50000 nM T05090 CDY18W 135407493 IC50 > 100000 nM T05090 CW2I4R 135412048 IC50 > 100000 nM T05090 C7U0AV 135412194 IC50 > 100000 nM T05090 CS54TL 135437514 IC50 = 86400 nM T05090 C36MUC 135441620 IC50 > 100000 nM T05090 CRB8M1 135444536 IC50 > 100000 nM T05090 CX5D6J 135446479 IC50 = 15200 nM T05090 C1TOK2 135449197 IC50 > 100000 nM T05090 CW25GL 135462117 IC50 > 100000 nM T05090 CCL28F 135473106 IC50 > 100000 nM T05090 CYA60G 135497781 IC50 > 100000 nM T05090 C01EZF 135567459 IC50 = 68000 nM T05090 CV3QP4 135886613 IC50 = 25.6 nM T05090 C8X5LO 135928012 Ki = 120 nM T05090 CI2YE8 135928628 IC50 > 100000 nM T05090 C50NIS 136025837 IC50 > 100000 nM T05090 C4OS0V 136025842 IC50 > 100000 nM T05090 CX7Z5B 136025843 IC50 > 100000 nM T05090 CB8EM9 136025984 IC50 > 100000 nM T05090 C49MUG 136025986 IC50 > 100000 nM T05090 CH7Y3C 136086920 IC50 > 100000 nM T05090 C3VDL5 136086921 IC50 > 100000 nM T05090 C9GOB5 136086922 IC50 = 40000 nM T05090 CE3ZL7 136086923 IC50 > 100000 nM T05090 CJZ5F3 136086924 IC50 > 100000 nM T05090 CY9U0E 136173089 IC50 = 20 nM T05090 CXHY69 136230092 IC50 = 690 nM T05090 CWK9U7 136230093 IC50 = 410 nM T05090 C7X1UL 136645449 IC50 = 854 nM T05090 CA5OY1 137628667 IC50 = 45 nM T05090 C67EFJ 137628684 IC50 = 1.47 nM T05090 CX0PH5 137628685 IC50 = 654 nM T05090 CG23FD 137631444 IC50 = 10390 nM T05090 C9UQD2 137631509 IC50 > 30000 nM T05090 CP0JL9 137631552 IC50 > 30000 nM T05090 CHL7E8 137631592 IC50 = 8007 nM T05090 CJ9GD5 137631769 IC50 > 30000 nM T05090 CJ7P1U 137631803 IC50 = 227 nM T05090 CQ54WK 137631915 IC50 > 30000 nM T05090 CD1L0I 137632135 IC50 > 30000 nM T05090 C6A4GK 137632422 IC50 > 30000 nM T05090 CQ4BK9 137632561 IC50 > 30000 nM T05090 CVB93K 137632723 IC50 = 1800 nM T05090 C9RWF1 137632979 IC50 > 30000 nM T05090 CI2G7B 137633049 IC50 > 30000 nM T05090 CMU42D 137633092 IC50 > 30000 nM T05090 CY08AM 137633123 IC50 > 30000 nM T05090 C84MIY 137633138 IC50 = 3570 nM T05090 C1HL3I 137633415 IC50 > 30000 nM T05090 CM6V3G 137633491 IC50 = 65.05 nM T05090 C8G4KJ 137634562 IC50 > 30000 nM T05090 CJ76DN 137634596 IC50 > 30000 nM T05090 C7JK8D 137634598 IC50 = 356.9 nM T05090 C7U1CE 137634604 IC50 > 30000 nM T05090 C28CEY 137634881 IC50 = 67.54 nM T05090 C90TSR 137634950 IC50 > 30000 nM T05090 CHA4E3 137635225 IC50 = 1940 nM T05090 CBMN61 137635405 IC50 > 30000 nM T05090 CZ29MT 137635651 IC50 = 5170 nM T05090 COF8J3 137635708 IC50 = 223 nM T05090 C7N5BG 137635855 IC50 > 30000 nM T05090 C2MB4U 137636234 IC50 = 1010 nM T05090 CA2S3J 137636481 IC50 = 220 nM T05090 C5GCO8 137636604 IC50 > 30000 nM T05090 C72SBN 137636632 IC50 > 30000 nM T05090 C9THE6 137636891 IC50 > 30000 nM T05090 CF3E8T 137637310 IC50 > 30000 nM T05090 C0VNM5 137637430 IC50 = 144.07 nM T05090 C6MVX0 137637661 IC50 = 4150 nM T05090 C3H2GO 137637718 IC50 = 750 nM T05090 CSH08B 137637787 IC50 = 2550 nM T05090 CEI0W2 137637915 IC50 = 2900 nM T05090 CZU9E2 137637958 IC50 = 24.71 nM T05090 CMU93I 137637990 IC50 > 30000 nM T05090 C6X0AW 137638091 IC50 = 19.8 nM T05090 CMD89K 137638151 IC50 = 1800 nM T05090 CQ3DR6 137638257 IC50 = 1210 nM T05090 CO9UY1 137638342 IC50 > 30000 nM T05090 C3RC2O 137638626 IC50 > 30000 nM T05090 CEMX30 137638687 IC50 > 30000 nM T05090 CTG6X0 137638748 IC50 > 30000 nM T05090 CZU31H 137638926 IC50 = 850 nM T05090 CQ86FE 137638947 IC50 > 30000 nM T05090 C7IJC2 137639014 IC50 = 430 nM T05090 C2DIM1 137639536 IC50 = 600 nM T05090 CW4DJ8 137639563 IC50 > 30000 nM T05090 CS9A6C 137639566 IC50 > 30000 nM T05090 CMI6Z0 137639764 IC50 = 1030 nM T05090 COV42L 137639829 IC50 > 30000 nM T05090 CL02GC 137640047 IC50 = 1320 nM T05090 C19GDO 137640291 IC50 = 7.1 nM T05090 CGKA54 137640295 IC50 > 30000 nM T05090 C7VIL6 137640304 IC50 = 3100 nM T05090 C0Q3ZW 137640468 IC50 = 12600 nM T05090 C39FQX 137641152 IC50 > 30000 nM T05090 CSA84O 137641263 IC50 = 590 nM T05090 CI4PM3 137641395 IC50 > 30000 nM T05090 C4OEC3 137641520 IC50 = 1600 nM T05090 CS1K3I 137641616 IC50 > 30000 nM T05090 C38HXT 137641735 IC50 = 4940 nM T05090 CV19SL 137642038 IC50 > 30000 nM T05090 CAF1N9 137642211 IC50 = 64.51 nM T05090 C40JZA 137642448 IC50 > 30000 nM T05090 CY02GK 137642671 IC50 > 30000 nM T05090 CF42GI 137643288 IC50 = 152.46 nM T05090 CJOS87 137643760 IC50 = 96 nM T05090 C4V1WC 137643841 IC50 = 830 nM T05090 CB59SN 137643993 IC50 = 147 nM T05090 C7DLO4 137644089 IC50 = 5626 nM T05090 CC38FN 137644424 IC50 > 30000 nM T05090 CVQ4J0 137644605 IC50 > 30000 nM T05090 CX37VS 137644658 IC50 > 30000 nM T05090 CCBN61 137645084 IC50 = 30850 nM T05090 CPL3J1 137645258 IC50 > 30000 nM T05090 C8XAR3 137645372 IC50 > 30000 nM T05090 C05LHW 137645511 IC50 > 30000 nM T05090 CX3E0H 137645675 IC50 = 138 nM T05090 C5REZ8 137645689 IC50 > 20000 nM T05090 CYSU67 137645967 IC50 > 30000 nM T05090 C8HKU4 137646033 IC50 = 98.79 nM T05090 CV7F6C 137646133 IC50 = 180 nM T05090 CMJ7D9 137646202 IC50 > 30000 nM T05090 CN08DL 137646214 IC50 > 30000 nM T05090 CNT3Y7 137647005 IC50 = 196.62 nM T05090 C4I9YE 137647260 IC50 = 5210 nM T05090 CX8C9V 137647325 IC50 > 30000 nM T05090 CHW8X4 137647384 IC50 > 30000 nM T05090 C5AFM1 137647889 IC50 = 50.27 nM T05090 CZ2RN9 137647935 IC50 > 30000 nM T05090 CO7H5A 137648171 IC50 = 151800 nM T05090 C5IK9F 137648357 IC50 = 215.48 nM T05090 C8S2TO 137648573 IC50 = 4310 nM T05090 C0VAB8 137648585 IC50 > 30000 nM T05090 CPK7Y5 137648623 IC50 = 5290 nM T05090 CL0XW1 137648762 IC50 = 660 nM T05090 CR0P6Z 137648837 IC50 = 910 nM T05090 CN3I9X 137648982 IC50 = 90 nM T05090 CG2PL8 137648996 IC50 = 3210 nM T05090 C05DNH 137649390 IC50 > 30000 nM T05090 CO20AE 137649565 IC50 > 30000 nM T05090 C0PGD9 137649617 IC50 = 62540 nM T05090 CH0ES8 137650022 IC50 > 30000 nM T05090 C4MC5X 137650991 IC50 > 30000 nM T05090 C4GNA5 137651338 IC50 > 30000 nM T05090 C8PWX1 137651771 IC50 > 30000 nM T05090 CGE1Z5 137651786 IC50 = 8710 nM T05090 CD89ZR 137651966 IC50 > 30000 nM T05090 C3EQ0D 137651991 IC50 = 33.77 nM T05090 CT05IE 137651994 IC50 = 570 nM T05090 CH3B5G 137652131 IC50 > 30000 nM T05090 C5FHD3 137652442 IC50 = 12500 nM T05090 CMP7G0 137652638 IC50 = 167 nM T05090 C83RBI 137652888 IC50 = 2570 nM T05090 CPI06O 137652951 IC50 = 133.06 nM T05090 C61VOF 137653427 IC50 = 490 nM T05090 C1OAE9 137654162 IC50 = 950 nM T05090 CFQ4T2 137654668 IC50 > 30000 nM T05090 C1SBN5 137654946 IC50 = 6530 nM T05090 CLWF87 137655165 IC50 > 30000 nM T05090 CS50BH 137655597 IC50 > 30000 nM T05090 CIA0V1 137656228 IC50 > 30000 nM T05090 CVG9T3 137656290 IC50 = 19 nM T05090 C0EQI2 137656898 IC50 = 42.9 nM T05090 C76OGQ 137656942 IC50 = 24000 nM T05090 C5BM7T 137657586 IC50 = 110 nM T05090 C97QUM 137657678 IC50 = 243 nM T05090 C21XDS 137657845 IC50 = 5800 nM T05090 CN0C1E 137658519 IC50 > 30000 nM T05090 COC9D2 137658833 IC50 > 30000 nM T05090 CPJL30 137659007 IC50 = 261 nM T05090 CFGW13 137659898 IC50 = 667 nM T05090 C7JGX8 137660397 IC50 = 45.55 nM T05090 C3Q7PX 137660404 IC50 = 1030 nM T05090 C02BSL 137661253 IC50 = 99.87 nM T05090 CQAY45 137662133 IC50 = 4290 nM T05090 CYZ43W 137662281 IC50 = 21.37 nM T05090 CAQ62X 137701235 Ki = 12 nM T05090 CIWG23 138393067 IC50 = 430 nM T05090 C7EM3I 138393071 IC50 = 4150 nM T05090 C4NFS3 138393072 IC50 = 178.3 nM T05090 CIT72O 139302883 IC50 = 3.78 nM T05090 CN1TH8 139302889 IC50 = 189 nM T05090 C0R1MD 139302991 IC50 = 42.51 nM T05090 C3GJQ8 139303021 IC50 = 17.06 nM T05090 CN73DV 139303049 IC50 = 260 nM T05090 CFAU90 139303050 IC50 = 38.41 nM T05090 CKQB30 139303051 IC50 = 13.88 nM T05090 CN2UH1 139303146 IC50 = 3.02 nM T05090 CE81VG 139303149 IC50 = 2.54 nM T05090 C9DJ3B 139303559 IC50 = 11.35 nM T05090 CP73QO 141504704 IC50 = 660 nM T05090 CX0E9B 142505968 IC50 = 10600 nM T05090 CBJC50 142505992 IC50 = 7075 nM T05090 C7N8LV 142506025 IC50 = 1031 nM T05090 CKBF56 142506033 IC50 = 427 nM T05090 CLND62 142506170 IC50 > 100000 nM T05090 CGNQ74 142506189 IC50 = 6699 nM T05090 C1T3IQ 142506210 IC50 = 2400 nM T05090 CXJ0Y4 145949850 IC50 = 32 nM T05090 CKG98W 145953085 IC50 > 30000 nM T05090 CBNG29 145957781 IC50 = 64 nM T05090 CK1XI0 145960971 IC50 > 10000 nM T05090 C3PWD4 145964064 IC50 = 2050 nM T05090 CDY56B 145964885 IC50 = 232 nM T05090 CJAE67 145966594 IC50 = 3910 nM T05090 C19POY 145967140 IC50 = 5090 nM T05090 CSJ81Y 145968726 IC50 = 59.6 nM T05090 CI43DY 145970786 IC50 > 100000 nM T05090 CO51JK 145973368 IC50 = 11.1 nM T05090 C4HTO2 145973543 IC50 = 861 nM T05090 CVM0Z3 145974125 IC50 = 2560 nM T05090 C8YEJ9 145974425 IC50 = 4400 nM T05090 CE8I5V 145975869 IC50 = 323 nM T05090 CMUA94 145976675 IC50 = 891 nM T05090 CN6UO4 145977003 IC50 = 996 nM T05090 CKAQ67 145977127 IC50 = 6050 nM T05090 COR40V 145978805 IC50 = 6620 nM T05090 C9BJW3 145979532 IC50 = 164 nM T05090 CZ7IQ9 145979841 IC50 = 0.41 nM T05090 C0UG8S 145980171 IC50 = 1220 nM T05090 CMB08D 145981960 IC50 = 60.3 nM T05090 C9VDE5 145982499 IC50 = 340 nM T05090 CKYP15 145982514 IC50 = 11780 nM T05090 CX2LY1 145982614 IC50 = 9320 nM T05090 C0SHF9 145982778 IC50 = 12000 nM T05090 CR63YW 145983218 IC50 = 100 nM T05090 C6OL1K 145983267 IC50 = 544 nM T05090 CE38WZ 145983432 IC50 = 1300 nM T05090 CPUJ75 145983482 IC50 = 27310 nM T05090 CWD0A9 145983712 Ki = 0.8 nM T05090 C2I7EQ 145983818 IC50 = 18830 nM T05090 CV8H2B 145983876 IC50 = 25380 nM T05090 C3I6VL 145983950 IC50 = 780 nM T05090 C7FBZ5 145984102 IC50 = 34860 nM T05090 CIWO70 145984314 IC50 = 1810 nM T05090 C9ZKC1 145984665 IC50 = 1890 nM T05090 CSA1K8 145984949 IC50 = 37190 nM T05090 CT50ZG 145985100 IC50 = 1600 nM T05090 CFLH65 145985111 IC50 = 24610 nM T05090 CN6KB9 145985243 IC50 = 160 nM T05090 CK90XR 145985933 IC50 = 100 nM T05090 CBF13W 145985947 IC50 = 5330 nM T05090 C56MWZ 145986208 Ki = 58 nM T05090 CL62QV 145986214 IC50 = 2650 nM T05090 CGN02Q 145986264 IC50 = 990 nM T05090 C51BUM 145986322 IC50 = 0.75 nM T05090 C82CIN 145988785 IC50 = 1500 nM T05090 CHR0U9 145990400 IC50 = 1.3 nM T05090 C68VKC 145993051 IC50 = 1190 nM T05090 C1W6CF 145994016 IC50 = 23000 nM T05090 C0GMR1 146585718 IC50 = 10990 nM T05090 C0YXS8 147254231 IC50 = 3951 nM T05090 CN71OS 149405396 IC50 = 1973 nM T05090 C9FIY4 153534005 IC50 = 75 nM T05090 CB8RS9 155512087 IC50 > 25000 nM T05090 CQ5BL7 155512551 IC50 > 50000 nM T05090 CPF6R7 155512997 IC50 = 213 nM T05090 CE4H7I 155513471 IC50 > 50000 nM T05090 CW3VT9 155514603 IC50 > 50000 nM T05090 CZ84WI 155515284 IC50 > 50000 nM T05090 CUKG21 155515602 IC50 > 50000 nM T05090 CY2DC1 155515836 IC50 = 148 nM T05090 CYJ53T 155515864 IC50 = 20000 nM T05090 CA1J3N 155517086 IC50 = 126 nM T05090 CEH2N5 155518106 IC50 = 235 nM T05090 C41AIO 155518963 IC50 > 1000 nM T05090 CDY5H6 155519645 IC50 = 1440 nM T05090 CAZ3S7 155521187 IC50 = 18000 nM T05090 CZ75FW 155521272 IC50 = 96 nM T05090 CEQ58R 155523224 IC50 = 83 nM T05090 CNW0D1 155524821 IC50 = 76 nM T05090 CN7B1T 155525782 IC50 > 100000 nM T05090 CHR4K5 155528532 IC50 > 100000 nM T05090 C0IC6W 155528706 IC50 = 146 nM T05090 CZ70PO 155529066 IC50 > 50000 nM T05090 C49NGT 155529137 IC50 > 50000 nM T05090 CZMC49 155530597 IC50 = 1.3 nM T05090 COTR30 155530602 IC50 = 708 nM T05090 CN3W5J 155531452 IC50 > 50000 nM T05090 CKV01F 155531688 IC50 = 380 nM T05090 CK2UY4 155531957 IC50 = 50000 nM T05090 CV2C8O 155532194 IC50 = 290 nM T05090 C1F4DU 155533216 IC50 = 680 nM T05090 CIZ46A 155533876 IC50 > 30000 nM T05090 CJH9L4 155535498 IC50 = 503 nM T05090 CAG9P4 155537573 IC50 > 50000 nM T05090 CLD19W 155539311 IC50 = 2060 nM T05090 CU6V4Q 155539319 IC50 > 50000 nM T05090 CP9O4L 155539654 IC50 = 2700 nM T05090 CE6G4A 155539837 IC50 = 16.29 nM T05090 C6U0FM 155540189 IC50 = 26000 nM T05090 CKZ9A5 155543845 IC50 = 276 nM T05090 CP4L1F 155544459 IC50 > 50000 nM T05090 C1VF5A 155544728 IC50 = 213 nM T05090 CXR86J 155545078 IC50 > 50000 nM T05090 CF2O4J 155546325 IC50 > 50000 nM T05090 C0AU1L 155546632 IC50 > 50000 nM T05090 CEF69A 155546817 IC50 = 185 nM T05090 C90FBZ 155549087 IC50 > 50000 nM T05090 CCTU12 155549163 IC50 > 1000 nM T05090 CE0YL6 155549538 IC50 = 30 nM T05090 CFA01C 155549905 IC50 = 148 nM T05090 C4Z5JX 155550827 IC50 = 50000 nM T05090 C05ZVG 155552130 IC50 = 10900 nM T05090 C46WHP 155552329 IC50 > 1000 nM T05090 CS5D0O 155552399 IC50 = 410 nM T05090 CV4Y5B 155552792 IC50 = 160 nM T05090 CGDF76 155554360 IC50 = 24000 nM T05090 CC56ED 155554844 IC50 = 1.7 nM T05090 CXGR50 155555191 IC50 = 60 nM T05090 CFW90N 155555562 IC50 = 4.21 nM T05090 C7QTU1 155555957 IC50 > 50000 nM T05090 CIN57Q 155556138 IC50 = 34 nM T05090 C0IO1Q 155557341 IC50 = 125 nM T05090 CJ9FW6 155557777 IC50 = 374 nM T05090 CJ3MZ1 155558467 IC50 = 372 nM T05090 C8AUB0 155558567 IC50 = 112 nM T05090 C0RZ7V 155558710 IC50 > 1000 nM T05090 C28CVZ 155559279 IC50 = 132 nM T05090 CPD50Q 155559583 IC50 = 1000 nM T05090 CY3XI1 155559600 IC50 > 1000 nM T05090 C4EQ8P 155561585 IC50 = 260 nM T05090 CGL24S 155562249 IC50 > 50000 nM T05090 C4IM1X 155564305 IC50 = 492 nM T05090 CPNA06 155564750 IC50 > 50000 nM T05090 CE0U7K 155564881 IC50 > 1000 nM T05090 CZDC03 155565491 IC50 > 30000 nM T05090 CG65CR 155565674 IC50 = 50000 nM T05090 C3G1JV 155565712 IC50 > 1000 nM T05090 CD05RS 155566122 IC50 = 43000 nM T05090 C4A0RK 155566461 IC50 > 50000 nM T05090 C04CGS 155567444 IC50 > 50000 nM T05090 CS03PJ 155568350 IC50 > 50000 nM T05090 CW5XB4 155569484 IC50 = 60.3 nM T05090 C3BAZ5 24861442 IC50 = 23.9 nM T05090 D00GBB 11449246 Ki = 23 nM T05090 D00HFS 46884057 IC50 = 114 nM T05090 D00HXX 56650312 IC50 = 80 nM T05090 D00SEE 11379392 IC50 = 201 nM T05090 D01FYB 23648267 IC50 > 20000 nM T05090 D01YBR 44591988 IC50 = 4080 nM T05090 D02NWS 279980 Ki = 1650 nM T05090 D03QOD 239512 IC50 > 50000 nM T05090 D04DOL 25032059 IC50 = 7 nM T05090 D04KQF 6675804 Ki = 275 nM T05090 D04UVL 1133083 IC50 = 3640 nM T05090 D05OVV 11993691 IC50 = 350 nM T05090 D07YZZ 5173 Ki = 125 nM T05090 D0B3ZM 11436024 IC50 = 725 nM T05090 D0E0TA 44454650 IC50 > 50000 nM T05090 D0E9DD 16095101 IC50 = 80 nM T05090 D0H7QA 46884056 IC50 = 58 nM T05090 D0K7QR 45269423 IC50 = 18 nM T05090 D0L6YF 46884016 IC50 = 137 nM T05090 D0M9LJ 44454415 IC50 = 11350 nM T05090 D0MD7H 44454143 IC50 = 11000 nM T05090 D0N9AK 44138031 IC50 = 2800 nM T05090 D0Q2CC 46884055 IC50 = 1348 nM T05090 D0Q2GM 44454416 IC50 = 7300 nM T05090 D0Q5DI 71462653 IC50 = 6680 nM T05090 D0Q5MC 24753719 IC50 > 30000 nM T05090 D0R7JA 53344908 IC50 > 43000 nM T05090 D0T0SK 44138032 IC50 = 160 nM T05090 D0T4JQ 264 IC50 = 9000 nM T05090 D0U8FC 759408 IC50 = 2800 nM T05090 D0W1PV 6918328 Ki = 0.26 nM T05090 D0XZ9Q 11149404 IC50 = 110 nM T05090 D0YO6M 785232 IC50 = 1400 nM T05090 D0Z8PX 24757913 IC50 = 245 nM T69563 D07DCG 71657455 IC50 = 7.5 nM T69563 D07GRH 2749 Ki > 50000 nM T69563 D07VYP 118955396 IC50 = 9 nM T69563 D0C6RM 118310260 IC50 < 10 nM T69563 D0K7FT 89683805 IC50 = 4950 nM T69563 D0K9PC 117817422 IC50 = 0.04 nM T69563 D0RZ9V 90415637 IC50 = 18 nM T69563 CK0JI9 1548955 IC50 = 37860 nM T69563 CV7YQ1 2942796 IC50 = 50000 nM T69563 CS9M6R 3047730 Ki > 50000 nM T69563 C4J5IH 3201893 IC50 = 1800 nM T69563 C0E2RO 3202856 IC50 = 390 nM T69563 CASM49 4016538 IC50 = 410 nM T69563 CY0CO2 5495925 Ki = 12000 nM T69563 C0Q3DC 5760176 Ki > 50000 nM T69563 COI9V5 10389037 IC50 = 270 nM T69563 C3V7MQ 13590964 Ki = 120 nM T69563 C2L5SU 13590965 Ki > 50000 nM T69563 CL5JD4 15187131 Ki = 30000 nM T69563 CN17UX 19287893 Ki > 50000 nM T69563 CG0XH9 20158121 Ki = 870 nM T69563 CX61GC 21520193 Ki > 50000 nM T69563 CBM72Z 25220414 Ki = 16700 nM T69563 C5IW0T 25361650 IC50 = 51400 nM T69563 C5TP6Y 44203254 Ki = 17400 nM T69563 CGCJ16 44541205 Ki = 30000 nM T69563 CPR67J 44541206 Ki > 50000 nM T69563 CCE93X 44541208 Ki > 50000 nM T69563 C3V2US 44543378 Ki = 50000 nM T69563 C3L5JM 45270871 IC50 = 1280 nM T69563 C2ILY9 46952127 IC50 = 704 nM T69563 CFG83B 46958630 IC50 = 3320 nM T69563 CKA58Y 46958631 IC50 = 238 nM T69563 CNP8Y2 54618317 IC50 = 190 nM T69563 CPL7Z4 54619107 IC50 = 6300 nM T69563 CFV27I 54619142 IC50 = 1700 nM T69563 C62ZPY 54619179 IC50 = 5300 nM T69563 CGE50Y 54619189 IC50 = 1000 nM T69563 CBP21C 54619212 IC50 = 3900 nM T69563 CQ4CZ7 54619246 IC50 = 600 nM T69563 C59QBG 54619248 EC50 = 300 nM T69563 C45IFU 54619285 IC50 > 20000 nM T69563 CO01JZ 54621040 IC50 = 550 nM T69563 CHY23G 54621327 IC50 = 91 nM T69563 C14LSD 54630941 IC50 = 6400 nM T69563 C48KIZ 54631125 IC50 = 37 nM T69563 CDO2I1 56645146 IC50 = 60 nM T69563 CFC0N1 56645147 IC50 = 60 nM T69563 CV90CE 56645355 IC50 = 80 nM T69563 C3WB8U 56645356 IC50 = 20 nM T69563 C2XV4G 56645357 IC50 = 40 nM T69563 C2AG6K 56646155 IC50 = 140 nM T69563 CPK0W1 56646779 IC50 = 50 nM T69563 C7RNB0 56832448 IC50 = 860 nM T69563 CFU0G9 56832449 IC50 < 100 nM T69563 CFK30C 56844254 IC50 > 57000 nM T69563 C4TE8X 56923423 IC50 = 50 nM T69563 C8LDQ3 66664967 IC50 = 7800 nM T69563 CX7PG5 66665307 IC50 = 900 nM T69563 C2P4KZ 66665324 IC50 = 5640 nM T69563 CS3U4V 68056458 IC50 = 640 nM T69563 CN0X4D 68056459 IC50 = 60 nM T69563 C7UET3 68056593 IC50 = 40 nM T69563 CRN8L7 68056678 IC50 = 420 nM T69563 C7I8YC 68057381 IC50 > 11000 nM T69563 CPBU43 68057382 IC50 = 80 nM T69563 C9OS2V 68057395 IC50 = 240 nM T69563 CEF19C 68057634 IC50 = 60 nM T69563 CNW1D3 71452045 IC50 = 1100 nM T69563 C8U2OI 71452046 IC50 = 1400 nM T69563 CE0WX3 71453859 IC50 = 3600 nM T69563 CR93TM 71453860 IC50 > 100000 nM T69563 C76JOC 71455563 IC50 = 1270 nM T69563 CBR65Z 71457355 IC50 = 1630 nM T69563 C9ZJR0 71457380 IC50 = 450 nM T69563 CV09MQ 71459238 IC50 = 290 nM T69563 CR8ZV7 71460994 IC50 = 140 nM T69563 C16IGX 71461015 IC50 = 2880 nM T69563 C6H5EQ 71461016 IC50 = 53100 nM T69563 CJ6VF9 71462745 IC50 = 570 nM T69563 C60AFH 71462746 IC50 = 190 nM T69563 C0YX6L 71462747 IC50 > 100000 nM T69563 C5K4SM 71533725 IC50 > 57000 nM T69563 C2A5LR 71541908 IC50 = 36 nM T69563 CX6HR5 71542283 IC50 = 39 nM T69563 C24FVX 71542286 IC50 = 14 nM T69563 C3U5RS 71606602 IC50 = 1580 nM T69563 CL4DW0 71816506 Ki = 270 nM T69563 C4H2SI 71816677 Ki = 270 nM T69563 C6JY3X 71816678 Ki = 2400 nM T69563 CO4UL8 73354948 Ki = 120 nM T69563 C8W5JL 73427242 IC50 = 11 nM T69563 C92IJQ 86268389 IC50 = 33 nM T69563 CPJ76F 86269829 IC50 = 4 nM T69563 CCKB17 86269832 IC50 = 30 nM T69563 C5GO6B 86270015 IC50 = 240 nM T69563 CLM23D 86299415 IC50 = 8.45 nM T69563 CEIX57 86299748 IC50 < 100 nM T69563 CO0E9H 86580656 IC50 = 1 nM T69563 CK0DO7 89479018 IC50 = 610 nM T69563 CR2CN8 89489859 IC50 = 94 nM T69563 CBP73I 89489907 IC50 = 820 nM T69563 CK7HO6 89489971 IC50 = 8800 nM T69563 C8J3EW 89684116 IC50 = 78 nM T69563 CR9TK5 89699486 IC50 = 8 nM T69563 C9X0CZ 89699544 IC50 < 100 nM T69563 C43NDF 89699781 IC50 < 100 nM T69563 CC2U5B 89700010 IC50 < 100 nM T69563 CAH2X0 89700075 IC50 < 100 nM T69563 CT1SH4 89700209 IC50 < 100 nM T69563 CFR82W 89711418 IC50 < 100 nM T69563 C21EGI 90422240 IC50 = 10.9 nM T69563 CM51KW 90452084 IC50 = 24 nM T69563 C4CO1H 90454346 IC50 = 22 nM T69563 C2ZPL7 90454349 IC50 = 15 nM T69563 CU12EN 90458225 IC50 < 100 nM T69563 CX7F2H 90466415 IC50 = 4 nM T69563 C5R3IX 91864709 IC50 = 4.6 nM T69563 C1P4KD 97161268 IC50 = 70 nM T69563 CO34YI 101884787 Ki = 150 nM T69563 C7NQB8 101884789 Ki = 340 nM T69563 CL03EK 101884790 Ki = 140 nM T69563 CFO13M 101884791 Ki = 950 nM T69563 CA1V7W 101884792 Ki = 380 nM T69563 C2B8SY 101884793 Ki = 250 nM T69563 CL9ZV3 101884794 Ki = 140 nM T69563 CF3HU5 101884795 Ki = 5600 nM T69563 CP4JS6 101884796 Ki = 4500 nM T69563 CHY62S 117603922 Ki > 50000 nM T69563 CK0NU9 117817076 IC50 = 2 nM T69563 CTA4U5 117817125 IC50 = 4 nM T69563 CM0W3N 117817132 IC50 = 1 nM T69563 CO4E9M 117817141 IC50 = 0.7 nM T69563 CFQ7I2 117817149 IC50 = 7 nM T69563 CI6BN3 117817339 IC50 = 0.25 nM T69563 CGRI81 117817435 IC50 = 0.3 nM T69563 C2R6FU 117817465 IC50 < 50 nM T69563 CXO21M 117817521 IC50 < 50 nM T69563 C3SPF6 117817536 IC50 < 50 nM T69563 CHOA78 117817538 IC50 < 50 nM T69563 C24YMC 118290999 IC50 = 110 nM T69563 CX1E9U 118291067 IC50 > 10000 nM T69563 C1L4YQ 118291499 IC50 = 210 nM T69563 C42UWZ 118291506 IC50 = 1500 nM T69563 CF6ZP1 118291647 IC50 = 1770 nM T69563 CQ78GD 118291683 IC50 = 8000 nM T69563 CJYC54 118310293 IC50 < 10 nM T69563 C89HIP 118310540 IC50 < 10 nM T69563 CK1GM4 118310766 IC50 < 10 nM T69563 CVC47U 118704643 IC50 = 2220 nM T69563 CE1F9G 118716664 IC50 = 7.27 nM T69563 CE8P7S 118716665 IC50 = 194 nM T69563 C4OHN1 118717060 Ki > 50000 nM T69563 CYK47T 118717061 Ki > 50000 nM T69563 CLS3X4 118717062 Ki = 46000 nM T69563 C20HYE 118717063 Ki > 50000 nM T69563 CW86RL 118717064 Ki > 50000 nM T69563 C6INW2 118717065 Ki > 50000 nM T69563 CI0G3J 118717066 Ki > 50000 nM T69563 CB8G2F 118717067 Ki = 10000 nM T69563 CWHK89 118717068 Ki = 27000 nM T69563 CJ9FT2 118717069 Ki = 4500 nM T69563 CCUM32 118717070 Ki = 9500 nM T69563 C0GAK8 118717071 Ki = 16200 nM T69563 CA94XC 118717072 Ki = 13600 nM T69563 CLRI67 118717073 Ki = 5500 nM T69563 CYOP14 118717074 Ki = 560 nM T69563 CNO9A8 118717075 Ki = 490 nM T69563 CKGO91 118717076 Ki = 650 nM T69563 C2CEK1 118717077 Ki = 2200 nM T69563 CY96SX 118717078 Ki = 2200 nM T69563 CMD28R 118717079 Ki = 12500 nM T69563 C1CT8Z 118717080 Ki = 1600 nM T69563 CU65HC 118717081 Ki > 50000 nM T69563 CM9R7E 118717082 Ki = 8500 nM T69563 C63RNW 118717083 Ki = 3200 nM T69563 C1VG8Y 118717084 Ki = 3100 nM T69563 CI5GF3 118717085 Ki = 600 nM T69563 C3YOI1 118717086 Ki = 750 nM T69563 C1AK2U 118717087 Ki = 950 nM T69563 CW36LO 118717088 Ki = 40500 nM T69563 CW4B7P 118717089 Ki = 27500 nM T69563 C14MZQ 118717090 Ki = 22500 nM T69563 CW23YJ 118717091 Ki = 270 nM T69563 CUH05G 118717092 Ki = 300 nM T69563 C6TRH5 118717093 Ki = 3800 nM T69563 CTCY15 118717094 Ki > 50000 nM T69563 CTC48X 118953591 IC50 = 1 nM T69563 C2F0HL 118953746 IC50 = 293 nM T69563 C3FH8U 118953752 IC50 = 9 nM T69563 CGV23R 118953762 IC50 = 43 nM T69563 CAY4W1 118953816 IC50 = 36.5 nM T69563 CIQ51N 118953858 IC50 = 18 nM T69563 C2TCK0 118953878 IC50 = 4 nM T69563 C6TS3A 118953907 IC50 < 10 nM T69563 C0LK2C 118953916 IC50 = 53 nM T69563 COYJ23 118954160 IC50 < 10 nM T69563 CT6ML1 118955389 IC50 = 223 nM T69563 CZ47QL 118955394 IC50 < 2 nM T69563 CS2GZ7 118955397 IC50 = 40.3 nM T69563 C90ETU 118955405 IC50 = 25 nM T69563 C8K1UB 118955416 IC50 = 358 nM T69563 CNWT10 118955424 IC50 = 4 nM T69563 C7NH0V 118955426 IC50 = 8 nM T69563 CV7SM5 118955430 IC50 = 694 nM T69563 CL3E8F 118955433 IC50 < 2 nM T69563 C2HF8P 118955448 IC50 = 160 nM T69563 C64OGA 118955458 IC50 = 64.7 nM T69563 C6L4WS 118955554 IC50 = 127 nM T69563 CJY41H 118955555 IC50 < 10 nM T69563 C0JMT1 118955563 IC50 = 998 nM T69563 CHF8G7 118955568 IC50 = 147 nM T69563 C63JBM 118955570 IC50 = 132 nM T69563 COUV04 118955574 IC50 = 6300 nM T69563 CNS5J9 118955576 IC50 = 1710 nM T69563 C2Z4XH 118955582 IC50 = 54 nM T69563 CV3O8K 118955589 IC50 = 455 nM T69563 C0EMW9 118955592 IC50 = 3710 nM T69563 CVIO61 118955597 IC50 = 32 nM T69563 C8Y2JP 118955601 IC50 = 267 nM T69563 C7ZD3C 118955606 IC50 = 16 nM T69563 C5K3BL 118955607 IC50 < 10 nM T69563 CC27OH 118955611 IC50 = 188 nM T69563 CG61SY 118955613 IC50 = 53 nM T69563 CBL1E3 118955615 IC50 = 481 nM T69563 CQI31L 118955618 IC50 = 56 nM T69563 C2JZ9E 118955625 IC50 = 316 nM T69563 C0I1AG 118955638 IC50 = 303 nM T69563 CWC9E0 118955642 IC50 = 23 nM T69563 CAUM15 118955650 IC50 = 225 nM T69563 C9ZR3Y 118955663 IC50 = 3480 nM T69563 C86JQU 118955667 IC50 = 138 nM T69563 CIDZ73 118955672 IC50 = 13 nM T69563 C4NF7Z 118955679 IC50 = 668 nM T69563 COU0K5 118955687 IC50 = 69 nM T69563 C2N8CB 118955691 IC50 = 913 nM T69563 C1W6RT 118955698 IC50 = 464 nM T69563 C5RCP1 118955701 IC50 = 77 nM T69563 COS41X 118955712 IC50 = 3110 nM T69563 C1XWG9 118955715 IC50 = 140 nM T69563 C5XVE9 118955721 IC50 = 76 nM T69563 CT24YZ 118955730 IC50 = 995 nM T69563 C5XLV0 118955734 IC50 = 382 nM T69563 CW81VD 118955741 IC50 = 231 nM T69563 CR74DW 118955742 IC50 = 9670 nM T69563 CLA3U0 118955743 IC50 = 487 nM T69563 CK2U0H 118955980 IC50 = 100.2 nM T69563 C15GHE 118956024 IC50 = 295 nM T69563 CH39KW 118956036 IC50 = 19300 nM T69563 CNL73Q 118956065 IC50 = 147 nM T69563 CQ5A6C 118956067 IC50 = 92 nM T69563 CW5A8Z 118956116 IC50 = 25000 nM T69563 CTQO83 118956124 IC50 = 344 nM T69563 CC60WG 118956129 IC50 = 365 nM T69563 C5T8NV 118956132 IC50 = 72 nM T69563 CYN69B 118956147 IC50 = 17 nM T69563 CT6X2G 118956170 IC50 = 1260 nM T69563 CK26OG 118956187 IC50 = 185.1 nM T69563 C5YNM0 118956202 IC50 = 5200 nM T69563 CKP1O6 118956227 IC50 = 20 nM T69563 CT58YU 121225870 IC50 > 57000 nM T69563 C2OV0L 121457603 IC50 > 57000 nM T69563 CB80PQ 121457701 IC50 > 57000 nM T69563 CLKW12 121457751 IC50 = 47400 nM T69563 C6ZTQ1 121457762 IC50 > 57000 nM T69563 CT82GB 121461607 IC50 = 33500 nM T69563 C1LDQ5 121461684 IC50 > 57000 nM T69563 CW62PD 121461708 IC50 > 57000 nM T69563 CEY1H9 121461710 IC50 = 33500 nM T69563 C42KHQ 121461721 IC50 > 57000 nM T69563 C2WU8I 121461723 IC50 > 57000 nM T69563 C1OZ2D 121461729 IC50 = 47400 nM T69563 COED87 121461743 IC50 > 57000 nM T69563 CT7PM0 121461757 IC50 > 57000 nM T69563 CV3L8S 121461774 IC50 > 57000 nM T69563 CMS1Q6 121461818 IC50 > 57000 nM T69563 CJG3D2 121461820 IC50 = 47400 nM T69563 CW8R2L 121461821 IC50 = 26600 nM T69563 CAM9R6 122186444 Ki > 50000 nM T69563 C2VYR3 122186445 Ki > 50000 nM T69563 CKX7M4 122186446 Ki = 13400 nM T69563 CC0P2W 122186447 Ki > 50000 nM T69563 CX9I1G 122186448 Ki > 50000 nM T69563 C0KT5U 122186449 Ki = 4800 nM T69563 CKP7G9 122186450 Ki = 9200 nM T69563 COG86J 122186451 Ki = 3600 nM T69563 CUC87V 122186452 Ki = 25000 nM T69563 CU5K8E 122186453 Ki = 750 nM T69563 C06PJL 122186454 Ki = 7800 nM T69563 C7QU8K 122186455 Ki = 420 nM T69563 CV3O7K 122186456 Ki > 50000 nM T69563 C1YDE3 122186457 Ki > 50000 nM T69563 C37CMN 122186458 Ki = 470 nM T69563 CGND61 122186459 Ki = 4600 nM T69563 CB81IV 122186460 Ki = 4300 nM T69563 C4UT5O 122186461 Ki = 5900 nM T69563 CJD79O 122186462 Ki = 25300 nM T69563 C2LNI6 122186463 Ki > 50000 nM T69563 C4C5QG 122186464 Ki = 34200 nM T69563 COT4C2 122186465 Ki = 11300 nM T69563 C80UNC 122186466 Ki = 2600 nM T69563 CPF8Q6 122186467 Ki = 9200 nM T69563 CGH60B 122186468 Ki > 50000 nM T69563 C0HB1P 122186469 Ki = 5600 nM T69563 CUO13Z 122186470 Ki = 3200 nM T69563 CAW9R2 122186471 Ki > 50000 nM T69563 CD26IH 122186472 Ki = 3100 nM T69563 CDC3Y1 122186473 Ki > 50000 nM T69563 C5AZ1C 122186474 Ki > 50000 nM T69563 CUJT30 122186477 Ki = 16500 nM T69563 C1AU6W 126540084 IC50 < 100 nM T69563 C3BR0C 126540358 IC50 < 100 nM T69563 C6O4DK 126540561 IC50 < 100 nM T69563 CA91IL 129080665 IC50 < 10 nM T69563 CEG3X2 129080727 IC50 < 10 nM T69563 CP5K7B 129080745 IC50 < 10 nM T69563 C5DOP3 129102401 IC50 = 3.5 nM T69563 CSH3V4 130356715 IC50 = 2 nM T69563 CY65ND 130418263 IC50 > 10000 nM T69563 C45PYN 130469646 IC50 < 100 nM T69563 CL01PO 130469826 IC50 < 100 nM T69563 CCMJ13 131955127 IC50 = 29800 nM T69563 C4BRM1 132212317 IC50 = 8.89 nM T69563 C1JK0W 132219367 IC50 < 100 nM T69563 CM81VB 132219371 IC50 < 100 nM T69563 CPM48R 132219770 IC50 < 100 nM T69563 CK1DI3 134132786 IC50 = 60 nM T69563 C9JG7W 134135029 IC50 = 260 nM T69563 CML85T 134136251 IC50 = 320 nM T69563 C39BMU 134136448 IC50 = 80 nM T69563 CIQ6Z8 134137347 IC50 = 19000 nM T69563 CFMG90 134140713 IC50 = 1000 nM T69563 CYF9N7 134141391 IC50 = 140 nM T69563 CH6J4X 134141647 IC50 = 32 nM T69563 CUF9M5 134141685 IC50 = 1600 nM T69563 CATD87 134142306 IC50 = 7900 nM T69563 CPCG95 134143587 IC50 = 140 nM T69563 C13YMT 134144334 IC50 = 1400 nM T69563 CO4D1Q 134145417 IC50 = 3100 nM T69563 CR84NZ 134145925 IC50 = 90 nM T69563 CTV9B8 134146140 IC50 = 160 nM T69563 CG7V6W 134146450 IC50 = 7400 nM T69563 CATO08 134147599 IC50 = 96 nM T69563 CXH8W3 134149147 IC50 = 360 nM T69563 CF9NA0 134149890 IC50 > 20000 nM T69563 C5ZLU2 134151046 IC50 = 75 nM T69563 CN6S0J 134151358 IC50 = 11000 nM T69563 CO74YZ 134152117 IC50 = 7700 nM T69563 CD5O3M 134152198 IC50 = 440 nM T69563 C81ESC 134153452 IC50 = 1600 nM T69563 COLF87 134153477 IC50 = 5700 nM T69563 C07YDQ 134153794 IC50 = 9100 nM T69563 CGC6P4 134153864 IC50 = 160 nM T69563 CIHC43 134154520 IC50 = 91 nM T69563 CAC65I 134155569 IC50 = 56 nM T69563 C5U2VM 134156397 IC50 = 28 nM T69563 CL1H7K 134464493 IC50 < 100 nM T69563 CW73JK 134693801 IC50 = 120 nM T69563 CKMU89 134693804 IC50 = 41 nM T69563 CL51MJ 136110950 Ki > 50000 nM T69563 CZF18P 136110951 Ki > 50000 nM T69563 CW3T4O 137333448 IC50 = 21 nM T69563 CAH41F 137440052 IC50 < 100 nM T69563 CQ19ZS 137496890 IC50 < 20 nM T69563 C3XTO9 137548127 IC50 < 300 nM T69563 CG5HS1 138753630 IC50 > 10000 nM T69563 CE0UK8 138976844 IC50 = 8.9 nM T69563 CHA68B 139373943 IC50 < 300 nM T69563 CLC12T 140267775 IC50 = 11 nM T69563 C0NQO6 140267826 IC50 = 1 nM T69563 CQYI50 140267835 IC50 = 3 nM T69563 CW1O0F 140267861 IC50 = 1 nM T69563 CC26QP 141451166 IC50 = 140 nM T69563 CR82BZ 141451167 IC50 = 950 nM T69563 C8TZ6R 141451170 IC50 = 230 nM T69563 C0Q2WJ 141451172 IC50 = 90 nM T69563 CZP73S 141451178 IC50 = 4420 nM T69563 C1FJ8M 141451182 IC50 = 50 nM T69563 C5N3VP 141451185 IC50 = 930 nM T69563 CG93ER 141451187 IC50 = 13620 nM T69563 C5HZB7 141451189 IC50 = 810 nM T69563 CB8W0Q 141492780 IC50 < 100 nM T69563 CJ6S4B 141503237 IC50 < 10 nM T69563 CM8ZT0 141503247 IC50 = 49 nM T69563 CUT16P 141503256 IC50 > 1000 nM T69563 CMB72E 141503257 IC50 = 5.6 nM T69563 CF35VQ 141503261 IC50 = 14 nM T69563 CW9D8I 142547299 IC50 < 20 nM T69563 C6V3PC 145426709 IC50 = 338 nM T69563 C3FJ1U 145426710 IC50 = 138 nM T69563 CPWT56 145426714 IC50 = 5 nM T69563 CT9J1D 145426720 IC50 = 95 nM T69563 C3UDY4 145426748 IC50 = 180 nM T69563 CU0Q3N 145426790 IC50 = 9 nM T69563 CW10RV 145426839 IC50 = 635 nM T69563 CXWN78 145426877 IC50 = 255 nM T69563 CISY09 145426959 IC50 = 266 nM T69563 C8TSE3 145426981 IC50 = 25 nM T69563 CVC37N 145426988 IC50 = 148 nM T69563 CPL8E6 145427034 IC50 = 21 nM T69563 CV63QK 145427036 IC50 = 186 nM T69563 C6BZA7 145427057 IC50 = 172 nM T69563 C8X0YZ 145427073 IC50 = 51 nM T69563 CP96LO 145721285 IC50 = 17310 nM T69563 CG58CF 145721286 IC50 > 50000 nM T69563 CRMU49 145721287 IC50 > 50000 nM T69563 C2IFB6 145721288 IC50 > 50000 nM T69563 CR53AV 145721289 IC50 > 50000 nM T69563 C2A4EJ 145721290 IC50 > 50000 nM T69563 C6X0NF 145950670 IC50 < 2 nM T69563 CLTN42 145951582 IC50 = 14 nM T69563 CBZ59V 145951646 IC50 = 47 nM T69563 CF5X9J 145954559 IC50 = 73 nM T69563 CUR5N4 145954702 IC50 = 145 nM T69563 CXR2W3 145955203 IC50 = 15 nM T69563 C8OM3X 145956839 IC50 = 116 nM T69563 C6HQJ5 145961862 IC50 = 42 nM T69563 C54CSY 145961866 IC50 = 41 nM T69563 C3M9NW 145963523 IC50 = 28 nM T69563 C7GC3U 145963920 IC50 > 10000 nM T69563 CM0T9L 145964379 IC50 = 560 nM T69563 CCM4K8 145965456 IC50 > 10000 nM T69563 CDM3X9 145965619 IC50 = 15 nM T69563 C7FR6H 145966084 IC50 > 10000 nM T69563 C6AM2R 145966168 IC50 = 27 nM T69563 C2FH9U 145966444 IC50 > 1000 nM T69563 CY7BQ5 145966713 IC50 = 15 nM T69563 C1T0UW 145971297 IC50 = 84 nM T69563 C8QCN3 145971400 IC50 = 13 nM T69563 CH50IP 145971583 IC50 = 21 nM T69563 C8P6QC 145971862 IC50 = 2965 nM T69563 C4L0VB 145972381 IC50 = 47 nM T69563 CSK1D4 145972835 IC50 = 42 nM T69563 CRH47A 145973499 IC50 = 260 nM T69563 C75YBO 145974168 IC50 = 275 nM T69563 C8WS0M 145974512 IC50 = 50 nM T69563 CC92FX 145975511 IC50 = 40 nM T69563 C7HVI9 145975779 IC50 = 270 nM T69563 C0VZ4H 145975944 IC50 = 2605 nM T69563 CS6X3V 145976283 IC50 = 108 nM T69563 CCY80A 145976820 IC50 = 22 nM T69563 CCY85M 145978022 IC50 = 128 nM T69563 C73HRS 145978840 IC50 = 19 nM T69563 C5J8NI 145980147 IC50 > 50000 nM T69563 CVJD53 145980478 IC50 = 34 nM T69563 CG0DS6 145980657 IC50 = 46 nM T69563 C1AOH7 145980705 IC50 = 32000 nM T69563 CVZS80 145981016 IC50 > 50000 nM T69563 CX35RT 145981660 IC50 > 50000 nM T69563 CBU6X1 145981803 IC50 > 50000 nM T69563 CAF30W 145981971 IC50 = 40 nM T69563 CREN84 145982246 IC50 = 8 nM T69563 CQS73W 145983417 IC50 = 13310 nM T69563 CBZ54K 145987434 IC50 = 230 nM T69563 CB1A0K 145987773 IC50 > 50000 nM T69563 CX6G9K 145987904 IC50 > 50000 nM T69563 CG39VW 145988250 IC50 > 50000 nM T69563 C3M8WP 145989869 IC50 = 297 nM T69563 C53EQF 145990414 IC50 = 23100 nM T69563 CTDA70 145992655 IC50 > 50000 nM T69563 CSKG09 145993293 IC50 = 45 nM T69563 CIZ83X 145993302 IC50 = 44 nM T69563 C6PR9F 145994156 IC50 > 50000 nM T69563 CJ12IY 146774513 IC50 = 18.8 nM T69563 C8FJ3A 148054621 IC50 = 16.3 nM T69563 CHK41W 149984817 IC50 = 61.9 nM T69563 CUY4O2 151050871 IC50 = 2.3 nM T69563 CU6FL5 151060963 IC50 = 24.1 nM T69563 CRN0K3 151095070 IC50 = 4 nM T69563 C1UW8G 151614103 IC50 = 9.7 nM T69563 C1ATK8 151745584 IC50 = 17.3 nM T69563 CP7B3F 152297087 IC50 = 24.8 nM T69563 CLC50D 152682805 IC50 = 8 nM T69563 CWA1K4 153354193 IC50 = 14.2 nM T69563 C7Z1RB 153354194 IC50 = 128.5 nM T69563 CXC8G3 153354195 IC50 = 43.5 nM T69563 CQ7R2X 153354196 IC50 = 5858 nM T69563 C3GLD4 153354197 IC50 = 9.4 nM T69563 C1CQ5W 153354198 IC50 = 119.1 nM T69563 C1KR3B 153354200 IC50 = 15 nM T69563 CJ2NI6 153354201 IC50 = 23.8 nM T69563 CS7OY3 153354202 IC50 = 1 nM T69563 CKD1H3 153354205 IC50 = 2.1 nM T69563 CC0T9V 153354208 IC50 = 2.12 nM T69563 CU3OF1 154709431 IC50 = 11660 nM T69563 CWKY46 154709433 IC50 = 13310 nM T69563 CB8F9R 155511968 IC50 = 90 nM T69563 CVF25J 155513757 IC50 = 2 nM T69563 C1YT5V 155514864 IC50 = 12 nM T69563 CLH3W0 155515484 IC50 = 112 nM T69563 CH24MR 155515991 IC50 = 1980 nM T69563 CDK81A 155516285 IC50 > 10000 nM T69563 CLJ5H1 155516944 IC50 = 21 nM T69563 CF60TJ 155517478 IC50 = 42 nM T69563 CT2Z8D 155518356 IC50 = 10 nM T69563 C53FQM 155518762 IC50 > 50000 nM T69563 CO4I8L 155519528 IC50 > 50000 nM T69563 C48QWJ 155519945 IC50 < 100 nM T69563 CT94CM 155520089 IC50 > 100000 nM T69563 C06QWY 155520182 IC50 > 50000 nM T69563 C4YO6W 155520615 IC50 = 28 nM T69563 C8A9HN 155520995 IC50 = 12790 nM T69563 CH7ZC1 155521584 IC50 < 100 nM T69563 C29SCL 155522425 IC50 = 3000 nM T69563 C4BK7X 155523227 IC50 = 11860 nM T69563 C1Y2MB 155523310 IC50 = 5000 nM T69563 COZ4K9 155524250 IC50 = 1400 nM T69563 CZ0CD8 155524347 IC50 = 8500 nM T69563 CC5W9E 155524570 IC50 > 200000 nM T69563 CZC8X9 155524600 IC50 = 32 nM T69563 C3VBJ1 155525283 IC50 > 50000 nM T69563 C8QA0B 155525540 IC50 = 290 nM T69563 CAD91T 155526125 IC50 = 81.5 nM T69563 C3LK2Q 155527455 IC50 = 50 nM T69563 CBR52U 155527494 IC50 > 100000 nM T69563 CO9UA0 155528439 IC50 = 38 nM T69563 C4H6ET 155529102 IC50 = 26.6 nM T69563 CPWO50 155529490 IC50 = 1450 nM T69563 CH3SC8 155531040 IC50 = 18000 nM T69563 C4XLB5 155531880 IC50 = 7910 nM T69563 CC2V9G 155532071 IC50 = 21 nM T69563 C30LMB 155532656 IC50 = 190 nM T69563 C4YFQ9 155533059 IC50 = 65 nM T69563 CAP54S 155533635 IC50 = 100 nM T69563 C8HL6B 155533681 IC50 = 2.2 nM T69563 CP9WL2 155533930 IC50 = 28 nM T69563 CJ2GF8 155534982 IC50 = 3050 nM T69563 CVE7U9 155534983 IC50 = 54 nM T69563 CL02MX 155536249 IC50 = 1480 nM T69563 C5LN0G 155536622 IC50 = 55500 nM T69563 CPS53T 155536735 IC50 < 10 nM T69563 C0BQ5V 155537997 IC50 = 18 nM T69563 CV1AE4 155538180 IC50 = 60 nM T69563 CS3X5Z 155540428 IC50 = 831 nM T69563 COAE19 155540545 IC50 = 55 nM T69563 CK4S2B 155540581 IC50 = 250 nM T69563 CQD6E7 155543356 IC50 = 266 nM T69563 C71CUQ 155544473 IC50 < 100 nM T69563 C1GJ2X 155546130 IC50 > 100000 nM T69563 CU1ST0 155547033 IC50 = 3720 nM T69563 CN46TF 155547202 IC50 = 25000 nM T69563 C5GK8W 155547940 IC50 > 25000 nM T69563 CIDO95 155548480 IC50 > 50000 nM T69563 CP27OJ 155548685 IC50 > 25000 nM T69563 C2S3OI 155548929 IC50 < 100 nM T69563 C9Z1RB 155549401 IC50 = 410 nM T69563 CG73WV 155549530 IC50 = 1540 nM T69563 C6UG0I 155549731 IC50 > 50000 nM T69563 CZ9AV3 155550739 IC50 < 100 nM T69563 C48VPJ 155553143 IC50 = 18 nM T69563 CJX6U0 155553326 IC50 > 100000 nM T69563 C18PRB 155553562 IC50 = 44.5 nM T69563 C7KJ4E 155553804 IC50 = 721 nM T69563 C4HT0M 155553871 IC50 = 39600 nM T69563 C7S1AK 155556534 IC50 = 26 nM T69563 C42KSY 155556957 IC50 = 4800 nM T69563 CD7IO6 155556974 IC50 = 82 nM T69563 C5KP4J 155557173 IC50 = 60 nM T69563 CRO21A 155557415 IC50 > 50000 nM T69563 C8AFH6 155557755 IC50 = 152 nM T69563 CV4H2Z 155559814 IC50 > 10000 nM T69563 CU8W4A 155560336 IC50 = 930 nM T69563 CKPE98 155561191 IC50 < 300 nM T69563 C27QFZ 155562355 IC50 > 10000 nM T69563 CHC0E2 155562949 IC50 = 800 nM T69563 C4FZ6B 155563652 IC50 = 50000 nM T69563 C26LSZ 155563728 IC50 = 393.9 nM T69563 CR3WQ5 155565507 IC50 = 43580 nM T69563 CDYB38 155565613 IC50 = 45300 nM T69563 CS01QM 155565995 IC50 > 50000 nM T69563 C5VZN7 155567367 IC50 = 220 nM T69563 D05IWY 5464078 Ki = 3170 nM T69563 D06PRC 5281650 Ki = 2850 nM T70539 D0A3CL 49801838 IC50 > 40000 nM T70539 CYIT28 9806086 IC50 = 10000 nM T70539 C5RIY7 9824428 IC50 > 100000 nM T70539 CTUO16 9955811 IC50 = 6310 nM T70539 CQL12P 10004545 IC50 > 10000 nM T70539 C6OI1A 10005009 IC50 = 6.8 nM T70539 CI8FM2 10025150 IC50 = 100 nM T70539 CS14OM 10027853 IC50 = 4.7 nM T70539 C9QZ0I 10046992 IC50 = 4 nM T70539 CR1ME4 10090198 IC50 = 100 nM T70539 CU7TP2 10091316 IC50 = 10 nM T70539 CG7Z9I 10128764 Ki > 3000 nM T70539 CEO59I 10129026 Ki > 3000 nM T70539 CW5O4B 10129036 Ki > 3000 nM T70539 C3FS7G 10129058 Ki > 3000 nM T70539 CJ05QL 10129135 Ki > 3000 nM T70539 CX9EI2 10143421 Ki > 3000 nM T70539 CZ95DQ 10143980 Ki > 3000 nM T70539 C2X9YI 10152629 Ki > 3000 nM T70539 C9VP5L 10152726 Ki > 3000 nM T70539 CVGB64 10152879 Ki > 3000 nM T70539 CZQ69G 10165656 Ki > 3000 nM T70539 C9EJT4 10166088 Ki > 3000 nM T70539 CC2F7Z 10173787 IC50 = 960 nM T70539 CM9KF2 10174522 Ki > 3000 nM T70539 CH25WF 10174984 Ki > 3000 nM T70539 C47RGT 10186370 Ki > 3000 nM T70539 C80YEW 10188732 Ki > 3000 nM T70539 CGJ7D9 10195667 Ki > 3000 nM T70539 C9OB3S 10196098 Ki > 3000 nM T70539 C2K1LR 10196214 Ki > 3000 nM T70539 CBX4C2 10196316 Ki > 3000 nM T70539 CD9N3H 10196460 Ki > 3000 nM T70539 CYT8S5 10196576 Ki > 3000 nM T70539 C5EGZ8 10196608 Ki > 3000 nM T70539 C0OB2A 10196742 Ki > 3000 nM T70539 CIC0H8 10218194 Ki > 3000 nM T70539 CH7BP9 10218547 Ki > 3000 nM T70539 CX7KR8 10218604 Ki > 3000 nM T70539 CEO3C0 10230947 Ki > 3000 nM T70539 C2AV9K 10239389 Ki > 3000 nM T70539 CWTM13 10239448 Ki > 3000 nM T70539 CY3B9V 10239505 Ki > 3000 nM T70539 C9ZR5W 10239639 Ki > 3000 nM T70539 C8R7NE 10239929 Ki > 3000 nM T70539 C2JY5L 10239930 Ki > 3000 nM T70539 CNY7O0 10280331 Ki > 3000 nM T70539 C7GFV9 10281308 Ki > 3000 nM T70539 CQAM65 10289494 Ki > 3000 nM T70539 CP4MX9 10303281 Ki > 3000 nM T70539 C5NVX2 10310772 Ki > 3000 nM T70539 C8X2OD 10311260 Ki > 3000 nM T70539 CS5YX7 10311798 Ki > 3000 nM T70539 CHR1A3 10312086 Ki > 3000 nM T70539 CCRI74 10312244 Ki > 3000 nM T70539 CMC1G5 10319824 IC50 > 100000 nM T70539 CVO3N7 10344176 IC50 > 10 nM T70539 CL83KQ 10388797 IC50 = 3.7 nM T70539 C6UO4Y 10410064 IC50 = 0.1 nM T70539 C6T7WB 10434776 IC50 > 100000 nM T70539 CFV7D4 10436090 IC50 = 10000 nM T70539 CGS89V 10455647 IC50 = 4 nM T70539 C07KPU 10456755 IC50 > 10 nM T70539 C38VGA 10457264 IC50 = 1 nM T70539 CUD3I6 11156790 Ki > 3000 nM T70539 C19UHW 11168186 Ki > 3000 nM T70539 CPS26T 11201645 IC50 = 6.4 nM T70539 CK9E2Y 11317465 Ki > 3000 nM T70539 CO7CX6 11318577 Ki > 3000 nM T70539 CCU9P8 11318709 Ki > 3000 nM T70539 CB51KQ 11433168 Ki > 3000 nM T70539 C6L8DU 11495754 IC50 > 10 nM T70539 C9YME5 11496313 IC50 > 10 nM T70539 C2B6YR 11512135 IC50 = 4.5 nM T70539 CQ08DH 11539632 IC50 = 8.7 nM T70539 CX6IL5 11548234 IC50 = 6.3 nM T70539 C59SVL 11563383 IC50 > 10 nM T70539 CPA3J7 11583744 IC50 = 7.1 nM T70539 CKI9D5 11599973 IC50 = 4600 nM T70539 CDA48G 11613696 Ki > 3000 nM T70539 C5A4YW 11648240 IC50 = 8.4 nM T70539 CP09GF 11655872 IC50 > 10 nM T70539 CFB78R 11752339 Ki > 3000 nM T70539 CX20YM 11785261 Ki > 3000 nM T70539 CJZ1S6 11785262 Ki > 3000 nM T70539 CL50KS 15983730 Ki > 10000 nM T70539 CB0JD2 16037921 Ki > 3000 nM T70539 C7K5AW 16721015 IC50 > 10000 nM T70539 CBR6Q7 20608969 Ki > 3000 nM T70539 COF9E8 20608974 Ki > 3000 nM T70539 CWSB30 20608975 Ki > 3000 nM T70539 C7PL9M 20608976 Ki > 3000 nM T70539 CG9R3I 20608977 Ki > 3000 nM T70539 C9U6JQ 20608981 Ki > 3000 nM T70539 CC1RB9 20608989 Ki > 3000 nM T70539 C2H1YF 20608991 Ki > 3000 nM T70539 C8Q0XO 20608992 Ki > 3000 nM T70539 C8CUT0 20608996 Ki > 3000 nM T70539 CVGY56 20609011 Ki > 3000 nM T70539 C7N6XY 20609018 Ki > 3000 nM T70539 C78UWI 20609028 Ki > 3000 nM T70539 CKHG76 23572819 IC50 = 30 nM T70539 C2DIJ7 23573799 Ki > 3000 nM T70539 CRCF01 30979231 IC50 = 1000 nM T70539 CMY45F 44188279 Ki > 9700 nM T70539 C76ONX 44219756 IC50 > 1000 nM T70539 C1RD0C 44394909 IC50 > 100000 nM T70539 C0KLA9 44394921 IC50 > 100000 nM T70539 CI7RP8 44394922 IC50 > 100000 nM T70539 C2KM0Q 44394959 IC50 > 100000 nM T70539 CUQ04R 44395076 IC50 = 2880 nM T70539 C4HR6C 44399507 Ki > 3000 nM T70539 CH39TA 44399610 Ki > 3000 nM T70539 CLGA83 44403765 IC50 = 6.8 nM T70539 CD3FE4 44405399 Ki > 3000 nM T70539 CW5KU8 44405417 Ki > 3000 nM T70539 CVP74K 44405418 Ki > 3000 nM T70539 C0N4IL 44405421 Ki > 3000 nM T70539 C79OPX 44405435 Ki > 3000 nM T70539 CDJF17 44405436 Ki > 3000 nM T70539 CT42XM 44405437 Ki > 3000 nM T70539 CF57KL 44405439 Ki > 3000 nM T70539 C37XOM 44405444 Ki > 3000 nM T70539 CW80JL 44405461 Ki > 3000 nM T70539 CN4KP9 44405501 Ki > 3000 nM T70539 CFSD50 44412624 Ki > 3000 nM T70539 C1CPT2 44412682 Ki > 3000 nM T70539 CG6J5R 44412683 Ki > 3000 nM T70539 CQ7P1N 44412686 Ki > 3000 nM T70539 CVJF97 44412837 Ki > 3000 nM T70539 CRPQ04 44412852 Ki > 3000 nM T70539 CV1ZX4 44412960 Ki > 3000 nM T70539 CAQ2D8 45487653 IC50 > 10 nM T70539 CN58HC 57391501 IC50 = 10 nM T70539 C0J6GT 57391502 IC50 = 678 nM T70539 C1W8ZE 57394991 IC50 = 250 nM T70539 CMNZ07 57394992 IC50 = 1 nM T70539 CAID96 57396733 IC50 = 15000 nM T70539 C8AOK6 57396734 IC50 = 200 nM T70539 CO0C6Y 57396735 IC50 = 10 nM T70539 CVN98L 57400176 IC50 = 300 nM T70539 CFXM54 57400177 IC50 = 200 nM T70539 CS05AF 57400178 IC50 = 80 nM T70539 C0SY9X 57400179 IC50 = 150 nM T70539 CRHS14 57400180 IC50 = 8 nM T70539 C98HEK 57401966 IC50 = 60000 nM T70539 CBEW17 57401967 IC50 = 100 nM T70539 C1E2LP 57401968 IC50 = 0.1 nM T70539 CS63IW 57401969 IC50 = 13 nM T70539 C9DF5Y 57403720 IC50 = 10000 nM T70539 C9PN3B 57403721 IC50 = 60000 nM T70539 CXZQ20 57403722 IC50 = 70 nM T70539 CH5EV8 57403723 IC50 = 250 nM T70539 D01NOZ 16665072 IC50 > 30000 nM T75888 D00SBN 4746 IC50 > 100000 nM T75888 D0L5WM 2157 IC50 > 100000 nM T75888 D0Q4YI 21109 IC50 > 100000 nM T75888 D01FCK 9843897 IC50 = 5400 nM T75888 D0P9JW 121830 IC50 > 100000 nM T75888 CSI0D4 355 IC50 = 11000 nM T75888 COK56H 36143 IC50 > 100000 nM T75888 CAUV41 11979264 IC50 = 6400 nM T75888 CY7XM3 13671155 IC50 = 21700 nM T75888 CFD2E4 15234003 IC50 = 160 nM T75888 CZ9JM6 15984085 IC50 > 100000 nM T75888 C7E2FM 16718554 IC50 = 3400 nM T75888 C7ZY1S 16736346 IC50 > 100000 nM T75888 C2WJQ5 23695524 IC50 > 50000 nM T75888 CMFN27 23729161 IC50 = 85300 nM T75888 CMW4E2 24825719 IC50 = 3500 nM T75888 C9KS1T 25095157 IC50 > 100000 nM T75888 CLS8H0 66857424 IC50 > 100000 nM T75888 CQR5T1 71457921 IC50 = 360 nM T15636 CV63UL 67240318 IC50 > 10000 nM T15636 C2MD1Q 155513187 IC50 > 10000 nM T15636 C41NLP 155544908 IC50 = 120 nM T15636 D0VC0I 5169 IC50 = 47200 nM T13453 CZ63PR 16133811 IC50 = 0.8 nM T13453 CP42JF 25180487 Ki = 22 nM T13453 C5VA6W 25180488 Ki = 108 nM T13453 CZ51CD 25180490 Ki = 65.5 nM T13453 C1IU8X 25180491 Ki = 15 nM T13453 C2WMX8 25180492 Ki = 75 nM T13453 CZ1N7I 25180493 Ki = 24 nM T13453 C3G8OJ 25180494 Ki = 28 nM T13453 CHRV59 25180496 Ki = 51 nM T13453 CVN29B 25180497 Ki = 214.5 nM T13453 C62QZX 25180498 Ki = 1323.5 nM T13453 C4DL5C 44469677 IC50 > 10000 nM T13453 CK4J9W 44584852 IC50 = 2.6 nM T13453 C0GTZ7 44587983 Ki = 160 nM T13453 C20WUX 44587984 Ki = 51.5 nM T13453 CGU02F 54764328 IC50 = 380 nM T13453 CD87IE 54764411 IC50 = 330 nM T13453 CPZ93G 54764412 IC50 = 380 nM T13453 C1TO0M 57390716 IC50 = 770 nM T13453 CKE01G 57390718 IC50 = 24850 nM T13453 C32ETJ 57392517 IC50 = 1060 nM T13453 CR25FK 57392518 IC50 = 1930 nM T13453 C7P8NA 57394235 IC50 = 3380 nM T13453 C7AT3L 57394236 IC50 = 930 nM T13453 CY5D0W 57394237 IC50 = 1750 nM T13453 CJ39YQ 57394238 IC50 = 560 nM T13453 C0WBK1 57394239 IC50 = 540 nM T13453 C16SNJ 57394240 IC50 = 430 nM T13453 C8G4OA 57394241 IC50 = 4180 nM T13453 CR7Z6D 57394303 IC50 = 4570 nM T13453 CN0MS2 57394304 IC50 = 6620 nM T13453 COJ7T1 57395992 IC50 = 8650 nM T13453 CU6K8A 57395993 IC50 = 12500 nM T13453 CU93SZ 57395994 IC50 = 2080 nM T13453 CCEG86 57395995 IC50 = 980 nM T13453 CB70EI 57396058 IC50 = 1090 nM T13453 CD3FK9 57397796 IC50 = 3690 nM T13453 CI2RP0 57397797 IC50 = 8040 nM T13453 C7GK1B 57397798 IC50 = 1920 nM T13453 CD35FB 57397799 IC50 = 440 nM T13453 C2W0JH 57399456 IC50 = 3400 nM T13453 C2H3XW 57399457 IC50 = 550 nM T13453 CZ9RD1 57399458 IC50 = 2030 nM T13453 CR9WH3 57399459 IC50 = 780 nM T13453 CS27BV 57401220 IC50 = 4150 nM T13453 C8DS7R 57401221 IC50 = 770 nM T13453 CO40GM 57401222 IC50 = 1180 nM T13453 CIO4Q9 57401223 IC50 = 2850 nM T13453 CT7PZ3 57401225 IC50 = 1340 nM T13453 CG1J8I 57401228 IC50 = 9070 nM T13453 CYR89Z 71508528 Ki = 15.6 nM T13453 C0O3CM 71720536 Ki = 119 nM T13453 CWH6T3 72548703 IC50 = 0.19 nM T13453 D01LMH 25180489 Ki = 17.5 nM T13453 D02GOE 44563954 Ki = 16.1 nM T13453 D02JQP 24760995 Ki = 51.5 nM T13453 D03ECE 44563952 Ki = 14.9 nM T13453 D05GFD 44563953 Ki = 14.4 nM T13453 D06DWA 44563958 Ki = 20.5 nM T13453 D07NOJ 45104655 Ki = 35 nM T13453 D09SDZ 44587982 Ki = 13 nM T13453 D0DD3F 44563955 Ki = 18.2 nM T13453 D0EO5F 44563956 Ki = 51.5 nM T13453 D0H4DF 16132126 Ki = 1.1 nM T13453 D0H9QA 25180495 Ki = 48 nM T13453 D0PY7O 6324638 Ki = 1.74 nM T13453 D0Q3CB 16133821 Ki = 1.5 nM T13453 D0S4VO 45104657 Ki = 20.2 nM T13453 D0TF7R 44563951 Ki = 24 nM T13453 D0V7UG 45104656 Ki = 15.9 nM T13453 D0Z3QG 44563957 Ki = 15 nM T89530 CW9G5L 150570 IC50 = 2170 nM T89530 C4QG8H 3508054 IC50 = 50 nM T89530 C0U6YX 3508059 IC50 = 1250 nM T89530 CMA40L 5092911 IC50 = 31700 nM T89530 CKP1Y4 90644339 IC50 > 100000 nM T89530 CYD71G 90644340 IC50 = 980 nM T89530 CMXY84 90644341 IC50 = 11800 nM T89530 CFVS82 90644342 IC50 = 15840 nM T89530 C2QDT0 90644343 IC50 = 13100 nM T89530 C8CXG2 90644344 IC50 = 5210 nM T89530 CHM46Z 90644345 IC50 = 660 nM T89530 CGM5N0 90644346 IC50 = 430 nM T89530 CM2J0G 90644347 IC50 = 2010 nM T89530 CL7CK6 90644348 IC50 = 33850 nM T89530 CS0AD6 90644349 IC50 = 210 nM T89530 C14GOM 90644350 IC50 = 180 nM T89530 C8GR5L 90644351 IC50 = 35400 nM T89530 C9OZ5L 90644352 IC50 > 100000 nM T89530 CLQ0C1 90644353 IC50 = 41990 nM T89530 CKL0B7 90644354 IC50 > 100000 nM T89530 CK31VW 90644355 IC50 = 31800 nM T89530 CET02U 90644356 IC50 = 180 nM T89530 C2I1VP 90644357 IC50 = 90 nM T89530 C8X9UO 90644358 IC50 = 140 nM T89530 CA7EU1 90644359 IC50 = 110 nM T89530 C7DPQ0 90644360 IC50 = 40 nM T89530 CZU1J4 90644361 IC50 = 3040 nM T89530 C4F6ZI 90644362 IC50 = 1090 nM T89530 CA21TC 90644363 IC50 = 730 nM T89530 CRL8E2 90644364 IC50 = 1350 nM T89530 C4E6WO 90644365 IC50 = 50900 nM T89530 CV76KR 90644366 IC50 = 22100 nM T03403 D03RTS 2662 IC50 = 89 nM T03403 D0GY5Z 2244 IC50 = 15000 nM T03403 D0R1RS 3715 IC50 = 10 nM T03403 D0U2FN 71321 IC50 = 6500000 nM T03403 D05WPQ 6438354 IC50 = 3200 nM T03403 D09QRO 55390 IC50 = 10000 nM T03403 D0DP8P 47795 IC50 = 5800 nM T03403 D0JY4Y 443292 IC50 > 100000 nM T03403 D0N1SU 133021 IC50 = 160 nM T03403 D0O8ZE 5059 IC50 = 5300 nM T03403 D0S8YL 3969 IC50 = 44000 nM T03403 CH0L7P 71697 IC50 = 950000 nM T03403 CI5D9O 92656 IC50 = 100 nM T03403 CV7L0G 112230 IC50 = 100000000 nM T03403 CT2XZ0 116545 IC50 = 7079457.84 nM T03403 CAT4E3 129615 IC50 = 3388441.56 nM T03403 CCJ76H 512829 IC50 = 9000 nM T03403 CE2BC3 512830 IC50 = 14000 nM T03403 C16VBD 512831 IC50 = 12000 nM T03403 CT7E6Y 573683 IC50 > 800000 nM T03403 CZ0AH3 638278 IC50 = 130000 nM T03403 C6EVL8 854057 IC50 = 3467368.5 nM T03403 CQM64G 3037018 IC50 = 800 nM T03403 COH1C4 3052566 IC50 = 446683.59 nM T03403 C82IPJ 3052567 IC50 = 912010.84 nM T03403 C4VBK3 3253091 IC50 = 50000 nM T03403 CU86JL 4618600 IC50 = 40000 nM T03403 C4M1JC 5709318 IC50 = 44000 nM T03403 COQ7T3 5973690 IC50 = 63000 nM T03403 C3G7DT 6365297 IC50 = 4200 nM T03403 C40FZG 6366698 IC50 = 1300 nM T03403 C02AQY 6366699 IC50 ~ 1000 nM T03403 CWK1F9 6438990 IC50 = 110 nM T03403 C62UOZ 6439221 IC50 = 780 nM T03403 CHQ4Z3 6439222 IC50 = 1300 nM T03403 COC86Q 6439421 IC50 = 390 nM T03403 CLJ91K 6439912 IC50 = 260 nM T03403 C82TEX 7515046 IC50 < 10000 nM T03403 CUS6L8 9822795 IC50 = 30 nM T03403 C5C9ET 10042219 IC50 > 100000 nM T03403 C9T7YV 10063338 IC50 > 100000 nM T03403 CBL7R3 10220019 IC50 = 400 nM T03403 C2WE0I 10246235 IC50 = 9600 nM T03403 C20BTQ 10313997 IC50 = 5500 nM T03403 C8EQI3 10334136 IC50 > 100000 nM T03403 CC1UF0 10335738 IC50 > 100000 nM T03403 C25MYB 10425738 IC50 > 100000 nM T03403 CPR7J0 10469807 IC50 = 12589254.12 nM T03403 C6JI5F 10492615 IC50 > 300000 nM T03403 C0NRO9 10513373 IC50 = 570000 nM T03403 CK0OL2 10704667 IC50 = 27000 nM T03403 CUOI16 10729548 IC50 = 26000 nM T03403 C8IBM2 10801359 IC50 = 250000 nM T03403 CC8S6O 10801786 IC50 = 37000 nM T03403 CDZ94R 10826230 IC50 = 29000 nM T03403 CGLQ72 11723348 IC50 > 100000 nM T03403 CH9VC8 13245625 IC50 > 10000 nM T03403 CRA87I 13556944 IC50 = 14125375.45 nM T03403 C0P5AK 13914227 IC50 > 100000 nM T03403 C49OGE 13914253 IC50 > 100000 nM T03403 C4U3RD 14006855 IC50 = 5000 nM T03403 C6EZ0K 14312565 IC50 > 10000 nM T03403 C2X8PQ 14416570 IC50 = 34 nM T03403 C5PT1G 14416572 IC50 670 nM T03403 C1SG0F 14416576 IC50 = 10000 nM T03403 CRYI80 14416580 IC50 = 610 nM T03403 C27NOS 14416585 IC50 < 10000 nM T03403 C6BP2F 14416587 IC50 < 1000 nM T03403 CER87K 14762923 IC50 = 13803842.65 nM T03403 CGYF09 14762938 IC50 = 501187233.6 nM T03403 CX9AH8 14762939 IC50 = 501187233.6 nM T03403 CU3OT4 14762940 IC50 = 165958690.7 nM T03403 CXT3B5 14762942 IC50 = 100000000 nM T03403 CNZ45J 14762943 IC50 = 91201083.94 nM T03403 CL2A1E 14762944 IC50 = 91201083.94 nM T03403 C78IHC 14762948 IC50 = 50118723.36 nM T03403 CBL2O8 14762951 IC50 = 14791083.88 nM T03403 C8NKZ7 14762954 IC50 = 7079457.84 nM T03403 C4PS0F 14771889 IC50 < 10000 nM T03403 CV41BE 14771890 IC50 = 3100 nM T03403 CCX7K5 14771891 IC50 = 1400 nM T03403 CG57JP 14771892 IC50 = 1300 nM T03403 C91VJM 14771893 IC50 = 230 nM T03403 C0EMA5 14771894 IC50 < 1000 nM T03403 CZ4WJ2 14771895 IC50 = 730 nM T03403 CV5YH8 14771896 IC50 < 10000 nM T03403 C3HNQ2 14771897 IC50 < 10000 nM T03403 CH0TC9 14771898 IC50 < 10000 nM T03403 CX3N7Z 14771899 IC50 = 11000 nM T03403 CX7VA0 14771900 IC50 < 10000 nM T03403 CZC2D4 14771901 IC50 < 10000 nM T03403 CTY60Q 14771902 IC50 < 10000 nM T03403 C0D5OC 14771903 IC50 = 1500 nM T03403 CS3V5C 14771904 IC50 < 10000 nM T03403 CNH5M1 14771905 IC50 = 3200 nM T03403 CXN94C 14771906 IC50 = 510 nM T03403 CY2HF8 14771907 IC50 = 1400 nM T03403 CP5M9A 14771908 IC50 = 190 nM T03403 CI3XK7 14771909 IC50 < 10000 nM T03403 C8NTK2 14771910 IC50 = 750 nM T03403 C8H6XA 14771911 IC50 = 2500 nM T03403 CK53TR 14771912 IC50 < 1000 nM T03403 C10DIY 14771913 IC50 < 1000 nM T03403 C2F9TX 14771915 IC50 = 1100 nM T03403 C83VPQ 14771916 IC50 = 710 nM T03403 CA0C7U 14771917 IC50 = 1000 nM T03403 CK0AR5 14771918 IC50 < 1000 nM T03403 C8SRH6 14771919 IC50 > 10000 nM T03403 CCS9Y4 14771920 IC50 > 10000 nM T03403 C47LJK 14771921 IC50 > 10000 nM T03403 C9OWP0 14771922 IC50 = 1300 nM T03403 C1Z6FX 14771923 IC50 = 780 nM T03403 CHI8M3 14771924 IC50 < 10000 nM T03403 C4JX5S 14771927 IC50 = 590 nM T03403 CRGJ45 14771928 IC50 < 10000 nM T03403 C7L2ZJ 14771929 IC50 = 400 nM T03403 CXAG49 14771930 IC50 < 1000 nM T03403 C54ITL 14771931 IC50 = 110 nM T03403 CC4LM1 14771932 IC50 < 10000 nM T03403 CU6TO3 14771933 IC50 < 10000 nM T03403 C08CRZ 14771934 IC50 = 630 nM T03403 CA3D5U 14771935 IC50 = 1000 nM T03403 CZU2H5 14771936 IC50 = 300 nM T03403 C3B0LX 14771937 IC50 < 10000 nM T03403 CRT9E4 14771938 IC50 > 10000 nM T03403 C18DXV 14977360 IC50 = 71000 nM T03403 CD8YK4 15256755 IC50 = 140000 nM T03403 C53TQI 19044744 IC50 > 100000 nM T03403 CGPW68 19044748 IC50 > 100000 nM T03403 CLN6S5 19044753 IC50 > 100000 nM T03403 CR1W2E 19934882 IC50 > 100000 nM T03403 CF30ID 23275601 IC50 = 66069344.8 nM T03403 CUC36F 23680215 IC50 = 9772372.21 nM T03403 CN6F4H 23680216 IC50 = 4365158.32 nM T03403 C2JUV4 23680221 IC50 = 17782794.1 nM T03403 CHY73S 23680224 IC50 = 524807460.3 nM T03403 C7HV8Y 23680227 IC50 = 70794578.44 nM T03403 CZV8U1 23680228 IC50 = 4677351.41 nM T03403 C54NWH 23680229 IC50 = 741310241.3 nM T03403 CNU43B 23680230 IC50 = 891250938.1 nM T03403 C8A9UV 23689693 IC50 = 562341325.2 nM T03403 CJ1Z9S 44315480 IC50 = 794328234.7 nM T03403 C7UG4F 44315519 IC50 = 15135612.48 nM T03403 C8FEV0 44319113 IC50 = 25000 nM T03403 C1ZH6U 90664380 IC50 > 100000 nM T03403 C5T4EQ 131801158 IC50 = 23 nM T03403 C6JF0E 135616214 IC50 = 2500 nM T03403 CH4YE6 135987613 IC50 > 10000 nM T03403 CFNO28 145950339 IC50 = 34 nM T03403 CG37FR 145950583 IC50 = 27 nM T03403 CCN16Y 145952805 IC50 = 44 nM T03403 C2FVO7 145953074 IC50 = 38 nM T03403 C19TPY 145958203 IC50 = 50 nM T03403 C1BLR8 145959460 IC50 = 33 nM T03403 CUXQ13 145971245 IC50 = 41 nM T03403 C8U9TX 145971276 IC50 = 28 nM T03403 D00GBX 71751 IC50 = 5.7 nM T03403 D01TOR 667555 IC50 = 50000 nM T03403 D05EMX 14076674 IC50 = 10000000 nM T03403 D06VWH 11758240 IC50 = 2 nM T03403 D08GOT 13752584 IC50 = 4897788.19 nM T03403 D09AUL 10266864 IC50 = 51000 nM T03403 D0EW3L 5281222 IC50 = 120000 nM T03403 D0M6UM 129265 IC50 = 22000 nM T03403 D0P1LP 7090 IC50 = 12000 nM T03403 D0U0YE 14762941 IC50 = 165958690.7 nM T03403 D0U2YL 131820 IC50 = 36000 nM T03403 D0U8YQ 921562 IC50 = 14000 nM T37417 D0E3TC 44259 IC50 = 1.47 nM T37417 CV63UL 67240318 IC50 > 10000 nM T37417 C2MD1Q 155513187 IC50 > 10000 nM T83193 D03LGG 1548942 EC50 = 28.2 nM T83193 D05JNI 8378 IC50 = 400 nM T83193 D07ILQ 4671 EC50 > 10000 nM T83193 D0BQ8Y 5971 EC50 = 160000 nM T83193 D0U5CE 1548943 EC50 = 2.512 nM T83193 D00CMV 11256560 IC50 = 0.7 nM T83193 D05XJW 5702546 EC50 = 0.019 nM T83193 D07AOL 16741 EC50 = 180000 nM T83193 D0CO6D 71144018 IC50 > 20000 nM T83193 D0EM4S 17751090 IC50 = 4.6 nM T83193 D0H7PW 638024 EC50 = 3162.28 nM T83193 D07LRT 8068410 IC50 = 2.1 nM T83193 D07EAV 66644203 Ki = 0.04 nM T83193 D09ZWU 66644325 Ki = 0.1 nM T83193 D0K3KE 24782891 IC50 = 25 nM T83193 D0NV2M 52949700 IC50 = 130 nM T83193 D0ZM8H 25265637 IC50 = 34 nM T83193 D0L5XI 16007367 IC50 = 0.6 nM T83193 D0VJ5N 9910486 IC50 = 100 nM T83193 D0Z0PB 11247522 IC50 = 1.1 nM T83193 CT3IS2 2346 EC50 = 223000 nM T83193 CNG85F 3473 EC50 = 3300 nM T83193 C1MO7R 8842 IC50 > 100000 nM T83193 CU94MR 9017 IC50 > 100000 nM T83193 C76SDU 75263 EC50 = 100000 nM T83193 C7UD3V 78151 EC50 = 100000 nM T83193 CTEY14 160611 EC50 = 170000 nM T83193 CF7G0R 160785 EC50 = 1.995 nM T83193 C0GD6Q 310417 IC50 = 3.5 nM T83193 C2QKN6 441539 EC50 = 26000 nM T83193 CE51PH 581676 EC50 = 6309.57 nM T83193 C8WO2M 609524 EC50 = 390 nM T83193 C37RCW 622545 EC50 = 6600 nM T83193 CI9TY8 641115 EC50 = 19952.62 nM T83193 CFMR42 641296 IC50 > 10000 nM T83193 CIX6Q2 643820 IC50 > 100000 nM T83193 C7JSO8 667594 IC50 = 270 nM T83193 CUN5Q0 671605 EC50 > 10000 nM T83193 CFZ3U9 677890 IC50 = 7100 nM T83193 C1YV5I 680436 IC50 = 140 nM T83193 CJ5HC3 692312 IC50 > 10000 nM T83193 CB6LT1 692324 IC50 > 10000 nM T83193 C0XD7N 692351 IC50 > 10000 nM T83193 CY0I3M 721917 IC50 = 147 nM T83193 CS61UR 723775 IC50 = 2500 nM T83193 C7INU2 727129 IC50 = 570 nM T83193 CV2R0I 732540 IC50 > 4000 nM T83193 C2RJ1B 749814 IC50 = 550 nM T83193 CYW3D8 766652 EC50 = 2700 nM T83193 CJD52G 790345 IC50 > 10000 nM T83193 C4M6AL 792621 IC50 = 10700 nM T83193 C5M0TR 871278 IC50 = 2100 nM T83193 CVL8W6 886896 IC50 = 1000 nM T83193 CPED72 887195 IC50 = 210 nM T83193 CVX97S 924972 IC50 > 10000 nM T83193 CY71JK 985818 IC50 > 10000 nM T83193 CR37XU 1245920 IC50 > 10000 nM T83193 CC5NZ4 1322679 IC50 = 320 nM T83193 CC0SH7 1549025 IC50 > 100000 nM T83193 CZ9UX2 1549026 IC50 > 100000 nM T83193 C6UK7A 2093845 IC50 = 210 nM T83193 COZ7X0 2163913 IC50 = 370 nM T83193 C3W6KF 2165451 IC50 > 10000 nM T83193 CD2U7F 2176913 IC50 = 190 nM T83193 CY2U4R 2272103 IC50 > 10000 nM T83193 CC1B7S 2671351 IC50 > 10000 nM T83193 C37EXF 2684177 IC50 > 10000 nM T83193 CG4N3Y 2773243 IC50 > 10000 nM T83193 C6TFN7 3024586 EC50 = 12.59 nM T83193 CN7L2E 3312764 EC50 = 700 nM T83193 CM62BA 3684843 IC50 = 3.9 nM T83193 CY2FP6 4169432 IC50 = 4230 nM T83193 C7WX8B 4391297 IC50 = 7350 nM T83193 CU6M8E 5280457 IC50 > 10000 nM T83193 CJ7NK6 5281719 IC50 = 15000 nM T83193 CZM7D8 5281794 EC50 = 320 nM T83193 CHL79T 5282363 IC50 > 10000 nM T83193 C1UI3F 5283663 IC50 = 1400 nM T83193 C2F8DE 5284650 IC50 > 10000 nM T83193 CA95OR 5311093 EC50 = 0.5012 nM T83193 CZ46HG 5315659 EC50 = 1300 nM T83193 CQM1P0 5316874 IC50 > 10000 nM T83193 C1RM8Q 5317148 IC50 = 5000 nM T83193 C14GJD 5320618 EC50 = 3981.07 nM T83193 CWAE41 5320621 EC50 = 6.31 nM T83193 CB1GY5 5330587 IC50 = 29 nM T83193 C5ZM8C 5330591 IC50 = 45 nM T83193 CETR65 5366045 EC50 = 4000 nM T83193 C3XA4D 5375465 IC50 > 10000 nM T83193 CU7MX6 5375953 IC50 > 10000 nM T83193 CLO2Q0 5375954 IC50 > 10000 nM T83193 CPX84Y 5394296 IC50 > 10000 nM T83193 C25YUO 5458190 EC50 = 20000 nM T83193 CVD3P2 5704872 IC50 > 10000 nM T83193 CX56UR 5704879 IC50 > 10000 nM T83193 C8JDF6 5775508 IC50 > 10000 nM T83193 CR9HU5 5795514 IC50 = 360 nM T83193 CQG8Z1 5930975 IC50 > 10000 nM T83193 CYU86S 5962587 IC50 > 10000 nM T83193 C6JTH9 6016362 IC50 > 10000 nM T83193 C61ZKG 6018729 IC50 > 4000 nM T83193 CIAL25 6029870 IC50 = 1800 nM T83193 CVC96K 6146604 IC50 = 21 nM T83193 CQ6W2K 6187443 IC50 = 82 nM T83193 C38SOC 6442187 IC50 > 10000 nM T83193 CH1ZX4 6445256 EC50 = 2511.89 nM T83193 CP6D9U 6450018 EC50 = 1.995 nM T83193 C3XYQ7 7354608 IC50 = 370 nM T83193 C1V8ZN 7825385 IC50 = 1200 nM T83193 C83PLM 7914251 IC50 = 120 nM T83193 CD9K5W 7926018 IC50 > 10000 nM T83193 C92YOX 8643775 IC50 = 3490 nM T83193 CVE26J 8668560 EC50 = 4620 nM T83193 CNWP54 8702029 IC50 = 46 nM T83193 C6QO1A 8763094 Ki = 400 nM T83193 C4BYR6 8802859 IC50 = 4100 nM T83193 CHD5I9 9191541 IC50 = 170 nM T83193 CIW52Q 9795270 EC50 = 1200 nM T83193 C8GA6Z 9800250 IC50 = 3.3 nM T83193 CW4Z5B 9802648 Ki = 1.2 nM T83193 CDSI92 9804872 Ki < 10 nM T83193 CY1IX4 9806014 EC50 = 1.34 nM T83193 CKDU64 9819027 Ki = 0.3 nM T83193 C9M0GR 9843337 EC50 = 21300 nM T83193 C7G4AN 9867739 Ki = 3 nM T83193 CS6FN7 9883254 IC50 > 30000 nM T83193 CZJV79 9885200 EC50 = 28100 nM T83193 C67XMD 9885883 EC50 = 22400 nM T83193 C91VSG 9892415 IC50 = 1627 nM T83193 CWXR69 9906556 IC50 = 28 nM T83193 C1QTI8 9950097 IC50 = 18 nM T83193 C79EXD 9950886 IC50 = 26.5 nM T83193 CC0NE7 9975006 IC50 = 24 nM T83193 C19YQR 9975762 IC50 = 10 nM T83193 CVA29T 9975827 Ki = 2.8 nM T83193 C7EK0F 9975828 Ki = 2 nM T83193 CELG21 9977590 IC50 = 3.8 nM T83193 CO7A0B 9983112 IC50 = 0.9 nM T83193 C5D3QA 9985117 IC50 = 0.5 nM T83193 CJ9VY2 9998549 IC50 = 19 nM T83193 C7RX8V 9998550 IC50 = 19 nM T83193 CC0KE3 10022547 IC50 = 15.5 nM T83193 CU02IO 10025997 EC50 = 3.981 nM T83193 C0GC4S 10027372 IC50 = 270 nM T83193 C2UHV7 10028367 Ki = 2 nM T83193 CF41ZU 10041746 IC50 = 680 nM T83193 C2K6IJ 10050089 IC50 = 4 nM T83193 CW29KD 10064626 Ki = 1110 nM T83193 CD84LG 10066181 IC50 = 4 nM T83193 CF4CJ3 10070949 IC50 = 200 nM T83193 CR93GP 10071063 Ki = 4 nM T83193 CB34HN 10084135 EC50 = 1100 nM T83193 CX1DC7 10089889 Ki = 1 nM T83193 C71NWR 10090630 EC50 = 0.5012 nM T83193 CHJB75 10090920 Ki = 1 nM T83193 CNU5H6 10097731 IC50 > 3000 nM T83193 C1RTO5 10125879 IC50 = 620 nM T83193 C8U6LR 10126213 IC50 = 210 nM T83193 C8FKH7 10127170 IC50 = 14 nM T83193 C0IRH4 10127277 IC50 = 7 nM T83193 C5GBZ9 10134409 IC50 = 2.2 nM T83193 CG7VD1 10137465 IC50 = 120 nM T83193 CPZ8N5 10149904 IC50 = 36 nM T83193 CF4Y2Q 10149955 IC50 = 170 nM T83193 C5UAW7 10151288 IC50 = 0.63 nM T83193 CA8J7D 10158754 IC50 = 3.4 nM T83193 CYL9Z3 10171348 IC50 > 10000 nM T83193 C4PA2N 10172003 EC50 = 440 nM T83193 CXT21K 10172112 IC50 = 110 nM T83193 CZRS09 10174189 IC50 = 25 nM T83193 CXRA70 10193842 IC50 = 58 nM T83193 C80JFQ 10194497 IC50 = 20 nM T83193 CHO90S 10194542 IC50 = 60 nM T83193 C30SET 10194869 IC50 = 15 nM T83193 CXOT69 10215278 IC50 = 960 nM T83193 C83KOY 10215307 IC50 = 57 nM T83193 CVR7Y5 10215323 IC50 = 100 nM T83193 C01ESY 10215461 IC50 = 6.5 nM T83193 CZV42N 10215462 IC50 = 270 nM T83193 CHL48Q 10216527 IC50 = 32 nM T83193 C84DFK 10237015 IC50 = 67 nM T83193 CR8W2O 10237016 IC50 = 33 nM T83193 CEB7X5 10238224 IC50 = 2.5 nM T83193 C46FGC 10238413 IC50 = 0.5 nM T83193 CI3CN0 10247042 IC50 = 5.3 nM T83193 CC5HS4 10248318 IC50 = 0.3 nM T83193 CX7UD3 10252323 EC50 = 3.162 nM T83193 CG42MQ 10254025 Ki = 20 nM T83193 CPY9C7 10255515 IC50 = 1015 nM T83193 C2O0AJ 10286990 IC50 = 360 nM T83193 CFL3R4 10288125 IC50 = 290 nM T83193 CCFL59 10291273 IC50 = 5.4 nM T83193 CU90PR 10296445 IC50 = 17 nM T83193 CUW8F6 10308903 IC50 = 2.5 nM T83193 CHXI91 10308951 IC50 = 100 nM T83193 CIGM15 10309581 IC50 = 16 nM T83193 CZ6AM2 10312273 IC50 = 8 nM T83193 CRJ50W 10317518 IC50 = 23.8 nM T83193 CP61TH 10320921 IC50 > 1000 nM T83193 C3HS0L 10322861 IC50 = 25 nM T83193 CJ30SL 10323420 IC50 = 380 nM T83193 CQG58D 10340730 IC50 = 156 nM T83193 C2PI9Q 10341359 Ki = 4 nM T83193 CJ3UF9 10344203 EC50 = 2.512 nM T83193 C0S8FJ 10344437 IC50 = 162 nM T83193 CZKJ20 10344725 Ki = 2 nM T83193 C3NQS1 10357804 Ki = 53 nM T83193 CSW7F0 10367774 IC50 = 1.5 nM T83193 C8DIR2 10382943 IC50 = 123 nM T83193 CC0WP2 10384501 IC50 = 26 nM T83193 C2JI8H 10385075 Ki = 0.8 nM T83193 CGP7U6 10385728 IC50 = 258 nM T83193 C9LFI6 10385845 IC50 = 2.8 nM T83193 CA1IV9 10386145 IC50 = 9.3 nM T83193 CYZG38 10387678 IC50 = 259 nM T83193 C3L9UM 10404960 IC50 = 143 nM T83193 CD2YP6 10406258 IC50 = 189 nM T83193 C29VNT 10406294 IC50 = 51 nM T83193 C6HQY1 10411678 IC50 = 392 nM T83193 CI9P1W 10425263 Ki > 10000 nM T83193 C13MQT 10425327 IC50 = 45 nM T83193 CEH01T 10426159 IC50 = 157 nM T83193 CI0JE6 10428579 Ki = 2.1 nM T83193 C57ZQU 10429018 IC50 = 3.7 nM T83193 CMG9A6 10429408 IC50 = 120 nM T83193 CWO2L8 10429507 IC50 = 3.3 nM T83193 C3LQN4 10447001 IC50 = 1000 nM T83193 CL8IZ5 10448190 IC50 = 6 nM T83193 CEQ06G 10450954 IC50 = 318 nM T83193 CBFE05 10451213 Ki = 1.3 nM T83193 C0U8LP 10452082 Ki = 6 nM T83193 CCAD19 10452485 Ki = 3280 nM T83193 CMPQ64 10452949 IC50 = 9.8 nM T83193 C4N1DL 10453522 IC50 = 0.4 nM T83193 CVFR67 10454306 Ki = 6 nM T83193 CYP0X1 10455072 IC50 = 93 nM T83193 C8AT1X 10455135 IC50 = 43 nM T83193 CV4J7H 10456001 Ki = 5 nM T83193 CAQF96 10472785 IC50 = 37 nM T83193 C25ZDB 10473617 IC50 = 22 nM T83193 CMK18G 10473758 EC50 > 4000 nM T83193 C6LOK4 10474580 Ki = 1 nM T83193 CBXL67 10478501 Ki = 2 nM T83193 C5P1KO 10873969 EC50 = 1.995 nM T83193 CI61XB 10914412 IC50 = 631 nM T83193 C2AHD6 10915682 IC50 = 251.6 nM T83193 C2J6TG 10919020 EC50 = 125.89 nM T83193 CA3B2H 10935516 EC50 = 794.33 nM T83193 CMQP95 10967355 EC50 > 100000 nM T83193 C2LN1R 10972111 EC50 = 6.31 nM T83193 C2VGU8 10974108 EC50 = 1.585 nM T83193 CJN8F0 11050348 EC50 = 501.19 nM T83193 CWE1X8 11081004 EC50 = 794.33 nM T83193 CFP20M 11081027 EC50 = 3.162 nM T83193 CS5FM3 11088005 EC50 = 39.81 nM T83193 C0JHT3 11111493 IC50 = 16.1 nM T83193 CVR3M4 11122626 IC50 = 126.2 nM T83193 CHU16K 11144513 EC50 = 1.259 nM T83193 CJ2FD9 11145177 EC50 = 79.43 nM T83193 C95ODG 11151251 EC50 = 7240 nM T83193 CFV06N 11152242 IC50 = 3 nM T83193 CDG10K 11154380 IC50 = 103 nM T83193 CPS86I 11154448 IC50 = 370 nM T83193 CLD61F 11154884 IC50 = 15 nM T83193 CI02FG 11162142 IC50 = 313 nM T83193 CP54RZ 11163439 IC50 = 3402 nM T83193 C6YWC5 11163678 IC50 = 489.5 nM T83193 CAE8L3 11164115 IC50 = 30 nM T83193 C1A4BU 11164323 IC50 = 21 nM T83193 CWM5V7 11169233 IC50 > 20000 nM T83193 CHY6X9 11174909 IC50 = 1.1 nM T83193 CAF06O 11176490 IC50 = 19 nM T83193 CXG1K0 11176566 IC50 = 104 nM T83193 C1J3LQ 11177997 IC50 = 27 nM T83193 C2SX3V 11185579 IC50 > 4000 nM T83193 CZL23J 11187009 IC50 = 11 nM T83193 C7RB6N 11187610 IC50 = 1500 nM T83193 CR4F1A 11201020 IC50 = 3900 nM T83193 C7M4GR 11202946 IC50 = 123 nM T83193 CM6I4W 11209975 IC50 = 987 nM T83193 CA7FV3 11210430 IC50 = 223 nM T83193 CW49IC 11210873 IC50 = 180 nM T83193 CHF3V9 11220874 IC50 = 68.2 nM T83193 C34WOG 11221698 IC50 = 42 nM T83193 C23SYW 11222319 IC50 = 618 nM T83193 C3XYU2 11233046 IC50 = 500 nM T83193 CU1FD5 11233174 IC50 = 33.4 nM T83193 C9VR3I 11234067 IC50 = 52.2 nM T83193 C6ZUV1 11234223 IC50 = 10 nM T83193 CF2AH5 11234438 IC50 = 124 nM T83193 CX8YP0 11234482 IC50 = 216 nM T83193 CJK04D 11234633 IC50 = 4.7 nM T83193 CGA41K 11235292 IC50 = 44 nM T83193 CZI71C 11235331 IC50 > 4000 nM T83193 CYW2F0 11235811 IC50 = 5030 nM T83193 CZ6MK4 11244984 IC50 = 6 nM T83193 CLOA71 11245391 EC50 = 1930 nM T83193 CR0K5D 11246068 IC50 > 10000 nM T83193 C97YAJ 11246431 IC50 = 3 nM T83193 C2NHQ7 11247081 IC50 = 708 nM T83193 CNW9A3 11247815 IC50 = 41 nM T83193 CKY53N 11255817 IC50 = 30 nM T83193 CKQ1P7 11256604 IC50 = 1220 nM T83193 CT2YA8 11257635 IC50 = 149 nM T83193 C9OWF3 11258604 EC50 > 10000 nM T83193 C6TY2P 11259004 IC50 > 538 nM T83193 CVC36Y 11266760 IC50 = 11 nM T83193 C8YO3L 11266761 IC50 = 46 nM T83193 C5WV4D 11267528 IC50 = 113 nM T83193 C0MJ8A 11268050 IC50 = 33 nM T83193 C56VSC 11268075 IC50 = 10 nM T83193 CR67LW 11278186 IC50 = 595 nM T83193 C9PM7U 11278403 IC50 = 110 nM T83193 C5OPQ9 11279403 IC50 = 87 nM T83193 CM08NB 11280561 IC50 = 170 nM T83193 CX5KL6 11281475 IC50 = 2746 nM T83193 CP5C7W 11281498 IC50 = 965 nM T83193 CH09YB 11290223 IC50 = 40 nM T83193 C5YH7T 11302584 IC50 > 4000 nM T83193 C8W2XI 11313411 IC50 = 10 nM T83193 CNP4Y7 11314287 IC50 = 9.8 nM T83193 CRK15B 11314719 IC50 = 223 nM T83193 CCR10K 11314913 IC50 = 3932 nM T83193 CMV01G 11317360 IC50 = 2700 nM T83193 C50RTJ 11325962 IC50 = 420 nM T83193 C6C5LA 11327231 Ki = 5.1 nM T83193 CU4QC7 11336651 IC50 = 2700 nM T83193 CN75HL 11337328 Ki = 8 nM T83193 CGR09J 11338019 IC50 = 14.2 nM T83193 CMV8T4 11338988 IC50 = 8 nM T83193 C02ELK 11348681 IC50 = 9544 nM T83193 CKD69Y 11360480 IC50 = 44 nM T83193 CD75ZO 11361213 IC50 = 1106 nM T83193 C1N5ED 11371933 IC50 = 2170 nM T83193 CU42XZ 11382833 IC50 = 10 nM T83193 CXO96B 11385287 IC50 = 2290 nM T83193 C8GJB1 11394405 IC50 = 1700 nM T83193 CID3X4 11394918 IC50 = 2415 nM T83193 CTK70N 11395736 IC50 = 15 nM T83193 C74LAW 11407011 IC50 = 6 nM T83193 C1C3TU 11407205 IC50 > 4000 nM T83193 CPU95G 11417553 IC50 = 52.3 nM T83193 CU7K1P 11420211 IC50 = 24 nM T83193 CDCB15 11426745 IC50 = 7200 nM T83193 CM15FO 11427765 IC50 = 150 nM T83193 CQTU13 11428484 IC50 = 290 nM T83193 CVL36R 11428656 IC50 = 270 nM T83193 CHZ75W 11428814 IC50 = 14 nM T83193 CQ13YN 11428847 IC50 = 58 nM T83193 CS2T0N 11430023 IC50 = 3 nM T83193 CE1IT2 11430396 IC50 = 64 nM T83193 CF9L0T 11439510 IC50 = 870 nM T83193 C4VDM3 11440418 IC50 > 4000 nM T83193 CEA7J0 11450944 IC50 = 5030 nM T83193 CD2Z3V 11451387 IC50 = 8 nM T83193 CB6O9N 11452823 IC50 = 3 nM T83193 C52AIL 11461948 IC50 = 3.7 nM T83193 CXC70P 11462535 IC50 = 3 nM T83193 CAW37B 11472797 IC50 = 27 nM T83193 C4J2HQ 11474026 IC50 = 78 nM T83193 CYUZ38 11474160 IC50 = 10 nM T83193 CP1KU4 11475509 IC50 = 44 nM T83193 C9M3QB 11476347 IC50 = 2450 nM T83193 C8XPK4 11484937 IC50 = 39 nM T83193 CRZ3D9 11485402 IC50 = 35 nM T83193 CN83SF 11486920 IC50 = 3383 nM T83193 CFU6A1 11487127 IC50 = 0.42 nM T83193 C07VMY 11494816 IC50 = 7 nM T83193 CM57GQ 11501549 IC50 = 670 nM T83193 C4YA8N 11501768 Ki = 125 nM T83193 CS3Z5T 11502982 IC50 = 29 nM T83193 CI9GW3 11510499 IC50 = 12 nM T83193 CQEK72 11515763 IC50 > 10000 nM T83193 C79ENI 11516347 IC50 = 43 nM T83193 CAVJ68 11516428 Ki = 314 nM T83193 CT30ZK 11516588 IC50 = 1070 nM T83193 CRL9B2 11516653 IC50 = 15 nM T83193 CY8JX7 11523773 IC50 = 1420 nM T83193 CKTQ89 11531155 IC50 = 230 nM T83193 CN6MQ9 11539037 IC50 = 1960 nM T83193 CWQ98U 11539631 Ki = 81 nM T83193 C08RMS 11545784 IC50 = 100 nM T83193 CJ0Y6C 11545915 Ki = 49 nM T83193 CL1DZ9 11545976 IC50 = 90 nM T83193 CDN4L6 11553027 IC50 = 70 nM T83193 CL6FO4 11554008 IC50 = 80 nM T83193 CVWG03 11560077 Ki = 93 nM T83193 C5CJ9Z 11566168 IC50 = 85.9 nM T83193 CB52VF 11566529 IC50 = 417.2 nM T83193 CXZG40 11568188 IC50 = 5610 nM T83193 CGZ52T 11568686 IC50 = 121 nM T83193 CDO0W8 11576806 IC50 = 870 nM T83193 C5ZA9N 11581212 IC50 = 46.7 nM T83193 CG2U8H 11581455 IC50 = 85.6 nM T83193 CV7KX2 11581829 Ki = 56 nM T83193 CMR49W 11582496 Ki = 65 nM T83193 C0BDS3 11588638 IC50 = 3 nM T83193 CS6G2H 11588890 IC50 = 4 nM T83193 CS5F7M 11594915 IC50 = 215 nM T83193 CG0L6V 11595037 IC50 = 1605 nM T83193 C4Z5JK 11595264 IC50 = 34 nM T83193 CDFN62 11595736 Ki = 225 nM T83193 CZ98PT 11601992 IC50 = 175.4 nM T83193 CYI2Z6 11603236 IC50 = 5 nM T83193 CZH2Y9 11610007 IC50 = 11.9 nM T83193 CI3RN0 11610880 Ki = 78 nM T83193 CSW1P8 11611379 IC50 = 66 nM T83193 C74UBE 11618868 IC50 = 800 nM T83193 C21AFU 11624859 Ki = 84 nM T83193 CZ60XH 11633359 Ki = 71 nM T83193 C6ET3R 11638123 IC50 = 234 nM T83193 C91TKC 11639553 IC50 = 41 nM T83193 C19YGI 11639605 Ki = 97 nM T83193 C0ZA2O 11646277 IC50 = 43 nM T83193 CHG1B2 11653471 IC50 = 5 nM T83193 CUDY54 11653760 Ki = 28 nM T83193 CJ15HT 11654024 IC50 = 8 nM T83193 CTD74A 11654160 IC50 = 6 nM T83193 CDZX61 11658617 EC50 = 115000 nM T83193 CB91CF 11661499 IC50 = 13 nM T83193 CD8EV7 11666821 EC50 = 600 nM T83193 CEC8W5 11668297 IC50 = 5 nM T83193 CJD1Q7 11668509 IC50 = 2871 nM T83193 CB0EI8 11669102 IC50 = 160 nM T83193 CIJD47 11674719 IC50 = 1810 nM T83193 CI9AN4 11675434 IC50 > 9000 nM T83193 CH04KW 11682087 IC50 = 19 nM T83193 CC2XH5 11682182 IC50 = 1688 nM T83193 C1QK7U 11688977 IC50 = 157 nM T83193 CHX6L1 11690649 IC50 = 8.4 nM T83193 C4AV3B 11696122 IC50 = 1072 nM T83193 CX6GH9 11696727 Ki = 137 nM T83193 C9QY1C 11696849 IC50 = 110 nM T83193 CFD2G5 11696967 IC50 = 600 nM T83193 CA83LO 11697246 IC50 = 11 nM T83193 CR49WU 11697696 IC50 > 9000 nM T83193 CQSV96 11704438 Ki = 68 nM T83193 CFPJ48 11704662 IC50 = 330 nM T83193 CPW83D 11709865 IC50 > 10000 nM T83193 C0YRW3 11711740 IC50 = 196 nM T83193 CB98GN 11717565 Ki = 61 nM T83193 C0UD1M 11718030 IC50 = 5575 nM T83193 CWV86L 11718098 IC50 = 16 nM T83193 C07CUH 11719337 IC50 = 5 nM T83193 CQ5K8J 11724001 Ki = 7 nM T83193 CHEX57 11725098 IC50 = 11 nM T83193 C8GL3E 11727340 EC50 = 3.162 nM T83193 CB2Q0P 11732417 EC50 = 1.259 nM T83193 CZN6Q7 11738421 IC50 = 52 nM T83193 CMBH71 11739242 IC50 = 670 nM T83193 C0NKI6 11739244 IC50 = 10970 nM T83193 C6VAE8 11739513 Ki = 1.3 nM T83193 CV5TK7 11740163 Ki = 581 nM T83193 CSB74R 11740932 Ki = 85 nM T83193 CBYF51 11749185 IC50 = 5 nM T83193 CT8JR0 11749393 IC50 = 175 nM T83193 C3KOH6 11750331 IC50 = 78 nM T83193 CNI40X 11750583 IC50 = 4 nM T83193 CNK13I 11750695 IC50 = 9 nM T83193 CN3XY8 11755886 IC50 = 2 nM T83193 C9NIB4 11759242 IC50 = 50.3 nM T83193 C5W8VO 11771660 IC50 > 4000 nM T83193 CMU4J6 11772590 IC50 = 280 nM T83193 C4HG5M 11772885 IC50 = 1100 nM T83193 CFB1Z4 11833616 EC50 = 199.53 nM T83193 C1DA0K 11951378 IC50 = 1.4 nM T83193 CCS69F 11951545 IC50 = 1.1 nM T83193 CTY37U 11951546 IC50 = 1.1 nM T83193 C2J7CO 11951910 IC50 = 0.62 nM T83193 CA3BL2 11951911 IC50 = 0.65 nM T83193 C8FJ0P 11955840 IC50 = 374 nM T83193 CV4OB6 11964241 IC50 = 327 nM T83193 CG1D8J 11964255 IC50 = 8.3 nM T83193 CIB79J 11964256 IC50 = 26 nM T83193 CJ3K6G 11964259 IC50 = 15 nM T83193 C2AP5B 11964260 IC50 = 101 nM T83193 C0ZFA2 11964262 IC50 = 62 nM T83193 C6S3AR 11964282 IC50 = 81 nM T83193 C3G2IB 11964283 IC50 = 187 nM T83193 CPM18J 11964284 IC50 = 416 nM T83193 CD6Z2K 11964285 IC50 = 157 nM T83193 C5BG8I 11964318 IC50 = 1820 nM T83193 C3ZXI9 11964319 IC50 = 277 nM T83193 CV3RW9 12110672 EC50 = 30000 nM T83193 CE38OM 12444907 IC50 = 200000 nM T83193 C6VR2A 13309825 EC50 = 60 nM T83193 C7ENX9 13559595 EC50 = 2.512 nM T83193 CBD2C4 13989871 IC50 = 17490 nM T83193 CD6N1T 14954814 IC50 > 10000 nM T83193 C08CSK 16007091 IC50 = 7.943 nM T83193 C2UML7 16035164 IC50 = 42 nM T83193 CPCZ62 16040329 IC50 > 10000 nM T83193 C5CJ0D 16045350 IC50 = 9120 nM T83193 C8Q6HW 16117762 IC50 > 10000 nM T83193 CP86RN 16117763 IC50 > 10000 nM T83193 CGDN09 16223445 Ki = 8.8 nM T83193 CKL25Q 16223447 Ki = 0.9 nM T83193 CZ2Q1X 16223604 Ki = 0.43 nM T83193 CFPN71 16223606 Ki = 1.3 nM T83193 C9I5RW 16223607 Ki = 19.1 nM T83193 C74WGS 16223608 Ki = 0.2 nM T83193 CB76QU 16223640 Ki = 0.3 nM T83193 CBC1R8 16223641 Ki = 0.5 nM T83193 CQ8MY6 16223642 Ki = 0.29 nM T83193 COS90Q 16223643 Ki = 1.1 nM T83193 C56AXM 16223644 Ki = 0.2 nM T83193 CVF6K8 16223645 Ki = 1.4 nM T83193 CH2ZC4 16223802 Ki = 2.1 nM T83193 CX8BV1 16223803 Ki = 0.4 nM T83193 C1RSQ8 16223806 Ki = 7.2 nM T83193 C1TOC0 16223839 Ki = 39.2 nM T83193 CAH18B 16223840 Ki = 9.1 nM T83193 CW7HQ6 16223841 Ki = 0.2 nM T83193 C7KM4H 16223842 Ki = 0.7 nM T83193 CE37HV 16223843 Ki = 0.9 nM T83193 COF9C5 16223844 Ki = 14 nM T83193 C3XHC6 16223998 Ki = 1 nM T83193 CQOF10 16224035 Ki = 0.02 nM T83193 CPL04S 16224036 Ki = 1 nM T83193 C3D1WU 16224037 Ki = 1.3 nM T83193 C6DNC7 16224038 Ki = 3.8 nM T83193 CRO21Z 16224039 Ki = 1.4 nM T83193 CU17TP 16224040 Ki = 3.5 nM T83193 CG3JR8 16224242 Ki = 0.9 nM T83193 C6ZGN2 16224243 Ki = 1.5 nM T83193 CT2E5Q 16224245 Ki = 0.8 nM T83193 C6QD9N 16224246 Ki = 59 nM T83193 CXC0I5 16224444 Ki = 5 nM T83193 CY54BU 16224445 Ki = 1.4 nM T83193 C76PDI 16224446 Ki = 0.6 nM T83193 CM6GV1 16224447 Ki = 4.2 nM T83193 C83EKL 16224449 Ki = 0.6 nM T83193 CQ24AK 16224638 Ki = 2.8 nM T83193 CX0G5W 16224639 Ki = 2 nM T83193 C07ASX 16224640 Ki = 3.4 nM T83193 C7YN2J 16224642 Ki = 1.3 nM T83193 CPS78U 16224643 Ki = 1.4 nM T83193 CHB3W0 16224833 Ki = 2.7 nM T83193 CHK78N 16224834 Ki = 1.2 nM T83193 CSA4V5 16224837 Ki = 6.1 nM T83193 C36QHN 16225030 Ki = 21.6 nM T83193 C7VM5G 16225031 Ki = 0.6 nM T83193 CL4UA3 16225032 Ki = 0.9 nM T83193 CG30SO 16225239 Ki = 1.1 nM T83193 C85JKQ 16225240 Ki = 54 nM T83193 C3S0GA 16225241 Ki = 42 nM T83193 C2T6CF 16225242 Ki = 32.7 nM T83193 CPVX56 16225243 Ki = 0.9 nM T83193 C81WVR 16225448 Ki = 0.9 nM T83193 C31LGV 16225451 Ki = 0.02 nM T83193 CNU8G3 16225452 Ki = 72.1 nM T83193 CZ12PD 16225453 Ki = 1.1 nM T83193 C4ZBD7 16225649 Ki = 0.6 nM T83193 CSR0J5 16225650 Ki = 0.8 nM T83193 CV1MH0 16225651 Ki = 2.4 nM T83193 CM5PT1 16225652 Ki = 0.7 nM T83193 CB0VG2 16225653 Ki = 0.3 nM T83193 CM4VX3 16225654 Ki < 1000 nM T83193 CF5AP8 16225855 Ki = 58 nM T83193 CJ5V2W 16225857 Ki = 9.2 nM T83193 CZ49PD 16389464 EC50 = 5888.44 nM T83193 CVD1R5 16655083 EC50 = 1.5 nM T83193 CQ3R0B 16747867 IC50 = 35.3 nM T83193 CHRA32 16747868 IC50 = 10.3 nM T83193 C6HF8Y 16748125 IC50 = 5.2 nM T83193 CJ7CV2 16748127 IC50 = 4.6 nM T83193 CR20DT 16748248 IC50 = 7360 nM T83193 CA5T8K 16748249 IC50 = 133 nM T83193 C94SBD 16748250 IC50 = 18 nM T83193 C2Q7FT 16748251 IC50 = 54.5 nM T83193 CA9GR3 16748252 IC50 = 43.2 nM T83193 CL2RP7 16748373 IC50 = 12.6 nM T83193 CPEG41 16748374 IC50 = 21.3 nM T83193 CAXZ17 16749111 EC50 > 4000 nM T83193 CVIT85 16749133 IC50 = 7.3 nM T83193 CST26C 16749136 IC50 = 9.3 nM T83193 C6TBH1 16749139 IC50 = 3.3 nM T83193 C1RJ3C 16749216 EC50 > 4000 nM T83193 CMF78C 16749217 EC50 > 4000 nM T83193 C3CY2E 16749218 EC50 > 4000 nM T83193 CJM80O 16749240 IC50 = 5.7 nM T83193 C2K7RW 16749243 IC50 = 14 nM T83193 CB13OV 16749244 IC50 = 190 nM T83193 C96BJP 16749324 EC50 > 4000 nM T83193 CMSA17 16749325 EC50 > 4000 nM T83193 C7U1NO 16749326 EC50 > 4000 nM T83193 C5YG7M 16749350 IC50 = 29.5 nM T83193 CLS61T 16749351 IC50 = 39.3 nM T83193 CMZ32J 16749352 IC50 = 58.8 nM T83193 C3W8DT 16749353 IC50 = 26.9 nM T83193 C0YS5E 16749354 IC50 = 20.4 nM T83193 CHA4N8 16749355 IC50 = 14.8 nM T83193 CWUP76 16749434 EC50 > 4000 nM T83193 CYHC97 16749435 EC50 > 4000 nM T83193 CP3AM6 16749438 IC50 = 1.9 nM T83193 CRQ73A 16749440 EC50 > 4000 nM T83193 CEJ56F 16749462 IC50 = 25.5 nM T83193 CG65CN 16749463 IC50 = 82 nM T83193 C9E4TJ 16749464 IC50 = 157 nM T83193 CI90SF 16749465 IC50 = 1850 nM T83193 CE8I4J 16749466 IC50 = 285 nM T83193 C2G7YQ 16749467 IC50 = 305 nM T83193 CZSC57 16749540 EC50 > 4000 nM T83193 C2EMH9 16749541 EC50 > 4000 nM T83193 CJ9D8L 16749542 EC50 > 4000 nM T83193 C2DK7L 16749543 EC50 > 4000 nM T83193 C4P5CU 16749544 EC50 > 4000 nM T83193 C8GVO1 16749545 EC50 > 4000 nM T83193 CR8EN6 16749565 IC50 = 902 nM T83193 C7AY3O 16749566 IC50 = 19.8 nM T83193 CBNQ43 16749567 IC50 = 29 nM T83193 CX05KR 16749568 IC50 = 22.4 nM T83193 C7EVJ4 16749569 IC50 = 19 nM T83193 CLN50R 17026579 IC50 = 2090 nM T83193 COL7M1 17421069 IC50 > 20000 nM T83193 CI73MC 17946552 IC50 > 10000 nM T83193 CSCY81 18229223 IC50 = 220 nM T83193 C0M4ZI 20090380 IC50 = 6300 nM T83193 CCR2N0 20807401 IC50 > 100000 nM T83193 C1G6OB 21404983 EC50 > 500000 nM T83193 CD6H7C 21598349 EC50 = 7000 nM T83193 CPJ06C 22030032 IC50 = 3 nM T83193 CS2H5P 22030052 IC50 = 0.3 nM T83193 CTI18S 22030066 IC50 = 0.4 nM T83193 CP40BJ 22030080 IC50 = 50 nM T83193 C5L7FA 22030144 IC50 = 24 nM T83193 C1UR9X 22030149 IC50 = 8 nM T83193 CC74QX 22030158 IC50 = 1.2 nM T83193 CZT0O2 22030173 IC50 = 12 nM T83193 CTU13R 22030183 IC50 = 6 nM T83193 C1HX4L 22030187 IC50 = 1 nM T83193 C7Y2SH 22030227 IC50 = 184 nM T83193 CRG70B 22030273 IC50 = 25 nM T83193 C6I7AP 22030278 IC50 = 35 nM T83193 C7O8AG 22030332 IC50 = 26 nM T83193 C8D4WK 22030340 IC50 = 2.1 nM T83193 C72FHC 22030363 IC50 = 2 nM T83193 C08ZUA 22030387 IC50 = 9 nM T83193 CMVA64 22030491 IC50 = 69 nM T83193 CDP5Y6 22030498 IC50 = 22 nM T83193 C0AS3O 22032592 IC50 = 19 nM T83193 CS9HJ7 22032616 IC50 = 94 nM T83193 CZRU05 22032622 Ki = 1.2 nM T83193 C17MCO 22032643 IC50 = 109 nM T83193 C6DGX1 22170442 IC50 = 0.8 nM T83193 C2W7TH 22258331 Ki = 0.8 nM T83193 CCG43N 22296670 IC50 = 141000 nM T83193 CR95GN 22337681 IC50 = 184 nM T83193 C3IEK4 23112208 IC50 = 350 nM T83193 CQ6XH2 23344732 IC50 = 320 nM T83193 C21YMA 23537063 IC50 = 62 nM T83193 C0B6WM 23537081 IC50 = 4.5 nM T83193 C9AI6U 23537111 IC50 = 25 nM T83193 CRF62A 23655242 IC50 = 41 nM T83193 CFK41Y 24106939 IC50 = 750 nM T83193 C2Z7MA 24749054 IC50 = 5250 nM T83193 CG0S9O 24749055 IC50 > 10000 nM T83193 CS3HD4 24749056 IC50 > 10000 nM T83193 C38RVI 24749057 IC50 > 10000 nM T83193 C3TRX4 24749058 IC50 > 10000 nM T83193 C5HCO9 24749162 IC50 = 470 nM T83193 C3L9PN 24749163 IC50 = 950 nM T83193 CJM71S 24749268 IC50 = 2570 nM T83193 CMNG82 24749269 IC50 > 10000 nM T83193 C7A1XM 24749272 IC50 = 2130 nM T83193 CM80VR 24749273 IC50 = 680 nM T83193 CU8EK4 24749373 IC50 = 240 nM T83193 C3FB1Y 24749374 IC50 = 430 nM T83193 CNVL17 24749375 IC50 = 3800 nM T83193 CI5P1B 24749376 IC50 = 2630 nM T83193 CWJ38Z 24749377 IC50 > 10000 nM T83193 CSD74Y 24749378 IC50 > 10000 nM T83193 C9F4CD 24749379 IC50 = 720 nM T83193 C5FJX1 24749485 IC50 > 10000 nM T83193 COY93F 24749486 IC50 > 10000 nM T83193 CAP1H6 24749487 IC50 = 2820 nM T83193 CC5Y4U 24749488 IC50 > 10000 nM T83193 CZ2H9N 24749489 IC50 > 10000 nM T83193 C6X1VD 24749490 IC50 > 10000 nM T83193 CI0L7N 24749586 IC50 = 2400 nM T83193 C6OXY3 24749587 IC50 > 10000 nM T83193 CHA2W7 24749588 IC50 > 10000 nM T83193 C4YU1Z 24749589 IC50 > 10000 nM T83193 CG32EF 24749590 IC50 > 10000 nM T83193 CG2E6O 24749591 IC50 > 10000 nM T83193 C2WF7Z 24749592 IC50 > 10000 nM T83193 CJ4E8Q 24749698 IC50 > 10000 nM T83193 CZ3TN1 24757992 IC50 = 300 nM T83193 CM8U7N 24758358 IC50 = 4.9 nM T83193 CIG1Z2 24758469 IC50 = 6 nM T83193 CAL0Z8 24758809 IC50 = 25 nM T83193 C8M2ZV 24758810 IC50 = 12 nM T83193 CHW1G2 24758811 IC50 = 140 nM T83193 CL1B4P 24758812 IC50 = 400 nM T83193 C9KHG4 24758813 IC50 = 40 nM T83193 CDQ6V0 24758928 IC50 = 2 nM T83193 CZ95VW 24758929 IC50 = 280 nM T83193 COS08A 24758930 IC50 = 210 nM T83193 CQLK06 24759035 IC50 = 10 nM T83193 CVI60T 24759038 IC50 = 120 nM T83193 C5ZB7W 24759039 IC50 = 45 nM T83193 C0D6BW 24759147 IC50 = 250 nM T83193 CSY3H1 24759484 IC50 = 76 nM T83193 C8QY4E 24759485 IC50 = 5.7 nM T83193 CWD7S2 24768191 Ki = 23 nM T83193 C7CNH2 24768197 IC50 = 147 nM T83193 CY02IF 24768198 IC50 = 125 nM T83193 CMC85W 24768199 IC50 = 171 nM T83193 CWY73R 24768200 IC50 = 46 nM T83193 CHL87D 24768201 IC50 = 20 nM T83193 CXO93T 24768202 IC50 = 17 nM T83193 CBMO21 24768204 IC50 = 31000 nM T83193 C9OL1G 24768205 IC50 = 15900 nM T83193 CUT5L4 24768206 IC50 = 476 nM T83193 CV31NY 24768207 IC50 = 287 nM T83193 C3NTZ4 24768208 IC50 = 47 nM T83193 CE27QX 24768209 IC50 = 248 nM T83193 CTQ1W2 24777535 IC50 = 19 nM T83193 C1NIH2 24777650 IC50 = 5 nM T83193 CF65KY 24777651 IC50 = 151 nM T83193 C03AVT 24777652 IC50 = 1350 nM T83193 C2Q4KN 24777657 IC50 = 127 nM T83193 C8IE1C 24777768 IC50 = 9 nM T83193 C63OSW 24777769 IC50 = 7 nM T83193 CTF76E 24777770 IC50 = 5 nM T83193 CYDV94 24777771 IC50 = 4 nM T83193 CV4E5Y 24777772 IC50 = 14 nM T83193 CBFM91 24777773 IC50 = 65 nM T83193 CVT9S0 24777889 IC50 = 5820 nM T83193 CE2I0G 24782892 IC50 = 188 nM T83193 CMN74Q 24782895 IC50 = 37 nM T83193 CUP61J 24783145 IC50 = 97 nM T83193 CT31VS 24783399 IC50 = 6160 nM T83193 C0NCS2 24783400 IC50 = 907 nM T83193 C7C9HL 24783403 IC50 = 6 nM T83193 C7D6JX 24783656 IC50 = 38 nM T83193 CL8T0V 24784683 IC50 = 361 nM T83193 C94OHQ 24784927 IC50 = 1450 nM T83193 CHYD03 24785963 IC50 = 2360 nM T83193 CB20PL 24795576 EC50 = 5000 nM T83193 CR40XN 24882612 IC50 = 23 nM T83193 C53HIK 24882754 IC50 = 2 nM T83193 CBW81E 24882793 IC50 = 5 nM T83193 CJN68G 24882876 IC50 = 13 nM T83193 CO7TH0 24882956 IC50 = 19 nM T83193 C75JOU 24882957 IC50 = 14 nM T83193 C1DQZ5 24882958 IC50 = 11 nM T83193 CFS9X6 24882959 IC50 = 21 nM T83193 CMV64G 24883004 IC50 = 23 nM T83193 CD6C5J 24883048 IC50 = 9 nM T83193 CRT08K 24883050 IC50 = 64 nM T83193 CI05FC 24883053 IC50 > 5000 nM T83193 CH0X7O 24883095 IC50 > 5000 nM T83193 C9K3MG 24883145 IC50 = 3 nM T83193 C0PUW7 24883305 IC50 = 63 nM T83193 C94XJC 24883307 IC50 = 12 nM T83193 CQKS73 24883308 IC50 = 59 nM T83193 C74BIP 24883353 IC50 = 3 nM T83193 CZRP90 24883354 IC50 = 41 nM T83193 CCN98Y 24883355 IC50 = 30 nM T83193 C7ODK0 24952932 IC50 = 101 nM T83193 C9YNW1 24952933 IC50 = 85 nM T83193 CRXY84 24970014 Ki = 3.79 nM T83193 CL0Q2W 25063516 Ki = 387 nM T83193 CJV2N6 25063517 Ki = 1.7 nM T83193 CGB14D 25063519 Ki = 0.2 nM T83193 C63HTY 25063555 Ki = 169 nM T83193 C2CLW4 25063559 Ki = 0.3 nM T83193 CUE06S 25063560 Ki = 0.6 nM T83193 CDIT59 25063596 Ki = 3.5 nM T83193 COCD41 25063598 Ki = 68.8 nM T83193 C6TSU3 25063599 Ki = 0.3 nM T83193 CZ6XV1 25063600 Ki = 0.9 nM T83193 CAZ23X 25063601 Ki = 6.4 nM T83193 C8CG5I 25063673 Ki = 2.3 nM T83193 CYIO54 25063675 Ki = 0.3 nM T83193 CF6O7A 25063709 Ki = 0.6 nM T83193 C16RAM 25063712 Ki = 59.4 nM T83193 CKQT89 25063747 Ki = 1.1 nM T83193 C0OTC3 25063748 Ki = 28.6 nM T83193 C0NUI7 25063787 Ki = 1.9 nM T83193 CV5JH8 25098503 Ki = 11.9 nM T83193 CSL79N 25098504 Ki = 55.5 nM T83193 CAW8P2 25102898 Ki = 0.1 nM T83193 CSG03M 25102901 Ki = 56.4 nM T83193 CCT35Q 25103505 Ki = 49.3 nM T83193 CN8X5E 25103635 Ki = 65.9 nM T83193 CV17BS 25103751 Ki = 49 nM T83193 C3JDL5 25103752 Ki = 62.5 nM T83193 C2C8ML 25103753 Ki = 65.7 nM T83193 C2X5RB 25103754 Ki = 1.3 nM T83193 CX2DO1 25103755 Ki = 124 nM T83193 C3G0BK 25104002 Ki = 7.5 nM T83193 CQ2BL0 25104247 Ki = 103 nM T83193 CT1MR7 25104361 Ki = 88.7 nM T83193 C90GAW 25104362 Ki = 42.9 nM T83193 C5XM0A 25104364 Ki = 3.4 nM T83193 C3PQ4U 25104478 Ki = 2.4 nM T83193 CM63CF 25104699 Ki = 1.1 nM T83193 CYA91N 25123379 Ki = 4.4 nM T83193 CB5LO8 25124040 Ki = 25 nM T83193 CXS51N 25124352 Ki = 0.9 nM T83193 CVM5H0 25124353 Ki = 0.7 nM T83193 CX6GR1 25124356 Ki = 9.6 nM T83193 C6K7FP 25141397 IC50 = 3000 nM T83193 CXT31S 25147549 IC50 = 15 nM T83193 CG5SI9 25181624 IC50 = 118 nM T83193 CP3JB6 25181625 IC50 = 5.012 nM T83193 CPH98K 25181768 IC50 = 79 nM T83193 CG7HA8 25181770 IC50 = 23 nM T83193 CW9J5U 25181771 IC50 = 0.5012 nM T83193 CPZA63 25181773 IC50 = 0.631 nM T83193 CRAE91 25181908 IC50 = 43 nM T83193 C21MGD 25181909 IC50 = 46 nM T83193 CA78YZ 25181911 IC50 = 55 nM T83193 CT8SH5 25182164 IC50 = 87 nM T83193 CG2K6M 25182166 IC50 = 92 nM T83193 CG5K9X 25182169 IC50 = 392 nM T83193 CO73NW 25182447 IC50 = 0.631 nM T83193 CHR4D8 25182737 IC50 = 1.995 nM T83193 CVM90Z 25182893 IC50 = 12.59 nM T83193 CK7F2C 25195123 IC50 = 8.5 nM T83193 CRC21B 25241873 IC50 = 3.2 nM T83193 CI8SQ7 25263541 IC50 = 17 nM T83193 CTW7E8 25263542 IC50 = 150 nM T83193 C6DX5M 25264621 IC50 = 4 nM T83193 CJO5R6 25264622 IC50 = 16 nM T83193 C8AIY7 25264623 IC50 = 4 nM T83193 CE04YM 25264757 IC50 = 7 nM T83193 C32USM 25264907 IC50 = 6 nM T83193 CR4T9V 25264908 IC50 = 7 nM T83193 CJ50IN 25265057 IC50 = 6 nM T83193 C20XDK 25265635 IC50 = 40 nM T83193 C7FBO1 25270198 IC50 = 15 nM T83193 CL3KW6 25270199 IC50 = 4.8 nM T83193 C4U3OE 25840617 IC50 > 10000 nM T83193 C1B0ZO 25840619 IC50 > 10000 nM T83193 CBR69Y 25840620 IC50 > 10000 nM T83193 C1YN3E 27838559 IC50 = 1930 nM T83193 CS43UD 29372808 IC50 = 74 nM T83193 CS3U9T 30294430 IC50 = 59 nM T83193 C1YT6G 35368250 IC50 > 10000 nM T83193 CJX06W 36223059 Ki > 3000 nM T83193 CBR9U4 42613351 EC50 = 1000 nM T83193 C9QF7X 42617987 EC50 = 26400 nM T83193 CYB0L5 42617988 EC50 = 40 nM T83193 CJR92V 44189702 Ki = 0.49 nM T83193 C8S9PC 44271987 Ki = 1.46 nM T83193 C3IJC8 44271988 Ki = 1.4 nM T83193 C1FJV0 44272140 Ki = 0.71 nM T83193 CNLI07 44276258 Ki = 66.1 nM T83193 CF10YJ 44276297 Ki = 149 nM T83193 CCY37M 44334307 IC50 = 38 nM T83193 C2A1TY 44334308 Ki = 4 nM T83193 CHXW51 44334309 Ki = 11 nM T83193 CV6RC0 44334375 Ki = 330 nM T83193 CU4T5Q 44334391 IC50 = 2.4 nM T83193 CJ8U2P 44334401 Ki = 19 nM T83193 CP5M4B 44334439 Ki = 160 nM T83193 C63ZPI 44334455 Ki = 17 nM T83193 C07IZG 44334734 Ki = 1.4 nM T83193 C71XAD 44348204 EC50 = 5.012 nM T83193 CJ4BM2 44348288 EC50 = 199.53 nM T83193 CB6D5O 44348320 EC50 = 5.012 nM T83193 C6KMD9 44348328 EC50 = 19.95 nM T83193 CI5JL6 44348331 EC50 = 0.3981 nM T83193 C0LOT7 44366106 Ki = 4.6 nM T83193 C09VPI 44366285 Ki = 4 nM T83193 CV3W5G 44366327 Ki = 9.8 nM T83193 CR12UP 44366328 IC50 = 770 nM T83193 C3CKU0 44386779 IC50 = 0.4 nM T83193 C96REQ 44387739 IC50 > 10000 nM T83193 C8GYE2 44387747 IC50 = 526 nM T83193 C6GQB7 44387748 EC50 = 1160 nM T83193 C78BVO 44387749 IC50 = 1310 nM T83193 C3UQS8 44387754 EC50 = 618 nM T83193 CUP59X 44387767 IC50 = 12100 nM T83193 C5EIO1 44387768 EC50 = 5260 nM T83193 C17ZVR 44387769 IC50 = 334 nM T83193 C2Q6TB 44387771 IC50 = 2280 nM T83193 CIE4Q2 44387778 IC50 = 367 nM T83193 C7A3UJ 44387779 IC50 = 8130 nM T83193 C46CST 44387781 IC50 = 908 nM T83193 CFOH27 44391151 IC50 = 776 nM T83193 C8T6VB 44391169 IC50 = 3128 nM T83193 CG9D1C 44391183 IC50 = 2143 nM T83193 CL3QU4 44391189 IC50 = 726 nM T83193 C25KZQ 44391190 IC50 = 305 nM T83193 C6I0DX 44391210 IC50 = 948 nM T83193 CN90WE 44391216 IC50 = 10000 nM T83193 CU3XC1 44391232 IC50 = 5773 nM T83193 CW83NP 44391233 IC50 = 325 nM T83193 CC43MN 44391249 IC50 = 665 nM T83193 C7X3EZ 44391250 IC50 = 5447 nM T83193 C5R2SC 44395836 IC50 = 2796 nM T83193 CT84UQ 44395837 IC50 = 4867 nM T83193 CTY85S 44395850 IC50 > 10000 nM T83193 C9CO4K 44395916 IC50 = 2178 nM T83193 C0ZG1C 44395917 IC50 > 10000 nM T83193 C2Q3EG 44395921 IC50 > 10000 nM T83193 CCA71Z 44395934 IC50 > 10000 nM T83193 C76MTS 44395937 IC50 = 8.5 nM T83193 CG92UT 44395945 IC50 = 8590.7 nM T83193 C8CH9T 44395955 IC50 = 3825.8 nM T83193 CFU3Q9 44395965 IC50 > 10000 nM T83193 C05DPN 44395979 IC50 > 10000 nM T83193 CEV27Q 44395981 IC50 > 10000 nM T83193 CB67VI 44395992 IC50 = 279 nM T83193 C84DTU 44395995 IC50 > 10000 nM T83193 C2W4RX 44395996 IC50 > 10000 nM T83193 CON6R0 44396004 IC50 > 10000 nM T83193 CX9C2V 44396013 IC50 > 10000 nM T83193 C58JNY 44396021 IC50 > 10000 nM T83193 C31NUC 44396024 IC50 > 10000 nM T83193 CXCQ03 44396026 IC50 = 67.5 nM T83193 CJ1BR0 44396035 IC50 = 8118.8 nM T83193 C5HO1D 44396060 IC50 = 176.6 nM T83193 C8RP3K 44396061 IC50 = 1623 nM T83193 CNET70 44396064 IC50 = 2154 nM T83193 CFDE76 44396075 IC50 > 10000 nM T83193 C0GHL8 44396080 IC50 > 10000 nM T83193 CM8HA5 44396081 IC50 > 10000 nM T83193 CL91XU 44396083 IC50 = 57.7 nM T83193 CJPK65 44396086 IC50 > 25000 nM T83193 C3LFO6 44396088 IC50 > 10000 nM T83193 C7DN0E 44396089 IC50 > 10000 nM T83193 CY69FU 44396093 IC50 > 10000 nM T83193 COQE95 44396094 IC50 > 10000 nM T83193 CC4K5Q 44396107 IC50 > 10000 nM T83193 CJK3B7 44396111 IC50 > 10000 nM T83193 CCP3L4 44396112 IC50 = 340 nM T83193 C9F0TP 44396115 IC50 = 5745 nM T83193 CHKC63 44396118 IC50 > 10000 nM T83193 CVZ2R9 44396121 IC50 > 10000 nM T83193 CQX6S5 44396143 IC50 > 10000 nM T83193 C09WPE 44396145 IC50 = 300.7 nM T83193 CHD94P 44396146 IC50 = 893 nM T83193 CTD74U 44396150 IC50 = 5021 nM T83193 CXY71J 44396164 IC50 = 2727 nM T83193 CC52ZU 44396172 IC50 = 6169 nM T83193 C0JYQ8 44398602 IC50 = 2740 nM T83193 CCDT79 44398616 IC50 = 389.6 nM T83193 CZP60S 44398654 IC50 = 355.3 nM T83193 CJZB34 44398661 IC50 = 10380 nM T83193 C1U4DF 44398772 IC50 > 20000 nM T83193 CR47MA 44400841 IC50 = 1800 nM T83193 C8R1NG 44406816 IC50 = 49 nM T83193 CYS04D 44412342 IC50 = 470 nM T83193 CA87CB 44412350 IC50 = 640 nM T83193 C69TCS 44412351 IC50 = 22 nM T83193 CUV46O 44412359 IC50 = 224 nM T83193 CB6U8P 44412367 IC50 = 170 nM T83193 C8NU9I 44412368 IC50 = 320 nM T83193 CB6N0V 44412369 IC50 = 290 nM T83193 C0T8JU 44412401 IC50 = 24 nM T83193 CZ6EH0 44412449 IC50 = 340 nM T83193 CP29AX 44412456 IC50 = 1500 nM T83193 C2YW6P 44412457 IC50 = 160 nM T83193 CV92RL 44412465 IC50 = 2400 nM T83193 C0RT4W 44412466 IC50 = 1100 nM T83193 C81QGK 44416398 IC50 = 42 nM T83193 C6GX3K 44416399 IC50 = 233 nM T83193 C74DWR 44416414 IC50 = 3669 nM T83193 C1W3EM 44416415 IC50 = 387 nM T83193 CQ90TZ 44416416 IC50 > 4000 nM T83193 CF8I9J 44416417 IC50 = 624 nM T83193 CY7ZI6 44416441 IC50 = 1779 nM T83193 C0JM2B 44416470 IC50 = 91 nM T83193 CQW7G5 44416491 IC50 > 4000 nM T83193 CT2HX5 44416493 IC50 > 4000 nM T83193 CUK10L 44416494 IC50 > 4000 nM T83193 CG7W3F 44416519 IC50 = 60 nM T83193 C0T8MF 44416550 IC50 = 746 nM T83193 CUG3C2 44416551 IC50 > 4000 nM T83193 C6KJG8 44416573 IC50 = 1412 nM T83193 CV4SR3 44416597 IC50 = 4303 nM T83193 C3KN2W 44416619 IC50 = 1527 nM T83193 CS94LP 44416642 IC50 = 257 nM T83193 C6M8EL 44416643 IC50 = 131 nM T83193 CT1BK4 44416662 IC50 > 4000 nM T83193 CI0P3Q 44416754 IC50 = 974 nM T83193 C9MB0K 44416755 IC50 = 189 nM T83193 CHC7D3 44416759 IC50 > 4000 nM T83193 CP80IX 44416784 IC50 > 4000 nM T83193 CQ1A2Z 44416785 IC50 = 65 nM T83193 C9HA3I 44416788 IC50 > 4000 nM T83193 CR5U4E 44416860 IC50 > 4000 nM T83193 C8GLZ1 44416863 IC50 = 49 nM T83193 CXST24 44416878 IC50 = 417 nM T83193 CVN68O 44416879 IC50 = 24 nM T83193 CSB61J 44416900 IC50 = 377 nM T83193 C84IAM 44416931 IC50 = 158 nM T83193 CCA8J4 44416932 IC50 = 190 nM T83193 CLFO48 44416952 IC50 = 49 nM T83193 CCZ8G2 44416971 IC50 = 62 nM T83193 C32FIC 44416972 IC50 = 152 nM T83193 CZV6L3 44416973 IC50 = 39 nM T83193 C1UHR8 44417047 IC50 = 73 nM T83193 CPND83 44417048 IC50 > 4000 nM T83193 CF71AH 44417070 IC50 > 4000 nM T83193 C7RW0A 44417071 IC50 = 1502 nM T83193 CKM17E 44417074 IC50 = 91 nM T83193 CQE0Z5 44417075 IC50 = 168 nM T83193 C3JC2H 44426231 IC50 = 3750 nM T83193 C2HR7A 44426233 IC50 = 123 nM T83193 CRFB27 44430071 EC50 = 9.4 nM T83193 CY8JL9 44430072 EC50 = 4.6 nM T83193 CDTP25 44430073 EC50 = 25.5 nM T83193 CZHI60 44430074 EC50 = 4.7 nM T83193 C52AJN 44430075 EC50 = 51.5 nM T83193 C2CD1Z 44430076 EC50 = 69.5 nM T83193 CXC58F 44430077 EC50 = 1.9 nM T83193 C21OIG 44430078 EC50 = 15.2 nM T83193 C3JKY0 44430082 EC50 = 8.6 nM T83193 CX1TW8 44430086 EC50 = 7.9 nM T83193 CH9XY0 44433395 IC50 = 42 nM T83193 CFP90W 44444341 IC50 = 680 nM T83193 CI56CT 44444349 IC50 = 184 nM T83193 C7JF0C 44444350 Ki = 4 nM T83193 CIVW16 44444351 IC50 = 5 nM T83193 C0HL3F 44444357 IC50 = 19 nM T83193 CZ2KI3 44444374 Ki = 10 nM T83193 CO04XT 44444381 Ki = 22 nM T83193 C2BP8Z 44444392 Ki = 11 nM T83193 CZ03IW 44444394 Ki = 4 nM T83193 C5JX2M 44444395 Ki = 16 nM T83193 CWU59D 44444396 Ki = 2 nM T83193 CY64IB 44444397 IC50 > 1000 nM T83193 CSI8P9 44444398 Ki = 8 nM T83193 CM7X2P 44444399 Ki = 17 nM T83193 C8Z1RQ 44444400 Ki = 1 nM T83193 CWF8P0 44444401 Ki = 1 nM T83193 C0SM7N 44444918 IC50 = 11 nM T83193 CIF3H2 44447609 IC50 = 70 nM T83193 C8UMG2 44447610 IC50 = 14 nM T83193 CI67JP 44447611 IC50 = 790 nM T83193 C4H5ZI 44447612 IC50 = 1400 nM T83193 CC7J0M 44447613 IC50 > 10000 nM T83193 CXQ64G 44447614 IC50 = 220 nM T83193 CGV17K 44447615 IC50 > 10000 nM T83193 C98GNL 44447617 IC50 > 10000 nM T83193 C07OUB 44447618 IC50 = 253 nM T83193 CLX6H3 44447619 IC50 > 10000 nM T83193 CJI0F1 44447620 IC50 > 10000 nM T83193 C59OWX 44447621 IC50 > 10000 nM T83193 CE67YB 44447622 IC50 > 10000 nM T83193 C9IE0S 44447623 IC50 > 10000 nM T83193 CVXH28 44447624 IC50 = 6000 nM T83193 CPJ0I5 44447625 IC50 > 10000 nM T83193 CK0BR6 44447626 IC50 > 10000 nM T83193 C7TGS0 44447627 IC50 = 380 nM T83193 CN30TO 44447628 IC50 = 477 nM T83193 CLJ6B8 44447629 IC50 = 1420 nM T83193 C5VH4R 44447630 IC50 = 4970 nM T83193 C7IU4D 44447631 IC50 > 10000 nM T83193 CQ89RW 44447632 IC50 = 1310 nM T83193 C9JW1X 44447633 IC50 = 1640 nM T83193 CJ28NP 44447634 IC50 = 1730 nM T83193 CKTP16 44447635 IC50 = 3720 nM T83193 CJXI21 44447636 IC50 > 10000 nM T83193 C7S9OY 44447637 IC50 = 2620 nM T83193 CAF50B 44447638 IC50 = 205 nM T83193 CO4HF6 44447639 IC50 = 776 nM T83193 C5A1IB 44447641 IC50 = 2560 nM T83193 CCV8W3 44447642 IC50 = 3700 nM T83193 CA3TM9 44447648 IC50 = 1890 nM T83193 C7ZKH5 44447649 IC50 = 1160 nM T83193 C7AO1C 44447650 IC50 = 3430 nM T83193 C6J5TL 44447651 IC50 > 10000 nM T83193 COCQ06 44447652 IC50 > 10000 nM T83193 CK4OE2 44447653 IC50 = 3940 nM T83193 C1YR8I 44447654 IC50 = 3400 nM T83193 CPO9Q6 44447655 IC50 > 10000 nM T83193 C26JRZ 44447667 IC50 = 400 nM T83193 CHB65M 44447668 IC50 = 550 nM T83193 C7T2DQ 44447669 IC50 = 5070 nM T83193 C0Y7IX 44447670 IC50 = 3280 nM T83193 CYR56O 44447671 IC50 = 490 nM T83193 CL4HR0 44447672 IC50 = 200 nM T83193 CD80OW 44447673 IC50 = 2600 nM T83193 C0P1QK 44447674 IC50 > 10000 nM T83193 CC6M4A 44447675 IC50 = 6700 nM T83193 CN5W9K 44447676 IC50 = 4600 nM T83193 CW4PO2 44447677 IC50 = 5400 nM T83193 C0TY7X 44447678 IC50 = 7300 nM T83193 CWK61M 44447679 IC50 = 1400 nM T83193 CM6FB3 44447680 IC50 > 10000 nM T83193 C4YV8G 44447681 IC50 > 10000 nM T83193 CVL4W5 44447682 IC50 > 10000 nM T83193 CO5MJ1 44447683 IC50 = 4650 nM T83193 COW25J 44447684 IC50 = 3550 nM T83193 CRNM76 44447685 IC50 = 150 nM T83193 CHEP38 44447686 IC50 = 76 nM T83193 CSWN64 44447687 IC50 = 1230 nM T83193 CP3WU4 44447688 IC50 = 960 nM T83193 CFW8G9 44447689 IC50 = 1350 nM T83193 CF5EB0 44447690 IC50 = 3100 nM T83193 CAZ4E9 44447691 IC50 > 10000 nM T83193 CQB6I3 44447692 IC50 = 81 nM T83193 CHO2B5 44447693 IC50 = 740 nM T83193 CW1VH4 44447972 IC50 = 70 nM T83193 CIJB18 44447973 IC50 = 32 nM T83193 CRY47W 44448494 EC50 > 100000 nM T83193 CA49WS 44448505 EC50 > 100000 nM T83193 C6AY8U 44448506 EC50 = 29600 nM T83193 C7ZJ9O 44448536 EC50 > 100000 nM T83193 C72IYN 44448539 EC50 = 15000 nM T83193 CZTQ62 44448540 EC50 = 53500 nM T83193 C4G9YD 44448542 EC50 > 100000 nM T83193 CBA36L 44448576 EC50 > 100000 nM T83193 CSB9M8 44448577 EC50 > 100000 nM T83193 C0J4VA 44448578 EC50 > 100000 nM T83193 CGL3J5 44448579 EC50 > 100000 nM T83193 COWF13 44448613 EC50 > 100000 nM T83193 C7VGI3 44448615 EC50 > 100000 nM T83193 CIR53D 44448618 EC50 > 100000 nM T83193 CVB6E5 44448647 EC50 > 100000 nM T83193 CS9YA3 44448648 EC50 > 100000 nM T83193 C7JYR2 44448650 EC50 > 100000 nM T83193 C7FU4D 44450275 Ki = 16 nM T83193 CH76LB 44450299 Ki = 1471 nM T83193 C64CPA 44450314 Ki = 24 nM T83193 CEF47K 44450323 Ki = 38 nM T83193 CJC7Y0 44450337 IC50 > 30000 nM T83193 C5F1JL 44450338 Ki = 267 nM T83193 CU6Q2L 44450367 Ki > 3000 nM T83193 C52CIP 44450378 Ki > 3000 nM T83193 C67ZYA 44454325 IC50 = 10 nM T83193 C0LWU9 44454328 IC50 = 2.9 nM T83193 C6GZ8V 44454360 IC50 = 2.1 nM T83193 CC31AH 44566752 IC50 > 200000 nM T83193 CC9Q7V 44569302 IC50 = 539 nM T83193 C3VZY7 44569303 IC50 = 224 nM T83193 CBYE01 44569304 IC50 = 274 nM T83193 CY6O1V 44569360 IC50 = 5000 nM T83193 CO54EV 44569361 IC50 = 184 nM T83193 CSG9U4 44569441 IC50 = 59 nM T83193 CJ82AH 44569442 IC50 = 48 nM T83193 CX25DT 44569484 IC50 = 39 nM T83193 CTI30N 44569485 IC50 = 1 nM T83193 C9R5XV 44569566 IC50 > 5000 nM T83193 C8BN2K 44569567 IC50 = 680 nM T83193 C6N8YA 44569568 IC50 > 5000 nM T83193 C9TR7S 44569601 IC50 = 502 nM T83193 CVW69G 44569602 IC50 = 43 nM T83193 C03OFA 44569641 IC50 = 234 nM T83193 CJ2X4R 44569642 IC50 = 51 nM T83193 CC8WO2 44569643 IC50 = 74 nM T83193 CP9DQ2 44569644 IC50 > 5000 nM T83193 CLAV98 44569672 IC50 = 95 nM T83193 CRP64A 44569673 IC50 = 125 nM T83193 CGN01P 44569738 IC50 = 69 nM T83193 C5K7OD 44569739 IC50 = 820 nM T83193 CN5K2H 44569740 IC50 > 5000 nM T83193 CJT58N 44569741 IC50 > 5000 nM T83193 C3SU5I 44569781 IC50 > 5000 nM T83193 CNK24D 44569782 IC50 > 5000 nM T83193 CFZ3H1 44569783 IC50 = 206 nM T83193 CJH87Z 44569784 IC50 > 5000 nM T83193 COW7F2 44569785 IC50 = 176 nM T83193 CD4O8U 44569814 IC50 = 33 nM T83193 C5JAG6 44569815 IC50 = 10 nM T83193 C5YGU6 44569816 IC50 = 31 nM T83193 CA2W1E 44569847 IC50 = 96 nM T83193 C6Y1ZB 44569848 IC50 > 5000 nM T83193 CB9F4A 44569849 IC50 > 5000 nM T83193 CR6UV4 44569850 IC50 > 5000 nM T83193 CUQ39B 44569893 IC50 > 5000 nM T83193 CS89MB 44569894 IC50 = 1 nM T83193 CMJ97X 44570894 IC50 = 9.4 nM T83193 C9YTH7 44570896 IC50 = 32 nM T83193 C2IWK3 44570932 IC50 = 226 nM T83193 C15JVN 44570933 IC50 = 205 nM T83193 CS6D5L 44570976 IC50 = 80 nM T83193 C4OJ3F 44571024 IC50 = 81 nM T83193 CCE67G 44579757 IC50 = 67 nM T83193 CQ25HD 44579758 IC50 = 35 nM T83193 CZA30W 44579759 IC50 = 95 nM T83193 C78CWZ 44579760 IC50 = 196 nM T83193 C9P5KO 44580000 IC50 = 78 nM T83193 C2C7NM 44580001 IC50 = 27 nM T83193 CQ84AH 44580002 IC50 = 19 nM T83193 C15HBR 44580003 IC50 = 14 nM T83193 CO13LW 44580004 IC50 = 10 nM T83193 CV1O7Z 44580033 IC50 = 265 nM T83193 C64AFD 44580034 IC50 = 41 nM T83193 CQLO61 44585756 IC50 > 50000 nM T83193 CBT81W 44587581 IC50 = 46 nM T83193 C3OKQ1 44587671 IC50 = 81 nM T83193 CAG32Q 44587705 IC50 = 36 nM T83193 C0J5AB 44587803 IC50 = 890 nM T83193 C0F6IE 44587823 IC50 = 2 nM T83193 CF89OM 44587857 IC50 = 1 nM T83193 CM8YS9 44587934 IC50 = 2 nM T83193 CKRZ26 44755933 EC50 = 4800 nM T83193 C4WS8T 45375957 IC50 = 1000 nM T83193 C80GPZ 45380559 IC50 = 7 nM T83193 CLK8O9 45380748 IC50 = 32 nM T83193 C84ORB 45380848 IC50 = 5 nM T83193 CQDI48 46191427 IC50 = 10 nM T83193 CAT9Z8 46191428 IC50 = 5 nM T83193 CP08ZD 46191499 IC50 = 32 nM T83193 C0ET7O 46191501 IC50 = 5 nM T83193 C4HSX5 46191502 IC50 = 3 nM T83193 CSD13A 46191565 IC50 = 22 nM T83193 CXIC58 46191567 IC50 = 9 nM T83193 C71CGU 46191622 IC50 = 2 nM T83193 CUHT54 46202912 IC50 = 0.83 nM T83193 CBL4C0 46202914 IC50 = 0.21 nM T83193 C6RJ0G 46203233 IC50 = 665 nM T83193 CI6Y5Q 46203537 IC50 = 1.65 nM T83193 C0Q5CE 46203540 IC50 = 308 nM T83193 C97LXB 46203543 IC50 = 6.1 nM T83193 CMB32E 46203864 IC50 = 2.2 nM T83193 CYQG10 46203867 IC50 = 0.2 nM T83193 CCDL39 46203868 IC50 = 79 nM T83193 CS57CK 46204201 IC50 = 460 nM T83193 CGY31W 46225223 EC50 = 19 nM T83193 C3E0RS 46225224 EC50 = 17.4 nM T83193 CA08KQ 46225225 EC50 = 0.65 nM T83193 CECI47 46225226 EC50 = 0.98 nM T83193 C6DM4B 46225227 EC50 = 0.15 nM T83193 CQ31DN 46225228 EC50 = 13.7 nM T83193 C28VIE 46225229 EC50 = 0.0047 nM T83193 CP6Q0D 46847337 IC50 = 3.162 nM T83193 CK5DW1 46847339 IC50 = 3.981 nM T83193 C8XC1H 46862564 IC50 = 794.33 nM T83193 C0SJO4 46865592 IC50 = 79.43 nM T83193 CB70JQ 46865593 IC50 = 19.95 nM T83193 C7ICH3 46865714 IC50 = 5011.87 nM T83193 C7TVB4 46865715 IC50 = 1000 nM T83193 CLM61U 46865716 IC50 = 125.89 nM T83193 CBI2C3 46879825 IC50 = 480 nM T83193 CP4T7X 46879826 IC50 > 10000 nM T83193 CAQ5R4 46879827 IC50 > 10000 nM T83193 C3DZ7T 46879828 IC50 = 3900 nM T83193 CE35RZ 46879878 IC50 > 10000 nM T83193 CVI20B 46879879 IC50 > 10000 nM T83193 C7YUV0 46879880 IC50 > 10000 nM T83193 CQ7BG8 46879881 IC50 = 260 nM T83193 C17SUC 46879882 IC50 > 10000 nM T83193 C3KJD7 46879962 IC50 > 10000 nM T83193 CBK1A2 46879963 IC50 = 4600 nM T83193 C27SQX 46879964 IC50 > 10000 nM T83193 CVTM60 46879965 IC50 > 10000 nM T83193 C2TCG9 46880022 IC50 > 10000 nM T83193 CPH2B0 46880023 IC50 > 10000 nM T83193 C0DPM5 46880024 IC50 > 10000 nM T83193 CM79PR 46880025 IC50 > 10000 nM T83193 CQ8CZ3 46880026 IC50 > 10000 nM T83193 C2PQ6Z 46880080 IC50 > 10000 nM T83193 CA0S7Z 46880081 IC50 > 10000 nM T83193 C3F9BQ 46880082 IC50 > 10000 nM T83193 C6BUT5 46887685 EC50 = 250 nM T83193 CUR8T5 46887699 EC50 = 10 nM T83193 C2DSH4 46887729 EC50 = 7600 nM T83193 C37TUH 46887730 EC50 = 4100 nM T83193 CC4BM2 46887741 EC50 = 2.512 nM T83193 C3DNY1 46887742 EC50 = 6.31 nM T83193 C72YRJ 46887775 EC50 = 5800 nM T83193 CG5US0 46887776 EC50 = 18300 nM T83193 CDOZ92 46887777 EC50 = 7100 nM T83193 CEV8T0 46887779 EC50 = 19200 nM T83193 C3LTH4 46887780 EC50 = 42800 nM T83193 CC5VF3 46887829 EC50 = 53800 nM T83193 CF20RK 46887830 EC50 = 1000 nM T83193 CX13FH 46887831 EC50 = 52200 nM T83193 CR15JT 46887832 EC50 = 230 nM T83193 CA05CQ 46890470 IC50 = 3.5 nM T83193 C4ZQT8 46890471 IC50 = 16 nM T83193 C4S5NR 46890472 IC50 = 14 nM T83193 CW7M5V 46890473 IC50 = 12 nM T83193 CN9Q1V 46890474 IC50 = 125 nM T83193 CF2MP7 46890519 IC50 = 9 nM T83193 C0F1OT 46890520 IC50 = 18 nM T83193 CNZA79 46890521 IC50 = 12 nM T83193 CFE72M 46890522 IC50 = 6 nM T83193 CMY9Q7 46890558 IC50 = 5 nM T83193 CRJZ40 46890559 IC50 = 8 nM T83193 CZ5L4F 46890560 IC50 = 8 nM T83193 CK03BA 46890561 IC50 = 9 nM T83193 CFT95E 46890599 IC50 = 9 nM T83193 CERU86 46890600 IC50 = 6 nM T83193 CGY5O8 46890601 IC50 = 4.3 nM T83193 C3HM1E 46890636 IC50 = 53 nM T83193 C7OG8I 46890637 IC50 = 69 nM T83193 C4DTN2 46911175 IC50 = 0.8 nM T83193 CB71DC 47297796 IC50 > 1000 nM T83193 C4CG8H 49799019 IC50 = 864 nM T83193 C28LCD 49799119 IC50 = 840 nM T83193 C6ZES7 49799164 IC50 = 120 nM T83193 CEOA34 49799165 IC50 = 150 nM T83193 C8ZEV3 49799281 IC50 = 2.1 nM T83193 C5YB3J 49799282 IC50 = 114 nM T83193 CN4IA2 49799319 IC50 = 9 nM T83193 CL1Y3D 49799400 IC50 = 229 nM T83193 C0YX5G 49799401 IC50 = 101 nM T83193 CJ2O8F 49799402 IC50 = 10 nM T83193 C0PYK3 49799487 IC50 = 2 nM T83193 CIB0O2 49799488 IC50 = 1.3 nM T83193 CBI95M 49800487 Ki = 0.4 nM T83193 CJ9QN5 49800488 Ki = 31.7 nM T83193 C4A0WZ 49800489 Ki = 0.3 nM T83193 CG3YU6 49800490 Ki = 0.3 nM T83193 CBX1V7 49804209 Ki = 27.7 nM T83193 CQ73ET 49804501 Ki = 21.6 nM T83193 CPB17S 49804502 Ki = 0.3 nM T83193 C5ROS2 49804506 Ki = 8 nM T83193 CA2N7C 49804795 Ki = 75.2 nM T83193 C72LYO 49804796 Ki = 3.7 nM T83193 CU0R5J 49804798 Ki = 0.5 nM T83193 CXDY96 49863783 IC50 = 5.5 nM T83193 C04BIX 49863784 IC50 = 4.4 nM T83193 CN45OH 49863799 IC50 = 81 nM T83193 CCS97I 49863800 IC50 = 25.4 nM T83193 CTD96F 49863801 IC50 = 48.7 nM T83193 C61LAF 49863802 IC50 = 1450 nM T83193 CDC3E9 49863825 IC50 = 47 nM T83193 CO4CR7 49863826 IC50 = 161 nM T83193 C3YRI7 49863827 IC50 = 134 nM T83193 C79MBF 49863867 IC50 = 13 nM T83193 CG3R4U 49863868 IC50 = 607 nM T83193 CF1K6M 49863889 IC50 = 30 nM T83193 C91ZEV 49863890 IC50 = 15 nM T83193 CXP96N 49863891 IC50 = 27 nM T83193 CLWI96 49870854 IC50 = 11 nM T83193 C90UKY 50899643 IC50 > 10000 nM T83193 COTK61 52918271 IC50 = 1 nM T83193 CRU86C 52918272 IC50 = 2.512 nM T83193 C75OUP 52941151 IC50 = 2520 nM T83193 C9TIQ8 52941239 IC50 = 70 nM T83193 CI3Y7H 52941260 IC50 = 1450 nM T83193 C3CI1S 52941261 IC50 = 4220 nM T83193 CSHU46 52941328 IC50 > 20000 nM T83193 C7VU8Z 52941372 IC50 = 18 nM T83193 CBZ8P2 52941429 IC50 = 18 nM T83193 CR2DV9 52941523 IC50 = 56 nM T83193 CUN29Y 52942454 IC50 = 2780 nM T83193 C76CYL 52942485 IC50 = 1940 nM T83193 C86XKP 52942506 IC50 = 449 nM T83193 CZ7AR6 52942548 IC50 = 462 nM T83193 CEL6A4 52942660 IC50 = 51 nM T83193 CRO4D0 52942705 IC50 = 37 nM T83193 CT80GC 52943679 IC50 = 21 nM T83193 CE8Q9H 52943953 IC50 = 61 nM T83193 CIL01O 52943954 IC50 = 58 nM T83193 C68QPI 52944760 IC50 = 19 nM T83193 C6B5GL 52944788 IC50 = 25 nM T83193 C2ZVJ9 52944807 IC50 = 3350 nM T83193 CSYL32 52944808 IC50 = 52 nM T83193 C5IB7F 52944955 IC50 > 6670 nM T83193 CS05EZ 52944995 IC50 > 10000 nM T83193 C3R4BQ 52945186 IC50 = 230 nM T83193 C1R5QI 52945343 IC50 = 1058 nM T83193 CLZ2Y0 52945367 IC50 = 7.1 nM T83193 C8YG4L 52946049 IC50 = 43 nM T83193 C12TYW 52946120 IC50 = 2460 nM T83193 C9YUE3 52946246 IC50 = 56 nM T83193 CGPN15 52946286 IC50 = 31 nM T83193 C06ZDI 52946380 IC50 = 87 nM T83193 C6QD9F 52947296 IC50 = 2330 nM T83193 CI68FS 52947502 IC50 = 2040 nM T83193 CY25PM 52948674 IC50 = 176 nM T83193 C8CZE7 52949686 IC50 > 20000 nM T83193 C25JSC 52949800 IC50 = 520 nM T83193 CEK05T 52949901 IC50 = 580 nM T83193 CWBH28 52950142 IC50 = 180 nM T83193 CV53UF 53251173 IC50 = 718 nM T83193 CW7I3P 53251330 IC50 = 933 nM T83193 CS95ME 53257733 IC50 = 275000 nM T83193 CSXZ90 53259578 IC50 = 1665000 nM T83193 C8ZJ9V 53316531 IC50 = 3600 nM T83193 CAC4B1 53316588 IC50 = 367 nM T83193 C2M5DZ 53316589 IC50 = 41 nM T83193 CP5IX2 53316590 IC50 = 65 nM T83193 CWK47I 53317334 IC50 = 1380 nM T83193 CTM5Y0 53317849 IC50 = 1756 nM T83193 C68GBO 53318190 IC50 = 404 nM T83193 CIJ02V 53318736 IC50 = 15 nM T83193 CY48EJ 53318883 IC50 = 238 nM T83193 CFG6X9 53318884 IC50 = 197 nM T83193 CWQ51H 53319165 IC50 = 140 nM T83193 CQI0V6 53319221 IC50 = 132 nM T83193 CK7TX5 53319909 IC50 = 3330 nM T83193 C59MGC 53320201 IC50 = 762 nM T83193 C4DC2Y 53320280 IC50 = 115 nM T83193 C4MXJ2 53320373 IC50 > 5000 nM T83193 C9Z7JY 53320484 IC50 > 5000 nM T83193 CXE4K1 53320485 IC50 = 250 nM T83193 CXV68G 53320830 IC50 = 50.12 nM T83193 C8R2ZC 53320831 IC50 = 201 nM T83193 C67QBL 53321243 IC50 = 6 nM T83193 C1RDE5 53321779 IC50 = 498 nM T83193 C12JTH 53321780 IC50 = 2667 nM T83193 C9H5AL 53321781 IC50 = 3700 nM T83193 CT0QG8 53321782 IC50 = 62 nM T83193 CY0TR1 53321783 IC50 = 53 nM T83193 C01CMS 53321847 IC50 = 11 nM T83193 C30HUE 53322166 IC50 = 1252 nM T83193 CRJY79 53322568 IC50 = 853 nM T83193 C6IWP5 53322847 IC50 = 263 nM T83193 CTK26S 53322848 IC50 = 434 nM T83193 C5VGA6 53323109 IC50 = 2000 nM T83193 C9ZU3V 53323161 IC50 = 91 nM T83193 CP6TV2 53323958 IC50 = 1200 nM T83193 CTO91A 53324108 IC50 = 112 nM T83193 CK2D5S 53324459 IC50 = 100 nM T83193 CIP2R6 53324813 IC50 = 410 nM T83193 CIC87Z 53324814 IC50 = 112 nM T83193 CQL80G 53325473 IC50 = 149 nM T83193 C3GJ1P 53325573 IC50 = 377 nM T83193 C0MG2V 53325658 IC50 = 24 nM T83193 C86PXA 53325663 IC50 = 243 nM T83193 CWEF56 53325770 IC50 = 150 nM T83193 CH0SJ3 53325771 IC50 = 185 nM T83193 CHPB78 53325772 IC50 = 3080 nM T83193 CK2GH1 53325956 IC50 = 2790 nM T83193 C2S9QF 53326093 IC50 = 4222 nM T83193 C1ZB5W 53326094 IC50 = 370 nM T83193 CU71RE 53326526 IC50 = 31 nM T83193 CP8YN4 53326730 IC50 = 595 nM T83193 C3OU8Z 53326731 IC50 = 2212 nM T83193 COJ05G 53326732 IC50 = 120 nM T83193 CX4T7C 53326733 IC50 = 48 nM T83193 CQ1CA3 53326824 IC50 = 476 nM T83193 CHCV32 53326862 IC50 = 65 nM T83193 CN9XB7 53341424 IC50 = 2.8 nM T83193 CPD9E0 53341464 IC50 = 10 nM T83193 CCE3M7 53341467 IC50 = 22 nM T83193 C54RAO 53341468 IC50 = 7 nM T83193 CGM0P7 53341469 IC50 = 9.2 nM T83193 C1DEO5 53344884 IC50 = 2.8 nM T83193 C1PVA2 53363480 IC50 = 63.1 nM T83193 CSYK59 54580312 IC50 = 3.162 nM T83193 CDV60E 54580597 IC50 = 5.9 nM T83193 CC6MY2 54581318 IC50 = 25.12 nM T83193 CX4W9B 54581319 IC50 = 25.12 nM T83193 C2Z5MI 54581320 IC50 = 10 nM T83193 CD7T6A 54581321 IC50 = 7.943 nM T83193 C05UWK 54581568 IC50 = 87 nM T83193 CY96DR 54581578 IC50 = 6.1 nM T83193 CHK9X8 54581579 IC50 = 11 nM T83193 CH79VA 54581580 IC50 = 8 nM T83193 CI6DG4 54581581 IC50 = 12 nM T83193 CG5OY0 54581582 IC50 = 4.9 nM T83193 C7URO0 54581583 IC50 = 31 nM T83193 CH45CT 54581605 IC50 = 34 nM T83193 C8RBZ2 54581606 IC50 = 7.5 nM T83193 CRI4D6 54582331 IC50 = 15.85 nM T83193 C2QT8D 54582332 IC50 = 1258.93 nM T83193 CTLX27 54582573 IC50 > 1000 nM T83193 CBY8X7 54583542 IC50 = 14 nM T83193 CC62IP 54583543 IC50 = 1.7 nM T83193 CRXD15 54583544 IC50 > 1000 nM T83193 CU87MQ 54584525 IC50 = 52 nM T83193 CMKC41 54584526 IC50 = 24 nM T83193 COYG60 54584527 IC50 = 13 nM T83193 CM39GI 54584539 IC50 = 260 nM T83193 CL7P1G 54585233 IC50 = 7.943 nM T83193 CLH59Y 54585234 IC50 = 3162.28 nM T83193 CA3D6M 54585460 IC50 = 12 nM T83193 C9G7BI 54585461 IC50 = 7.5 nM T83193 CYSJ96 54585485 IC50 = 32 nM T83193 CS8GO5 54586192 IC50 = 0.1585 nM T83193 CJCT30 54586193 IC50 = 79.43 nM T83193 CVH34C 54586194 IC50 = 5.012 nM T83193 CJK4A9 54586430 IC50 = 28 nM T83193 CZ7UO6 54586431 IC50 > 1000 nM T83193 CB7OU9 54586432 IC50 = 520 nM T83193 CNZ87H 54586433 IC50 = 12 nM T83193 CF7N3X 54586458 IC50 = 44 nM T83193 CLAJ60 54587208 IC50 = 1.259 nM T83193 CHMU16 54587209 IC50 = 12.59 nM T83193 CXCT26 54587210 IC50 = 10 nM T83193 CY7WO8 54587294 IC50 = 1320000 nM T83193 CX6K9Z 54587295 IC50 = 227000 nM T83193 C1R8EC 54587460 IC50 = 5.7 nM T83193 CIY57J 54587479 IC50 = 340 nM T83193 CCO2I3 54587480 IC50 > 1000 nM T83193 C47PDY 54587481 IC50 = 6.8 nM T83193 CUV69N 54669855 EC50 = 4400 nM T83193 C2L3AP 56659764 IC50 = 199.53 nM T83193 CI51JF 56659769 IC50 = 125.89 nM T83193 CKY93J 56659770 IC50 = 158.49 nM T83193 CA13MO 56659771 IC50 = 5011.87 nM T83193 CIE1F0 56659772 IC50 = 316.23 nM T83193 CCBE24 56666677 IC50 = 158.49 nM T83193 C41IRL 56666678 IC50 = 794.33 nM T83193 CX3C4N 56670093 IC50 = 12.59 nM T83193 CCOP96 56670094 IC50 = 1584.89 nM T83193 CK9L6R 56673610 IC50 = 1584.89 nM T83193 COV8T6 56673613 IC50 = 1584.89 nM T83193 C64FYX 56676933 IC50 = 3162.28 nM T83193 CP0V8Y 56676934 IC50 = 1995.26 nM T83193 C57HIX 56676935 IC50 = 63.1 nM T83193 C2V7DN 56683573 IC50 = 3.162 nM T83193 C9WUS8 56683582 IC50 = 39.81 nM T83193 CRG8X7 56896484 IC50 = 314 nM T83193 C7TC2E 56966490 IC50 = 21 nM T83193 CY8NQ9 57334560 EC50 = 110 nM T83193 CDW28C 57334561 EC50 = 500 nM T83193 C34DKP 57334562 IC50 > 10000 nM T83193 C8OTV0 57334563 IC50 > 10000 nM T83193 C96KIT 57334564 IC50 > 50000 nM T83193 CADV61 57390833 IC50 > 100000 nM T83193 CH6D3G 57392653 IC50 > 50000 nM T83193 C6J5IZ 57394365 IC50 > 50000 nM T83193 CWD30P 57394366 IC50 > 10000 nM T83193 C19LBS 57394367 EC50 = 100 nM T83193 CIX28C 57396122 EC50 = 14600 nM T83193 CZ9DL6 57397938 IC50 > 50000 nM T83193 C5MU1H 57397939 EC50 = 14300 nM T83193 CIXP67 57399580 IC50 = 35300 nM T83193 CQ5P7U 57401337 IC50 = 4800 nM T83193 C32NVG 57927125 IC50 = 320 nM T83193 CL10GR 58381102 IC50 = 6 nM T83193 CQV67K 58381208 IC50 = 19 nM T83193 CVY71G 58543815 IC50 > 100000 nM T83193 C0AI3H 58639564 IC50 = 750 nM T83193 C19NCQ 58755739 Ki = 217 nM T83193 CIV21U 58873250 Ki = 2.5 nM T83193 C1QJN0 58873252 Ki = 0.7 nM T83193 C42NXZ 58873256 Ki = 8.7 nM T83193 CL8IE5 58873257 Ki = 142 nM T83193 C9NU8M 58873260 Ki = 4 nM T83193 C5API8 58873263 Ki = 2 nM T83193 C7L2MN 58873266 Ki = 2.1 nM T83193 CQFL38 58873268 Ki = 0.7 nM T83193 C3V9HU 58873274 Ki = 0.3 nM T83193 C37AKC 58873277 Ki = 0.9 nM T83193 CKJ8B5 58873278 Ki = 14.6 nM T83193 CY47JC 58873281 Ki = 1.43 nM T83193 CMC0K2 58873283 Ki = 2.8 nM T83193 C61IXR 58873285 Ki = 2.9 nM T83193 CN4AE9 58873286 Ki = 1.8 nM T83193 C20NLZ 58873288 Ki = 0.7 nM T83193 C6UT7V 58873299 Ki = 1 nM T83193 CCI49K 58873310 Ki = 0.6 nM T83193 CME01F 58873315 Ki = 0.9 nM T83193 C92XOC 58873319 Ki = 0.6 nM T83193 CJUG90 58873320 Ki = 36.1 nM T83193 CFG70L 58873323 Ki = 146 nM T83193 C5WQ2C 58873326 Ki = 2.9 nM T83193 C63DYW 58873336 Ki = 1.2 nM T83193 CBZU20 58873340 Ki = 1.8 nM T83193 CP9Q3K 58873345 Ki = 7.7 nM T83193 CM3RC0 58873352 Ki = 1.3 nM T83193 CL74KX 58873360 Ki = 25.6 nM T83193 C2LF0B 58873361 Ki = 0.4 nM T83193 CFRO67 58873367 Ki = 0.8 nM T83193 CDO01G 58873371 Ki = 0.7 nM T83193 CB9TN3 58873374 Ki = 3.4 nM T83193 CG37QC 58873376 Ki = 13.8 nM T83193 C9NB8V 58873379 Ki = 0.8 nM T83193 CH21ET 58873383 Ki = 0.8 nM T83193 CEV28U 58873386 Ki < 1000 nM T83193 C14SMQ 58873396 Ki = 20.4 nM T83193 CNHX52 58873403 Ki = 3.2 nM T83193 CBK28Y 58873408 Ki = 4.2 nM T83193 C8YAB1 58873411 Ki = 2.3 nM T83193 CWT26G 58873412 Ki = 0.9 nM T83193 CU81DX 58873414 Ki = 0.8 nM T83193 CEN4Y5 58873424 Ki = 5.8 nM T83193 CTS30F 58873427 Ki = 0.3 nM T83193 CFL8W2 58873438 Ki = 15.3 nM T83193 C1FC4S 58873447 Ki = 1.9 nM T83193 CO47KG 58873448 Ki = 1.3 nM T83193 C9M2QG 58873450 Ki = 0.5 nM T83193 CWP8X0 58873451 Ki = 2.5 nM T83193 CRZS39 58873454 Ki = 0.7 nM T83193 C1UV7I 58873461 Ki = 51 nM T83193 C39AWE 58873465 Ki = 8.6 nM T83193 CLT9Z1 58873467 Ki = 2.5 nM T83193 CNET76 58873468 Ki = 2.5 nM T83193 CEN23Q 58873470 Ki = 1.7 nM T83193 C3VFN0 58873473 Ki = 0.7 nM T83193 CR8YK9 58873474 Ki = 2.7 nM T83193 CQ6SE3 58873475 Ki = 0.7 nM T83193 CDZ35O 58873481 Ki = 0.7 nM T83193 CG4NB0 58873497 Ki = 0.8 nM T83193 CCO6D0 58873499 Ki = 1.6 nM T83193 C61YMS 58873504 Ki = 3.2 nM T83193 C6GZT3 58873505 Ki = 0.6 nM T83193 CNKA45 58873506 Ki = 0.8 nM T83193 C6Q7FU 58873513 Ki = 65.7 nM T83193 CWI9U6 58873514 Ki = 1 nM T83193 CV3OU4 58873516 Ki = 0.4 nM T83193 C6IX7N 58873517 Ki = 68.7 nM T83193 C9EPG7 58873529 Ki = 1.9 nM T83193 C02TSG 58873530 Ki = 4.4 nM T83193 CQB4G1 58873536 Ki = 4.4 nM T83193 CDNF58 58873545 Ki = 91 nM T83193 C41BJQ 58873549 Ki = 39.3 nM T83193 CYJ73G 58873550 Ki = 0.001 nM T83193 C9T0NB 58873556 Ki = 0.5 nM T83193 CE4BO0 58873559 Ki = 3 nM T83193 CF7PH2 58873561 Ki = 0.5 nM T83193 CPK9D3 58873562 Ki = 43.7 nM T83193 CTJX93 58873563 Ki = 0.7 nM T83193 CWZ91P 58873575 Ki = 2.4 nM T83193 C1Y6GE 58873578 Ki = 2.2 nM T83193 CLBE06 58873579 Ki = 1 nM T83193 C3JP5E 58873581 Ki = 0.04 nM T83193 CW36FK 58873584 Ki = 1.5 nM T83193 CCI1S0 58873592 Ki = 1.5 nM T83193 C7B0FK 58873593 Ki = 2.5 nM T83193 C5OJI2 58873598 Ki = 8.1 nM T83193 C8D0XQ 58873600 Ki = 12.7 nM T83193 CU9SY5 58873608 Ki = 29.5 nM T83193 CY9FU3 58873610 Ki = 0.3 nM T83193 CG18HW 58873616 Ki = 1.6 nM T83193 C6J9MV 58873625 Ki = 44 nM T83193 CR4XA7 58873626 Ki = 15.8 nM T83193 CCB69W 58873638 Ki = 6.4 nM T83193 CUW53L 58873640 Ki = 1.1 nM T83193 C8C7MW 58873642 Ki = 0.5 nM T83193 C50PHI 58873652 Ki = 0.9 nM T83193 C3MB6C 58873654 Ki = 0.2 nM T83193 CJ72CP 58873655 Ki = 1 nM T83193 CY1HG9 58873658 Ki = 0.9 nM T83193 CI0MC5 58873667 Ki = 0.6 nM T83193 C7ZN6P 58873674 Ki = 16 nM T83193 C8K1XH 58873675 Ki = 4.4 nM T83193 CCXH69 58873678 Ki = 0.9 nM T83193 CDG2Z6 58873681 Ki = 0.9 nM T83193 CJDS23 58873682 Ki = 0.5 nM T83193 C7HR9E 58873691 Ki = 63.3 nM T83193 CQ2VK5 58873692 Ki = 2.7 nM T83193 C82NCS 58873694 Ki = 0.6 nM T83193 CG09QP 58873697 Ki = 9.7 nM T83193 CYD4M9 58873698 Ki = 0.3 nM T83193 CEI47W 58873712 Ki = 1.6 nM T83193 C7JOV4 58873713 Ki = 59.6 nM T83193 C5SNQ0 58873716 Ki = 0.7 nM T83193 C1CN7E 58873717 Ki = 1.6 nM T83193 CSHP94 58873734 Ki = 1.6 nM T83193 CIZN23 58873735 Ki = 3.3 nM T83193 CW4XP9 58873742 Ki = 17.5 nM T83193 CAY81O 58873745 Ki = 0.4 nM T83193 CPK63B 58873748 Ki = 1 nM T83193 C2QH3P 58873756 Ki = 0.7 nM T83193 CKJ40C 58873760 Ki = 0.8 nM T83193 CA13EB 58873763 Ki = 1 nM T83193 C48FVB 58873765 Ki = 0.8 nM T83193 CVC98P 58873771 Ki = 4.8 nM T83193 C91BTK 58873774 Ki = 2.4 nM T83193 CE36NO 58873778 Ki = 2.8 nM T83193 CB98IU 58873784 Ki = 19.3 nM T83193 CC63GV 58873793 Ki = 1.8 nM T83193 C9KNA0 58873796 Ki = 2.1 nM T83193 C3E9RN 58873810 Ki = 1.4 nM T83193 CH64QG 59007833 IC50 = 8 nM T83193 C7YT8V 59007841 IC50 = 22 nM T83193 CQ03ID 59007872 IC50 = 7 nM T83193 C6HDS2 59007884 IC50 = 240 nM T83193 CH6NX5 59007900 IC50 = 7 nM T83193 CSZ0B9 59007942 IC50 = 20 nM T83193 CSL09Q 59007969 IC50 = 5.9 nM T83193 C6J2ML 59008004 IC50 = 190 nM T83193 C0GFE3 59008008 IC50 = 17 nM T83193 CQ76CT 59008012 IC50 = 26 nM T83193 C4I1ME 59008027 IC50 = 13 nM T83193 CAM28G 59008035 IC50 = 40 nM T83193 C72EBR 59008085 IC50 = 4.5 nM T83193 CK79PR 59666268 IC50 = 93 nM T83193 C06TKS 59666298 IC50 = 87 nM T83193 CUN39P 60011733 IC50 = 180 nM T83193 C3VZ4T 60021981 IC50 = 16 nM T83193 C1Z0PC 60022072 IC50 = 56 nM T83193 CUH87T 66644289 Ki = 26.5 nM T83193 CM79IJ 67438722 Ki = 1.1 nM T83193 CTH71U 67438734 Ki = 1.3 nM T83193 C3CHO9 67439038 Ki = 2.3 nM T83193 CRS75Y 67439048 Ki = 100 nM T83193 CM02ZH 67439190 Ki = 3.7 nM T83193 CABX60 67439400 Ki = 14.8 nM T83193 CZ82FC 67439430 Ki = 2.1 nM T83193 C98OFW 67439460 Ki = 0.8 nM T83193 C0MUZ3 67439540 Ki = 3 nM T83193 CO0QB2 67439554 Ki = 1.4 nM T83193 CW4I6M 67439763 Ki = 0.4 nM T83193 CH1NR3 67439768 Ki = 3.4 nM T83193 CY70SV 67439821 Ki < 1000 nM T83193 C4VW6Q 67439823 Ki = 3.8 nM T83193 C32ONF 67439992 Ki = 5.6 nM T83193 CXF3U6 67440023 Ki = 0.7 nM T83193 CY79ZC 67440125 Ki = 0.9 nM T83193 CR2K7S 67440200 Ki = 4.2 nM T83193 CA03ES 67440314 Ki = 14.3 nM T83193 C1Y3QE 67440351 Ki = 2.1 nM T83193 C10CJQ 67440400 Ki = 0.8 nM T83193 CGB6I3 67440621 Ki = 2.2 nM T83193 CW8CK3 67440652 Ki = 1.7 nM T83193 C23SYL 67440783 Ki = 11.5 nM T83193 C1FK5L 67440786 Ki = 0.7 nM T83193 C38NTG 67440919 Ki = 0.4 nM T83193 C6AF8R 67440951 Ki = 5 nM T83193 CW07HE 67441243 Ki = 0.7 nM T83193 CV8T9K 67441528 Ki = 4.1 nM T83193 C63IOB 67441550 Ki = 20.3 nM T83193 CJM17W 67441632 Ki = 0.8 nM T83193 CX5PT0 67441643 Ki = 4 nM T83193 CM92GF 67441906 Ki = 23.9 nM T83193 C49ZSB 68653853 Ki = 22.7 nM T83193 C8DBE3 68718852 Ki = 48.7 nM T83193 C04EJH 68718961 Ki = 31.1 nM T83193 CBSY42 68721207 Ki = 37.6 nM T83193 C5OXZ3 69830044 IC50 > 1000 nM T83193 C4T1EY 69830874 IC50 = 34 nM T83193 C6D9XF 69903675 IC50 = 530 nM T83193 C1I6GO 70681468 IC50 = 230 nM T83193 C3T8HN 70682776 IC50 > 10000 nM T83193 CA0FG3 70682777 IC50 > 10000 nM T83193 C3ZKG0 70683578 IC50 = 45 nM T83193 CE6T5P 70683579 IC50 = 140 nM T83193 CNK40G 70684861 IC50 > 10000 nM T83193 CFDV81 70684862 IC50 = 833 nM T83193 CABQ74 70685686 IC50 = 9.1 nM T83193 CX3L9A 70685687 IC50 > 1000 nM T83193 CL0IK9 70685694 IC50 = 220 nM T83193 C4OFS1 70685695 IC50 = 330 nM T83193 CDJ51K 70687840 IC50 = 18 nM T83193 CFS60E 70687841 IC50 = 710 nM T83193 CN9B7M 70689871 IC50 = 130 nM T83193 C91TQS 70689872 IC50 > 1000 nM T83193 C1MLN9 70689873 IC50 = 460 nM T83193 CKX5D0 70692033 IC50 = 84 nM T83193 C25FYO 70694071 IC50 = 30 nM T83193 CMJ68Z 70694078 IC50 > 1000 nM T83193 CM70ZK 70898363 EC50 = 4897.79 nM T83193 CD6BV5 71237020 Ki = 8.4 nM T83193 C36KJR 71237040 Ki = 0.7 nM T83193 CI5NQ7 71237069 Ki = 7.1 nM T83193 C8M9YX 71237098 Ki = 0.4 nM T83193 C8FH5A 71237137 Ki = 1.8 nM T83193 C7XMW4 71237161 Ki = 8.9 nM T83193 CU52OL 71237192 Ki = 7.2 nM T83193 CI18GC 71237213 Ki = 9.5 nM T83193 CANF28 71237326 Ki = 0.02 nM T83193 CYU80Z 71237407 Ki = 91.6 nM T83193 C5U7AF 71237443 Ki = 48.1 nM T83193 CFHJ43 71237649 Ki = 7.8 nM T83193 CM9P0Z 71449757 IC50 = 1995.26 nM T83193 CSDE19 71449975 Ki = 0.2 nM T83193 CW3J4K 71450023 Ki = 0.3 nM T83193 C1BZR6 71451555 IC50 = 3162.28 nM T83193 C4X5RC 71451556 IC50 = 7943.28 nM T83193 CE45PR 71453396 IC50 = 1258.93 nM T83193 C5SEQ9 71453410 IC50 = 1584.89 nM T83193 CPA80H 71453411 IC50 = 630.96 nM T83193 C39LVF 71453662 Ki = 0.2 nM T83193 CWS2T3 71453663 Ki = 1.4 nM T83193 C27XOP 71455090 IC50 = 5011.87 nM T83193 C4JH2D 71455346 Ki = 11 nM T83193 CL86AH 71455347 Ki = 0.3 nM T83193 C2PL5G 71456898 IC50 = 794.33 nM T83193 CE2M1B 71456899 IC50 = 100 nM T83193 CUEX93 71456916 IC50 = 158.49 nM T83193 C6QVT0 71456917 IC50 = 1000 nM T83193 C3M9KC 71456918 IC50 = 501.19 nM T83193 CCF78E 71456919 IC50 = 3981.07 nM T83193 C6COI9 71457119 Ki = 0.4 nM T83193 CK28DR 71457120 Ki = 3.9 nM T83193 C6VU3T 71457121 Ki = 0.01 nM T83193 CE27CB 71457122 Ki = 7.5 nM T83193 CLDG16 71457160 Ki = 101 nM T83193 CPV3O2 71458753 IC50 = 1000 nM T83193 CM2F1A 71458754 IC50 = 2511.89 nM T83193 CPST04 71458774 IC50 = 1258.93 nM T83193 CZX76C 71458990 Ki = 2.1 nM T83193 C6NK2W 71458991 Ki = 9.8 nM T83193 CPQ4C6 71459032 Ki = 103 nM T83193 C0JB7W 71460583 IC50 = 199.53 nM T83193 CN0TC6 71460584 IC50 = 501.19 nM T83193 C1IKD0 71460788 Ki = 7.1 nM T83193 CKW28L 71460827 Ki = 2.6 nM T83193 CKP7J0 71462280 IC50 = 5011.87 nM T83193 CKO8C9 71462281 IC50 = 501.19 nM T83193 CKYO86 71462283 IC50 = 251.19 nM T83193 CX4OP7 71462545 Ki = 27.2 nM T83193 C4W8XS 71517050 IC50 = 440 nM T83193 C28CKU 71517051 EC50 = 6420 nM T83193 C1RG2N 71517052 EC50 = 11800 nM T83193 C0B2JQ 71517053 EC50 = 5100 nM T83193 C2HK8W 71517054 IC50 = 6400 nM T83193 C7T0YV 71517055 IC50 = 5100 nM T83193 C86OEX 71517056 EC50 = 400 nM T83193 C0ZGK9 71517199 EC50 = 5200 nM T83193 CE2UH4 71517200 EC50 = 7750 nM T83193 CDQ20R 71517201 EC50 = 1890 nM T83193 C5WE8T 71517202 IC50 = 1 nM T83193 CTL61C 71517203 EC50 = 7430 nM T83193 CQTR79 71517204 EC50 = 260 nM T83193 CG7FR3 71517205 EC50 = 2270 nM T83193 C7YH9K 71517356 EC50 = 170 nM T83193 C64RHP 71517357 EC50 = 1200 nM T83193 CX8HQ4 71517358 EC50 = 470 nM T83193 C6S8HN 71517359 EC50 = 5290 nM T83193 CD41WT 71517360 EC50 = 2400 nM T83193 C9O4FN 71517361 IC50 = 4360 nM T83193 CS46UC 71519502 IC50 = 9300 nM T83193 CQ0N9J 71519503 IC50 = 10600 nM T83193 CRK85C 71519504 IC50 = 9600 nM T83193 CM67KB 71528847 EC50 = 18620.87 nM T83193 CICU74 71537378 Ki = 6.77 nM T83193 C9HJ6P 71538504 Ki = 27.6 nM T83193 CT8OU5 71625073 IC50 = 516 nM T83193 CR0NS1 71625201 IC50 = 583 nM T83193 C1YG3H 71625202 IC50 = 33 nM T83193 CF4D3Z 71625203 IC50 = 130 nM T83193 C57ABI 71625204 IC50 = 44 nM T83193 CDG3B5 71625205 IC50 = 2620 nM T83193 CB7R9O 71625206 IC50 = 796 nM T83193 CGH9Q3 71625318 IC50 > 10000 nM T83193 C4F5XT 71625319 IC50 = 110 nM T83193 CQ31CB 71625320 IC50 > 10000 nM T83193 CB6Z0H 71625321 IC50 > 10000 nM T83193 C4F7LM 71625322 IC50 = 107 nM T83193 CXZ51P 71625323 IC50 = 86 nM T83193 CIMO89 71625324 IC50 = 941 nM T83193 CP74ZA 71698456 Ki = 1.3 nM T83193 C4JI2R 71698540 Ki = 0.3 nM T83193 C7NFG8 71698721 Ki = 0.3 nM T83193 CE6BS4 71698888 Ki = 2.6 nM T83193 C34HYQ 71698889 Ki = 0.8 nM T83193 CNE29A 71698890 Ki = 4.9 nM T83193 CXT35W 71698979 Ki = 1 nM T83193 CHRY76 71698980 Ki = 2.6 nM T83193 C0GJ2K 71699635 Ki = 49 nM T83193 CBT0I6 71699636 Ki = 50 nM T83193 CFTM13 71812230 EC50 = 0.99 nM T83193 CW20HQ 71818431 IC50 = 1260 nM T83193 C2L7TX 71818575 IC50 = 6300 nM T83193 C4IP1G 72197089 EC50 = 5900 nM T83193 C9EVP5 72197090 EC50 = 13400 nM T83193 CUAX51 72197091 EC50 = 1500 nM T83193 CWP34U 72197092 EC50 = 2500 nM T83193 CDN29K 72197093 EC50 = 1800 nM T83193 CA9CX5 72197094 EC50 = 250 nM T83193 C5QGC9 72197264 EC50 = 1700 nM T83193 C3C5FR 72197265 EC50 = 11900 nM T83193 CO5Z4D 72197266 IC50 > 100000 nM T83193 CX1J5H 72197267 IC50 > 100000 nM T83193 CXS6H8 72197268 IC50 > 100000 nM T83193 COMJ27 72197269 IC50 > 100000 nM T83193 CC95RF 72197270 IC50 > 100000 nM T83193 CSB3M1 72197441 EC50 = 25000 nM T83193 CC26EQ 72197442 IC50 > 100000 nM T83193 C2HD9F 72197443 EC50 = 32300 nM T83193 CV9DU7 72197444 IC50 > 100000 nM T83193 C9F1KH 72197445 IC50 > 100000 nM T83193 C0KL4H 72197446 EC50 = 22500 nM T83193 CO9TL8 72197447 IC50 > 100000 nM T83193 CHF0K8 72197628 IC50 > 100000 nM T83193 C5UT4O 72197629 IC50 > 100000 nM T83193 CNB9D0 72197630 IC50 > 100000 nM T83193 CT8LB2 72197631 IC50 > 100000 nM T83193 COJ5V6 72197632 IC50 > 100000 nM T83193 CVB7R8 72197633 IC50 > 100000 nM T83193 CVUH81 72197634 IC50 = 91800 nM T83193 C6W2NK 72197807 IC50 > 100000 nM T83193 C9VGP6 72197808 IC50 = 78900 nM T83193 C1Q5DT 72197809 EC50 = 4800 nM T83193 C28SBK 72203625 Ki = 2.3 nM T83193 CFP71H 72203627 Ki = 27.4 nM T83193 C2E3CW 72203628 Ki = 3.3 nM T83193 CH47JO 72203629 Ki = 3 nM T83193 CAG12S 72203823 Ki = 2.9 nM T83193 CT5OI8 72203826 Ki = 48.2 nM T83193 C8NK7U 72203827 Ki = 85 nM T83193 CV8Y0S 72204004 Ki = 1.2 nM T83193 CI1Q5C 72204007 Ki = 0.5 nM T83193 C16QGV 72204008 Ki = 1.9 nM T83193 CSG97M 72204177 Ki = 1 nM T83193 CTS3X9 72204178 Ki = 2.6 nM T83193 C7J0UX 72204179 Ki = 2.3 nM T83193 CM70LI 72204180 Ki = 8.7 nM T83193 CKF0D1 72204181 Ki = 3.2 nM T83193 C65HFT 72204376 Ki = 2.3 nM T83193 C9E6WU 72204377 Ki = 4.9 nM T83193 CZFU81 72204378 Ki = 3.9 nM T83193 CX7H6K 72204379 Ki = 14.6 nM T83193 CT81FE 72204380 Ki = 15 nM T83193 CUL51P 72204570 Ki = 1.9 nM T83193 CD1HF7 72204571 Ki = 0.05 nM T83193 CA1D0M 72204572 Ki = 43.5 nM T83193 C96BEP 72205499 IC50 = 841.6 nM T83193 CXR7L8 72205500 IC50 > 1000 nM T83193 CO57MJ 72205501 IC50 > 1000 nM T83193 C74JTD 72205502 IC50 = 266.3 nM T83193 C8NT4P 72205682 IC50 = 217.8 nM T83193 CDI82J 72205683 IC50 = 412.9 nM T83193 C16WFJ 72206428 Ki = 2.5 nM T83193 C34URG 72206429 Ki = 5.6 nM T83193 C1LP7R 72206430 Ki = 0.7 nM T83193 C2FL5C 72206431 Ki = 4.3 nM T83193 CN48VY 72206432 Ki = 7 nM T83193 CM13IT 72946681 Ki = 6.58 nM T83193 C5LP9N 72946682 Ki = 17.2 nM T83193 C5AQ2V 72946683 Ki = 63 nM T83193 C01WJG 73347328 IC50 = 411 nM T83193 CZ7U6Y 73349242 Ki = 330 nM T83193 COH89Q 73350826 EC50 = 16.5 nM T83193 CZB6C3 73352314 Ki = 212 nM T83193 CBDT72 73353428 Ki = 0.5 nM T83193 CDW07U 73355312 EC50 = 16.3 nM T83193 CW6ZP3 73355313 Ki = 50 nM T83193 CJQL93 73355314 Ki = 33.3 nM T83193 CEN85W 73355315 EC50 = 6.28 nM T83193 CC56EI 73356500 Ki = 1.5 nM T83193 C7QG1L 73356858 Ki = 990 nM T83193 CMF59G 73356859 EC50 = 17.9 nM T83193 CYT0M3 76327921 IC50 = 34 nM T83193 CR62OL 76335194 IC50 = 97 nM T83193 CXJI74 87401321 Ki = 0.9 nM T83193 CD9TA0 89469070 Ki = 199 nM T83193 CW12XC 89717400 IC50 = 70000 nM T83193 CXUH46 90645310 IC50 > 10000 nM T83193 CL0O7Q 90645312 IC50 > 10000 nM T83193 CN61RW 90645447 IC50 > 30000 nM T83193 CISP03 90645459 IC50 = 16700 nM T83193 CM5FN9 90645460 IC50 = 5100 nM T83193 C31TXQ 90645465 IC50 > 30000 nM T83193 C6OF3B 90645468 IC50 = 8100 nM T83193 C0VW1K 90645470 IC50 = 11500 nM T83193 C6SU4X 90665452 IC50 > 3900 nM T83193 CJCR26 90665456 IC50 > 16000 nM T83193 C7Y3DA 92045037 Ki = 1.99 nM T83193 COGJ67 92131136 Ki = 0.03 nM T83193 CF1D6S 101898797 EC50 = 6900 nM T83193 CVZ14O 101922675 EC50 = 2600 nM T83193 CFYD15 110877153 IC50 = 6100 nM T83193 CDNC39 118246723 IC50 > 30000 nM T83193 CEJ1A3 118707572 Ki = 22.7 nM T83193 CYC47B 118707573 Ki = 0.3 nM T83193 CQH41Y 118707574 Ki = 0.4 nM T83193 CK10OS 118707575 Ki = 0.3 nM T83193 CL6VZ5 118707576 Ki = 0.2 nM T83193 CPS2D8 118707577 Ki = 0.3 nM T83193 C9O3FI 118707578 Ki = 0.4 nM T83193 C75WKY 118707579 Ki = 0.3 nM T83193 C3C5NE 118707580 Ki = 1.5 nM T83193 CES2D3 118707581 Ki = 1.5 nM T83193 C7Q8GM 118707582 Ki = 0.8 nM T83193 CP3Y7C 118707583 Ki = 0.3 nM T83193 CQ17KB 118707584 Ki = 0.2 nM T83193 C0CIH4 118707585 Ki = 0.2 nM T83193 C21JUV 118707586 Ki = 0.1 nM T83193 CMAR-86 118707587 Ki = 0.1 nM T83193 CDBN38 118707588 Ki = 0.2 nM T83193 C8CIT6 118707589 Ki = 0.1 nM T83193 CE1B7V 118707590 Ki = 0.2 nM T83193 CQ4ZN2 118707591 Ki = 0.1 nM T83193 C3R5OM 118708168 Ki = 2 nM T83193 CQN36C 118708169 Ki = 5.8 nM T83193 CFX49V 118708170 Ki = 1.4 nM T83193 C9J1NK 118708171 Ki = 1 nM T83193 CO9EJ8 118708172 Ki = 141 nM T83193 CZH02O 118711168 IC50 > 200000 nM T83193 CT91SV 118711722 IC50 = 5 nM T83193 CO60KW 118711975 IC50 = 74 nM T83193 C1P0DX 118711976 IC50 = 97 nM T83193 C1X9PL 118711977 IC50 = 60 nM T83193 C9AGF7 118711978 IC50 = 350 nM T83193 C0A5NJ 118711979 IC50 = 22 nM T83193 CH1Q9Y 118711980 IC50 = 36 nM T83193 CP7N2U 118720705 EC50 = 6000 nM T83193 CFL2M7 118720706 IC50 > 100000 nM T83193 C29ZPL 118720707 IC50 > 100000 nM T83193 CUP7E9 118720708 IC50 > 100000 nM T83193 CPBE74 118720709 IC50 > 100000 nM T83193 C10QZR 118720710 EC50 = 8000 nM T83193 C4C6IY 118720711 EC50 = 1100 nM T83193 CC3JI2 118720712 EC50 = 16200 nM T83193 CU41SM 118720713 EC50 = 2500 nM T83193 CMHI10 118720714 EC50 = 10700 nM T83193 CP51VQ 118720715 EC50 = 8700 nM T83193 CC2A4O 118720716 IC50 > 100000 nM T83193 CV58RZ 118720717 IC50 > 100000 nM T83193 CAS16Q 118720718 IC50 > 100000 nM T83193 C19AGC 118720719 IC50 > 100000 nM T83193 CDL9U8 118720720 IC50 > 100000 nM T83193 CE7Q3M 118720721 IC50 > 100000 nM T83193 CG8JZ5 118720722 IC50 > 100000 nM T83193 C8XEA1 118720723 IC50 > 100000 nM T83193 CK9SH2 118720724 IC50 > 100000 nM T83193 CFBS82 118720725 EC50 = 430 nM T83193 CB17KL 118720726 IC50 > 100000 nM T83193 C9SD8T 118720727 EC50 = 1700 nM T83193 CI53FJ 118720728 EC50 = 8900 nM T83193 CH9WE1 118720729 EC50 = 6500 nM T83193 C8D9NZ 118720730 EC50 = 7800 nM T83193 C9S7AD 118720731 IC50 > 100000 nM T83193 CUR3X5 118720732 IC50 > 100000 nM T83193 CL0J1A 118720733 IC50 > 100000 nM T83193 CQF2M9 118723540 IC50 = 203000 nM T83193 C8P6NQ 118723541 IC50 = 10000 nM T83193 CCA4I7 118723542 IC50 = 19000 nM T83193 C5B8RU 118723543 IC50 = 48000 nM T83193 C8XMY5 118723544 IC50 = 70000 nM T83193 C8NB1I 118723545 IC50 = 45000 nM T83193 CFH7X4 118723546 IC50 = 8000 nM T83193 CZDF29 118723547 IC50 = 13000 nM T83193 C1PM6B 118723548 IC50 = 6000 nM T83193 CPJL95 118723549 IC50 = 9000 nM T83193 CP3R7M 118730332 Ki = 0.9 nM T83193 C5WG9H 118730333 Ki = 1.1 nM T83193 CN63MX 118730445 Ki = 3 nM T83193 CZTH58 118735927 IC50 > 10000 nM T83193 CEXG34 118735928 IC50 = 4300 nM T83193 CS7P9K 118735929 IC50 > 10000 nM T83193 C38JDV 118737608 Ki = 40.3 nM T83193 C6C9EF 121304827 IC50 > 3000 nM T83193 CAYH20 121364823 EC50 = 5.05 nM T83193 C1XNR3 121513880 IC50 > 10000 nM T83193 CB08PN 122193011 Ki = 3.9 nM T83193 C9NE4L 122193012 Ki = 2 nM T83193 C2S4NZ 122193013 Ki = 0.7 nM T83193 CIG7L0 122193014 Ki = 0.8 nM T83193 CBL0C9 122193015 Ki = 0.5 nM T83193 CZY7I1 122193016 Ki = 0.5 nM T83193 C6RL2A 122193017 Ki = 1.9 nM T83193 COU4P1 122193018 Ki = 2.3 nM T83193 CWS0T6 122193019 Ki = 1.8 nM T83193 C9UC0H 122193020 Ki = 1.4 nM T83193 CL93XU 122193022 Ki = 0.03 nM T83193 C7NEC1 122193023 Ki = 0.5 nM T83193 C2QW9Y 122193024 Ki = 13.9 nM T83193 C67NQR 122193025 Ki = 0.5 nM T83193 CM1V9A 122193026 Ki = 1.1 nM T83193 C9Y3XG 122194129 Ki = 0.9 nM T83193 C85KXR 122194130 Ki = 2.3 nM T83193 C9Q6PD 122194131 Ki = 3.2 nM T83193 CPS08K 122194132 Ki = 0.4 nM T83193 C2FYP9 122194133 Ki = 0.6 nM T83193 CE0H9Q 122194238 Ki = 1.2 nM T83193 CKW14B 122194340 Ki = 0.4 nM T83193 C2XOI4 122194341 Ki = 0.4 nM T83193 CA5HR7 122489394 IC50 > 20000 nM T83193 C74SXU 127025660 EC50 = 3970 nM T83193 C01GNA 127026006 Ki = 2.32 nM T83193 C2N8AP 127026007 Ki = 6 nM T83193 CWFH46 127026247 Ki = 0.76 nM T83193 CZV1H2 127026248 Ki = 0.71 nM T83193 CZ76GR 127026249 Ki = 0.9 nM T83193 C0CT8B 127026250 Ki = 1.65 nM T83193 CZGX18 127026253 Ki = 3.28 nM T83193 C4P3JA 127026320 Ki = 7.3 nM T83193 C6TJE7 127026548 IC50 > 10000 nM T83193 CY5L2R 127026553 EC50 = 320 nM T83193 C96DOK 127026858 IC50 > 10000 nM T83193 C63FIE 127026927 Ki = 1.29 nM T83193 CL2J1U 127026928 Ki = 2.14 nM T83193 C04QRN 127026929 Ki = 1.85 nM T83193 CE8BQ3 127026930 Ki = 1.56 nM T83193 C7QPD9 127027216 IC50 > 10000 nM T83193 C5EZR8 127027217 EC50 = 1530 nM T83193 CYWS67 127027218 EC50 = 1000 nM T83193 C7ST5H 127027220 EC50 = 1460 nM T83193 C32MSO 127027221 IC50 = 34 nM T83193 CP6UK0 127027222 IC50 > 10000 nM T83193 C4RGC5 127027223 IC50 > 10000 nM T83193 C2ESL3 127027524 EC50 = 310 nM T83193 CX8K3W 127027525 EC50 = 1990 nM T83193 C5IJF2 127027526 EC50 = 2250 nM T83193 C29BWY 127027527 EC50 = 370 nM T83193 CVHZ19 127028102 IC50 = 1950 nM T83193 CG5S3H 127028103 IC50 = 41 nM T83193 CBH98Z 127028104 EC50 = 660 nM T83193 CBI86M 127028105 EC50 = 170 nM T83193 CT4EN3 127028474 EC50 = 520 nM T83193 CO6C7E 127028475 IC50 > 10000 nM T83193 CXS10T 127028476 IC50 > 10000 nM T83193 CS1RH4 127028477 IC50 > 10000 nM T83193 C2J4XO 127028758 EC50 = 22 nM T83193 CE2NK5 127028759 EC50 = 20 nM T83193 C4RSM7 127028760 EC50 = 4230 nM T83193 C13LHT 127028800 IC50 > 10000 nM T83193 C7U3MP 127029033 IC50 = 1390 nM T83193 CD2TB1 127029037 IC50 > 10000 nM T83193 CHRE59 127029038 IC50 = 4130 nM T83193 C5BX0A 127029039 IC50 = 8110 nM T83193 CAP7Y6 127029097 Ki = 2.3 nM T83193 C4E8QM 127029371 Ki = 0.54 nM T83193 CS3ER8 127029372 Ki = 100 nM T83193 CB8S2H 127029373 Ki = 27.6 nM T83193 CXI5F8 127029645 Ki = 25 nM T83193 CO2NT6 127029646 Ki = 11.9 nM T83193 C4MYB0 127029647 Ki = 6.19 nM T83193 CI80PT 127029648 Ki = 3.13 nM T83193 C62AWV 127034988 IC50 = 173 nM T83193 CZU6J0 127034993 IC50 = 28 nM T83193 CCJ8G9 127035008 IC50 = 370 nM T83193 C4ORS9 127035153 IC50 = 783 nM T83193 C82YBF 127035453 IC50 = 653 nM T83193 C5MN6C 127035454 IC50 = 549 nM T83193 CB4E5T 127035456 IC50 = 67 nM T83193 CW6H7Q 127035457 IC50 = 75 nM T83193 CPFS58 127035458 IC50 = 125 nM T83193 C07TUH 127035459 IC50 = 136 nM T83193 C9V3CE 127035617 IC50 = 347 nM T83193 CFZ95J 127035618 IC50 = 325 nM T83193 CQ4MH9 127035822 IC50 = 127 nM T83193 C30NVR 127035823 IC50 = 239 nM T83193 CH94SE 127035824 IC50 = 381 nM T83193 CAMI26 127035825 IC50 = 24 nM T83193 C8Q1SD 127036261 IC50 = 591 nM T83193 CHB49J 127036589 IC50 = 359 nM T83193 CR16XZ 127036590 IC50 = 86 nM T83193 CDP78L 127037569 IC50 = 403 nM T83193 C6CXG5 127037570 IC50 = 38 nM T83193 C5YZ1L 127049919 Ki = 18.7 nM T83193 C3ZWT2 127049920 Ki = 28.1 nM T83193 CBU1F8 127049921 Ki = 59 nM T83193 C0ZC8V 127049922 Ki = 490 nM T83193 C2RHZ8 127050730 Ki = 83 nM T83193 C74JPG 127050731 Ki = 210 nM T83193 CJZ7Y8 132569635 IC50 > 10000 nM T83193 CMD64J 132942889 IC50 = 49700 nM T83193 C7Y4FE 132942890 IC50 = 68500 nM T83193 CD8P7C 132942891 IC50 = 53000 nM T83193 C4XK9Z 132942893 IC50 = 68900 nM T83193 CTJF87 134134782 IC50 > 10000 nM T83193 C3TW0A 134374895 IC50 > 30000 nM T83193 CPA8R4 135373178 EC50 = 200 nM T83193 CMX3A6 135373212 EC50 = 320 nM T83193 CB3FD2 135373234 EC50 = 370 nM T83193 CXZ6F7 135373249 IC50 = 930 nM T83193 CC5DJ8 135373260 IC50 = 90 nM T83193 CYHW05 135373273 EC50 = 450 nM T83193 CE0DR3 135373275 EC50 = 40 nM T83193 C28RFL 135373302 EC50 = 410 nM T83193 CU8PR6 135373307 EC50 = 330 nM T83193 C4PH1D 135373311 EC50 = 40 nM T83193 CR7S8O 135373364 EC50 = 90 nM T83193 CL87FA 135373389 EC50 = 170 nM T83193 CLAY04 135373392 EC50 = 140 nM T83193 C4N7MS 135373395 IC50 = 1340 nM T83193 C0R8IK 135433889 IC50 = 13 nM T83193 C0Y7WF 135444669 IC50 = 50 nM T83193 C3O9XM 135465551 IC50 = 14 nM T83193 C67MSV 135474346 IC50 = 31 nM T83193 C4EN0K 135492547 IC50 = 12 nM T83193 C1IV8U 136027059 IC50 = 1343 nM T83193 C7BW3K 136094797 IC50 = 487 nM T83193 C0GIS5 136094798 IC50 = 557 nM T83193 C73EKQ 136094799 IC50 = 40 nM T83193 C63WKI 136094800 IC50 = 133 nM T83193 C4LS1T 136094801 IC50 = 42 nM T83193 CF18ME 136094802 IC50 = 144 nM T83193 CPQ7Y1 136094803 IC50 = 23 nM T83193 CQ9EP5 136094804 IC50 > 1000 nM T83193 CF3KG8 136094805 IC50 = 82 nM T83193 CIS4K7 136094806 IC50 = 201 nM T83193 CA8MI2 136094807 IC50 = 216 nM T83193 C41JRM 136094808 IC50 = 286 nM T83193 C4Z3GW 136094809 IC50 > 1000 nM T83193 CV40RL 136094810 IC50 = 100 nM T83193 CPNF93 136094811 IC50 = 37 nM T83193 CZY5X9 137007154 EC50 = 6900 nM T83193 CHO40Y 137007155 EC50 = 5500 nM T83193 C0NU7J 137007156 EC50 = 37500 nM T83193 CF5IN0 137007157 IC50 > 100000 nM T83193 CX52EQ 137634042 Ki = 6.7 nM T83193 CW35LN 137634053 Ki = 112 nM T83193 CGME50 137634139 Ki = 51.8 nM T83193 C35VLF 137634200 Ki = 1.9 nM T83193 CG6E3D 137634936 Ki = 1.5 nM T83193 C3NYE0 137636166 Ki = 4.1 nM T83193 CJH2V9 137637559 IC50 > 30000 nM T83193 CJS75L 137639554 Ki = 3.4 nM T83193 CZ4SA7 137640006 Ki = 0.7 nM T83193 CFMN82 137642621 Ki = 8.5 nM T83193 CE17JM 137643454 Ki = 17.1 nM T83193 CGT02Z 137644147 Ki = 2.8 nM T83193 CZM60X 137644630 Ki = 6 nM T83193 CXC8H3 137646362 Ki = 4.4 nM T83193 CL97NH 137646641 Ki = 4 nM T83193 C46HTO 137647720 Ki = 5.9 nM T83193 CNB4W7 137648188 Ki = 1 nM T83193 C7T5UR 137649873 Ki = 6 nM T83193 CHB60E 137649975 Ki = 89.2 nM T83193 CR35QL 137649976 Ki = 3.2 nM T83193 CZ4B1S 137650495 Ki = 3.4 nM T83193 C0K7PN 137650773 Ki = 0.3 nM T83193 C6R5OF 137651359 Ki = 9.8 nM T83193 CJ9L0P 137652512 Ki = 3.5 nM T83193 C15RPF 137652934 Ki = 2.5 nM T83193 C9UWO7 137654328 Ki = 3.1 nM T83193 CQ5K4S 137654340 Ki = 0.63 nM T83193 C21JIB 137654381 Ki = 3.8 nM T83193 CC5HF6 137654715 Ki = 0.6 nM T83193 C6GWK3 137656096 Ki = 6.2 nM T83193 CFA87N 137656645 Ki = 7.4 nM T83193 CQO4K3 137656714 Ki = 3.1 nM T83193 CX5BP4 137656937 Ki = 0.8 nM T83193 C6WM9Z 137657008 Ki = 0.3 nM T83193 CK7SZ1 137657211 Ki = 0.1 nM T83193 CRL18A 137658691 Ki = 8.1 nM T83193 C0QTE6 137659796 Ki = 3.8 nM T83193 CW1IL7 137660362 Ki = 0.5 nM T83193 C32YDL 137660439 Ki = 2.9 nM T83193 C2KX3V 137661020 IC50 > 30000 nM T83193 CY46UQ 137661067 Ki = 0.8 nM T83193 C39HPA 137661261 IC50 > 10000 nM T83193 C8FWK9 137662018 Ki = 1.2 nM T83193 CRI14T 137662297 Ki = 36.4 nM T83193 CEK6B1 139300630 IC50 > 10000 nM T83193 CD4OJ3 141507741 IC50 = 12.8 nM T83193 CC7PG9 141507742 IC50 = 76 nM T83193 C2OGN0 141507743 IC50 = 46.8 nM T83193 CGN93F 141507744 IC50 = 12.2 nM T83193 CPBZ17 141507745 IC50 = 39.6 nM T83193 C8ZM7G 141507746 IC50 = 14 nM T83193 C70TDA 141507748 IC50 = 250.3 nM T83193 C6X2BP 141507750 IC50 = 125.2 nM T83193 CZI7O3 141507751 IC50 = 12.3 nM T83193 CG08HC 141507753 IC50 = 16.4 nM T83193 C7M1DR 141507754 IC50 = 80.3 nM T83193 C0FE1B 141507755 IC50 = 45.2 nM T83193 C3OA9W 141507756 IC50 = 10.2 nM T83193 CP3BC5 141507757 IC50 = 36.4 nM T83193 C98MWI 141507758 IC50 = 37 nM T83193 CW9A4T 141507759 IC50 = 22 nM T83193 CU1HB0 141507760 IC50 = 40.7 nM T83193 C3RX5K 141507761 IC50 = 43.5 nM T83193 CQ0K8F 141507762 IC50 = 37.6 nM T83193 C6NA4O 141507763 IC50 = 12.7 nM T83193 CK53FW 141507764 IC50 = 46 nM T83193 CD69ZJ 141507765 IC50 = 136.2 nM T83193 C2C1ND 141507767 IC50 = 47.1 nM T83193 CF6XQ0 141507768 IC50 = 70.3 nM T83193 C9D1QP 141507769 IC50 = 40.5 nM T83193 CJ7I0E 141507770 IC50 = 14 nM T83193 CIC73G 141756420 IC50 = 243 nM T83193 C3VHP9 141756421 IC50 = 385 nM T83193 C19VLF 141756424 IC50 = 495 nM T83193 CD7OE4 141756426 IC50 = 2156 nM T83193 CG4P5R 141756427 IC50 = 1122 nM T83193 CM4IX7 141756430 IC50 = 3489 nM T83193 C81AOD 141756431 IC50 = 1674 nM T83193 C24LJR 141756433 IC50 = 121 nM T83193 C2PZB6 145952645 Ki = 2.3 nM T83193 CJ1WT7 145952872 IC50 = 200 nM T83193 C43IUN 145953312 IC50 = 98 nM T83193 CU71FI 145953315 IC50 = 1800 nM T83193 CO9JR6 145953318 IC50 = 72 nM T83193 CWFX19 145954238 IC50 = 95 nM T83193 C4ZH3R 145954944 IC50 = 510 nM T83193 CQ0T2U 145954951 IC50 = 150 nM T83193 CZX10U 145955162 IC50 = 29 nM T83193 CEFH61 145955415 IC50 = 1300 nM T83193 CX0IJ3 145955646 IC50 = 890 nM T83193 CUT2Z8 145955878 Ki = 3.2 nM T83193 C15VSY 145960411 Ki = 0.7 nM T83193 C5RLE1 145960771 IC50 = 470 nM T83193 C52ALB 145960801 Ki = 0.2 nM T83193 CU8L7X 145960890 IC50 = 150 nM T83193 CG3U1B 145961025 IC50 = 820 nM T83193 CB7L9N 145961796 Ki = 0.3 nM T83193 CDYL02 145961805 Ki = 2.4 nM T83193 C1INS9 145962051 IC50 = 700 nM T83193 CJ9BA4 145962156 IC50 = 580 nM T83193 CSCL29 145962213 IC50 = 140 nM T83193 C0O2DH 145962509 Ki = 1.6 nM T83193 CIHR57 145962782 IC50 = 23 nM T83193 CVH7K8 145962832 IC50 = 150 nM T83193 C5TE0L 145962994 IC50 = 320 nM T83193 CG2DY1 145963166 IC50 = 73 nM T83193 CXCD86 145963177 IC50 = 530 nM T83193 CCUD75 145963228 IC50 = 86 nM T83193 CI34EM 145963457 IC50 = 480 nM T83193 C2T1CI 145965659 Ki = 819 nM T83193 CTMX69 145968194 EC50 = 3690 nM T83193 C1N5FP 145968965 IC50 = 81.9 nM T83193 C8C5OW 145969594 IC50 = 10.6 nM T83193 CQL1I9 145972802 Ki = 0.1 nM T83193 C9ME8W 145974998 Ki = 8 nM T83193 C80UTE 145976266 Ki = 50.2 nM T83193 C0WR3F 145976623 Ki = 5.1 nM T83193 C1ZA4F 145977088 IC50 = 25.7 nM T83193 C6KW1F 145983017 IC50 = 297 nM T83193 C4DPI9 145983348 Ki = 20 nM T83193 C5OL8C 145983461 Ki = 66.5 nM T83193 C40INH 145983507 IC50 > 50000 nM T83193 CS9Z6B 145983717 IC50 = 46 nM T83193 CH9AW8 145983743 IC50 = 25 nM T83193 CYVP70 145983755 IC50 = 352 nM T83193 C2TQK7 145983963 Ki = 7.4 nM T83193 CYGR61 145983976 Ki = 5.3 nM T83193 C79POF 145984006 Ki = 0.1 nM T83193 CJ9X5Q 145984060 IC50 = 684 nM T83193 C6H0QM 145984205 IC50 > 100000 nM T83193 C2AO8L 145984443 IC50 = 20 nM T83193 CO54SW 145984817 Ki = 51.9 nM T83193 CB61OL 145985025 IC50 = 458 nM T83193 CL8WN5 145985126 Ki = 21 nM T83193 C0YQ6D 145985141 Ki = 2.4 nM T83193 CWZ1U5 145985255 Ki = 26.4 nM T83193 CF6DU3 145985290 IC50 = 621 nM T83193 C5WVH1 145985756 IC50 > 100000 nM T83193 CC4Q1B 145985949 EC50 = 4900 nM T83193 C2MAB1 145986122 EC50 = 1800 nM T83193 C6EF2M 145986126 IC50 = 461 nM T83193 C4EFS1 145986233 IC50 = 33 nM T83193 CXJH67 155510378 Ki = 0.67 nM T83193 C93ETV 155511833 IC50 = 89 nM T83193 CXS52I 155512061 IC50 = 204 nM T83193 C3E0TA 155512687 IC50 = 22573 nM T83193 CG6MB4 155513334 IC50 = 232 nM T83193 CX4Z3F 155513383 Ki = 0.95 nM T83193 CI65OP 155513602 Ki = 10.8 nM T83193 CYRX70 155515945 Ki = 12.3 nM T83193 C05DLO 155517206 IC50 = 75 nM T83193 CBHC08 155517653 IC50 = 341 nM T83193 CZS69J 155518412 IC50 = 27071 nM T83193 CZ79SG 155518694 IC50 = 1543 nM T83193 CT93LK 155520217 EC50 = 43.7 nM T83193 CVL45A 155523755 IC50 = 788 nM T83193 CY8XL4 155524179 Ki = 7.33 nM T83193 CS0LP7 155525545 Ki = 62 nM T83193 CSL9T1 155525842 EC50 = 31.3 nM T83193 C3IG2A 155526856 IC50 = 1195 nM T83193 CEJI39 155527289 Ki = 14.1 nM T83193 CA16DV 155528800 IC50 = 112 nM T83193 C3NEY4 155530370 IC50 = 394 nM T83193 C0W2GI 155531907 IC50 = 12572 nM T83193 C7QW0U 155532849 IC50 = 1878 nM T83193 C38MQU 155533274 IC50 = 19416 nM T83193 CG6C1I 155535201 Ki = 0.46 nM T83193 CG27DS 155537117 IC50 = 494 nM T83193 CD34OK 155537741 IC50 = 108 nM T83193 CUX51M 155538186 EC50 = 85.9 nM T83193 C8EQ5U 155538902 IC50 = 81600 nM T83193 C6IJA4 155539728 Ki = 1159 nM T83193 CS79MX 155547713 IC50 = 2531 nM T83193 CL36YR 155548389 Ki = 15.3 nM T83193 CPT0Q4 155553946 IC50 = 4945 nM T83193 CN61OU 155554804 IC50 = 1217 nM T83193 CEY91R 155556936 IC50 = 416 nM T83193 CB3DO5 155556993 Ki = 27.9 nM T83193 CHU9L6 155559739 Ki = 1.67 nM T83193 C8I3RS 155562884 Ki = 16.4 nM T83193 D00AII 5281727 IC50 > 10000 nM T83193 D00AJB 73255 IC50 = 50000 nM T83193 D00HCI 1598 EC50 = 129000 nM T83193 D00RDS 797382 Ki = 24 nM T83193 D00XZZ 4286311 EC50 = 300 nM T83193 D00ZWU 1860395 Ki = 53 nM T83193 D01DIT 5283446 EC50 = 630 nM T83193 D01WDS 44450288 Ki = 156 nM T83193 D02GOH 6604822 EC50 = 26 nM T83193 D03HFM 42617984 EC50 = 23 nM T83193 D03LVL 53464483 IC50 > 25000 nM T83193 D03SCD 44448616 EC50 > 100000 nM T83193 D03SJY 24749270 IC50 = 760 nM T83193 D04AMC 11559610 EC50 = 260 nM T83193 D04ECZ 42617986 EC50 = 13 nM T83193 D04XXE 73489 IC50 = 170000 nM T83193 D05APW 46890602 IC50 = 7 nM T83193 D05NTO 5149140 IC50 = 10 nM T83193 D06CDW 3035862 Ki = 0.12 nM T83193 D06MRN 44450313 Ki = 15 nM T83193 D07BKU 11451659 IC50 = 14 nM T83193 D07LCG 44450366 Ki = 6272 nM T83193 D07MBC 5283454 EC50 = 40 nM T83193 D07YQG 5282105 EC50 = 50 nM T83193 D08KRX 4375060 Ki = 980 nM T83193 D08KYH 44450322 Ki = 70 nM T83193 D08WAW 2796370 Ki = 421 nM T83193 D09AZO 44416783 IC50 = 2585 nM T83193 D09BEW 44450379 Ki = 15000 nM T83193 D09OSN 151253 IC50 > 10000 nM T83193 D09SXM 24768211 IC50 = 73 nM T83193 D09WYF 44450365 EC50 > 5000 nM T83193 D0A9PS 5281969 EC50 = 15.8 nM T83193 D0BB7F 44450355 Ki = 72 nM T83193 D0C3XF 44450381 Ki = 607 nM T83193 D0D0DW 11302766 IC50 = 170 nM T83193 D0D4SO 3904199 Ki = 2080 nM T83193 D0D6MC 1150897 IC50 > 20000 nM T83193 D0D6OH 104895 EC50 = 10 nM T83193 D0D7QH 6449767 EC50 = 0.5012 nM T83193 D0D9MW 4298023 Ki = 60 nM T83193 D0DJ6G 44450356 Ki = 29 nM T83193 D0DL4Y 22020504 IC50 = 51 nM T83193 D0DY4E 11339118 IC50 = 65 nM T83193 D0E2XP 24749267 IC50 = 1820 nM T83193 D0E4FJ 5283381 IC50 = 35 nM T83193 D0F1UD 4589192 IC50 = 9100 nM T83193 D0F4NA 1019468 IC50 = 330 nM T83193 D0FF6S 16038374 IC50 > 10000 nM T83193 D0G2EQ 42617990 EC50 = 47 nM T83193 D0G8BN 2733484 IC50 = 4 nM T83193 D0H6GW 44450346 Ki = 1740 nM T83193 D0H6TX 24768210 IC50 = 749 nM T83193 D0J3VX 10248092 IC50 = 91 nM T83193 D0J7CR 42617983 EC50 = 610 nM T83193 D0K7QP 44591633 EC50 = 19 nM T83193 D0K8MN 44448617 EC50 = 10000 nM T83193 D0L9DR 9951636 IC50 = 49 nM T83193 D0M7NA 25224408 IC50 = 21 nM T83193 D0N2QH 6324614 Ki = 5.87 nM T83193 D0N8EI 44450336 IC50 = 66 nM T83193 D0O9NE 5388063 IC50 > 10000 nM T83193 D0P7VQ 9929425 IC50 = 0.18 nM T83193 D0Q0XV 44591632 EC50 = 180 nM T83193 D0Q2ZO 44450380 Ki = 546 nM T83193 D0Q4GB 637566 IC50 > 100000 nM T83193 D0Q8QH 11638703 EC50 = 400 nM T83193 D0R7QF 42617989 EC50 = 2400 nM T83193 D0R8XX 24749271 IC50 = 740 nM T83193 D0SH1L 10473280 IC50 = 600 nM T83193 D0T3CP 11645841 EC50 = 320 nM T83193 D0T8DR 44450347 IC50 = 150 nM T83193 D0U5LL 2543 EC50 = 6200 nM T83193 D0W3VM 11472986 IC50 = 11 nM T83193 D0W6TX 7927254 IC50 = 280 nM T83193 D0W7XR 11507802 IC50 > 100000 nM T83193 D0WK3N 44450300 Ki = 23 nM T83193 D0X7AM 10295883 EC50 = 8 nM T83193 D0X8XU 24768203 IC50 = 2580 nM T83193 D0XO2G 680502 IC50 = 150 nM T83193 D0Y1MM 11710300 EC50 = 250 nM T83193 D0Y7QY 5885566 IC50 = 330 nM T83193 D0Y9EU 3884807 Ki = 3520 nM T83193 D0Z1NH 42617985 EC50 = 150 nM T35465 D01KKQ 135400182 IC50 = 6.3 nM T35465 D02LWU 148121 IC50 = 0.69 nM T35465 D0SV8E 126941 IC50 = 12 nM T35465 D0Y4GO 135410875 IC50 = 138 nM T35465 CO2DY5 11247965 Ki = 280 nM T35465 C8Q6ZT 11248313 Ki = 1100 nM T35465 CM4Z7A 44421498 Ki = 530 nM T35465 CPM3L5 67092576 IC50 = 54 nM T35465 CTK64O 67092918 IC50 > 1000 nM T35465 C87FBU 135455948 IC50 = 59.8 nM T35465 CF8D5O 135465664 IC50 > 1000 nM T35465 C9Z4ES 135567027 IC50 > 1000 nM T35465 C14LTO 135567028 IC50 > 1000 nM T35465 CF39AI 135567029 IC50 = 101 nM T35465 C8N7ES 135567030 IC50 > 1000 nM T35465 CFE2O7 135567034 IC50 = 197 nM T35465 C8KVP5 135567035 IC50 = 189 nM T35465 CSQX75 135567163 IC50 = 510 nM T35465 CQF8P5 135800109 IC50 = 304 nM T35465 CL8VN5 136015502 IC50 = 116 nM T35465 CR7UY3 136044173 IC50 > 1000 nM T35465 C0Q5FI 136044174 IC50 > 1000 nM T35465 CGX68Y 136044175 IC50 > 1000 nM T35465 C4C9FN 136044176 IC50 > 1000 nM T35465 CIPD35 136044177 IC50 > 1000 nM T35465 CZG8W6 136059167 IC50 = 634 nM T35465 CZC95Y 136059168 IC50 > 1000 nM T35465 CG2ID9 136059169 IC50 > 1000 nM T35465 C2WH0S 136059178 IC50 > 1000 nM T35465 CB3GL7 136059191 IC50 > 1000 nM T35465 CCHG08 136059192 IC50 > 1000 nM T35465 C4Q1HF 136180345 IC50 = 38.3 nM T35465 CDC83K 136180346 IC50 = 243.2 nM T35465 CF7NW6 136180347 IC50 > 1000 nM T35465 CPH52E 137150145 IC50 > 1000 nM T35465 C9XD1M 137150146 IC50 > 1000 nM T35465 CHDB56 137150160 IC50 > 1000 nM T35465 CMKA64 155517044 IC50 = 808 nM T35465 CCL3Y9 155518053 IC50 = 66.2 nM T35465 C91SVN 155519837 IC50 = 641 nM T35465 CO7BN6 155524531 IC50 > 1000 nM T35465 CT70WU 155530762 IC50 = 213 nM T35465 CX42MF 155532591 IC50 > 1000 nM T35465 CFU98A 155534971 IC50 = 642 nM T35465 C4K2RU 155538415 IC50 > 1000 nM T35465 C27BIX 155539477 IC50 > 1000 nM T35465 C6S7OC 155548982 IC50 = 62 nM T35465 CX3K8F 155549935 IC50 > 1000 nM T35465 CJ0MK5 155554671 IC50 = 468 nM T35465 CYQ0I9 155555353 IC50 = 783 nM T46828 D01AZG 5073 Ki = 1000 nM T46828 D01FFA 72301 Ki = 305 nM T46828 D01ZII 2726 Ki = 172 nM T46828 D03KQF 4011 Ki = 429 nM T46828 D05XGO 11154555 Ki = 7900 nM T46828 D0B0CP 667467 Ki = 9 nM T46828 D0CQ0Z 33630 Ki = 125 nM T46828 D0D1AL 3559 Ki = 38 nM T46828 D0G8NN 119570 Ki > 10000 nM T46828 D0H3HM 60795 Ki > 1000 nM T46828 D0H7KF 5002 Ki > 1000 nM T46828 D0KS6W 7077 Ki = 414 nM T46828 D0P5SA 3372 Ki = 21 nM T46828 D0R9EQ 5095 Ki = 41211 nM T46828 D0T7OW 681 EC50 = 2 nM T46828 D0V4QS 135398745 Ki = 90 nM T46828 D0Y5UG 2160 Ki = 170 nM T46828 D0Z1RV 135398737 Ki = 198 nM T46828 D0N1HW 5311200 Ki > 10000 nM T46828 D0Y6HW 107930 Ki = 2 nM T46828 D07YLK 4350931 Ki = 7.5 nM T46828 D02DHU 1218 EC50 = 1.4 nM T46828 D06DZI 107780 Ki > 10000 nM T46828 D0M7LV 5761 Ki = 340 nM T46828 D0OU7P 1242 Ki = 124 nM T46828 D0OW1R 9802631 Ki > 10000 nM T46828 C5H9CN 9287 Ki > 10000 nM T46828 C9E6DA 21171 Ki = 62.1 nM T46828 C17TDE 23269 Ki > 10000 nM T46828 CBJ5R0 65340 Ki = 1023.29 nM T46828 C6CU1T 70515 Ki > 10000 nM T46828 CPZ5N6 98358 Ki > 10000 nM T46828 C1ND9W 161665 Ki = 242 nM T46828 C09JTU 199798 Ki > 10000 nM T46828 C5RC4G 231915 Ki > 10000 nM T46828 CYO3R2 300430 Ki > 10000 nM T46828 CG2JX9 440229 Ki = 9.5 nM T46828 CQZ4A9 636934 Ki > 10000 nM T46828 CD7P8Y 763194 Ki > 10000 nM T46828 C6QLR0 763343 Ki > 10000 nM T46828 CLR75J 763625 Ki = 2059 nM T46828 C5SXQ1 763774 Ki = 3523 nM T46828 C9IK2J 792265 Ki > 10000 nM T46828 C13TYL 792460 Ki > 10000 nM T46828 C4AY9X 792584 Ki > 10000 nM T46828 CVTP62 1811569 Ki > 10000 nM T46828 C4TB0I 3036864 Ki = 0.48 nM T46828 C64CZV 3038494 Ki = 1223 nM T46828 C82GMT 3246443 Ki = 15.1 nM T46828 C0U6EW 3504099 Ki > 10000 nM T46828 C6AQP8 5249952 Ki = 112 nM T46828 C9AZ2I 5249956 Ki = 3.09 nM T46828 CO3N1A 6440792 IC50 = 0.15 nM T46828 C8QM7B 6852376 Ki = 245.47 nM T46828 C7EZ2L 9859861 Ki > 10000 nM T46828 C5WYN4 9865858 Ki > 1000 nM T46828 C3DB5H 9884781 Ki > 3000 nM T46828 C6WY0D 9891901 Ki > 10000 nM T46828 CYWQ50 9906447 Ki > 10000 nM T46828 CP41ZO 9992499 Ki = 337 nM T46828 CZKG96 10200496 Ki = 16.6 nM T46828 C6J2ZL 10402378 Ki = 1.8 nM T46828 C2B0IU 10421236 Ki > 10000 nM T46828 COV85C 10472143 Ki = 400 nM T46828 CPI5M7 10476504 Ki = 3700 nM T46828 CEF2O6 10478367 Ki > 10000 nM T46828 CRI50E 10885636 IC50 = 988 nM T46828 CNP08C 10891703 Ki > 10000 nM T46828 CX65PW 10907460 IC50 = 1450 nM T46828 CQ62UO 10918307 IC50 = 3660 nM T46828 CNB39C 10947658 Ki = 1000 nM T46828 CJC9K4 11005810 IC50 = 513 nM T46828 CFJG64 11059058 IC50 = 4890 nM T46828 CG41BK 11071079 IC50 = 1550 nM T46828 C7DE0U 11113605 IC50 = 3020 nM T46828 CVE8T3 11121216 Ki = 590 nM T46828 CUD5A0 11134444 Ki = 1756 nM T46828 C3NEM0 11151473 Ki = 9600 nM T46828 C5JS0L 11151831 Ki = 12000 nM T46828 C4FTD9 11153135 Ki = 83000 nM T46828 C3Q9UG 11154178 Ki = 13 nM T46828 CN06GJ 11186895 Ki = 313 nM T46828 C8FKS6 11198948 Ki = 5900 nM T46828 C7MY8T 11210215 Ki = 19000 nM T46828 CVT04Q 11221294 Ki = 9000 nM T46828 C8RJ3D 11223303 Ki = 7.1 nM T46828 CKX06B 11235174 Ki = 5.8 nM T46828 C1Z4WT 11246806 Ki = 26000 nM T46828 CM72YX 11269330 Ki = 10.5 nM T46828 CUJ2R7 11280344 Ki > 10000 nM T46828 CF1C7M 11290269 Ki = 8300 nM T46828 CLZ9S1 11290688 Ki = 7200 nM T46828 CG95WP 11301268 Ki = 71000 nM T46828 C45WLN 11324023 Ki = 16000 nM T46828 CXWH42 11358377 Ki = 1812 nM T46828 CY24NV 11374299 Ki = 5.9 nM T46828 CP3Y2E 11394805 Ki = 32000 nM T46828 C6O9QT 11405458 Ki = 7700 nM T46828 CT32OJ 11406143 Ki = 620 nM T46828 C95WMQ 11415988 Ki = 7600 nM T46828 C1OUA4 11416809 Ki = 20000 nM T46828 CKQ6F7 11416811 Ki = 16000 nM T46828 CF2V6Y 11438636 Ki = 16000 nM T46828 CBN91Q 11439190 Ki = 89 nM T46828 C6A0EF 11439436 Ki = 15000 nM T46828 CD4UV2 11441173 Ki = 54000 nM T46828 C37RKD 11449266 Ki = 19000 nM T46828 CS34HD 11449669 Ki = 19000 nM T46828 C4YT6M 11450584 Ki = 9600 nM T46828 C86CJB 11451022 Ki > 10000 nM T46828 CB3P6S 11452916 Ki = 5.6 nM T46828 CK39HZ 11486421 Ki = 3.3 nM T46828 CTU1Z7 11488247 Ki = 1.2 nM T46828 CKV25P 11493746 Ki = 1.2 nM T46828 CR1HO4 11500181 Ki > 10000 nM T46828 CAU1R7 11500677 Ki = 1050 nM T46828 CQ5IN9 11522339 Ki = 10.4 nM T46828 CC6U7R 11522476 Ki = 2610 nM T46828 C75YUO 11536580 Ki > 10000 nM T46828 C2JT3I 11536995 Ki = 54.6 nM T46828 CN3W7S 11543350 Ki > 10000 nM T46828 C8X0EM 11543992 Ki > 10000 nM T46828 C0AN1Y 11551474 Ki > 10000 nM T46828 C7S2WZ 11558055 Ki = 1.5 nM T46828 CM8G3B 11558247 Ki = 39.5 nM T46828 C4HDA6 11558324 Ki > 10000 nM T46828 C8GK0U 11566745 Ki = 2.32 nM T46828 CP8MF4 11573628 Ki = 3.1 nM T46828 C1TBC8 11573806 Ki = 11.5 nM T46828 C5Q8XM 11595240 Ki = 0.98 nM T46828 CFC25K 11601627 Ki > 10000 nM T46828 C9D7OU 11616435 Ki > 10000 nM T46828 CN1P4I 11623343 Ki = 0.54 nM T46828 CIZ53S 11623652 Ki > 10000 nM T46828 CS4CR7 11631304 Ki = 893 nM T46828 CMX4K8 11633643 Ki > 10000 nM T46828 CG1C3D 11637457 Ki = 15 nM T46828 CLZQ65 11644613 Ki > 10000 nM T46828 CHIW07 11652965 Ki > 10000 nM T46828 CO69ZI 11666419 Ki > 10000 nM T46828 CE34SW 11668495 Ki > 10000 nM T46828 CI26JH 11674133 Ki > 10000 nM T46828 CSQ4B1 11681599 Ki = 0.053 nM T46828 C06BEA 11694873 Ki > 10000 nM T46828 CRO95K 11695189 Ki > 10000 nM T46828 CN1SJ8 11696598 Ki > 10000 nM T46828 CDLW51 11701907 Ki > 10000 nM T46828 C0G1WQ 11709500 Ki > 10000 nM T46828 CI3N1K 11716230 Ki > 10000 nM T46828 CZ6NB8 11716438 Ki = 37.5 nM T46828 CZ7SJ2 11716449 Ki = 14.7 nM T46828 C9FTL5 11718008 Ki = 59 nM T46828 C7PVL8 11730467 IC50 = 1860 nM T46828 CA4W1P 11739113 Ki = 13000 nM T46828 CV91RG 11778580 Ki = 0.57 nM T46828 CH5T6L 11818686 Ki = 16000 nM T46828 CXLW54 11948707 Ki > 10000 nM T46828 C8JQL7 11957735 IC50 > 10000 nM T46828 C7NV4W 12068769 Ki > 10000 nM T46828 C4NWX9 12301195 Ki > 10000 nM T46828 CCG14E 13091356 Ki > 10000 nM T46828 CC74ND 13373172 Ki = 41.1 nM T46828 CI5Y6N 13611248 Ki > 10000 nM T46828 C7VAI1 15011772 Ki > 10000 nM T46828 C0G2EO 16007117 Ki = 73 nM T46828 CWMC70 16090814 Ki = 0.61 nM T46828 CP09RQ 16090821 Ki = 71.6 nM T46828 CZ2IS9 16660294 Ki > 10000 nM T46828 CGX0D5 16665071 Ki = 0.23 nM T46828 C7KP5T 17755866 Ki = 17 nM T46828 CX7VE8 17755867 Ki = 9.8 nM T46828 CUW8S4 17755868 Ki = 95 nM T46828 C3KA6Z 17755875 Ki > 10000 nM T46828 C4N1LS 17755991 Ki = 314 nM T46828 C6BE2Y 17755992 Ki > 10000 nM T46828 C10UQJ 17755999 Ki = 55 nM T46828 C6WO9X 17756101 Ki = 4.6 nM T46828 CI9RW0 17756102 Ki = 53 nM T46828 CDPT42 17756110 Ki > 10000 nM T46828 C0XG9B 17756212 Ki = 75 nM T46828 C6JQ1K 17756213 Ki = 69 nM T46828 CG5NT4 20035572 Ki > 10000 nM T46828 C94BPG 21460314 Ki > 10000 nM T46828 C3T5HF 21509921 Ki = 575.44 nM T46828 CFN81Q 21527771 Ki = 103 nM T46828 CH59WN 21533446 Ki = 113 nM T46828 CL5A2V 21554999 Ki > 10000 nM T46828 C61LUT 21555004 Ki > 10000 nM T46828 CAH39X 21564536 Ki > 10000 nM T46828 CO4C6M 23653115 Ki > 10000 nM T46828 CBUJ02 23653176 Ki = 202 nM T46828 CDH38J 23992579 Ki > 10000 nM T46828 C3W6DQ 25096873 IC50 > 1000 nM T46828 CX04LB 25142456 Ki = 7 nM T46828 C78HME 25212275 Ki = 265 nM T46828 CE6Z9I 25212276 Ki = 265 nM T46828 C4MRQ0 27842480 IC50 > 50000 nM T46828 CK3QD2 42625354 Ki = 80 nM T46828 CLH7Y0 42626289 Ki = 75.4 nM T46828 C5VTZ6 42626293 Ki = 313 nM T46828 CVG6X1 44209472 Ki = 2392 nM T46828 CD5AB7 44209480 Ki = 1451 nM T46828 C98VPM 44275670 Ki = 5.62 nM T46828 C1B4QL 44403095 Ki > 10000 nM T46828 C1YL7Z 44403098 Ki > 10000 nM T46828 CFV98A 44403101 Ki > 10000 nM T46828 C6OY9S 44403102 Ki > 10000 nM T46828 CH4SX6 44403105 Ki > 10000 nM T46828 C12FIH 44403106 Ki > 10000 nM T46828 C4LKC1 44404394 Ki > 10000 nM T46828 C3EJ4G 44404396 Ki > 10000 nM T46828 CO2H3T 44406799 Ki > 10000 nM T46828 CI70SN 44406862 Ki > 10000 nM T46828 C0R6PK 44406863 Ki > 10000 nM T46828 CDA3R0 44406866 Ki > 10000 nM T46828 CU52FA 44406881 Ki > 10000 nM T46828 CZ24HP 44408818 Ki = 7.2 nM T46828 C93NGH 44414299 Ki = 411 nM T46828 CU2FG6 44415569 Ki = 38 nM T46828 CDU6Y5 44415593 Ki = 105 nM T46828 CH0BY5 44415672 Ki = 7 nM T46828 CK59CO 44415689 Ki = 53 nM T46828 C7AZ5D 44415690 Ki = 31 nM T46828 CEVY54 44415704 Ki = 58 nM T46828 CY0QJ2 44427970 Ki = 510 nM T46828 C2AZ6B 44436300 Ki = 386 nM T46828 C30QMX 44436301 Ki = 230 nM T46828 C9AJ0D 44436302 Ki = 1132 nM T46828 C3NVL0 44436303 Ki > 10000 nM T46828 CREM27 44436304 Ki = 507 nM T46828 C53XYK 44436305 Ki = 1703 nM T46828 C2LF9K 44436306 Ki = 190 nM T46828 C9H8ST 44436307 Ki = 33.6 nM T46828 C7IBE2 44436308 Ki = 80.8 nM T46828 CBI86V 44439942 Ki = 3.6 nM T46828 C3HMI2 44439943 Ki = 0.39 nM T46828 C63PQV 44439944 Ki = 31.5 nM T46828 C2P4CI 44439945 Ki = 5.4 nM T46828 C12XGE 44456400 Ki > 10000 nM T46828 C16HEZ 44555445 Ki > 10000 nM T46828 CRCH48 44582675 Ki = 7419 nM T46828 CEJ4R8 44582676 Ki = 7398 nM T46828 CP6ZA9 44591012 Ki > 1000 nM T46828 CU37BO 44591098 Ki > 1000 nM T46828 CU48CL 44591099 Ki = 273 nM T46828 C7H9SE 44591134 Ki = 153 nM T46828 C6RLW0 44591135 Ki = 297 nM T46828 CYJ7P8 45379368 Ki > 10000 nM T46828 CU2CA7 45379369 Ki = 2.5 nM T46828 CT3K8Y 45379370 Ki = 10.3 nM T46828 CT3A1Q 45379373 Ki > 10000 nM T46828 C8TRE1 45379377 Ki = 1525 nM T46828 CML67J 45379515 Ki > 10000 nM T46828 CSV1P2 46216855 Ki = 1.9 nM T46828 CY7NM6 46227242 Ki > 10000 nM T46828 CR9S7B 46227243 Ki > 10000 nM T46828 C9A8FV 46227273 Ki > 10000 nM T46828 CL3KU2 46227284 Ki = 1508 nM T46828 CS4O6A 46227317 Ki = 185 nM T46828 CE1L6H 46227320 Ki > 10000 nM T46828 CSQ9D5 46227325 Ki = 1810 nM T46828 CDI10H 46231541 Ki = 3.9 nM T46828 C9KI4E 46231646 Ki = 8.3 nM T46828 C8SFI5 46231768 Ki = 7 nM T46828 C1EW4S 46231782 Ki = 3.7 nM T46828 C6JM5T 46231784 Ki = 1.4 nM T46828 CD6IC3 46231845 Ki = 7.5 nM T46828 C38WBY 46231846 Ki = 3.3 nM T46828 C0A7GW 46231847 Ki = 7.4 nM T46828 CVT82S 46231848 Ki = 26.9 nM T46828 C9W1US 46231924 Ki = 22 nM T46828 CL7WX9 46231925 Ki = 10 nM T46828 CVG26Z 46231926 Ki = 2.5 nM T46828 CKJ09A 46231927 Ki = 2.1 nM T46828 C2BX8U 46231994 Ki = 3.4 nM T46828 C7FD2G 46231995 Ki = 4.7 nM T46828 CYV52A 46232066 Ki = 6.2 nM T46828 C03LTM 46869265 Ki = 2800 nM T46828 C2LZJ0 49783209 Ki = 972 nM T46828 C57SMG 49783415 Ki > 10000 nM T46828 C0TG6I 49783419 Ki > 10000 nM T46828 C2RY0J 50878551 Ki > 10000 nM T46828 C1W6TV 50898777 Ki > 10000 nM T46828 CXMZ73 50898778 Ki > 10000 nM T46828 CE4KP1 51050257 Ki > 10000 nM T46828 C19ZKQ 52946556 Ki = 1.5 nM T46828 CPA2G4 52951481 Ki > 10000 nM T46828 CYP0I3 52951482 Ki > 10000 nM T46828 CSX14G 53321869 Ki > 10000 nM T46828 C32YWL 53324045 Ki = 121 nM T46828 CRQF15 53325242 Ki = 529 nM T46828 CLZ09P 53359025 Ki > 10000 nM T46828 CG24AT 53381002 Ki > 10000 nM T46828 CQ3AR0 56589560 Ki = 4.4 nM T46828 C4XGR3 56589561 Ki = 91.4 nM T46828 C9PHZ3 56594402 Ki = 657 nM T46828 C82IVX 56594533 Ki = 389 nM T46828 CT4J5C 56594534 Ki = 11.4 nM T46828 CH37LU 56663451 Ki > 10000 nM T46828 C1TC7Q 56963799 Ki > 10000 nM T46828 CV08WY 57391216 Ki = 1370 nM T46828 C07PMA 57391307 Ki = 2684 nM T46828 CWT20M 57393083 Ki = 3812 nM T46828 C3GW6L 57398351 Ki = 867 nM T46828 CZX05B 57401706 Ki = 3223 nM T46828 CYN38R 57401819 Ki = 1758 nM T46828 CO0XD2 57401820 Ki = 2808 nM T46828 CX0B5M 57403525 Ki = 414 nM T46828 C5RUP6 60167166 Ki > 10000 nM T46828 C34GMW 69599704 Ki > 10000 nM T46828 C9VZ8J 71450550 Ki > 10000 nM T46828 CE92DF 71528209 Ki = 5210 nM T46828 C31THM 72164180 Ki = 1743 nM T46828 C56VLM 72164181 Ki > 10000 nM T46828 CD8A9K 72164182 Ki = 1534 nM T46828 C4C0BH 72164183 Ki > 10000 nM T46828 CQU81Y 72164299 Ki > 10000 nM T46828 CF0H7K 72164300 Ki > 10000 nM T46828 C7WM5U 72164301 Ki > 10000 nM T46828 C4HO2U 72164302 Ki > 10000 nM T46828 CC65OA 73213195 Ki > 10000 nM T46828 CW83DK 73213196 Ki > 10000 nM T46828 CW8A0Y 73349359 Ki > 10000 nM T46828 CH2B4Y 73350932 Ki > 10000 nM T46828 C1NJ0R 73353884 Ki > 10000 nM T46828 CA4CP6 73355416 Ki > 10000 nM T46828 C81CIL 73355418 Ki > 10000 nM T46828 CN5V0R 73355421 Ki > 10000 nM T46828 C2E7QW 75201901 Ki = 4.8 nM T46828 CJG57Z 75202022 EC50 = 4.4 nM T46828 C8IDL3 75306277 Ki = 199.53 nM T46828 CZFW19 76314267 Ki = 17378.01 nM T46828 CIB40D 76321554 Ki = 3548.13 nM T46828 CS9F1X 76321556 Ki = 3467.37 nM T46828 C97LOB 76325150 Ki = 4570.88 nM T46828 CCR29U 76325152 Ki = 2454.71 nM T46828 CLP59V 76325156 Ki = 2754.23 nM T46828 C17YTI 76328715 Ki = 9700 nM T46828 CSW58A 76336021 Ki = 19498.45 nM T46828 C28RIZ 76518514 Ki > 10000 nM T46828 C8EWX5 85658088 Ki = 1613 nM T46828 CJ9K3T 86290953 EC50 > 10000 nM T46828 CM6X4U 86764103 EC50 = 12 nM T46828 C80SXV 90644057 Ki > 10000 nM T46828 CY8TP0 90644061 Ki = 2511.89 nM T46828 CKV24H 90644062 Ki = 1995.26 nM T46828 CW2ZC4 90644063 Ki = 3162.28 nM T46828 CLG60I 90644064 Ki > 10000 nM T46828 CKLN72 90644065 Ki > 10000 nM T46828 CDPE48 90644071 Ki = 1522 nM T46828 C35WTP 122177641 Ki = 24000 nM T46828 C8OS7B 122177642 Ki = 48000 nM T46828 CV2AT4 122177644 Ki = 21000 nM T46828 CB16GY 122177645 Ki = 700 nM T46828 CH9SX5 122180956 Ki = 3800 nM T46828 CCV9D5 122181326 Ki = 2800 nM T46828 C5D1NC 122181329 Ki = 2900 nM T46828 C05RGV 122181330 Ki = 7000 nM T46828 C3XGN0 122181333 Ki = 11000 nM T46828 CVJ3R4 122191605 Ki = 3600 nM T46828 C2J4ZX 122191607 Ki = 1300 nM T46828 C71KZQ 122205437 Ki = 3 nM T46828 C30ZRC 122205438 Ki = 1.9 nM T46828 CM57GR 126720252 Ki = 1070 nM T46828 C09YOS 127027905 Ki > 10000 nM T46828 CE9MN1 127028185 Ki > 10000 nM T46828 C9SC6E 127028505 Ki > 10000 nM T46828 CO53TS 127035828 Ki > 1000 nM T46828 CY7LP9 127035829 Ki > 1000 nM T46828 CR29BS 127035830 Ki > 1000 nM T46828 C50GOC 130442480 Ki = 82 nM T46828 CM04RF 130442572 Ki = 47 nM T46828 CAVB41 132584404 Ki > 10000 nM T46828 CBU81N 134149168 Ki > 10000 nM T46828 C5KE3N 135986088 Ki = 921 nM T46828 CN8BJ2 137632607 Ki > 20000 nM T46828 C3R2LO 137632761 Ki > 20000 nM T46828 C3PF9Z 137633454 Ki > 20000 nM T46828 CN1I7A 137634153 Ki > 20000 nM T46828 C6FRJ5 137634397 Ki > 15000 nM T46828 CPHI76 137635364 Ki = 3800 nM T46828 C8ZFQ6 137635685 Ki = 5800 nM T46828 CZ36LE 137636066 Ki = 15000 nM T46828 CAL1W4 137636298 Ki > 20000 nM T46828 CQ20FO 137636498 Ki = 3400 nM T46828 CZU6N5 137636581 Ki > 50000 nM T46828 C0YDQ5 137637428 Ki > 20000 nM T46828 C1HX3Z 137639304 Ki > 20000 nM T46828 CC16HE 137640152 Ki > 20000 nM T46828 CZP68A 137640189 Ki = 4200 nM T46828 C8IO0R 137640836 Ki > 20000 nM T46828 C6PT7L 137642033 Ki > 20000 nM T46828 CAC6W0 137643122 Ki > 20000 nM T46828 C71XIQ 137643132 Ki = 5700 nM T46828 C4PV8U 137645196 Ki > 20000 nM T46828 CNH95X 137645574 Ki = 9300 nM T46828 C3TP2G 137645830 Ki = 19000 nM T46828 CPI68E 137646281 Ki = 3016 nM T46828 CYH5U9 137647533 Ki > 20000 nM T46828 CW4T6D 137651322 Ki = 7700 nM T46828 CX30HQ 137653096 Ki > 20000 nM T46828 C4C6EV 137653986 Ki > 20000 nM T46828 COTX19 137654511 Ki > 20000 nM T46828 CF5Y2A 137654675 Ki = 13000 nM T46828 CLI4D8 137655029 Ki > 20000 nM T46828 CJAZ13 137655556 Ki > 20000 nM T46828 C6CA5H 137655594 Ki > 20000 nM T46828 CD16SQ 137655795 Ki = 16000 nM T46828 CE0Y7P 137657322 Ki > 20000 nM T46828 CRT86S 137657427 Ki > 20000 nM T46828 CH76FP 137657951 Ki > 20000 nM T46828 CP6US4 137660046 Ki = 16000 nM T46828 C5V4DQ 137660707 Ki > 20000 nM T46828 CL58XS 145967572 Ki = 286 nM T46828 C58WSL 145967904 Ki = 640 nM T46828 CB1FD8 145968810 Ki = 312 nM T46828 C48XNG 145969667 Ki = 101 nM T46828 CNZY06 145969934 Ki = 438 nM T46828 C61MSO 145970938 Ki = 605 nM T46828 C87MSW 145980271 Ki = 744 nM T46828 CNJH37 145986752 Ki = 623 nM T46828 CO4LK7 145988180 Ki = 143 nM T46828 CUGO10 145988693 Ki = 437 nM T46828 CC2G1V 146025727 Ki = 27 nM T46828 C6P3SR 153287553 Ki > 10000 nM T46828 CV9G7Z 153287572 Ki > 10000 nM T46828 CO85KL 153287574 Ki > 10000 nM T46828 CQ83KZ 155512662 Ki > 10000 nM T46828 CHXY56 155513802 Ki > 5000 nM T46828 CL5G9Q 155513837 Ki > 5000 nM T46828 CH34RK 155514798 Ki = 1204 nM T46828 CUE5J3 155515907 Ki > 5000 nM T46828 CUM2N4 155515982 Ki = 340 nM T46828 CV12SD 155516041 Ki > 5000 nM T46828 CJ98ZK 155516236 Ki > 5000 nM T46828 C9ZAW0 155517266 Ki = 5799 nM T46828 CUSA24 155519891 Ki > 10000 nM T46828 C8IYD1 155520455 Ki = 1995.3 nM T46828 C5DSE0 155520996 Ki = 1584.9 nM T46828 CV7IG5 155522663 Ki > 5000 nM T46828 C2H3JL 155523073 Ki = 1721 nM T46828 CQA76T 155523112 Ki > 5000 nM T46828 C3E9DJ 155523127 Ki > 5000 nM T46828 CVQ68Y 155523770 Ki = 2203 nM T46828 COH1Q5 155524191 Ki > 5000 nM T46828 CW7NT8 155524423 Ki = 3500 nM T46828 CQX27T 155525357 Ki > 5000 nM T46828 CW65KS 155525705 Ki = 1104 nM T46828 CKZ35G 155532475 Ki > 5000 nM T46828 C4LOR5 155532477 Ki > 5000 nM T46828 CQ12KS 155533996 Ki = 6109 nM T46828 C8AX5N 155534186 Ki = 7703 nM T46828 CHP2Z9 155535866 Ki = 9290 nM T46828 CB79ZW 155536080 Ki > 10000 nM T46828 CVFD68 155537516 Ki > 5000 nM T46828 C13CSU 155537907 Ki > 5000 nM T46828 C3DIY2 155539246 Ki = 926.1 nM T46828 CPV48W 155539557 Ki = 1000 nM T46828 CVK2M9 155543189 Ki = 8670 nM T46828 C4ANI0 155543691 Ki > 5000 nM T46828 C08FTE 155544239 Ki > 5000 nM T46828 C7MCZ0 155546478 Ki = 789 nM T46828 CN6I4P 155550431 Ki = 10532 nM T46828 C6N9PG 155550640 Ki > 5000 nM T46828 CG7NR9 155550756 Ki = 5580 nM T46828 C82QWR 155551173 Ki = 571 nM T46828 CX8JA1 155552185 Ki = 1000 nM T46828 CG70XQ 155552591 Ki = 8844 nM T46828 CB4F8Y 155552676 Ki = 1079.8 nM T46828 CD5LC6 155554006 Ki = 4227 nM T46828 C36SYJ 155558844 Ki > 5000 nM T46828 C7OZM6 155561446 Ki > 5000 nM T46828 CALB48 155561861 Ki > 10000 nM T46828 C2Z0HB 155562353 Ki = 2154.4 nM T46828 C0UN4V 155564747 Ki > 5000 nM T46828 CMH8I1 155565768 Ki = 8191 nM T46828 CK20WA 155566662 Ki > 5000 nM T46828 C6DPR8 155566974 Ki > 5000 nM T46828 C95RAP 155567835 Ki = 588.8 nM T46828 C5A6YM 155567869 Ki = 4018 nM T46828 CV24CW 155568676 Ki > 5000 nM T46828 C73ERT 155568786 Ki = 1847.9 nM T46828 C42JKO 155569198 Ki > 5000 nM T46828 C3N9VU 10251906 Ki > 500 nM T46828 CP9TR0 10324985 Ki > 10000 nM T46828 D00NQV 5041 Ki > 10000 nM T46828 D00SDJ 11237664 IC50 > 10000 nM T46828 D01ENR 2993172 Ki = 366 nM T46828 D04TWX 9794475 IC50 > 10000 nM T46828 D07RYR 44396235 Ki = 951 nM T46828 D09RPR 16737207 Ki > 10000 nM T46828 D0E1RX 11335419 Ki = 113 nM T46828 D0E3AL 56597938 Ki = 1100 nM T46828 D0F0IA 11301655 Ki > 8000 nM T46828 D0FF6S 16038374 IC50 > 10000 nM T46828 D0HH3R 11698643 Ki = 939 nM T46828 D0J1HP 10378389 Ki = 3715.35 nM T46828 D0L5MW 181743 Ki = 2397 nM T46828 D0L7OM 6917970 Ki = 4.4 nM T46828 D0L8PI 5018 IC50 = 0.56 nM T46828 D0LV7U 10667433 Ki = 330 nM T46828 D0R8UU 44396220 Ki = 43 nM T95913 D09XZB 123631 IC50 > 50000 nM T95913 D0B3HD 2519 IC50 = 1000000 nM T95913 D0E3SH 6918837 IC50 > 10000 nM T95913 D0E6XR 3062316 IC50 > 50000 nM T95913 D0F8RA 2153 IC50 = 800000 nM T95913 D0J5VR 11625818 IC50 = 60 nM T95913 D0K8KX 5280343 IC50 = 13790 nM T95913 D0R0MW 5329102 IC50 = 13000 nM T95913 D0RU0O 50905713 IC50 = 2 nM T95913 D0S5LD 135565596 IC50 = 0.7 nM T95913 D0W5HK 216239 IC50 > 50000 nM T95913 D01PGR 16123056 IC50 = 9 nM T95913 D01QSO 16654980 IC50 = 256 nM T95913 D03BHZ 52913813 IC50 = 675 nM T95913 D03EZE 25167777 IC50 = 0.61 nM T95913 D03FOP 68947304 IC50 = 850 nM T95913 D03IJO 11618268 IC50 = 3000 nM T95913 D03KAC 1893730 IC50 = 23 nM T95913 D03XAQ 49784945 IC50 = 36 nM T95913 D06GUA 49784002 IC50 = 6309.57 nM T95913 D07EHV 44814409 IC50 > 9100 nM T95913 D07HPJ 11476171 IC50 = 3200 nM T95913 D08QGT 17755052 Ki = 1.4 nM T95913 D0C3ZR 10427712 IC50 = 83 nM T95913 D0D8JB 44516953 IC50 = 6 nM T95913 D0E6UZ 54575456 IC50 = 311 nM T95913 D0I3LO 91933883 IC50 = 0.29 nM T95913 D0LG7X 86291103 IC50 = 33 nM T95913 D0O1LD 11647372 IC50 = 5 nM T95913 D0O6VZ 25254071 IC50 = 14 nM T95913 D0O8SJ 72950888 IC50 > 120 nM T95913 D0TU7B 58507717 IC50 = 708 nM T95913 D0U3DP 46912230 IC50 = 25 nM T95913 D0UP1Z 51001932 Ki = 0.97 nM T95913 D0VG0D 11977753 IC50 = 6 nM T95913 D0W7HE 56649450 IC50 = 250 nM T95913 D0X7IN 11978790 IC50 = 38 nM T95913 D0XD4I 118502708 IC50 = 1100 nM T95913 D0Y2NS 70798655 IC50 = 1900 nM T95913 D03BNU 59604787 IC50 > 5000 nM T95913 D0C9JZ 58111426 IC50 = 2297 nM T95913 D05HIJ 135565159 IC50 = 10000 nM T95913 D09SFV 3973 IC50 = 950 nM T95913 D0D0QA 44137675 IC50 = 1090 nM T95913 D0P1JI 312145 IC50 = 19 nM T95913 CX74ND 40237 IC50 = 380000 nM T95913 CEL9D8 79972 IC50 = 1498000 nM T95913 CNW59X 95001 IC50 = 53000 nM T95913 C3FRX9 131989 IC50 > 83300 nM T95913 C1MOD6 165595 IC50 = 2415000 nM T95913 CW1B9X 226105 IC50 = 1570000 nM T95913 C6KL2D 235602 IC50 = 992000 nM T95913 C4I2PT 244740 IC50 = 134000 nM T95913 C6ET7X 247414 IC50 = 5184000 nM T95913 CGC10Q 249363 IC50 = 2700 nM T95913 CQ7B2K 252311 IC50 = 187000 nM T95913 CBY29G 260801 IC50 = 105000 nM T95913 C1Y0JB 263480 IC50 = 324000 nM T95913 CTU12Q 267310 IC50 > 1600000 nM T95913 CJ43OR 270557 IC50 = 6074000 nM T95913 CV8DJ6 274101 IC50 = 241000 nM T95913 C2M5YF 275065 IC50 = 1460000 nM T95913 CEW10F 291727 IC50 = 234000 nM T95913 C1M3IR 309591 IC50 = 9157000 nM T95913 C6E4HJ 347279 IC50 = 5876000 nM T95913 CFW2K4 414938 IC50 = 2437000 nM T95913 COE1I6 426449 IC50 = 7333000 nM T95913 CK30NI 520127 IC50 > 1670000 nM T95913 CY3D4G 617191 IC50 = 16670 nM T95913 CS5O7B 622000 IC50 > 40000 nM T95913 CXC3V1 622262 IC50 = 1660 nM T95913 CU73NO 736009 IC50 > 83300 nM T95913 CZN6S9 743974 IC50 > 25118.86 nM T95913 C3P4OY 1093514 IC50 = 27950 nM T95913 C3KPX5 1270546 IC50 = 920 nM T95913 CP0QU1 1355022 IC50 = 3600 nM T95913 CWOQ49 1627922 IC50 = 10000 nM T95913 CAN89K 2762479 IC50 > 100000 nM T95913 C56YDF 2762944 IC50 > 100000 nM T95913 C8E3HY 2796894 IC50 = 5495.41 nM T95913 C09VKD 2816900 IC50 > 83300 nM T95913 C4RH3J 3106064 IC50 = 25000 nM T95913 C4PQ7T 3128427 IC50 = 5 nM T95913 C1O4KS 4416330 IC50 = 4200 nM T95913 CIN5F7 4904109 IC50 <= 10000 nM T95913 C1YJM9 4912089 IC50 > 83300 nM T95913 CE74CV 5059890 IC50 = 100000 nM T95913 C9N4MH 5765281 IC50 = 20000 nM T95913 CKX0F4 5806797 IC50 = 4300 nM T95913 C8CL1W 6053578 IC50 = 612000 nM T95913 CS26IV 6089668 IC50 = 3800 nM T95913 CGF7R0 6196488 IC50 = 20000 nM T95913 C2OZ0W 6484194 IC50 > 83300 nM T95913 CK2IR4 6852165 IC50 = 2030 nM T95913 CX18LU 9342140 IC50 = 1200 nM T95913 CE1Y8A 9815659 IC50 = 37000 nM T95913 CJ79RC 9879653 IC50 = 31 nM T95913 CC2Q6T 9925404 IC50 = 217800 nM T95913 CLT13A 10088066 IC50 = 4000 nM T95913 C9HWF6 10114067 IC50 = 3630 nM T95913 C57FPB 10115147 IC50 = 5450 nM T95913 CZ15SC 10125446 IC50 = 380 nM T95913 C02SQE 10141582 IC50 = 7620 nM T95913 CZ4D7S 10181657 IC50 = 145200 nM T95913 CF6Y2U 10202973 IC50 = 1820 nM T95913 C1RDW9 10203280 IC50 = 6170 nM T95913 CC82QV 10204538 IC50 = 137900 nM T95913 CO5VP9 10296641 IC50 = 2540 nM T95913 C7SFI1 10296883 IC50 > 10000 nM T95913 C7ZG0A 10296917 IC50 = 13070 nM T95913 CW7Q0R 10315189 IC50 = 18150 nM T95913 C32NQS 10357196 IC50 = 21 nM T95913 CC67FL 10383101 IC50 = 46000 nM T95913 C2VG4L 10455817 IC50 = 2.42 nM T95913 CAZT53 10475366 IC50 = 570 nM T95913 CL8YE3 11230964 IC50 = 6400 nM T95913 C8Y6IM 11234514 IC50 = 67 nM T95913 CK65NF 11418892 Ki = 3060 nM T95913 CL3Z4O 11419728 Ki = 20 nM T95913 CYBD21 11428504 IC50 = 100000 nM T95913 CHJ30L 11492951 IC50 = 250 nM T95913 C5E2PO 11500850 IC50 = 13500 nM T95913 CV8J3I 11514586 IC50 = 950 nM T95913 CTXF73 11515474 IC50 = 80 nM T95913 C0O4SQ 11522078 IC50 = 30 nM T95913 C7HMO6 11526786 IC50 = 8000 nM T95913 C15XPT 11529859 IC50 = 43 nM T95913 C5KV8L 11530037 IC50 = 530 nM T95913 CGK17J 11536358 IC50 = 110 nM T95913 C38YWS 11541283 IC50 = 6 nM T95913 C1VA4C 11543481 IC50 = 970 nM T95913 C4T8IQ 11550986 IC50 = 290 nM T95913 C63TOQ 11551198 IC50 = 39 nM T95913 CN2MS6 11562853 IC50 = 1258.93 nM T95913 C9JF1G 11565677 IC50 = 2600 nM T95913 CPXS32 11566902 IC50 = 56 nM T95913 CMVQ43 11576772 IC50 = 20 nM T95913 CUZP58 11580302 IC50 = 1000 nM T95913 CX92QM 11581007 IC50 = 29 nM T95913 CEHZ82 11599141 IC50 = 794.33 nM T95913 C6U0BN 11601532 IC50 > 10000 nM T95913 CL5F3Z 11601890 IC50 = 20 nM T95913 C58QVA 11601930 IC50 = 37 nM T95913 C1ZPM5 11630874 IC50 = 30 nM T95913 CLK3Y4 11638999 IC50 = 1000 nM T95913 CU2CK3 11644621 IC50 = 840 nM T95913 CQIX52 11645168 IC50 = 260 nM T95913 C08DUS 11645350 IC50 = 20000 nM T95913 CC64OJ 11652531 IC50 = 40 nM T95913 CP04JC 11666231 IC50 = 2.3 nM T95913 CK8T1S 11666950 IC50 = 29 nM T95913 CU0E8O 11690457 Ki > 4000 nM T95913 CLQ02O 11695207 IC50 = 20000 nM T95913 C3BT1M 11702204 IC50 = 20 nM T95913 CB0AP2 11705863 Ki > 4000 nM T95913 CY8C9P 11751126 IC50 = 382 nM T95913 CAJV97 11955205 IC50 = 21 nM T95913 CBR6D5 11955693 IC50 = 1860 nM T95913 C68SND 11955695 IC50 = 1873 nM T95913 C60DBM 11998444 IC50 > 40000 nM T95913 C5FTB0 11998445 IC50 = 6259 nM T95913 C68WMR 11998447 IC50 = 19790 nM T95913 CYL24B 11998448 IC50 = 16700 nM T95913 CNPI54 11998563 IC50 = 3506 nM T95913 C6AK0Y 11998564 IC50 = 1674 nM T95913 CMVA72 11998565 IC50 = 386 nM T95913 CJ3YP8 11998685 IC50 = 2076 nM T95913 CV8PB5 11998690 IC50 = 829 nM T95913 CB9T1H 11998803 IC50 = 49 nM T95913 C59SKD 11999032 IC50 = 31 nM T95913 CT58GS 12171624 IC50 = 333.96 nM T95913 C0RF3U 14501859 IC50 = 773000 nM T95913 CY7A0T 14638904 IC50 = 10900 nM T95913 CW2XK6 16050925 IC50 = 390 nM T95913 CW5FD8 16081736 IC50 = 16060 nM T95913 C2IF3P 16678352 IC50 > 30000 nM T95913 C3IO1C 16679060 IC50 > 30000 nM T95913 CV9US5 16736978 IC50 > 30000 nM T95913 C72THB 16739368 IC50 = 250 nM T95913 CF6JS9 16757570 IC50 = 54 nM T95913 CB19TH 16757576 IC50 = 10000 nM T95913 C9BJ7Q 16757577 IC50 = 660 nM T95913 C9DM4T 16757578 IC50 = 230 nM T95913 C1NZC7 16757579 IC50 > 10000 nM T95913 CY0S6G 17751063 IC50 = 127 nM T95913 CTP62W 17755300 IC50 = 9000 nM T95913 CQYN41 17755304 IC50 = 3000 nM T95913 C1G7NC 17755392 IC50 = 32700 nM T95913 CI87FV 17755495 IC50 = 17000 nM T95913 CI71OB 17755611 IC50 = 51000 nM T95913 C9W7ID 17755613 IC50 = 12.6 nM T95913 C1SN9M 17756679 IC50 >= 100000 nM T95913 CJAM62 18452190 IC50 = 11.2 nM T95913 C48LCH 18452193 IC50 = 4.27 nM T95913 CVH65S 18452195 IC50 = 2.66 nM T95913 C31KPH 18452198 IC50 = 4.76 nM T95913 CPSJ85 18452200 IC50 = 6.57 nM T95913 C14WMZ 18452237 IC50 = 2.59 nM T95913 CQ89PW 18452323 IC50 = 7.16 nM T95913 C1O3CJ 18452350 IC50 = 23 nM T95913 CXFA80 18452409 IC50 = 37.3 nM T95913 C9Q0EK 18452424 IC50 = 27.5 nM T95913 C5WV4J 18452430 IC50 = 103.4 nM T95913 CVDL81 22036885 IC50 = 6 nM T95913 C61ZGT 22135435 IC50 > 50118.72 nM T95913 CC5QS1 22263527 IC50 = 10890 nM T95913 CP05ZB 22346757 IC50 = 50000 nM T95913 C1F2TM 23582995 IC50 = 1500 nM T95913 CEYL29 23585510 Ki = 88 nM T95913 CR08WX 23586742 IC50 = 7260 nM T95913 CBL37C 23642173 Ki = 1020 nM T95913 C8J1SI 23642272 IC50 = 5285 nM T95913 C59CTR 23652981 IC50 = 97 nM T95913 C29SFI 24768579 IC50 = 829 nM T95913 C3M1OC 24802861 IC50 = 230 nM T95913 CP4G9Z 24855584 Ki = 120 nM T95913 CJV7D9 24855887 IC50 = 50 nM T95913 CM9C0R 24866805 IC50 = 6800 nM T95913 CB79YC 24905143 IC50 = 1500 nM T95913 C2DC9J 24905144 IC50 = 570 nM T95913 CN6V8Z 24905145 IC50 = 100 nM T95913 CSB7P5 24905148 IC50 = 2400 nM T95913 CGSF21 24905149 IC50 = 200 nM T95913 CVDG02 24905150 IC50 = 1800 nM T95913 CWH6C5 24905152 IC50 = 43 nM T95913 C0HE2Q 24905153 IC50 = 72 nM T95913 C7QSC9 24905154 IC50 = 990 nM T95913 CO9D0K 24905155 IC50 = 860 nM T95913 C5W9UR 24905157 IC50 = 1400 nM T95913 CC1DA3 24905158 IC50 = 940 nM T95913 COW79F 24905159 IC50 = 680 nM T95913 CFPA53 24905160 IC50 = 2400 nM T95913 C2O0JX 24905161 IC50 = 7200 nM T95913 CA72BE 24905162 IC50 = 900 nM T95913 CQN6X9 24905163 IC50 = 2400 nM T95913 CD4O1F 24905165 IC50 = 5900 nM T95913 CKL48T 24905166 IC50 = 10000 nM T95913 C76VYL 24905167 IC50 = 1300 nM T95913 C7K5PU 24905168 IC50 = 1400 nM T95913 CZ57ID 24905169 IC50 = 1100 nM T95913 C2DHX9 24905170 IC50 = 2300 nM T95913 CSB96E 24905171 IC50 = 100000 nM T95913 CWZ0R2 24905172 IC50 = 1100 nM T95913 CY3B6M 24905175 IC50 = 551 nM T95913 CW7UA3 24905176 IC50 = 821 nM T95913 CW1V0H 24905177 IC50 = 100000 nM T95913 CO6Y0L 24905178 IC50 = 100000 nM T95913 C60NQW 24905179 IC50 = 8020 nM T95913 C4MO8B 24905180 IC50 = 1470 nM T95913 COJI47 24905181 IC50 = 1210 nM T95913 CS0B2C 24905182 IC50 = 640 nM T95913 C1H4BT 24905183 IC50 = 271 nM T95913 C4WHK9 24905184 IC50 = 4250 nM T95913 C7Q4MZ 24905185 IC50 = 799 nM T95913 CS4IP1 24905186 IC50 = 270 nM T95913 C69QWO 24905187 IC50 = 873 nM T95913 C85ANB 24905188 IC50 = 123 nM T95913 CNHD75 24905189 IC50 = 87 nM T95913 C9JUO2 24905190 IC50 = 1022 nM T95913 CPR03K 24905191 IC50 = 1140 nM T95913 CTAG19 24905193 IC50 = 435 nM T95913 C7VJM5 24905194 IC50 = 430 nM T95913 CEP1L3 24905195 IC50 = 347 nM T95913 CP68ZD 24905196 IC50 = 239 nM T95913 C8Z0RJ 24905197 IC50 = 381 nM T95913 CN9RT0 24905198 IC50 = 100000 nM T95913 CHI78P 24905200 IC50 = 2700 nM T95913 CO6PE8 24905201 IC50 = 2000 nM T95913 CZ63HS 24905202 IC50 = 1300 nM T95913 C2X0FC 24905203 IC50 = 330 nM T95913 C0WCE3 24905204 IC50 = 220 nM T95913 CNK50B 24905205 IC50 = 590 nM T95913 C12DPB 24905206 IC50 = 830 nM T95913 C8N0RH 24905207 IC50 = 2700 nM T95913 CYA5G2 24905208 IC50 = 461 nM T95913 CDV2B4 24905209 IC50 = 1800 nM T95913 CEFK68 24905210 IC50 = 640 nM T95913 CUFP12 24905211 IC50 = 1300 nM T95913 C0JG8L 24905212 IC50 = 1500 nM T95913 CP47MK 24905213 IC50 = 15000 nM T95913 CB61QC 24905214 IC50 = 3000 nM T95913 CQ13ZI 24905215 IC50 = 100000 nM T95913 C6VI8F 24905216 IC50 = 184 nM T95913 CXNH25 24905217 IC50 = 167 nM T95913 C2PN9S 24905218 IC50 = 95 nM T95913 C9O2AL 24905219 IC50 = 228 nM T95913 CIT7U8 24905220 IC50 = 100000 nM T95913 CMD26S 24905221 IC50 = 627 nM T95913 C4R8WC 24905222 IC50 = 31000 nM T95913 C47SHA 24905223 IC50 = 113 nM T95913 C1DY2R 24905224 IC50 = 90 nM T95913 CS0XF9 24905225 IC50 = 100000 nM T95913 CG5VX2 24905226 IC50 = 100000 nM T95913 C57QEO 24905227 IC50 = 100000 nM T95913 C7CG5E 24905228 IC50 = 586 nM T95913 CHP5D1 24905229 IC50 = 3000 nM T95913 CXP09S 24905230 IC50 = 60 nM T95913 CY7XG1 24905231 IC50 = 7300 nM T95913 C7JFQ2 24905232 IC50 = 242 nM T95913 C2JM1P 24905233 IC50 = 6900 nM T95913 CC3BF0 24905234 IC50 = 3000 nM T95913 CE57FI 24905235 IC50 = 4200 nM T95913 CUP20O 24905236 IC50 = 3500 nM T95913 CLC6Q2 24905237 IC50 = 6200 nM T95913 C9M1GI 24905238 IC50 = 2400 nM T95913 CVD72F 24905239 IC50 = 101 nM T95913 CK38IZ 24905240 IC50 = 28 nM T95913 CO2V5E 24905241 IC50 = 22000 nM T95913 CZBA19 24905244 IC50 = 625 nM T95913 CQ8OI1 24905246 IC50 = 100000 nM T95913 C5URC6 24905247 IC50 = 4000 nM T95913 C03SVO 24905250 IC50 = 7700 nM T95913 CIF2J5 24905251 IC50 = 700 nM T95913 CPTE58 24905252 IC50 = 1450 nM T95913 CX1JB8 24905253 IC50 = 2400 nM T95913 COZ3H7 24905254 IC50 = 25000 nM T95913 CDT1H9 24905255 IC50 = 15000 nM T95913 C54QKA 24905256 IC50 = 1700 nM T95913 CRU3P2 24905257 IC50 = 100000 nM T95913 C9U0JA 24905259 IC50 = 11000 nM T95913 CO4YS7 24905260 IC50 = 9600 nM T95913 CEG0B5 24905261 IC50 = 100000 nM T95913 C9VE5F 24905262 IC50 = 100000 nM T95913 C3I4HK 24905264 IC50 = 20000 nM T95913 C0VMI6 24905265 IC50 = 100000 nM T95913 CWE3V0 24905267 IC50 = 100000 nM T95913 CH4T3A 24905268 IC50 = 50000 nM T95913 C6QDN7 24905271 IC50 = 3600 nM T95913 C6XHJ7 24905272 IC50 = 4500 nM T95913 CTB9A3 24905273 IC50 = 17000 nM T95913 C0NB1Q 24905274 IC50 = 6300 nM T95913 C9KQ0L 24905275 IC50 = 5100 nM T95913 C9O8QZ 24905277 IC50 = 4000 nM T95913 CP50RD 24905280 IC50 = 209 nM T95913 CG13ZM 24905281 IC50 = 735 nM T95913 CF0S6X 24905282 IC50 = 5160 nM T95913 C5HBL0 24905284 IC50 = 3340 nM T95913 C2Z5DN 24905285 IC50 = 852 nM T95913 CL6GH8 24905286 IC50 = 523 nM T95913 CKYO98 24905287 IC50 = 435 nM T95913 CRNQ65 24905288 IC50 = 340 nM T95913 COD7I5 24905289 IC50 = 772 nM T95913 C4LP7E 24905290 IC50 = 550 nM T95913 CE9JC2 24905291 IC50 = 200 nM T95913 C2GI1R 24905292 IC50 = 909 nM T95913 CHW8C4 24905293 IC50 = 355 nM T95913 CQF0H1 24905294 IC50 = 120 nM T95913 CNO7X0 24905295 IC50 = 140 nM T95913 C5WRG7 24905296 IC50 = 116 nM T95913 CQ1S0U 24905297 IC50 = 311 nM T95913 C4UES7 24905298 IC50 = 353 nM T95913 CMS69P 24905299 IC50 = 12500 nM T95913 CC0U5M 24905300 IC50 = 147 nM T95913 CW7X6S 24905301 IC50 = 16400 nM T95913 C97IQV 24905302 IC50 = 257 nM T95913 CSJ47V 24905303 IC50 = 1530 nM T95913 CPN74C 24905304 IC50 = 1820 nM T95913 C5CS3N 24905305 IC50 = 1390 nM T95913 CK4XE9 24905307 IC50 = 1070 nM T95913 CTU6Z3 24905308 IC50 = 100000 nM T95913 C9SQX1 24905309 IC50 = 780 nM T95913 CM75JP 24905310 IC50 = 1190 nM T95913 C9Q2BJ 24905311 IC50 = 1270 nM T95913 C9VUA1 24905312 IC50 = 366 nM T95913 CU3RS1 24905313 IC50 = 460 nM T95913 CYG3H2 24905314 IC50 = 633 nM T95913 CV5Q7O 24905315 IC50 = 283 nM T95913 C8SA3O 24905316 IC50 = 113 nM T95913 CI5MN3 24905317 IC50 = 58 nM T95913 CJ1P7K 24905318 IC50 = 43 nM T95913 C1T6YQ 24905319 IC50 = 554 nM T95913 CAU86X 24905320 IC50 = 342 nM T95913 C54ISY 24905321 IC50 = 808 nM T95913 C2GE5I 24905322 IC50 = 637 nM T95913 C8D6YK 24905323 IC50 = 606 nM T95913 C5NZH9 24905324 IC50 = 80 nM T95913 C9D6JR 24905325 IC50 = 1070 nM T95913 CLZT41 24905326 IC50 = 293 nM T95913 CW8FD3 24905327 IC50 = 808 nM T95913 CHB7A2 24905328 IC50 = 502 nM T95913 CA8EI3 24905329 IC50 = 448 nM T95913 CCQ0O7 24905330 IC50 = 1080 nM T95913 CJ81AS 24905331 IC50 = 39 nM T95913 C8PW4H 24905332 IC50 = 44 nM T95913 C2Y5TF 24905333 IC50 = 54 nM T95913 CH9FL5 24905334 IC50 = 2300 nM T95913 C1S0PC 24905335 IC50 = 1900 nM T95913 C8N9MV 24905336 IC50 = 7900 nM T95913 C9E8BJ 24905338 IC50 = 4000 nM T95913 CKZ80E 24905342 IC50 = 340 nM T95913 CO8SH1 24905343 IC50 = 200 nM T95913 C7IZL6 24905344 IC50 = 890 nM T95913 CLD3X6 24936051 IC50 = 47 nM T95913 C43VSW 24936353 IC50 = 501.19 nM T95913 C98MEW 24946175 IC50 = 6.7 nM T95913 CC7H3U 24946706 IC50 = 5.2 nM T95913 C78NJE 24955795 IC50 = 3130 nM T95913 C8P6NT 24956158 IC50 = 854 nM T95913 CJI29P 24956159 IC50 = 6654 nM T95913 C6C4RH 24993871 IC50 = 19 nM T95913 CL0TI6 24993895 IC50 = 6165.95 nM T95913 CS3Q8B 24995659 Ki > 4000 nM T95913 C8W3FZ 25023762 IC50 = 77.7 nM T95913 CZ9WE5 25023763 IC50 = 29.5 nM T95913 C3RL8W 25023764 IC50 = 36.1 nM T95913 CI6M9D 25023765 IC50 = 43.7 nM T95913 CF76VL 25023766 IC50 = 2.79 nM T95913 CC1KV3 25023767 IC50 = 2.34 nM T95913 CX7HP1 25023768 IC50 = 18.4 nM T95913 CEO7L0 25023769 IC50 = 33.2 nM T95913 CPA38V 25023770 IC50 = 1.92 nM T95913 C6QML7 25023771 IC50 = 4.28 nM T95913 C3VI4L 25023772 IC50 = 4.96 nM T95913 C6IOR9 25023773 IC50 = 4.84 nM T95913 CEW91Q 25032963 IC50 = 20 nM T95913 CY50OT 25052783 IC50 = 78 nM T95913 CHR51O 25057242 IC50 = 2600 nM T95913 CTM16Y 25069911 IC50 = 7909 nM T95913 CVI2S5 25070227 IC50 = 7582 nM T95913 CNL4Y2 25070228 IC50 = 11000 nM T95913 CSDN18 25070229 IC50 = 7907 nM T95913 CK92QL 25070230 IC50 = 10322 nM T95913 CKZ7X2 25070231 IC50 = 5830 nM T95913 C0T4NK 25070551 IC50 = 683 nM T95913 C1UKQ4 25070552 IC50 = 1378 nM T95913 CZRA03 25070553 IC50 = 2378 nM T95913 CO20FT 25070554 IC50 = 10000 nM T95913 CL4B5Z 25070555 IC50 = 1650 nM T95913 C7U0SC 25070882 IC50 = 1134 nM T95913 CCN36H 25071204 IC50 = 44 nM T95913 CQ7P4X 25071206 IC50 = 119 nM T95913 C14SFA 25071208 IC50 = 204 nM T95913 CNCJ40 25071516 IC50 = 61 nM T95913 CXWO13 25071518 IC50 = 776 nM T95913 CBH13R 25071519 IC50 = 1102 nM T95913 CJM7O0 25071520 IC50 = 594 nM T95913 C68PFD 25073081 IC50 = 583 nM T95913 CBJ20X 25073385 IC50 = 306 nM T95913 CZN7W0 25073388 IC50 = 368 nM T95913 CD69RK 25097993 IC50 = 33 nM T95913 CLP07J 25110819 IC50 > 10000 nM T95913 CVM89J 25128663 IC50 = 79.43 nM T95913 C4HRL9 25128667 IC50 = 39.81 nM T95913 C4SWT5 25128668 IC50 = 158.49 nM T95913 CIO6A4 25129024 IC50 = 630.96 nM T95913 CLS7P0 25129381 IC50 = 1995.26 nM T95913 C9R2EA 25129383 IC50 = 3981.07 nM T95913 C4YZL9 25129386 IC50 = 316.23 nM T95913 CDO9Q0 25129729 IC50 = 3981.07 nM T95913 CX86YV 25129734 IC50 = 398.11 nM T95913 CA2K4U 25130429 IC50 = 316.23 nM T95913 C1J8KH 25132804 IC50 = 3981.07 nM T95913 CI04XW 25132806 IC50 = 1000 nM T95913 C5WC4L 25133141 IC50 = 251.19 nM T95913 CSH37X 25133142 IC50 = 63.1 nM T95913 CW3HN6 25133144 IC50 = 1584.89 nM T95913 C4LHV1 25165368 IC50 > 10000 nM T95913 C2CXH3 25165371 IC50 > 10000 nM T95913 CQWL59 25165372 IC50 > 10000 nM T95913 CL87JW 25165773 IC50 = 7000 nM T95913 CB89TL 25165774 IC50 > 10000 nM T95913 CFZI92 25165961 IC50 > 10000 nM T95913 CK2YI4 25168990 IC50 = 6309.57 nM T95913 CC1D8V 25172062 IC50 = 14 nM T95913 CPW2D9 25172477 IC50 = 11 nM T95913 CLW96O 25207689 IC50 = 15 nM T95913 CWP29U 25242324 IC50 = 16 nM T95913 C4V2EJ 25261231 IC50 = 148 nM T95913 C3IDN0 25266674 IC50 = 12589.25 nM T95913 CIXE02 28063903 IC50 = 915000 nM T95913 C2IM0O 39733146 IC50 = 2511.89 nM T95913 CO4PL8 42606076 IC50 > 100000 nM T95913 C20VGT 42606077 IC50 = 40000 nM T95913 C7N5EC 42606078 IC50 > 100000 nM T95913 CIF63E 42623219 IC50 = 100 nM T95913 C3DNM9 42623223 IC50 = 25.12 nM T95913 COR5I0 42623224 IC50 = 251.19 nM T95913 CX1DC2 42623385 IC50 = 6.31 nM T95913 CR6N3I 42623632 IC50 = 15.85 nM T95913 C4EM0W 42623869 IC50 = 630.96 nM T95913 C5TY9Q 42623950 IC50 = 158.49 nM T95913 C10RBA 42636535 IC50 = 8000 nM T95913 C8N6CY 44119296 IC50 = 156000 nM T95913 C3ROX1 44124863 Ki = 1.9 nM T95913 CI3K7H 44129042 IC50 = 7900 nM T95913 CIE0J3 44129043 IC50 > 10000 nM T95913 CUW85V 44129044 IC50 > 10000 nM T95913 C2B9DE 44129118 IC50 = 8300 nM T95913 C0R1PH 44129198 IC50 > 10000 nM T95913 C6LGD5 44129200 IC50 = 3000 nM T95913 C03RLS 44129270 IC50 > 10000 nM T95913 CU4H1I 44129274 IC50 > 10000 nM T95913 C79QOC 44129275 IC50 = 6100 nM T95913 C0W3ZF 44129348 IC50 > 10000 nM T95913 CH6RO4 44129351 IC50 > 10000 nM T95913 CPAU59 44129353 IC50 > 10000 nM T95913 CN5O4I 44129429 IC50 = 2900 nM T95913 C3ZSV2 44129432 IC50 = 6300 nM T95913 CM5U2I 44137407 IC50 = 211 nM T95913 CQ82MS 44138035 IC50 = 23000 nM T95913 CZA3N9 44138128 IC50 = 34000 nM T95913 CF17OS 44180029 IC50 = 808 nM T95913 CHK8Z6 44180034 IC50 = 1170 nM T95913 CEJ5F7 44180035 IC50 = 9180 nM T95913 CQNT23 44180155 IC50 = 158 nM T95913 CIKM57 44180156 IC50 = 1310 nM T95913 CBP2T3 44180157 IC50 = 1090 nM T95913 C9CGB4 44180282 IC50 = 503 nM T95913 C2S5LC 44180395 IC50 = 410 nM T95913 C40NOQ 44180397 IC50 = 1080 nM T95913 CTB46H 44180398 IC50 = 547 nM T95913 CRS2G3 44180853 IC50 = 3945 nM T95913 C2VZX7 44181492 IC50 > 50000 nM T95913 C7SYM2 44181493 IC50 = 8780 nM T95913 CB8KF1 44181494 IC50 = 5460 nM T95913 C5AI8R 44181598 IC50 = 4220 nM T95913 CK03RW 44181599 IC50 = 2310 nM T95913 CXL61J 44181600 IC50 = 1570 nM T95913 C6TZK5 44181601 IC50 = 385 nM T95913 CCIV74 44181602 IC50 = 553 nM T95913 C36WUP 44181603 IC50 > 50000 nM T95913 CS2U7R 44181604 IC50 = 6300 nM T95913 CL6W0C 44181605 IC50 = 314 nM T95913 CFD41Z 44181718 IC50 = 7500 nM T95913 C2RB1P 44181719 IC50 = 5200 nM T95913 CMC75I 44181720 IC50 = 1390 nM T95913 CWTS93 44181721 IC50 = 667 nM T95913 CT1JL2 44181722 IC50 = 586 nM T95913 CE9HO1 44181723 IC50 = 5560 nM T95913 CFSB29 44181724 IC50 = 4990 nM T95913 CS0M9A 44187604 IC50 = 18.5 nM T95913 C0BRI9 44187779 IC50 = 37 nM T95913 CDA81B 44187783 IC50 = 25 nM T95913 C0LB8S 44187784 IC50 = 11.5 nM T95913 CCTO21 44187951 IC50 = 84.5 nM T95913 CVYS60 44187952 IC50 = 12 nM T95913 C8X3UZ 44187955 IC50 = 9 nM T95913 CJU85Z 44188321 IC50 = 33 nM T95913 CHU02A 44188322 IC50 = 17.2 nM T95913 C69HQS 44188840 IC50 = 13.5 nM T95913 CD78AG 44188841 IC50 = 19.5 nM T95913 CY7EL1 44188842 IC50 = 21.5 nM T95913 C0SE1X 44188843 IC50 = 48.5 nM T95913 CG13ZF 44188844 IC50 = 24.8 nM T95913 CR0BF9 44189010 IC50 = 78 nM T95913 C71NFL 44189011 IC50 = 69 nM T95913 C39ABJ 44189192 IC50 = 17.5 nM T95913 CK73NR 44219749 IC50 = 6315 nM T95913 CZ3L7W 44233390 IC50 = 1697 nM T95913 CA7R1U 44233391 IC50 = 1772 nM T95913 CU2F9E 44413107 IC50 = 29 nM T95913 C9SK8P 44413114 IC50 = 200 nM T95913 C9ZML1 44454396 IC50 = 117 nM T95913 CVG75D 44473371 IC50 = 8 nM T95913 C30NZA 44475985 IC50 = 69 nM T95913 CAT8F7 44475986 IC50 = 185 nM T95913 CSR73H 44475987 IC50 = 1300 nM T95913 CDAX92 44475988 IC50 = 113 nM T95913 CBH0S5 44475989 IC50 = 20000 nM T95913 CW5A7L 44475990 IC50 = 4 nM T95913 CLKU13 44481151 Ki = 39 nM T95913 CX3FK1 44513884 IC50 = 28.5 nM T95913 CL4RO5 44513885 IC50 = 34 nM T95913 C6RC9J 44513886 IC50 = 27 nM T95913 CGS7Q4 44513887 IC50 = 23 nM T95913 CSVD32 44513888 IC50 = 438 nM T95913 CLN2M5 44514201 IC50 = 52.5 nM T95913 C2Y8ML 44514203 IC50 = 219.5 nM T95913 CA9H8D 44514205 IC50 = 528 nM T95913 C01ZJI 44514208 IC50 = 18 nM T95913 CZ8WK6 44514210 IC50 = 24.5 nM T95913 CI8H3K 44514481 IC50 = 814.5 nM T95913 C51SEJ 44515083 IC50 = 21.5 nM T95913 CXBV98 44515084 IC50 = 14.5 nM T95913 C73HNB 44515696 IC50 = 85 nM T95913 CB7XW5 44516307 IC50 = 48.5 nM T95913 C4W5EM 44516309 IC50 = 9 nM T95913 C8VAU1 44516310 IC50 = 20 nM T95913 C8I1ZB 44516311 IC50 = 9 nM T95913 CSJ95V 44516635 IC50 = 10 nM T95913 CV6Z0N 44516636 IC50 = 10 nM T95913 CB3MV8 44517288 IC50 = 49.5 nM T95913 CDEQ97 44520808 IC50 = 993 nM T95913 CB4RN0 44520812 IC50 = 2367 nM T95913 CFC65B 44539960 IC50 <= 1000 nM T95913 C03IGD 44540030 IC50 = 7943.28 nM T95913 C5LWU1 44540126 IC50 = 7943.28 nM T95913 CYD4Z8 44540130 IC50 = 50.12 nM T95913 CAT2R7 44540316 IC50 = 15848.93 nM T95913 C36NRP 44540403 IC50 <= 1000 nM T95913 C2T9GC 44540407 IC50 = 6309.57 nM T95913 CQ4PE7 44540492 IC50 > 25118.86 nM T95913 C6HC3L 44548482 IC50 = 72.5 nM T95913 CH3L9P 44551660 IC50 > 1000 nM T95913 CYMD49 44552663 IC50 = 1358 nM T95913 C6B7LH 44552664 IC50 = 473 nM T95913 C3QZX0 44552666 IC50 = 283 nM T95913 C64OQC 44552667 IC50 = 155 nM T95913 C7LG6Q 44552844 IC50 = 404 nM T95913 C9T2CZ 44552845 IC50 = 76 nM T95913 CXLD75 44552846 IC50 = 109 nM T95913 CALT95 44554240 IC50 = 2781 nM T95913 CVDA08 44554755 IC50 = 1458 nM T95913 C25EGX 44554909 IC50 = 1820 nM T95913 CR4J0X 44554913 IC50 = 1625 nM T95913 CWV2T9 44554915 IC50 = 402 nM T95913 CCW12H 44555222 IC50 = 269 nM T95913 CTM8S9 44555225 IC50 = 2419 nM T95913 C7PSO6 44555226 IC50 = 646 nM T95913 C3VRO9 44557921 IC50 = 12.59 nM T95913 CRE61W 44577592 IC50 = 258 nM T95913 CH63GM 44577593 IC50 = 113 nM T95913 CA8MV5 44577594 IC50 = 321 nM T95913 C9IXW8 44577638 IC50 = 159 nM T95913 C8A5RT 44577639 IC50 = 28 nM T95913 CNP02V 44577640 IC50 = 73 nM T95913 CT6GN5 44577641 IC50 = 189 nM T95913 CIQR97 44577850 IC50 = 959 nM T95913 CCG8P9 44577851 IC50 = 16840 nM T95913 CLBA40 44577853 IC50 = 357 nM T95913 COU6V7 44577854 IC50 = 531 nM T95913 C8M5FY 44577914 IC50 = 318 nM T95913 C3MGZ9 44577915 IC50 > 20000 nM T95913 CGO09K 44577916 IC50 = 80 nM T95913 CRJ3B7 44577917 IC50 = 210 nM T95913 CTR89C 44577918 IC50 > 20000 nM T95913 CO05YG 44577919 IC50 = 163 nM T95913 CT70WA 44577920 IC50 = 77 nM T95913 C5KXS4 44577921 IC50 = 145 nM T95913 CZ2HI5 44577922 IC50 = 107 nM T95913 CGTU34 44577950 IC50 = 819 nM T95913 CQC50R 44577951 IC50 = 52 nM T95913 C8ZTW2 44577952 IC50 = 440 nM T95913 CIL93G 44577953 IC50 = 617 nM T95913 C8NB5H 44578037 IC50 > 40000 nM T95913 CX9TO2 44578038 IC50 = 35730 nM T95913 C7AHR4 44578039 IC50 > 50000 nM T95913 C13LGI 44578040 IC50 > 50000 nM T95913 CNZ06H 44578074 IC50 > 50000 nM T95913 C41TYA 44578108 IC50 = 63 nM T95913 C2W3SQ 44578109 IC50 = 223 nM T95913 CYM69I 44580064 IC50 = 51 nM T95913 CV09JM 44580065 IC50 = 34 nM T95913 CF37TO 44580066 IC50 = 35 nM T95913 CA0BU6 44580067 IC50 = 203 nM T95913 COQ85J 44580235 IC50 = 24 nM T95913 CD4ER0 44580236 IC50 = 20 nM T95913 CHVQ28 44580237 IC50 = 34 nM T95913 C8N2AF 44580238 IC50 = 767 nM T95913 C40LVX 44580274 IC50 = 1288 nM T95913 CO9LD8 44580275 IC50 = 138 nM T95913 C5QWG4 44580276 IC50 = 222 nM T95913 CFZS45 44580277 IC50 = 174 nM T95913 CQ4CR6 44580635 IC50 = 201 nM T95913 CJHK57 44580636 IC50 = 257 nM T95913 CC6M2E 44580684 IC50 = 70 nM T95913 CA3KP5 44580685 IC50 = 180 nM T95913 C40VHS 44580686 IC50 = 52 nM T95913 CXV92J 44580687 IC50 = 767 nM T95913 CG3PH2 44580721 IC50 = 327 nM T95913 CIO46B 44580722 IC50 = 48 nM T95913 CNLS71 44580723 IC50 = 35 nM T95913 C1N0MF 44580724 IC50 = 18 nM T95913 CAHQ76 44580766 IC50 = 131 nM T95913 C2XN6B 44580767 IC50 = 51 nM T95913 CC36YN 44580768 IC50 = 70 nM T95913 CZ56FY 44580769 IC50 = 46 nM T95913 CL8S0Y 44592136 IC50 >= 50000 nM T95913 C9E6JV 44592170 IC50 = 10000 nM T95913 C8DUA1 44592171 IC50 < 10000 nM T95913 CY8VU1 44592172 IC50 < 10000 nM T95913 C56TOC 44592173 IC50 < 10000 nM T95913 CGP6M7 44592216 IC50 >= 100000 nM T95913 CS38JL 44592217 IC50 = 100000 nM T95913 CJ1FW0 44592218 IC50 > 100000 nM T95913 C70VRG 44592219 IC50 > 100000 nM T95913 CW5RQ0 44592258 IC50 > 100000 nM T95913 CVB1I3 44592259 IC50 > 100000 nM T95913 CV9MY8 44592260 IC50 > 100000 nM T95913 CA65CE 44592261 IC50 > 100000 nM T95913 CEHY48 44592262 IC50 > 100000 nM T95913 C09OLK 44592299 IC50 = 42000 nM T95913 CJM35R 44592300 IC50 > 100000 nM T95913 C54DKW 44592302 IC50 = 42000 nM T95913 CJX76V 44592338 IC50 > 100000 nM T95913 CNY53M 44592339 IC50 > 100000 nM T95913 CXPK04 44592340 IC50 > 100000 nM T95913 C0L2HO 44593630 IC50 = 107 nM T95913 C2NQ6Z 44593631 IC50 = 22 nM T95913 CHKQ45 44593990 IC50 > 10000 nM T95913 CY3SV7 44596118 IC50 > 10000 nM T95913 C28QLM 44605035 IC50 = 6224 nM T95913 C75XHS 44605037 IC50 = 495 nM T95913 C3F4UX 44605249 IC50 = 1431 nM T95913 CQ0FZ7 44605426 IC50 = 3765 nM T95913 CC7G2L 44605427 IC50 = 3554 nM T95913 CDLP04 44605428 IC50 = 409 nM T95913 CSKN09 44605429 IC50 = 2526 nM T95913 CA79QG 44605430 IC50 = 1290 nM T95913 CH6V9F 44608754 IC50 = 6.5 nM T95913 C0IY9N 44608757 IC50 = 16 nM T95913 C90ITS 44608915 IC50 = 8.1 nM T95913 CZH1P9 44609387 IC50 = 2.4 nM T95913 CNDX48 44609388 IC50 = 13 nM T95913 CE95RQ 44620964 IC50 = 15 nM T95913 CVYJ36 44620965 IC50 = 33 nM T95913 CA8BY7 44621440 IC50 = 31.62 nM T95913 C5M1FR 44621441 IC50 = 25.12 nM T95913 C5LD7E 44621442 IC50 = 7.943 nM T95913 CO4GT0 44621447 IC50 = 25.12 nM T95913 CUV26H 44621448 IC50 = 19.95 nM T95913 CV2MG9 44621449 IC50 = 19.95 nM T95913 C24IYW 44621451 IC50 = 39.81 nM T95913 C0F9YW 44621452 IC50 = 100 nM T95913 C0GRD8 44621454 IC50 = 79.43 nM T95913 C4YHJ0 44621456 IC50 = 19.95 nM T95913 C31VBF 44621458 IC50 = 15.85 nM T95913 CQD03G 44623048 Ki = 770 nM T95913 C54IUP 44818842 IC50 = 435 nM T95913 C16IMZ 44819024 IC50 = 49 nM T95913 CN38JF 44819199 IC50 = 48.5 nM T95913 CVW6L8 44819200 IC50 = 22 nM T95913 CZ7M6D 44819201 IC50 = 12.2 nM T95913 C7MU8J 44819203 IC50 = 12.3 nM T95913 C8FU0W 44819375 IC50 = 22 nM T95913 C4N8CK 44819376 IC50 = 25 nM T95913 CP6DB9 45265864 IC50 = 40 nM T95913 C5I1VH 45379222 IC50 = 789 nM T95913 CA4JZ8 45379223 IC50 = 65 nM T95913 CZ68MG 45488079 IC50 > 10000 nM T95913 CV1U7I 46180604 IC50 = 8.4 nM T95913 CED2B3 46180606 IC50 = 5100 nM T95913 CDV85O 46180663 IC50 = 1300 nM T95913 CZGB46 46180666 IC50 = 15 nM T95913 C61ZLI 46190736 IC50 = 265 nM T95913 C6H3GT 46196486 IC50 = 33 nM T95913 CAU17V 46202808 IC50 = 3.162 nM T95913 CDA3R9 46220225 IC50 = 8 nM T95913 CIJ5V9 46224766 IC50 = 223 nM T95913 CIPV59 46224808 IC50 = 640 nM T95913 CRQ5M4 46225259 IC50 = 10000 nM T95913 C65IPQ 46225280 IC50 = 133 nM T95913 C8A7QJ 46225281 IC50 = 341 nM T95913 CPL45H 46225307 IC50 = 6907 nM T95913 CTN8J2 46225308 IC50 = 8297 nM T95913 CL34IK 46227801 IC50 = 510 nM T95913 C6D2RL 46227820 IC50 = 975 nM T95913 CSIK15 46228569 IC50 = 7470 nM T95913 C94YRI 46853654 IC50 = 3.981 nM T95913 CZ3WS1 46861592 IC50 = 5 nM T95913 CRO8W0 46865423 IC50 = 25 nM T95913 C47VTS 46865424 IC50 = 11 nM T95913 CO3P0J 46866604 IC50 = 1256 nM T95913 CQ2Y1V 46866705 Ki = 0.111 nM T95913 C63RCG 46870269 IC50 = 2.512 nM T95913 CTQ25M 46871497 IC50 = 6.31 nM T95913 CXRI03 46872177 Ki = 0.048 nM T95913 CC0R5U 46872178 Ki = 0.017 nM T95913 C8SRB0 46872297 Ki = 0.157 nM T95913 C67QZY 46872298 Ki = 0.33 nM T95913 CQB16A 46872415 Ki = 0.003 nM T95913 C7V8RJ 46873664 Ki = 0.066 nM T95913 CJB8T7 46873665 Ki = 0.011 nM T95913 CU7Z9M 46873667 Ki = 0.013 nM T95913 C6MZ1J 46884121 IC50 = 6949 nM T95913 CLA40T 46885426 IC50 = 3628 nM T95913 CC8T1E 46885496 IC50 = 2220 nM T95913 CCS20H 46885565 IC50 = 10 nM T95913 CG47YP 46885566 IC50 = 587 nM T95913 C4R3XP 46885599 IC50 = 54 nM T95913 CV5MK6 46885601 IC50 = 976 nM T95913 C42WVO 46885648 IC50 = 322 nM T95913 C3HMQ2 46891474 IC50 = 2.4 nM T95913 CB6Z8P 46892208 IC50 = 6200 nM T95913 CZX46Y 46892342 IC50 = 110 nM T95913 C5FN6I 46892845 IC50 = 320 nM T95913 CQ32BN 46892970 IC50 = 8 nM T95913 COJA32 46892971 Ki = 69 nM T95913 C5QFB3 46893088 IC50 = 200 nM T95913 CS30AI 46893754 IC50 = 3600 nM T95913 CPO1N7 46927938 Ki = 179 nM T95913 CJ0VB4 46932297 IC50 = 430 nM T95913 CL84AF 46946248 Ki > 500 nM T95913 CF14PE 46947264 IC50 = 74 nM T95913 COE37N 49778924 IC50 = 790 nM T95913 C7ZK3D 49783923 IC50 = 316.23 nM T95913 CHX76J 49784892 Ki = 29 nM T95913 CA1H8S 49784893 Ki = 88 nM T95913 CP2QD0 49784894 Ki = 4 nM T95913 CTZG05 49784988 Ki = 45 nM T95913 CE9AC5 49785078 Ki = 23 nM T95913 CG2IO7 49785079 Ki = 12 nM T95913 C8EYN4 49785083 Ki = 17 nM T95913 CBNZ47 49785166 Ki = 136 nM T95913 CZI34V 49785167 Ki = 330 nM T95913 CJK65T 49785253 Ki = 51 nM T95913 CXK8F5 49785436 Ki = 2 nM T95913 CWL5C6 49785518 Ki = 6 nM T95913 C3NV0J 49785827 Ki = 12 nM T95913 C0OZM2 49785828 Ki = 200 nM T95913 C1AR4G 49785829 Ki = 450 nM T95913 C39HAK 49785832 Ki = 12 nM T95913 C90JBE 49834576 IC50 > 10000 nM T95913 C5UR4A 49843944 IC50 = 720 nM T95913 CS40YB 49853846 IC50 = 230 nM T95913 C7PER0 49853953 IC50 = 660 nM T95913 CU9A8O 49854022 IC50 > 10000 nM T95913 C51QVH 49854023 IC50 = 10000 nM T95913 CM4HQ2 49854024 IC50 > 10000 nM T95913 C1LBX3 49854049 IC50 = 430 nM T95913 CVC2H6 49854052 IC50 = 290 nM T95913 CC2X9N 49854121 IC50 > 10000 nM T95913 CAJ58E 49854156 IC50 = 180 nM T95913 CAU39Y 49854158 IC50 = 200 nM T95913 CPK6X3 49854360 IC50 = 1400 nM T95913 CBVT70 49854361 IC50 = 4000 nM T95913 CQ1TZ6 49854365 IC50 = 1100 nM T95913 CJ5I9X 49854461 IC50 = 330 nM T95913 CDXQ69 49854462 IC50 = 8000 nM T95913 C0ORZ9 49854466 IC50 = 200 nM T95913 CY14XF 49854572 IC50 = 1200 nM T95913 CEC10T 49854573 IC50 = 15 nM T95913 C39KQW 49854679 IC50 = 200 nM T95913 C8VDR2 49854680 IC50 = 160 nM T95913 CN2V8R 49854681 IC50 = 990 nM T95913 CSN96A 49855001 IC50 = 230 nM T95913 CALY90 49855192 IC50 = 5000 nM T95913 CJPE20 49855193 IC50 = 2500 nM T95913 C1OM3I 49855237 IC50 = 17780 nM T95913 C26IQK 49857091 IC50 = 5300 nM T95913 CR0PN9 49857092 IC50 = 5700 nM T95913 CCJN26 49857093 IC50 = 1900 nM T95913 C3YG5L 49857275 IC50 > 10000 nM T95913 CHO65B 49857279 IC50 = 2640 nM T95913 C9HMY1 49857280 IC50 = 1800 nM T95913 CGW9L1 49857476 IC50 = 5150 nM T95913 CRD84P 49857479 IC50 = 1400 nM T95913 COF78C 49857678 IC50 > 10000 nM T95913 C4H7XG 49857865 IC50 = 2200 nM T95913 CY8MP7 49867926 IC50 = 9 nM T95913 CR0IA5 49871864 IC50 = 1100 nM T95913 C13WJZ 49872243 IC50 = 290 nM T95913 C5OY7B 49872246 IC50 = 146 nM T95913 C2KD5E 49872344 IC50 = 62 nM T95913 CV5BF3 49872645 IC50 = 634 nM T95913 CN97FO 49872646 IC50 = 22.5 nM T95913 CD6P5R 49872735 IC50 = 507 nM T95913 CL64NB 49872737 IC50 = 4650 nM T95913 CRNG04 49872831 IC50 = 11 nM T95913 CQC8B4 49872835 IC50 = 13 nM T95913 CPS3O1 49872924 IC50 = 120 nM T95913 CUBX74 49872925 IC50 = 19 nM T95913 CAW69U 49872927 IC50 = 220 nM T95913 CV1L4P 49873242 IC50 = 964 nM T95913 C5BA2V 49873243 IC50 = 3590 nM T95913 CSN45W 49873329 IC50 = 35.4 nM T95913 CLC2N7 50913517 IC50 = 20500 nM T95913 CJ4L8Y 50938829 Ki = 364 nM T95913 CJG65L 50939078 Ki = 509 nM T95913 CI8QM1 50939080 Ki = 28 nM T95913 CT0IP3 50939081 Ki = 90 nM T95913 C54EUL 50939212 Ki = 7340 nM T95913 CS7Z6U 50939338 Ki = 92 nM T95913 C2I9PS 50939992 IC50 = 18000 nM T95913 C9TUE4 50940108 IC50 = 1400 nM T95913 C2Q0GE 50990922 IC50 = 100 nM T95913 CKY3V1 50990924 Ki = 4.7 nM T95913 C5ZF9W 51003380 IC50 = 77000 nM T95913 CY36EH 51003592 IC50 = 398.11 nM T95913 CLB85F 51346892 IC50 = 740 nM T95913 C65ILG 51346893 IC50 = 44 nM T95913 CRJ5W8 51358113 IC50 = 5.67 nM T95913 CT91WR 52040626 IC50 = 371 nM T95913 CG7T4H 52913198 IC50 = 25 nM T95913 CD84MT 52913592 IC50 = 2200 nM T95913 C2TLG6 52913931 IC50 = 1800 nM T95913 CQ5GF2 52917084 Ki = 126 nM T95913 CAFR91 52917382 Ki = 361 nM T95913 C2DQK4 52917534 Ki = 50.1 nM T95913 C5ON6F 52919356 IC50 = 14 nM T95913 CM5BX0 52919492 IC50 = 68 nM T95913 CU1P2L 52940797 IC50 = 2010 nM T95913 CD62QJ 52940982 IC50 = 358 nM T95913 C43SVQ 52941322 IC50 = 189.5 nM T95913 CK59HM 52941479 IC50 = 150 nM T95913 C2KI6V 52942202 IC50 = 100000 nM T95913 CFRN73 52942850 IC50 = 122 nM T95913 C4D1KT 52942879 IC50 = 44 nM T95913 C4VCY0 52943258 IC50 = 16000 nM T95913 C1XEV2 52943394 IC50 = 2410 nM T95913 C73WTL 52943744 IC50 = 45.2 nM T95913 C6Q1AH 52943745 IC50 = 100 nM T95913 CHI0P6 52944356 IC50 = 100000 nM T95913 CWD27C 52945142 IC50 = 240 nM T95913 CWPC54 52945348 IC50 = 140 nM T95913 CXL53B 52945589 IC50 = 154 nM T95913 C4NLX7 52945630 IC50 = 723 nM T95913 CXD6T8 52945845 IC50 = 1200 nM T95913 CN8F0V 52946289 IC50 = 717 nM T95913 CMQY93 52946368 IC50 = 149 nM T95913 C5X9VO 52948007 IC50 = 290 nM T95913 C7ET6Z 52948010 IC50 = 1600 nM T95913 CW9Z1T 52949347 IC50 = 51 nM T95913 CV5B2C 52949497 IC50 = 25000 nM T95913 CB0KM5 52949869 IC50 = 98 nM T95913 CAJQ03 52950001 IC50 = 99 nM T95913 C5HQ2E 52950102 IC50 = 74 nM T95913 CH1Q5D 53234281 IC50 = 3 nM T95913 C45JKN 53234283 IC50 = 8.4 nM T95913 CVK28S 53235062 IC50 = 0.7 nM T95913 COW61E 53235216 IC50 = 1.5 nM T95913 CWE56X 53235217 IC50 = 3.7 nM T95913 CDXM59 53235451 IC50 = 55 nM T95913 CT8IN1 53242225 IC50 = 3200 nM T95913 C9NF0C 53302364 Ki = 42.4 nM T95913 C4J9WZ 53307606 IC50 = 5 nM T95913 C7ZH0D 53308041 IC50 = 1170 nM T95913 CRD3A9 53316967 IC50 = 340 nM T95913 C84YNK 53317325 IC50 > 83300 nM T95913 CS8DJ3 53318252 IC50 = 150 nM T95913 C58NQJ 53318614 IC50 = 55400 nM T95913 C10YUH 53318615 IC50 = 9700 nM T95913 C24GBF 53319075 IC50 = 15 nM T95913 CFJD70 53319932 IC50 = 70000 nM T95913 C3EJB1 53319933 IC50 = 9100 nM T95913 C2V7AX 53320017 IC50 = 380 nM T95913 CKGJ60 53320018 IC50 = 730 nM T95913 CJRM64 53322563 IC50 = 43500 nM T95913 CN92LK 53322732 IC50 = 9 nM T95913 CJZ29M 53325374 IC50 = 830 nM T95913 C1TE8J 53325515 IC50 = 7600 nM T95913 C6LAI9 53326166 IC50 = 960 nM T95913 CCU75P 53327266 Ki = 6 nM T95913 C1TWE6 53327269 Ki = 3 nM T95913 COSB47 53327579 Ki = 20 nM T95913 C62JOP 53327629 Ki = 4 nM T95913 CCX7M5 53353847 Ki = 20.7 nM T95913 C23HAU 53361718 IC50 = 7.7 nM T95913 CM60WQ 53361719 IC50 = 13 nM T95913 CL69DK 53377727 IC50 = 81 nM T95913 C6Q8RC 53378051 IC50 = 1584.89 nM T95913 CG3C1J 53379513 IC50 = 4.8 nM T95913 CSV9X2 54579940 IC50 = 13 nM T95913 CN51TL 54579941 IC50 = 4100 nM T95913 C7VZU2 54579942 IC50 = 2300 nM T95913 C4R9JB 54579943 IC50 = 610 nM T95913 CG26HQ 54579944 IC50 = 3700 nM T95913 CC5R3O 54580924 IC50 = 340 nM T95913 C3OIY4 54580925 IC50 = 250 nM T95913 C60TYL 54581049 IC50 = 470 nM T95913 CF2UH5 54581983 IC50 = 20 nM T95913 C23EVN 54582916 IC50 = 26 nM T95913 CT2SV7 54583916 IC50 = 480 nM T95913 CY87EC 54583917 IC50 = 30 nM T95913 C8CPI4 54584859 IC50 = 860 nM T95913 C9TZ2V 54584860 IC50 = 2300 nM T95913 CME81Q 54585830 IC50 = 190 nM T95913 CFI7E6 54754350 IC50 = 760 nM T95913 CE4TS9 56589559 IC50 = 32 nM T95913 CR24WQ 56595421 IC50 = 56 nM T95913 CJ41GT 56595686 IC50 = 52 nM T95913 C2PN4S 56599298 IC50 = 6600 nM T95913 CT64SR 56599306 IC50 = 23 nM T95913 CFUT05 56648675 IC50 = 17 nM T95913 C1GAB6 56648677 IC50 = 37 nM T95913 CWDF40 56648757 IC50 = 20 nM T95913 CE35CB 56648758 IC50 = 10 nM T95913 CJO39U 56648759 IC50 = 25 nM T95913 CNKC90 56654649 IC50 > 9100 nM T95913 C83QGP 56660108 IC50 = 9.5 nM T95913 CYM1D0 56660109 IC50 = 6 nM T95913 CHA35L 56663573 IC50 = 4 nM T95913 CF7PY5 56667023 IC50 = 7 nM T95913 CC1DJ8 56670464 IC50 = 20.5 nM T95913 CZH95G 56673952 IC50 = 8 nM T95913 CHR8K0 56677282 IC50 = 10.5 nM T95913 C79AMB 56677283 IC50 = 13.5 nM T95913 CG17TZ 56683916 IC50 = 9.5 nM T95913 C7B2OH 56683917 IC50 = 6.5 nM T95913 C6LMP8 56683918 IC50 = 14.3 nM T95913 C94JIT 56832510 Ki = 0.55 nM T95913 C0IJP8 56927258 IC50 > 6309.57 nM T95913 CM28GU 56928390 IC50 = 280 nM T95913 C9MJG4 56929824 IC50 = 50 nM T95913 CYFB96 56932203 IC50 = 63.1 nM T95913 CJ9R2C 56932209 IC50 = 630.96 nM T95913 C8C2FG 56932238 IC50 = 125.89 nM T95913 CX6Q2K 56932240 IC50 = 10 nM T95913 CPGC81 56947516 Ki = 1 nM T95913 CO6K5Q 56955953 IC50 = 441 nM T95913 CAK91L 56955954 IC50 = 18 nM T95913 C8B6JG 56955955 IC50 = 18 nM T95913 CX4W6G 57325497 IC50 = 1750 nM T95913 CVK5A3 57328247 Ki > 500 nM T95913 CW8B4D 57330208 IC50 = 850 nM T95913 C6JMN9 57345685 IC50 = 1600 nM T95913 CZ7RE0 57345686 IC50 = 1000 nM T95913 CA53SC 57351276 Ki = 183 nM T95913 C9RB7K 57391333 Ki > 500 nM T95913 CH37SE 57391335 Ki > 500 nM T95913 C1GVK3 57391362 IC50 > 4000 nM T95913 C0PR9J 57391364 IC50 > 6300 nM T95913 C6L9HO 57391365 IC50 = 3200 nM T95913 C2QX0T 57391366 IC50 = 1600 nM T95913 CLQ9J1 57391367 IC50 = 1300 nM T95913 CQ1W0C 57393124 IC50 = 7900 nM T95913 CZ0RW2 57393125 IC50 = 1600 nM T95913 COT0L2 57394595 IC50 = 19000 nM T95913 CA93ZE 57394864 IC50 = 3200 nM T95913 C6CL4F 57395172 IC50 = 980 nM T95913 CS14ZH 57396608 Ki > 500 nM T95913 CDG2F3 57396625 IC50 = 3200 nM T95913 CD73TE 57396626 IC50 > 6300 nM T95913 CQRU75 57396627 IC50 > 6300 nM T95913 CI34XH 57396628 IC50 > 6300 nM T95913 CYM02V 57397667 IC50 = 2060 nM T95913 CQO74C 57398382 Ki > 500 nM T95913 CV2Z0C 57398383 Ki > 500 nM T95913 C3Q2ZP 57398390 IC50 > 6300 nM T95913 C56TEZ 57398391 IC50 = 5000 nM T95913 CP9Q4U 57398392 IC50 = 10000 nM T95913 C0O5KE 57398393 IC50 = 320 nM T95913 C3G9HW 57399126 IC50 > 10000 nM T95913 CYE09F 57400062 IC50 = 4000 nM T95913 CN5PY7 57400063 IC50 > 7900 nM T95913 CT0Y7E 57400064 IC50 = 2500 nM T95913 C3Q2NF 57401565 IC50 = 395000 nM T95913 CRO5Z6 57401846 Ki > 500 nM T95913 CM63CS 57401865 IC50 = 1300 nM T95913 CG6M4H 57401867 IC50 > 6300 nM T95913 CP8FY5 57401868 IC50 = 1600 nM T95913 CQ5P4X 57401869 IC50 = 2500 nM T95913 CPG6N5 57402167 IC50 = 1310 nM T95913 C8LKZ3 57402168 IC50 = 1980 nM T95913 CF68RN 57403576 IC50 = 6300 nM T95913 CL2R7T 57403577 IC50 > 6300 nM T95913 CC5N9R 57403578 IC50 > 10000 nM T95913 CZ8M5F 57403579 IC50 = 1600 nM T95913 C5NT7R 57403580 IC50 = 1300 nM T95913 CHBV63 57403581 IC50 = 400 nM T95913 CAC72X 57403582 IC50 > 6300 nM T95913 CQ5Z4S 57404801 IC50 = 39.81 nM T95913 C78YHO 57404804 IC50 = 50.12 nM T95913 CNR95F 57404840 IC50 = 1900 nM T95913 CQ4E8N 57405149 IC50 = 50.12 nM T95913 CA8BT7 57405314 IC50 = 794.33 nM T95913 CI40MW 57405315 IC50 = 501.19 nM T95913 CGN72O 57405485 IC50 = 6.31 nM T95913 C5B9XS 57406164 IC50 = 3.981 nM T95913 CEI2S9 57406702 IC50 = 3162.28 nM T95913 CED47A 57410062 IC50 > 10000 nM T95913 C1BVX6 57411134 IC50 > 10000 nM T95913 C39JSW 57411135 IC50 > 10000 nM T95913 CL8F6Q 57411137 IC50 > 10000 nM T95913 CW97FT 57411139 IC50 > 10000 nM T95913 CU0R3A 57411250 IC50 > 10000 nM T95913 C6C5TU 57411252 IC50 > 10000 nM T95913 CD0W2I 57411254 IC50 = 8135 nM T95913 CW1DA3 57411255 IC50 > 10000 nM T95913 C6U4LO 57411256 IC50 > 10000 nM T95913 CP9G7L 57411366 IC50 = 4203 nM T95913 CC5DO3 57411369 IC50 > 10000 nM T95913 C56RBS 57411372 IC50 > 10000 nM T95913 CX9O3T 57411485 IC50 > 10000 nM T95913 CQBM65 57411486 IC50 > 10000 nM T95913 CK5QX7 57411488 IC50 > 10000 nM T95913 C90LNK 57411715 IC50 > 10000 nM T95913 CPXE40 57411716 IC50 > 10000 nM T95913 CE6RY5 57411836 IC50 > 10000 nM T95913 C5JOX3 57411837 IC50 > 10000 nM T95913 C0I5JM 57419280 IC50 > 10000 nM T95913 CT6XL0 57466811 Ki = 36 nM T95913 CRB5P2 57495287 IC50 > 9100 nM T95913 C59YAC 57495353 IC50 = 2230 nM T95913 CJE19S 57523686 IC50 > 10000 nM T95913 CHIU94 57545876 IC50 = 2.512 nM T95913 C0JQ8P 57584929 Ki = 36 nM T95913 CQU8A1 57585145 Ki = 36 nM T95913 C6L4FZ 57599744 IC50 = 810 nM T95913 CV9J7D 57748162 IC50 = 320 nM T95913 CL57CP 57789333 IC50 = 870 nM T95913 CZ21KP 57900314 IC50 = 2.2 nM T95913 CO20YT 58203712 IC50 = 0.6 nM T95913 C7X0OJ 58203779 IC50 = 8.4 nM T95913 CW1M9X 58203976 IC50 = 36 nM T95913 COFN62 58203995 IC50 = 80 nM T95913 C16GRS 58204034 IC50 = 19.1 nM T95913 CM62NB 58204076 IC50 = 3.5 nM T95913 CGA01N 58204242 IC50 = 4.3 nM T95913 CVR9Q2 58233988 IC50 = 25.12 nM T95913 CB9AH8 58234990 IC50 = 6000 nM T95913 CJ8YI2 58234995 IC50 = 830 nM T95913 CZF3U5 58235016 IC50 = 1000 nM T95913 CM0ND7 58235018 IC50 = 930 nM T95913 C25RXY 58235020 IC50 = 1600 nM T95913 CAY94U 58235030 IC50 = 4200 nM T95913 CAJC03 58235033 IC50 = 710 nM T95913 CN7MZ8 58235039 IC50 = 2600 nM T95913 CPW84H 58235041 IC50 = 630 nM T95913 C70CRN 58235043 IC50 = 3500 nM T95913 C5SQV3 58235052 IC50 = 700 nM T95913 CEZ4T5 58235053 IC50 = 2400 nM T95913 C82LIS 58235061 IC50 = 520 nM T95913 C3SO4E 58235062 IC50 = 530 nM T95913 CZ0SD5 58235073 IC50 = 1200 nM T95913 CQP25T 58235077 IC50 = 700 nM T95913 C0LDZ2 58235079 IC50 = 13000 nM T95913 C2YG5L 58235088 IC50 = 2600 nM T95913 CTVF29 58290044 Ki = 13 nM T95913 CJ6R8Q 59251679 IC50 = 8.2 nM T95913 CWF9Z7 59251848 Ki = 13 nM T95913 CRZ5B1 59251991 IC50 = 1190 nM T95913 C6A3KL 59293676 IC50 = 690 nM T95913 CC14ZL 59293709 IC50 = 1100 nM T95913 C0R3TX 59293715 IC50 = 1400 nM T95913 C9TVC6 59293721 IC50 = 1400 nM T95913 CZ5OV1 59293740 IC50 = 410 nM T95913 CB2Z4R 59293755 IC50 = 830 nM T95913 C8AL6C 59293763 IC50 = 610 nM T95913 CT3CF1 59477024 IC50 = 100 nM T95913 CF6YB8 59477038 IC50 = 3162.28 nM T95913 CK3H9O 59477041 IC50 = 199.53 nM T95913 C7KG5E 59477042 IC50 = 1000 nM T95913 C01DZW 59477048 IC50 = 251.19 nM T95913 CPE9X3 59507470 IC50 = 142 nM T95913 C2X8TY 59548177 Ki = 80 nM T95913 C71GBC 59548184 Ki = 7 nM T95913 CGRO45 59548196 Ki = 210 nM T95913 CD39AG 59548207 Ki = 750 nM T95913 C6KP4G 59548220 Ki = 110 nM T95913 CL82RM 59548221 Ki = 7 nM T95913 CTNU85 59548226 Ki = 54 nM T95913 CLB6N4 59548232 Ki = 1100 nM T95913 C2KBG8 59548236 Ki = 9 nM T95913 CSWV07 59548243 Ki = 130 nM T95913 CN48VL 59548245 Ki = 9 nM T95913 CMT2R0 59548250 Ki = 690 nM T95913 C3I8NE 59548256 Ki = 100 nM T95913 C8W5HT 59548263 Ki = 380 nM T95913 CT8Q5B 59548274 Ki = 8 nM T95913 CBG52T 59548278 Ki = 9 nM T95913 CVF1B2 59548283 Ki = 59 nM T95913 CY31EA 59548284 Ki = 99 nM T95913 CO4GT7 59548288 Ki = 1 nM T95913 CFR7S8 59548302 Ki = 24 nM T95913 CRE8B3 59548316 Ki = 16 nM T95913 CRM20Z 59548320 Ki = 140 nM T95913 CX1KJ9 59548322 Ki = 8 nM T95913 CJE5I4 59548341 Ki = 22 nM T95913 C8O1VS 59548349 Ki = 5 nM T95913 CE9W0K 59548355 Ki = 24 nM T95913 CWC65A 59548356 Ki = 9 nM T95913 CMKP95 59548371 Ki = 9 nM T95913 CC8UV3 59548383 Ki = 12 nM T95913 C4SN3U 59548390 Ki = 21 nM T95913 CD4ET2 59548402 Ki = 58 nM T95913 CES59T 59548403 Ki = 90 nM T95913 CE8P3G 59548407 Ki = 14 nM T95913 CO4K2W 59548419 Ki = 2.2 nM T95913 CSDB78 59548424 Ki = 8 nM T95913 C81FCQ 59548431 Ki = 9 nM T95913 CLGY34 59548453 Ki = 11 nM T95913 CBT21W 59548454 Ki = 91 nM T95913 C9DIB3 59548458 Ki = 9 nM T95913 CJT68K 59548460 Ki = 40 nM T95913 C9LFT3 59548462 Ki = 7 nM T95913 CA47YQ 59548474 Ki = 12 nM T95913 CX8C2U 59548480 Ki = 3600 nM T95913 C8S0ED 59605870 IC50 = 540 nM T95913 C4Y3GL 59609976 IC50 = 441 nM T95913 C1PC0J 59634638 IC50 = 210 nM T95913 CP2UY3 59634686 IC50 = 3530 nM T95913 C1TH2N 59634692 IC50 = 1420 nM T95913 CPA0L2 59634709 IC50 = 5360 nM T95913 C7DC6R 59662371 IC50 = 2398.83 nM T95913 C5S0FG 59662506 IC50 = 5754.4 nM T95913 CBI0M6 59688563 IC50 = 398.11 nM T95913 CUYB59 60148924 IC50 = 6600 nM T95913 CM8PD7 60150509 IC50 = 160 nM T95913 C5KD3Z 60154714 Ki > 10000 nM T95913 CS0L4D 60154996 Ki > 10000 nM T95913 C1UI3P 60155086 Ki = 2600 nM T95913 CX08ON 60155087 Ki = 480 nM T95913 CX8J1I 60155265 Ki = 9 nM T95913 CAT40I 60155266 Ki = 4 nM T95913 CD56VA 60155268 Ki = 21 nM T95913 CCQB56 60155375 IC50 = 10 nM T95913 CH5X2S 60155376 IC50 = 18 nM T95913 C74FEN 60155377 IC50 = 326 nM T95913 CZ6G4B 60155378 IC50 = 39 nM T95913 C10AHQ 60155379 IC50 = 17 nM T95913 C5FI4P 60155451 Ki = 18 nM T95913 CX9G4U 60155452 Ki = 8 nM T95913 C9Q7DE 60155469 IC50 = 26 nM T95913 CH8UY5 60155470 IC50 = 65 nM T95913 C3EDY4 60155471 IC50 = 507 nM T95913 CE0ZX1 60155472 IC50 = 152 nM T95913 CG90MC 60155473 IC50 = 53 nM T95913 C82PVI 60155474 IC50 = 167 nM T95913 CX49FT 60155475 IC50 = 161 nM T95913 CR7EG9 60155538 Ki = 46 nM T95913 CU6YB9 60155539 Ki = 30 nM T95913 CW6N1S 60155552 IC50 = 11 nM T95913 CIB08V 60155553 IC50 = 48 nM T95913 CZE28G 60155554 IC50 = 43 nM T95913 CZD2W7 60155555 IC50 = 31 nM T95913 CO6IU3 60155556 IC50 = 49 nM T95913 C6HN5O 60155557 IC50 = 18 nM T95913 CMQ9G1 60155638 IC50 = 507 nM T95913 CG56KT 60155639 IC50 = 26 nM T95913 CBJ65P 60155640 IC50 = 42 nM T95913 C8OJK0 60155641 IC50 = 5 nM T95913 CT9XJ6 60155642 IC50 = 21 nM T95913 C5BYQ3 60155643 IC50 = 8 nM T95913 C57RBF 60155722 IC50 = 587 nM T95913 CU7J6L 60155723 IC50 = 102 nM T95913 CSZA16 60155724 IC50 = 34 nM T95913 C21DWT 60155725 IC50 = 497 nM T95913 C12CQU 60155726 IC50 = 60 nM T95913 CA5TM3 60155805 IC50 = 20 nM T95913 C60RIO 60155806 IC50 = 6 nM T95913 CIRO73 66493714 IC50 = 167 nM T95913 C71LPV 66493729 IC50 = 302 nM T95913 C54NOW 66552297 IC50 > 100000 nM T95913 CX4HW1 66552298 IC50 > 50118.72 nM T95913 CEJ54A 66552343 IC50 = 501.19 nM T95913 CUQ5Y2 66552345 IC50 > 3981.07 nM T95913 C5F8ZE 66552346 IC50 > 100000 nM T95913 CHQC56 66552347 IC50 = 3162.28 nM T95913 CS6BQ0 66552348 IC50 > 12589.25 nM T95913 CGT2V9 66552407 IC50 = 3981.07 nM T95913 CIJ3C5 66552408 IC50 = 39.81 nM T95913 C6ZFI1 66552410 IC50 > 31622.78 nM T95913 C8S7CM 66552411 IC50 = 316.23 nM T95913 C9A7IK 66552412 IC50 > 39810.72 nM T95913 CRC24S 66552467 IC50 > 100000 nM T95913 CHU5V3 66552468 IC50 > 100000 nM T95913 C46POH 66552523 IC50 = 1995.26 nM T95913 C68LXT 66552524 IC50 = 25118.86 nM T95913 C91JZL 66553214 IC50 = 8280 nM T95913 CUC7B3 66557964 IC50 = 190 nM T95913 C9X2TB 66558056 IC50 = 340 nM T95913 CWZ54O 66600540 Ki = 20 nM T95913 C6Q0KU 66612050 Ki = 34 nM T95913 C1R3SI 66653673 IC50 = 3290 nM T95913 CF8BZ7 66677439 IC50 = 1060 nM T95913 C8L9DK 66743362 Ki = 14 nM T95913 C1IKT2 66743443 Ki = 11 nM T95913 CN0RE8 66779813 IC50 = 1000 nM T95913 C3IP5D 66779815 IC50 = 1000 nM T95913 CH86MR 66779905 IC50 = 1600 nM T95913 CX2N6E 66779920 IC50 > 790 nM T95913 C9O4TC 66779989 IC50 = 400 nM T95913 CF2UM8 66780001 IC50 = 4000 nM T95913 CHU0C5 66780007 IC50 = 500 nM T95913 CGL4V1 66780016 IC50 = 2000 nM T95913 C5F6OA 66780027 IC50 = 6300 nM T95913 C8DN7A 66780034 IC50 = 4000 nM T95913 C4AM6R 66780100 IC50 = 1300 nM T95913 CZ5P2N 66780118 IC50 = 160 nM T95913 CREA54 66780266 IC50 = 1300 nM T95913 CRCA72 66780292 IC50 = 2500 nM T95913 CW2SM6 66780337 IC50 = 250 nM T95913 CU54DY 66780379 IC50 = 2500 nM T95913 CQ70YA 66780434 IC50 > 7900 nM T95913 C8F9UY 66780515 IC50 = 250 nM T95913 CFH6C2 66780644 IC50 = 2500 nM T95913 CTZB46 66780835 IC50 = 7900 nM T95913 CEP5A2 66780844 IC50 > 6300 nM T95913 C51ARE 66788835 Ki = 5.3 nM T95913 C3PL1S 66800530 IC50 = 63.1 nM T95913 CJN4M2 66806967 IC50 = 630.96 nM T95913 CW12XO 66882257 IC50 > 10000 nM T95913 C6IO1S 66883557 IC50 > 10000 nM T95913 C1HSE0 67035086 IC50 = 980 nM T95913 C38RGB 67035556 IC50 > 9100 nM T95913 C5E4AJ 67050504 IC50 = 11 nM T95913 CMWO25 67061712 IC50 = 1.4 nM T95913 C0OX5N 67103709 IC50 = 1500 nM T95913 C9J2EO 67103712 IC50 = 210 nM T95913 CM4W1Y 67103722 IC50 = 2500 nM T95913 C5TYQ3 67103909 IC50 = 140 nM T95913 CVJ49E 67103974 IC50 = 1200 nM T95913 C3VFY7 67104025 IC50 = 3500 nM T95913 CC07KA 67104052 IC50 = 2900 nM T95913 C4Z0HT 67159178 IC50 <= 10000 nM T95913 C7EZW6 67192973 IC50 = 1600 nM T95913 CQHF85 67284779 IC50 = 2010 nM T95913 CT6BX3 67285457 Ki = 16000 nM T95913 C9LI0M 67294297 Ki = 49.1 nM T95913 C5BZ2V 67981475 IC50 = 1000 nM T95913 CK86XZ 67982080 IC50 = 316.23 nM T95913 CS0TY5 67982485 IC50 = 398.11 nM T95913 C9A2RD 67982543 IC50 = 3981.07 nM T95913 C7A0GH 67982639 IC50 = 1584.89 nM T95913 CW79LA 67982712 IC50 = 1258.93 nM T95913 CEG3F8 67983123 IC50 = 3000 nM T95913 C25AHY 67984037 IC50 = 8500 nM T95913 C7N4ZS 68034365 IC50 = 2400 nM T95913 CG53JO 68044823 Ki = 11 nM T95913 CGA82Q 68044837 Ki = 35 nM T95913 C4RLP9 68044907 Ki = 9 nM T95913 C6U8RP 68045063 Ki = 8 nM T95913 C0LQN1 68045070 Ki = 60 nM T95913 C7DL6V 68045162 Ki = 28 nM T95913 CA4JF3 68045179 Ki = 7 nM T95913 C57DTK 68045182 Ki = 4 nM T95913 CUQ2W1 68095924 IC50 = 158.49 nM T95913 CUR8N0 68096082 IC50 = 501.19 nM T95913 C8I7GC 68293638 IC50 > 10000 nM T95913 C45TIJ 69489467 Ki = 59.8 nM T95913 C8MTV6 70674592 IC50 = 280 nM T95913 CXB45Q 70674939 IC50 = 108 nM T95913 CAR46Z 70675172 IC50 = 72 nM T95913 CN09DI 70675846 IC50 = 97400 nM T95913 C6BQE1 70681248 IC50 = 1600 nM T95913 CPE36T 70681262 IC50 = 200 nM T95913 CPX41V 70682086 IC50 = 6.31 nM T95913 CZ5TI9 70682135 IC50 = 5120 nM T95913 CQW54O 70682591 Ki = 230 nM T95913 CPV59G 70682592 Ki = 1140 nM T95913 CB3ZN5 70683337 IC50 = 2500 nM T95913 C1I5PH 70683338 IC50 = 250 nM T95913 CSM0A6 70684204 IC50 = 2.512 nM T95913 CXD08N 70684690 Ki = 61 nM T95913 CG95EC 70684794 Ki = 84 nM T95913 C8O2QH 70685440 IC50 = 500 nM T95913 CZG9M1 70685441 IC50 = 2000 nM T95913 CH7KO0 70685442 IC50 = 1300 nM T95913 C6G4WB 70686339 IC50 = 251.19 nM T95913 CON8X4 70686340 IC50 = 63.1 nM T95913 C1ASW4 70686341 IC50 = 25.12 nM T95913 C0PWL5 70686455 IC50 = 125.89 nM T95913 CN4CR2 70686584 IC50 = 4100 nM T95913 C85FWA 70686829 Ki = 110 nM T95913 CQS8G7 70686830 Ki = 530 nM T95913 C8QSD2 70688455 IC50 = 7.943 nM T95913 CFCJ02 70688558 IC50 = 15.85 nM T95913 CSX6I7 70688908 Ki = 110 nM T95913 C1U5FC 70689024 Ki = 124 nM T95913 C5YN6U 70689166 IC50 = 5000 nM T95913 C6L4WY 70689639 IC50 = 790 nM T95913 CGT1X2 70690496 IC50 = 25.12 nM T95913 CTY78N 70690549 IC50 = 5740 nM T95913 CW3U5J 70690994 Ki = 260 nM T95913 CC6I1Q 70691259 IC50 = 3200 nM T95913 CD3JL4 70691776 IC50 = 500 nM T95913 CDK52M 70692650 IC50 = 15.85 nM T95913 CGQJ68 70692914 IC50 = 7.943 nM T95913 C7G5UV 70692915 IC50 = 7.943 nM T95913 C3TM1F 70693128 Ki = 57 nM T95913 C2VAU8 70693129 Ki = 32 nM T95913 CU3WF2 70693248 Ki = 26.7 nM T95913 C65FHO 70694723 Ki = 62.9 nM T95913 CPFO83 70694805 IC50 = 12.59 nM T95913 CRNY76 70695188 Ki = 62 nM T95913 C3N5YJ 70695189 Ki = 5810 nM T95913 C75YGN 70695469 IC50 > 3200 nM T95913 C61CFG 70696737 IC50 = 31.62 nM T95913 C7KL5X 70696852 IC50 = 125.89 nM T95913 CRH8E2 71270723 IC50 = 501.19 nM T95913 CWR58A 71270783 IC50 > 1479.11 nM T95913 CF9LU4 71270807 IC50 = 501.19 nM T95913 C7FDL2 71270817 IC50 = 398.11 nM T95913 CNR1G9 71270824 IC50 = 2511.89 nM T95913 C38LBA 71270831 IC50 = 316.23 nM T95913 CTL6R5 71270836 IC50 = 398.11 nM T95913 CM4LX7 71270848 IC50 > 6309.57 nM T95913 C2GWX6 71270906 IC50 = 1995.26 nM T95913 CX0DL3 71270910 IC50 > 3981.07 nM T95913 C0COW6 71270913 IC50 > 6309.57 nM T95913 CB0S8G 71270927 IC50 = 251.19 nM T95913 C24IOW 71270948 IC50 > 5011.87 nM T95913 C5BJ2Y 71270957 IC50 > 3162.28 nM T95913 C03NFY 71271625 IC50 > 5011.87 nM T95913 CL47JU 71271739 IC50 > 7943.28 nM T95913 CS5JG6 71271910 IC50 > 6309.57 nM T95913 C4PSK8 71271965 IC50 = 316.23 nM T95913 CB4N1M 71272066 IC50 > 5011.87 nM T95913 CD8E1Y 71272453 IC50 = 630.96 nM T95913 C8EW9V 71272757 IC50 = 3162.28 nM T95913 C0LO8I 71272765 IC50 = 398.11 nM T95913 C1MVL0 71273460 Ki = 40.6 nM T95913 CK58RV 71449587 IC50 = 91 nM T95913 C0ROQ6 71450451 IC50 = 22 nM T95913 CTL30H 71450452 IC50 = 12 nM T95913 CNX18D 71450453 IC50 = 24 nM T95913 C7HT4F 71450454 IC50 = 46 nM T95913 CNHJ63 71451228 IC50 = 777 nM T95913 CD8Y3S 71451617 Ki = 2350 nM T95913 C9SC2V 71452282 IC50 = 16 nM T95913 CY62VF 71452283 IC50 = 181 nM T95913 CQ7C5R 71452284 IC50 = 14 nM T95913 C6VF7J 71453206 IC50 = 63 nM T95913 CR84JX 71453419 Ki = 4 nM T95913 CZ61FJ 71454160 IC50 = 25.12 nM T95913 CZ8Q5P 71454238 Ki = 2.4 nM T95913 CF74SL 71454944 IC50 = 93 nM T95913 CO82IY 71455167 Ki = 21 nM T95913 CA7L1Y 71455168 Ki = 31 nM T95913 CSW47K 71455817 IC50 = 117 nM T95913 CT32GB 71455818 IC50 = 10 nM T95913 CE1IX7 71456728 IC50 = 59 nM T95913 CLUR84 71457607 IC50 = 12 nM T95913 C4ACV9 71457608 IC50 = 95 nM T95913 CM1ND2 71458573 IC50 = 82 nM T95913 C3S0NP 71458574 IC50 = 72 nM T95913 CY6WI2 71458575 IC50 = 60 nM T95913 C13KJV 71459500 IC50 = 250 nM T95913 CO8U5R 71459501 IC50 = 223 nM T95913 CL30DJ 71459502 IC50 = 346 nM T95913 C1Y8WD 71459503 IC50 = 12 nM T95913 CT7K3A 71460422 IC50 = 54 nM T95913 CW9YM2 71461240 IC50 = 3 nM T95913 CA2V9S 71461241 IC50 = 161 nM T95913 C65RJY 71461242 IC50 = 25 nM T95913 C2HOB7 71461243 IC50 = 3 nM T95913 CO26VM 71462973 IC50 = 24 nM T95913 CU3EO6 71520393 IC50 > 10000 nM T95913 CYC6S1 71520394 IC50 > 10000 nM T95913 C1KMX0 71520395 IC50 > 10000 nM T95913 CYK7N8 71520396 IC50 > 10000 nM T95913 CTC0O8 71520397 IC50 > 10000 nM T95913 C0UZ3D 71526877 IC50 = 2000 nM T95913 CP05SQ 71526878 IC50 = 100000 nM T95913 CZK6X9 71526879 IC50 > 10000 nM T95913 C8QRE4 71526880 IC50 > 10000 nM T95913 CT3QI8 71526881 IC50 > 10000 nM T95913 CO4MY1 71527005 IC50 > 10000 nM T95913 CJC64F 71527006 IC50 > 10000 nM T95913 C96WZG 71527007 IC50 = 3900 nM T95913 CUC7I1 71527008 IC50 = 8000 nM T95913 C09WKC 71527009 IC50 > 10000 nM T95913 CSPO76 71527716 IC50 > 5011.87 nM T95913 CIN7O1 71527842 IC50 > 6309.57 nM T95913 CO6CI7 71528725 IC50 = 9900 nM T95913 C5U2ZC 71528726 IC50 = 380 nM T95913 CTKO36 71528727 IC50 = 3600 nM T95913 C2KF3X 71533728 IC50 = 1046 nM T95913 CI7Q4K 71548718 IC50 = 2700 nM T95913 CED62L 71548719 IC50 = 9200 nM T95913 C4B0KN 71549093 IC50 = 20000 nM T95913 C6PRV1 71655831 IC50 = 12 nM T95913 CU48RN 71657825 IC50 = 154 nM T95913 CWG8M3 71682651 IC50 = 210 nM T95913 C6UGW3 71682652 IC50 = 4600 nM T95913 C7BX4K 71682653 IC50 = 930 nM T95913 CQX8N3 71682654 IC50 > 10000 nM T95913 CS32HB 71716798 IC50 > 6309.57 nM T95913 C07GCV 71716799 IC50 = 5011.87 nM T95913 CFW01E 71718034 IC50 = 2530 nM T95913 CXJC41 72188489 IC50 = 1000 nM T95913 C29KOU 72709209 IC50 > 10000 nM T95913 CT73IW 72709284 IC50 = 2500 nM T95913 CIL6S8 72737375 IC50 = 28 nM T95913 CTYJ25 72737376 IC50 = 158 nM T95913 CPL27S 72737377 IC50 = 52 nM T95913 C5RQB7 72737378 IC50 = 68 nM T95913 C8H7VT 72737379 IC50 = 121 nM T95913 CV2G1F 72737380 IC50 = 62 nM T95913 CHX84Q 72737381 IC50 = 7.2 nM T95913 CI5OT1 72737382 IC50 = 203 nM T95913 CSN5U8 72737551 IC50 = 17 nM T95913 CHC5J2 72737552 IC50 = 29 nM T95913 CB5PM9 72737553 IC50 = 68 nM T95913 CIF36E 72737554 IC50 = 57 nM T95913 C87HDL 72737555 IC50 = 100 nM T95913 CVU2J9 72949025 IC50 = 42 nM T95913 CC6KY3 72949203 IC50 = 16 nM T95913 CYGV85 73051332 IC50 = 5 nM T95913 CV4BH5 73051810 IC50 = 34 nM T95913 CE2IG4 73051811 IC50 = 271 nM T95913 CKUF15 73051812 IC50 = 4 nM T95913 CRF25X 73051813 IC50 = 12 nM T95913 C56JVH 73051977 IC50 = 67 nM T95913 C7N0AF 73052137 IC50 = 11 nM T95913 CNTD65 73052455 IC50 = 6 nM T95913 CZY9U8 73441896 IC50 = 31622.78 nM T95913 CL0XZ1 73659199 Ki = 2 nM T95913 CK7XM5 73659200 Ki = 1 nM T95913 C8EI1X 73673707 IC50 = 1.5 nM T95913 C0W1TK 73774799 IC50 = 120 nM T95913 C4W3IL 73774944 IC50 = 420 nM T95913 CH75QS 73774946 IC50 = 11 nM T95913 C5NKS4 73774948 IC50 = 40 nM T95913 C23MSN 73775105 IC50 = 160 nM T95913 CQG43I 73775546 IC50 = 3.3 nM T95913 CBXV38 73775549 IC50 = 3.1 nM T95913 C6O4PV 73775675 IC50 = 15 nM T95913 CQI4G9 73775798 IC50 = 81 nM T95913 CG0VK1 73775800 IC50 = 17 nM T95913 C7N0ME 73775931 IC50 = 3.6 nM T95913 CA5DJ3 73775934 IC50 = 13 nM T95913 CD6M4Q 73776065 IC50 = 10 nM T95913 C6X3LA 73776070 IC50 = 0.3 nM T95913 C5PKH6 73776209 IC50 = 430 nM T95913 C4WLT1 73776507 IC50 = 12 nM T95913 CPH39S 73776508 IC50 = 45 nM T95913 CT6ZB1 73776511 IC50 = 64 nM T95913 CI9K0J 73776652 IC50 = 0.7 nM T95913 CMHK83 73776786 IC50 = 0.6 nM T95913 CMT13V 73776787 IC50 = 6.8 nM T95913 CBYN18 73977439 IC50 = 1995 nM T95913 C9V1YR 73977449 IC50 = 251 nM T95913 CXA90D 73977451 IC50 = 316 nM T95913 CEZ7L2 73977461 IC50 = 126 nM T95913 CD0T9V 74539799 IC50 = 0.74 nM T95913 C16KOS 74539862 IC50 = 1.1 nM T95913 CN2MI8 76310247 IC50 > 50000 nM T95913 CKO41J 76310248 IC50 = 741 nM T95913 CEN9Q5 76310249 IC50 > 50000 nM T95913 CJCF67 76310250 IC50 = 26 nM T95913 CBF70W 76310805 IC50 = 316.23 nM T95913 CA2VR6 76311340 IC50 = 194.98 nM T95913 CMR07I 76313939 IC50 > 50000 nM T95913 C5P2CJ 76313940 IC50 = 30700 nM T95913 CAV5Q9 76313941 IC50 = 22000 nM T95913 CO13XZ 76314937 IC50 = 386 nM T95913 C7W2HI 76314938 IC50 = 341.98 nM T95913 C6H9EL 76314939 IC50 = 230.99 nM T95913 C0J6PL 76317466 IC50 > 50000 nM T95913 CVW35P 76317467 IC50 > 50000 nM T95913 CZ1T3C 76317468 IC50 > 50000 nM T95913 C4MKN3 76317469 IC50 = 62 nM T95913 C3JA4F 76317470 IC50 = 353 nM T95913 C4XJ5Y 76317471 IC50 = 153 nM T95913 CS6ME5 76318566 IC50 = 235 nM T95913 CG4I2R 76318567 IC50 = 217 nM T95913 C8E4GI 76321204 IC50 = 183 nM T95913 CF4OI8 76321205 IC50 = 12300 nM T95913 C1YFK9 76322218 IC50 = 267.98 nM T95913 CL0T7B 76322219 IC50 <= 65 nM T95913 CDG8V4 76324821 IC50 = 87 nM T95913 CJW39V 76324822 IC50 > 50000 nM T95913 C2BFA1 76324823 IC50 = 4700 nM T95913 CM4N8A 76325342 IC50 = 6309.57 nM T95913 C92ZAB 76325343 IC50 = 25118.86 nM T95913 C1HFI9 76325446 IC50 = 3259 nM T95913 C4GZ1Q 76325833 IC50 = 357.03 nM T95913 CQ31CA 76325834 IC50 = 312.97 nM T95913 C4A8XZ 76328376 IC50 = 3400 nM T95913 C39CLE 76329428 IC50 = 247 nM T95913 CYR0G6 76332050 IC50 = 6300 nM T95913 C4MID5 76332051 IC50 = 7880 nM T95913 C70WJE 76332052 IC50 = 79 nM T95913 CQ8YC1 76332568 IC50 = 7.943 nM T95913 CE6BI0 76332666 IC50 = 4350 nM T95913 C16SRX 76333068 IC50 = 143 nM T95913 CW81MC 76333069 IC50 = 264.97 nM T95913 C26CKL 76333070 IC50 = 153.99 nM T95913 C47NLT 76333071 IC50 = 250 nM T95913 CN38BK 76335378 IC50 = 81 nM T95913 C69ATM 76335666 IC50 > 50000 nM T95913 C0SI4C 76335667 IC50 > 50000 nM T95913 C31NEK 76335668 IC50 = 574 nM T95913 CL6BV5 76335669 IC50 > 50000 nM T95913 C73KJD 76335670 IC50 = 227 nM T95913 CY3LO5 76336173 IC50 = 1258.93 nM T95913 CJ3V6Y 76336695 IC50 = 274 nM T95913 CD03GB 76336696 IC50 = 277.97 nM T95913 C2JTH8 77107528 IC50 = 112 nM T95913 C42HDP 77107927 IC50 = 42 nM T95913 C04SRC 77147259 IC50 = 1774 nM T95913 C9I7TY 78319187 IC50 = 1584.89 nM T95913 C24LQH 78320362 IC50 = 35 nM T95913 C9T8KF 78320671 IC50 = 70 nM T95913 CI2YN8 78320672 IC50 = 24 nM T95913 CI6K4J 78320673 IC50 = 305 nM T95913 COFJ16 78320996 IC50 = 5200 nM T95913 CMU5P2 78321310 IC50 = 150 nM T95913 CE13AJ 78321314 IC50 = 200 nM T95913 CSP2H4 78321635 IC50 = 280 nM T95913 CWA0B1 78322567 IC50 = 140 nM T95913 CH6P9D 78322877 IC50 > 10000 nM T95913 C4IW9V 78323193 IC50 = 230 nM T95913 CD1JC8 78324443 IC50 = 129 nM T95913 C04IKP 86268622 IC50 = 28 nM T95913 C5P3RO 86647783 IC50 = 1200 nM T95913 CDXM47 86677874 IC50 > 10000 nM T95913 CP3W1B 86695297 IC50 > 20000 nM T95913 CA17UE 86732669 IC50 = 4630 nM T95913 C2PCS7 87061302 IC50 = 181 nM T95913 CNVS32 87343636 Ki = 16.7 nM T95913 CV6PI8 87562294 IC50 = 125.89 nM T95913 CZ2AU4 87570781 IC50 = 375 nM T95913 C3HD5O 88570842 Ki = 9 nM T95913 CLEX32 89034287 Ki = 4 nM T95913 C1AKZ4 89034365 Ki = 6 nM T95913 CEQ80V 89034380 Ki = 5 nM T95913 C1HB3F 89051931 IC50 = 330 nM T95913 C61SCX 89493851 IC50 = 5 nM T95913 C1LU3X 89493904 IC50 = 31 nM T95913 CTE1L0 89517065 IC50 = 9300 nM T95913 C56KSC 89517226 IC50 > 10000 nM T95913 C6M0QF 89841854 IC50 = 400 nM T95913 C61GIO 89841941 IC50 = 40 nM T95913 C6FI0A 89842032 IC50 = 110 nM T95913 COL45N 89842055 IC50 = 60 nM T95913 C7FNP8 89842123 IC50 = 25 nM T95913 CF50MO 89842136 IC50 = 1100 nM T95913 C6CKP2 89842150 IC50 = 50 nM T95913 CVZH15 89842186 IC50 = 240 nM T95913 C2LQ9V 89842220 IC50 = 150 nM T95913 C83SXM 89842240 IC50 = 1100 nM T95913 CQ1U2Y 89842245 IC50 = 1000 nM T95913 CQO85K 89842249 IC50 > 7000 nM T95913 CX70NQ 89842250 IC50 = 14 nM T95913 CN5Y9A 90064110 IC50 = 27 nM T95913 C7FP2M 90064111 IC50 = 4 nM T95913 CN51BK 90064299 IC50 = 2 nM T95913 CUZ13D 90102336 IC50 = 0.7 nM T95913 CQO9J0 90103194 IC50 = 1.7 nM T95913 C28WQY 90431726 IC50 = 20 nM T95913 C08UWK 90665816 IC50 = 100000 nM T95913 CMWB58 91757958 IC50 <= 10000 nM T95913 C3Y0DS 91801158 IC50 = 2.6 nM T95913 CAS7W6 91864650 IC50 = 8440 nM T95913 CA3ZC1 92172785 IC50 = 575000 nM T95913 C4JMV1 118003503 IC50 = 330 nM T95913 C6YRW7 118003617 IC50 = 110 nM T95913 C8QHY9 118003714 IC50 = 75 nM T95913 CLDA15 118003719 IC50 = 360 nM T95913 C5LW9G 118004010 IC50 = 100 nM T95913 CK0W1T 118004012 IC50 = 170 nM T95913 C0BIP8 118004016 IC50 = 350 nM T95913 CB4PM3 118004022 IC50 = 110 nM T95913 CNCK58 118004064 IC50 = 280 nM T95913 C14WCU 118131317 IC50 > 1000 nM T95913 C67VQE 118341819 IC50 = 850 nM T95913 CC9P5H 118341835 IC50 = 750 nM T95913 CUMA23 118341844 IC50 = 1840 nM T95913 C3IP9X 118341852 IC50 = 190 nM T95913 C6TI0Z 118341865 IC50 = 520 nM T95913 C4U7NC 118341870 IC50 = 360 nM T95913 CVL03K 118341884 IC50 = 1370 nM T95913 CPZN96 118341923 IC50 = 150 nM T95913 C9E3DU 118341927 IC50 = 6950 nM T95913 CVN87P 118433737 IC50 = 36 nM T95913 C8W1RN 118445922 IC50 = 7 nM T95913 CGYA58 118445928 IC50 = 182 nM T95913 CL29BI 118445929 IC50 = 52 nM T95913 CI24WZ 118445978 IC50 = 3 nM T95913 CA20CO 118445983 IC50 = 13 nM T95913 CQF1V4 118446049 IC50 = 4 nM T95913 C90OAT 118446064 IC50 = 43 nM T95913 CJQ92T 118572891 IC50 < 10 nM T95913 CVY45K 118575373 IC50 > 10000 nM T95913 CS20UM 118575423 IC50 > 10000 nM T95913 CCPV26 118575517 IC50 = 632 nM T95913 C0L9JQ 118575526 IC50 = 1300 nM T95913 CH6AB7 118575540 IC50 > 10000 nM T95913 C97QIN 118575555 IC50 = 990 nM T95913 CEDC48 118575654 IC50 = 3466 nM T95913 COYJ84 118575663 IC50 > 10000 nM T95913 CS1Z8W 118575682 IC50 = 4407 nM T95913 CC0S4G 118575689 IC50 = 199 nM T95913 C6X8HG 118575694 IC50 > 10000 nM T95913 CUJ30I 118575784 IC50 = 1247 nM T95913 CAT54V 118575791 IC50 = 1277 nM T95913 C1K6HU 118575835 IC50 = 4262 nM T95913 C2OQ4U 118575893 IC50 > 10000 nM T95913 C6HEA7 118575940 IC50 = 990 nM T95913 CIU7J3 118575971 IC50 = 267 nM T95913 CAD39P 118575986 IC50 = 4150 nM T95913 CCYI54 118576050 IC50 = 1131 nM T95913 CW9T6F 118576060 IC50 = 7836 nM T95913 C7Y4AT 118576103 IC50 > 10000 nM T95913 C47WMX 118576166 IC50 = 7989 nM T95913 C1UT8B 118576192 IC50 > 10000 nM T95913 C0F7JV 118576207 IC50 = 2311 nM T95913 CU61WD 118576212 IC50 > 10000 nM T95913 CE3V8W 118576268 IC50 = 54 nM T95913 CO0YC8 118616775 IC50 = 1 nM T95913 CS5C8W 118684133 IC50 = 4.3 nM T95913 CRX24W 118709077 IC50 = 6000 nM T95913 CV2EJ7 118709081 IC50 = 6900 nM T95913 CZ41AQ 118709092 IC50 = 83000 nM T95913 CR6ML1 118709578 IC50 = 670 nM T95913 C0OH7I 118709579 IC50 = 13500 nM T95913 C73YIO 118709582 IC50 = 3000 nM T95913 CGWX02 118709583 IC50 = 510 nM T95913 CY2QG0 118711873 IC50 = 10890 nM T95913 CH4XY2 118711874 IC50 = 10710 nM T95913 C94GZM 118712046 IC50 = 3600 nM T95913 CPXQ86 118721834 Ki = 44 nM T95913 CH9D8G 118721835 Ki = 19 nM T95913 CYHG95 118721836 Ki = 21 nM T95913 CP6SR7 118721837 Ki = 9 nM T95913 CW4N7Q 118721838 Ki = 7 nM T95913 CZG78A 118721839 Ki = 190 nM T95913 C2BQS3 118721840 Ki = 6 nM T95913 C2T9RN 118721841 Ki = 1 nM T95913 C6GJ0Q 118721842 Ki = 7 nM T95913 C9RPN4 118721843 Ki = 2 nM T95913 CYNZ53 118721844 Ki = 22 nM T95913 C5R1VP 118721845 Ki = 19 nM T95913 CB53EU 118728320 IC50 = 34624 nM T95913 C6KJL1 118728321 IC50 = 21668 nM T95913 CKJ3S6 118728322 IC50 = 27916 nM T95913 CT0L3Y 118728325 IC50 = 24342 nM T95913 CHS2E4 118728326 IC50 = 11812 nM T95913 CRUP47 118728328 IC50 = 44117 nM T95913 CQR41G 118728330 IC50 = 19479 nM T95913 CN4Q9R 118728332 IC50 = 9443 nM T95913 CDI10F 118728336 IC50 = 41626 nM T95913 CHT6K9 118728811 Ki = 2900 nM T95913 CUA3Y2 118728812 Ki > 4000 nM T95913 CDQ78G 118728813 Ki = 400 nM T95913 CZ6XL7 118728814 Ki = 630 nM T95913 CMO67K 118728815 Ki = 750 nM T95913 CR2M0Q 118728816 Ki = 1500 nM T95913 C62SCL 118728817 Ki = 690 nM T95913 CSB30C 118728819 Ki = 1100 nM T95913 CV7XU8 118728820 Ki = 710 nM T95913 C3J1EX 118728821 Ki > 4000 nM T95913 CIWB78 118728822 Ki > 4000 nM T95913 CP18SE 118728823 Ki = 780 nM T95913 CM42CA 118728824 Ki = 1400 nM T95913 C9Q7CL 118728825 Ki = 2800 nM T95913 CCR3S0 118728826 Ki = 1200 nM T95913 CB1WC5 118729946 IC50 = 380 nM T95913 CQ4G9M 118729947 IC50 = 1600 nM T95913 C43IPJ 118729948 IC50 = 250 nM T95913 C3I9CQ 118729949 IC50 = 510 nM T95913 CZQ17M 118729950 IC50 = 200 nM T95913 C3G1ZP 118729951 IC50 = 4950 nM T95913 CY60FC 118730033 IC50 = 17087 nM T95913 CN3B4U 118730711 IC50 = 320 nM T95913 C0IL3N 118730712 IC50 = 1400 nM T95913 C3CH1A 118730713 IC50 = 350 nM T95913 CHX5L9 118730714 IC50 = 250 nM T95913 CNJ32C 118730715 IC50 = 3200 nM T95913 C1MKB3 118730716 IC50 = 1400 nM T95913 C81RJA 118730717 IC50 = 13000 nM T95913 CFZ16R 118737301 IC50 <= 10000 nM T95913 C27CPQ 118737302 IC50 <= 10000 nM T95913 C59VXA 118737303 IC50 <= 10000 nM T95913 CGO1N4 118737304 IC50 <= 10000 nM T95913 CS85FM 118737305 IC50 <= 10000 nM T95913 C8UCO1 118737306 IC50 <= 10000 nM T95913 CR0BZ2 118737307 IC50 <= 10000 nM T95913 C3N4DJ 118737308 IC50 <= 10000 nM T95913 CGY5B1 118737309 IC50 <= 10000 nM T95913 CV85EL 118981804 IC50 = 38 nM T95913 C91PVZ 121428416 IC50 = 204 nM T95913 CA2DM0 121428489 IC50 = 164 nM T95913 CQLX36 121428567 IC50 = 288 nM T95913 CFN12W 121445751 IC50 = 28 nM T95913 C04NDW 121445810 IC50 = 41 nM T95913 C81IFQ 122163152 IC50 = 1340 nM T95913 C2VGD5 122178120 IC50 = 21.1 nM T95913 C24XUZ 122178124 IC50 = 10.2 nM T95913 CN5AB3 122179486 IC50 = 4.4 nM T95913 CLEK13 122179487 IC50 = 10 nM T95913 C0OW8H 122179490 IC50 = 52 nM T95913 C0VD5F 122179491 IC50 = 2 nM T95913 CQ87FB 122179492 IC50 = 4 nM T95913 CBJ29X 122179493 IC50 > 10000 nM T95913 CA5N1B 122179494 IC50 = 25 nM T95913 CM4AW9 122180514 Ki = 0.024 nM T95913 CM89OL 122180515 Ki = 0.016 nM T95913 CU0C1D 122180516 Ki = 0.01 nM T95913 CB6PR7 122180517 Ki = 0.034 nM T95913 CQ63DW 122180518 Ki = 0.006 nM T95913 C9N8JT 122180519 Ki = 0.003 nM T95913 C42GSX 122180520 Ki = 0.002 nM T95913 CVA3P2 122180521 Ki = 0.009 nM T95913 C0A7CQ 122180522 Ki = 0.025 nM T95913 CEFS13 122180793 IC50 = 91560 nM T95913 CFZ2E1 122180794 IC50 = 125800 nM T95913 C5YKG7 122180795 IC50 = 465500 nM T95913 C9ID7U 122180796 IC50 = 345900 nM T95913 C08XOC 122180839 IC50 = 781500 nM T95913 C2HM6P 122180840 IC50 = 967700 nM T95913 CT9Y6U 122180841 IC50 = 23640 nM T95913 C6FOM0 122180842 IC50 = 18480 nM T95913 COX90L 122180843 IC50 = 12570 nM T95913 CP40RU 122180844 IC50 = 26870 nM T95913 CC0EK9 122180845 IC50 = 15560 nM T95913 CS85CU 122181413 IC50 = 280 nM T95913 CQS67B 122181416 IC50 = 650 nM T95913 C58XRY 122184465 IC50 = 1995.26 nM T95913 C16ALM 122184466 IC50 = 1000 nM T95913 CDZY02 122184468 IC50 = 50118.72 nM T95913 CTH70U 122184469 IC50 = 12589.25 nM T95913 C9ZXR7 122184470 IC50 = 3981.07 nM T95913 CNJ9Z4 122184471 IC50 = 3981.07 nM T95913 CS41EG 122184473 IC50 = 1258.93 nM T95913 CZ36GL 122184474 IC50 = 1000 nM T95913 CU4ZT6 122184475 IC50 = 10000 nM T95913 C3H9PR 122184476 IC50 = 1258.93 nM T95913 CU40TW 122184477 IC50 = 3162.28 nM T95913 CAMD31 122184479 IC50 = 19952.62 nM T95913 C1F9RK 122184480 IC50 = 251.19 nM T95913 C7XW1K 122184481 IC50 = 12589.25 nM T95913 CRUX54 122184482 IC50 = 31622.78 nM T95913 CQ7W0P 122184526 IC50 = 3981.07 nM T95913 CA5YB2 122184529 IC50 = 2511.89 nM T95913 C64YPH 122184530 IC50 = 2511.89 nM T95913 C4AGX5 122184531 IC50 = 3162.28 nM T95913 CQL4K5 122184532 IC50 = 1584.89 nM T95913 CRKV74 122184533 IC50 = 3981.07 nM T95913 CX14YD 122184534 IC50 = 1000 nM T95913 CM6A4S 122184535 IC50 = 1258.93 nM T95913 CF86YS 122184536 IC50 = 1995.26 nM T95913 CYRH97 122184538 IC50 = 3162.28 nM T95913 CD4W0Z 122184539 IC50 = 10000 nM T95913 CH8Y3Q 122184540 IC50 = 15848.93 nM T95913 CDA85R 122184541 IC50 = 63095.73 nM T95913 CF36XJ 122184542 IC50 > 199526.23 nM T95913 CQ6O7H 122184543 IC50 = 50118.72 nM T95913 CS4MN0 122184544 IC50 = 10000 nM T95913 CKT74G 122185265 IC50 = 14 nM T95913 CJ6C1O 122185267 IC50 = 22 nM T95913 CGW35U 122387497 IC50 = 259 nM T95913 C38BML 122387499 IC50 = 265 nM T95913 CCW0M1 122387500 IC50 = 174 nM T95913 CKA90Y 122387501 IC50 = 89 nM T95913 CH4LC6 122387502 IC50 = 56 nM T95913 C8OC3E 122387504 IC50 = 169 nM T95913 C34AHY 122387505 IC50 = 185 nM T95913 CUG1T6 122387506 IC50 = 98 nM T95913 CE7K5C 122387507 IC50 = 173 nM T95913 C4HL3N 122387508 IC50 = 111 nM T95913 CA7L3S 122387509 IC50 = 112 nM T95913 CR9NF3 122542400 IC50 = 5.7 nM T95913 CZE35C 122648343 IC50 > 10000 nM T95913 C54RNT 122648367 IC50 > 10000 nM T95913 C1UVI7 122648600 IC50 = 255 nM T95913 CMX59K 122648648 IC50 = 8.1 nM T95913 CVZ64I 122648649 IC50 > 10000 nM T95913 CPTY78 124518210 IC50 = 89 nM T95913 CB7G5E 126476620 IC50 = 501.19 nM T95913 C74BNR 126480568 IC50 = 1584.89 nM T95913 C1N6YP 126480569 IC50 = 2511.89 nM T95913 CE52HC 126480570 IC50 = 630.96 nM T95913 CQ74WU 126480571 IC50 = 3981.07 nM T95913 C0AFE2 126480572 IC50 = 1000 nM T95913 C3E7JB 126480573 IC50 = 6309.57 nM T95913 CPW54V 126480574 IC50 = 1000 nM T95913 CVJ3Q5 127025094 IC50 = 285 nM T95913 C2E4LO 127025141 IC50 = 6570 nM T95913 CO94KJ 127025144 IC50 > 25000 nM T95913 CKO53P 127025146 IC50 = 21450 nM T95913 CF7H0V 127025161 IC50 = 1260 nM T95913 CE4C3J 127025163 IC50 = 12360 nM T95913 CAV24Z 127025164 IC50 = 9360 nM T95913 C98DKI 127025346 IC50 = 4 nM T95913 CDZ56M 127025449 IC50 > 25000 nM T95913 CBXJ67 127025628 IC50 = 2.7 nM T95913 CH2Q7A 127027634 IC50 = 280 nM T95913 CSV3R7 127029064 IC50 = 64 nM T95913 CQTG79 127029604 IC50 = 279 nM T95913 CZHT45 127031017 IC50 = 3700 nM T95913 CU0F4R 127031332 IC50 = 1500 nM T95913 C2IN4Q 127031333 IC50 > 50000 nM T95913 CS12RU 127031435 IC50 = 2.3 nM T95913 CGU4H3 127031891 IC50 = 21 nM T95913 CGKR53 127032915 IC50 = 502 nM T95913 C41YQI 127035981 IC50 = 939 nM T95913 C7V4WA 127036623 IC50 = 13780 nM T95913 CJ1LH4 127036935 IC50 = 3120 nM T95913 CG8DA9 127045861 IC50 = 99 nM T95913 CVF8Z9 127045862 IC50 = 5 nM T95913 CH68NT 127046076 IC50 = 77 nM T95913 CA2XD5 127046077 IC50 = 230 nM T95913 COJ68G 127046117 IC50 = 1900 nM T95913 C34REM 127046317 IC50 = 570 nM T95913 CC4ND8 127046862 IC50 = 302 nM T95913 CY2P1X 127047138 IC50 = 440 nM T95913 CZ2R0C 127047140 IC50 = 120 nM T95913 CT89GI 127047683 IC50 = 720 nM T95913 C7D0FN 127047685 IC50 = 240 nM T95913 CN94CQ 127047797 IC50 = 140 nM T95913 C3IC2Z 127052212 IC50 = 5803 nM T95913 CN9XL1 129262531 IC50 = 90 nM T95913 CW7A5X 129626595 IC50 = 3981.07 nM T95913 C18NHD 130302549 IC50 <= 10000 nM T95913 CL13RZ 130302558 IC50 <= 10000 nM T95913 CF5JZ3 130302563 IC50 <= 10000 nM T95913 CD46EL 130302605 IC50 <= 10000 nM T95913 CNI8M6 130302620 IC50 <= 10000 nM T95913 CI6WN9 130302651 IC50 <= 10000 nM T95913 C5ZP0L 130302658 IC50 <= 10000 nM T95913 CW61SG 130302663 IC50 <= 10000 nM T95913 CB27ZG 130302668 IC50 <= 10000 nM T95913 C5VYM6 130302674 IC50 <= 10000 nM T95913 C0FQR2 130302675 IC50 <= 10000 nM T95913 CB34HQ 130302676 IC50 <= 10000 nM T95913 CQR1I8 130302685 IC50 <= 10000 nM T95913 C17DZF 130302698 IC50 <= 10000 nM T95913 CBC6W7 130302701 IC50 <= 10000 nM T95913 CBT21G 130302702 IC50 <= 10000 nM T95913 CDZ45O 130302703 IC50 <= 10000 nM T95913 C2GWU8 130302709 IC50 <= 10000 nM T95913 CV3M6Y 130302710 IC50 <= 10000 nM T95913 C39UQN 130302731 IC50 <= 10000 nM T95913 CL9O8X 130302732 IC50 <= 10000 nM T95913 CL69GM 130302740 IC50 <= 10000 nM T95913 CH8YK9 130302741 IC50 <= 10000 nM T95913 CQR2W9 130302781 IC50 <= 10000 nM T95913 C9HC8A 130302803 IC50 <= 10000 nM T95913 CIK25W 130302809 IC50 <= 10000 nM T95913 CI08PF 130332501 IC50 <= 10000 nM T95913 C1H4UT 130332505 IC50 <= 10000 nM T95913 CZPI64 130332579 IC50 <= 10000 nM T95913 CDS9F3 130332582 IC50 <= 10000 nM T95913 C3G0HF 130332585 IC50 <= 10000 nM T95913 CX13UC 130332620 IC50 <= 10000 nM T95913 CED6F3 130332657 IC50 <= 10000 nM T95913 C73KWM 130338615 IC50 = 100 nM T95913 CLC06T 130406587 IC50 = 1 nM T95913 C47CAY 130421765 IC50 = 0.631 nM T95913 C84YKI 130422161 IC50 = 0.7943 nM T95913 C2MVE6 130422162 IC50 = 0.631 nM T95913 CK68CA 130453737 IC50 = 3000 nM T95913 CUO41K 130470684 IC50 = 7100 nM T95913 CDE7T3 132005217 IC50 = 49 nM T95913 CL26YS 132005219 IC50 = 310 nM T95913 CP32GB 132005220 IC50 = 15 nM T95913 CG1NC4 132005221 IC50 = 3300 nM T95913 C0UV2M 132005224 IC50 = 58 nM T95913 CUN18W 132005225 IC50 = 6.5 nM T95913 CD84OI 132005228 IC50 = 2.8 nM T95913 C9VDI0 132005229 IC50 = 110 nM T95913 CB1Z7P 132005231 IC50 = 340 nM T95913 C7ASP9 132005246 IC50 = 11 nM T95913 C8VE6T 132005248 IC50 = 560 nM T95913 C7LCW1 132005249 IC50 = 110 nM T95913 C5W9LN 132005323 IC50 = 120 nM T95913 CQ6GO2 132005326 IC50 = 330 nM T95913 C6OXE3 132134663 IC50 = 10 nM T95913 C4M8WN 132209922 IC50 = 1.3 nM T95913 CFI23B 132210082 IC50 = 21 nM T95913 C8RK4V 132218631 IC50 = 300 nM T95913 CZD9F3 132219135 IC50 > 10000 nM T95913 CH8DP7 132220479 IC50 = 41 nM T95913 C4Q5LF 132471857 IC50 = 10 nM T95913 CJE34F 132597748 IC50 = 3220 nM T95913 CCV46G 132606879 IC50 = 199.53 nM T95913 CT2PN8 132990561 IC50 = 75 nM T95913 CFG90E 134132909 IC50 = 642 nM T95913 CI49TK 134133218 IC50 = 65 nM T95913 C4YNH0 134134126 IC50 = 698 nM T95913 C0EK8P 134134680 IC50 = 828 nM T95913 C0A1UM 134138053 IC50 = 282 nM T95913 CQ2S4X 134138703 IC50 > 9100 nM T95913 CL3Q6G 134140420 IC50 = 1210 nM T95913 CDJ10M 134142931 IC50 = 1230 nM T95913 CUE85S 134143151 IC50 > 50000 nM T95913 CQ9G7H 134145670 IC50 = 220 nM T95913 C6G8EJ 134146051 IC50 = 40000 nM T95913 CIPL93 134147099 IC50 = 2070 nM T95913 C8ITR3 134147904 IC50 > 50000 nM T95913 CXA3V0 134148445 IC50 = 3780 nM T95913 CXU92M 134150578 IC50 = 366 nM T95913 CG8LE2 134151667 IC50 < 10000 nM T95913 CK43EY 134152988 IC50 = 2940 nM T95913 CS2QP7 134154582 IC50 = 194 nM T95913 C2QGB3 134156160 IC50 = 978 nM T95913 C42RJH 134157534 IC50 = 5859 nM T95913 C9C3XT 134163708 IC50 = 0.631 nM T95913 CD9ZR6 134372929 IC50 = 440 nM T95913 CCS6I3 134372959 IC50 = 4156 nM T95913 CTD03Q 134611885 IC50 >= 199.53 nM T95913 CJXA12 134611894 IC50 <= 0.7943 nM T95913 CX0UR7 134694318 IC50 > 1000 nM T95913 C6LYD2 135121892 IC50 = 63.1 nM T95913 C9FUK2 135151360 IC50 = 52 nM T95913 CT0GQ6 135197577 IC50 = 1.7 nM T95913 C87VKA 135197594 IC50 = 0.93 nM T95913 C0YK5W 135197617 IC50 = 1.6 nM T95913 CF6DJ2 135197621 IC50 = 2.1 nM T95913 CDT25A 135197623 IC50 = 1.5 nM T95913 CQXS07 135197635 IC50 = 1.2 nM T95913 C7KXF1 135197643 IC50 = 1.3 nM T95913 CY38TL 135391000 IC50 = 89.7 nM T95913 COG86Z 135397763 IC50 = 3162.28 nM T95913 CWL67T 135397764 IC50 = 1000 nM T95913 CX8AI4 135398491 IC50 = 180 nM T95913 CQN49C 135409495 IC50 = 4000 nM T95913 C6AZ2R 135435018 IC50 > 25118.86 nM T95913 CMGY62 135485500 IC50 = 273 nM T95913 CM9NV6 135492341 IC50 = 1200 nM T95913 CWJQ64 135492555 IC50 = 968 nM T95913 C3QJ8W 135566371 IC50 = 20 nM T95913 C24ZGX 135566644 IC50 > 10000 nM T95913 C2QDV5 135566741 IC50 > 10000 nM T95913 CTJ6B2 135610083 IC50 = 5900 nM T95913 CN2ME4 135610084 IC50 = 4700 nM T95913 C4G6JF 135610087 IC50 = 5100 nM T95913 CPV59N 135685787 Ki = 1000 nM T95913 C2UN0D 135742360 IC50 > 83300 nM T95913 CI98OY 135750190 IC50 = 195 nM T95913 CF0VL3 135750206 IC50 = 48000 nM T95913 CY4CZ0 135750219 IC50 = 1300 nM T95913 CU29YK 135750268 IC50 = 680 nM T95913 C02PHA 135927892 IC50 > 25118.86 nM T95913 CS8T3D 135927897 IC50 = 5011.87 nM T95913 CF1PS8 135934877 Ki = 1300 nM T95913 C12UDA 135947972 IC50 = 187 nM T95913 CN42ZS 135947973 IC50 = 1500 nM T95913 CF8AO3 135947974 IC50 = 118 nM T95913 CW08GJ 135947976 IC50 = 89 nM T95913 C8O9HG 135947977 IC50 = 50000 nM T95913 CJN7E2 135947978 IC50 = 190 nM T95913 CFKH34 135947979 IC50 = 587 nM T95913 C58FHM 135961523 IC50 = 6918.31 nM T95913 CTRL59 135976660 Ki = 540 nM T95913 C9OAV5 135986100 IC50 = 100000 nM T95913 C3USL8 135986101 IC50 > 100000 nM T95913 C4G2HP 135995897 IC50 = 5780 nM T95913 CNF15Q 135995898 IC50 = 1340 nM T95913 C98HZG 135995899 IC50 = 7640 nM T95913 CIQ82W 135995900 IC50 = 4560 nM T95913 CP1US5 136041737 IC50 = 7070 nM T95913 CXH63V 136041747 IC50 > 10000 nM T95913 C6B5TC 136041748 IC50 > 10000 nM T95913 CU6XG1 136041749 IC50 > 10000 nM T95913 C0U5DB 136041750 IC50 > 10000 nM T95913 C48KAQ 136041752 IC50 > 10000 nM T95913 C74PRL 136041753 IC50 > 10000 nM T95913 CT4FJ1 136041757 IC50 = 10000 nM T95913 CCS2G6 136041761 IC50 > 10000 nM T95913 CEZP21 136041762 IC50 > 10000 nM T95913 CJ58TD 136041764 IC50 > 10000 nM T95913 CX67QW 136041765 IC50 > 10000 nM T95913 CK0H2Q 136041766 IC50 > 10000 nM T95913 CQP7B6 136041767 IC50 > 10000 nM T95913 CM65BS 136041773 IC50 = 8270 nM T95913 C6P7JB 136041775 IC50 > 10000 nM T95913 C5CJF7 136041776 IC50 > 10000 nM T95913 C3XIZ8 136041777 IC50 > 10000 nM T95913 C32LKO 136041785 IC50 > 10000 nM T95913 C90ARP 136041787 IC50 > 10000 nM T95913 CZ3BN1 136041792 IC50 = 6215 nM T95913 CG19DI 136041799 IC50 > 10000 nM T95913 CXJA29 136041804 IC50 = 10000 nM T95913 CHT31V 136041805 IC50 = 1590 nM T95913 CO8C4J 136041817 IC50 = 3315 nM T95913 C4QU6G 136041827 IC50 = 10000 nM T95913 CNE10X 136041834 IC50 = 10000 nM T95913 CS3AE1 136041847 IC50 > 10000 nM T95913 CZC47Y 136041848 IC50 > 10000 nM T95913 C7PHA5 136044403 IC50 = 60 nM T95913 CLA3C2 136068720 IC50 = 96.5 nM T95913 CA91JG 136069599 IC50 = 1532 nM T95913 CGAB91 136069600 IC50 = 7418 nM T95913 C3ZAW2 136069605 IC50 = 8400 nM T95913 C8JXL5 136069609 IC50 = 1000 nM T95913 C9I0EQ 136069610 IC50 = 8966 nM T95913 C25EYJ 136069611 IC50 = 2461 nM T95913 C2S5QF 136069615 IC50 = 10000 nM T95913 CI1LY8 136096349 IC50 = 60 nM T95913 CC4UM3 136176116 IC50 > 10000 nM T95913 CJRK81 136176117 IC50 > 10000 nM T95913 C63IOS 136176118 IC50 > 10000 nM T95913 C3KW7H 136176119 IC50 > 10000 nM T95913 C69AKQ 136176120 IC50 > 10000 nM T95913 CF17KO 136176121 IC50 > 10000 nM T95913 CU3TE0 136176122 IC50 = 3333 nM T95913 C3X5KE 136176124 IC50 > 10000 nM T95913 CA8C5E 136176125 IC50 > 10000 nM T95913 C5OMG2 136176126 IC50 > 10000 nM T95913 CP2YM7 136176127 IC50 > 10000 nM T95913 C8XIJ0 136176128 IC50 = 5742 nM T95913 CUY8N4 136176129 IC50 > 10000 nM T95913 C3J4ME 136176130 IC50 > 10000 nM T95913 CR1NZ2 136176131 IC50 > 10000 nM T95913 C4WG2F 136176132 IC50 > 10000 nM T95913 CJ8EC5 136176139 IC50 > 10000 nM T95913 CQ84IZ 136180335 Ki > 4000 nM T95913 C1LK9U 136183381 IC50 = 3975 nM T95913 C27TKQ 136196449 IC50 = 10000 nM T95913 CHF3R5 136200721 IC50 = 4810 nM T95913 CV2X9O 136200837 IC50 = 3690 nM T95913 CK9S4X 136229137 IC50 = 18500 nM T95913 C7S1YJ 136230225 IC50 > 10000 nM T95913 C3Q6ED 136230226 IC50 > 10000 nM T95913 CKPF02 136230227 IC50 > 10000 nM T95913 CZY9O0 136230228 IC50 = 5090 nM T95913 CRET01 136230229 IC50 > 10000 nM T95913 CX1KI8 136230230 IC50 > 10000 nM T95913 C3Z5MH 136230231 IC50 > 10000 nM T95913 CUE6N8 136230232 IC50 = 8010 nM T95913 C8Q1AP 136230233 IC50 = 6710 nM T95913 C70RXE 136230234 IC50 > 10000 nM T95913 C4W0KN 136230235 IC50 = 6610 nM T95913 CMZN01 136230236 IC50 > 10000 nM T95913 CCU0H5 136241428 IC50 = 1780 nM T95913 C75RWX 136244223 IC50 = 7410 nM T95913 CXI04C 136244224 IC50 = 6480 nM T95913 C0YW6L 136244283 IC50 = 1340 nM T95913 CF3DK1 136245085 IC50 = 9360 nM T95913 CEU87Z 136245089 IC50 = 10000 nM T95913 CUF56H 136245251 IC50 = 2170 nM T95913 CKPR81 136245252 IC50 = 7120 nM T95913 C7C5ZV 136249323 IC50 = 2600 nM T95913 CI6HG4 136249373 IC50 = 264 nM T95913 CL4MO3 136249382 IC50 = 10000 nM T95913 C68CRX 136254271 IC50 = 2870 nM T95913 C0GZV9 136254283 IC50 > 10000 nM T95913 CMWA86 136264282 IC50 = 9149 nM T95913 CSD78N 136264452 IC50 = 6390 nM T95913 C1HI5T 136264454 IC50 = 1131 nM T95913 CV3UE9 137333450 IC50 = 202.7 nM T95913 CH8WU5 137348751 IC50 = 12.59 nM T95913 CP34TI 137631388 IC50 = 130 nM T95913 CF0PQ2 137632018 IC50 > 794.33 nM T95913 CZ4WN6 137633048 Ki = 66.7 nM T95913 CIX4S7 137633081 IC50 = 630.96 nM T95913 CR17XH 137634463 IC50 = 499 nM T95913 CM63EP 137634801 IC50 = 6309.57 nM T95913 CYAL31 137634808 Ki = 113 nM T95913 C34MHP 137634951 IC50 = 35 nM T95913 C9GXM1 137635017 IC50 = 794.33 nM T95913 C06BDR 137635072 IC50 = 150 nM T95913 CY86AJ 137635564 IC50 = 630.96 nM T95913 CYK6C4 137635941 IC50 >= 199.53 nM T95913 CMN6T7 137636115 IC50 = 125 nM T95913 CZ74XF 137636132 IC50 = 316.23 nM T95913 CPJ43Y 137636841 IC50 = 220 nM T95913 C7BE2O 137636964 IC50 = 10000 nM T95913 CV38QX 137637076 IC50 > 1000 nM T95913 CK4V7A 137637244 IC50 = 2511.89 nM T95913 CK2HR6 137637299 IC50 = 4300 nM T95913 CXPI97 137637422 IC50 >= 199.53 nM T95913 CX8NI0 137637899 IC50 = 15848.93 nM T95913 CMZV19 137639099 IC50 = 199.53 nM T95913 CJ3LX4 137639119 IC50 = 4.7 nM T95913 CS78JW 137639139 IC50 = 43 nM T95913 CHK7G9 137639570 IC50 = 6309.57 nM T95913 C4TSZ8 137639858 IC50 = 316.23 nM T95913 CK9GP8 137640140 Ki > 490 nM T95913 C7HA4V 137640279 IC50 >= 199.53 nM T95913 CA0QO6 137640453 IC50 = 91.9 nM T95913 CWK2F4 137640548 IC50 > 31622.78 nM T95913 C67NLM 137640896 IC50 >= 199.53 nM T95913 CQ8X0E 137641383 IC50 = 99 nM T95913 C0I6RQ 137641405 IC50 = 1000 nM T95913 CN3F5A 137641753 IC50 >= 199.53 nM T95913 C5X3TH 137642662 IC50 = 27 nM T95913 C1EBS6 137642764 Ki > 490 nM T95913 C8M9TX 137642801 IC50 = 16 nM T95913 CL4Q9G 137643238 IC50 > 1000 nM T95913 CP3JK1 137643598 IC50 = 794.33 nM T95913 CAPQ93 137644458 IC50 = 251.19 nM T95913 C4KAU7 137644907 IC50 = 7943.28 nM T95913 CKI2G8 137645541 IC50 = 398.11 nM T95913 C6SW7U 137646075 IC50 >= 199.53 nM T95913 C9SU6F 137646331 IC50 = 630.96 nM T95913 C5ERV3 137646413 IC50 = 29 nM T95913 CZC27Y 137646667 IC50 = 158.49 nM T95913 CA4V8H 137646998 IC50 >= 199.53 nM T95913 C5HIM9 137647114 IC50 = 398.11 nM T95913 CPMG65 137647250 IC50 = 8.4 nM T95913 C3TXN9 137647591 IC50 = 291 nM T95913 CPX42N 137647765 IC50 = 190 nM T95913 C6OK0J 137647964 IC50 > 19952.62 nM T95913 CS39XP 137648085 IC50 = 251.19 nM T95913 C4Z0NQ 137648826 IC50 = 1584.89 nM T95913 CE54DO 137648917 IC50 >= 199.53 nM T95913 CSML14 137649696 IC50 = 47 nM T95913 CCM18K 137650283 IC50 = 794.33 nM T95913 CHT1R8 137650579 IC50 = 794.33 nM T95913 C9QA0W 137652944 IC50 >= 199.53 nM T95913 CI64CW 137653468 IC50 > 25118.86 nM T95913 CN78RE 137653565 IC50 = 501.19 nM T95913 CTKQ38 137653713 IC50 = 199.53 nM T95913 C9M4PI 137653924 IC50 = 398.11 nM T95913 C9E5JK 137654836 IC50 = 316.23 nM T95913 CD19ZS 137654937 IC50 = 61 nM T95913 C4N5LS 137655123 IC50 = 1000 nM T95913 C82EOF 137655140 IC50 = 316.23 nM T95913 CHV26G 137655828 IC50 = 20 nM T95913 CC5NK4 137655965 IC50 = 501.19 nM T95913 CLC7N4 137656507 IC50 = 630.96 nM T95913 CE9H8D 137657006 IC50 = 1995.26 nM T95913 C3TD6A 137657429 Ki = 84.3 nM T95913 C2JX1W 137657572 IC50 >= 199.53 nM T95913 C41OPW 137658031 IC50 = 3162.28 nM T95913 C6BF8E 137658458 IC50 = 390 nM T95913 C35DPY 137658611 IC50 = 398.11 nM T95913 CU9PB7 137659393 IC50 = 501.19 nM T95913 CZ36BW 137659557 IC50 = 501.19 nM T95913 C3CF4O 137659746 IC50 = 316.23 nM T95913 CCX64Q 137660055 IC50 = 398.11 nM T95913 C1F6QN 137660818 IC50 >= 199.53 nM T95913 CP5K4E 137660883 IC50 = 132 nM T95913 C1OLQ3 137660961 IC50 = 1258.93 nM T95913 CM6FS2 137661095 IC50 = 398.11 nM T95913 C8R3JK 137661301 IC50 = 158.49 nM T95913 C9HPG8 137661516 IC50 = 1584.89 nM T95913 C90ELH 137661890 IC50 = 187 nM T95913 CA3C4O 138454792 IC50 = 67 nM T95913 CKDZ26 138504497 IC50 = 2900 nM T95913 C0BFS3 139327957 IC50 = 140 nM T95913 C7ZAQ1 141406387 IC50 = 24640 nM T95913 C7NUI8 141406388 IC50 = 42570 nM T95913 CQYI18 141406390 IC50 = 9470 nM T95913 CUA1D0 141406392 IC50 = 38290 nM T95913 CP0R6Y 141406393 IC50 = 1900 nM T95913 C1EVQ0 141406394 IC50 = 17810 nM T95913 C2QP0F 141406396 IC50 = 18240 nM T95913 CY2M0B 141406399 IC50 = 5100 nM T95913 CC3OU2 141406400 IC50 = 32180 nM T95913 CKV13Y 141406404 IC50 = 19030 nM T95913 C3Q1VL 141419885 IC50 = 174.2 nM T95913 C3EJX8 141419888 IC50 = 198.5 nM T95913 CKX4P3 141446054 IC50 > 158489.32 nM T95913 C9IV8R 141461655 IC50 = 268 nM T95913 C4C0QL 141461656 IC50 = 37 nM T95913 CG6O8P 141461658 IC50 = 63 nM T95913 C6I1VW 141461659 IC50 = 155 nM T95913 CES84U 141461662 IC50 = 1593 nM T95913 CM8HT7 141461664 IC50 = 381 nM T95913 CZV17F 141461667 IC50 = 7 nM T95913 CFR0I4 141461668 IC50 = 2062 nM T95913 CD5VE0 141461669 IC50 = 17 nM T95913 CU6LE4 141461671 IC50 = 15 nM T95913 CHJ93Y 141461672 IC50 = 2966 nM T95913 CV54CS 141471198 IC50 = 11 nM T95913 C25HYI 141471200 IC50 = 10 nM T95913 CZS03J 141509623 IC50 = 684 nM T95913 C1R9AN 141518981 IC50 = 45 nM T95913 C4MH5U 141518989 IC50 = 37 nM T95913 CQT27N 141520958 IC50 = 116 nM T95913 CH5F2X 141716982 IC50 = 1.259 nM T95913 CRU08D 141717009 IC50 = 0.7943 nM T95913 C8Q0VB 141717016 IC50 = 1.259 nM T95913 CQ34YR 142506035 IC50 = 162 nM T95913 CU03GW 142506036 IC50 = 2 nM T95913 C74MXW 142506065 IC50 = 3 nM T95913 CX6BQ7 142506102 IC50 = 2 nM T95913 CY3BM0 142506119 IC50 = 1769 nM T95913 CC6MD0 142506155 IC50 = 8 nM T95913 C05QOM 142506157 IC50 = 203 nM T95913 CGNQ74 142506189 IC50 = 103 nM T95913 CT3U9R 142506192 IC50 = 2 nM T95913 C1T3IQ 142506210 IC50 = 43 nM T95913 CEGV67 142506220 IC50 = 234 nM T95913 CP5HF8 142506225 IC50 = 995 nM T95913 C1U3CA 142506238 IC50 = 45 nM T95913 C7QMG9 145108300 IC50 = 17 nM T95913 C1FIE4 145439085 IC50 = 2293 nM T95913 CGF4I3 145946093 IC50 = 316.23 nM T95913 CI40JE 145951013 IC50 = 602.1 nM T95913 C6YT8E 145951131 IC50 > 9100 nM T95913 CFW62M 145951569 IC50 = 120.5 nM T95913 CHA84K 145951830 IC50 > 10000 nM T95913 CT4I9A 145952160 IC50 = 31 nM T95913 C91GVH 145952598 IC50 = 76 nM T95913 C1W0GJ 145952796 IC50 = 25118.86 nM T95913 CVMF13 145953272 IC50 = 1207 nM T95913 CYL5T1 145953372 IC50 <= 10000 nM T95913 CP14AV 145953653 IC50 = 751 nM T95913 CY8D5Q 145953886 IC50 = 596.3 nM T95913 C3ZUW8 145954195 IC50 = 358.3 nM T95913 C1NJB7 145955070 IC50 = 47 nM T95913 CRHE01 145955133 IC50 <= 10000 nM T95913 C7MP9Z 145955279 IC50 = 255.7 nM T95913 C7K8VT 145955565 IC50 = 118.1 nM T95913 CPU4X2 145955670 IC50 = 1898 nM T95913 C3ST5Y 145955693 IC50 = 140 nM T95913 C1VH5X 145955836 IC50 = 2628 nM T95913 C7K2YF 145956631 IC50 <= 10000 nM T95913 CQW74M 145956683 IC50 = 110 nM T95913 CJ1F6A 145956725 IC50 = 1036 nM T95913 C12IFO 145956886 IC50 = 456.7 nM T95913 C9O2PL 145958063 IC50 = 193.7 nM T95913 CQH01X 145958257 IC50 <= 10000 nM T95913 C3DGU7 145958571 IC50 = 708 nM T95913 C9NS6T 145958690 IC50 = 245.5 nM T95913 C7ZO9V 145959196 IC50 = 236 nM T95913 CSC81H 145959429 IC50 = 62 nM T95913 C0S1YM 145959980 IC50 = 303 nM T95913 CT3I2R 145960112 IC50 = 893.1 nM T95913 C8MJ9X 145960272 IC50 = 170 nM T95913 CLH5J2 145960703 IC50 = 6.31 nM T95913 CF36RA 145961004 IC50 = 64 nM T95913 CZO6T7 145961089 IC50 = 2511.89 nM T95913 CX6T3J 145961172 IC50 > 10000 nM T95913 C9I7EC 145961182 IC50 = 7.943 nM T95913 C54ZQA 145961234 IC50 = 3981.07 nM T95913 C83FPK 145961240 IC50 = 100 nM T95913 C31QBE 145961348 IC50 > 10000 nM T95913 CHF56O 145961403 IC50 > 9100 nM T95913 C2GT9Y 145961404 IC50 > 9100 nM T95913 COCG81 145961565 IC50 = 6309.57 nM T95913 C73MVW 145961583 IC50 = 1584.89 nM T95913 CKF0I1 145961740 IC50 = 1.259 nM T95913 C6HB9M 145961899 IC50 = 6309.57 nM T95913 CS46RM 145962397 Ki = 160 nM T95913 CT42OW 145962848 IC50 = 25.12 nM T95913 CLFQ85 145963006 IC50 = 12.59 nM T95913 CAI0D6 145963117 IC50 = 256 nM T95913 CA4FO3 145963201 IC50 = 10 nM T95913 CYZ14S 145963250 IC50 = 7943.28 nM T95913 CAD5Q9 145963302 IC50 > 10000 nM T95913 C35ZRP 145963416 IC50 > 10000 nM T95913 CQBU31 145963478 IC50 > 1000 nM T95913 C0S1ZI 145963484 IC50 = 1.259 nM T95913 C4JI8B 145963558 IC50 = 158.49 nM T95913 C87HFG 145964719 IC50 = 4752 nM T95913 CRE3Q1 145966313 IC50 = 68 nM T95913 CU9XC4 145966764 IC50 = 0.7 nM T95913 C97IKW 145969580 IC50 = 223.9 nM T95913 CK82QG 145969816 IC50 = 1783 nM T95913 C71YAK 145970017 IC50 = 3000 nM T95913 C3Y7RS 145970202 IC50 > 10000 nM T95913 CP6YC2 145970436 IC50 = 117.5 nM T95913 CZ98FH 145971490 IC50 = 1591 nM T95913 CTB97Z 145971948 IC50 = 408 nM T95913 CGQJ04 145972017 IC50 = 1590 nM T95913 C96IUM 145973569 IC50 = 0.5 nM T95913 CD7PS3 145973794 IC50 = 420 nM T95913 CZ9G6E 145974533 IC50 = 146 nM T95913 C3XIT8 145974725 IC50 = 1491 nM T95913 C1N5TZ 145975623 IC50 = 445 nM T95913 C3LR4O 145976442 IC50 = 3560 nM T95913 C3YG4Z 145977475 IC50 = 0.7 nM T95913 CPZS56 145982349 EC50 = 10000 nM T95913 CH90CT 145983168 IC50 = 184.7 nM T95913 CJU02I 145983624 IC50 = 62 nM T95913 CVS2U0 145983808 IC50 = 363 nM T95913 CF8MR5 145986347 IC50 = 1000 nM T95913 C6XMQ8 145989163 EC50 = 9890 nM T95913 CBU86Y 145991850 IC50 = 10000 nM T95913 C8X2IT 145996536 IC50 > 10000 nM T95913 C4K0JW 145996540 IC50 = 1.2 nM T95913 C6RPG0 146014481 IC50 = 831.76 nM T95913 C59KOM 146585662 IC50 = 9 nM T95913 CFQO97 146585699 IC50 = 752 nM T95913 C0GMR1 146585718 IC50 = 135 nM T95913 CI85VS 146731761 IC50 = 81 nM T95913 CWZ05D 148564044 IC50 = 22 nM T95913 C4MC0S 149169124 IC50 = 1870 nM T95913 CVW62P 149242889 IC50 = 10530 nM T95913 CN87RZ 149370890 IC50 = 810 nM T95913 CK4FJ1 149556361 IC50 = 2300 nM T95913 C8UQL4 153940691 IC50 = 1320 nM T95913 CMZ68Q 153940692 IC50 = 110 nM T95913 C5X7JK 154734328 IC50 = 1000 nM T95913 C8Q9UG 155510876 IC50 = 222 nM T95913 CDT8F2 155510913 IC50 = 1258.93 nM T95913 C6WIC9 155511977 IC50 = 1258.93 nM T95913 CPH8N1 155512095 IC50 = 251.19 nM T95913 CZJ9D6 155512258 IC50 = 5533 nM T95913 CG9I4X 155512515 IC50 = 140 nM T95913 CR1Z8A 155512529 IC50 > 10000 nM T95913 CQZY50 155512775 IC50 = 39.81 nM T95913 C5V2GO 155512947 IC50 = 2511.89 nM T95913 C1DIT4 155513047 IC50 = 125.89 nM T95913 C8PG6Z 155513084 IC50 = 794.33 nM T95913 C5M6NS 155513226 IC50 = 9550 nM T95913 C45SYX 155513615 IC50 = 6 nM T95913 CBH57O 155514764 IC50 = 2511.89 nM T95913 C5C9EG 155515047 IC50 = 1000 nM T95913 CEFS61 155515135 IC50 = 2650 nM T95913 C0AXF7 155515394 IC50 = 1584.89 nM T95913 CTS48F 155515676 IC50 = 3 nM T95913 C7Q3FR 155515734 IC50 = 1995.26 nM T95913 C30ZFN 155516445 IC50 = 630.96 nM T95913 CJDG04 155516604 IC50 = 100 nM T95913 C42JXQ 155517064 IC50 = 1995.26 nM T95913 CYO19V 155517071 IC50 = 125.89 nM T95913 CYWX76 155517213 IC50 = 1584.89 nM T95913 CT53XD 155517442 IC50 = 12589.25 nM T95913 C4G8YN 155517534 IC50 = 1983 nM T95913 CS2JT9 155518175 IC50 = 3162.28 nM T95913 CW7OM6 155518918 IC50 = 708 nM T95913 CC51GM 155519635 IC50 = 158.49 nM T95913 CHFJ25 155519726 IC50 = 12589.25 nM T95913 CZ78HW 155519830 IC50 = 316.23 nM T95913 CQEK39 155520373 IC50 = 4.3 nM T95913 C3D7FJ 155520444 IC50 = 6309.57 nM T95913 C5D6YX 155521099 IC50 > 10000 nM T95913 CEA3M1 155521494 IC50 = 63.1 nM T95913 CBSR95 155522042 IC50 = 3480 nM T95913 CZO7Q8 155522149 IC50 = 536 nM T95913 CCGW06 155523124 IC50 = 6309.57 nM T95913 CNB70P 155523246 IC50 = 1000 nM T95913 C4TLQ7 155523447 IC50 > 10000 nM T95913 CZG27I 155523570 IC50 = 38 nM T95913 C37RVF 155523599 IC50 = 4500 nM T95913 C4H2AB 155524238 IC50 = 15.85 nM T95913 CP18VT 155524467 IC50 = 1995.26 nM T95913 CUP7L2 155524901 IC50 = 1258.93 nM T95913 C2BL5I 155525312 IC50 = 25.12 nM T95913 C10RZQ 155525477 IC50 = 1000 nM T95913 CF76OV 155525717 IC50 = 19.3 nM T95913 C0UA4D 155525996 IC50 = 63.1 nM T95913 C0AR4W 155526097 IC50 = 3981.07 nM T95913 C3EAR8 155526323 IC50 = 1000 nM T95913 C82NUW 155527501 IC50 = 445 nM T95913 CK07GS 155527559 IC50 = 64 nM T95913 CX12MK 155527651 IC50 = 4 nM T95913 C8Z3TK 155528581 IC50 = 1584.89 nM T95913 C0B2NV 155528644 IC50 = 853 nM T95913 C3VAI9 155528997 IC50 = 501.19 nM T95913 C9L6OC 155529247 IC50 = 467 nM T95913 C2FE1S 155529479 IC50 = 25.12 nM T95913 CB90AR 155529643 IC50 = 199.53 nM T95913 CFV1S0 155529706 IC50 = 434 nM T95913 C14QOF 155530163 IC50 = 1584.89 nM T95913 C4I5UP 155530224 IC50 = 158.49 nM T95913 CX6N3Y 155531155 IC50 = 79.43 nM T95913 C9AXO7 155531257 IC50 = 1258.93 nM T95913 CGAI60 155531409 IC50 = 3162.28 nM T95913 CDI4V8 155531526 IC50 = 194 nM T95913 CE6QP1 155532037 IC50 = 501.19 nM T95913 CJH9U4 155532237 IC50 = 12589.25 nM T95913 C6W0JX 155532471 IC50 = 6309.57 nM T95913 CKMD29 155532546 IC50 = 6309.57 nM T95913 C3XFB8 155532820 IC50 = 19.95 nM T95913 CIYA39 155532858 IC50 = 34 nM T95913 C0GR1J 155533050 IC50 = 2 nM T95913 CQS8P1 155533070 IC50 = 1584.89 nM T95913 C0SZR9 155533335 IC50 = 2511.89 nM T95913 CAT9V1 155533370 IC50 = 5600 nM T95913 C67ERP 155533384 IC50 = 158.49 nM T95913 CL8OM7 155533564 IC50 = 6081 nM T95913 CBM24U 155533579 IC50 = 3981.07 nM T95913 CR5H8B 155533591 IC50 = 1995.26 nM T95913 CA7T0Y 155533911 IC50 = 9340 nM T95913 C8XQ4W 155534168 IC50 = 87 nM T95913 CN1ST4 155534269 IC50 = 1258.93 nM T95913 CBEG39 155534594 IC50 = 1258.93 nM T95913 CTZ3E0 155534905 IC50 = 112 nM T95913 CG1JR7 155535513 IC50 = 630.96 nM T95913 CN6KJ5 155535520 IC50 = 794.33 nM T95913 C5F2TY 155535537 IC50 = 1995.26 nM T95913 CKB2U4 155535691 IC50 = 63.1 nM T95913 CY7X3M 155535740 IC50 = 39.81 nM T95913 CUWE49 155535963 IC50 = 794.33 nM T95913 C70UDF 155536179 IC50 = 3162.28 nM T95913 CEJ6L1 155536226 IC50 = 210.7 nM T95913 CNB24M 155536473 IC50 = 1000 nM T95913 C2CG1A 155537016 IC50 = 3981.07 nM T95913 C8AJ6C 155538256 IC50 = 250.4 nM T95913 CQ1E6H 155538266 IC50 = 39.81 nM T95913 CZ19AN 155538609 IC50 = 496 nM T95913 CHR8M1 155538990 IC50 = 7510 nM T95913 CC1BG2 155539321 IC50 > 10000 nM T95913 CF20PS 155539394 IC50 = 2511.89 nM T95913 C8LKW4 155540264 IC50 = 2511.89 nM T95913 C6I5DK 155541290 IC50 = 1258.93 nM T95913 CECX47 155541544 IC50 = 501.19 nM T95913 C4FC0V 155541900 IC50 = 630.96 nM T95913 CKBW37 155542030 IC50 = 1905 nM T95913 CASE16 155542363 IC50 = 3162.28 nM T95913 C8AXF9 155542633 IC50 = 5011.87 nM T95913 C8OC2P 155542800 IC50 = 5600 nM T95913 C42BIZ 155542813 IC50 = 12589.25 nM T95913 CVNR95 155542898 IC50 = 1400 nM T95913 C1SY0G 155543154 IC50 = 23200 nM T95913 C7IWJ2 155543389 IC50 = 10000 nM T95913 CZY0N4 155543588 IC50 = 10 nM T95913 CJB8C9 155543659 IC50 = 231 nM T95913 CX1C8I 155544561 IC50 > 10000 nM T95913 CBN29V 155544583 IC50 = 204 nM T95913 C98FXC 155544955 IC50 = 3594 nM T95913 CTSW53 155546042 IC50 > 10000 nM T95913 CQ6J7U 155546361 IC50 = 280 nM T95913 C8SQA2 155546999 IC50 = 12.59 nM T95913 C8D4ZH 155547166 IC50 = 630.96 nM T95913 CI6KO7 155548518 IC50 = 251.19 nM T95913 CL4F8P 155549003 IC50 = 7.943 nM T95913 CM6S8K 155549098 IC50 = 5011.87 nM T95913 C4PEJ5 155549895 IC50 > 10000 nM T95913 CFP94J 155550309 IC50 = 794.33 nM T95913 CQ5OD0 155550395 IC50 = 45 nM T95913 CK1JR7 155551961 IC50 = 6.5 nM T95913 CJ75BO 155552100 IC50 > 1000 nM T95913 CXN3Y8 155553327 IC50 = 3981.07 nM T95913 CL04BD 155554125 IC50 = 934 nM T95913 CX9C6O 155554180 IC50 = 1000 nM T95913 CC13QL 155555170 IC50 = 1378 nM T95913 CZX06J 155555458 IC50 = 1995.26 nM T95913 C2OGW1 155555483 IC50 = 521 nM T95913 CRO5Z3 155556073 IC50 = 5756 nM T95913 CH2P4T 155556124 IC50 = 25118.86 nM T95913 CCU8M1 155556480 IC50 = 15848.93 nM T95913 CIU29Z 155556576 IC50 > 10000 nM T95913 CM3LI6 155556593 IC50 > 10000 nM T95913 CZ8CX1 155556887 IC50 = 501.19 nM T95913 CG2FS6 155557123 IC50 = 2511.89 nM T95913 CFS63H 155557182 IC50 = 301 nM T95913 C0FE4G 155557988 IC50 = 2183 nM T95913 CR8J0E 155558167 IC50 = 50.12 nM T95913 CN96JH 155558197 IC50 = 316.23 nM T95913 CSO4M3 155558261 IC50 = 5011.87 nM T95913 C52TSP 155558262 IC50 = 440 nM T95913 CS70ER 155559192 IC50 = 247 nM T95913 CVG49I 155560688 IC50 = 4010 nM T95913 C5S7AL 155560766 IC50 = 199.53 nM T95913 CQ7PS9 155560780 IC50 = 3981.07 nM T95913 CLO3B1 155561152 IC50 = 7900 nM T95913 C8XS0L 155561165 IC50 = 794.33 nM T95913 C72CQG 155561233 IC50 = 125.89 nM T95913 C1INL7 155561328 IC50 = 794.33 nM T95913 CX6U2T 155562388 IC50 = 3981.07 nM T95913 C5E9TP 155562641 IC50 = 79432.82 nM T95913 CCF4W2 155563986 IC50 = 6309.57 nM T95913 CHK4E8 155565269 IC50 = 1258.93 nM T95913 C7PXA0 155565551 IC50 = 630.96 nM T95913 CY4N7O 155565715 IC50 = 15848.93 nM T95913 CVQ6Z4 155565763 IC50 = 2511.89 nM T95913 CA1RX3 155565771 IC50 = 2511.89 nM T95913 CQ3AU4 155565828 IC50 = 19952.62 nM T95913 CMK4I3 155565845 IC50 = 1995.26 nM T95913 C59VPW 155565958 IC50 = 1584.89 nM T95913 CAP9F2 155566187 IC50 = 15 nM T95913 CM7E2G 155566279 IC50 = 3162.28 nM T95913 C3BNY5 155566309 IC50 = 10000 nM T95913 C9KQW3 155567372 IC50 = 740 nM T95913 C98NZE 155567616 IC50 = 5011.87 nM T95913 C1HQ5J 155568324 IC50 = 354 nM T95913 CLA46O 155568356 IC50 = 800 nM T95913 C7SLR8 155568452 IC50 = 501.19 nM T95913 C1S8ZB 155568922 IC50 > 1000 nM T95913 C14LVO 155569074 IC50 = 158.49 nM T95913 CFWP17 155569113 IC50 = 587 nM T95913 CUH38L 155569363 IC50 = 8420 nM T95913 C4H0NE 155569598 IC50 = 3162.28 nM T95913 D00GQM 25069592 IC50 = 7972 nM T95913 D00ZIK 9908783 IC50 = 61000 nM T95913 D01ILN 223355 IC50 = 8500 nM T95913 D01SSI 24937012 IC50 > 10000 nM T95913 D03EHM 24905142 IC50 = 1100 nM T95913 D03QQH 16760391 IC50 = 100000 nM T95913 D05USL 5278396 IC50 > 1000 nM T95913 D06DNH 9907093 IC50 > 10000 nM T95913 D06HVH 54613583 IC50 = 3100 nM T95913 D06PWI 42623951 IC50 = 25.12 nM T95913 D07JKB 135955185 IC50 = 5135 nM T95913 D07PMP 44187953 IC50 = 16 nM T95913 D08KSQ 11637090 IC50 > 10000 nM T95913 D08NQM 5289247 IC50 = 8 nM T95913 D09FBN 135955186 IC50 = 8558 nM T95913 D09ZNV 447682 IC50 > 200000 nM T95913 D0AH8Q 25074311 IC50 = 6742 nM T95913 D0EU1R 46215815 IC50 = 25118 nM T95913 D0F1SI 25074312 IC50 = 8000 nM T95913 D0H0HR 49836027 IC50 = 171 nM T95913 D0H2CM 135565635 IC50 = 1300 nM T95913 D0P5TI 58441401 IC50 = 240.3 nM T95913 D0R0TW 11964036 IC50 = 590 nM T95913 D0R2UG 52936849 IC50 = 104 nM T95913 D0S5YV 6852167 Ki = 7 nM T95913 D0T3PW 5281672 IC50 = 4720 nM T95913 D0TC5H 16049458 IC50 = 2343 nM T95913 D0W8XH 9884685 IC50 = 15 nM T95913 D0Y1DR 46225260 IC50 = 7371 nM T95913 D0Y3OO 11327430 IC50 = 220 nM T66011 CM86EA 25082538 IC50 = 12000 nM T66011 C8J7CH 44560082 IC50 = 19000 nM T66011 C2GXT8 44560086 IC50 = 19000 nM T66011 CA03BN 46883572 IC50 = 19000 nM T66011 CV0W3Y 46883575 IC50 = 23000 nM T66011 C8R2WL 46883576 IC50 = 13000 nM T66011 CGFC59 46883582 IC50 = 4000 nM T66011 C87DPG 46883583 IC50 = 5000 nM T66011 CR51BY 46883590 IC50 = 5000 nM T66011 CKA62U 46883591 IC50 = 12000 nM T66011 C5Z7YU 46883592 IC50 = 3000 nM T66011 CHWU39 46883593 IC50 = 3000 nM T66011 C1SB3M 46883594 IC50 = 50000 nM T66011 CC6SH3 46883595 IC50 = 7000 nM T66011 C14TGE 86282201 IC50 = 30 nM T66011 C5T3ZX 91755031 IC50 = 23 nM T66011 CVMB75 118046356 IC50 = 1 nM T66011 CL74ZP 145985971 IC50 = 250 nM T66011 D09JGO 46883596 IC50 = 10000 nM T16016 D0I1FQ 54671008 Ki = 5 nM T16016 D00XBC 46861584 IC50 > 10000 nM T16016 D05VTN 135565361 IC50 = 2 nM T16016 D0O2XQ 11256587 IC50 > 10000 nM T16016 D0UX2V 44537841 IC50 = 1.5 nM T16016 D0W0LS 183789 IC50 > 10000 nM T16016 C7Y8VS 1318 EC50 = 5900 nM T16016 CB4Z9P 1474 EC50 = 31622.78 nM T16016 C78GSK 14338 EC50 = 3600 nM T16016 CW6J7R 15664 EC50 = 15848.93 nM T16016 CBX47E 20445 EC50 = 12000 nM T16016 CD72TB 65237 IC50 < 1000000 nM T16016 CF1UA4 70848 EC50 = 63095.73 nM T16016 CR15FN 72791 EC50 = 1800 nM T16016 C8SC9N 72792 EC50 = 794.33 nM T16016 C7SIE4 74265 EC50 = 1500 nM T16016 CMJ4V7 77524 EC50 < 100000 nM T16016 CGZ1C6 77865 EC50 = 1995.26 nM T16016 CBW4N5 93149 EC50 = 1000 nM T16016 CTUE81 336912 IC50 > 1000000 nM T16016 C2P3FM 353741 EC50 = 15000 nM T16016 CQ3KO7 483339 IC50 > 1000 nM T16016 C7AP9W 483340 IC50 > 1000 nM T16016 CAB79M 483341 IC50 > 1000 nM T16016 C7XW2D 483342 IC50 > 1000 nM T16016 C7PMT6 483343 IC50 > 1000 nM T16016 CP25RI 483344 IC50 > 1000 nM T16016 CSF9D4 602123 IC50 = 5011.87 nM T16016 CXMY27 619353 EC50 < 1000000 nM T16016 CYU56N 667748 EC50 = 1200 nM T16016 C1SFP9 1370410 IC50 = 93 nM T16016 CAF8P7 2733927 EC50 = 10000 nM T16016 CJ73WC 2868511 Ki = 537.03 nM T16016 CAVN29 3063066 Ki = 203 nM T16016 CP65DT 3063068 Ki = 164 nM T16016 C1TX2Y 3794409 Ki = 67 nM T16016 CPZ6S1 3796276 Ki = 85.11 nM T16016 CI4N9O 3798520 Ki = 162 nM T16016 CI73AQ 5311125 Ki = 24 nM T16016 CMT8K7 5481702 IC50 = 10000 nM T16016 CHCY06 6918496 IC50 = 0.9 nM T16016 C18KRM 6918497 IC50 = 0.9 nM T16016 C5IXA6 7693048 IC50 > 10000 nM T16016 CEA5Y0 9804868 Ki = 44 nM T16016 CXM5S9 9845614 IC50 = 400 nM T16016 CUES31 9850002 Ki = 22 nM T16016 CC9U3T 9857981 Ki = 54.95 nM T16016 CN25EM 9869274 Ki = 56 nM T16016 CK7FJ6 9870185 IC50 = 5011.87 nM T16016 CK97YH 9870787 Ki = 54 nM T16016 CE13DO 9889700 Ki = 52 nM T16016 CN92IT 9894713 IC50 = 5.2 nM T16016 C2R6KA 9902204 Ki = 38.9 nM T16016 C0RH2D 9902578 Ki = 28.84 nM T16016 CY4B8U 9924108 Ki = 57 nM T16016 CQ86OZ 9935062 IC50 = 23 nM T16016 C24MLV 9935588 IC50 > 50000 nM T16016 C7LY1M 9945265 Ki = 54.95 nM T16016 C7WM0Z 9954423 IC50 = 0.96 nM T16016 C91RTG 9956238 IC50 > 10000 nM T16016 C56NZO 9956380 Ki = 45 nM T16016 CTO01C 9956488 Ki = 34 nM T16016 CAVL67 9959839 Ki = 9 nM T16016 CL3KT8 9967166 Ki = 165.96 nM T16016 CTFZ89 9967349 Ki = 27.54 nM T16016 CBVP31 9967465 Ki = 524.81 nM T16016 CJ2HT6 9979012 IC50 = 4200 nM T16016 C3TB8W 9980155 IC50 = 0.9 nM T16016 C3L7CB 9999626 IC50 = 860 nM T16016 CH5C2N 10000888 IC50 = 7100 nM T16016 CG8R5H 10001921 IC50 = 58 nM T16016 C0PDB1 10003548 IC50 = 1 nM T16016 CWD3B7 10030344 IC50 = 6.7 nM T16016 C6V8MF 10032207 IC50 = 0.92 nM T16016 C1T2FI 10049290 IC50 = 650 nM T16016 CIYE32 10049340 IC50 = 28 nM T16016 C81WKZ 10072252 IC50 = 20 nM T16016 C5QHG3 10072781 IC50 = 2.8 nM T16016 CYAJ69 10073725 IC50 = 12 nM T16016 C9RM2X 10076509 Ki = 22 nM T16016 CG0MA2 10094211 IC50 = 3.2 nM T16016 CV18TY 10094212 IC50 = 0.52 nM T16016 CC03WA 10111333 Ki = 10.47 nM T16016 CM48CP 10132885 Ki = 21.88 nM T16016 CFH9U0 10133557 Ki = 138.04 nM T16016 CU90AP 10195332 Ki = 5 nM T16016 CIGL41 10254761 IC50 = 8.9 nM T16016 CL0BS6 10255511 IC50 = 32 nM T16016 CK49NQ 10272003 IC50 > 10000 nM T16016 CDU26C 10293022 Ki = 23.99 nM T16016 CZNP37 10300214 Ki = 15.85 nM T16016 CWFB30 10323427 IC50 > 1000 nM T16016 CFH29X 10367570 IC50 = 1.4 nM T16016 C93OHM 10368175 IC50 = 1.8 nM T16016 C2JX8W 10368788 IC50 = 7.9 nM T16016 CFAY08 10371087 Ki = 1.8 nM T16016 C58GLR 10388824 IC50 = 13 nM T16016 C5LJ4B 10389562 IC50 = 0.9 nM T16016 CM9R2K 10391877 IC50 = 71 nM T16016 C9WC5D 10393066 IC50 = 3.2 nM T16016 CQU29H 10409538 IC50 = 0.96 nM T16016 C56SLV 10412648 IC50 = 1.4 nM T16016 CI9A3D 10434371 IC50 = 1.5 nM T16016 C4R6KU 10435088 IC50 = 400 nM T16016 C5GQF1 10436125 IC50 = 1.9 nM T16016 CY9B4E 10456104 IC50 = 9 nM T16016 CP1X2E 10478859 IC50 = 0.64 nM T16016 C4LB6P 10480588 IC50 = 2.5 nM T16016 CEW7C9 10482996 IC50 = 5.6 nM T16016 C6VI1Y 10499297 Ki = 54 nM T16016 C0AF4N 10501338 Ki = 306 nM T16016 CRK86P 10502989 IC50 = 1600 nM T16016 CP0OT1 10503474 Ki = 385 nM T16016 C4R5MW 10503785 Ki = 130 nM T16016 CH0F6V 10505512 IC50 = 240 nM T16016 CB6C7M 10507822 IC50 = 3.6 nM T16016 C9DY4N 10509338 IC50 = 3.1 nM T16016 C8CX5H 10524463 Ki = 4010 nM T16016 CVT27G 10525291 IC50 = 200 nM T16016 C2XON9 10525695 Ki = 906 nM T16016 CSRY03 10528677 Ki = 1330 nM T16016 CV42OK 10530837 Ki = 224 nM T16016 CIR60O 10531238 IC50 = 2100 nM T16016 CNO9H4 10531631 IC50 = 2.8 nM T16016 C4HSF7 10547456 Ki = 128 nM T16016 CUMX19 10548809 Ki = 93 nM T16016 CO6V8R 10549688 Ki = 510 nM T16016 CDC1Z2 10554359 Ki = 233 nM T16016 CAFS58 10555067 IC50 = 1800 nM T16016 C0CM5H 10555107 IC50 = 2.5 nM T16016 C83NYU 10555351 IC50 = 150 nM T16016 CWS49E 10571296 Ki = 429 nM T16016 COE8I1 10572669 Ki = 98 nM T16016 C6YW1U 10573219 Ki = 463 nM T16016 C0GWC7 10575889 Ki = 78 nM T16016 COM01N 10576419 Ki = 99 nM T16016 C15TUC 10579692 IC50 = 5 nM T16016 CUG16A 10580014 IC50 = 17 nM T16016 C05PCB 10591473 IC50 > 50000 nM T16016 CE1O4F 10596333 Ki = 371 nM T16016 C9J3PF 10597049 Ki = 359 nM T16016 C4KXS5 10599794 Ki = 1155 nM T16016 C53DCW 10623381 Ki = 244 nM T16016 CYE90Z 10643770 Ki = 790 nM T16016 C2DF5Z 10645313 Ki = 206 nM T16016 CJV7U8 10645391 Ki = 1425 nM T16016 CKBR38 10647579 Ki = 330 nM T16016 CRKL63 10649043 Ki = 32 nM T16016 C2CAG8 10652532 IC50 = 3.9 nM T16016 CV27LS 10667913 Ki = 533 nM T16016 CS93VO 10670301 IC50 = 51 nM T16016 CH65OG 10670785 Ki = 347 nM T16016 CND87M 10672205 Ki = 3430 nM T16016 C3BM7V 10676519 IC50 = 3.3 nM T16016 CB4PJ6 10690854 Ki = 236 nM T16016 C4U5IV 10693630 Ki = 7500 nM T16016 CY4D2Q 10694874 Ki = 400 nM T16016 CGL09P 10695227 Ki = 497 nM T16016 C0Q3PC 10695296 IC50 = 800 nM T16016 C80BGV 10698567 IC50 = 2 nM T16016 CT02HZ 10717972 Ki = 33 nM T16016 CAYG15 10722082 Ki = 8 nM T16016 COMN02 10737864 Ki = 584 nM T16016 C60FAV 10741203 IC50 > 10000 nM T16016 CK2VW3 10742114 IC50 > 10000 nM T16016 C5CPM3 10743274 Ki = 153 nM T16016 CNX07L 10764931 Ki = 53 nM T16016 C7I2NG 10765199 IC50 = 140 nM T16016 C3XVO7 10766333 Ki = 234 nM T16016 C68ILN 10766998 Ki = 74 nM T16016 CFV5B7 10767747 IC50 > 10000 nM T16016 C3P9OQ 10768343 Ki = 623 nM T16016 C02OLI 10769446 IC50 = 14 nM T16016 CS2JC3 10786180 Ki = 460 nM T16016 CBMA67 10788075 Ki = 1020 nM T16016 C6G7KV 10789018 Ki = 92 nM T16016 CXVY80 10789482 Ki = 51 nM T16016 C5QU0S 10793529 IC50 = 5100 nM T16016 C6XEU2 10809142 Ki = 1000 nM T16016 CTB07E 10810107 Ki = 975 nM T16016 C9AST2 10811393 Ki = 125 nM T16016 CG8FW4 10811980 IC50 = 1100 nM T16016 C6DCL5 10812461 Ki = 136 nM T16016 CSN93A 10813846 Ki = 715 nM T16016 CZX0G4 10814504 Ki = 406 nM T16016 CN0W4S 10816698 IC50 = 800 nM T16016 CRZ43V 10833944 Ki = 156 nM T16016 CE0JO2 10837160 Ki = 366 nM T16016 C36WKP 10838033 Ki = 405 nM T16016 C9EZ4N 10873705 IC50 = 260 nM T16016 C47TRP 10875472 IC50 = 167 nM T16016 C6HE2M 10916572 IC50 > 50000 nM T16016 C0EM4G 10928173 IC50 > 10000 nM T16016 CX1GK6 10928228 IC50 > 50000 nM T16016 C86DMO 10934382 IC50 > 50000 nM T16016 CX2K8E 10974378 IC50 = 310 nM T16016 CB2CG7 10984360 IC50 > 10000 nM T16016 CN87LP 10985078 IC50 = 890 nM T16016 CZM5K3 10993686 IC50 > 10000 nM T16016 CWS9J7 10995218 IC50 = 31 nM T16016 CDO30J 10995329 IC50 = 240 nM T16016 CPC19I 11004663 IC50 > 10000 nM T16016 CGY15F 11015975 IC50 > 10000 nM T16016 CK70OY 11026367 IC50 > 10000 nM T16016 C82RPC 11026461 IC50 > 50000 nM T16016 CJGS81 11026634 IC50 > 10000 nM T16016 CNE74S 11037958 IC50 = 450 nM T16016 CZ3CB6 11048445 IC50 > 10000 nM T16016 C9UK2E 11049424 IC50 < 780 nM T16016 CVX0M9 11060510 IC50 < 780 nM T16016 C8JG0H 11060814 IC50 < 780 nM T16016 CL82DR 11069916 IC50 > 10000 nM T16016 CH0DL9 11072063 IC50 = 780 nM T16016 CSUH61 11072275 IC50 = 500 nM T16016 CFG06R 11082578 IC50 = 1340 nM T16016 CCD3L5 11091447 IC50 > 10000 nM T16016 C90YHK 11104005 IC50 = 360 nM T16016 C4FB5K 11113940 IC50 = 3600 nM T16016 CZ9U7O 11124782 IC50 = 125 nM T16016 C9P3ME 11133428 IC50 > 10000 nM T16016 CIP20Q 11134412 IC50 > 10000 nM T16016 CWJ69P 11166434 IC50 = 59 nM T16016 C8L4JY 11211557 IC50 = 600 nM T16016 CA39QR 11227406 IC50 > 10000 nM T16016 CW6S9U 11236656 IC50 = 50 nM T16016 CQ6KW0 11272103 IC50 = 10000 nM T16016 C06TUD 11285791 IC50 > 10000 nM T16016 C1A5ET 11329244 IC50 = 10000 nM T16016 C8I2LV 11351191 IC50 = 16 nM T16016 C2L8BH 11397004 IC50 = 6 nM T16016 C39QNY 11464915 IC50 = 32 nM T16016 CY7S2M 11554849 IC50 = 10 nM T16016 C1HAT5 11719164 IC50 = 200 nM T16016 C3KU0D 11722772 IC50 > 50000 nM T16016 CB34MH 11729258 IC50 > 50000 nM T16016 CVB47P 11733139 IC50 > 10000 nM T16016 CVLM30 11734303 IC50 = 71 nM T16016 CPG15O 11743399 IC50 = 1 nM T16016 CL54BJ 11744314 IC50 = 0.36 nM T16016 CQN35J 11764610 IC50 = 7.9 nM T16016 CI29EG 11794863 IC50 = 510 nM T16016 CU1EP6 11798220 Ki = 908 nM T16016 CTB87F 11801019 Ki = 6 nM T16016 C0B9XN 11803141 IC50 = 1.9 nM T16016 CSX85G 11811443 IC50 > 10000 nM T16016 COZ69K 11813735 IC50 = 67 nM T16016 CT8D3H 11814253 IC50 = 1410 nM T16016 CO23LC 11825113 IC50 > 10000 nM T16016 C96ZJD 11828013 IC50 < 780 nM T16016 C6QN3V 11828215 IC50 = 295 nM T16016 C5F3ZC 12015739 IC50 = 11800 nM T16016 C8BM0H 12041800 EC50 = 2000 nM T16016 CRY83B 12093162 Ki = 251.19 nM T16016 C2QWR3 12093163 Ki = 489.78 nM T16016 C79CBJ 12093167 Ki = 15 nM T16016 C3E1FW 12112109 IC50 = 8 nM T16016 CK80NA 12987698 EC50 = 4900 nM T16016 CJGC50 14434082 IC50 < 1000000 nM T16016 CV3O8X 14770534 IC50 > 32000 nM T16016 C7X3CQ 15604497 Ki = 1000 nM T16016 CIZ8C1 15783796 EC50 = 1258.93 nM T16016 CQJ7Y2 15985912 Ki = 398.11 nM T16016 C0G1SC 15985914 Ki = 501.19 nM T16016 C8IKY6 17553211 IC50 > 3000 nM T16016 C9EHC5 17753030 IC50 = 7 nM T16016 CRM90U 19430534 Ki = 501.19 nM T16016 C1ZYS2 21070982 IC50 = 182 nM T16016 C13PWC 21070983 IC50 = 12 nM T16016 C0AOI7 21070984 IC50 = 77 nM T16016 C1CA6D 21070989 IC50 = 2.5 nM T16016 C7FA0C 21070990 IC50 = 3400 nM T16016 CB03CZ 21070993 IC50 = 100 nM T16016 CM27EA 21071046 IC50 = 340 nM T16016 CU8Q7B 21071066 IC50 = 5600 nM T16016 C28JBU 21071070 IC50 = 1100 nM T16016 CV6NF4 21071081 IC50 = 11000 nM T16016 CNM1A8 21071083 IC50 = 2700 nM T16016 C2AS6B 21071094 IC50 = 98 nM T16016 C4WI1R 21071096 IC50 = 32000 nM T16016 C57SVE 21071098 IC50 = 5650 nM T16016 CWMA26 21071099 IC50 = 9800 nM T16016 CZT7J5 21071106 IC50 = 3300 nM T16016 CVQU01 21071108 IC50 = 3650 nM T16016 CC9YA1 22335665 Ki = 47.86 nM T16016 CTO2A8 22335694 Ki = 42.66 nM T16016 CKO01W 22725647 Ki = 30.9 nM T16016 CRM12J 23283073 IC50 = 9.7 nM T16016 C27VNB 24712289 IC50 > 3000 nM T16016 C0J1HA 24738063 IC50 = 4.1 nM T16016 C48OHP 24740167 IC50 = 525 nM T16016 CYX72D 24740170 IC50 = 375 nM T16016 C25HKJ 24758044 IC50 = 28 nM T16016 CW2CM4 24758045 IC50 = 26 nM T16016 C8KC5X 24758046 IC50 = 118 nM T16016 CJF53V 24758047 IC50 = 70 nM T16016 CC7N3T 24758171 IC50 = 40 nM T16016 C1JHY4 24758172 IC50 = 32 nM T16016 C8F0CE 24758173 IC50 = 32 nM T16016 C0P3BR 24758174 IC50 = 24 nM T16016 CXE3M1 24758175 IC50 = 58 nM T16016 C2EP9Y 24758176 IC50 = 25 nM T16016 CA5C3R 24758294 IC50 = 30 nM T16016 C7UE5H 24758295 IC50 = 8 nM T16016 C0OU9Z 24758296 IC50 = 13 nM T16016 CD0XB9 24758297 IC50 = 14 nM T16016 CQ9WX7 24758298 IC50 = 18 nM T16016 CI0V6U 24758299 IC50 = 19 nM T16016 CKH7M2 24758406 IC50 = 20 nM T16016 C93QGZ 24758408 IC50 = 22 nM T16016 CIY5Q4 24758517 IC50 = 44 nM T16016 C32AZH 24758518 IC50 = 45 nM T16016 CD5JH7 24758630 IC50 = 121 nM T16016 CS6NW4 24758743 IC50 = 152 nM T16016 C7ZRE8 24758744 IC50 = 50 nM T16016 C6F1NH 24758745 IC50 = 85 nM T16016 CF9S7E 24758856 IC50 = 40 nM T16016 C9H6MY 24759081 IC50 = 35 nM T16016 C5YDC2 24759191 IC50 = 36 nM T16016 CF6GO2 24759420 IC50 = 80 nM T16016 C6CET2 24759740 IC50 = 388 nM T16016 CPD05R 24782574 IC50 = 50 nM T16016 CISV81 24782826 IC50 = 22 nM T16016 CLG7M5 25022507 IC50 = 90 nM T16016 C7NJ1B 25109291 Ki = 0.043 nM T16016 C54LQF 25230828 IC50 > 50000 nM T16016 CZX9B0 25231298 IC50 > 75000 nM T16016 C74EOA 25231299 IC50 = 3600 nM T16016 C98VPY 25231300 IC50 = 270 nM T16016 CF76KB 25231301 IC50 = 270 nM T16016 CZXC46 25231302 IC50 = 43000 nM T16016 C0RZJ5 25231303 IC50 > 100000 nM T16016 C2J4GS 25231477 IC50 > 13000 nM T16016 C6YW9F 25231478 IC50 > 77000 nM T16016 C6JNK1 25231479 IC50 > 100000 nM T16016 CRP1H8 25231480 IC50 = 1300 nM T16016 C9H2LY 25231481 IC50 = 5700 nM T16016 COHI45 25231482 IC50 > 100000 nM T16016 C5C8DA 25233577 IC50 = 4000 nM T16016 CIX06B 25233578 IC50 = 4700 nM T16016 CVCF50 25233579 IC50 = 680 nM T16016 CE1FK6 25233580 IC50 = 700 nM T16016 CD8F7W 25233581 IC50 = 720 nM T16016 CEF52O 25233582 IC50 = 290 nM T16016 C8H5EP 25233753 IC50 = 2950 nM T16016 CAL67P 25233754 IC50 = 120 nM T16016 CNVF07 25233755 IC50 = 22 nM T16016 C8W5VE 25233756 IC50 = 6 nM T16016 CCGL97 25233757 IC50 > 28000 nM T16016 C72FBZ 25233758 IC50 > 100000 nM T16016 C3CAP1 25233941 IC50 > 28000 nM T16016 CDJ67K 25233947 IC50 = 540 nM T16016 C07BSM 25252974 IC50 = 4 nM T16016 CS0XW4 25253284 IC50 = 20 nM T16016 CUKC71 25254218 IC50 = 22 nM T16016 C8E3GU 26042546 IC50 > 30000 nM T16016 CQD8U5 31900420 IC50 > 3000 nM T16016 CIKC26 32637491 IC50 > 3000 nM T16016 C5D0XT 36715516 IC50 > 3000 nM T16016 CXI89R 37664972 IC50 = 790 nM T16016 CC3D2Q 40636824 IC50 > 3000 nM T16016 CA79PZ 40636827 IC50 > 3000 nM T16016 CAR7X3 42602328 IC50 = 1.8 nM T16016 C8A5TC 42602331 IC50 = 1.4 nM T16016 CU2PO5 44180522 IC50 > 25118.86 nM T16016 C5YFB9 44252324 IC50 > 10000 nM T16016 CKNR65 44281427 IC50 = 370 nM T16016 CPS75A 44308794 IC50 < 50000 nM T16016 C0MU9T 44308812 IC50 < 50000 nM T16016 CJZ54H 44308819 IC50 = 840 nM T16016 C1T9VK 44308837 IC50 < 50000 nM T16016 CW29KX 44308850 IC50 < 50000 nM T16016 C03USP 44308902 IC50 = 30000 nM T16016 C2MA1N 44308997 IC50 = 2490 nM T16016 CCRW52 44309046 IC50 > 32000 nM T16016 CBC5G2 44309060 IC50 = 10300 nM T16016 CI4P5Z 44309061 IC50 = 55100 nM T16016 CW2JL5 44309067 IC50 < 50000 nM T16016 CDF92Y 44309074 IC50 = 64 nM T16016 C8O0UX 44309077 IC50 = 5600 nM T16016 CWXN65 44309087 IC50 = 18500 nM T16016 C9K2EI 44309091 IC50 = 8000 nM T16016 CWNB28 44309094 IC50 > 32000 nM T16016 CJ3WS4 44309105 IC50 = 280 nM T16016 CW3FI1 44309112 IC50 = 5150 nM T16016 COK2M0 44309119 IC50 < 50000 nM T16016 CF28NB 44309120 IC50 > 32000 nM T16016 CPTJ37 44309122 IC50 = 27 nM T16016 C3NG7S 44309124 IC50 = 740 nM T16016 C49FZD 44309128 IC50 = 4600 nM T16016 COWL46 44309136 IC50 < 50000 nM T16016 CC5ZE8 44309143 IC50 = 1 nM T16016 C81JTN 44309155 IC50 = 15000 nM T16016 C41TRZ 44309156 IC50 < 50000 nM T16016 CE52DG 44309161 IC50 = 3460 nM T16016 C7UV9B 44309163 IC50 = 22 nM T16016 CYE9C4 44309165 IC50 = 15 nM T16016 C3ZD4J 44309166 IC50 = 3500 nM T16016 CVA24D 44309171 IC50 = 420 nM T16016 C0XA4Q 44309178 IC50 = 2600 nM T16016 CJSP94 44309185 IC50 = 670 nM T16016 C3SHY2 44309192 IC50 = 610 nM T16016 C93LQN 44309194 IC50 = 580 nM T16016 C2ENG9 44309195 IC50 = 20 nM T16016 CRU6E3 44309213 IC50 = 2900 nM T16016 C2P1KQ 44309219 IC50 = 560 nM T16016 CT7DV5 44309222 IC50 = 4200 nM T16016 C7KLP0 44309235 IC50 = 580 nM T16016 CL8P6W 44309236 IC50 = 510 nM T16016 C6V8DR 44309237 IC50 = 16700 nM T16016 CVIJ87 44309244 IC50 = 44800 nM T16016 CU52KE 44309245 IC50 = 850 nM T16016 C0GY2J 44309267 IC50 = 130 nM T16016 CE2I6H 44309286 IC50 = 7 nM T16016 C71LNC 44309312 IC50 = 8 nM T16016 CGDF80 44309313 IC50 = 52 nM T16016 CA5YD0 44309318 IC50 = 48 nM T16016 CHS3F9 44309327 IC50 = 26 nM T16016 C8CY4Z 44309337 IC50 = 8 nM T16016 CXQ38W 44309347 IC50 = 160 nM T16016 C7B5LR 44309353 IC50 = 46 nM T16016 CVO98N 44309364 IC50 = 130 nM T16016 C8DTH6 44309365 IC50 > 25000 nM T16016 CPQ8T7 44309397 IC50 = 9 nM T16016 C27LRK 44309407 IC50 = 540 nM T16016 CNQ0G4 44309414 IC50 = 2570 nM T16016 CJFV61 44361881 Ki = 29 nM T16016 CR5S9Y 44362079 Ki = 1188 nM T16016 C8C9LX 44405180 IC50 = 360 nM T16016 C8TS2N 44405181 IC50 = 2.4 nM T16016 CO16BT 44405194 IC50 = 1700 nM T16016 C47JTD 44405196 IC50 = 800 nM T16016 C87DSA 44405202 IC50 = 9.6 nM T16016 CGKV93 44405203 IC50 = 28 nM T16016 C4FS7U 44405211 IC50 = 300 nM T16016 CLDC78 44405212 IC50 = 6 nM T16016 CP3O7Y 44405234 IC50 = 1600 nM T16016 C9ZT8S 44430713 IC50 = 18 nM T16016 CM1E0I 44430714 IC50 = 350 nM T16016 CPI3C7 44430715 IC50 = 78 nM T16016 C53WIQ 44430716 IC50 = 270 nM T16016 CNAZ59 44430717 IC50 = 97 nM T16016 CMJ8I2 44430718 IC50 = 2340 nM T16016 CNA21M 44430720 IC50 = 2910 nM T16016 CKA2R9 44430721 IC50 = 200 nM T16016 C61NLQ 44430722 IC50 = 920 nM T16016 CG9E5H 44430723 IC50 = 14 nM T16016 CQKT60 44430724 IC50 = 160 nM T16016 CBVJ95 44430725 IC50 = 90 nM T16016 CG49JY 44430726 IC50 = 140 nM T16016 CE5AF1 44430727 IC50 > 10000 nM T16016 CSG7K4 44430732 IC50 = 72 nM T16016 CZ9WM3 44430735 IC50 = 170 nM T16016 CWLX40 44430736 IC50 = 800 nM T16016 CV62CF 44430742 IC50 = 160 nM T16016 C8PK5W 44430745 IC50 = 54 nM T16016 CC6YP2 44430746 IC50 = 13 nM T16016 CPM05Z 44430748 IC50 = 6 nM T16016 C9BE1D 44430750 IC50 = 64 nM T16016 CU39TN 44430752 IC50 = 12 nM T16016 CP37VK 44430753 IC50 = 5 nM T16016 C47MRZ 44430754 IC50 = 15 nM T16016 CQSY30 44430755 IC50 = 8 nM T16016 C9BVX3 44430756 IC50 = 26 nM T16016 CSH43L 44430758 IC50 = 6 nM T16016 CF4EM2 44430759 IC50 = 76 nM T16016 CX2Q8V 44430836 IC50 = 220 nM T16016 CQGX84 44431523 IC50 = 480 nM T16016 CU9V8X 44431524 IC50 = 30 nM T16016 C4VN5J 44431527 IC50 = 38 nM T16016 CU42MW 44431528 IC50 = 44 nM T16016 CNZ4R0 44431529 IC50 = 13 nM T16016 C68QOX 44453084 IC50 = 1650 nM T16016 C4QAH9 44453157 IC50 = 390 nM T16016 C5URL9 44453161 IC50 = 280 nM T16016 CZ6QR5 44453162 IC50 = 120 nM T16016 CH9D7P 44453163 IC50 = 7330 nM T16016 CYN36R 44453164 IC50 = 190 nM T16016 C62OVR 44453165 IC50 = 3650 nM T16016 C6HVU9 44453167 IC50 = 2200 nM T16016 CEY32C 44453195 IC50 = 2260 nM T16016 C3VK9H 44453197 IC50 = 2260 nM T16016 CA70QE 44453198 IC50 = 4650 nM T16016 C1QZE2 44453199 IC50 = 120 nM T16016 CAO60C 44453200 IC50 = 50 nM T16016 CXZ96H 44453202 IC50 = 30 nM T16016 CL2YO8 44453225 IC50 = 970 nM T16016 CZ85CL 44453226 IC50 = 670 nM T16016 C1RMH2 44453227 IC50 = 330 nM T16016 CW82CO 44453228 IC50 = 80 nM T16016 CHW4U3 44453229 IC50 = 210 nM T16016 C8NX4K 44453263 IC50 = 370 nM T16016 CSA8W9 44453265 IC50 = 380 nM T16016 CT5LK7 44453289 IC50 > 10000 nM T16016 CRP5D2 44453290 IC50 = 370 nM T16016 CUE83S 44453291 IC50 = 110 nM T16016 CHSC39 44453292 IC50 = 180 nM T16016 CASM45 44453293 IC50 = 140 nM T16016 CMVW23 44453317 IC50 = 7980 nM T16016 CE3UW0 44453320 IC50 = 200 nM T16016 CYA2S8 44453321 IC50 = 420 nM T16016 CJL5T4 44453356 IC50 > 10000 nM T16016 CRM58W 44453357 IC50 = 1240 nM T16016 C4DY0R 44453359 IC50 = 90 nM T16016 C59PBZ 44453361 IC50 = 40 nM T16016 C1VA0H 44453363 IC50 = 180 nM T16016 CQPG50 44453399 IC50 > 10000 nM T16016 CE1PR7 44453400 IC50 = 100 nM T16016 CJIZ23 44453401 IC50 > 10000 nM T16016 CZY72M 44453402 IC50 = 1340 nM T16016 CRN83S 44453403 IC50 = 30 nM T16016 CX4PU5 44453433 IC50 = 1850 nM T16016 CT3D4B 44453435 IC50 = 280 nM T16016 CI9BZ7 44453436 IC50 = 520 nM T16016 CT9D0R 44453437 IC50 = 360 nM T16016 CV0KP8 44453464 IC50 = 1330 nM T16016 C35SCE 44453466 IC50 = 430 nM T16016 C8I5SN 44453467 IC50 = 180 nM T16016 C15TOP 44453469 IC50 = 510 nM T16016 CKX1I6 44453472 IC50 > 1000 nM T16016 C58PQU 44453499 IC50 = 510 nM T16016 CK9E6M 44453501 IC50 = 180 nM T16016 CC7XV8 44453502 IC50 = 6210 nM T16016 CX12CN 44453503 IC50 = 350 nM T16016 C2OED7 44453504 IC50 = 240 nM T16016 CO4ZW0 44453525 IC50 = 1170 nM T16016 CD4Y8C 44453527 IC50 = 1000 nM T16016 CO8TK2 44453528 IC50 = 385 nM T16016 C6G3XF 44453529 IC50 = 160 nM T16016 C1V0EH 44453557 IC50 = 600 nM T16016 CI9E5K 44453559 IC50 > 30000 nM T16016 CDHV21 44453579 IC50 = 400 nM T16016 CV6TD4 44453584 IC50 = 84 nM T16016 C4SLA8 44453611 IC50 > 30000 nM T16016 CMCN57 44453612 IC50 > 10000 nM T16016 C4EM8C 44453614 IC50 = 1400 nM T16016 CUP6R8 44453615 IC50 = 1300 nM T16016 C7CMI0 44453637 IC50 = 1900 nM T16016 CD5QK4 44453638 IC50 = 1290 nM T16016 C2Z1YR 44453639 IC50 = 480 nM T16016 CBA20D 44453641 IC50 = 3880 nM T16016 CL2WB7 44468439 IC50 > 3000 nM T16016 C94VWK 44468440 IC50 = 1200 nM T16016 C5OIK9 44468442 IC50 = 1200 nM T16016 CYXR38 44468570 IC50 = 68 nM T16016 CX6U4M 44468708 IC50 = 61 nM T16016 CR6W8U 44469380 IC50 = 2500 nM T16016 C4DL5C 44469677 IC50 > 10000 nM T16016 CO3D8M 44469804 IC50 = 120 nM T16016 C35AHO 44469942 IC50 = 44 nM T16016 CHE1A2 44470083 IC50 = 5 nM T16016 CHNM79 44470374 IC50 = 12 nM T16016 CA7V8M 44480348 IC50 = 47 nM T16016 C3UMK5 44480600 IC50 = 15 nM T16016 CT5N4E 44555481 IC50 > 50000 nM T16016 CS9U6X 44560288 IC50 = 9.6 nM T16016 CF5X2U 45138007 IC50 = 3 nM T16016 CK50UD 45138010 IC50 = 34 nM T16016 CID15S 45138012 IC50 = 450 nM T16016 C6A3XH 45138458 IC50 = 19 nM T16016 CXC4M1 45138759 IC50 = 0.3 nM T16016 CK3N1G 46206137 IC50 > 10000 nM T16016 CQ3FX0 46858281 IC50 = 2400 nM T16016 C80WVI 49796696 Ki = 206 nM T16016 CVY1G2 49796697 Ki = 116 nM T16016 C95CPY 49798264 Ki = 316.23 nM T16016 C3SUN1 49798265 Ki = 125.89 nM T16016 CBG4T2 49798289 Ki = 125.89 nM T16016 C6C8AV 49865900 IC50 = 16 nM T16016 C87BYU 49865901 IC50 = 810 nM T16016 CJV7Z9 49865951 IC50 = 2.9 nM T16016 C8K6CQ 52916803 IC50 = 1.8 nM T16016 C3P7QF 52917500 IC50 = 2 nM T16016 C0NT2M 52932654 IC50 > 3000 nM T16016 CCI58B 54712652 Ki = 199.53 nM T16016 CH3UL5 57390926 IC50 = 261 nM T16016 CK2Y8P 57396208 IC50 = 387 nM T16016 CR09LY 57400127 IC50 > 25118.86 nM T16016 CAT9F4 57840192 IC50 = 10 nM T16016 CT1JC7 57840210 IC50 = 5200 nM T16016 CTAH32 57840282 IC50 = 20 nM T16016 CJ90DZ 57840295 IC50 = 10 nM T16016 C4RC3N 57840302 IC50 = 6 nM T16016 C3LMG6 57840312 IC50 = 120 nM T16016 C9QO4L 57840315 IC50 = 97 nM T16016 C89RVZ 57840356 IC50 = 18 nM T16016 C5S7FB 57840363 IC50 = 2 nM T16016 CVW80D 57840380 IC50 = 68 nM T16016 CFJ80G 57840427 IC50 = 40 nM T16016 CE3V0N 57840435 IC50 = 8 nM T16016 C9KW6F 57840437 IC50 = 5 nM T16016 CNA3W0 57840460 IC50 = 92 nM T16016 CFS8P5 57840482 IC50 = 7 nM T16016 CM6UK5 57840511 IC50 = 10 nM T16016 C5CU2J 57840512 IC50 = 23 nM T16016 CM32AV 57840515 IC50 = 47 nM T16016 CD5Z6H 57840518 IC50 = 37 nM T16016 C4I2OZ 57840522 IC50 = 740 nM T16016 CI2B1E 57840556 IC50 = 19 nM T16016 CI6XW0 57840557 IC50 = 500 nM T16016 C25SLU 57888652 IC50 = 130 nM T16016 C7TBL8 57888663 IC50 = 233 nM T16016 CM31AW 57888688 IC50 = 303 nM T16016 C6NLY7 57888690 IC50 = 46 nM T16016 CTX8J4 57888707 IC50 = 107 nM T16016 CTY08U 57888715 IC50 = 100 nM T16016 C1EGP2 57888718 IC50 = 1077 nM T16016 CD08VL 57888746 IC50 = 194 nM T16016 CUX61B 57888747 IC50 = 4.7 nM T16016 C70ZKN 57888758 IC50 = 2940 nM T16016 C32IGS 57888775 IC50 = 152 nM T16016 CUG73D 57888785 IC50 = 6 nM T16016 CD8XO3 57888812 IC50 = 259 nM T16016 CQ79WS 57888832 IC50 = 115 nM T16016 CBS39N 57888834 IC50 = 1.7 nM T16016 CG15IU 57888886 IC50 = 854 nM T16016 CGK3S6 57888895 IC50 = 3.3 nM T16016 C7USZ8 57888900 IC50 = 9.9 nM T16016 CSR0N6 57888907 IC50 = 2 nM T16016 C7S5XP 57888919 IC50 = 0.8 nM T16016 CG3JO6 57888925 IC50 = 262 nM T16016 C14OID 57888938 IC50 = 40 nM T16016 CWKP07 57888949 IC50 = 616 nM T16016 CUHR07 57888953 IC50 = 55 nM T16016 C8EBZ4 57888963 IC50 = 370 nM T16016 C56BOX 57888966 IC50 = 9.9 nM T16016 C9FM2N 57888993 IC50 = 1 nM T16016 C05HEB 57889002 IC50 = 423 nM T16016 COP15F 57889003 IC50 = 0.8 nM T16016 CO67FJ 57889006 IC50 = 539 nM T16016 CUCX67 57889023 IC50 = 3.4 nM T16016 C4VC6R 57889047 IC50 = 20 nM T16016 CCD01J 57889071 IC50 = 1.8 nM T16016 CLT76V 57889077 IC50 = 2.2 nM T16016 CCQ8G1 57889099 IC50 = 2 nM T16016 C69CJK 57889121 IC50 = 4.4 nM T16016 CW4S5A 57889141 IC50 = 180 nM T16016 CBMJ90 57889158 IC50 = 15 nM T16016 CM8IY2 57889164 IC50 = 2.9 nM T16016 CP13VI 57889180 IC50 = 4 nM T16016 CMZQ02 57889181 IC50 = 3 nM T16016 C1J5RH 57889188 IC50 = 3 nM T16016 CH9V4I 57889230 IC50 = 1.7 nM T16016 CY9F3C 57889234 IC50 = 933 nM T16016 CUW9Z5 57889255 IC50 = 140 nM T16016 CPD8S4 57889291 IC50 = 7.6 nM T16016 CJ5C3D 57889314 IC50 = 3 nM T16016 CMT6C1 57889327 IC50 = 1 nM T16016 CDOA16 57889334 IC50 = 1.9 nM T16016 C4DMF2 57889346 IC50 = 543 nM T16016 C9SR2K 57889347 IC50 = 2.6 nM T16016 C9AMN1 57889407 IC50 = 341 nM T16016 CN0WX5 57889423 IC50 = 2.5 nM T16016 C0YCH2 57889430 IC50 = 1.1 nM T16016 C5EU1V 57889478 IC50 = 45 nM T16016 CM9PI7 57889484 IC50 = 153 nM T16016 CFOK45 57889591 IC50 = 120 nM T16016 C8KEZ3 57889592 IC50 = 185 nM T16016 C26KEZ 57889613 IC50 = 10 nM T16016 CF2E5A 57889625 IC50 = 191 nM T16016 CJ2P3S 57889635 IC50 = 9 nM T16016 CY28OV 57889649 IC50 = 7.1 nM T16016 C0AOP9 57889660 IC50 = 13 nM T16016 C70YGB 57889664 IC50 = 105 nM T16016 C7OQV8 57889667 IC50 = 172 nM T16016 CW4Q2Z 57889679 IC50 = 10 nM T16016 C5G6PM 57889696 IC50 = 121 nM T16016 C31ZKO 57889736 IC50 = 3 nM T16016 CL29GA 57889758 IC50 = 5.8 nM T16016 CA46BV 57889764 IC50 = 1.2 nM T16016 CL8GT3 57889796 IC50 = 180 nM T16016 CLKA82 57889843 IC50 = 3.6 nM T16016 C7ZF9O 57889874 IC50 = 265 nM T16016 C3SZL5 57889880 IC50 = 521 nM T16016 CNV92I 57889883 IC50 = 70 nM T16016 CX82KS 57889897 IC50 = 4.1 nM T16016 C7KL5M 57889944 IC50 = 88 nM T16016 C9U8JV 57889972 IC50 = 324 nM T16016 C4Z3GA 57889974 IC50 = 6.3 nM T16016 CG1M7U 57889975 IC50 = 18 nM T16016 C9LKQ5 57889979 IC50 = 4.3 nM T16016 C9VE5T 57991685 IC50 = 1603 nM T16016 CAL9F2 57991690 IC50 = 95 nM T16016 CLH4Y8 57991707 IC50 = 2.3 nM T16016 CUNM10 57991713 IC50 = 208 nM T16016 CBQ7I3 58138764 IC50 > 3000 nM T16016 C84IXN 58138765 IC50 = 1100 nM T16016 CPWO40 58138766 IC50 > 3000 nM T16016 CIP73G 58138781 IC50 = 450 nM T16016 CY5G6S 58138788 IC50 = 750 nM T16016 C7IVB1 58138789 IC50 = 4.5 nM T16016 C1PAV2 58138800 IC50 > 3000 nM T16016 C1FV4A 58138826 IC50 = 22 nM T16016 CW20DR 58138832 IC50 = 1700 nM T16016 CM3L2A 58138839 IC50 > 3000 nM T16016 CQXC68 58138841 IC50 = 55 nM T16016 CKMW80 58138845 IC50 = 210 nM T16016 C6I3ED 58138852 IC50 = 170 nM T16016 C12JLA 58138868 IC50 = 17 nM T16016 CFHQ71 58138880 IC50 = 6 nM T16016 CNG5X3 58138893 IC50 = 180 nM T16016 CD01TW 58138911 IC50 = 260 nM T16016 C0YWT1 58509213 IC50 > 10000 nM T16016 C5P0GD 58778003 IC50 = 8 nM T16016 C08OME 58778007 IC50 = 6400 nM T16016 C0I2HN 59278115 IC50 = 1.4 nM T16016 CJW8D2 59278123 IC50 = 8 nM T16016 C8CZ7T 59278147 IC50 = 1.2 nM T16016 C03SHK 59278235 IC50 = 61 nM T16016 C4KU2S 59278286 IC50 = 0.2 nM T16016 CRH6S5 59278305 IC50 = 12 nM T16016 CA23BD 59278307 IC50 = 12 nM T16016 CEAY32 59278314 IC50 = 6.8 nM T16016 C1L2SC 59278332 IC50 = 0.2 nM T16016 CLS59N 59278436 IC50 = 2 nM T16016 CO78WQ 59278474 IC50 = 41 nM T16016 CK2CB9 59687824 IC50 = 5 nM T16016 CODB07 66686405 IC50 = 0.8 nM T16016 CO74RQ 68416145 IC50 > 3000 nM T16016 CG46AF 68816399 IC50 = 560 nM T16016 CQ34PJ 68817337 IC50 = 32 nM T16016 CAN47O 68818375 IC50 = 9 nM T16016 C9S1NP 68818964 IC50 = 79 nM T16016 C6KH1J 68956901 IC50 = 7.1 nM T16016 CRWB79 68958915 IC50 = 130 nM T16016 CZHF19 68959770 IC50 = 1.4 nM T16016 C8HM7E 68959963 IC50 = 0.36 nM T16016 C3H9CD 68962095 IC50 = 5 nM T16016 C8Y3PB 68963393 IC50 = 2.5 nM T16016 C1E4QF 68963562 IC50 = 12 nM T16016 C1KAN5 68963686 IC50 = 1.1 nM T16016 C52BVJ 68963698 IC50 = 89 nM T16016 C6Z7UL 69435853 IC50 = 7.1 nM T16016 CQVW46 69437029 IC50 = 160 nM T16016 CNY8G5 69437067 IC50 = 1300 nM T16016 C37WGU 69437285 IC50 = 560 nM T16016 C6XQ3C 69439557 IC50 = 37 nM T16016 CG3DM1 71214709 Ki = 398.11 nM T16016 CG5V6I 71214710 Ki = 1584.89 nM T16016 CA72CU 71214725 Ki = 1000 nM T16016 CMSH09 71214976 Ki = 1258.93 nM T16016 CSD6R9 71450657 Ki = 501.19 nM T16016 C8A0XW 71450658 Ki = 316.23 nM T16016 C4SH7L 71452035 IC50 = 177 nM T16016 C8YW2L 71452487 Ki = 1584.89 nM T16016 C1TOE8 71452488 Ki = 1000 nM T16016 CT7FK3 71453837 IC50 = 66 nM T16016 C71FXH 71454246 Ki = 3981.07 nM T16016 CD8I7C 71454247 Ki = 1584.89 nM T16016 CSL01M 71454248 Ki = 316.23 nM T16016 CSN6K4 71455572 IC50 = 14930 nM T16016 C3EYK5 71456007 Ki = 7943.28 nM T16016 CHV16Z 71456008 Ki = 1584.89 nM T16016 C7K2XU 71457361 IC50 = 38 nM T16016 CCYR75 71457362 IC50 = 34 nM T16016 C6MHX5 71457815 Ki = 2511.89 nM T16016 C76AQC 71460999 IC50 = 2832 nM T16016 C3BXS9 71461438 Ki = 1000 nM T16016 CRV73F 71461439 Ki = 1000 nM T16016 C3P5HM 71461440 Ki = 1000 nM T16016 CIP7D8 71462570 Ki = 2.3 nM T16016 C5E1FJ 71463165 Ki = 7943.28 nM T16016 C8VX0L 71463166 Ki = 1995.26 nM T16016 CTZ63Y 71560163 IC50 = 120 nM T16016 CVH9S8 71570633 IC50 = 0.79 nM T16016 C6ZBW8 71570634 IC50 = 18 nM T16016 C46RFP 71655299 IC50 = 1.3 nM T16016 CUI4D7 71655559 IC50 = 110 nM T16016 CHZ92K 71680936 IC50 = 2.3 nM T16016 CS1X3B 71681244 IC50 = 20 nM T16016 C86DGB 71681399 IC50 = 2.2 nM T16016 CGFZ24 71681400 IC50 = 17 nM T16016 C1IX0A 71682816 IC50 = 2240 nM T16016 CNE87P 71717436 IC50 = 5 nM T16016 CVM47W 71717437 IC50 = 420 nM T16016 C30LKZ 71718022 IC50 = 12 nM T16016 CG18BJ 71718023 IC50 = 16 nM T16016 C5N7RO 71718646 IC50 = 107 nM T16016 CM45XP 71718647 IC50 = 220 nM T16016 CSF0T9 71719253 IC50 = 11 nM T16016 C3EUY7 71719254 IC50 = 14 nM T16016 C9F0XG 71719255 IC50 = 210 nM T16016 C05FBT 71719855 IC50 = 10 nM T16016 CEPD62 71719856 IC50 = 52 nM T16016 CWH6T3 72548703 IC50 = 0.081 nM T16016 C4S2OT 72945111 IC50 = 13 nM T16016 C7MS4G 72945112 IC50 = 3.2 nM T16016 CV74IH 72945310 IC50 = 4.5 nM T16016 CXOI39 72945311 IC50 = 1.3 nM T16016 C5TS1M 72945313 IC50 = 1.8 nM T16016 CH63BO 72945314 IC50 = 1.8 nM T16016 C2VU8F 72945510 IC50 = 0.89 nM T16016 CAO2L3 72945511 IC50 = 2.2 nM T16016 CQ5MD0 72945512 IC50 = 0.63 nM T16016 C42LID 72947880 IC50 = 1300 nM T16016 CWSX63 73345959 IC50 > 8333 nM T16016 CH0R4L 73347500 IC50 = 196 nM T16016 CBWU87 73349030 IC50 = 1800 nM T16016 C9E6RP 73350585 IC50 = 7.2 nM T16016 C15IOL 73353555 IC50 = 25000 nM T16016 CUA0J7 73353556 IC50 > 8333 nM T16016 CR79ZO 73353557 IC50 > 8333 nM T16016 CJ3L5M 73355055 IC50 = 3.7 nM T16016 C7V1JG 76311396 IC50 = 9100 nM T16016 CH7B9N 76311400 IC50 = 260 nM T16016 CGP1F3 76315009 IC50 = 5700 nM T16016 C5IJN1 76318623 IC50 = 12700 nM T16016 C4TYD3 76322249 IC50 = 10000 nM T16016 C2YJR4 76322269 IC50 = 10000 nM T16016 CR4IO8 76325891 IC50 = 4000 nM T16016 CW12KH 76336764 IC50 = 260 nM T16016 CP3C1F 118714001 IC50 = 2 nM T16016 C3P4VQ 118714034 IC50 = 11 nM T16016 C79CKF 118714035 IC50 = 2 nM T16016 CFB78G 118714036 IC50 = 2 nM T16016 CM5F8Z 118714037 IC50 = 2 nM T16016 C2KET6 118714038 IC50 = 2 nM T16016 C5I8EN 134817249 IC50 > 30000 nM T16016 C4Z3XS 145983516 IC50 > 30000 nM T16016 C9NDM5 145983631 IC50 > 30000 nM T16016 C3ZPR5 145985518 IC50 > 30000 nM T16016 CHTY23 145985766 IC50 > 30000 nM T16016 C54YUG 155511496 IC50 > 3000 nM T16016 C3CJ8L 155511620 IC50 = 10 nM T16016 C7R1SZ 155513751 Ki = 40.74 nM T16016 CM7Y9H 155514261 Ki = 50 nM T16016 C7HW9V 155514720 IC50 > 3000 nM T16016 CW1K9P 155515101 IC50 > 3000 nM T16016 CDI07N 155515240 IC50 > 3000 nM T16016 CT45DJ 155515471 IC50 > 3000 nM T16016 CZ29FQ 155521447 Ki = 5 nM T16016 CNH6D0 155522863 IC50 > 3000 nM T16016 C8Q0SV 155526212 IC50 = 350 nM T16016 CW0R6Z 155526680 Ki = 64.57 nM T16016 C86PTC 155528640 IC50 > 3000 nM T16016 CA6QL2 155529800 IC50 > 3000 nM T16016 CDRM08 155530458 IC50 = 1200 nM T16016 C15NKD 155532102 Ki = 181 nM T16016 C7KI0H 155533083 IC50 > 3000 nM T16016 CTW3H0 155533145 IC50 = 1900 nM T16016 CF6DQ7 155535265 Ki = 18.2 nM T16016 CM5R3Q 155538641 IC50 > 3000 nM T16016 CR0A2Y 155538947 IC50 = 28 nM T16016 CE5SU4 155539148 Ki = 30 nM T16016 C0KX7I 155539505 IC50 > 3000 nM T16016 CSP9L2 155543214 IC50 > 3000 nM T16016 COK7D3 155544726 IC50 = 1700 nM T16016 C4J1ZL 155545804 Ki = 31 nM T16016 C0D3CS 155547454 IC50 > 3000 nM T16016 C62DPU 155548977 Ki = 77 nM T16016 CIU9M4 155549273 IC50 = 960 nM T16016 C8DX4C 155549724 IC50 = 500 nM T16016 C0QHR1 155549943 IC50 > 3000 nM T16016 C80MNA 155553428 Ki = 198 nM T16016 C05PNE 155554350 IC50 > 3000 nM T16016 CHX96A 155556819 IC50 > 3000 nM T16016 C7X6VW 155559153 Ki = 27.54 nM T16016 CDUT06 155561022 Ki = 194.98 nM T16016 CC1JE8 155561040 IC50 = 420 nM T16016 CDS87R 155562877 IC50 = 2100 nM T16016 C2KB9Y 155564974 IC50 = 13 nM T16016 CMZ94A 155565119 IC50 > 3000 nM T16016 CY1BK9 155565496 IC50 > 3000 nM T16016 CT6P7E 155566515 IC50 > 3000 nM T16016 CV8IG3 155568751 IC50 > 3000 nM T16016 CT27HO 155569186 IC50 > 3000 nM T16016 D01JZV 9913085 IC50 = 1900 nM T16016 D05XZF 512282 Ki = 1 nM T16016 D06QRP 5311123 IC50 = 39 nM T16016 D0FF6S 16038374 IC50 > 10000 nM T38200 D0ED7U 60648 IC50 = 917000 nM T38200 D08ESA 198693 IC50 = 333000 nM T38200 D0C9XA 119 IC50 = 1000 nM T38200 CJ9V4G 40598 IC50 > 1000000 nM T38200 CXSD61 155246 IC50 = 43700 nM T38200 CHV0G9 639062 IC50 > 1000000 nM T38200 C97FYX 702501 IC50 > 300000 nM T38200 C8X9TQ 1069892 Ki > 100000 nM T38200 C1A0UL 1502074 IC50 = 2300 nM T38200 C3DR8J 1502075 IC50 = 2511.89 nM T38200 C9EI4M 1530639 IC50 > 1000000 nM T38200 CU23IC 4531494 IC50 = 10000 nM T38200 CG1ZF6 5311322 Ki = 6100 nM T38200 CN2C7Q 6604883 IC50 = 86000 nM T38200 C4A6SU 8181355 IC50 > 500000 nM T38200 CQ64IH 9797818 IC50 = 1990000 nM T38200 C31HNE 9884272 Ki > 100000 nM T38200 CY2IS7 9888224 IC50 = 46000 nM T38200 CI06JL 9982662 IC50 = 198000 nM T38200 CTZ5Q7 9983570 IC50 = 1080000 nM T38200 C75BDY 10031163 IC50 = 212000 nM T38200 CZ4PO2 10050339 IC50 = 6740000 nM T38200 CZQ52G 10052359 IC50 = 169000 nM T38200 CP2WF1 10072112 IC50 = 142000 nM T38200 CG1A4H 10073933 IC50 = 25000 nM T38200 C57RVK 10075407 IC50 = 142000 nM T38200 C4S1CO 10096504 IC50 = 25000 nM T38200 CXJR61 10252950 IC50 = 178000 nM T38200 CC8V4E 10412575 IC50 = 20000 nM T38200 CZ8FQ2 10481573 IC50 = 29000 nM T38200 CU40KP 11743493 IC50 = 91000 nM T38200 CH6GX1 13314232 IC50 > 500000 nM T38200 C03OAI 14810154 IC50 = 8128.31 nM T38200 C6VK4E 17173775 IC50 > 1000000 nM T38200 CE92MX 17174058 IC50 > 1000000 nM T38200 C3OQD7 17250318 IC50 > 500000 nM T38200 CME93B 43345728 IC50 > 1000000 nM T38200 C5JUW9 47058964 IC50 > 1000000 nM T38200 CLIK30 50941729 IC50 > 100000 nM T38200 CQ4XJ7 55285849 IC50 = 13900 nM T38200 CY9O8W 55285850 IC50 = 13900 nM T38200 C8UTR2 67642717 IC50 = 1900 nM T38200 C6ME5H 70684991 IC50 = 876000 nM T38200 C79CYX 70689234 IC50 = 2043000 nM T38200 CD9EV5 70691307 IC50 = 782000 nM T38200 CJ7P8C 70691309 IC50 = 3233000 nM T38200 C53QGB 118711599 IC50 = 76300 nM T38200 CO18BS 137635197 IC50 = 405000 nM T38200 CQL64H 137637846 IC50 > 1000000 nM T38200 CZ73DV 137638595 IC50 > 100000 nM T38200 CARI53 137638617 IC50 > 100000 nM T38200 CUM2T0 137638836 IC50 > 100000 nM T38200 C3PY5G 137638838 IC50 > 50000 nM T38200 CP7OV5 137639241 IC50 > 100000 nM T38200 C21IZT 137639281 IC50 > 1000000 nM T38200 CP24OX 137642163 IC50 > 100000 nM T38200 CK2VU3 137650102 IC50 > 1000000 nM T38200 C52PYO 137650910 IC50 > 1000000 nM T38200 CS6FX4 137651374 IC50 > 1000000 nM T38200 CPLJ94 137651669 IC50 > 1000000 nM T38200 CN04QK 137652511 IC50 > 1000000 nM T38200 CGC1Z4 137654858 IC50 > 50000 nM T38200 CADN74 137657292 IC50 > 100000 nM T38200 C4NK1W 137658990 IC50 > 50000 nM T38200 CPI4S8 137659917 IC50 > 50000 nM T38200 CI7S8H 155516242 IC50 > 100000 nM T38200 CL2TZ4 155518880 IC50 = 2754.23 nM T38200 C4U8QT 155524561 IC50 > 100000 nM T38200 CJ4OV6 155530359 IC50 > 100000 nM T38200 C4RL9X 155535776 IC50 > 100000 nM T38200 C7XS6Z 155549186 IC50 = 9332.54 nM T38200 CL2Q6G 155567178 IC50 > 100000 nM T38200 D02ANG 5216267 IC50 = 125892.54 nM T38200 D03IWW 6575389 IC50 = 2320000 nM T38200 D08YGM 92409 IC50 = 944000 nM T38200 D0D2EF 1796510 IC50 = 51000 nM T38200 D0H7WK 10458835 IC50 = 5000 nM T38200 D0P3KI 9888030 IC50 = 8920 nM T38200 D0RF2M 4498 IC50 = 106000 nM T38200 D0V5OY 16725912 Ki > 100000 nM T38200 D0V7RG 3532 IC50 = 110000 nM T38200 D0W8SX 239 IC50 = 41200 nM T38200 D0X3CF 442879 IC50 > 500000 nM T29355 D02VTV 117968550 EC50 = 1100 nM T29355 D03LZO 117967861 EC50 = 4400 nM T29355 C70QRI 1026354 IC50 = 64000 nM T29355 CJF29V 2965792 IC50 = 46500 nM T29355 CJ4ID2 3718032 IC50 = 38000 nM T29355 CBX8T9 16451230 IC50 > 200000 nM T29355 C85NAQ 24858111 EC50 = 900 nM T29355 CM4J7H 44379494 EC50 = 36000 nM T29355 CPL71I 54596764 IC50 > 100000 nM T29355 CER5F1 67466175 IC50 > 100000 nM T29355 CYB1U4 76318201 IC50 = 2800 nM T29355 CVM64R 117967504 EC50 = 1400 nM T29355 CJY5W0 117967660 EC50 = 6800 nM T29355 C9F3YV 117967663 EC50 = 1000 nM T29355 CM5N2A 117967691 EC50 = 3400 nM T29355 C2G4ND 117967705 EC50 = 1200 nM T29355 CY1V9T 117976066 EC50 = 4900 nM T29355 CY2R4J 117976176 EC50 = 300 nM T29355 CGQ82T 118732749 IC50 = 50000 nM T29355 CIZF42 122178085 IC50 > 50000 nM T29355 CR53MN 122186750 EC50 = 3000 nM T29355 CX3NU8 122186767 EC50 = 4000 nM T29355 CEW2X8 122186780 EC50 = 2100 nM T29355 C6G0CZ 122580323 EC50 = 1600 nM T29355 CU50GO 134154293 IC50 = 41000 nM T29355 CL0WR7 134386479 EC50 = 5400 nM T29355 C6GC0O 137028680 EC50 = 6200 nM T29355 CWMH49 137638632 EC50 = 1900 nM T29355 C05DFP 137653852 EC50 = 2100 nM T29355 C8LEV4 139267760 IC50 = 7600 nM T29355 CUVO30 155515610 EC50 = 2400 nM T29355 CX5G9E 155528619 EC50 = 5200 nM T29355 CS3PF1 155533577 EC50 = 4600 nM T29355 CRH9J5 155534178 EC50 = 5100 nM T29355 CAE51Q 155534378 EC50 = 4800 nM T29355 C29RHJ 155544579 EC50 = 5400 nM T29355 CIN57Q 155556138 IC50 = 74000 nM T29355 CB8SD4 155557649 EC50 = 8700 nM T29355 C0BU1J 155560963 EC50 = 5400 nM T29355 D02TVQ 71268957 IC50 > 100000 nM T29355 D09CLP 439155 IC50 > 50000 nM T01092 D05ROI 44462760 IC50 = 53200 nM T01092 D0H0EQ 24826799 IC50 = 12 nM T01092 D0W5HK 216239 IC50 = 1500 nM T01092 D02XNW 5494449 IC50 = 208 nM T01092 D0LQ3L 77108121 IC50 = 0.4 nM T01092 C09BCS 23578 Ki = 63.1 nM T01092 C76XNU 643953 IC50 = 754 nM T01092 C5IOS0 670041 EC50 = 4100 nM T01092 C7X5WE 2828334 EC50 = 182 nM T01092 C86MXJ 3063662 IC50 = 794 nM T01092 CDLJ02 3078467 IC50 = 2000 nM T01092 C8B3WY 3078469 IC50 = 2000 nM T01092 CMV76B 3078470 IC50 = 10 nM T01092 CYE04H 3078480 IC50 = 1.6 nM T01092 CZ4WV2 3670283 IC50 = 126 nM T01092 CA82YG 4628569 EC50 > 10000 nM T01092 CL70MG 4634732 EC50 = 457 nM T01092 C7TA9J 10113568 Ki = 2.042 nM T01092 CIV15Q 10113978 IC50 = 873 nM T01092 CFB81R 10317604 IC50 = 160 nM T01092 CF8Q2B 11288934 EC50 = 18 nM T01092 C8ET0Q 12791776 IC50 > 10000 nM T01092 CD2E5U 13142332 EC50 > 10000 nM T01092 C4V0BX 20895670 IC50 = 79 nM T01092 C25UKC 21081761 IC50 = 1500 nM T01092 CSFK63 23646936 IC50 = 32 nM T01092 CJ5H1Z 23646938 IC50 = 10 nM T01092 CIP7T2 23646939 IC50 = 2500 nM T01092 CI32JB 23646942 IC50 = 100 nM T01092 CX30ZW 25023828 IC50 = 73.6 nM T01092 C38PUJ 45271185 IC50 = 600 nM T01092 CS9T8F 53466952 IC50 = 61 nM T01092 C0HY3M 53467389 IC50 = 58 nM T01092 CLP04A 53467390 IC50 = 14 nM T01092 CV7C0D 53469060 IC50 = 69 nM T01092 CY04AP 53469630 IC50 = 56 nM T01092 CU4B0V 53469825 IC50 = 116 nM T01092 C5B4NV 55157876 EC50 = 1077 nM T01092 CKFP29 57971132 IC50 = 13 nM T01092 CUB9N0 60236671 EC50 = 378 nM T01092 CD8AV0 60698388 IC50 > 10000 nM T01092 CXIQ15 60723604 IC50 = 316 nM T01092 CVY1Z2 62679367 EC50 > 10000 nM T01092 CX30KT 62679368 EC50 = 8562 nM T01092 COQ08Y 62679370 EC50 = 1233 nM T01092 C9DYZ5 71816195 IC50 = 630 nM T01092 CY8O3K 72724969 IC50 = 20 nM T01092 CW7YD6 72725026 IC50 = 16 nM T01092 C5SQ7I 72725027 IC50 = 32 nM T01092 CFB69C 72725028 IC50 = 10 nM T01092 CE7G9T 72725029 IC50 = 4 nM T01092 CFR80L 72725083 IC50 = 160 nM T01092 COP05E 76310255 IC50 = 10 nM T01092 CHB93K 76313942 IC50 = 200 nM T01092 CCS63Z 76317480 IC50 = 40 nM T01092 CL0BO7 76317481 IC50 = 320 nM T01092 CFYP81 76317482 IC50 = 32 nM T01092 CFX5S0 76321210 IC50 = 4000 nM T01092 C7SD8Z 76321211 IC50 = 500 nM T01092 CKD2R6 76321212 IC50 = 63 nM T01092 C9X6CZ 76321213 IC50 = 160 nM T01092 C1EMH2 76321214 IC50 = 10 nM T01092 CW95IP 76324828 IC50 = 160 nM T01092 C35VHG 76328382 IC50 = 320 nM T01092 CUB91G 76328383 IC50 = 10 nM T01092 CAD50N 76328384 IC50 = 16 nM T01092 C4MT3A 76332057 IC50 = 25 nM T01092 C9IC1L 76332058 IC50 = 3200 nM T01092 C0K5MP 76332059 IC50 = 6.3 nM T01092 CO7J2V 76332061 IC50 = 16 nM T01092 CE09XW 76335674 IC50 = 200 nM T01092 CPUD78 77230897 IC50 = 1030 nM T01092 CB5H7C 82244347 IC50 > 10000 nM T01092 CC0US3 90345286 IC50 = 7.9 nM T01092 CM73SR 90345378 IC50 = 0.94 nM T01092 CNTP05 90345427 IC50 = 50 nM T01092 CS43ZG 90351311 Ki = 0.8 nM T01092 CR9ZV7 90351952 IC50 = 0.5 nM T01092 C4LT3Y 91885439 IC50 = 8.6 nM T01092 C28GLZ 110728326 IC50 > 1000 nM T01092 CF20OX 118557066 IC50 = 5 nM T01092 C6V5XY 118557110 IC50 = 0.4 nM T01092 C5ZQ4I 118557139 IC50 = 0.79 nM T01092 C78DEX 118557145 IC50 = 1600 nM T01092 C98CAG 118557162 IC50 = 0.4 nM T01092 CFJ27P 118557220 IC50 = 400 nM T01092 CSJR15 118557245 IC50 = 79 nM T01092 C21IGS 118557254 IC50 = 320 nM T01092 C3LR2H 118557293 IC50 = 1.6 nM T01092 CCYI79 118557322 IC50 = 0.79 nM T01092 CSD2H6 118557338 IC50 = 3.2 nM T01092 C5O4ZV 118557362 IC50 = 0.079 nM T01092 C6S0NT 118557462 IC50 = 63 nM T01092 CE8J7H 118557468 IC50 = 25 nM T01092 C02OGI 118557491 IC50 = 1 nM T01092 C42EMA 118557502 IC50 = 0.5 nM T01092 C12PXU 118557507 IC50 = 0.5 nM T01092 CS6JK9 118557559 IC50 = 794 nM T01092 CU7I5M 118564393 IC50 = 200 nM T01092 C2U3FR 118564396 IC50 = 32 nM T01092 CU0DW4 118564398 IC50 = 5 nM T01092 C7TBH3 118564402 IC50 = 0.32 nM T01092 C3KNZ5 121439991 EC50 = 28 nM T01092 CCX27F 121440014 EC50 = 74 nM T01092 CUR74H 121440015 EC50 > 3000 nM T01092 CH3CO4 121440032 EC50 = 262 nM T01092 CE0QC9 121440033 EC50 = 49 nM T01092 CJ0A5S 121440051 EC50 = 64 nM T01092 CLJI17 121446658 EC50 = 628 nM T01092 CY5A1S 121446659 EC50 = 125 nM T01092 C0HFX3 121446661 EC50 > 10000 nM T01092 C04IQZ 121446667 EC50 > 3000 nM T01092 C19DEL 121446676 EC50 = 490 nM T01092 C4FAO7 121446682 EC50 = 1234 nM T01092 CKUM01 121446684 EC50 = 56 nM T01092 CTM6K0 121446695 EC50 > 3000 nM T01092 CY61UA 121446710 EC50 = 1526 nM T01092 CWN4T7 121446721 EC50 = 1735 nM T01092 C0ZE8M 121446729 EC50 > 10000 nM T01092 CTXO48 121446730 EC50 = 898 nM T01092 C57TND 121446732 EC50 = 1254 nM T01092 CQH48Z 121446733 EC50 > 10000 nM T01092 CYTZ27 121446735 EC50 > 10000 nM T01092 C1ENL2 121446737 EC50 > 10000 nM T01092 CH68FX 121446738 EC50 = 221 nM T01092 C8SK7Y 121446739 EC50 = 628 nM T01092 C54DCI 121446741 EC50 > 10000 nM T01092 C1K5ZD 121446742 EC50 > 5000 nM T01092 CO32FQ 121446750 EC50 > 10000 nM T01092 C1FU2G 121446752 EC50 > 10000 nM T01092 CJ08HW 121446757 EC50 = 627 nM T01092 CX06JV 121446760 EC50 = 2527 nM T01092 C2ZF7V 121446761 EC50 = 8237 nM T01092 CB3I0L 121446764 EC50 = 656 nM T01092 C1H3VY 121446771 EC50 = 1308 nM T01092 C0B1WO 121446775 EC50 = 198 nM T01092 CU92HQ 121446778 EC50 = 58 nM T01092 C08KJZ 121446782 EC50 = 72 nM T01092 CVM06Q 121446783 EC50 = 36 nM T01092 CCD94Y 121446786 EC50 > 10000 nM T01092 CT8K2N 121446791 EC50 > 10000 nM T01092 C4NT5D 121446843 EC50 > 3000 nM T01092 CGP13F 121446847 EC50 = 12 nM T01092 CNH04D 121446878 EC50 = 98 nM T01092 C4QV9N 121446902 EC50 = 815 nM T01092 C8P4AE 122703561 IC50 = 10 nM T01092 C9E5DT 122703570 IC50 = 2 nM T01092 CM7C5F 122703576 IC50 = 7.9 nM T01092 CF5WY1 122703578 IC50 = 10 nM T01092 CF4PR9 122703579 IC50 = 16 nM T01092 C74SQF 122703581 IC50 = 13 nM T01092 CPA2Z5 122703584 IC50 = 10 nM T01092 CW70QA 122703585 IC50 = 63 nM T01092 CA6Z5C 122703586 IC50 = 10 nM T01092 CYIP81 122703588 IC50 = 10 nM T01092 C5LYJ9 122703599 IC50 = 126 nM T01092 CL7MB6 122703611 IC50 = 16 nM T01092 CJ3RT5 122703613 IC50 = 1.6 nM T01092 C6NT4C 122703637 IC50 = 10 nM T01092 C2TE3N 122703644 IC50 = 9 nM T01092 CP31IH 122703646 IC50 = 200 nM T01092 CIA2M8 122703656 IC50 = 6.3 nM T01092 CX7BC0 122703665 IC50 = 4 nM T01092 CKY5L7 122703666 IC50 = 316 nM T01092 C6R7MN 122703671 IC50 = 10 nM T01092 CAEG59 122703680 IC50 = 10 nM T01092 C8ODW1 122703682 IC50 = 10 nM T01092 CXA83K 122703688 IC50 > 10000 nM T01092 CR1C5H 122703691 IC50 = 4.8 nM T01092 CU7TI5 122703692 IC50 = 10 nM T01092 C27BKA 122703700 IC50 = 1.6 nM T01092 C26JOL 122703705 IC50 = 10 nM T01092 CR75IM 122703716 IC50 = 10 nM T01092 CEG87H 122703723 IC50 = 10 nM T01092 CG7RC6 122703734 IC50 = 398 nM T01092 CK2D8E 122703743 IC50 = 0.5 nM T01092 CZ6R3X 124086061 IC50 = 35 nM T01092 C9XVO7 124086067 IC50 = 10 nM T01092 C7MLB2 124086077 IC50 = 16 nM T01092 CJXY94 124180534 IC50 = 32 nM T01092 CY8JW7 127033346 IC50 > 10000 nM T01092 C3ASY7 127033640 IC50 = 35 nM T01092 C4BKW6 127033641 IC50 = 210 nM T01092 C1KNJ3 127033642 IC50 = 0.2 nM T01092 C1U6TC 130299179 IC50 = 631 nM T01092 C6IZ3V 130299401 IC50 = 3162 nM T01092 CNI1W2 132016672 IC50 = 79 nM T01092 CPF5E3 132471860 Ki = 0.912 nM T01092 CK4HX5 134521326 IC50 = 10 nM T01092 CRT5O7 134521520 IC50 = 8.5 nM T01092 C2E7AT 134521814 IC50 = 1 nM T01092 CG9R3J 134522007 IC50 = 10 nM T01092 CZB75S 134522265 IC50 = 2.5 nM T01092 CSCT10 134536604 IC50 = 7.9 nM T01092 CSL60X 135308861 Ki = 0.912 nM T01092 C0ZQP5 135308877 Ki = 1.738 nM T01092 CS1DF9 135308888 Ki = 13.8 nM T01092 CFX4W3 135308904 Ki = 251.19 nM T01092 CNF6O4 135308906 Ki = 1.778 nM T01092 C6M9FG 135308913 Ki = 2.57 nM T01092 CF1LY8 135308922 Ki = 6918.31 nM T01092 C3XG8C 135308924 Ki = 2.512 nM T01092 C8Z7AU 135308925 Ki = 1.148 nM T01092 C6EW1J 135308927 Ki = 3.467 nM T01092 C8NC5R 135308928 Ki = 2.951 nM T01092 C2C5TL 135308931 Ki = 4265.8 nM T01092 CZP1T3 135308934 Ki = 5.129 nM T01092 CNI5C3 135308946 Ki = 38.02 nM T01092 C8AVZ0 135308996 Ki = 3.89 nM T01092 CSOZ57 135309005 Ki = 7.943 nM T01092 CGFM04 135309027 Ki = 117.49 nM T01092 CQIU03 135309039 Ki = 107.15 nM T01092 CRJ8H5 135309049 Ki = 54.95 nM T01092 C5GAV8 135309066 Ki = 0.8511 nM T01092 CZ53KU 135309069 Ki = 33.88 nM T01092 CA28GI 135309090 Ki = 0.4074 nM T01092 CI8Z2F 135309102 Ki = 1.148 nM T01092 C5E6UB 135314480 IC50 = 39.81 nM T01092 CXC69T 137321158 IC50 = 11 nM T01092 CVGN14 137632484 IC50 = 0.05 nM T01092 C8PV3G 137632977 IC50 > 10000 nM T01092 COL6Q7 137634539 IC50 = 12600 nM T01092 C1FTS9 137634957 IC50 > 10000 nM T01092 C5KYE7 137635049 IC50 = 100 nM T01092 C3EIS6 137635629 IC50 = 0.4 nM T01092 CA8GF2 137637401 IC50 = 2468 nM T01092 CQ32NB 137638108 EC50 > 10000 nM T01092 C58MXE 137640092 IC50 = 2 nM T01092 C5B9NR 137640099 IC50 = 501 nM T01092 CZS13Q 137640111 IC50 = 295 nM T01092 C62DVJ 137640435 EC50 > 3000 nM T01092 CGC9T1 137641614 IC50 > 10000 nM T01092 CESF45 137644276 IC50 = 167 nM T01092 C4TBJ8 137647324 IC50 > 10000 nM T01092 CLP5H9 137647405 IC50 = 0.63 nM T01092 C4JH8A 137647835 IC50 > 10000 nM T01092 CYP70I 137651336 IC50 > 10000 nM T01092 CCK03W 137652965 IC50 > 10000 nM T01092 CKX2D8 137654471 IC50 > 10000 nM T01092 CRH18Z 137656846 IC50 = 178 nM T01092 CP51KG 137657894 IC50 = 1259 nM T01092 CFH52E 137659234 IC50 = 251 nM T01092 C3BCN1 138377545 IC50 = 0.3 nM T01092 CGX92C 138393291 IC50 = 5500 nM T01092 CCT23N 141340950 IC50 > 15000 nM T01092 CTS9Q8 142416001 IC50 = 2.512 nM T01092 CFGH25 142416011 IC50 = 10 nM T01092 C2X1CR 145978863 IC50 = 190 nM T01092 C85UBM 145978937 IC50 = 10 nM T01092 CAW7B1 145980780 IC50 = 468 nM T01092 C43ZUJ 145981140 IC50 = 49 nM T01092 C10HDT 145981335 IC50 = 134 nM T01092 C8DKN3 145981423 IC50 = 94 nM T01092 C89BNR 145982306 IC50 = 531 nM T01092 CO57FT 145982439 IC50 = 3457 nM T01092 CUZQ37 145985171 IC50 = 704 nM T01092 C41ZBR 145986358 IC50 = 105 nM T01092 C4D8HB 145986929 IC50 = 18 nM T01092 C3FN9P 145987011 IC50 = 424 nM T01092 CST1O6 145987202 IC50 = 31 nM T01092 CGM18W 145987557 IC50 = 10 nM T01092 CAC0M7 145988480 IC50 = 13 nM T01092 C7DWU4 145988653 IC50 = 26 nM T01092 CUJL09 145988701 IC50 = 77 nM T01092 C58ULD 145988885 IC50 = 49 nM T01092 CVH28K 145989341 IC50 = 128 nM T01092 COTX64 145989416 IC50 = 2994 nM T01092 C8VND5 145989851 IC50 = 10 nM T01092 C4P8HQ 145990145 IC50 = 264 nM T01092 CZ0RI5 145990208 IC50 = 107 nM T01092 CGF6E4 145990858 IC50 = 17 nM T01092 C96XWF 145991904 IC50 = 28 nM T01092 C3D6OB 145992043 IC50 = 79 nM T01092 CAOQ30 145992060 IC50 = 392 nM T01092 C1NYL4 145993423 IC50 = 634 nM T01092 C05WAM 146344085 IC50 = 90 nM T01092 CN7MS2 154023591 IC50 = 5 nM T01092 CKW68P 155393270 IC50 = 7940 nM T01092 CS0T6E 155510707 IC50 = 17000 nM T01092 C37FPZ 155510738 IC50 > 15000 nM T01092 CX0T1C 155512182 IC50 = 10 nM T01092 C0AUE4 155512296 IC50 = 10 nM T01092 COA84W 155512492 IC50 = 200 nM T01092 C23DJP 155512860 IC50 = 19.95 nM T01092 C2MD1Q 155513187 IC50 > 10000 nM T01092 CZ7K6H 155513660 IC50 > 15000 nM T01092 CC3T0M 155518699 IC50 = 10 nM T01092 CWZ5J8 155519113 IC50 = 5012 nM T01092 CXD9M4 155520427 IC50 = 10 nM T01092 C4FW0B 155522577 IC50 = 6.3 nM T01092 CLW39S 155522794 IC50 = 10 nM T01092 CQIR50 155523679 IC50 = 200 nM T01092 C9M2ZT 155523831 IC50 = 10 nM T01092 CPK67I 155524868 IC50 = 180 nM T01092 CJ3M5T 155524881 IC50 > 1000 nM T01092 CU9H3G 155525351 Ki = 21 nM T01092 C1ICR3 155529856 IC50 > 10000 nM T01092 CIP84Q 155530191 IC50 = 90 nM T01092 C0V9QN 155532882 IC50 > 15000 nM T01092 CTJ84E 155533767 IC50 = 1.3 nM T01092 CQOE59 155534156 IC50 = 310 nM T01092 CF09IN 155535999 IC50 = 10 nM T01092 C8JR2S 155537020 IC50 = 20.8 nM T01092 CSU48D 155537554 IC50 = 10 nM T01092 CZR0J9 155537757 IC50 = 11000 nM T01092 CTP72E 155538424 IC50 = 200 nM T01092 CZ80HO 155547269 IC50 = 10 nM T01092 CSQ28H 155548887 IC50 = 2.5 nM T01092 C5L7HY 155551127 IC50 > 15000 nM T01092 CQ92XF 155552769 IC50 = 126 nM T01092 CDT06B 155555771 IC50 = 600 nM T01092 CL2CH8 155556595 IC50 = 10 nM T01092 C4Z8UW 155569299 IC50 = 1.3 nM T01092 D0K8YD 76332060 IC50 = 16 nM T01092 D0N4LR 53469448 IC50 = 18 nM T99149 D04XVN 11707110 IC50 = 1.6 nM T99149 D0E3TC 44259 IC50 = 37.4 nM T99149 D0K0YC 9826528 IC50 = 110 nM T99149 D0A9KI 9863367 IC50 > 50 nM T99149 C8KED5 4713 IC50 = 50000 nM T99149 CQ7PL4 1235170 IC50 > 20000 nM T99149 C5VPH9 16129448 IC50 = 391 nM T99149 C0H8UN 16730109 IC50 > 30000 nM T99149 C6P1CX 25066843 IC50 > 20000 nM T99149 C3VRO9 44557921 IC50 > 10000 nM T99149 CIPX17 45485590 Ki = 9700 nM T99149 CI10RQ 45485600 Ki = 13000 nM T99149 CPVU61 45485609 Ki = 6200 nM T99149 C58VXQ 45485625 Ki = 710 nM T99149 CMI83V 45485640 Ki = 2400 nM T99149 CP87FU 45485645 Ki = 1400 nM T99149 CLJF04 45485646 Ki = 1800 nM T99149 CQE7Z0 45485654 Ki = 3700 nM T99149 C5J4CW 45485664 Ki = 1400 nM T99149 C63VLU 45485665 Ki = 1800 nM T99149 C7VRC1 45485666 Ki = 2100 nM T99149 CK8Q9R 45485676 Ki = 16000 nM T99149 C7SX0U 45485677 Ki = 670 nM T99149 C4UB6E 45485687 Ki = 1400 nM T99149 CRA74I 49842779 IC50 = 6840 nM T99149 C37NKO 67129970 IC50 > 10000 nM T99149 CK80LJ 67130050 IC50 > 10000 nM T99149 CV63UL 67240318 IC50 > 10000 nM T99149 C7GRV2 68755406 IC50 > 10000 nM T99149 C2LAM7 126591927 IC50 = 82 nM T99149 CI2YE9 132606873 IC50 = 186.7 nM T99149 C0TE5S 135651612 IC50 = 1300 nM T99149 CI1E8V 137634241 IC50 > 10000 nM T99149 CU62AO 145712394 IC50 = 590 nM T99149 C6VB3O 145925651 IC50 >= 5000 nM T99149 C2MD1Q 155513187 IC50 > 10000 nM T99149 C4NKP6 155518298 IC50 = 1500 nM T99149 C86HPW 155518524 IC50 = 74000 nM T99149 D08LYB 5166 IC50 > 50 nM T99149 D0GD8Y 3006531 IC50 = 58 nM T48780 CZ7HO2 24139 IC50 = 125892.54 nM T48780 CSO4E3 644170 IC50 = 1000000000 nM T48780 C0FSW1 2733653 IC50 = 4.3 nM T48780 CDPK78 7177184 IC50 = 1000000000 nM T48780 CNC34Y 11182549 IC50 = 0.5012 nM T48780 C7HF4C 13018787 IC50 = 630957.34 nM T48780 CD7TM6 15423759 IC50 = 398107.17 nM T48780 C90UTG 15471714 IC50 = 12.59 nM T48780 CUB5A3 16182677 IC50 = 63.1 nM T48780 C3TJZ4 46233136 IC50 = 14 nM T48780 CRK14X 46233137 IC50 = 251188.64 nM T48780 CXYW80 46233138 IC50 = 79432.82 nM T48780 C0EO5S 46233140 IC50 = 79.43 nM T48780 CZ7UL4 46233142 IC50 = 31622.78 nM T48780 C8ZC9X 49798491 IC50 = 3981.07 nM T48780 CSRN46 49863275 IC50 = 501187.23 nM T48780 CQT6X8 49863277 IC50 = 31622.78 nM T19531 C71SIH 253167 IC50 > 200000 nM T19531 CWC34Q 259205 IC50 > 200000 nM T19531 C8QM7B 6852376 EC50 = 80 nM T19531 CAD72T 9817518 IC50 = 10800 nM T19531 CZTH29 9834991 IC50 = 78000 nM T19531 CR52JI 9910619 IC50 = 7.2 nM T19531 CB3I8J 10014327 IC50 = 7900 nM T19531 CXZ8F3 10469457 IC50 = 13600 nM T19531 C2FP5Q 10617830 IC50 > 200000 nM T19531 CXMT71 10858184 IC50 > 200000 nM T19531 CA2ZN5 10869068 IC50 = 4600 nM T19531 CUM3X1 10912229 IC50 > 200000 nM T19531 C3VSN6 10912305 IC50 = 200 nM T19531 CQ4J5L 10934245 IC50 > 100000 nM T19531 CTX59A 10934704 IC50 = 600 nM T19531 C51JOG 10945208 IC50 > 200000 nM T19531 CQ45ND 10956699 IC50 = 16300 nM T19531 C72IAN 10989023 IC50 = 4900 nM T19531 CC4K0Z 10989442 IC50 = 400 nM T19531 CR7VM3 11000246 IC50 = 2600 nM T19531 CL06OV 11021644 IC50 > 200000 nM T19531 C8IO0S 11032616 IC50 = 188000 nM T19531 CM5XW9 11043528 IC50 = 28800 nM T19531 CK0IO4 11054944 IC50 = 55000 nM T19531 C3TOQ4 11086961 IC50 = 4300 nM T19531 CH91TK 11097296 IC50 = 100000 nM T19531 C7OTX5 11108129 IC50 > 70000 nM T19531 C5I0MZ 11139808 IC50 = 8200 nM T19531 C3NEH9 11776872 IC50 = 7600 nM T19531 CN4SE5 11780214 IC50 = 73200 nM T19531 CIX40T 11780786 IC50 = 9400 nM T19531 CUVM56 11832149 IC50 > 200000 nM T19531 C4R9QU 11832661 IC50 = 25100 nM T19531 CTM46O 14787969 EC50 = 210 nM T19531 CS6BV5 44309263 IC50 = 35400 nM T19531 CPA3N4 44335158 IC50 > 200000 nM T19531 CZM7L2 44335253 IC50 > 200000 nM T19531 CC5D0B 44335255 IC50 > 200000 nM T19531 CS75WN 44335277 IC50 > 200000 nM T19531 CCH3Y5 44335278 IC50 = 15300 nM T19531 CX7S8F 44335279 IC50 > 200000 nM T19531 CAQ09P 44335291 IC50 > 200000 nM T19531 C73QWO 44335292 IC50 > 200000 nM T19531 C2DX5B 44335293 IC50 > 200000 nM T19531 C8RME2 44335295 IC50 > 200000 nM T19531 CEY06B 44335296 IC50 > 200000 nM T19531 CV51XU 44335303 IC50 > 200000 nM T19531 COHV64 44335304 IC50 > 200000 nM T19531 C3T8LU 44335305 IC50 > 200000 nM T19531 CXT80K 44335306 IC50 > 200000 nM T19531 CB2HR3 44335308 IC50 > 200000 nM T19531 C2VU5P 44335316 IC50 > 200000 nM T19531 CLJ93K 44335335 IC50 = 140500 nM T19531 C60VLZ 44335352 IC50 > 200000 nM T19531 C47QRL 44335393 IC50 = 94000 nM T19531 C84RSA 44335432 IC50 > 200000 nM T19531 CCJB21 44335433 IC50 > 200000 nM T19531 CU25TG 44335465 IC50 > 200000 nM T19531 C1Y6QO 44335470 IC50 > 200000 nM T19531 C2JTN3 44335685 IC50 > 200000 nM T19531 CLK79Y 44335691 IC50 > 200000 nM T19531 C93OIU 44335698 IC50 > 200000 nM T19531 CIGM53 44335700 IC50 = 72000 nM T19531 C3MWY8 44335701 IC50 = 110000 nM T19531 CF7MS0 44335709 IC50 = 13600 nM T19531 CY8E2J 44335711 IC50 > 200000 nM T19531 CH5J4P 44335712 IC50 = 78000 nM T19531 CI4R0U 44335725 IC50 = 79000 nM T19531 CD7LE2 44335742 IC50 = 102000 nM T19531 C68TLS 44335939 IC50 = 98000 nM T19531 CGBF56 44335982 IC50 = 10800 nM T19531 C3NA5F 44461049 EC50 = 8 nM T97174 C13QNP 65127 IC50 = 23000 nM T97174 CAO2X9 25169386 IC50 = 150000 nM T97174 C5TBY8 25169388 IC50 = 71000 nM T97174 CVX2B3 25169390 IC50 = 22000 nM T97174 COXH93 44589903 IC50 = 230000 nM T31543 D05EAM 4735 Ki = 1160 nM T31543 D07XHO 4413 Ki = 0.02 nM T31543 D0KG3R 9875401 Ki = 3350 nM T31543 C2KE5Q 1508 Ki = 60000 nM T31543 CUSM50 11974 Ki = 535 nM T31543 C5P3TH 65130 Ki = 924 nM T31543 CZ1QL5 411406 Ki = 191 nM T31543 CB9VP7 432298 Ki = 200 nM T31543 C8VB4U 480183 Ki = 719 nM T31543 CROX25 480185 Ki = 397 nM T31543 CO5Y7H 725447 IC50 = 111000 nM T31543 CPJ28H 828532 IC50 = 420 nM T31543 CJ1GN3 869194 IC50 = 98000 nM T31543 CBFT53 975107 IC50 > 30000 nM T31543 CQUP23 2208579 IC50 = 75000 nM T31543 C97ZIP 2262135 IC50 = 120000 nM T31543 C74DMH 2262990 IC50 = 103000 nM T31543 CQPJ74 2938648 IC50 > 30000 nM T31543 C4S9WR 3000497 Ki = 816 nM T31543 C4Z0XK 3010932 Ki = 2280 nM T31543 C6WU4N 5000438 IC50 > 30000 nM T31543 CQ26VM 5289531 Ki = 170 nM T31543 CHY56L 5729350 IC50 = 138000 nM T31543 CI69XU 5739522 IC50 = 128000 nM T31543 CN2B6S 6852211 Ki = 4.3 nM T31543 CKDP84 9895193 Ki = 320 nM T31543 CDT95S 9939426 Ki = 370 nM T31543 CEC95B 9997816 Ki = 9600 nM T31543 CB1S5N 11363919 Ki = 7180 nM T31543 CJZ09N 11512593 Ki = 340 nM T31543 C28BMR 11513105 Ki = 13 nM T31543 CRNU10 11534959 Ki = 50 nM T31543 CD1A6T 11542037 Ki = 61 nM T31543 CA8KD7 11542038 Ki = 65 nM T31543 CBP69L 11557024 Ki = 1.8 nM T31543 CCG84F 11563457 Ki = 89 nM T31543 CV46NL 11563632 Ki = 730 nM T31543 CEAZ46 11569930 Ki = 160 nM T31543 C3TJ7M 11570580 Ki = 88 nM T31543 C6RHD8 11570700 Ki = 1.5 nM T31543 C1DN2L 11570759 Ki = 690 nM T31543 C6FG8V 11577055 Ki = 110 nM T31543 CIY34V 11577968 Ki = 200 nM T31543 CJ38EP 11577970 Ki = 690 nM T31543 C7MF9N 11578158 Ki = 89 nM T31543 CTSK74 11584729 Ki = 3.8 nM T31543 C1RQ6P 11592130 Ki = 3.9 nM T31543 CBC84M 11592593 Ki = 140 nM T31543 C7ZS8L 11592600 Ki = 44 nM T31543 C7QTY8 11606981 Ki = 4.2 nM T31543 CU07NO 11607091 Ki = 100 nM T31543 CL9TZ2 11614477 Ki = 140 nM T31543 CB4O2Q 11621579 Ki = 61 nM T31543 CD3R1E 11627899 Ki = 75 nM T31543 CB9P0Q 11628768 Ki = 8.7 nM T31543 CO3Q9N 11635973 Ki = 330 nM T31543 CRX98P 11636026 Ki = 53 nM T31543 CW10CL 11642802 Ki = 45 nM T31543 C2W5XF 11656797 Ki = 28 nM T31543 C4SAR0 11657278 Ki = 1500 nM T31543 CVQ16C 11664107 Ki = 42 nM T31543 CPZG49 11664334 Ki = 400 nM T31543 CT9E0G 11664643 Ki = 57 nM T31543 CWV87X 11671266 Ki = 5 nM T31543 CE0A6N 11671776 Ki = 96 nM T31543 C85GCY 11671956 Ki = 130 nM T31543 C1DHO6 11678360 Ki = 120 nM T31543 C4IBO3 11678764 Ki = 13 nM T31543 C69YSR 11693028 Ki = 380 nM T31543 CCQY30 11693049 Ki = 21 nM T31543 CPFW75 11699600 Ki = 72 nM T31543 C3VS2H 11699903 Ki = 53 nM T31543 CNV09Z 11699913 Ki = 38 nM T31543 CKQ4O2 11721188 Ki = 210 nM T31543 C4UB2X 11721375 Ki = 250 nM T31543 CRD97T 14477068 Ki > 10000 nM T31543 C1Z9SX 24776379 Ki = 200 nM T31543 CAO2V4 25030840 Ki = 7.5 nM T31543 CU82IO 25030929 Ki = 3 nM T31543 C7MCT6 25031099 Ki = 37 nM T31543 C5PO7A 25031100 Ki = 255 nM T31543 CH7Z1K 25031101 Ki = 12 nM T31543 CEW9X2 25031102 Ki = 6.1 nM T31543 C9NC4S 25031541 Ki = 33 nM T31543 CK5R8Q 25032200 Ki = 13 nM T31543 CG8HY2 25032202 Ki = 31 nM T31543 CH76XK 25032204 Ki = 65 nM T31543 CG76TR 25181493 Ki = 7 nM T31543 CA81RS 44144381 Ki = 220 nM T31543 CMZ05T 44324727 Ki = 40500 nM T31543 CE9I1R 44362422 Ki = 1800 nM T31543 CF5XO4 44413343 Ki = 84 nM T31543 CTD42X 44413355 Ki = 240 nM T31543 C9KQM2 44413356 Ki = 26 nM T31543 CQDX92 44413619 Ki = 100 nM T31543 CBSG69 44413636 Ki = 82 nM T31543 CU4AE5 44436348 Ki = 0.92 nM T31543 CVI26C 44436349 Ki = 4750 nM T31543 CZX07Q 44436350 Ki > 250000 nM T31543 C3X8OV 44436352 Ki = 90000 nM T31543 C9MOC3 44436353 Ki = 22500 nM T31543 CZF8M1 44436354 Ki = 28000 nM T31543 C3PGJ7 44436356 Ki = 107000 nM T31543 CRP6D7 44436357 Ki = 2330 nM T31543 CDI8A3 44436358 Ki = 450 nM T31543 C64FDS 44436359 Ki = 1000 nM T31543 C7PN9C 44436360 Ki = 890 nM T31543 C1RZ4Y 44436365 Ki = 857 nM T31543 CPEM68 44436366 Ki = 380 nM T31543 C8LQS9 44436368 Ki = 160 nM T31543 CEW6G1 44569299 Ki = 0.08 nM T31543 C9JNT3 44569300 Ki = 28 nM T31543 C9XE7Q 44569301 Ki = 56 nM T31543 CZI8D7 44569333 Ki = 2800 nM T31543 CK9YI3 44569356 Ki = 10000 nM T31543 C7XE6N 44569357 Ki > 1000000 nM T31543 C5ZG0T 44569358 Ki > 1000000 nM T31543 CR4CP6 44569359 Ki = 145 nM T31543 C9JF7W 44569667 Ki = 1 nM T31543 C61IJB 44569732 Ki = 6.7 nM T31543 CR36MB 44569733 Ki = 120 nM T31543 CE25UL 44569767 Ki = 180 nM T31543 C0CZ4I 44569768 Ki = 41 nM T31543 CIR4M0 44569769 Ki = 110 nM T31543 C02SHD 44569811 Ki = 29 nM T31543 CG3LE9 44569812 Ki = 91 nM T31543 CCU7V0 44569813 Ki = 26 nM T31543 C8BR6E 44569843 Ki = 6 nM T31543 C7Q9BH 44569844 Ki = 12 nM T31543 CZ35OW 44569845 Ki = 5.4 nM T31543 CHV9C1 44569846 Ki = 2.5 nM T31543 C5JQ4W 44569889 Ki = 60 nM T31543 CE1O4I 44569890 Ki = 47 nM T31543 C4JU7I 44569891 Ki = 13 nM T31543 CGS83Z 44569892 Ki = 1.6 nM T31543 C4BN3H 44573109 Ki = 6.3 nM T31543 COR57Y 44573272 Ki = 53 nM T31543 C6DX3Y 44573273 Ki = 17 nM T31543 CM2R1P 44573274 Ki = 53 nM T31543 CSP1I0 44573310 Ki = 150 nM T31543 C6EG9V 44573311 Ki = 180 nM T31543 CYV3X2 44573378 Ki = 470 nM T31543 CWUA41 44573379 Ki = 100 nM T31543 CYA64G 44573380 Ki = 2400 nM T31543 CLG42S 44573428 Ki = 11000 nM T31543 C4RSI0 46899736 Ki = 770 nM T31543 CX0Y2G 46899738 Ki = 2100 nM T31543 CLC94G 46918674 Ki = 972.9 nM T31543 C54AGL 46918753 Ki = 1710.7 nM T31543 CG7K0O 46937165 Ki = 457 nM T31543 CXUM36 49820499 Ki = 200 nM T31543 CX7SA8 49820500 Ki = 40 nM T31543 CQ3R6L 49820501 Ki = 200 nM T31543 CSFD83 49820654 Ki = 1200 nM T31543 CS8FY6 49820655 Ki = 545 nM T31543 C6OIW8 49820657 Ki = 600 nM T31543 CJ5G9Q 49820816 Ki = 1131 nM T31543 CL8UV3 49820969 Ki = 40 nM T31543 C2B5EC 49820973 Ki = 301 nM T31543 CAM3V7 50939649 Ki = 2 nM T31543 CHC74O 50939651 Ki = 23 nM T31543 CSAQ19 66818162 Ki = 40 nM T31543 COAY94 66818433 Ki = 1790 nM T31543 CG9UM3 66818450 Ki = 141 nM T31543 CG0TZ3 66818504 Ki = 1982 nM T31543 CU6E0A 66818541 Ki = 3 nM T31543 C89BXR 66818555 Ki = 400 nM T31543 C6LD2R 66818559 Ki = 10 nM T31543 C6CP8D 66818568 Ki = 6 nM T31543 CKD8I1 66818569 Ki = 10 nM T31543 C05LHZ 66818575 Ki = 592 nM T31543 CDA2M4 66818582 Ki = 1698 nM T31543 C9LTK3 66818589 Ki = 500 nM T31543 C9FQY8 66818629 Ki = 2032 nM T31543 C9GM3F 66818639 Ki = 260 nM T31543 C4U7SZ 66818677 Ki = 18 nM T31543 CL8D0V 66818717 Ki = 18 nM T31543 C41RKZ 66818743 Ki = 200 nM T31543 C6Q8FO 66818744 Ki = 411 nM T31543 CE53KG 66818763 Ki = 1060 nM T31543 CJA30C 66818765 Ki = 204 nM T31543 C5LU1Z 66818766 Ki = 1 nM T31543 CR94HZ 66818781 Ki = 1850 nM T31543 CP18VA 66818813 Ki = 770 nM T31543 CF4PT6 66818819 Ki = 824 nM T31543 CYB76J 66818882 Ki = 116 nM T31543 CRH5O7 66818889 Ki = 100 nM T31543 CGI6B3 66819113 Ki = 61 nM T31543 C4JV1L 66820910 Ki = 730 nM T31543 C62LDA 66821311 Ki = 94 nM T31543 CK59IZ 68788696 Ki = 1617 nM T31543 CGA3T2 68789018 Ki = 3 nM T31543 CC0J3V 68790735 Ki = 23 nM T31543 C5S0OC 70682854 Ki = 0.088 nM T31543 CUM4H3 70684929 Ki = 6124 nM T31543 CAU0K6 70689168 Ki = 9.5 nM T31543 C70YQU 70689169 Ki = 1.4 nM T31543 C47HLV 70689173 Ki = 4.6 nM T31543 CVD3W9 71495381 Ki = 13 nM T31543 CNVH43 71495466 Ki = 13 nM T31543 CA5N2S 71495467 Ki = 51 nM T31543 CQ98NY 71495468 Ki = 120 nM T31543 CE15GB 71495559 Ki = 130 nM T31543 CW1Y2L 71495560 Ki = 52 nM T31543 C5Q9BD 71495561 Ki = 33 nM T31543 C36MRI 71495659 Ki = 8 nM T31543 C7PDA9 71495660 Ki = 1 nM T31543 CF3C8E 71495661 Ki = 11 nM T31543 CECD13 71495765 Ki = 74 nM T31543 C7LXK1 71495766 Ki = 18 nM T31543 CKQ82B 71495974 Ki = 14 nM T31543 CSV38K 71495975 Ki = 56 nM T31543 C7QPA0 71495976 Ki = 35 nM T31543 CI4P9Z 71495977 Ki = 39 nM T31543 CE03BA 71496089 Ki = 8 nM T31543 CLO24G 71496201 Ki = 14 nM T31543 CIE7A6 71496202 Ki = 26 nM T31543 CAM0I4 71496204 Ki = 120 nM T31543 C5MVT3 76310068 Ki = 2900 nM T31543 CWZA05 76320988 Ki = 40 nM T31543 CV7IW5 87167024 Ki = 793 nM T31543 CMC3L7 89399327 Ki = 11 nM T31543 CJ6CN0 90644019 Ki = 591 nM T31543 CB8KY3 90644020 Ki = 1182 nM T31543 CB3Z7W 90644021 Ki = 0.08 nM T31543 C0G6SP 90644022 Ki = 305 nM T31543 CH3US6 90644023 Ki = 470 nM T31543 C1SAZ8 90666139 Ki = 49 nM T31543 C2ERV8 90666140 Ki = 7 nM T31543 CSO5R7 90666141 Ki = 12 nM T31543 C3F0PB 90666142 Ki = 23 nM T31543 CG1W0R 90666143 Ki = 17 nM T31543 CI3AX1 90666144 Ki = 1.8 nM T31543 C43YWM 90666145 Ki = 0.9 nM T31543 CT45NA 90666146 Ki = 2.7 nM T31543 C56KQL 90666147 Ki = 5.1 nM T31543 CA90QH 91827690 Ki = 530 nM T31543 C65TLW 101862198 Ki > 1000000 nM T31543 C46MSP 118542774 Ki = 1280 nM T31543 C20WBY 118542785 Ki = 830 nM T31543 CI65YK 118542879 Ki = 850 nM T31543 CEH93P 118542958 Ki = 580 nM T31543 CITU59 118548755 Ki = 470 nM T31543 CMF5R6 118548758 Ki = 280 nM T31543 C1IH2W 118548759 Ki = 810 nM T31543 C6LZQ3 118548760 Ki = 330 nM T31543 C62ZNW 118548761 Ki = 520 nM T31543 C3WQ9D 118548776 Ki = 1510 nM T31543 CU01RP 118548813 Ki = 350 nM T31543 CYUL31 118720337 Ki = 0.061 nM T31543 C4SUL9 118720338 Ki = 0.18 nM T31543 CP4F0X 118720339 Ki = 0.23 nM T31543 C0QI8C 118720340 Ki = 0.14 nM T31543 C6UG4N 118720341 Ki = 0.72 nM T31543 COFR38 118720342 Ki = 0.15 nM T31543 CA7O2K 118720343 Ki = 0.092 nM T31543 C3E7IH 118720344 Ki = 14.67 nM T31543 C9Z4AQ 118720345 Ki = 0.91 nM T31543 CKLU87 118720346 Ki = 0.45 nM T31543 C2NE9Q 118720347 Ki = 7.98 nM T31543 CS2G7Z 118720348 Ki = 31.54 nM T31543 CC2EV6 118720349 Ki = 3.22 nM T31543 CL28SC 118720350 Ki = 1.4 nM T31543 CF64QE 118720351 Ki = 0.89 nM T31543 C7NG3I 118721642 Ki = 0.92 nM T31543 CTV97I 118721643 Ki = 22 nM T31543 C1NS7F 118721644 Ki = 32 nM T31543 C3OCD1 118721645 Ki = 0.69 nM T31543 CQK2U8 118721646 Ki = 15 nM T31543 C4HB3G 118721647 Ki = 0.32 nM T31543 CNP30X 118721648 Ki = 9.2 nM T31543 CRPV34 118721649 Ki = 1.1 nM T31543 CU5KB2 118721650 Ki = 5.5 nM T31543 CJA76N 118721651 Ki = 58 nM T31543 CS3GX9 118721652 Ki = 104 nM T31543 C0Y9EU 118721653 Ki = 8.6 nM T31543 CJ4FI3 118721654 Ki = 3 nM T31543 CK2QX9 118721655 Ki = 12 nM T31543 C4UYE3 118721656 Ki = 5.8 nM T31543 CP9L7H 118721657 Ki = 8.7 nM T31543 C2MI1J 118721658 Ki = 69 nM T31543 CIPY54 118721659 Ki = 0.83 nM T31543 CSAZ58 118728084 Ki = 14900 nM T31543 C4K6HY 118729129 Ki = 1500 nM T31543 C4MX0T 118729130 Ki = 6700 nM T31543 CUC7N1 118729131 Ki = 620 nM T31543 C1KWF0 118729132 Ki = 760 nM T31543 CS7QD3 118729855 Ki = 300 nM T31543 CWK9I0 118729856 Ki = 2600 nM T31543 C73DSK 118729857 Ki = 1200 nM T31543 CM2E0V 118729858 Ki = 4600 nM T31543 C63TEA 118729859 Ki = 480 nM T31543 CPD68M 118729860 Ki = 2500 nM T31543 C3NK4O 121232387 Ki = 2100 nM T31543 C0IAV8 122182389 Ki = 558 nM T31543 CXT84D 122182390 Ki = 526 nM T31543 CG4LR5 122194707 Ki = 4400 nM T31543 CA6U5Q 122194708 Ki = 4800 nM T31543 CZ8CH4 122194709 Ki = 500 nM T31543 CLDC14 122194710 Ki = 1500 nM T31543 C6NGM7 122194711 Ki = 800 nM T31543 CR4CY8 122194712 Ki = 1100 nM T31543 COY83A 122535266 Ki = 0.13 nM T31543 CG5S2R 122535267 Ki = 0.65 nM T31543 CAI69W 123238067 Ki = 1540 nM T31543 C76BAD 123424620 Ki = 850 nM T31543 CA30BN 127033248 Ki = 48900 nM T31543 CO7PY0 127033521 Ki = 13500 nM T31543 CE0QZ4 127033522 Ki = 15400 nM T31543 C7ZIR9 127034099 Ki = 510 nM T31543 C1BWV2 127035672 Ki > 1000000 nM T31543 CVRY56 127036086 Ki > 1000000 nM T31543 C9B6LT 127037264 Ki > 1000000 nM T31543 C60HLK 127037469 Ki > 1000000 nM T31543 C90LJI 127045142 Ki = 492 nM T31543 CD06PE 134313025 Ki = 3.1 nM T31543 CH74VX 135435498 Ki = 4500 nM T31543 CX52AQ 137631869 Ki = 44 nM T31543 CMB40N 137632239 Ki = 28 nM T31543 CDN14Z 137635697 Ki = 48 nM T31543 CDQ62V 137637214 Ki = 40000 nM T31543 CV3I9R 137637849 Ki = 240 nM T31543 CI5VX9 137639355 Ki = 63 nM T31543 C2K8JV 137639385 Ki = 15000 nM T31543 C5PHM2 137640910 Ki = 71 nM T31543 CI3JQ8 137640977 Ki = 150 nM T31543 C3TZH7 137640998 Ki = 120 nM T31543 CQ7N3P 137642872 Ki = 19 nM T31543 CVTM59 137644771 Ki = 12 nM T31543 CA7F3M 137645031 Ki = 200 nM T31543 C51JAT 137646077 Ki = 26 nM T31543 C94KVB 137646622 Ki = 12000 nM T31543 C6G4RT 137647792 Ki = 20 nM T31543 C3P0CS 137648443 Ki = 1380 nM T31543 C30ZQS 137648450 Ki = 120 nM T31543 CS03HK 137648571 Ki = 4 nM T31543 C6Z7LI 137653508 Ki = 7 nM T31543 CC0OE6 137653752 Ki = 39 nM T31543 C6HKV9 137654166 Ki = 43 nM T31543 CNX46H 137654508 Ki = 50000 nM T31543 CZW3F6 137655661 Ki = 15000 nM T31543 CT6X1A 137657743 Ki = 34 nM T31543 C38KYF 137658118 Ki = 5.6 nM T31543 C0Z8RH 137658426 Ki = 51 nM T31543 CXEV32 137659374 Ki = 230 nM T31543 CAE43N 137659536 Ki = 34 nM T31543 C0SJX8 137661290 Ki = 20 nM T31543 CXZ3O7 137662143 Ki = 65 nM T31543 CUZ35A 138115400 IC50 = 25118.86 nM T31543 C0A3MI 145959466 IC50 > 50000 nM T31543 CJP64T 155510867 IC50 = 90 nM T31543 CZR36C 155511554 IC50 = 7943.28 nM T31543 CUP78D 155512098 IC50 = 640 nM T31543 CYT20V 155514020 Ki > 50000 nM T31543 C1RYT8 155517297 Ki = 486 nM T31543 C6NX4K 155519661 IC50 = 1995.26 nM T31543 C4MS1B 155519676 IC50 = 39810.72 nM T31543 CX6C5Y 155520312 IC50 = 4000 nM T31543 CE01NY 155523107 IC50 = 730 nM T31543 CW9K3R 155523263 IC50 = 1100 nM T31543 CGMP07 155523803 Ki = 0.55 nM T31543 CRC6L7 155524551 IC50 > 10000 nM T31543 C4HN6V 155525157 Ki = 271 nM T31543 C6L1WU 155525184 Ki = 200 nM T31543 CN3BH5 155527998 IC50 = 1258.93 nM T31543 C7SB9X 155528083 Ki = 25 nM T31543 CHYW65 155528639 IC50 = 15848.93 nM T31543 CG68UH 155529134 IC50 = 810 nM T31543 CN0B2S 155529433 Ki = 106 nM T31543 C5QT3D 155529505 Ki = 294 nM T31543 CD7O2G 155530095 IC50 = 63095.73 nM T31543 CA82SM 155530516 Ki = 2.5 nM T31543 C46AZL 155530642 Ki > 25000 nM T31543 C35QWO 155531023 IC50 = 1995.26 nM T31543 CDT7A9 155531797 IC50 > 10000 nM T31543 CER1Z8 155532768 Ki = 7.2 nM T31543 C1HAW5 155533558 IC50 = 20 nM T31543 CEFK81 155534191 Ki = 0.22 nM T31543 C7M2UT 155534310 IC50 = 30 nM T31543 C2YB0P 155535378 Ki = 4.9 nM T31543 C6AE0I 155535379 Ki = 18 nM T31543 CUV1I4 155535874 IC50 = 10000 nM T31543 C12HON 155536142 IC50 = 31622.78 nM T31543 CY6DK3 155540964 IC50 = 12.59 nM T31543 C4P2GV 155543617 Ki > 25000 nM T31543 CT4S3M 155544624 IC50 = 2100 nM T31543 C5FZ3I 155545003 Ki = 294 nM T31543 CA08GE 155545013 Ki = 188 nM T31543 CQ51DI 155546002 IC50 = 70 nM T31543 C5MB9R 155547962 IC50 = 7943.28 nM T31543 CLFB25 155548371 IC50 = 25118.86 nM T31543 CK0E7M 155548720 IC50 = 4500 nM T31543 C3R9TO 155551160 IC50 = 2400 nM T31543 CU9FL4 155551858 Ki > 50000 nM T31543 COM52R 155551892 IC50 = 10000 nM T31543 CJ3FI5 155553630 IC50 = 25118.86 nM T31543 CU8LR3 155555208 Ki > 25000 nM T31543 CM3X6Y 155555703 Ki = 11 nM T31543 CXYR84 155556203 Ki = 5.4 nM T31543 CM63SG 155557605 IC50 = 7500 nM T31543 CSW48V 155557718 IC50 = 1258.93 nM T31543 C0IW5Z 155557962 IC50 > 20000 nM T31543 C3VJ5W 155559076 Ki = 0.36 nM T31543 CY60RV 155559158 Ki = 253 nM T31543 CQ3MJ4 155559840 Ki = 3.9 nM T31543 C0B3ID 155562970 Ki = 0.5 nM T31543 C6N0LM 155564043 IC50 > 10000 nM T31543 CM8XB1 155565537 IC50 = 6309.57 nM T31543 CTF0S7 155566456 Ki = 1.3 nM T31543 CP4F1U 155567613 Ki = 480000 nM T31543 D00LOL 970375 IC50 = 570 nM T31543 D01TWD 126363 Ki = 14000 nM T31543 D07SFI 2332 Ki = 400000 nM T31543 D07ZRG 46899577 Ki = 55 nM T31543 D08KCA 72429 Ki = 696 nM T31543 D0SP2I 6852210 Ki = 46 nM T31543 D0W2SV 70689167 Ki = 0.011 nM T17140 D01BYB 5957 EC50 = 340 nM T17140 D07BSQ 5994 IC50 = 1600 nM T17140 D0H2UB 5361 EC50 = 3000 nM T17140 D0PL3N 24764487 IC50 = 45 nM T17140 D0UF2N 21706 EC50 = 500 nM T17140 CCJ8P0 440317 EC50 = 690 nM T17140 CIWV85 746996 IC50 = 7980 nM T17140 CMUV80 766793 IC50 = 14200 nM T17140 CEBX03 779113 IC50 = 29800 nM T17140 CGJ9S2 921624 IC50 = 28000 nM T17140 CYV85L 2320735 IC50 > 10000 nM T17140 CI76GD 3119320 IC50 = 4790 nM T17140 CJEV94 5287422 EC50 = 0.9 nM T17140 CDON91 5310949 EC50 = 350 nM T17140 C97WCE 5310950 EC50 = 17 nM T17140 C6P7VU 5311303 EC50 = 13000 nM T17140 CQC5W8 5702690 IC50 = 1000 nM T17140 CXUA54 5796006 IC50 = 20 nM T17140 CLF3B8 5861195 IC50 = 130 nM T17140 CLU4D6 5891789 IC50 > 10000 nM T17140 CD67GR 5897666 IC50 = 30 nM T17140 CMB71S 5922935 IC50 > 10000 nM T17140 CBA53G 5935441 IC50 = 370 nM T17140 CT5V6E 5935932 IC50 = 130 nM T17140 CDG68S 5936815 IC50 = 20 nM T17140 CX92YW 6093160 IC50 = 28500 nM T17140 CQ7U2M 6298699 IC50 = 90 nM T17140 CGAX04 6436223 IC50 = 755 nM T17140 CX7J8F 11636756 IC50 = 354.81 nM T17140 CR8U0Y 11663667 IC50 > 100000 nM T17140 C6J8WC 16066783 IC50 = 1580 nM T17140 CSXO69 16680454 IC50 = 86.1 nM T17140 C6AR3Q 16757019 IC50 = 353 nM T17140 CP0NB8 25060060 IC50 = 10 nM T17140 CG91NW 25097210 IC50 = 10 nM T17140 CG2Z1N 25097457 IC50 = 140 nM T17140 C5UOK2 25097734 IC50 = 260 nM T17140 C6ETK1 25117612 IC50 = 618 nM T17140 CJ7HT2 25117615 IC50 = 398 nM T17140 CGR1W4 25117983 IC50 = 5689 nM T17140 C8BZ0T 25117985 IC50 = 4214 nM T17140 CK06LQ 25118337 IC50 = 64 nM T17140 CQE1C2 25118338 IC50 = 69 nM T17140 C98MNR 25120809 IC50 = 441 nM T17140 CT06WO 25121155 IC50 = 2057 nM T17140 C3OC1Y 25121511 IC50 = 1271 nM T17140 CMCH17 25121856 IC50 = 613 nM T17140 CM7WO3 25122581 IC50 = 20 nM T17140 CA25BL 42603033 IC50 = 18 nM T17140 CI60EN 42666540 IC50 = 810 nM T17140 CWK71B 42795648 IC50 = 1300 nM T17140 CE25GL 42795663 IC50 = 7500 nM T17140 CQ46IG 44353592 EC50 = 80 nM T17140 CBPD97 46175179 IC50 = 398.11 nM T17140 C2W8ID 46832336 IC50 > 10000 nM T17140 C50QVP 53262865 IC50 = 438 nM T17140 C1UV0E 54590854 IC50 = 797 nM T17140 C9B6DZ 54590935 IC50 = 460 nM T17140 C2HZW4 54590936 IC50 = 920 nM T17140 CX4R5G 54590937 IC50 = 458 nM T17140 CZ41CM 54591029 IC50 = 824 nM T17140 C0Y5CL 54591030 IC50 = 1250 nM T17140 CM3T2V 57431767 IC50 = 2523 nM T17140 CE85TF 57431769 IC50 = 262 nM T17140 C8LVD4 57431775 IC50 = 324 nM T17140 C7AO1Q 57431779 IC50 = 1665 nM T17140 CS2ID6 57431780 IC50 = 1311 nM T17140 CWA65N 57431796 IC50 = 268 nM T17140 C94OEW 57431799 IC50 = 1360 nM T17140 CP4HN8 57431802 IC50 = 440 nM T17140 C06QYE 57431806 IC50 = 327 nM T17140 CVF9A8 57431849 IC50 = 67 nM T17140 CI4V2N 57431852 IC50 = 24 nM T17140 C0MBP3 57431914 IC50 = 24 nM T17140 CZTG87 57480939 IC50 = 255 nM T17140 C9ZMQ1 57480972 IC50 = 22 nM T17140 CKF4N7 57500055 IC50 = 13950 nM T17140 CBRF16 57500058 IC50 > 30000 nM T17140 CSD0M2 57658880 IC50 = 38 nM T17140 C81GJB 57658902 IC50 = 521 nM T17140 CGIP34 57658907 IC50 = 21 nM T17140 CA9WJ6 57658920 IC50 = 1947 nM T17140 CIFW58 57658935 IC50 = 115 nM T17140 C1B9DW 57658971 IC50 = 212 nM T17140 CBG3O4 58044900 IC50 = 11 nM T17140 C25PHF 58044933 IC50 > 10000 nM T17140 C2TAY8 58045034 IC50 = 203 nM T17140 CIZ69B 58045105 IC50 = 44 nM T17140 CN4Q7D 58045231 IC50 = 52 nM T17140 CG2ZR3 58045273 IC50 > 10000 nM T17140 CW5G9P 58045279 IC50 = 1020 nM T17140 CMXC37 58365250 IC50 = 16 nM T17140 C4EPA5 58365345 IC50 = 16 nM T17140 CO53TZ 58365501 IC50 = 15 nM T17140 CXY58G 58365527 IC50 = 13 nM T17140 CON6K1 58365686 IC50 = 16 nM T17140 CVP17Q 58365704 IC50 = 74 nM T17140 CB72VP 58365714 IC50 = 49 nM T17140 CZ6X0Y 58365744 IC50 = 73 nM T17140 CX8Y6Z 58365813 IC50 = 11 nM T17140 C3WB9I 58365828 IC50 = 16 nM T17140 C5CRB1 58365867 IC50 = 13 nM T17140 CF6A8Y 58365941 IC50 = 1089 nM T17140 C35RYZ 58365945 IC50 = 82 nM T17140 CJI25C 58365995 IC50 = 13 nM T17140 C3QI6Y 58366053 IC50 = 35 nM T17140 C6AC9L 58366064 IC50 = 999 nM T17140 CC67BX 58366073 IC50 = 700 nM T17140 CQAG37 59447778 IC50 = 553 nM T17140 CO7PZ5 60168729 IC50 = 10000 nM T17140 C32ADF 66895517 IC50 = 24 nM T17140 CH9Q0R 71450180 IC50 > 10000 nM T17140 CR64QG 71457337 IC50 > 10000 nM T17140 CR1L5W 71459185 IC50 = 429 nM T17140 CSV43Z 71459189 IC50 >= 10000 nM T17140 C0Y1JN 71462707 IC50 > 10000 nM T17140 C3U1YM 73669299 IC50 = 7180 nM T17140 CJYH20 76309929 IC50 = 587 nM T17140 CR93FA 76309930 IC50 = 723 nM T17140 CYQ01L 76313648 IC50 = 3300 nM T17140 C82PEC 76317151 IC50 = 145 nM T17140 CF1KS0 76320868 IC50 = 60 nM T17140 CD30RO 76324525 IC50 = 2930 nM T17140 CYPC45 76324526 IC50 = 928 nM T17140 CG5RF9 76324527 IC50 = 377 nM T17140 C4U3DT 76324528 IC50 = 652 nM T17140 CB69EX 76324694 IC50 = 15200 nM T17140 C43VZB 76328091 IC50 = 474 nM T17140 CB2G0F 76331762 IC50 = 636 nM T17140 CJN18X 76331763 IC50 = 366 nM T17140 CJ63YT 76331764 IC50 = 638 nM T17140 C71DLU 76331765 IC50 = 856 nM T17140 CMH31Y 76335353 IC50 = 1050 nM T17140 CHX09Y 108679493 IC50 = 360 nM T17140 CVQU96 118733194 IC50 = 600 nM T17140 CPO7N5 124125214 IC50 = 8300 nM T17140 CDX97M 134691714 IC50 = 840 nM T17140 CUSH91 135431092 IC50 = 2800 nM T17140 C50GNB 136082632 IC50 = 79.8 nM T17140 CQHU28 136088910 IC50 = 106 nM T17140 CO23GR 142737932 IC50 = 910 nM T17140 C3ZOV5 142737950 IC50 = 2660 nM T17140 CI7P6A 142737955 IC50 = 800 nM T17140 C4M3FP 145952869 IC50 = 21 nM T17140 C3P0KM 145953319 IC50 = 9800 nM T17140 C5IMK3 145953533 IC50 = 100 nM T17140 C8S1NH 145953535 IC50 = 3930 nM T17140 CKT0E1 145953538 IC50 = 19 nM T17140 CQ2GB7 145953759 IC50 = 72 nM T17140 CR95YQ 145954711 IC50 = 9 nM T17140 CLFO06 145954942 IC50 = 1370 nM T17140 CKMB59 145954945 IC50 = 4240 nM T17140 C8FJE9 145956116 IC50 = 560 nM T17140 CJ5XS2 145959607 IC50 = 3000 nM T17140 C3Q1DO 145960696 IC50 > 10000 nM T17140 CLS0X7 145960885 IC50 = 25 nM T17140 C9JQ8N 145961138 IC50 = 140 nM T17140 CT7UF3 145961319 IC50 > 10000 nM T17140 CC62FN 145962500 IC50 > 10000 nM T17140 CIP21K 145963223 IC50 = 5920 nM T17140 CK4R6B 145963480 IC50 = 135 nM T17140 CSF84N 145963490 IC50 = 3280 nM T17140 CEB6C4 145963681 IC50 = 10 nM T17140 CMO5J6 155511397 IC50 = 130 nM T17140 C75XNF 155511587 IC50 = 6300 nM T17140 C4J6BF 155512768 IC50 = 60 nM T17140 CB9XT1 155513864 IC50 = 15 nM T17140 CPE58H 155514125 IC50 = 8 nM T17140 CF6LV4 155514310 IC50 > 100000 nM T17140 C4JZB6 155514547 IC50 = 40 nM T17140 CM39YO 155514691 IC50 = 140 nM T17140 C7W9LA 155514822 IC50 = 85 nM T17140 CVK82Z 155514869 IC50 = 7500 nM T17140 CM3H9Q 155514887 IC50 = 8700 nM T17140 CKVY03 155515950 IC50 = 35 nM T17140 CRY41S 155517023 IC50 = 40 nM T17140 C6GCH5 155517065 IC50 = 3000 nM T17140 CLMW53 155518757 IC50 = 9900 nM T17140 C0BRX7 155519441 IC50 = 1400 nM T17140 C9HK4E 155519617 IC50 > 10000 nM T17140 CT7W8K 155519826 IC50 = 20 nM T17140 CG6JE1 155520066 IC50 = 380 nM T17140 C4LH3M 155520244 IC50 = 25 nM T17140 CT01XB 155521633 IC50 = 180 nM T17140 CY1IU5 155521709 IC50 = 35 nM T17140 CP58CD 155523291 IC50 = 180 nM T17140 CZD97E 155524156 IC50 = 440 nM T17140 CJ58QP 155524530 IC50 = 5 nM T17140 C2NWE8 155525058 IC50 = 900 nM T17140 C8R4GF 155525867 IC50 = 45 nM T17140 CM9CW2 155526224 IC50 = 5830 nM T17140 CDJ31N 155526369 IC50 = 7500 nM T17140 CU2I4R 155526703 IC50 = 20 nM T17140 C3B6EX 155526972 IC50 = 590 nM T17140 C2CQI3 155527693 IC50 = 2400 nM T17140 CL4RC9 155528080 IC50 > 2000 nM T17140 C9EL4D 155528131 IC50 = 50 nM T17140 C1NOD4 155529242 IC50 = 4110 nM T17140 CL4NQ9 155529657 IC50 = 650 nM T17140 CX12AU 155529713 IC50 = 611 nM T17140 C5BC9V 155529971 IC50 = 17500 nM T17140 C3LU9N 155530055 IC50 = 6 nM T17140 CXGC97 155530178 IC50 = 7400 nM T17140 CQX4F0 155530320 IC50 = 668 nM T17140 CKY09W 155531083 IC50 = 580 nM T17140 CYQ84G 155532585 IC50 = 10700 nM T17140 CBD9L6 155533139 IC50 = 19 nM T17140 C8QR1E 155534154 IC50 = 5000 nM T17140 C7GZ8C 155534904 IC50 = 2100 nM T17140 CJB82P 155535066 IC50 = 1310 nM T17140 CP97ML 155535352 IC50 = 65 nM T17140 CH47QU 155535354 IC50 = 390 nM T17140 C4L0SX 155537072 IC50 = 20 nM T17140 CTG39Y 155537553 IC50 = 1500 nM T17140 COQC96 155537975 IC50 = 95 nM T17140 CH9Y0J 155538262 IC50 = 10 nM T17140 CA26YF 155538734 IC50 = 11200 nM T17140 CH92GY 155539221 IC50 = 65 nM T17140 CHI78B 155540008 IC50 = 40 nM T17140 C45GAY 155540285 IC50 = 720 nM T17140 C4ZAM2 155540414 IC50 = 400 nM T17140 C9BGA0 155540772 IC50 = 700 nM T17140 C0K9FV 155542440 IC50 = 3700 nM T17140 C5OIQ7 155542766 IC50 = 7 nM T17140 COD7Q8 155543044 IC50 = 883 nM T17140 C0I3WD 155543378 IC50 = 170 nM T17140 C5AFJ7 155543528 IC50 = 850 nM T17140 CI0E4P 155544725 IC50 = 6800 nM T17140 C6L2JE 155544746 IC50 = 140 nM T17140 CCB2O4 155545366 IC50 = 7500 nM T17140 C2CZ7O 155545879 IC50 = 10000 nM T17140 CR5D3Q 155548909 IC50 = 5700 nM T17140 CS57LN 155549377 IC50 > 10000 nM T17140 C1MYS0 155549544 IC50 = 40 nM T17140 CET18Q 155550268 IC50 = 21 nM T17140 CC7AN2 155550493 IC50 = 1300 nM T17140 CSQ05B 155551563 IC50 = 15 nM T17140 CI9B5Y 155551797 IC50 = 640 nM T17140 CTBK15 155552357 IC50 = 33 nM T17140 CDH06Y 155552819 IC50 = 15 nM T17140 C0F6RT 155553704 IC50 = 48 nM T17140 C3I7BT 155553879 IC50 = 190 nM T17140 CPV2E3 155554392 IC50 = 1600 nM T17140 CJ07RZ 155554473 IC50 = 80 nM T17140 CQH57Z 155555213 IC50 = 7300 nM T17140 C09SOB 155557542 IC50 = 1400 nM T17140 CPO1H2 155557786 IC50 = 150 nM T17140 C2NBD5 155558024 IC50 = 280 nM T17140 CB5Y7A 155558453 IC50 = 1000 nM T17140 C2WFY3 155558639 IC50 = 3700 nM T17140 CZ9G8K 155559078 IC50 > 100000 nM T17140 C47VBE 155559341 IC50 = 55 nM T17140 CJCO90 155560573 IC50 = 140 nM T17140 C0PYX1 155562454 IC50 >= 100000 nM T17140 CDQ97I 155562606 IC50 = 1300 nM T17140 COL84V 155563568 IC50 = 65 nM T17140 CPM6Y0 155564816 IC50 = 1000 nM T17140 C9T5VU 155564839 IC50 = 45 nM T17140 C0AK8B 155565293 IC50 = 660 nM T17140 CJTV86 155566512 IC50 = 15 nM T17140 CVT0H6 155567668 IC50 = 3800 nM T17140 C4QDL9 155568671 IC50 = 3300 nM T17140 C9TRF0 155568988 IC50 = 750 nM T17140 CQA3R5 155569370 IC50 = 648 nM T17140 D00QLM 91557 EC50 = 740 nM T17140 D03EEO 3960826 IC50 = 58300 nM T17140 D05BFC 3978952 IC50 = 96.2 nM T17140 D05NWF 6022 EC50 > 100000 nM T17140 D05RRF 17756317 IC50 = 82.4 nM T17140 D07QYU 4881 EC50 = 240 nM T17140 D0B1KT 15953802 IC50 = 20 nM T17140 D0FF6S 16038374 IC50 > 10000 nM T17140 D0M8HU 25054651 IC50 = 32.4 nM T17140 D0U1OJ 5310983 EC50 = 350 nM T17140 D0UG4S 91532 EC50 = 9200 nM T17140 D0V4GQ 5310996 EC50 = 8800 nM T17140 D0Z0QD 3081832 IC50 = 0.0083 nM T17140 D0Z1DQ 9829395 IC50 = 35 nM T17140 D0Z6UE 25054398 IC50 = 14.3 nM T58589 D06BHG 11953367 Ki = 0.3 nM T58589 D0LI1C 44469321 IC50 > 30000 nM T58589 D0X0BI 439201 Ki > 10 nM T58589 C1ZTN0 2818985 IC50 = 3200 nM T58589 C93QUY 3102216 Ki = 500 nM T58589 C0TV9U 4227718 Ki = 45 nM T58589 C73ZFI 9804704 IC50 = 86 nM T58589 CO36FU 9852117 Ki = 5.6 nM T58589 CWL4Q7 9894973 Ki = 0.59 nM T58589 CU15TR 9897921 Ki < 10000 nM T58589 CM45KH 9919335 Ki = 24.1 nM T58589 CQ39DL 9961595 Ki = 10 nM T58589 CCP49I 9988753 Ki < 10000 nM T58589 CJ37QY 10001334 Ki = 390 nM T58589 C0X3IQ 10008626 Ki <= 5.5 nM T58589 C7YH1R 10010104 Ki <= 5.5 nM T58589 C7JE8F 10010669 Ki <= 5.5 nM T58589 C9QZ6G 10031511 Ki = 0.59 nM T58589 CGI57Y 10032895 Ki < 10000 nM T58589 CNQL86 10055774 Ki <= 5.5 nM T58589 CSYU04 10056816 Ki <= 5.5 nM T58589 C68GEM 10079793 Ki < 10000 nM T58589 CIXU90 10079797 Ki < 10000 nM T58589 CU39IK 10101294 Ki <= 5.5 nM T58589 CF4WK8 10102296 Ki < 10000 nM T58589 CXF5K1 10102599 Ki <= 5.5 nM T58589 CY8R9E 10102701 Ki < 10000 nM T58589 CNY18T 10120979 Ki = 97.5 nM T58589 CZY3I5 10128103 Ki = 2.05 nM T58589 C8POE9 10128412 Ki = 1.39 nM T58589 C27URE 10151875 Ki = 0.57 nM T58589 C4U6AG 10166801 Ki = 141 nM T58589 C0W2IY 10168110 Ki = 100 nM T58589 C3RTP5 10173772 Ki = 0.4 nM T58589 CC6M9P 10187167 Ki = 78 nM T58589 C05VWM 10187347 Ki = 28 nM T58589 CH16RG 10196170 Ki = 0.68 nM T58589 CN9G3L 10217706 Ki = 0.51 nM T58589 C7FAN6 10233880 Ki = 1.5 nM T58589 CLB35I 10239095 Ki = 0.6 nM T58589 C4OVQ0 10260476 Ki <= 5.5 nM T58589 CJ9G2K 10282203 Ki = 55 nM T58589 C01IRZ 10288906 Ki = 0.13 nM T58589 CX5CV4 10300688 Ki > 10000 nM T58589 CC87GI 10311064 Ki = 22 nM T58589 CJ1W6X 10349694 Ki <= 5.5 nM T58589 C8EP5X 10350966 Ki < 10000 nM T58589 C1TQ7U 10373970 Ki < 10000 nM T58589 CXS0E7 10388673 Ki = 11.8 nM T58589 CP14YR 10396101 Ki < 10000 nM T58589 CUS3Q8 10418252 Ki <= 5.5 nM T58589 C7X2OY 10418495 Ki <= 5.5 nM T58589 CMNA43 10418701 Ki < 10000 nM T58589 CXP97A 10439868 Ki <= 5.5 nM T58589 C90DQN 10441167 Ki < 10000 nM T58589 CX79PI 10441194 Ki < 10000 nM T58589 C49PQN 10441297 Ki < 10000 nM T58589 CLEX38 10456579 Ki = 40 nM T58589 C45PFV 10463758 Ki <= 5.5 nM T58589 CWHI15 10463818 Ki <= 5.5 nM T58589 C3ZU0G 10463883 Ki < 10000 nM T58589 C4TV3E 10875606 Ki = 1023 nM T58589 CC7VZ4 10940858 Ki > 10000 nM T58589 C2OCH6 11017305 Ki = 1.33 nM T58589 CL31CX 11039234 Ki = 13.4 nM T58589 CE26TD 11050306 Ki = 1.37 nM T58589 CNJZ59 11071992 Ki = 5.73 nM T58589 CB8PH3 11167607 Ki = 0.8 nM T58589 C6VDM5 11168954 Ki = 0.41 nM T58589 C67ZQB 11180561 Ki = 0.07 nM T58589 C3CD4H 11180748 Ki = 250 nM T58589 C84IRP 11203826 IC50 = 16 nM T58589 CR9V6S 11204003 IC50 = 11 nM T58589 CW3QO7 11213709 IC50 = 1700 nM T58589 CB31LO 11214151 Ki = 10 nM T58589 C04LNE 11214480 IC50 = 0.075 nM T58589 CK8R5Q 11214819 Ki = 0.3 nM T58589 CEWC14 11214998 IC50 = 110 nM T58589 CKA87Y 11215189 IC50 = 13 nM T58589 C3UPQ2 11215488 Ki = 0.15 nM T58589 C9NT7H 11215677 Ki = 0.1 nM T58589 CP0DT6 11215913 Ki = 1.3 nM T58589 C8VN1E 11224694 Ki = 120 nM T58589 C0N5LC 11225601 Ki = 0.5 nM T58589 CQ04GL 11227059 Ki = 3.73 nM T58589 CWON94 11238372 IC50 = 54 nM T58589 C5S9IC 11259064 Ki = 2 nM T58589 CINP41 11259614 IC50 = 82 nM T58589 CE21NL 11260745 Ki = 4.5 nM T58589 CJ2BZ3 11272685 IC50 = 1.2 nM T58589 C8R1KF 11281533 Ki = 0.83 nM T58589 CC09KZ 11283865 Ki = 0.4 nM T58589 CTJW92 11284303 Ki = 3000 nM T58589 CY1EC9 11284304 IC50 = 1.46 nM T58589 C2TW3L 11284458 Ki = 23 nM T58589 C3DQ7P 11284564 Ki = 0.5 nM T58589 CUQF93 11293092 Ki = 13 nM T58589 C2K4CM 11306090 Ki = 1.1 nM T58589 CHD87N 11307467 Ki = 1.4 nM T58589 CH4V5L 11307733 IC50 = 59 nM T58589 CG7BW3 11317669 IC50 = 16 nM T58589 CS5EH9 11319515 Ki = 0.02 nM T58589 CE4A7D 11320189 Ki = 1 nM T58589 C2J1GL 11326315 IC50 = 700 nM T58589 C41ZHJ 11330286 IC50 = 48 nM T58589 CVEZ45 11331054 Ki = 3.3 nM T58589 CE2N5Z 11340940 Ki = 1.6 nM T58589 CH2NA9 11341448 Ki = 3.8 nM T58589 C9QE3H 11341479 Ki = 0.29 nM T58589 C7IL8N 11342079 IC50 = 183 nM T58589 CGSA32 11342350 Ki = 0.46 nM T58589 CUR5A1 11342704 Ki = 0.1 nM T58589 CGU5O9 11352746 Ki = 0.2 nM T58589 CHS08F 11363856 Ki = 0.5 nM T58589 C4UXC1 11364466 IC50 = 0.48 nM T58589 CJ8LZ5 11365433 Ki = 0.07 nM T58589 CTZ8E1 11373520 IC50 = 560 nM T58589 CN95TV 11375297 Ki = 73 nM T58589 C21NFQ 11376509 Ki = 230 nM T58589 C31XME 11377529 Ki = 10 nM T58589 C2U7SZ 11386138 Ki = 0.7 nM T58589 CKB2E6 11387387 IC50 = 0.2 nM T58589 CBQ4G7 11387624 Ki = 0.2 nM T58589 CFN4Q3 11387915 Ki = 0.7 nM T58589 CPV9F1 11398971 Ki = 1.9 nM T58589 COS6U4 11399429 Ki > 1000 nM T58589 C8RH5J 11405561 IC50 = 2000 nM T58589 CUQ4X8 11420875 IC50 = 130 nM T58589 CW3R8K 11421944 Ki = 17.9 nM T58589 CF41TX 11422305 Ki = 140 nM T58589 CV68QE 11433587 Ki = 3.5 nM T58589 CI15ME 11442712 IC50 = 0.25 nM T58589 C2V5ED 11444165 IC50 = 22 nM T58589 CM03JU 11444270 IC50 = 14 nM T58589 CBIY13 11444668 Ki = 1.1 nM T58589 CFG04P 11444808 Ki = 0.01 nM T58589 CY9KC3 11452874 Ki = 200 nM T58589 CGV08Y 11454567 Ki = 30 nM T58589 C89TLC 11456015 Ki = 2.6 nM T58589 C4XW1I 11466010 Ki = 6 nM T58589 C6DGB7 11467345 Ki = 31 nM T58589 CGS0Y9 11476944 Ki = 106 nM T58589 C2DX7T 11477390 Ki = 0.7 nM T58589 C0ER8C 11478613 IC50 = 21 nM T58589 C8M0XU 11478717 IC50 = 5.2 nM T58589 C03DKV 11479448 Ki = 10 nM T58589 CUC91I 11488817 Ki = 0.7 nM T58589 C4RKM5 11495796 Ki = 3450 nM T58589 C13DVN 11498691 Ki <= 5.5 nM T58589 C4BD2X 11498853 Ki < 10000 nM T58589 CNT5H8 11505970 Ki <= 5.5 nM T58589 C5SPA8 11506007 Ki <= 5.5 nM T58589 CGH4A1 11512379 IC50 = 150 nM T58589 CO7HB4 11513104 Ki <= 5.5 nM T58589 C5M2QO 11513163 Ki <= 5.5 nM T58589 CVL4R2 11513471 Ki <= 5.5 nM T58589 CZ1QS6 11519239 Ki = 19.1 nM T58589 C8QW9F 11526655 Ki = 6.4 nM T58589 C4AZO9 11526891 Ki = 16.9 nM T58589 CV97KH 11527838 Ki <= 5.5 nM T58589 C4QK9A 11527892 Ki <= 5.5 nM T58589 CR14MO 11527906 Ki <= 5.5 nM T58589 CF37AZ 11542210 Ki <= 5.5 nM T58589 CWLX79 11546560 Ki = 63 nM T58589 C4B8LI 11549335 Ki <= 5.5 nM T58589 CMIS36 11549560 Ki <= 5.5 nM T58589 CU95QM 11549562 Ki <= 5.5 nM T58589 CR5V6E 11553268 Ki = 52000 nM T58589 C0SDP6 11555433 IC50 = 39.2 nM T58589 CD02NX 11555599 IC50 = 79 nM T58589 C2Z4WP 11561240 IC50 = 3.3 nM T58589 CU7CR4 11570120 Ki = 0.045 nM T58589 CUDQ72 11571204 Ki <= 5.5 nM T58589 C3ZQ1H 11575578 Ki = 25.5 nM T58589 CCF8U0 11577748 Ki <= 5.5 nM T58589 CD7TL4 11584184 IC50 = 84.2 nM T58589 C5JY3H 11585604 Ki <= 5.5 nM T58589 C7KN1L 11585627 Ki <= 5.5 nM T58589 CG0Q6N 11589876 Ki > 50000 nM T58589 C7XDG2 11592927 Ki <= 5.5 nM T58589 C9D7LB 11596635 Ki = 478 nM T58589 CL9M5H 11600186 Ki <= 5.5 nM T58589 CF5YX0 11600235 Ki <= 5.5 nM T58589 C90SJN 11600324 Ki < 10000 nM T58589 CW28IT 11604201 Ki = 1580 nM T58589 CCPQ75 11605512 Ki = 565 nM T58589 C1D2NQ 11614670 Ki <= 5.5 nM T58589 CXV40U 11620238 Ki = 1.8 nM T58589 C34GHD 11620871 Ki = 0.045 nM T58589 CJ06QY 11620980 Ki = 43.8 nM T58589 CRW92U 11621618 Ki <= 5.5 nM T58589 C0XZ1G 11621850 Ki <= 5.5 nM T58589 CXU7G5 11635364 IC50 = 44.9 nM T58589 CG07XP 11635365 Ki = 4.1 nM T58589 CJAD90 11636064 Ki <= 5.5 nM T58589 CC0P7Y 11636119 Ki <= 5.5 nM T58589 CPR35B 11636121 Ki <= 5.5 nM T58589 CL7N1Z 11641218 Ki = 462 nM T58589 C5PZ3J 11650337 Ki <= 5.5 nM T58589 CFB32S 11650783 Ki <= 5.5 nM T58589 C9DON1 11657717 Ki <= 5.5 nM T58589 CQXI09 11663606 Ki = 41.4 nM T58589 C9ESF1 11663809 Ki = 1.7 nM T58589 C42RFY 11670114 Ki = 752 nM T58589 C82AWM 11670860 Ki = 23.5 nM T58589 CO5R3C 11671905 Ki <= 5.5 nM T58589 CFA5K1 11672186 Ki <= 5.5 nM T58589 C65VUE 11672243 Ki <= 5.5 nM T58589 C7QCH6 11676747 Ki = 1645 nM T58589 C06SLD 11679144 Ki <= 5.5 nM T58589 CKF81H 11685446 IC50 = 9.9 nM T58589 C5QC8X 11686256 Ki <= 5.5 nM T58589 C1R7VL 11686399 Ki <= 5.5 nM T58589 C2BTI0 11691896 Ki = 59.9 nM T58589 C8Y4US 11699718 Ki <= 5.5 nM T58589 CZB59C 11707335 Ki <= 5.5 nM T58589 C4PY9R 11707423 Ki <= 5.5 nM T58589 C4CA1S 11707528 Ki <= 5.5 nM T58589 CYG71V 11714620 Ki <= 5.5 nM T58589 C28ZVE 11719314 Ki = 119 nM T58589 CH9P6I 11752335 Ki = 9.5 nM T58589 C8Q6ZV 11757682 Ki = 0.02 nM T58589 C3NI6Q 11766718 Ki < 10000 nM T58589 C31JUX 11786597 Ki = 1.09 nM T58589 C9LRU7 11848206 Ki = 0.26 nM T58589 C4MQ2U 12085129 Ki = 65 nM T58589 CI2Z4V 12085130 Ki = 15 nM T58589 CI72ED 12085131 Ki = 12 nM T58589 CK6OS9 12085225 Ki = 63.5 nM T58589 CC76XK 12085227 Ki = 85 nM T58589 C1V9EY 16041612 Ki = 0.2 nM T58589 CNFS70 16047262 Ki = 4.4 nM T58589 C48JMD 16102881 Ki = 2.95 nM T58589 CCHB78 16102882 Ki = 13.5 nM T58589 C6EJP9 16102883 Ki = 0.54 nM T58589 C03DLN 16102884 Ki = 2.5 nM T58589 CAQ93H 16102885 Ki = 2.8 nM T58589 CYS6P1 16102896 Ki = 0.81 nM T58589 C2DI6U 16102897 Ki = 0.44 nM T58589 CQT8E1 16102898 Ki = 0.66 nM T58589 CF89EI 16102899 Ki = 1.44 nM T58589 CYN40W 16102907 Ki = 1.47 nM T58589 CXZ5J9 16102908 Ki = 11.6 nM T58589 C68KPL 16102909 Ki = 119 nM T58589 CO7L1Z 16102918 Ki = 0.93 nM T58589 CCP79J 16102919 Ki = 10.3 nM T58589 C9GF5P 16102920 Ki = 1.35 nM T58589 CMIV80 16102922 Ki = 62.5 nM T58589 CUF20D 16102923 Ki = 1.95 nM T58589 CB43PJ 16105690 Ki < 10000 nM T58589 CC7S8Z 16105694 Ki < 10000 nM T58589 CLM34B 16105696 Ki < 10000 nM T58589 CZ8PH5 16105698 Ki < 10000 nM T58589 CXK4E7 16105701 Ki < 10000 nM T58589 CB4N2X 16105703 Ki < 10000 nM T58589 C8U2YI 16105727 Ki < 10000 nM T58589 CVI42S 16105729 Ki < 10000 nM T58589 CICB86 16105734 Ki < 10000 nM T58589 CR85GM 16105742 Ki < 10000 nM T58589 CFQ42K 16105746 Ki < 10000 nM T58589 C6LSG9 16105751 Ki < 10000 nM T58589 CL4ZQ8 16108953 IC50 <= 4000 nM T58589 CQAH63 16108958 IC50 > 4000 nM T58589 CL7R0B 16108960 Ki = 1.6 nM T58589 C12LZJ 16108962 Ki = 17 nM T58589 CNPJ98 16108963 Ki = 143 nM T58589 CKM75I 16108964 IC50 = 1700 nM T58589 CBL7U8 16108965 IC50 = 14 nM T58589 C3VC2M 16108966 Ki = 17 nM T58589 CL90BF 16108967 IC50 = 359 nM T58589 CX0BL6 16108968 Ki = 132 nM T58589 CMX85A 16108969 Ki = 0.24 nM T58589 CZ84ND 16202227 Ki = 1.2 nM T58589 C8H9YA 16220913 Ki = 308 nM T58589 CC2ZD8 16220914 Ki = 138 nM T58589 C7GX3R 16220915 Ki = 8.3 nM T58589 CA20GX 16220916 Ki = 5.4 nM T58589 CYIC03 16220917 Ki = 84.8 nM T58589 CO6KJ2 16220918 Ki = 3.7 nM T58589 C1QE6G 16220986 Ki = 393 nM T58589 CIAQ15 16220987 Ki = 27.7 nM T58589 CKJX76 16220988 Ki = 367 nM T58589 CS4U5I 16220989 Ki = 77.6 nM T58589 CV3AI0 16220990 Ki = 7.6 nM T58589 CC65FR 16221053 Ki = 25.2 nM T58589 CRP3N0 16221054 Ki = 20.6 nM T58589 CX2J9P 16221055 Ki = 4.8 nM T58589 C96BGW 16221056 Ki = 14 nM T58589 CSP6I0 16221057 Ki = 5.9 nM T58589 C04COE 16221108 Ki = 5.5 nM T58589 C3NF9J 16221109 Ki = 5 nM T58589 CK0XQ9 16221110 Ki = 8.9 nM T58589 CJG3C2 16221111 Ki = 5 nM T58589 CE83RF 16221160 Ki = 21.8 nM T58589 CG4D0Z 16221161 Ki = 5.7 nM T58589 C7QS0G 16221162 Ki = 13.4 nM T58589 C8CP4Q 16221163 Ki = 132 nM T58589 C4HP1S 16221164 Ki = 24.8 nM T58589 C2M8KF 16221225 Ki = 127 nM T58589 CMJ02P 16221226 Ki = 40.6 nM T58589 CSA49K 16221227 Ki = 120 nM T58589 CD67GW 16221228 Ki = 4.7 nM T58589 CTI5B7 16221229 Ki = 10 nM T58589 CIWM58 16221282 Ki = 0.4 nM T58589 CX2E1R 16221283 Ki = 6.7 nM T58589 C6M4LX 16726096 Ki = 0.5 nM T58589 CUG94I 16726109 Ki = 0.77 nM T58589 CX2MU3 16747694 IC50 = 0.45 nM T58589 C90IKR 17751347 IC50 = 1.53 nM T58589 CDE6M1 17751422 IC50 = 130 nM T58589 C8F4VI 17751599 IC50 = 1210 nM T58589 C0L5FH 17751827 IC50 = 25.2 nM T58589 CS8RD0 17751868 IC50 = 2040 nM T58589 CN82VK 23627396 Ki = 3.1 nM T58589 CIFA02 23627458 Ki = 4.7 nM T58589 C52ZOX 23627520 Ki = 15.5 nM T58589 C9C3UF 23627521 Ki = 1.7 nM T58589 CK8XN7 23627523 Ki = 9.1 nM T58589 CAT48V 23627583 Ki = 8.9 nM T58589 CY46XI 23628223 Ki = 0.4 nM T58589 CL45YA 23630509 IC50 = 290 nM T58589 C0LI6H 23630510 IC50 = 210 nM T58589 C86RLI 23630511 IC50 = 3.9 nM T58589 CZMB41 23630512 IC50 = 9.3 nM T58589 C0KME3 23630513 IC50 = 49 nM T58589 C8C1FO 23630514 IC50 > 10000 nM T58589 CN9MI8 23630612 IC50 = 640 nM T58589 CX8UN7 23630613 IC50 = 12 nM T58589 C30ZPG 23630614 IC50 = 71 nM T58589 CKE90S 23630615 IC50 = 1600 nM T58589 CVW34A 23630715 IC50 = 1.8 nM T58589 CQ65JF 23630809 IC50 = 60 nM T58589 C2VFP3 23630810 IC50 = 200 nM T58589 CV4SN3 23630811 IC50 = 23 nM T58589 C2TNP5 23630812 IC50 > 10000 nM T58589 CPM6B8 23630813 IC50 = 10 nM T58589 C9XQZ8 23630814 IC50 = 650 nM T58589 CR43ZH 23630918 IC50 = 44 nM T58589 C9CH0A 23630919 IC50 = 3.5 nM T58589 C9EQ7K 23630920 IC50 = 1200 nM T58589 CJ85EN 23630923 IC50 > 10000 nM T58589 CLOX15 23631015 IC50 = 320 nM T58589 CF0GB7 23631902 IC50 = 3 nM T58589 C9ZAV1 23631903 IC50 = 13 nM T58589 CET97P 24884552 Ki = 0.41 nM T58589 CRAK17 24893993 Ki = 0.7 nM T58589 CE8G9Z 24895111 Ki = 251 nM T58589 C38XVG 24895112 Ki = 65 nM T58589 C24RIT 24895113 Ki > 10000 nM T58589 CD4S1J 24895114 Ki = 108 nM T58589 CCF80B 24895181 Ki = 56 nM T58589 CT9V3Q 24895182 Ki = 28 nM T58589 C2MIR3 24895183 Ki = 72 nM T58589 CC2UH9 24895184 Ki = 24 nM T58589 C4BAU6 24895185 Ki > 10000 nM T58589 C4Z6JT 24895186 Ki = 217 nM T58589 C07VXH 24895252 Ki = 19 nM T58589 C4LQ8N 24895253 Ki = 1.2 nM T58589 CRDU93 24895255 Ki = 5.6 nM T58589 CT5GY9 24895256 Ki = 24 nM T58589 C1N0CZ 24895351 Ki = 23 nM T58589 CRQ6V5 24895352 Ki = 70 nM T58589 CZV68P 24895353 Ki = 331 nM T58589 C4GP1S 24895354 Ki = 202 nM T58589 CKN0E1 24895355 Ki = 431 nM T58589 CY9LI6 24895449 Ki = 43 nM T58589 C60SUP 24895450 Ki = 215 nM T58589 CI2S7Y 24895452 Ki = 0.25 nM T58589 CQ9N6Z 24895454 Ki = 2.1 nM T58589 C32FHS 24895455 Ki = 15 nM T58589 CU31LR 24895550 Ki = 0.6 nM T58589 CVDK89 24970287 IC50 = 0.12 nM T58589 CNIX27 24970501 Ki = 67 nM T58589 CGO65I 24970503 Ki = 1996 nM T58589 CPR90J 25181410 Ki = 11 nM T58589 C0I6QH 25181411 Ki = 93 nM T58589 CF3ZB9 25195622 Ki = 0.12 nM T58589 C79QTD 25207727 IC50 = 125 nM T58589 CQ0K9H 42605727 IC50 = 3100 nM T58589 C7B4AG 42606173 IC50 = 500 nM T58589 CKD3V8 42606292 IC50 = 5 nM T58589 CK19AE 44355038 Ki > 10000 nM T58589 C7JZ8G 44391943 Ki > 5000 nM T58589 CUA0Z6 44391956 Ki > 5000 nM T58589 CD90BO 44391962 Ki = 385 nM T58589 C91YGR 44391977 Ki = 250 nM T58589 CPAZ59 44391980 Ki = 35 nM T58589 C1O8FA 44391982 Ki > 5000 nM T58589 CB6M8N 44392010 Ki = 3500 nM T58589 CIR9X3 44392012 Ki = 130 nM T58589 C27IOC 44392025 Ki = 11 nM T58589 C1S6KP 44392040 Ki = 38 nM T58589 C2A8BO 44392045 Ki = 25 nM T58589 C0D9QZ 44392064 Ki > 5000 nM T58589 CZP3F2 44392068 Ki = 2 nM T58589 CZV49W 44392113 Ki = 730 nM T58589 CD24PS 44392133 Ki = 54 nM T58589 CGDY20 44392138 Ki = 126 nM T58589 C82CAK 44392156 Ki = 2.2 nM T58589 CN3T6R 44392544 Ki = 130 nM T58589 C3QK1W 44401703 Ki = 230 nM T58589 CN3CQ8 44401768 Ki = 1280 nM T58589 CE30XP 44401834 Ki = 33 nM T58589 CDS12U 44401887 Ki = 119 nM T58589 CW5TK9 44401932 Ki = 11 nM T58589 CI9Z8T 44402028 Ki = 11.5 nM T58589 C8H2YK 44402075 Ki = 200 nM T58589 CTW7N2 44402076 Ki = 11 nM T58589 C93VON 44402279 Ki = 88 nM T58589 CO5D1X 44402298 Ki = 6 nM T58589 CU64BX 44410020 IC50 = 1100 nM T58589 C4FD7Y 44410026 IC50 = 95 nM T58589 CM1JP7 44410059 IC50 > 40000 nM T58589 CR9WY5 44410084 IC50 = 700 nM T58589 CA7PS8 44410143 IC50 = 1700 nM T58589 CRP3X2 44410179 IC50 = 540 nM T58589 C2GR1F 44410186 IC50 = 210 nM T58589 CTP46F 44410250 IC50 = 220 nM T58589 CW8G2V 44410254 IC50 = 4300 nM T58589 C91LOM 44410269 IC50 = 590 nM T58589 C03ZNS 44410273 IC50 = 560 nM T58589 CNV1L9 44410313 IC50 = 780 nM T58589 CZQX26 44410316 IC50 = 73 nM T58589 C2B5EM 44410328 IC50 = 62 nM T58589 C3RCW8 44410368 IC50 = 960 nM T58589 C4R3HA 44410972 Ki = 2100 nM T58589 C9D6BT 44411050 Ki = 184 nM T58589 C5MEF4 44411051 Ki = 3.4 nM T58589 CI2Q5H 44411054 Ki = 1.7 nM T58589 C9EWK7 44411058 Ki = 9.5 nM T58589 C7OBM1 44411062 Ki = 1.4 nM T58589 CLM3B0 44411068 Ki = 5.2 nM T58589 CE43KC 44411071 Ki = 28 nM T58589 CD9EZ1 44411080 Ki = 26 nM T58589 CZS4U1 44411091 Ki = 70 nM T58589 C9K2LJ 44411092 Ki = 80 nM T58589 CB41DZ 44411093 Ki = 1.7 nM T58589 CQKX13 44411095 Ki = 2.2 nM T58589 C07CPD 44411101 Ki = 1.5 nM T58589 C6NC8V 44411134 Ki = 893 nM T58589 CCLW04 44411135 Ki = 9.1 nM T58589 CGRY62 44411138 Ki = 3.5 nM T58589 C31BMX 44411153 Ki = 52 nM T58589 CKU49L 44411245 Ki = 62 nM T58589 C2VKS7 44411252 Ki = 65 nM T58589 C8M6FY 44411294 Ki = 0.71 nM T58589 CQE41C 44411297 Ki = 815 nM T58589 C5H1NY 44411338 Ki = 611 nM T58589 C1EA5B 44411343 Ki = 4 nM T58589 CDY70Z 44411344 Ki > 3000 nM T58589 C23YEB 44411345 Ki > 3000 nM T58589 CQ2BI1 44411347 Ki = 25 nM T58589 C68QXN 44411349 Ki = 213 nM T58589 CE74PI 44411353 Ki = 2.9 nM T58589 CDH8E9 44411355 Ki = 17 nM T58589 CI8O0K 44411358 Ki = 1.5 nM T58589 CO31SL 44411360 Ki = 23 nM T58589 CZ6P9W 44411364 Ki = 1.5 nM T58589 CN5P0A 44411368 Ki = 3.3 nM T58589 C0G9HJ 44411372 Ki = 8 nM T58589 CGF61K 44411392 Ki = 34 nM T58589 CTW96R 44411393 Ki = 5.5 nM T58589 CN2G9R 44411442 Ki = 2.8 nM T58589 CUE29X 44411452 Ki = 0.85 nM T58589 C2W3DT 44411457 Ki = 3.4 nM T58589 CLI08P 44412007 Ki <= 5.5 nM T58589 C4KJR5 44412412 Ki <= 5.5 nM T58589 CNZG76 44418930 Ki = 0.81 nM T58589 C6MQF3 44419045 IC50 = 6.4 nM T58589 C1YPW0 44419046 IC50 = 325 nM T58589 C9KZ5O 44419100 IC50 = 540 nM T58589 C79FXT 44421279 Ki = 1.2 nM T58589 CEO74Z 44428099 IC50 > 10000 nM T58589 CP4Y3S 44428100 IC50 = 1100 nM T58589 CX5C2J 44430679 Ki = 1451 nM T58589 CM6NO2 44430680 Ki = 14 nM T58589 CGP0N8 44430681 Ki = 18 nM T58589 CY4WJ2 44430682 Ki = 3.7 nM T58589 CA8Q7N 44430683 Ki = 60 nM T58589 C0WTZ7 44430684 Ki = 24.5 nM T58589 C8OLK2 44430685 Ki = 49 nM T58589 COI8Z0 44430686 Ki = 2 nM T58589 C65ONB 44430687 Ki = 30 nM T58589 C0H1ES 44430688 Ki = 4.9 nM T58589 CBR46X 44430692 Ki = 3.7 nM T58589 C8S2ZG 44430694 Ki = 3.6 nM T58589 CRF25T 44430696 Ki = 0.4 nM T58589 C5G6TD 44432176 Ki = 134 nM T58589 CFB18H 44432178 Ki = 7.6 nM T58589 CRBX21 44432181 Ki = 1.45 nM T58589 CVN93I 44432186 Ki = 0.68 nM T58589 C49NAQ 44432198 Ki = 1.85 nM T58589 C3ZJ5F 44432207 Ki = 2.4 nM T58589 CC5TL6 44432212 Ki = 1.58 nM T58589 CYGL73 44432215 Ki = 1.1 nM T58589 C64XDP 44432220 Ki = 2.6 nM T58589 COR0T7 44432221 Ki = 1.2 nM T58589 CC47IB 44432222 Ki = 1.8 nM T58589 CGC75O 44432223 Ki = 3.8 nM T58589 CVZ18Y 44455004 Ki = 0.43 nM T58589 CZ39GO 44455035 Ki = 0.59 nM T58589 COGS39 44455038 Ki = 0.66 nM T58589 CTV8X4 44455073 Ki = 0.79 nM T58589 CEPR21 44455074 Ki = 579 nM T58589 C50PNH 44455075 Ki = 0.35 nM T58589 C0F3MC 44455087 Ki = 0.4 nM T58589 C9T0EJ 44455089 Ki = 1.5 nM T58589 C07XKW 44455090 Ki = 0.6 nM T58589 C0B1NM 44455107 Ki = 83.5 nM T58589 CY0JU1 44455108 Ki = 24.5 nM T58589 CXSR48 44455145 Ki = 88.5 nM T58589 CJ1MN2 44455147 Ki = 479 nM T58589 C9UKR8 44455148 Ki = 71.5 nM T58589 CSFA12 44455150 Ki = 109 nM T58589 CL37VJ 44455181 Ki = 660 nM T58589 C9X0BM 44455182 Ki = 1050 nM T58589 CL1Q8W 44455227 Ki = 1090 nM T58589 CNVJ71 44455228 Ki = 95 nM T58589 CDB65J 44455229 Ki = 125 nM T58589 CD9CZ7 44455255 Ki = 516 nM T58589 CXE54J 44455256 Ki = 59.1 nM T58589 CD64NE 44455268 Ki = 0.4 nM T58589 C8Q6JE 44455364 Ki = 1.2 nM T58589 C9XP0N 44455366 Ki = 1.5 nM T58589 CQ5EP2 44455492 Ki = 2.3 nM T58589 C8UBI3 44455519 Ki = 0.2 nM T58589 CT7HW2 44455549 Ki = 1.3 nM T58589 CZ1O6I 44455574 Ki = 0.9 nM T58589 C72CFO 44455853 Ki = 1.8 nM T58589 C8YF9S 44455875 Ki = 0.9 nM T58589 CP8A9I 44561641 Ki = 100 nM T58589 C4LZH6 44561643 IC50 = 4.5 nM T58589 CF0B5N 44561786 Ki = 1.5 nM T58589 CHM8G3 44569935 Ki = 21 nM T58589 CPS43A 44569936 Ki = 34 nM T58589 CN8DZ2 44569937 Ki = 113 nM T58589 C2MK9Z 44569938 Ki = 149 nM T58589 CKE5P6 44569939 Ki = 210 nM T58589 CSA47P 44569940 Ki = 410 nM T58589 C1SOB8 44570026 Ki = 1090 nM T58589 C5I0QO 44570136 Ki = 1210 nM T58589 CC36VK 44570137 Ki = 1570 nM T58589 CTRU56 44570138 Ki = 2200 nM T58589 CGD34W 44570139 Ki = 13010 nM T58589 C3C2YB 44579694 IC50 = 1.8 nM T58589 C3J1KC 44580047 Ki = 1.6 nM T58589 C5E8RX 44580048 Ki = 0.69 nM T58589 C5J1YQ 44580049 Ki = 0.67 nM T58589 C3WPQ9 44580209 Ki = 0.96 nM T58589 CNM2H1 44580742 Ki = 0.8 nM T58589 CTD24M 44580743 Ki = 0.48 nM T58589 CBLK51 44580744 Ki = 0.39 nM T58589 C0GI6R 44587041 IC50 = 1.2 nM T58589 C2PD7R 44587181 IC50 = 0.8 nM T58589 CLT2G5 44587182 IC50 = 1 nM T58589 C58RKS 44587183 Ki = 0.7 nM T58589 C90QHG 44587184 Ki = 0.44 nM T58589 CL3IJ1 44587185 Ki = 1.1 nM T58589 C7USG0 44587186 Ki = 0.15 nM T58589 CYW1F6 44587187 Ki = 0.1 nM T58589 CF0C2O 44587188 IC50 = 0.37 nM T58589 CE23AR 44587189 IC50 = 0.14 nM T58589 CC3R0G 44587206 IC50 = 62 nM T58589 C8ZOV4 44587207 IC50 = 23 nM T58589 C2BXO7 44593650 Ki = 0.67 nM T58589 CC9S4T 46216675 IC50 = 0.19 nM T58589 C8JZI3 46216744 IC50 = 4.6 nM T58589 CTU3R5 46216844 IC50 = 1.5 nM T58589 CB0I2Z 46216845 IC50 = 1.8 nM T58589 CT4D1V 46216846 IC50 = 1 nM T58589 C12HXW 46216847 IC50 = 0.6 nM T58589 C6LK7W 46229895 IC50 > 10000 nM T58589 CL4N5G 46229967 IC50 = 1.3 nM T58589 C13TMX 46229968 IC50 = 28 nM T58589 C2YNW1 46230011 IC50 > 1000 nM T58589 C9JK7D 46230012 IC50 > 1000 nM T58589 CD7ZC6 46230013 IC50 > 1000 nM T58589 CAI50D 46230067 IC50 = 1 nM T58589 C7RJH9 46230068 IC50 = 4.4 nM T58589 CWJ9F0 46230069 IC50 = 15 nM T58589 C8JA3U 46230119 IC50 = 0.43 nM T58589 CT01AD 46230120 IC50 = 0.26 nM T58589 C4M3EK 46230121 IC50 = 0.13 nM T58589 CJ41PR 46230160 IC50 = 0.2 nM T58589 CH1RE9 46230161 IC50 = 0.14 nM T58589 CX20BL 46230162 IC50 = 1.3 nM T58589 CJ6FU3 46230163 IC50 = 0.48 nM T58589 CPE7O4 46230202 IC50 = 0.64 nM T58589 CQY4E2 46230203 IC50 = 0.28 nM T58589 CW2D5A 46230258 IC50 = 180 nM T58589 C9H0CP 46230259 IC50 = 35000 nM T58589 CI9JZ4 46230306 IC50 = 42000 nM T58589 C5LB0M 46230307 IC50 = 6100 nM T58589 CLHZ96 46230308 IC50 = 3500 nM T58589 CHD4I0 46230309 IC50 = 0.7 nM T58589 C4KT1A 46230310 IC50 = 85 nM T58589 CI9K6A 46230352 IC50 = 1.7 nM T58589 C42UCQ 46230354 IC50 = 3.5 nM T58589 CUW9M7 46230403 IC50 = 1.6 nM T58589 C1A6WU 46230404 IC50 = 0.3 nM T58589 C9D3PW 46230458 IC50 = 7.7 nM T58589 C4VHS6 46230459 IC50 = 1.7 nM T58589 C2E8PK 46230833 IC50 = 1.2 nM T58589 C1H7LY 46230834 IC50 = 17 nM T58589 C06HIR 46230835 IC50 = 2.3 nM T58589 CXS6D0 46230836 IC50 = 31 nM T58589 C26ZJX 46230889 IC50 = 3.6 nM T58589 CD7CV8 46230890 IC50 = 32 nM T58589 C1LIK9 46230891 IC50 > 100 nM T58589 C2VEI6 46230892 IC50 = 59 nM T58589 CG5N0L 46230893 IC50 = 17 nM T58589 CNO24Q 46230938 IC50 = 4.6 nM T58589 CLX87C 46230939 IC50 = 1 nM T58589 CA34LI 46230940 IC50 = 1.4 nM T58589 CGK92B 46230941 IC50 = 0.8 nM T58589 C98JCN 46230989 IC50 = 3.9 nM T58589 CG03LI 46230990 IC50 = 0.5 nM T58589 CK74NF 46911683 IC50 = 1.3 nM T58589 C8A5JH 46911684 Ki = 4.6 nM T58589 COWR30 49863227 Ki = 34 nM T58589 C2S4KB 49863228 Ki = 14 nM T58589 CN6CE1 49863229 Ki = 12 nM T58589 C08ENG 49863230 Ki = 12 nM T58589 CSO1T6 49863231 Ki = 78 nM T58589 CAY62R 49863232 Ki = 21 nM T58589 C42HRX 49863233 IC50 = 23 nM T58589 CGYV42 49863234 Ki = 16 nM T58589 CWI61B 49863235 Ki = 11 nM T58589 C7L9WC 49863236 Ki = 3.4 nM T58589 CU2Y0N 49863237 Ki = 30 nM T58589 C2YXJ6 53248885 Ki = 0.1 nM T58589 CQSV19 53360054 IC50 = 0.43 nM T58589 CK7F3Y 54580628 Ki = 0.17 nM T58589 CQ8C9G 54580655 Ki = 17.6 nM T58589 C3KW6G 54581634 Ki = 0.21 nM T58589 CYDG96 54581635 IC50 = 0.43 nM T58589 CN3GY5 54581664 IC50 = 3.6 nM T58589 CXZ2T7 54581665 Ki = 718 nM T58589 CZD8U9 54581666 Ki = 1.98 nM T58589 CDHJ78 54581667 Ki = 0.52 nM T58589 CAFY01 54582655 Ki = 0.11 nM T58589 CKC3G4 54582656 Ki = 1.09 nM T58589 CTRO07 54583583 IC50 = 475 nM T58589 C84KJN 54583617 Ki = 0.18 nM T58589 C9TVP7 54584600 IC50 = 2.2 nM T58589 CL92WT 54585539 Ki = 60 nM T58589 CJIV69 54585540 IC50 = 1.28 nM T58589 C4STF5 54586518 IC50 = 98.6 nM T58589 CJ04HM 54586519 Ki = 0.22 nM T58589 CDP6V3 54587514 IC50 = 0.49 nM T58589 C45WVG 54587550 Ki = 31.8 nM T58589 CCU28P 54587551 Ki = 541 nM T58589 CI38WG 54587552 Ki = 0.5 nM T58589 C0VM3Y 54587553 Ki = 1.6 nM T58589 CHA35B 54772237 IC50 = 0.09 nM T58589 CSIT41 56589598 IC50 = 0.3 nM T58589 CCGQ04 56594241 Ki = 64 nM T58589 CQK5I0 56594242 Ki = 183 nM T58589 CRBD81 56594243 Ki = 331 nM T58589 CWL18E 56594244 Ki > 10000 nM T58589 CW78HM 56594371 Ki = 159 nM T58589 C4G2SE 56594372 Ki = 18 nM T58589 C3UI1N 56594373 IC50 = 3405 nM T58589 CHUP45 56594374 Ki = 35 nM T58589 CI27CK 56594375 Ki > 10000 nM T58589 C2GJ3O 56594504 Ki = 614 nM T58589 CWXM09 56594505 Ki = 52 nM T58589 CTN0H2 56594506 Ki = 29 nM T58589 CW75EL 56594507 Ki = 214 nM T58589 CPAQ52 56594508 Ki = 98 nM T58589 C2L9SG 56594639 Ki = 418 nM T58589 CD3E4Y 56594640 Ki = 1.9 nM T58589 CNIP32 56594641 Ki = 3.5 nM T58589 CW1A5M 56594642 Ki = 0.9 nM T58589 C6HLO4 56594643 Ki = 198 nM T58589 C9LF2Q 56594768 Ki = 4.7 nM T58589 C92MLU 56594769 IC50 = 0.18 nM T58589 CY9JD5 56594770 Ki = 3.1 nM T58589 CS76GP 56594771 Ki = 69.9 nM T58589 CVK17L 56594772 IC50 = 1.1 nM T58589 C0UW1N 56658544 Ki = 296 nM T58589 CU9NQ4 56668920 Ki = 565 nM T58589 CV80AB 56672397 IC50 = 1371 nM T58589 CJ0A1B 56679097 Ki = 311 nM T58589 CU0Z1C 56835162 Ki = 4 nM T58589 C7VM9I 56835163 IC50 = 12 nM T58589 CQO75F 56951319 IC50 = 83.9 nM T58589 CTV6P0 57342336 Ki = 2.1 nM T58589 C7O2KQ 57342494 Ki = 3.1 nM T58589 CIY7G9 57342496 Ki = 4.2 nM T58589 C5B9QU 57342845 Ki = 2.8 nM T58589 CH0Q2J 57342847 Ki = 5.5 nM T58589 CF3ET1 57342849 Ki = 4.3 nM T58589 C2N0VG 57342852 Ki = 6.8 nM T58589 C3M1OD 57343016 Ki = 142 nM T58589 CZG03B 57390218 IC50 = 0.4 nM T58589 CJI47Q 57390219 IC50 = 18.7 nM T58589 C49OBW 57390411 IC50 = 7.51 nM T58589 C7W1CO 57390466 Ki > 10000 nM T58589 C5U6AL 57390932 IC50 = 17 nM T58589 C8T5HQ 57390933 IC50 = 279 nM T58589 C14PSN 57391172 IC50 = 25.9 nM T58589 C38SYJ 57391173 IC50 = 0.28 nM T58589 CUAX92 57391276 Ki > 10000 nM T58589 CEI42Q 57391278 Ki > 10000 nM T58589 CR4CU9 57392146 Ki > 10000 nM T58589 C24BYU 57392728 IC50 = 186 nM T58589 CK65VI 57392940 IC50 = 0.42 nM T58589 CD68LS 57392941 IC50 = 0.247 nM T58589 CYDF85 57393059 Ki > 10000 nM T58589 CAC8M5 57393061 Ki > 10000 nM T58589 C2CO0A 57394682 IC50 = 990 nM T58589 CZ6KQ1 57394683 IC50 = 1.38 nM T58589 C7FR2W 57394684 IC50 = 1.09 nM T58589 CRZL24 57394685 IC50 = 1.12 nM T58589 CTB9H6 57394686 IC50 = 19 nM T58589 C9TU1X 57394687 IC50 = 38 nM T58589 CH1JC4 57394688 IC50 = 23.4 nM T58589 CD2J8Z 57394689 IC50 = 4.75 nM T58589 COG8S6 57394779 Ki > 10000 nM T58589 C8PVE2 57394782 Ki > 10000 nM T58589 C2TQ5A 57394783 Ki > 10000 nM T58589 CWYQ56 57395448 IC50 = 0.28 nM T58589 CXN8Q3 57395449 IC50 = 836 nM T58589 CDH04R 57395450 IC50 = 94.7 nM T58589 CVX7F9 57395451 IC50 = 36.1 nM T58589 CYKA40 57395702 IC50 = 40.8 nM T58589 COK0D3 57396212 Ki = 1616 nM T58589 CS58YL 57396445 IC50 = 17.7 nM T58589 C95WJK 57396446 IC50 = 0.63 nM T58589 CW5K9S 57396447 IC50 = 0.22 nM T58589 CJE35F 57396534 Ki > 10000 nM T58589 C97VSN 57396535 Ki > 10000 nM T58589 C8UG2C 57396537 Ki > 10000 nM T58589 C5FV8O 57396539 Ki > 10000 nM T58589 C7H6TJ 57397292 IC50 = 0.084 nM T58589 CK3S0J 57397547 Ki > 10000 nM T58589 C20SLV 57398013 IC50 = 799 nM T58589 CWG42N 57398235 IC50 = 0.51 nM T58589 C4FRJ1 57398236 IC50 = 0.74 nM T58589 C7GA2X 57398237 IC50 = 0.65 nM T58589 C0B9RS 57398238 IC50 = 0.28 nM T58589 C17FCZ 57398239 IC50 = 20.3 nM T58589 CM07WZ 57398323 Ki > 10000 nM T58589 CG5S2A 57398325 Ki > 10000 nM T58589 CDVK40 57398327 Ki > 10000 nM T58589 C3RS9A 57398978 IC50 = 0.21 nM T58589 CM7VX0 57398979 IC50 = 178 nM T58589 CI4H6K 57398980 IC50 = 21.6 nM T58589 CV2NF8 57399227 Ki > 10000 nM T58589 CGFP58 57399382 IC50 = 2.7 nM T58589 CC5B3W 57399670 IC50 = 7 nM T58589 CEY8B9 57399671 Ki = 15 nM T58589 CU03OI 57399885 IC50 = 314 nM T58589 C1W6YL 57399886 IC50 = 152 nM T58589 CZ61BH 57399887 IC50 = 136 nM T58589 C8VG0D 57399981 Ki > 10000 nM T58589 C5BK7O 57399982 Ki > 10000 nM T58589 CH8K5Y 57400696 IC50 = 0.23 nM T58589 CU57BH 57400697 IC50 = 72.2 nM T58589 CJ3AE0 57400937 IC50 = 96 nM T58589 C4KTX6 57400985 Ki > 10000 nM T58589 CON6W8 57401425 IC50 = 98 nM T58589 CJ5M3L 57401426 Ki = 42 nM T58589 C2R6WU 57401663 IC50 = 1.47 nM T58589 C39QYA 57401664 IC50 = 0.31 nM T58589 C05JCX 57401770 Ki > 10000 nM T58589 C1JMA0 57401772 Ki > 10000 nM T58589 C91ALU 57401773 Ki > 10000 nM T58589 CJX89L 57401775 Ki > 10000 nM T58589 CB0I3M 57401777 Ki > 10000 nM T58589 C0HP6R 57401779 Ki > 10000 nM T58589 CB4T8H 57401781 Ki > 10000 nM T58589 CB2XH5 57401783 Ki > 10000 nM T58589 CXLU20 57402467 IC50 = 8.95 nM T58589 C3C9JU 57402744 Ki > 10000 nM T58589 COK10P 57402745 Ki > 10000 nM T58589 CGW59E 57403174 IC50 = 78 nM T58589 CW5O2D 57403175 IC50 = 188 nM T58589 CT6PB0 57403390 IC50 = 1.32 nM T58589 C9KLZ4 57403391 IC50 = 0.86 nM T58589 CG0VE7 57403503 Ki > 10000 nM T58589 CT74HP 57403504 Ki > 10000 nM T58589 CWO85L 68867798 Ki = 3.5 nM T58589 C69UHS 68868627 Ki = 5.8 nM T58589 C79JCF 68868975 Ki = 10 nM T58589 CP8FI7 68869351 Ki = 34 nM T58589 C06EMT 68869570 Ki = 3.3 nM T58589 C0VL1X 68869647 Ki = 0.8 nM T58589 CP0O3A 68870388 Ki = 4.7 nM T58589 CJ5XU4 70683374 Ki = 138 nM T58589 C3X0JV 70685470 Ki = 481 nM T58589 C2O3AY 70685471 Ki = 1 nM T58589 CP7QY1 70687620 Ki = 3.8 nM T58589 C6Z9WM 70688994 Ki = 2300 nM T58589 CXHO48 70688995 Ki = 59 nM T58589 CXAC04 70689675 Ki = 480 nM T58589 C49OIX 70691811 Ki = 1400 nM T58589 C13AMV 70691812 Ki = 6.3 nM T58589 C61JIR 70691813 Ki = 628 nM T58589 CKHP92 70691814 Ki = 2.9 nM T58589 CMV3F0 70692051 IC50 > 10000 nM T58589 C03TXD 70693872 Ki = 166 nM T58589 CZ41AD 70693873 Ki = 4.3 nM T58589 C0YZ2D 70695304 Ki = 2300 nM T58589 CL41AT 70695989 Ki = 2.2 nM T58589 CUX47G 71449505 IC50 = 2500 nM T58589 C6B0OV 71450888 Ki > 10000 nM T58589 C8YG2E 71454501 Ki = 1.8 nM T58589 CTIA35 71454502 Ki = 2.6 nM T58589 CHMG56 71456247 Ki = 7.1 nM T58589 CK01OM 71459890 Ki > 10000 nM T58589 C3Z7AR 71719128 Ki < 0.2 nM T58589 CJ2I4X 73346673 IC50 > 10000 nM T58589 C4QLS2 73346675 IC50 > 10000 nM T58589 CE1WK4 73348186 IC50 = 3019.95 nM T58589 CS27DN 73348187 IC50 = 1621.81 nM T58589 C2GO9F 73349741 IC50 > 10000 nM T58589 CNBL34 73351264 IC50 > 10000 nM T58589 CT72YC 73351265 IC50 > 10000 nM T58589 CO7W1C 73354242 IC50 = 389.05 nM T58589 CF49RH 73354498 Ki = 0.9 nM T58589 CDX4V9 73354499 Ki = 24 nM T58589 CUK4W3 73355813 IC50 = 4570.88 nM T58589 CWMR48 76331576 Ki = 0.023 nM T58589 C61FVX 90662943 Ki = 0.035 nM T58589 CSW30M 90662945 Ki > 10 nM T58589 CYEV01 137640759 IC50 = 4040 nM T58589 CRX0E4 137657568 IC50 = 2000 nM T58589 D00FAE 44316621 Ki = 5.6 nM T58589 D00FUT 123884 Ki = 382 nM T58589 D02DGP 44316161 Ki = 0.22 nM T58589 D04KFR 9831083 Ki = 8 nM T58589 D04WHO 9916412 Ki = 0.0078 nM T58589 D05TZN 122227 Ki < 0.2 nM T58589 D0L3GT 16108961 Ki = 0.7 nM T58589 D0N2GM 44316620 Ki = 83 nM T58589 D0U4SG 10281725 Ki = 85 nM T58589 D0V0LY 5310951 IC50 = 990 nM T62815 D01XYJ 35370 Ki = 150000 nM T62815 D0D1AL 3559 Ki = 590000 nM T62815 D0Y3KG 3121 Ki = 1600000 nM T62815 CF8W5U 68929 Ki = 162000 nM T62815 C57YCN 640695 IC50 = 507000 nM T62815 C2XI6Z 6971242 IC50 = 513000 nM T62815 CM4KP8 6971243 IC50 = 275000 nM T62815 CLI53U 6976566 IC50 = 214000 nM T62815 CX3B2N 6976567 IC50 = 130000 nM T62815 C16OIX 6976568 IC50 = 105000 nM T62815 C1CLV4 6976569 IC50 = 79000 nM T62815 CM6UB5 6992933 IC50 = 532000 nM T62815 C7RVQ1 7004960 IC50 = 344000 nM T62815 CBYR84 7058027 IC50 = 518000 nM T62815 CCAZ92 7058028 IC50 = 337000 nM T62815 C2D6MG 7058029 IC50 = 489000 nM T62815 C2JAE6 11491985 IC50 = 225000 nM T62815 CQJ29R 11513913 IC50 = 651000 nM T62815 C9VD3N 11550148 IC50 = 599000 nM T62815 C9PD1C 11557377 IC50 = 366000 nM T62815 C5XLW0 11564555 IC50 = 284000 nM T62815 C8LDV4 11607933 IC50 = 394000 nM T62815 CEFO25 11615192 IC50 = 179000 nM T62815 CCO5B8 11629630 IC50 = 317000 nM T62815 CD08XY 11636907 IC50 = 166000 nM T62815 CL1A3Y 11643947 IC50 = 540000 nM T62815 CP4ZE5 11658372 IC50 = 158000 nM T62815 CI5WQ9 11708159 IC50 = 301000 nM T62815 CX67NF 11715277 IC50 = 351000 nM T62815 CV3TC0 11831435 IC50 = 2000 nM T62815 C5VS2K 12328973 Ki = 113000 nM T62815 CQ47CA 12328974 IC50 = 182000 nM T62815 CNA17L 12337217 Ki = 301000 nM T62815 CA0M7Q 15148407 Ki = 101000 nM T62815 CR2I5A 16719568 IC50 = 4000 nM T62815 CCIK89 16720943 IC50 = 10000 nM T62815 C3XL7S 16720946 IC50 = 5000 nM T62815 CVS98C 17749637 IC50 = 5000 nM T62815 CE3O7S 18503890 IC50 = 500 nM T62815 C9RJD7 18503891 IC50 = 600 nM T62815 C50QKO 18503892 IC50 = 200 nM T62815 C1CT0N 18503893 IC50 = 400 nM T62815 CGO9E8 18503894 IC50 = 200 nM T62815 CC61VS 18503895 IC50 = 900 nM T62815 CN9FM4 18503899 IC50 = 500 nM T62815 CNS15Y 18503900 IC50 = 3000 nM T62815 CCS8Y9 18503901 IC50 = 16000 nM T62815 C29BLC 18503902 IC50 = 32000 nM T62815 CF72UR 18503905 IC50 = 800 nM T62815 CO63PD 18503907 IC50 = 3000 nM T62815 C30EWI 18503908 IC50 = 900 nM T62815 C3ZYJ1 18503909 IC50 = 400 nM T62815 C9EZF1 18503911 IC50 = 10000 nM T62815 C59OUH 18503912 IC50 = 18000 nM T62815 CHS8L5 18503913 IC50 = 4000 nM T62815 CSW96O 18503915 IC50 = 300 nM T62815 CHU60D 18503916 IC50 = 500 nM T62815 CXBU90 18503917 IC50 = 300 nM T62815 CB36RZ 18503918 IC50 = 400 nM T62815 CR9F0S 18503919 IC50 = 400 nM T62815 CDE1G2 18503920 IC50 = 800 nM T62815 C53NHK 18503921 Ki = 18.4 nM T62815 C5XMF7 18523698 IC50 = 900 nM T62815 CJ8XY0 18523699 IC50 = 700 nM T62815 CM6R0L 18523707 IC50 = 2000 nM T62815 CARN24 18523708 IC50 = 3000 nM T62815 CX8IJ4 18523709 IC50 = 12000 nM T62815 C7D5BX 18523710 IC50 = 8000 nM T62815 CCX5K6 18523711 IC50 = 41000 nM T62815 C2XMT1 18523712 IC50 = 1000 nM T62815 CGX30S 18523713 IC50 = 300 nM T62815 C69YMN 18523714 IC50 = 13000 nM T62815 CS28DQ 18523716 IC50 = 28000 nM T62815 CA9R0S 18523717 IC50 = 3000 nM T62815 C9LE0F 18523719 IC50 = 200 nM T62815 CBOW96 18523720 IC50 = 200 nM T62815 C87YIX 18523721 IC50 = 200 nM T62815 C25YFP 44423322 IC50 = 500 nM T62815 CULW28 44423323 IC50 = 700 nM T62815 CA34IP 89826402 IC50 > 300000 nM T62815 CZE16B 146026197 IC50 > 50000 nM T62815 D0M7YB 12311096 IC50 = 100 nM T62815 D0Z8EV 446541 Ki = 1500 nM T98264 D03DXN 66435 IC50 > 300000 nM T98264 D0I2AN 86298439 IC50 = 1440 nM T98264 CW68ZS 61672 IC50 = 2630 nM T98264 C7KJ3B 114917 IC50 = 1970 nM T98264 C5X1YU 160254 IC50 = 39500 nM T98264 C4IRY2 164676 IC50 = 2140 nM T98264 CCEG90 259329 IC50 = 40400 nM T98264 CONR62 444765 Ki = 350000 nM T98264 C9B3YM 444766 Ki > 2000000 nM T98264 CM0IQ3 446665 IC50 = 31000 nM T98264 C5Y3DJ 446871 Ki = 289000 nM T98264 C7GU8T 470607 IC50 = 12360 nM T98264 CELG48 998012 IC50 = 38760 nM T98264 CJ90PO 1159989 IC50 = 85000 nM T98264 CB7OS1 2964738 IC50 = 160000 nM T98264 C3NL9W 3246406 IC50 = 68000 nM T98264 C35LZP 4774445 Ki = 100000 nM T98264 CPM09B 5327156 IC50 = 203000 nM T98264 C4BE0F 9874843 IC50 = 9000 nM T98264 COX2J8 9930943 IC50 = 19000 nM T98264 CA75NG 9985013 IC50 = 15000 nM T98264 C3A8JL 10256983 IC50 = 6300 nM T98264 CZTN01 10675368 IC50 = 5000 nM T98264 CT4H0O 11006141 IC50 = 16000 nM T98264 C1JAC5 11425923 IC50 = 3670 nM T98264 C5K9MX 17748269 Ki = 17000 nM T98264 C3TV7F 19779154 IC50 = 129000 nM T98264 C54IUM 21778115 IC50 > 50000 nM T98264 C1OR3D 22084082 Ki = 28000 nM T98264 CDTE90 24180456 IC50 = 4000 nM T98264 C21ECL 24180507 Ki = 9700 nM T98264 CE9B6H 25014222 IC50 > 20000 nM T98264 C1Y0KM 25101546 Ki = 14000 nM T98264 CZ4M3C 25141412 IC50 = 15000 nM T98264 C4WM9S 25262527 IC50 = 15700 nM T98264 C3P8XN 42644186 IC50 > 40000 nM T98264 C98IOF 42644187 IC50 > 40000 nM T98264 CL04IU 44156271 IC50 = 14000 nM T98264 C1V7WS 44334321 Ki = 29000 nM T98264 CEL2Q6 44334377 Ki > 200000 nM T98264 CT20HY 44359237 Ki = 60000 nM T98264 C5YV1R 44359299 Ki > 2000000 nM T98264 C76DPK 44387848 EC50 = 50000 nM T98264 C36CRP 44387849 EC50 = 150000 nM T98264 CXU27L 44401026 EC50 = 50000 nM T98264 CZ6S7W 44401113 EC50 = 85000 nM T98264 CXL68A 44401147 EC50 = 160000 nM T98264 CGHV34 44401148 EC50 = 70000 nM T98264 CZC37T 44401149 EC50 = 140000 nM T98264 C01BYZ 44401229 EC50 = 80000 nM T98264 CL9BV8 44401230 EC50 = 180000 nM T98264 C7ABG4 44401231 EC50 = 220000 nM T98264 CLU5N2 44434676 IC50 = 38000 nM T98264 CWN8V5 44434677 IC50 = 13000 nM T98264 CA9X5W 44434678 IC50 = 9000 nM T98264 CY4LH6 44434679 IC50 = 25000 nM T98264 CBUP13 44434680 IC50 = 12000 nM T98264 C3R2HL 44563278 IC50 = 12640 nM T98264 CR50UK 44563344 IC50 = 27380 nM T98264 C9PC6L 44563345 IC50 = 5200 nM T98264 C3HDB9 44563372 IC50 = 4080 nM T98264 CT94FG 44563387 IC50 = 710 nM T98264 CDP45M 44563447 IC50 = 4050 nM T98264 C8MXT3 44563448 IC50 = 890 nM T98264 C7MP5Y 44563570 IC50 = 6000 nM T98264 C5Q2FM 44563588 IC50 = 126000 nM T98264 C7D5GS 44563589 IC50 = 140000 nM T98264 CBV8J9 44563590 IC50 = 78000 nM T98264 CP2H1Y 44563591 IC50 = 231000 nM T98264 CHNU48 44563656 IC50 = 10000 nM T98264 C3LMP9 44563657 IC50 = 6000 nM T98264 CO1GI5 45482833 Ki = 2200 nM T98264 CYRC54 45482878 IC50 > 40000 nM T98264 CK98JB 45482885 IC50 > 40000 nM T98264 CQ5U3C 45482886 IC50 > 40000 nM T98264 C8Z7HX 45482894 IC50 > 40000 nM T98264 CCKE09 45482895 IC50 > 40000 nM T98264 C1ULD8 45483667 Ki = 94000 nM T98264 CLGB06 46830252 IC50 > 10000000 nM T98264 C81CPM 46861833 IC50 = 10600 nM T98264 C0A9LD 46861834 IC50 = 9790 nM T98264 C2IU1Z 49796692 IC50 = 61000 nM T98264 CSBV96 50898774 IC50 = 3000 nM T98264 C4AEZ1 50925509 IC50 = 378 nM T98264 C95QWO 50925510 IC50 = 335 nM T98264 CK1YX2 50941649 IC50 = 5760 nM T98264 C1PJL0 50941745 IC50 = 408 nM T98264 CRF1O3 50942131 IC50 = 486 nM T98264 C2NJ3B 51003508 IC50 = 14000 nM T98264 CMDB84 53316640 IC50 > 50000 nM T98264 C9GVU5 53317937 IC50 > 50000 nM T98264 CV4QD5 53317938 IC50 = 17700 nM T98264 CWT10N 53319270 IC50 > 50000 nM T98264 CRC82E 53320578 IC50 > 50000 nM T98264 C8Y4KW 53320579 IC50 = 25700 nM T98264 CF35GK 53320580 IC50 = 18500 nM T98264 C04CYS 53320581 IC50 > 50000 nM T98264 CBI29Z 53321875 IC50 = 53100 nM T98264 C94WKB 53324565 IC50 > 50000 nM T98264 CCNG89 54576098 IC50 = 9840 nM T98264 CV3YH5 54576318 IC50 = 26500 nM T98264 C4CAU1 54576319 IC50 = 2430 nM T98264 CYK80P 54576320 IC50 = 16340 nM T98264 CKD3W9 54576321 IC50 = 10970 nM T98264 C1P4QM 54576322 IC50 = 13020 nM T98264 C1GDN4 54768308 IC50 = 15550 nM T98264 C1VCJ9 54768351 IC50 = 18500 nM T98264 CF7X2K 54768352 IC50 = 13220 nM T98264 C48KOI 54768353 IC50 = 12500 nM T98264 CK3W0Z 54768391 IC50 = 10720 nM T98264 C01LRT 54768392 IC50 = 16440 nM T98264 CNZY43 56589511 IC50 > 10000000 nM T98264 C53XYO 56589513 IC50 > 10000000 nM T98264 CHM5V3 56660070 IC50 > 120000 nM T98264 CHOF39 56670422 IC50 > 120000 nM T98264 CI9R8M 56670423 IC50 > 120000 nM T98264 CL3N0K 56673907 IC50 > 120000 nM T98264 CAL96I 56673908 IC50 > 120000 nM T98264 CEK3S2 56680547 IC50 > 120000 nM T98264 C72JTU 56681854 IC50 = 68900 nM T98264 CJ50EL 56681855 IC50 = 52600 nM T98264 CN3EW7 56683882 IC50 > 120000 nM T98264 C5CQY2 56683883 IC50 > 120000 nM T98264 CV4PW2 56683884 IC50 = 40400 nM T98264 CZP28F 57327772 IC50 = 24450 nM T98264 CG71TE 57380427 IC50 > 10000000 nM T98264 C4QJD7 57380429 IC50 > 10000000 nM T98264 CLTX25 57380431 IC50 > 10000000 nM T98264 CU94DW 57380433 IC50 = 129000 nM T98264 CCY75L 57380662 IC50 > 10000000 nM T98264 CE24LJ 57380664 IC50 = 167000 nM T98264 CWZ9E2 57380666 IC50 > 10000000 nM T98264 C9H7GI 57380668 IC50 > 10000000 nM T98264 CXW05S 57390693 IC50 > 10000000 nM T98264 CE57HQ 57395972 IC50 > 10000000 nM T98264 CGC16T 57397768 IC50 > 10000000 nM T98264 C18FTX 57397769 IC50 > 10000000 nM T98264 CQNG21 57397770 IC50 > 10000000 nM T98264 CX3A5R 57399431 IC50 > 10000000 nM T98264 CU5ND3 57514697 IC50 = 21000 nM T98264 C2BT9H 70673568 IC50 = 5000 nM T98264 C3AJ7H 70981706 IC50 = 2300 nM T98264 CP4H6L 70981726 IC50 = 2300 nM T98264 C2KS7Y 70982811 IC50 = 2490 nM T98264 C7VES4 71449486 IC50 = 16810 nM T98264 C5XB2N 71456091 IC50 > 100000 nM T98264 CP43AS 71461531 IC50 > 100000 nM T98264 CXI0F3 71561559 IC50 > 100000 nM T98264 CE0Y3O 71561685 IC50 = 4900 nM T98264 C3M4CF 71561686 IC50 = 4200 nM T98264 C82KCZ 71561687 IC50 = 3400 nM T98264 CDA8P2 71561688 IC50 = 34000 nM T98264 C87EXF 71561689 IC50 = 2600 nM T98264 CP9HX5 71561815 IC50 = 760 nM T98264 C9H5YS 71561816 IC50 = 5700 nM T98264 C61MWP 71561817 IC50 = 5100 nM T98264 C9GO5M 71561818 IC50 = 11500 nM T98264 CWA30F 71561819 IC50 = 5300 nM T98264 CBC4G0 71561820 IC50 = 7100 nM T98264 CPV8Y3 71561944 IC50 = 3700 nM T98264 CPWU40 71597177 IC50 > 50000 nM T98264 CT4MK9 71717989 IC50 > 100000 nM T98264 CCY15D 71734765 IC50 = 910 nM T98264 CS0XU2 72163288 IC50 = 10910 nM T98264 C6F1TD 72163289 IC50 = 14050 nM T98264 C0FWS2 72163422 IC50 = 24370 nM T98264 C2RNH4 72163424 IC50 = 17940 nM T98264 CNLB62 72163425 IC50 = 15770 nM T98264 C2JNO9 73345604 EC50 = 75000 nM T98264 C68EIC 73351713 EC50 = 60000 nM T98264 C20TML 73351714 EC50 = 140000 nM T98264 C1DWU4 73353952 IC50 = 7530 nM T98264 C9UP3V 73353954 IC50 = 12640 nM T98264 CS5O4J 73355491 IC50 = 6930 nM T98264 CMDC47 73357035 IC50 = 8790 nM T98264 CY0K7L 73357036 IC50 = 10610 nM T98264 CT1JH8 86766297 IC50 = 18180 nM T98264 CL4IN3 86766306 IC50 = 17760 nM T98264 CBK96X 90666455 IC50 > 20000 nM T98264 C61PBQ 90666456 IC50 > 20000 nM T98264 C40WCO 90666457 IC50 > 20000 nM T98264 C2ZGE9 90666458 IC50 > 20000 nM T98264 CG5TY1 90666459 IC50 > 20000 nM T98264 CWQN87 90666460 IC50 > 20000 nM T98264 CLU52N 90666461 IC50 = 15020 nM T98264 C0DW7A 90666462 IC50 > 20000 nM T98264 CXMC74 90666463 IC50 > 20000 nM T98264 C19JKD 101884098 IC50 = 78000 nM T98264 CX81PZ 118706101 IC50 = 6.8 ug.mL-1 T98264 CV5Q8J 118706102 IC50 = 5.1 ug.mL-1 T98264 CX2A8G 118722143 IC50 > 120000 nM T98264 CV5F0I 118722144 IC50 > 120000 nM T98264 C32ODE 118729111 IC50 = 5130 nM T98264 CTV62N 118729112 IC50 = 38420 nM T98264 CP9E4Q 118729113 IC50 = 19250 nM T98264 CS2XI7 118729114 IC50 = 8670 nM T98264 C3LN4T 118729115 IC50 = 10000 nM T98264 CF9KD7 118729116 IC50 = 9210 nM T98264 C27YKT 118729117 IC50 = 9250 nM T98264 C5FXC0 118729118 IC50 = 23650 nM T98264 C90UMX 118729119 IC50 = 24880 nM T98264 C4XZ2J 118729123 IC50 = 32240 nM T98264 C5GM1D 118729125 IC50 = 11120 nM T98264 CHF7U0 118729126 IC50 = 15680 nM T98264 C0IJ2X 118737463 IC50 = 8000 nM T98264 CN02HB 122182193 IC50 = 2310 nM T98264 CI87OL 122182194 IC50 = 9080 nM T98264 C12OHP 122187565 IC50 = 7300 nM T98264 CXHR32 122187566 IC50 = 4800 nM T98264 C59OUG 122187567 IC50 = 6000 nM T98264 CKT67D 122196241 IC50 = 2310 nM T98264 C2PVC5 122196288 IC50 = 9610 nM T98264 CV2H8T 122196290 IC50 = 11360 nM T98264 C46PST 127024952 IC50 > 120000 nM T98264 CF05SB 127025572 IC50 > 120000 nM T98264 C0KDZ2 127025573 IC50 > 120000 nM T98264 CI0NR9 127025574 IC50 > 120000 nM T98264 C6RI3J 127025575 IC50 > 120000 nM T98264 C5Z4PH 127025576 IC50 > 120000 nM T98264 C94EIF 127025577 IC50 > 120000 nM T98264 CR87HW 127025578 IC50 > 120000 nM T98264 CM9CP5 127027398 IC50 > 120000 nM T98264 C2A4GS 127027399 IC50 > 120000 nM T98264 CYOQ30 127027703 IC50 > 120000 nM T98264 CX52UN 127027704 IC50 > 120000 nM T98264 C6TIJ1 127027705 IC50 > 120000 nM T98264 C6H9SE 127027706 IC50 > 120000 nM T98264 C2X4JK 127027707 IC50 > 120000 nM T98264 C6UR4C 127027724 IC50 > 120000 nM T98264 C0RQ1U 127027725 IC50 > 120000 nM T98264 C0K2UI 127028022 IC50 > 120000 nM T98264 C1WA5T 127028346 IC50 > 120000 nM T98264 CC8HW0 127028347 IC50 > 120000 nM T98264 C6T0DY 127028683 IC50 > 120000 nM T98264 CL6QV7 127028684 IC50 > 120000 nM T98264 CG68NT 127028685 IC50 > 120000 nM T98264 C3MCH5 127028686 IC50 > 120000 nM T98264 CIAX67 127050086 IC50 = 2450 nM T98264 CEL9C4 127052247 IC50 = 6460 nM T98264 CF5HN6 132938289 IC50 = 8800 nM T98264 CZC42X 135924009 IC50 = 27700 nM T98264 C5BL1Z 135924010 IC50 = 103700 nM T98264 C9UA3N 135924011 IC50 = 32600 nM T98264 C1V8JE 135924012 IC50 = 7100 nM T98264 C8HP1O 135924013 IC50 = 18000 nM T98264 CHUD85 135924014 IC50 = 18100 nM T98264 CTZ5K1 135924015 IC50 = 15900 nM T98264 CAF8B6 135924016 IC50 = 32400 nM T98264 CK4X8S 135924017 IC50 = 10800 nM T98264 CE1FB0 135924018 IC50 = 122800 nM T98264 C39EPD 135924019 IC50 = 43100 nM T98264 CEH2M5 135924020 IC50 = 74200 nM T98264 CN6I5O 135924021 IC50 = 72500 nM T98264 CKW8X5 135924023 IC50 = 19400 nM T98264 CO3EX1 135924024 IC50 = 15700 nM T98264 CBJ7F8 135924025 IC50 = 40900 nM T98264 C81SHP 135924026 IC50 = 42500 nM T98264 CI62JU 135924027 IC50 = 60800 nM T98264 CAL83P 135924028 IC50 = 18300 nM T98264 CJ14VX 135924029 IC50 = 73400 nM T98264 C5C4EP 135924030 IC50 = 15400 nM T98264 C5QIK7 137174949 IC50 > 120000 nM T98264 CDZN68 137635090 IC50 = 10600 nM T98264 C28DUQ 137642390 IC50 = 34620 nM T98264 C48YBW 137646377 IC50 = 5290 nM T98264 CRU6Z7 137796282 IC50 = 72720 nM T98264 C0WMZ4 139593950 IC50 > 36800 nM T98264 C6NQ9I 145720956 IC50 = 14000 nM T98264 C4DWG8 145950748 IC50 = 3450 nM T98264 CIZE64 145960181 IC50 = 2940 nM T98264 CT6I5O 145961409 IC50 = 1090 nM T98264 C58OBV 145971193 IC50 = 850 nM T98264 CUE85W 145971302 IC50 = 4280 nM T98264 CV3FS9 145972458 IC50 = 8630 nM T98264 CB2I5V 155517051 IC50 = 2800 nM T98264 CGUP05 155517773 IC50 = 1520 nM T98264 C1HL4K 155519234 IC50 = 2800 nM T98264 CZ75SL 155521073 IC50 = 2950 nM T98264 C2WP6O 155522824 IC50 = 2800 nM T98264 CW1V5X 155522892 IC50 = 2800 nM T98264 CQ63GA 155537698 IC50 = 1110 nM T98264 CRU6F2 155538623 IC50 = 3990 nM T98264 C3Y6ZF 155538861 IC50 = 29900 nM T98264 CRH8J5 155548680 IC50 = 2540 nM T98264 CL1S9J 155565716 IC50 = 5160 nM T98264 C7W5HT 155566457 IC50 = 27100 nM T98264 D01BZE 73659 IC50 > 40000 nM T98264 D07LUJ 64945 IC50 = 25780 nM T98264 D0E0BU 444763 Ki = 16000 nM T98264 D0F9RO 6918774 IC50 = 24560 nM T98264 D0SJ2Q 10494 IC50 = 14190 nM T98264 D0U8IF 10114 IC50 = 65400 nM T98264 D0Y1RO 1829 Ki = 80000 nM T98264 D0Y5SB 444764 Ki = 510000 nM T48195 D06YPU 39912 IC50 = 100 nM T48195 D00QKI 9865554 IC50 = 16 nM T48195 D0LJ1B 9838712 IC50 = 5.3 nM T48195 D0ZL4F 180540 IC50 = 34 nM T48195 CNB6V7 114864 IC50 = 110 nM T48195 CMJ91Y 667550 IC50 = 50 nM T48195 CCVO02 9972278 IC50 = 360 nM T48195 C1L2WF 10018018 IC50 > 20000 nM T48195 CG2F7V 10200589 IC50 = 398 nM T48195 C7M8NX 10267982 IC50 = 42 nM T48195 C2BM1R 10402760 IC50 = 110 nM T48195 CC7T5M 11414892 IC50 = 80 nM T48195 C6H5VS 11625425 IC50 = 40 nM T48195 CYU1N8 12146502 IC50 = 46 nM T48195 CP6C4M 15980787 IC50 = 43 nM T48195 CT2D7W 15980830 IC50 = 410 nM T48195 CWEK41 15980918 IC50 > 20000 nM T48195 CM31SA 15980919 IC50 = 5100 nM T48195 C2OW0T 15981315 IC50 = 760 nM T48195 CV5M7D 15981316 IC50 = 160 nM T48195 CEW06X 15981317 IC50 = 200 nM T48195 C9KT1A 15981347 IC50 = 220 nM T48195 CY79RO 15981348 IC50 = 94 nM T48195 CT4C8A 15981349 IC50 = 50 nM T48195 CFJ3N8 15981350 IC50 = 680 nM T48195 CQGO53 16098481 IC50 = 251 nM T48195 C5NPO3 44284796 IC50 = 83 nM T48195 CCZ79T 44285113 IC50 > 20000 nM T48195 CO2Z4F 44285114 IC50 > 20000 nM T48195 C7CAM3 44285230 IC50 = 1000 nM T48195 C9VTS1 44285279 IC50 = 220 nM T48195 C30HNE 44285280 IC50 = 2700 nM T48195 CA52QI 44285430 IC50 = 12500 nM T48195 CFA7G2 44298268 Ki = 23000 nM T48195 CK45QG 44298269 Ki = 1700 nM T48195 CX7RL3 44298270 Ki = 68000 nM T48195 CVB2L1 44298317 Ki = 300 nM T48195 C6AE8K 44298340 Ki = 10000 nM T48195 CM3NT2 44298341 Ki = 13000 nM T48195 CKEX94 44298371 Ki = 120000 nM T48195 C6Q3WF 44298372 Ki = 190000 nM T48195 CAY2Q5 44298412 Ki = 750000 nM T48195 C3V1OQ 44298415 Ki = 3100000 nM T48195 C4EZ1W 44298416 Ki = 1850000 nM T48195 CAZG75 44298417 Ki = 890000 nM T48195 CWJX62 44298478 Ki > 1000 nM T48195 CEPB90 44298479 Ki > 1000 nM T48195 CWIA49 44298480 Ki > 30000 nM T48195 C8A9ZY 44298517 Ki > 30000 nM T48195 CRB25O 44298566 Ki = 55000 nM T48195 C5HB7Q 44298567 Ki = 27000 nM T48195 CE1FD5 44298568 Ki = 400000 nM T48195 C8WR7Q 44298569 Ki = 61000 nM T48195 C46FCX 44298606 Ki = 265000 nM T48195 CY3NW7 44298652 Ki = 155000 nM T48195 CK15HY 44298653 Ki = 15000 nM T48195 C06XVP 44298672 Ki = 62000 nM T48195 CED36R 44298676 Ki = 42000 nM T48195 C7QI1B 44298677 Ki = 29000 nM T48195 C6IW4P 44298701 Ki = 14000 nM T48195 C0QCP8 44298702 Ki = 5000 nM T48195 CL8E5P 44298703 Ki = 107000 nM T48195 C37RPZ 44298719 Ki = 42000 nM T48195 CO40US 44298729 Ki = 32000 nM T48195 C91FYI 44298730 Ki = 49000 nM T48195 CYI87G 44298744 Ki = 55000 nM T48195 C0RV8X 44298745 Ki = 27000 nM T48195 CUGS48 44298788 Ki = 28000 nM T48195 CY58NT 44298789 Ki = 2050000 nM T48195 CIZ42J 44298801 Ki = 2700000 nM T48195 C7RS5H 46896782 IC50 = 52 nM T48195 CX57UB 46896783 IC50 = 80 nM T48195 C0CEV2 46897163 IC50 = 22 nM T48195 C8E3GN 46897164 IC50 = 1220 nM T48195 CPL1N2 46897165 IC50 = 90 nM T48195 CI2J0B 46897254 IC50 = 387 nM T48195 CV7HR1 46897255 IC50 = 689 nM T48195 CE2D6V 77844109 IC50 > 10000 nM T48195 CC7Y9A 77844110 IC50 > 10000 nM T48195 C0VD5A 122187268 IC50 = 185 nM T48195 CW51VO 135485575 IC50 = 8990 nM T48195 C6J7ZP 135673987 IC50 = 2000 nM T48195 D09FHA 11322291 IC50 = 1.8 nM T48195 D09MAZ 46897162 IC50 = 36 nM T40332 D04AIT 5280445 Ki = 10100 nM T40332 D0FT4R 107706 Ki = 37 nM T40332 D0K8KX 5280343 Ki = 11900 nM T40332 D0SH3I 387447 Ki = 2300 nM T40332 D0V3YT 10324367 IC50 = 17000 nM T40332 D0X7JN 5280980 IC50 < 40000 nM T40332 D0X9CH 3010818 IC50 = 680 nM T40332 D00LOB 9866964 Ki > 26000 nM T40332 D06KJQ 42601552 IC50 > 30000 nM T40332 D08PBB 177992 IC50 = 23 nM T40332 D0A0SI 66601502 IC50 = 0.065 nM T40332 D0U2BH 65064 IC50 = 12800 nM T40332 D0VO0T 24800541 IC50 = 3550 nM T40332 D0Y6SQ 2536 IC50 > 100000 nM T40332 D00AWA 9938355 Ki = 0.013 nM T40332 D02PHE 46861623 IC50 = 12 nM T40332 D02YSI 44316902 Ki = 12 nM T40332 D06DET 9807572 IC50 = 29 nM T40332 D08ZCW 9910174 IC50 > 10 nM T40332 D0I0FM 44445940 Ki = 10 nM T40332 D0R9ON 65837 IC50 = 1000 nM T40332 D0U7OU 3220 IC50 = 52000 nM T40332 D0WY9H 9892148 Ki = 1.3 nM T40332 C19TYR 44343121 IC50 = 10500000 nM T40332 C3N6FP 44342779 IC50 = 13500000 nM T40332 CT8RD6 1526 Ki = 15 nM T40332 CX09SM 1636 Ki = 18 nM T40332 C7ET4R 6773 IC50 = 39000 nM T40332 C4RT3E 10208 IC50 = 18000 nM T40332 C73JPZ 10639 IC50 = 6200 nM T40332 C0WN5U 13926 Ki = 9549.93 nM T40332 CE1GQ3 68236 Ki = 4786.3 nM T40332 CF7O4D 125700 IC50 = 40 nM T40332 CB17TY 128954 IC50 = 2000 nM T40332 CLX4V7 130395 IC50 > 100000 nM T40332 C5Q7EX 160817 IC50 = 11000 nM T40332 CW4AE7 178662 Ki = 0.014 nM T40332 C0Z8UG 191187 IC50 = 10000 nM T40332 CIGP91 196813 IC50 = 9000 nM T40332 CQJD84 216294 Ki = 12 nM T40332 C05PDV 223000 Ki = 831763.77 nM T40332 C4HLA8 223062 IC50 = 100000 nM T40332 CC9E0Y 232547 IC50 = 15600 nM T40332 CPJW07 294660 Ki = 4365.16 nM T40332 CH46ID 296003 Ki = 1778.28 nM T40332 C1WRQ6 309231 IC50 >= 28000 nM T40332 CXOC26 339156 Ki = 112.2 nM T40332 CB39JK 343129 IC50 = 13000 nM T40332 CJ1R7C 433517 IC50 > 100000 nM T40332 CCX8A5 468714 Ki = 6 nM T40332 CT79FC 468715 IC50 = 44 nM T40332 CG2SL7 468760 IC50 = 92 nM T40332 C5XV2G 481422 IC50 > 1000000 nM T40332 CW1KP3 481437 IC50 > 300000 nM T40332 C7ZUS1 481440 IC50 > 600000 nM T40332 C9EAL6 482277 IC50 > 75000 nM T40332 C58PLQ 482278 IC50 > 75000 nM T40332 C2G9IH 482279 IC50 > 75000 nM T40332 C5L4ED 482280 IC50 > 75000 nM T40332 CTW1J9 482282 IC50 > 75000 nM T40332 CK0O9U 482283 IC50 > 75000 nM T40332 CX0SQ5 482284 IC50 > 75000 nM T40332 C6Y5SA 482285 IC50 > 75000 nM T40332 C2D7MH 482286 IC50 > 75000 nM T40332 CAZV26 482287 IC50 > 75000 nM T40332 C2QP9I 482288 IC50 > 75000 nM T40332 C3L9TI 482289 IC50 > 75000 nM T40332 CO3N0A 482290 IC50 > 75000 nM T40332 CZ15KR 482291 IC50 > 75000 nM T40332 C0HV7G 482292 IC50 > 75000 nM T40332 CC1RP8 483672 IC50 < 60 nM T40332 C3N7CD 487110 IC50 = 30000 nM T40332 C6B1KZ 504659 Ki = 6.457 nM T40332 CVE0Y8 504661 Ki = 0.1148 nM T40332 CTD7X8 504663 Ki = 0.04266 nM T40332 CN67CR 555078 Ki = 28 nM T40332 C32HXT 589588 Ki = 1905.46 nM T40332 CRQ98S 589620 Ki = 645.65 nM T40332 CM7T6V 589629 Ki = 302 nM T40332 C9Y3FN 589883 Ki = 10964.78 nM T40332 C9YWX0 607716 IC50 = 16000 nM T40332 C0LDK9 611090 Ki = 7244.36 nM T40332 CD23NS 628877 IC50 >= 28000 nM T40332 CFO5M9 630168 IC50 >= 28000 nM T40332 CQ94TR 639465 Ki = 15700 nM T40332 CD5P8N 644145 IC50 = 5000 nM T40332 CTDG97 644152 IC50 = 168000 nM T40332 CAJ4F5 644153 IC50 = 21000 nM T40332 C7Q0UO 644154 IC50 = 41000 nM T40332 CREX84 644155 IC50 = 151000 nM T40332 C28PBX 644930 IC50 > 100000 nM T40332 CCKZ79 668744 IC50 = 51500 nM T40332 C53FNM 674593 Ki = 15 nM T40332 C45NBS 674629 Ki = 107 nM T40332 C21HDC 674632 Ki = 24 nM T40332 CG2UK8 674633 Ki = 1000 nM T40332 CX1W4S 674635 Ki = 7200 nM T40332 C9PI4L 674639 Ki = 9000 nM T40332 C3M8OE 674640 Ki = 9000 nM T40332 CI9LH0 674642 Ki = 1100 nM T40332 CBX3U0 674652 Ki = 6 nM T40332 COD8V2 674657 Ki = 3100 nM T40332 CW5ZA1 680939 Ki = 24 nM T40332 CN06WE 685663 Ki = 10700 nM T40332 CXDC18 714833 Ki = 24500 nM T40332 CFP1A9 730175 Ki = 820 nM T40332 C87WLA 753830 Ki = 50900 nM T40332 C0ER8S 767161 IC50 = 124900 nM T40332 CDVJ42 767163 IC50 = 15500 nM T40332 CE10WO 776842 IC50 = 160200 nM T40332 CYF3T7 806239 Ki = 8912.51 nM T40332 CU85MI 823661 Ki = 2884.03 nM T40332 C8BQU5 833517 Ki = 300 nM T40332 C2O5LR 849299 IC50 = 20000 nM T40332 CLR3H1 899247 Ki = 21 nM T40332 CV23JB 914899 Ki = 169.82 nM T40332 C5SN4P 928297 Ki = 3630.78 nM T40332 CLR10O 928795 Ki = 11.48 nM T40332 CQ2R0M 1011274 IC50 = 78300 nM T40332 C5AM9V 1169804 IC50 > 100000 nM T40332 CWJL58 1169805 IC50 > 100000 nM T40332 CX1W4I 1170184 IC50 > 100000 nM T40332 C2PRY6 1269450 IC50 = 6700 nM T40332 CUL5Y4 1331170 IC50 > 100000 nM T40332 CW90DG 1457429 IC50 > 100000 nM T40332 CENL04 1523065 IC50 = 5100 nM T40332 CYH46M 1993219 IC50 > 100000 nM T40332 C0D8LM 2213207 Ki = 29900 nM T40332 CO4AB7 2264784 IC50 = 52200 nM T40332 C3A9BT 2302435 Ki = 1.8 nM T40332 C8DW1C 2372853 IC50 > 100000 nM T40332 CC5R9U 2796528 Ki = 34673.69 nM T40332 CKJ5T0 2812522 IC50 = 61 nM T40332 CYW3M6 3223864 IC50 > 100000 nM T40332 C45ZIU 3368775 IC50 >= 28000 nM T40332 CAEW98 3435549 IC50 > 100000 nM T40332 CNJM56 3534338 IC50 > 60000 nM T40332 CPC72H 3835811 IC50 = 32100 nM T40332 CJDR03 3963048 Ki = 1600 nM T40332 C6JF0O 4155991 IC50 = 2700 nM T40332 C9FTM3 5113707 Ki = 71 nM T40332 C9UOQ3 5151183 Ki = 2570.4 nM T40332 CF9VK2 5236960 IC50 = 26900 nM T40332 CK2X1T 5271294 IC50 > 75000 nM T40332 CWIC65 5279637 IC50 = 36100 nM T40332 CAF61Z 5289347 Ki = 25 nM T40332 CV20QH 5294946 IC50 > 100000 nM T40332 CO58XD 5311161 IC50 > 100000 nM T40332 CA63CX 5367020 Ki = 8128.31 nM T40332 CCUM24 5467627 IC50 = 2900 nM T40332 C4VIT3 5480997 IC50 = 20 nM T40332 CDV72G 5480998 IC50 = 3200 nM T40332 CZ1XU5 5876194 IC50 = 19600 nM T40332 COD34R 6451966 Ki = 954.99 nM T40332 CQS5E1 6888904 IC50 = 17600 nM T40332 C8OE6S 6913584 IC50 > 100000 nM T40332 CG2A7X 7028541 IC50 = 84800 nM T40332 CECO04 8967103 IC50 >= 28000 nM T40332 CF4TK5 8967105 IC50 >= 28000 nM T40332 C89JBK 9636571 IC50 > 100000 nM T40332 CZ8V7U 9799757 IC50 = 1000 nM T40332 CE56CV 9804093 Ki = 114 nM T40332 CUX59Q 9804457 Ki = 0.066 nM T40332 CL8TN0 9806936 Ki = 170 nM T40332 CRJ6I2 9808548 Ki = 1.66 nM T40332 C4DIG6 9808564 Ki = 0.022 nM T40332 C84XOY 9808874 Ki = 0.025 nM T40332 C92HSW 9809309 IC50 = 24 nM T40332 CZ6W1Y 9809577 IC50 = 21 nM T40332 CFSX09 9815828 Ki = 1.5 nM T40332 CT2WM1 9827187 Ki = 4.9 nM T40332 C4I0UG 9829396 IC50 = 6.6 nM T40332 C9YO0Z 9830006 Ki = 0.7 nM T40332 CH31WN 9830037 Ki = 0.008 nM T40332 CGNB60 9830581 IC50 = 9500 nM T40332 CR54JK 9830622 IC50 = 30 nM T40332 CZFT64 9830860 IC50 = 20 nM T40332 C6NIU3 9831417 Ki = 0.2 nM T40332 CM53FA 9834041 Ki = 63000 nM T40332 C2NX3Q 9852363 IC50 = 27 nM T40332 C6R7XS 9852378 IC50 = 23 nM T40332 CDL5O0 9866692 Ki = 0.7 nM T40332 CBC5V7 9866842 Ki = 0.035 nM T40332 CX92DE 9871592 Ki = 26 nM T40332 CI5T7N 9873436 IC50 = 17 nM T40332 C2T6QH 9875205 Ki = 0.45 nM T40332 CS3C0L 9887581 IC50 < 150 nM T40332 CL61HY 9888442 Ki = 0.014 nM T40332 CG2EZ0 9889108 Ki = 0.31 nM T40332 C3H0LQ 9892781 Ki = 3.35 nM T40332 CCX4N0 9893147 Ki = 170 nM T40332 COA8T5 9894208 IC50 = 6.6 nM T40332 CEO04L 9894378 Ki = 5.1 nM T40332 CZQ97P 9895636 IC50 = 14 nM T40332 C9IZB4 9904055 IC50 = 4000 nM T40332 C7KJP3 9908917 Ki = 1.73 nM T40332 C1T5VN 9912574 Ki = 725 nM T40332 CJ6M8N 9915812 IC50 > 300000 nM T40332 C08KHW 9917190 IC50 = 62 nM T40332 C2HY9N 9917412 IC50 = 47 nM T40332 CQ84MG 9917430 Ki = 6.3 nM T40332 C8D5CH 9920598 Ki = 51 nM T40332 CGT3K4 9932145 Ki = 0.16 nM T40332 CRK8F2 9933704 Ki = 44.3 nM T40332 CG2Q1F 9934160 Ki = 79.7 nM T40332 CA8DY4 9938068 IC50 = 28 nM T40332 CXA7B4 9953653 Ki = 0.3 nM T40332 C3EPC4 9955758 Ki > 22000 nM T40332 CUY4S5 9960766 IC50 = 27 nM T40332 C2VU3Y 9962219 IC50 = 84 nM T40332 C2CE1A 9962331 Ki = 0.2 nM T40332 C3HI6E 9972080 IC50 = 47 nM T40332 CM06CQ 9973338 Ki = 100 nM T40332 C1UKM3 9977679 Ki = 320 nM T40332 C4J0GP 9978440 Ki = 52 nM T40332 CW56ZP 9978595 Ki = 500 nM T40332 C1VB6K 9980302 Ki = 0.6 nM T40332 C7E9BA 9980407 Ki = 54 nM T40332 C5ZNO7 9980554 Ki = 43 nM T40332 C58VXC 9982602 Ki = 51 nM T40332 C09EYT 9983109 Ki = 94 nM T40332 C12ITA 9984374 Ki = 190 nM T40332 C2B9IN 9985199 Ki = 13 nM T40332 CME79C 9985374 Ki = 25 nM T40332 CIJ5L2 9987080 IC50 = 6700 nM T40332 CCE26Y 10002661 Ki = 0.03 nM T40332 CPO47T 10002668 Ki = 46 nM T40332 C7UON4 10002900 Ki = 270 nM T40332 C6ANW0 10004044 Ki = 280 nM T40332 C7YSW2 10004682 Ki = 340 nM T40332 CW2G0I 10005629 Ki = 261 nM T40332 CMV31E 10006663 Ki = 4300 nM T40332 CBXZ29 10007724 Ki = 13 nM T40332 CC1JY8 10008607 Ki = 4.2 nM T40332 CTEQ15 10008826 Ki = 0.55 nM T40332 C95FMS 10009631 Ki = 1.5 nM T40332 CFBX35 10014336 IC50 > 1000000 nM T40332 C1MKH6 10015569 IC50 > 1000000 nM T40332 CI8PL9 10016936 IC50 = 221.5 nM T40332 CN16OT 10022457 Ki = 8 nM T40332 C87NHX 10023592 Ki = 1100 nM T40332 CWB04G 10023940 IC50 = 28000 nM T40332 CO75QM 10024023 Ki = 0.8 nM T40332 CHC6E8 10024782 Ki = 101 nM T40332 CH32TU 10026529 Ki = 6.5 nM T40332 CPMA30 10026572 IC50 = 200 nM T40332 CEO32W 10027816 Ki = 9.3 nM T40332 CG0H4T 10028039 Ki = 10 nM T40332 CL1RN4 10028081 Ki = 19 nM T40332 C6GMX9 10028968 Ki > 500000 nM T40332 CQ9A2O 10029003 Ki = 7.7 nM T40332 C9XH3K 10029428 Ki = 49 nM T40332 CL8WU9 10029465 Ki = 1.2 nM T40332 CEA89V 10029470 Ki = 270 nM T40332 CDM5V2 10029484 Ki = 0.8 nM T40332 CEN3S7 10029919 Ki = 15 nM T40332 CF1SN8 10029970 Ki = 33 nM T40332 C07UYT 10030271 Ki = 66 nM T40332 C1KIE7 10030460 Ki = 21000 nM T40332 CYW21E 10030835 Ki = 20 nM T40332 CGK82S 10031500 Ki = 88 nM T40332 CUM1S3 10032109 Ki = 12 nM T40332 C1FM9L 10032899 Ki = 0.33 nM T40332 C35XZA 10036576 Ki = 257.04 nM T40332 C8RNZ5 10043396 Ki = 60 nM T40332 CG7F8T 10048188 Ki = 210 nM T40332 CVHQ60 10048700 Ki = 22 nM T40332 CEH7X8 10049090 Ki = 6.2 nM T40332 CS9U8H 10052095 Ki = 80000 nM T40332 C5HYK8 10052622 Ki = 130 nM T40332 CH3NT1 10052689 Ki = 300 nM T40332 CNK54H 10052690 Ki = 16 nM T40332 C14TNZ 10053504 Ki = 89 nM T40332 CH7B0C 10053891 Ki = 2.3 nM T40332 C4K3QL 10054085 Ki = 0.11 nM T40332 CVZU17 10054360 Ki = 0.07 nM T40332 CRJ2W9 10054620 Ki = 0.011 nM T40332 C8DHG9 10054626 Ki = 1.1 nM T40332 CH8YI6 10054689 Ki = 16 nM T40332 CF2V0Y 10055681 Ki = 0.3 nM T40332 CH70LT 10055869 Ki = 0.81 nM T40332 CRL8D2 10060710 Ki = 1.349 nM T40332 CM7XN1 10067940 Ki = 24 nM T40332 CO6QV4 10069016 Ki = 350 nM T40332 CBAU50 10071439 Ki = 4.9 nM T40332 CWJ29L 10071504 Ki = 3400 nM T40332 CIO8S2 10071747 Ki = 57 nM T40332 C8GVA0 10072025 Ki = 0.06 nM T40332 C7MZL9 10073426 Ki = 16 nM T40332 CVGW19 10074999 Ki = 22000 nM T40332 C4DG6S 10075424 Ki = 40 nM T40332 C8YT1B 10076039 Ki = 24 nM T40332 C8BHG0 10076168 Ki = 5600 nM T40332 C3WCV4 10076315 Ki = 87000 nM T40332 C5V1YC 10076625 Ki = 8.4 nM T40332 C8TVW3 10076806 Ki = 5.7 nM T40332 CL59QU 10076807 Ki = 42 nM T40332 C2H5PM 10076832 Ki = 330 nM T40332 C9MZ0X 10076908 Ki = 1.9 nM T40332 C6FUN8 10077271 Ki = 42 nM T40332 CZG6L4 10077327 Ki = 4.4 nM T40332 C67HUG 10077412 Ki = 0.2 nM T40332 CO4NR6 10077495 Ki = 2.8 nM T40332 CMG13S 10077534 Ki = 0.4 nM T40332 C1CFV6 10078395 Ki = 0.43 nM T40332 C7CW1P 10080504 IC50 = 58 nM T40332 CD3N9Q 10084731 Ki = 5.754 nM T40332 C45MKR 10087296 IC50 > 50000 nM T40332 CEH86P 10088912 Ki = 4 nM T40332 CKX3J8 10092679 Ki = 0.07 nM T40332 C5YF2B 10092898 Ki = 18 nM T40332 CEN06H 10093642 IC50 > 100000 nM T40332 CNS73M 10093670 IC50 = 140 nM T40332 CPSY01 10093766 Ki = 8.7 nM T40332 CZU18G 10094548 Ki = 730 nM T40332 CA6WS0 10095870 Ki = 1 nM T40332 CPY1Q7 10097512 Ki = 0.55 nM T40332 CNX98I 10098504 Ki = 6.6 nM T40332 CU4N0V 10098932 Ki = 3.6 nM T40332 CC7WV4 10099005 Ki = 8.2 nM T40332 CNZ68F 10099030 Ki = 22 nM T40332 CKM91H 10099223 Ki = 3.5 nM T40332 CWG0Q4 10099305 Ki = 8.5 nM T40332 CSXU07 10099653 Ki = 1.18 nM T40332 CP2D8N 10099715 Ki = 2.4 nM T40332 C83RTX 10100215 Ki = 0.37 nM T40332 C57PNI 10101455 Ki = 3 nM T40332 CSY56V 10101683 Ki = 0.66 nM T40332 CV8U6L 10101834 Ki = 0.1 nM T40332 C58BWQ 10113382 Ki = 14 nM T40332 C3VA2F 10116108 Ki = 6.38 nM T40332 C3RFT8 10118557 Ki = 2.55 nM T40332 CJLB36 10138967 Ki = 43.8 nM T40332 CXR76P 10138974 Ki = 16.6 nM T40332 CVBL74 10160118 Ki = 26.4 nM T40332 CG6Z3R 10165977 Ki = 1.37 nM T40332 CPU95M 10198315 Ki = 83.18 nM T40332 C5BEP1 10227093 Ki = 6.76 nM T40332 CD8OU0 10241309 Ki = 6900 nM T40332 CDLR68 10250073 Ki = 62 nM T40332 CUY45Q 10251702 Ki = 350 nM T40332 CEHC01 10254338 Ki = 8.5 nM T40332 CA3E1W 10256440 Ki = 8 nM T40332 CK1NB4 10257209 Ki = 34 nM T40332 CZ1B8M 10257257 Ki = 87 nM T40332 CY8NL9 10257279 Ki = 11 nM T40332 CKX95D 10257311 Ki = 6.6 nM T40332 CR8D4G 10257948 Ki = 0.93 nM T40332 CEC58D 10258115 Ki = 4.4 nM T40332 C04XJL 10264928 Ki = 13 nM T40332 CXWQ38 10274774 Ki = 23.5 nM T40332 CB28OA 10275675 Ki = 8.75 nM T40332 CA2YG9 10297988 Ki = 10.7 nM T40332 C97QRW 10298752 Ki = 15.3 nM T40332 CT3A2S 10300047 Ki = 24.8 nM T40332 C8DU7V 10300829 Ki = 2.25 nM T40332 C0X2CU 10302080 Ki = 0.52 nM T40332 CQA3X0 10321894 Ki = 0.023 nM T40332 CD5QM2 10323328 Ki = 39 nM T40332 CW8A4E 10325129 Ki = 52 nM T40332 CW3X4Q 10325189 Ki = 3400 nM T40332 CNXE05 10325233 Ki = 1.4 nM T40332 CA9X6O 10326668 Ki = 8000 nM T40332 CWV2A9 10327283 Ki = 25 nM T40332 C0PJN3 10331933 Ki = 2.73 nM T40332 COA7X1 10338134 Ki = 8 nM T40332 CYCO34 10341700 Ki = 0.07079 nM T40332 CU7FE3 10342642 Ki = 26 nM T40332 C0FME8 10343129 Ki = 27 nM T40332 CS16AL 10343238 Ki = 43000 nM T40332 CIE4G0 10343847 Ki = 3.59 nM T40332 C2GLK6 10346121 IC50 > 50000 nM T40332 C1PI8K 10346591 Ki = 150 nM T40332 C9GL1U 10346870 Ki = 15 nM T40332 CKJC76 10347501 Ki = 23 nM T40332 CO3WL8 10347655 Ki = 33 nM T40332 CC3NH2 10347721 Ki = 4.1 nM T40332 CZ58RW 10347871 Ki = 3.5 nM T40332 C0VL6K 10347891 Ki = 1.8 nM T40332 C1XV8P 10348077 Ki = 4.8 nM T40332 C2VWM9 10348957 Ki = 0.013 nM T40332 CMW89Q 10349323 Ki = 36 nM T40332 C6YUW8 10349541 Ki = 25 nM T40332 CY3L2F 10358434 Ki = 31 nM T40332 C1B6UP 10361206 Ki = 2800 nM T40332 C2I1XM 10363347 Ki = 51000 nM T40332 CK60UV 10366641 Ki = 15 nM T40332 C7K9PJ 10367217 Ki = 2500 nM T40332 CE6VW2 10368099 Ki = 6.7 nM T40332 CS4UX5 10368963 Ki = 16000 nM T40332 C62KEB 10369593 Ki = 4 nM T40332 CK2YU1 10369681 Ki = 4.5 nM T40332 C01CPM 10369682 Ki = 480 nM T40332 CATB56 10370141 Ki = 31 nM T40332 CU3ZF4 10370563 Ki = 8.1 nM T40332 CAT02C 10370853 Ki = 1.8 nM T40332 CGH83D 10371178 Ki = 3.8 nM T40332 CH1RY5 10371190 Ki = 150000 nM T40332 CG9UT0 10371325 Ki = 1.3 nM T40332 CC7RW2 10371949 Ki = 43 nM T40332 CDP4T7 10372563 Ki = 0.5 nM T40332 C5FYM0 10372900 Ki = 0.2 nM T40332 CND9F2 10378134 Ki = 12.59 nM T40332 C1P9VJ 10389512 Ki = 42 nM T40332 CKY94N 10389844 Ki = 34 nM T40332 C8I3WV 10390162 IC50 = 20300 nM T40332 C6RHB5 10390443 Ki = 48 nM T40332 CL49JD 10391720 Ki = 13 nM T40332 CMZ05N 10391723 Ki = 15 nM T40332 CX0KM7 10392329 IC50 = 1 nM T40332 CD6MQ8 10392657 Ki = 5.6 nM T40332 C2FLG8 10392960 Ki = 79 nM T40332 CF05VG 10393052 Ki = 71 nM T40332 C48IQH 10393970 Ki = 47 nM T40332 CH32ZO 10394405 Ki = 32 nM T40332 C3TU6O 10394985 Ki = 25 nM T40332 CBF97Q 10397988 Ki = 91 nM T40332 CC5Q6K 10405508 Ki = 15000 nM T40332 CL48XK 10412920 Ki = 80 nM T40332 C4IUT8 10414698 Ki = 0.011 nM T40332 CSDZ76 10414749 Ki = 30 nM T40332 CPE67V 10414810 Ki = 11 nM T40332 CSH83N 10414990 Ki = 40 nM T40332 C36VYB 10415426 Ki = 12000 nM T40332 CHV37A 10415461 Ki = 15 nM T40332 CQY79A 10415479 Ki = 6.9 nM T40332 CSKX23 10415744 Ki = 17 nM T40332 CNT27F 10415810 Ki = 60 nM T40332 CN7D3W 10415869 Ki = 12 nM T40332 C4MC7H 10416037 Ki = 9.4 nM T40332 C2KJR0 10426076 Ki = 2700 nM T40332 C3IC8F 10432526 Ki = 1100 nM T40332 CW2D3O 10432804 Ki = 1000 nM T40332 CTF92S 10434048 Ki = 37 nM T40332 C84QZG 10434385 Ki = 28 nM T40332 C0CPI1 10435585 Ki = 23 nM T40332 C1RI4C 10435834 Ki = 6.6 nM T40332 CK2SL0 10435916 Ki = 170 nM T40332 C1Z6TU 10436952 Ki = 48 nM T40332 COST60 10436956 Ki = 7 nM T40332 CV7YC6 10436990 Ki = 320 nM T40332 CH6Q2J 10437166 Ki = 6 nM T40332 CV1LD0 10437728 Ki = 18 nM T40332 CXR12A 10438569 Ki = 42 nM T40332 C59OXM 10439034 Ki = 20 nM T40332 C5N0OZ 10439282 Ki = 0.35 nM T40332 C5Z1IB 10440161 Ki = 0.66 nM T40332 C79OYK 10440316 Ki = 0.1 nM T40332 C08TPL 10440405 Ki = 0.06 nM T40332 CQ5DM6 10452703 Ki = 1.995 nM T40332 CQ6G5E 10453174 Ki = 290 nM T40332 CHNG31 10453578 Ki = 1.995 nM T40332 COX97B 10454399 Ki = 30 nM T40332 CJ5FS1 10456006 Ki = 26 nM T40332 CTF5G1 10457246 Ki = 6100 nM T40332 CW7FT8 10457506 Ki = 40 nM T40332 CRH7I5 10457598 Ki = 71 nM T40332 C06QJW 10457653 IC50 > 50000 nM T40332 CKY0C5 10459649 Ki = 8.8 nM T40332 C6BQL9 10459820 Ki = 57 nM T40332 C5N9DB 10460031 IC50 > 300000 nM T40332 C1L0VN 10460376 Ki = 23 nM T40332 CB4K1S 10460522 Ki = 11 nM T40332 COL58Y 10460549 Ki = 18 nM T40332 CQ0S8Y 10460720 Ki = 9 nM T40332 CH17CO 10460911 Ki = 1.1 nM T40332 C15YVO 10461918 IC50 = 33 nM T40332 CO1XS4 10462803 Ki = 9.4 nM T40332 CHJ27G 10462942 Ki = 0.65 nM T40332 C9Y2MK 10468056 Ki = 1.43 nM T40332 CYD67S 10475537 Ki = 0.1 nM T40332 C8C9YS 10477377 Ki = 26 nM T40332 C7DHG4 10478230 Ki = 510 nM T40332 CCNA48 10479704 Ki = 360 nM T40332 CO6U0V 10479967 Ki = 20.5 nM T40332 C9XB8D 10481065 Ki = 17 nM T40332 CJNT56 10481404 Ki = 190 nM T40332 C09HJD 10481557 Ki = 410 nM T40332 C5U6DL 10481845 Ki = 469 nM T40332 C2GEQ9 10482544 Ki = 52 nM T40332 CR5F0K 10483274 Ki = 9.6 nM T40332 CU0EA3 10483607 IC50 = 260000 nM T40332 C90THX 10484261 Ki = 4.6 nM T40332 CWN6L8 10484563 Ki = 72 nM T40332 CF5W6B 10491098 Ki = 133 nM T40332 CFP53Y 10502109 IC50 = 2260 nM T40332 C60MXW 10505465 Ki = 0.027 nM T40332 CQW51O 10506703 IC50 = 183000 nM T40332 CYQB28 10507021 IC50 > 300000 nM T40332 CFNK35 10507077 IC50 > 300000 nM T40332 CPET76 10517251 Ki = 238 nM T40332 CA4RW1 10517868 IC50 = 11000 nM T40332 CG34WR 10518548 Ki = 100 nM T40332 C5Y1XO 10527174 Ki = 0.5 nM T40332 CYJ58Q 10528103 Ki = 15 nM T40332 CQES53 10529707 Ki = 130 nM T40332 C84WLX 10531366 Ki = 5.7 nM T40332 CQC62W 10531634 Ki = 1.6 nM T40332 CZ29RX 10537951 Ki = 3.981 nM T40332 C7B8LG 10549313 Ki = 0.85 nM T40332 C5J7MX 10550886 Ki = 4281 nM T40332 C5KO9W 10553305 Ki = 0.81 nM T40332 C5G6SC 10553739 Ki = 15 nM T40332 CAKY60 10554399 Ki = 3 nM T40332 C7NJQ1 10554839 IC50 > 300000 nM T40332 C0T6QD 10556018 Ki = 5500 nM T40332 CER1M4 10560388 Ki = 41.69 nM T40332 CC2DB8 10564561 Ki = 12.59 nM T40332 CVX74R 10569244 IC50 < 200 nM T40332 CP1HE3 10571766 Ki = 0.06 nM T40332 C6Y1XV 10573143 Ki = 0.03 nM T40332 C3F4KN 10577308 Ki = 12 nM T40332 C9EK8W 10579293 Ki = 1100000 nM T40332 CJ5MB0 10579493 Ki = 0.35 nM T40332 C3VR0Q 10579612 Ki = 1.1 nM T40332 C3HJ4N 10579613 Ki = 3.4 nM T40332 CXF17L 10579679 Ki = 3.1 nM T40332 CBM4L7 10591621 IC50 > 1000000 nM T40332 C7HM6O 10599457 Ki = 0.22 nM T40332 CZB90H 10601497 Ki = 330 nM T40332 CQ9BP2 10601989 Ki = 4200 nM T40332 CGS56E 10610038 Ki = 5.61 nM T40332 CKN60O 10612715 Ki = 51 nM T40332 CQ38DS 10615154 IC50 = 6600 nM T40332 CYQC10 10615902 IC50 = 1200 nM T40332 C53MHY 10616362 Ki = 288.4 nM T40332 CPN7X5 10624194 Ki = 11.8 nM T40332 C8XA3U 10626170 Ki = 8 nM T40332 CDLP35 10628028 Ki = 70 nM T40332 CS18WR 10635550 Ki = 5.7 nM T40332 COL8B0 10636536 Ki = 91 nM T40332 CG69CZ 10638623 IC50 = 36000 nM T40332 CD86WR 10647120 Ki = 0.72 nM T40332 CDL36E 10647461 Ki = 0.14 nM T40332 CQ0O5J 10648323 Ki = 160 nM T40332 C5T8WG 10650026 Ki = 57.8 nM T40332 CZ78MR 10651388 Ki = 9.9 nM T40332 CME37Y 10651433 Ki = 6.4 nM T40332 CBHW74 10653967 Ki = 1000 nM T40332 CMXS14 10653995 Ki = 20 nM T40332 CW75PO 10661946 IC50 > 500 nM T40332 CM2IJ0 10665528 IC50 = 75000 nM T40332 CQAG87 10670178 Ki = 0.025 nM T40332 C71RBG 10670907 Ki = 0.025 nM T40332 CX36QE 10671458 Ki = 0.034 nM T40332 CJ1B0W 10671534 Ki = 0.013 nM T40332 CDB35L 10673162 Ki = 74 nM T40332 CP1V5D 10673918 Ki = 44 nM T40332 CN0I1R 10673962 Ki = 2.3 nM T40332 CCF8L6 10674356 IC50 > 300000 nM T40332 COSG14 10675303 Ki = 58 nM T40332 C8A0EJ 10680902 Ki = 28.84 nM T40332 COM2A7 10687511 IC50 = 900 nM T40332 CVCW48 10694581 Ki = 310 nM T40332 CC35DA 10695507 IC50 = 2660 nM T40332 CNEA57 10696461 Ki = 42 nM T40332 CT6ME5 10696947 Ki = 19 nM T40332 CZ8C2D 10697242 Ki = 0.64 nM T40332 CGR40J 10697956 Ki = 12 nM T40332 CC2G9E 10698640 Ki = 14000 nM T40332 C8BX1N 10710010 IC50 = 25000 nM T40332 C2SK5B 10718228 Ki = 690 nM T40332 CH1B5D 10727846 Ki = 130 nM T40332 C2UGD0 10728016 Ki = 34.67 nM T40332 CY0B3X 10729570 Ki = 5.74 nM T40332 CB2ZE0 10732420 Ki = 204.17 nM T40332 CNK38E 10733818 Ki = 17.78 nM T40332 CMBL13 10738994 Ki = 910 nM T40332 C58TAI 10739339 Ki = 0.18 nM T40332 CWZ92Y 10741446 Ki = 0.11 nM T40332 CL7RC5 10742017 IC50 = 1440 nM T40332 CV6D9X 10744508 Ki = 0.9 nM T40332 C3MXP5 10744523 Ki = 16 nM T40332 CZC57E 10744893 Ki = 22 nM T40332 C5VGC3 10744962 Ki = 3.4 nM T40332 C3L7VF 10745054 Ki = 21 nM T40332 C7AEI6 10745144 IC50 > 300000 nM T40332 CZAT51 10747107 Ki = 18 nM T40332 CZP63T 10756289 IC50 > 75000 nM T40332 CB7V0K 10763054 Ki = 14 nM T40332 CL20BQ 10765017 Ki = 0.09 nM T40332 CLU87Q 10765018 Ki = 0.078 nM T40332 CR6S4Z 10767409 Ki = 13.9 nM T40332 CB50RU 10768396 Ki = 0.85 nM T40332 C0EC3Z 10769317 Ki = 8.9 nM T40332 CE38KS 10769657 Ki = 4.1 nM T40332 CZG97S 10783016 IC50 = 300 nM T40332 CEMV61 10786746 Ki = 0.05 nM T40332 CWM1X4 10788924 Ki = 0.21 nM T40332 CV0O8I 10789380 Ki = 0.25 nM T40332 CS9F4X 10789763 Ki = 5.8 nM T40332 C97TFC 10791626 Ki = 230 nM T40332 C0WZ5S 10792102 Ki = 15 nM T40332 CD4P6H 10793294 Ki = 8.4 nM T40332 C1NK2I 10793641 Ki = 0.35 nM T40332 CT56CL 10793708 Ki = 1.7 nM T40332 C7K4RS 10794780 Ki = 100 nM T40332 CIC52D 10799209 Ki = 10.7 nM T40332 C20LYK 10799960 Ki = 446.68 nM T40332 CH0TA1 10805857 IC50 = 3000 nM T40332 CFHQ20 10813515 Ki = 29.1 nM T40332 C0H9BP 10815491 Ki = 0.058 nM T40332 C3L1DQ 10815914 Ki = 0.38 nM T40332 CL0E8T 10816188 Ki = 7.5 nM T40332 C28DOK 10816650 IC50 > 300000 nM T40332 CGP01V 10817508 IC50 > 300000 nM T40332 CG9B1J 10819798 Ki = 1300 nM T40332 C04IOW 10827508 Ki = 43.65 nM T40332 CDN04R 10831749 Ki = 0.033 nM T40332 CJ9FT6 10832773 Ki = 0.052 nM T40332 CE9NM4 10835541 Ki = 0.083 nM T40332 CIHY04 10837647 Ki = 490 nM T40332 CGX75W 10839361 Ki = 100 nM T40332 CSK04U 10839694 Ki = 21.2 nM T40332 CP6S9N 10854087 IC50 = 200 nM T40332 C07UEM 10889772 Ki = 707.95 nM T40332 C9Q2XI 11230895 IC50 = 1900 nM T40332 C7CHR5 11236753 IC50 = 17000 nM T40332 CS0CP2 11247668 Ki = 11700 nM T40332 C92PMV 11253808 IC50 = 9900 nM T40332 CKPO36 11272981 IC50 = 0.9 nM T40332 C2M7UP 11343089 IC50 > 30000 nM T40332 C4VX3G 11534280 IC50 = 0.5 nM T40332 CLAK97 11540629 IC50 = 100000 nM T40332 CT4FV1 11563929 Ki = 5300 nM T40332 CD7JU2 11590336 IC50 = 6700 nM T40332 C7FV6O 11592854 Ki = 340 nM T40332 CV82NQ 11619625 IC50 = 44 nM T40332 C93USP 11626693 IC50 > 10000 nM T40332 CWQ25N 11741764 Ki = 2 nM T40332 CHS6B5 11742000 Ki = 2600 nM T40332 C6FBJ4 11742006 Ki = 17 nM T40332 CTFS51 11742114 Ki = 4.5 nM T40332 C6B2TV 11743404 Ki = 100 nM T40332 CB95LW 11754431 Ki = 6.1 nM T40332 CS1TC0 11754640 Ki = 0.08 nM T40332 CD5W1A 11755516 Ki = 70 nM T40332 C5EQ9D 11756768 Ki = 9.1 nM T40332 CD7E0H 11757806 Ki = 32 nM T40332 C34FJZ 11757887 Ki = 52 nM T40332 CSM9F4 11758548 Ki = 0.34 nM T40332 C53SEA 11760115 IC50 = 14000 nM T40332 CJ6IG2 11765406 Ki = 0.6 nM T40332 CFG62D 11777027 Ki = 56.23 nM T40332 CJ0E8V 11779851 IC50 = 610 nM T40332 CO6A8F 11795366 Ki = 620 nM T40332 CN7LE6 11796530 Ki = 36 nM T40332 C3BN8Q 11797855 Ki = 33 nM T40332 CW5KF3 11798332 Ki = 830 nM T40332 C7QM3S 11799612 Ki = 290 nM T40332 CYRC95 11800689 IC50 > 300000 nM T40332 CWK1G8 11801735 Ki = 0.35 nM T40332 C7L9FS 11802328 Ki = 150 nM T40332 CCNX57 11983863 IC50 = 36000 nM T40332 C4IYM7 12134435 IC50 = 62 nM T40332 C3TIQ7 12248312 Ki = 52 nM T40332 C4O9HJ 12290092 Ki = 7413.1 nM T40332 CU0RL3 12689300 IC50 = 4800 nM T40332 CN6Z8X 12689316 IC50 = 400 nM T40332 CI8BH7 12689319 IC50 = 50 nM T40332 CKQ0W6 12689323 IC50 = 20 nM T40332 C7DV9I 12689324 IC50 = 5700 nM T40332 CY0RD7 12689332 IC50 = 19000 nM T40332 C0OIN2 12735875 Ki = 64565.42 nM T40332 C0S1VX 12942058 IC50 = 1390000 nM T40332 C4O5EV 13129200 IC50 = 19000 nM T40332 C32VSL 13221326 Ki = 30902.95 nM T40332 C19FEY 13629121 IC50 = 2000 nM T40332 C41KQG 13629122 IC50 > 40000 nM T40332 CY0U2X 13629126 IC50 = 4000 nM T40332 C4LKW6 13787283 Ki = 933.25 nM T40332 CVJU63 13827088 Ki = 17.78 nM T40332 C73UJB 13827090 Ki = 4.898 nM T40332 C64HRM 13827091 Ki = 0.06761 nM T40332 C4UOW2 13827093 Ki = 0.1905 nM T40332 C8PBE1 13827094 Ki = 5.754 nM T40332 CG6L2Y 13849881 Ki = 75.5 nM T40332 CU6H5B 13849894 Ki = 144.54 nM T40332 C9HVJ5 13853503 Ki = 38.02 nM T40332 C7XH2D 13853505 Ki = 43 nM T40332 CUC1S9 13853506 Ki = 3600 nM T40332 CIN97K 13853507 Ki = 31622.78 nM T40332 C56YEI 13853508 Ki = 954.99 nM T40332 CYIJ53 13853509 Ki = 588.84 nM T40332 CBK13D 13853511 Ki = 22.91 nM T40332 CL28MT 13853512 Ki = 1995.26 nM T40332 CY8ZP3 13853515 Ki = 181.97 nM T40332 CSE35Q 13853516 Ki = 776.25 nM T40332 C8BC3R 13853517 Ki = 407.38 nM T40332 CM1F9R 13853519 Ki = 4.169 nM T40332 C1JYQ0 13853520 Ki = 0.9333 nM T40332 CKD31E 13853528 Ki = 5.888 nM T40332 CE17QS 13853530 Ki = 707.95 nM T40332 CSU9J2 13853531 Ki = 6.607 nM T40332 CHG37U 13853534 Ki = 147.91 nM T40332 CQK4T2 13853537 Ki = 20.89 nM T40332 CJO19A 13853538 Ki = 177.83 nM T40332 CG85UW 13853539 Ki = 239.88 nM T40332 C3YUS1 13853541 Ki = 37.15 nM T40332 C3KO7X 13853551 Ki = 18620.87 nM T40332 C50ERO 13853552 Ki = 66.07 nM T40332 CZ5R9T 13853553 Ki = 37.15 nM T40332 CV57RA 13853554 Ki = 169.82 nM T40332 CF2J8E 13853555 Ki = 46.77 nM T40332 CQ7SY6 13853556 Ki = 27.54 nM T40332 COV0G6 13853560 Ki = 12.02 nM T40332 C34BNK 13880838 IC50 = 40000 nM T40332 CXYN02 14010380 IC50 = 620 nM T40332 CKF19U 14010382 IC50 = 6200 nM T40332 C4P0AK 14010383 IC50 = 250 nM T40332 CZ16DP 14010384 IC50 = 1400 nM T40332 C6MY3O 14010385 IC50 = 19000 nM T40332 CAH1W7 14010386 IC50 = 6000 nM T40332 CUH75S 14010387 IC50 = 1000 nM T40332 C24WHI 14010388 IC50 = 850 nM T40332 C4Z5NT 14010389 IC50 = 800 nM T40332 CK5T2I 14010390 IC50 = 320 nM T40332 CGA68E 14010391 IC50 = 1500 nM T40332 C6CKZ7 14010392 IC50 = 350 nM T40332 C1C9FM 14010393 IC50 = 800 nM T40332 C15ACF 14010394 IC50 = 2200 nM T40332 C3QB5A 14010395 IC50 = 170 nM T40332 C7KV4T 14010396 IC50 = 12000 nM T40332 CFJ0O9 14010397 IC50 = 670 nM T40332 CF52UJ 14010398 IC50 = 150 nM T40332 C5ZVC9 14010399 IC50 = 900 nM T40332 CO6QD1 14010400 IC50 = 27 nM T40332 CZBO42 14010401 IC50 = 1500 nM T40332 C3S2KZ 14010402 IC50 = 55 nM T40332 C0Z8EN 14010403 IC50 = 84 nM T40332 C1VWO8 14010404 IC50 = 10000 nM T40332 CMS3V7 14010405 IC50 = 8000 nM T40332 CUT3S2 14010407 IC50 = 140 nM T40332 CPQ5N2 14010408 IC50 = 360 nM T40332 CT3HG6 14010410 IC50 = 460 nM T40332 CR27UM 14010411 IC50 = 1500 nM T40332 CY82DH 14010414 IC50 = 130 nM T40332 CFON34 14010415 IC50 = 450 nM T40332 CQ18TM 14010416 IC50 = 83 nM T40332 C59EVI 14010418 IC50 = 1800 nM T40332 CB8XQ1 14052374 IC50 = 10000 nM T40332 C87RMA 14089169 IC50 = 110 nM T40332 CS8BF9 14089170 IC50 = 100 nM T40332 CAF82P 14089172 IC50 = 300 nM T40332 CHZ75Q 14089173 IC50 = 210 nM T40332 C9KM6B 14089174 IC50 = 160 nM T40332 C5RWV4 14089175 IC50 = 1900 nM T40332 CUT74L 14089176 IC50 = 200 nM T40332 CO2C7I 14089177 IC50 = 5400 nM T40332 CAZM38 14089178 IC50 = 27 nM T40332 C2U7LD 14089179 IC50 = 100 nM T40332 C38RIF 14089180 IC50 = 8400 nM T40332 CGO1Q5 14089181 IC50 = 600 nM T40332 C68VEU 14089182 IC50 = 130 nM T40332 C5QE8G 14089184 IC50 = 80000 nM T40332 CQ3YT2 14089185 IC50 = 72 nM T40332 C7LBW3 14089186 IC50 = 9000 nM T40332 CXI47P 14089187 IC50 = 1000 nM T40332 C0A8HV 14207561 Ki = 0.4677 nM T40332 CUGW80 14207563 Ki = 0.3981 nM T40332 C0EIF7 14379792 IC50 > 40000 nM T40332 C3NK7L 14379796 IC50 = 60 nM T40332 CC9A3G 14379800 IC50 = 3000 nM T40332 CJFB97 14379803 IC50 = 30000 nM T40332 CCM8E6 14379806 IC50 = 2000 nM T40332 CGEU96 14488442 IC50 = 4000 nM T40332 CVI43O 14488443 IC50 > 40000 nM T40332 C3TG7L 14493342 Ki = 102 nM T40332 CC10KI 14513750 Ki = 3400 nM T40332 CV7A3W 14539951 Ki = 4300 nM T40332 C9G4DC 14542117 Ki = 512.86 nM T40332 C0AUT7 14760206 IC50 = 200 nM T40332 C1MR8P 14760208 IC50 = 500 nM T40332 CYC20A 14760210 IC50 = 100 nM T40332 CD1OC8 14760212 IC50 = 100 nM T40332 CG7J0I 14760231 IC50 = 800 nM T40332 CU3H5M 14760233 IC50 = 70 nM T40332 C2LS8V 14760235 IC50 = 100 nM T40332 C4SF7Z 14760237 IC50 = 200 nM T40332 CY76IR 14760239 IC50 = 100 nM T40332 CCNE24 14760241 IC50 = 400 nM T40332 C2A3HQ 14760243 IC50 = 40 nM T40332 C2FQ3E 14760247 IC50 = 400 nM T40332 C0P6KI 14760249 IC50 = 400 nM T40332 CY4HQ3 14760260 IC50 = 5000 nM T40332 C46LBG 14760262 IC50 = 100 nM T40332 CEZ3A4 14760264 IC50 = 800 nM T40332 CWK7S9 14760266 IC50 = 2000 nM T40332 CARP67 14760298 IC50 = 1000 nM T40332 CJ2HR7 14760300 IC50 = 200 nM T40332 CYJ3K2 14760306 IC50 > 50000 nM T40332 C5UP4K 14760308 IC50 > 50000 nM T40332 C5FVQ2 14760310 IC50 = 5000 nM T40332 CDW0S3 14760319 IC50 = 400 nM T40332 C0FA5S 14760334 IC50 = 430 nM T40332 CR6ZV5 14760337 IC50 = 2400 nM T40332 CL78BW 14760339 IC50 = 2230 nM T40332 CK3YT2 14760341 IC50 = 2330 nM T40332 C96RUH 14760343 IC50 = 1620 nM T40332 CBG83A 14760345 IC50 = 1820 nM T40332 CZO79G 14760347 IC50 = 630 nM T40332 C13ABK 14760351 IC50 = 940 nM T40332 C72HTW 14760353 IC50 = 910 nM T40332 CH7ZT3 14760355 Ki = 220 nM T40332 CZGD18 14760368 IC50 = 130 nM T40332 C4UM1D 14760370 IC50 = 1000 nM T40332 CBQ0Z1 14760376 IC50 = 1800 nM T40332 CAXH03 14760380 IC50 = 57800 nM T40332 C5F3MZ 14861885 IC50 = 3.7 ug.mL-1 T40332 COE37G 15035342 Ki = 290000 nM T40332 C3NM4I 15035343 Ki = 16500 nM T40332 CCWF97 15198479 IC50 = 6700 nM T40332 CQ0RU9 15200486 Ki = 28 nM T40332 C4Y8KR 15230194 Ki = 15 nM T40332 CG1NR2 15230196 Ki = 81 nM T40332 C1UH7S 15338151 Ki = 0.08 nM T40332 CT48FA 15407997 IC50 > 300000 nM T40332 CLGV32 15547238 IC50 > 10000 nM T40332 CN05KP 15573427 IC50 > 40000 nM T40332 CKR59B 15589985 IC50 > 10000000 nM T40332 CU1TD9 15726831 IC50 > 40000 nM T40332 C32CWO 15726832 IC50 > 40000 nM T40332 C6L5MJ 15726833 IC50 > 40000 nM T40332 CJQ6V7 15726835 IC50 > 40000 nM T40332 CAYS45 15726841 IC50 = 40000 nM T40332 C26CQI 15726842 IC50 > 40000 nM T40332 CVPL97 15726843 IC50 = 28000 nM T40332 CH7KS8 15726844 IC50 > 40000 nM T40332 CED5G0 15726845 IC50 = 1000 nM T40332 C0UYJ4 15726846 IC50 > 10000 nM T40332 C3VE9S 15726847 IC50 = 5000 nM T40332 CZG4F5 15726851 IC50 = 10000 nM T40332 CA4R1Z 15726852 IC50 = 36000 nM T40332 CSC4K3 15726857 IC50 = 300 nM T40332 C0YBI9 15726858 IC50 = 6000 nM T40332 CT6W4L 15726859 IC50 = 10000 nM T40332 C6TYB5 15726860 IC50 > 40000 nM T40332 CKJU90 15726861 IC50 = 10000 nM T40332 C8BD3T 15726862 IC50 = 6000 nM T40332 C3MIX7 15726863 IC50 = 1000 nM T40332 CRO39F 15726866 IC50 = 24000 nM T40332 C2EGD3 15726867 IC50 = 40000 nM T40332 CX1LM4 15726868 IC50 = 2000 nM T40332 CQY3B4 15726869 IC50 = 20000 nM T40332 CG9X0Z 15726871 IC50 > 40000 nM T40332 CO5MC2 15726874 IC50 > 40000 nM T40332 CYTK20 15726875 IC50 > 40000 nM T40332 CF49XE 15726876 IC50 = 4000 nM T40332 CDP91C 15743471 IC50 = 8700 nM T40332 CJ41CN 15743472 IC50 = 4200 nM T40332 C8YR1W 15743473 IC50 = 5900 nM T40332 CWU90T 15743474 Ki = 150 nM T40332 CZ6WU7 15838071 Ki = 5.47 nM T40332 COG9C4 15885812 Ki = 33.88 nM T40332 C5XRE1 15886812 Ki = 0.49 nM T40332 CPZU83 15928334 IC50 = 830 nM T40332 C72JFE 15955759 Ki = 251.19 nM T40332 C9M1EK 16104379 IC50 > 10000 nM T40332 CRQV57 16104920 IC50 = 49 nM T40332 C9OSM6 16144480 Ki = 120 nM T40332 CDR0G7 16145606 Ki = 100 nM T40332 CY20PW 16147332 Ki = 130 nM T40332 CF5Y3L 16147570 Ki = 8300 nM T40332 C7S6IT 16148231 Ki = 200 nM T40332 C0WX5C 16163030 Ki = 1300 nM T40332 CSXO69 16680454 IC50 = 352 nM T40332 C6AR3Q 16757019 IC50 = 316 nM T40332 CL8M0W 17755151 IC50 = 0.21 nM T40332 C0JBH9 18395047 IC50 > 50000 nM T40332 C2XTI9 18395048 IC50 > 50000 nM T40332 C63HAE 18572952 IC50 = 18000 nM T40332 CV86RX 18603196 Ki = 41 nM T40332 CRW81C 18607241 Ki = 1258.93 nM T40332 C50UPT 18607265 Ki = 870.96 nM T40332 C8MD2B 18607267 Ki = 213.8 nM T40332 CJ03UC 18633082 IC50 = 200 nM T40332 CZP68C 18633083 IC50 = 2000 nM T40332 CN85LE 18633087 IC50 = 200 nM T40332 CIYD09 18633089 IC50 = 10000 nM T40332 C3YRI4 18633090 IC50 = 150 nM T40332 CI9A1H 18643724 IC50 = 1330 nM T40332 CXF13I 18801003 IC50 > 5000 nM T40332 C7U4PY 19030591 Ki = 5.754 nM T40332 C7DPB4 19389555 Ki = 91.2 nM T40332 C6K1QN 19845653 Ki = 0.07079 nM T40332 CD4L1N 19845806 Ki = 0.2291 nM T40332 C5UDO2 20139259 Ki = 10 nM T40332 CRQ9Y6 20139310 Ki = 10 nM T40332 C1DRH4 20208290 Ki = 2818.38 nM T40332 CJ7TH3 20208319 Ki = 10.96 nM T40332 CP6UN4 20208423 Ki = 1348.96 nM T40332 C2M8AW 20208435 Ki = 16.98 nM T40332 CX59VG 20208455 Ki = 1202.26 nM T40332 CUG1K3 20208523 Ki = 645.65 nM T40332 CXHA26 21033975 Ki = 63 nM T40332 CGB92N 21731457 Ki = 109.65 nM T40332 C20KJO 21823504 Ki = 219 nM T40332 CD7CI2 22124919 Ki = 416.87 nM T40332 CS2X9Z 22152164 Ki = 77.62 nM T40332 CT58FO 22392859 IC50 > 10000000 nM T40332 CLU18Y 22881851 Ki = 28 nM T40332 CA2S6B 23151285 Ki = 1000 nM T40332 C5VSO2 23276168 Ki = 288403.15 nM T40332 CB63KH 23276169 Ki = 338844.16 nM T40332 C7QD8E 23276182 Ki = 346736.85 nM T40332 CR8LI0 23437569 Ki = 218.78 nM T40332 CUH0K4 23444468 Ki = 109.65 nM T40332 CS13PY 23657291 IC50 = 23 nM T40332 CTBO93 23664980 IC50 = 44 nM T40332 C9XJP3 23711928 IC50 = 3000 nM T40332 CBD3H5 23728722 Ki = 15 nM T40332 CN0VA7 24822701 IC50 > 50000 nM T40332 CW9D6P 24823445 Ki = 23.8 nM T40332 C2WI4S 24823446 Ki = 0.71 nM T40332 CU2O6S 24823609 Ki = 63.5 nM T40332 CT78NC 24854122 IC50 = 59100 nM T40332 CCD95H 24854123 IC50 = 71300 nM T40332 C9J2QD 24974797 Ki = 4570.88 nM T40332 C9TKJ6 24999408 IC50 = 390 nM T40332 CVI40X 24999724 IC50 = 93 nM T40332 C8G7FX 24999726 IC50 = 64 nM T40332 C8SNG4 25000364 IC50 = 110 nM T40332 C1UH4R 25000365 IC50 = 6000 nM T40332 C0GJ4N 25000368 IC50 = 8100 nM T40332 CUC8N5 25141405 IC50 = 3100 nM T40332 CX05JT 25205745 IC50 = 19 nM T40332 C3GS6F 33009902 IC50 > 10000 nM T40332 C2DEG7 42642360 IC50 < 0.3 nM T40332 CL0M7R 44143089 IC50 = 85113.8 nM T40332 CPT2B6 44266363 IC50 = 6100 nM T40332 CH9O7C 44266372 IC50 = 130 nM T40332 CX89JI 44266374 IC50 = 43000 nM T40332 C54FSU 44266698 IC50 = 110 nM T40332 CDS31V 44267097 Ki = 0.21 nM T40332 C9X4QL 44267147 Ki = 0.96 nM T40332 CUW9I2 44267176 Ki = 1.6 nM T40332 CR8O5J 44267221 Ki = 27 nM T40332 C97EWG 44267427 Ki = 1.2 nM T40332 C8EQ9C 44267442 Ki = 0.24 nM T40332 C43NJL 44267444 Ki = 0.17 nM T40332 C75REN 44267447 Ki = 0.47 nM T40332 C8QVJ6 44267462 Ki = 0.34 nM T40332 C3ZU7Q 44267468 Ki = 0.049 nM T40332 CMSI17 44272976 Ki = 19000 nM T40332 CN2X4F 44272977 Ki = 27000 nM T40332 CYV1W8 44273732 Ki = 270000 nM T40332 CFA21P 44273766 Ki = 190000 nM T40332 CNV18Y 44274239 Ki > 300000 nM T40332 CD84XF 44279475 IC50 > 50000 nM T40332 C0RQ3V 44279712 IC50 > 30000 nM T40332 CFJ2Z1 44279771 IC50 > 30000 nM T40332 C3IBQ0 44279792 IC50 > 50000 nM T40332 CQ57HR 44279823 IC50 > 50000 nM T40332 C5YF0J 44279873 IC50 > 50000 nM T40332 CROD68 44279951 IC50 > 50000 nM T40332 C6ZXK0 44280152 IC50 > 50000 nM T40332 CVZ54E 44280172 IC50 > 50000 nM T40332 C8D6VK 44282051 IC50 > 75000 nM T40332 CN7SA3 44287645 IC50 = 3900 nM T40332 C1GU7P 44287670 IC50 = 13000 nM T40332 C7QSK8 44287706 IC50 = 11000 nM T40332 CB8L9Q 44287782 IC50 = 8000 nM T40332 CR6QO0 44287881 IC50 = 6000 nM T40332 C5NR3Q 44287906 IC50 = 12000 nM T40332 CT98XO 44287910 IC50 = 5900 nM T40332 C3F9LM 44287918 IC50 = 21000 nM T40332 C42JSV 44287920 IC50 = 13000 nM T40332 C6AZV8 44287930 IC50 = 2500 nM T40332 C4KWZ8 44287967 IC50 = 6400 nM T40332 CR9YA8 44288052 Ki = 7500 nM T40332 C6KJ4D 44288060 IC50 = 6100 nM T40332 CMO3X2 44288136 IC50 = 4200 nM T40332 CDT93F 44288297 IC50 = 1300 nM T40332 CN04DK 44288315 Ki = 430 nM T40332 COP5H9 44288316 Ki = 1900 nM T40332 CJH40B 44295808 Ki = 17500 nM T40332 CSC8X9 44295983 Ki = 32 nM T40332 C6POB4 44296152 Ki = 0.7 nM T40332 CJC83Z 44296212 Ki = 13.6 nM T40332 C49ZTQ 44296213 Ki = 15 nM T40332 CNI4K8 44296327 Ki = 80 nM T40332 CSEG82 44296328 Ki = 2000 nM T40332 CA9R6Z 44296341 Ki = 60 nM T40332 CYO86L 44296343 Ki = 0.6 nM T40332 CWL62G 44296396 Ki = 3 nM T40332 CI0EM5 44296406 Ki = 32 nM T40332 C12XSO 44296649 Ki = 246 nM T40332 CN1I6M 44296666 Ki = 17.5 nM T40332 CJ37GI 44298562 Ki = 6.1 nM T40332 COB9F7 44298605 Ki = 0.41 nM T40332 C14GUD 44298619 Ki = 0.87 nM T40332 CKEA52 44298620 Ki = 1.8 nM T40332 CQAG41 44298819 Ki = 3.3 nM T40332 C6URN0 44298842 Ki = 43 nM T40332 CP50DO 44298855 Ki = 1.1 nM T40332 C94FOM 44298860 Ki = 1.7 nM T40332 CAK97H 44298884 Ki = 1.2 nM T40332 CMWF68 44298885 Ki = 5.4 nM T40332 CPN6G7 44298886 Ki = 60 nM T40332 CU8Z3V 44298888 Ki = 1.8 nM T40332 C0K2QM 44298908 Ki = 1.6 nM T40332 CGB10R 44298921 Ki = 4.2 nM T40332 CQ8B2N 44298922 Ki = 2 nM T40332 CT3DQ8 44298927 Ki = 55 nM T40332 C1FM8K 44298929 Ki = 2.7 nM T40332 C8U2WZ 44298945 Ki = 2.3 nM T40332 CO6MA7 44298966 Ki = 8 nM T40332 CUCW51 44298967 Ki = 10 nM T40332 CQGX12 44298970 Ki = 3.2 nM T40332 C62MQB 44298980 Ki = 2.5 nM T40332 C80XBS 44298984 Ki = 5.2 nM T40332 C4KTI6 44298990 Ki = 15 nM T40332 CB39FC 44298992 Ki = 11 nM T40332 C47SOH 44298993 Ki = 0.43 nM T40332 C2BYH3 44299001 Ki = 1.7 nM T40332 CGBR39 44299062 Ki = 190 nM T40332 CM54OT 44299064 Ki = 1.2 nM T40332 CIOE85 44299235 Ki = 12 nM T40332 CPO75N 44299253 Ki = 1.3 nM T40332 C8IL5V 44299896 IC50 = 36 nM T40332 C3A1YN 44299897 IC50 = 38 nM T40332 C5G6LV 44299976 IC50 = 15 nM T40332 CM24TU 44299977 IC50 = 24 nM T40332 C9G5QX 44299990 IC50 = 24 nM T40332 CZMJ96 44300040 IC50 = 18 nM T40332 CEW05I 44300059 IC50 = 59 nM T40332 CS28OU 44300070 IC50 = 0.1 nM T40332 CGE9W3 44300076 IC50 = 84 nM T40332 C69WJZ 44300092 IC50 = 30 nM T40332 C5FDJ3 44300093 IC50 = 36 nM T40332 C20JDX 44300119 IC50 = 40 nM T40332 CUKL54 44300133 IC50 = 43 nM T40332 C6V4XE 44300174 IC50 = 46 nM T40332 C6EU7G 44300177 IC50 = 38 nM T40332 C5G9KX 44300179 IC50 = 70 nM T40332 CV7F8N 44300180 IC50 = 34 nM T40332 C5RSX9 44300181 IC50 = 26 nM T40332 C30HJX 44300217 IC50 = 20 nM T40332 C9M3NU 44300289 IC50 = 46 nM T40332 COX87D 44304039 IC50 = 50 nM T40332 C68UDG 44306172 Ki = 320000 nM T40332 C6ZO2A 44306517 Ki = 1800000 nM T40332 CO42PE 44306533 Ki = 1000000 nM T40332 CY0M9E 44306778 IC50 = 40000 nM T40332 C51ZLR 44308482 Ki = 18 nM T40332 CZK3U8 44308945 Ki = 1.6 nM T40332 CKA3B8 44308946 Ki = 0.35 nM T40332 CF61VA 44308955 Ki = 0.81 nM T40332 C2Z9QB 44309043 Ki = 4.1 nM T40332 CQ80NX 44309049 Ki = 130 nM T40332 CSFN37 44309050 Ki = 0.39 nM T40332 CR4XO9 44309051 Ki = 1.1 nM T40332 CX80SC 44309073 Ki = 3.4 nM T40332 C18AZL 44309216 IC50 = 3.5 nM T40332 C8E0AZ 44309228 Ki = 15 nM T40332 CBEA34 44309326 Ki = 0.65 nM T40332 C60GWS 44312415 Ki > 100000 nM T40332 CDGX29 44312419 Ki = 3200 nM T40332 C75DJS 44312600 Ki > 100000 nM T40332 C9LT2C 44312642 IC50 = 20000 nM T40332 C61MLD 44312660 IC50 = 12000 nM T40332 CKHV96 44312681 IC50 = 3000 nM T40332 CK08ZX 44312691 IC50 = 9000 nM T40332 CIWU48 44312692 IC50 > 20000 nM T40332 CE06PC 44312711 IC50 = 800 nM T40332 C6HV5N 44312736 IC50 = 700 nM T40332 C6D8ZP 44312737 IC50 = 3000 nM T40332 CCBJ53 44312740 IC50 = 1000 nM T40332 C25UOL 44312741 IC50 = 2000 nM T40332 CB3A9W 44312771 IC50 > 20000 nM T40332 C1P7ED 44312773 IC50 = 3000 nM T40332 C4HJZ9 44312840 Ki = 4000 nM T40332 COYR46 44312861 Ki = 12000 nM T40332 C28YCZ 44312862 Ki = 400 nM T40332 C5GMQ9 44312896 Ki = 1500 nM T40332 C40UFA 44312925 IC50 > 20000 nM T40332 C37LOU 44312957 IC50 = 20000 nM T40332 CJQI56 44312958 IC50 = 4000 nM T40332 CQO41D 44312969 IC50 = 4000 nM T40332 C08ZBI 44312990 IC50 = 700 nM T40332 CU3E4B 44312991 IC50 = 100 nM T40332 CQJ5F9 44312992 IC50 = 4000 nM T40332 C2YA6T 44312993 Ki = 10000 nM T40332 CRZX02 44313005 IC50 = 2000 nM T40332 CCM2R1 44313033 IC50 = 2000 nM T40332 CT69SA 44313040 IC50 = 4000 nM T40332 CZ24YH 44313056 IC50 = 600 nM T40332 CG0Y5Z 44313064 IC50 = 700 nM T40332 CO01JG 44313077 IC50 = 300 nM T40332 CN1E5H 44313087 IC50 = 5000 nM T40332 C9LT4Z 44313114 IC50 = 4000 nM T40332 CJ5UI3 44313122 Ki = 50000 nM T40332 CC7A1J 44313131 Ki = 53000 nM T40332 C4UNO3 44313149 IC50 = 20000 nM T40332 CZ07MG 44313176 IC50 = 5000 nM T40332 C8VCL3 44313177 IC50 = 5000 nM T40332 CD2FS4 44313342 Ki = 22000 nM T40332 CQK72I 44313345 Ki = 1500 nM T40332 C2XHU4 44313650 Ki = 14000 nM T40332 CH18RW 44313833 Ki = 1300 nM T40332 CKN8C1 44316486 IC50 > 10000 nM T40332 C60AVB 44317117 Ki >= 30000 nM T40332 C4T0AC 44317137 Ki >= 88000 nM T40332 CCVZ83 44317149 Ki >= 72000 nM T40332 C83FQT 44317256 Ki = 43000 nM T40332 CP03CV 44317262 Ki >= 45000 nM T40332 CJ2B9M 44317267 Ki = 29000 nM T40332 C3T6YK 44317274 Ki >= 78000 nM T40332 C5AR9V 44317284 Ki >= 30000 nM T40332 CKP03R 44317285 Ki >= 104000 nM T40332 CAK4P6 44318572 IC50 = 40000 nM T40332 C84AGV 44319331 IC50 = 1400 nM T40332 C0CWH7 44319367 IC50 = 76000 nM T40332 C5Z8KW 44319375 IC50 = 43000 nM T40332 C1RL4T 44319383 IC50 = 45000 nM T40332 CO5CA2 44319384 IC50 = 94000 nM T40332 C3VH1X 44319419 IC50 = 13000 nM T40332 CAC49M 44319423 IC50 = 11000 nM T40332 C3GO1N 44319641 IC50 = 1600 nM T40332 CMPE25 44319642 IC50 = 18000 nM T40332 CM5HO4 44321916 Ki = 0.008 nM T40332 C4MJ8H 44322029 Ki = 0.01 nM T40332 CB3Q9U 44322389 Ki = 0.007 nM T40332 CA6KV2 44331082 Ki = 14.5 nM T40332 CBFS14 44331115 Ki = 2 nM T40332 CJ19RM 44337844 Ki = 0.64 nM T40332 C0TE6U 44337930 Ki = 0.64 nM T40332 CHT61Y 44338018 Ki = 8 nM T40332 C14UGI 44338019 Ki = 0.65 nM T40332 C0JY7C 44338029 Ki = 0.06 nM T40332 CWI7N9 44338415 IC50 = 5000 nM T40332 CN4C5X 44338416 IC50 = 5700 nM T40332 CZX39H 44338433 IC50 = 60 nM T40332 CXF5Z2 44338508 IC50 = 400 nM T40332 CBM7L9 44338509 IC50 = 3500 nM T40332 CU5H2I 44338658 IC50 = 900 nM T40332 CC0O3Q 44338659 IC50 = 220 nM T40332 C09SZK 44338660 IC50 = 450 nM T40332 C32EVN 44338707 IC50 = 1600 nM T40332 C06BSK 44338737 IC50 = 1400 nM T40332 CGM1H7 44338738 IC50 = 1800 nM T40332 C4XDT1 44338807 IC50 = 340 nM T40332 C6K3YE 44338808 IC50 = 900 nM T40332 CUFS02 44338809 IC50 = 560 nM T40332 CZD3L7 44338820 IC50 = 400 nM T40332 CMK10R 44338821 IC50 = 20 nM T40332 CP56NM 44338822 IC50 = 7300 nM T40332 CKP0B1 44339163 Ki = 34 nM T40332 CA1D5G 44339167 Ki = 1.6 nM T40332 C2FZD6 44339168 Ki = 51.6 nM T40332 C4HY8G 44339183 Ki > 100 nM T40332 C5R4DQ 44339184 Ki = 10 nM T40332 CPQ47M 44339196 Ki = 13.6 nM T40332 CEX5G4 44339197 Ki = 42 nM T40332 CG87DW 44339210 Ki > 1000 nM T40332 CWM73S 44339220 Ki > 100 nM T40332 C5JZA6 44340361 Ki = 1 nM T40332 C75HMC 44340504 Ki = 18 nM T40332 COE37X 44340528 Ki = 1 nM T40332 CE71WL 44340543 Ki = 5 nM T40332 CZE75W 44340561 Ki = 1 nM T40332 C54RWE 44340595 Ki = 100 nM T40332 CR4OT3 44341284 Ki = 1.1 nM T40332 C8J1KC 44341355 Ki = 2.2 nM T40332 C0XZO4 44341377 Ki = 0.2 nM T40332 CR8KP4 44341378 Ki = 5.2 nM T40332 CLQ2W9 44341406 Ki = 0.03 nM T40332 C2AT7J 44342409 Ki = 17 nM T40332 CUR86C 44342423 Ki = 20 nM T40332 CF60PZ 44342469 Ki = 1380 nM T40332 C8DV6S 44342778 IC50 = 9000000 nM T40332 CH3CE9 44342794 IC50 = 5400000 nM T40332 CWLT78 44342805 IC50 > 10000000 nM T40332 CWQ13J 44342806 IC50 > 10000000 nM T40332 CB7HO1 44342811 Ki = 4 nM T40332 C01YDQ 44342827 IC50 = 8900000 nM T40332 CX2HK7 44342836 IC50 > 10000000 nM T40332 C64PAR 44342837 IC50 = 2600000 nM T40332 CH39PO 44342847 IC50 > 10000000 nM T40332 CLI0B3 44342857 IC50 = 8900000 nM T40332 CP7RQ6 44342869 IC50 > 10000000 nM T40332 CJU1K9 44342887 IC50 = 2560000 nM T40332 CMR6I2 44342888 IC50 = 6410000 nM T40332 CXO27U 44342890 IC50 > 10000000 nM T40332 C95EXJ 44342891 IC50 = 210000 nM T40332 C9BKY1 44342937 IC50 = 5350000 nM T40332 CX6M5P 44342953 IC50 = 6000000 nM T40332 CN1VD4 44342954 IC50 = 1180000 nM T40332 CA93TW 44342991 IC50 = 490000 nM T40332 CBED26 44342992 IC50 > 10000000 nM T40332 CF0XD7 44343000 IC50 > 10000000 nM T40332 CTI5A0 44343012 IC50 = 2070000 nM T40332 C14ITM 44343019 IC50 = 13900000 nM T40332 CS8E1H 44343022 IC50 = 4270000 nM T40332 C9QD7A 44343029 IC50 = 6000000 nM T40332 COY26B 44343032 IC50 > 10000000 nM T40332 CKT05N 44343039 IC50 = 7100000 nM T40332 CNS1W4 44343061 IC50 = 6100000 nM T40332 C0JP1W 44343069 IC50 = 280000 nM T40332 C3KGY9 44343124 IC50 > 10000000 nM T40332 C4HFN2 44343139 IC50 = 3360000 nM T40332 CZT68I 44343164 IC50 = 390000 nM T40332 CJ6R9X 44343194 IC50 > 10000000 nM T40332 CQ7A9W 44343906 Ki > 100000 nM T40332 C9X0ZR 44343907 Ki > 100000 nM T40332 C6FY8O 44345532 IC50 = 12000 nM T40332 CPW75O 44348239 Ki = 250 nM T40332 C5U7YX 44348372 Ki = 500 nM T40332 CD8AL2 44351097 IC50 = 69 nM T40332 CHGE39 44351104 IC50 = 74 nM T40332 C2RMW4 44351162 IC50 = 88 nM T40332 C2Y7GN 44352045 Ki = 0.5 nM T40332 C68KSH 44352097 Ki = 1 nM T40332 C0D4CK 44353344 Ki = 1 nM T40332 C38RJF 44353357 Ki = 200 nM T40332 CQU69T 44353358 Ki = 7 nM T40332 COPM05 44353364 Ki = 66000 nM T40332 C20CYN 44353485 Ki < 0.1 nM T40332 CN85XQ 44354163 IC50 > 300000 nM T40332 CGL18R 44359861 Ki = 19 nM T40332 CLM3H4 44359870 Ki = 70 nM T40332 CL9GT7 44359932 Ki = 70 nM T40332 CD0PS5 44359934 Ki = 59 nM T40332 C80BKQ 44359984 Ki = 7 nM T40332 C9Z2IU 44359985 Ki = 2 nM T40332 C53AJT 44360051 Ki = 21 nM T40332 CY24NZ 44360093 Ki = 43 nM T40332 CJEC32 44360131 Ki = 44 nM T40332 CZ5JL3 44360132 Ki = 24 nM T40332 CIX34U 44360133 Ki = 39 nM T40332 C5NE7W 44360270 Ki = 29 nM T40332 CLO39R 44361701 Ki = 0.016 nM T40332 C1RS0F 44361716 Ki = 0.021 nM T40332 CO6VL0 44362002 Ki = 0.093 nM T40332 CHF49P 44362414 Ki = 120.23 nM T40332 CT04RY 44362423 Ki = 257.04 nM T40332 CAP5Y6 44362424 Ki = 102.33 nM T40332 C0W7TH 44362425 Ki = 14454.4 nM T40332 C93FWR 44362443 Ki = 0.0955 nM T40332 CKTI90 44362458 Ki = 1096.48 nM T40332 CGAN05 44362471 Ki = 12882.5 nM T40332 CHAQ14 44362472 Ki = 6918.31 nM T40332 C41XZU 44362486 Ki = 758.58 nM T40332 CSZ03H 44362546 Ki = 7585.78 nM T40332 CCHM90 44362570 Ki = 398.11 nM T40332 C2UZC3 44362571 Ki = 2570.4 nM T40332 C51UBY 44362573 Ki = 549.54 nM T40332 CLG37U 44362583 Ki = 363.08 nM T40332 C4FK2R 44362584 Ki = 70.79 nM T40332 C4XCT3 44362585 Ki = 467.74 nM T40332 C8O5YU 44362587 Ki = 104.71 nM T40332 CMK28R 44362631 Ki = 39.81 nM T40332 CT2X0F 44362640 Ki = 1548.82 nM T40332 CND9Z3 44362653 Ki = 1.585 nM T40332 C5XU6E 44362657 Ki = 181.97 nM T40332 CNEI94 44362661 Ki = 5100 nM T40332 C41HKG 44362664 Ki = 10 nM T40332 CH4YV7 44362667 Ki = 660.69 nM T40332 C7CR2Y 44362668 Ki = 741.31 nM T40332 C78ROB 44362669 Ki = 3388.44 nM T40332 C52GSX 44362683 Ki = 151.36 nM T40332 C7O9RC 44362688 Ki = 6456.54 nM T40332 C9U3FY 44362694 Ki = 97723.72 nM T40332 C2EIU0 44362697 Ki = 1122.02 nM T40332 C3Z6BO 44362707 Ki = 2137.96 nM T40332 CCDJ03 44362708 Ki = 109.65 nM T40332 CZ8BI0 44362721 Ki = 478.63 nM T40332 CO59RP 44362722 Ki = 338.84 nM T40332 C24FNJ 44362734 Ki = 169.82 nM T40332 CCD2N8 44362741 IC50 = 107 nM T40332 CLV72W 44362755 Ki = 1202.26 nM T40332 C4GRW1 44362756 Ki = 1445.44 nM T40332 CED8M4 44362761 Ki = 0.9333 nM T40332 C9YM0R 44362762 Ki = 72.44 nM T40332 C6N1FA 44362778 Ki = 1258.93 nM T40332 C8QFN6 44362779 Ki = 30.9 nM T40332 C0QG4Z 44362780 Ki = 537.03 nM T40332 CLI68E 44362789 Ki = 109.65 nM T40332 CNWF06 44362845 Ki = 8.128 nM T40332 CTAY98 44362846 Ki = 1.413 nM T40332 C06INC 44362848 Ki = 20.89 nM T40332 CY6QH7 44362849 Ki = 177.83 nM T40332 C6ZM5V 44362850 Ki = 114.82 nM T40332 C71WGV 44362853 Ki = 1230.27 nM T40332 CVH3L1 44362854 Ki = 1584.89 nM T40332 C2K7JM 44362855 Ki = 158489.32 nM T40332 C6P1AQ 44362869 Ki = 1698.24 nM T40332 CSEZ31 44362877 Ki = 446.68 nM T40332 C9FC7V 44362890 Ki = 1995.26 nM T40332 CKE47Z 44362891 Ki = 2137.96 nM T40332 CPL17T 44362892 Ki = 316.23 nM T40332 C67KRN 44362900 Ki = 724.44 nM T40332 CT0SE7 44362901 Ki = 239.88 nM T40332 CXZS62 44362903 Ki = 154.88 nM T40332 C3R8CM 44362909 Ki = 199.53 nM T40332 C6C8RO 44362910 Ki = 2.692 nM T40332 CK5AJ0 44362944 Ki = 28.18 nM T40332 CN43FB 44362945 Ki = 20.89 nM T40332 C2FRU6 44362954 Ki = 1000 nM T40332 CG48UP 44362959 Ki = 5495.41 nM T40332 C1ETU0 44362969 Ki = 39.81 nM T40332 CS3H1F 44362970 Ki = 7.762 nM T40332 CAO25V 44362980 IC50 = 365 nM T40332 CR8MD1 44362982 Ki = 72.44 nM T40332 CV4Z7R 44363005 Ki = 691.83 nM T40332 CPU7L1 44363006 Ki = 281.84 nM T40332 C72KXW 44363019 Ki = 21.38 nM T40332 CT7V2L 44363025 Ki = 54954.09 nM T40332 CUCE12 44363030 Ki = 21.38 nM T40332 C27SKX 44363034 Ki = 7943.28 nM T40332 CZK7I9 44363091 Ki = 65000 nM T40332 C7Q5UZ 44363092 Ki = 595000 nM T40332 CO6Z8K 44366639 Ki = 55 nM T40332 CFL1J0 44366665 Ki = 4 nM T40332 C27VSQ 44366666 Ki = 15.9 nM T40332 C35YGE 44367854 IC50 = 7800 nM T40332 C7FBC3 44367865 IC50 > 10000 nM T40332 CV4L8A 44367935 IC50 = 7.6 nM T40332 CD0IM7 44368008 IC50 = 8.9 nM T40332 C8E7CZ 44368051 IC50 = 130 nM T40332 CVM6S7 44368057 IC50 = 66 nM T40332 C9RLA3 44368068 IC50 > 10000 nM T40332 CR53IL 44368071 IC50 = 290 nM T40332 CU3F6L 44368072 IC50 = 230 nM T40332 C97NDU 44368076 IC50 > 10000 nM T40332 C4SFV3 44368077 IC50 > 10000 nM T40332 C5TQ1G 44368099 IC50 > 10000 nM T40332 C41CWE 44368121 IC50 > 10000 nM T40332 C1ZW4D 44368174 IC50 > 10000 nM T40332 C0BC2Q 44368175 IC50 > 10000 nM T40332 C6L9DK 44368178 IC50 = 450 nM T40332 CPE92K 44368218 IC50 = 7.2 nM T40332 C19ARS 44368431 IC50 > 10000 nM T40332 CMN18Z 44368433 IC50 = 13 nM T40332 C3S7YX 44368434 IC50 = 7.4 nM T40332 CIP7M3 44368435 IC50 > 10000 nM T40332 C62RSP 44368445 IC50 = 280 nM T40332 CV0Y2M 44368446 IC50 = 72 nM T40332 CCY58J 44368452 IC50 = 3.5 nM T40332 CSYO09 44368455 IC50 > 10000 nM T40332 CP6V1Y 44368456 IC50 > 10000 nM T40332 C0G6XP 44372603 Ki = 2 nM T40332 CQ6UZ3 44373218 IC50 > 5000 nM T40332 C0UE9N 44375714 IC50 = 0.365 ug.mL-1 T40332 CNFA42 44380213 IC50 = 380 nM T40332 CA84BI 44380230 IC50 = 74 nM T40332 CY5QC9 44380439 IC50 = 330 nM T40332 CD6AM9 44380440 IC50 = 320 nM T40332 CDMP49 44380948 Ki = 0.6 nM T40332 CVT80Q 44380960 Ki = 1.8 nM T40332 CED81F 44381178 Ki = 1.6 nM T40332 CKW3N0 44381293 Ki = 1.6 nM T40332 CO0X8N 44381295 Ki = 8000 nM T40332 CHI6Q5 44383146 IC50 = 26 nM T40332 C17LOX 44383308 IC50 = 274 nM T40332 CI3KG4 44383348 IC50 = 120 nM T40332 C0CW7E 44383468 IC50 = 242 nM T40332 CB3ED9 44383545 IC50 = 22 nM T40332 C1FCZ3 44384633 IC50 > 1000000 nM T40332 C8HL9B 44384637 IC50 = 810000 nM T40332 CR0T6A 44384638 IC50 = 665000 nM T40332 CTF25D 44384701 IC50 > 1000000 nM T40332 C2WSZ7 44384797 IC50 = 989000 nM T40332 CA0F5I 44384840 IC50 = 742000 nM T40332 CN0XD8 44384856 IC50 = 305000 nM T40332 CUBE67 44385436 IC50 = 454000 nM T40332 C8G1VT 44385622 IC50 = 92000 nM T40332 CLW2F7 44385646 IC50 = 895000 nM T40332 CF3GW6 44385689 IC50 > 1000000 nM T40332 C92XES 44385735 IC50 = 292000 nM T40332 CB35TE 44385740 IC50 > 1000000 nM T40332 C7W9MR 44385741 IC50 > 1000000 nM T40332 CU85DE 44385747 IC50 > 1000000 nM T40332 CK9I0A 44385748 IC50 > 1000000 nM T40332 CUAJ67 44385919 IC50 > 1000000 nM T40332 CJ98UI 44387451 IC50 = 41 nM T40332 C3JQH9 44398885 Ki = 2900 nM T40332 C0THI1 44415189 IC50 = 89800 nM T40332 CGDY32 44415219 IC50 = 75800 nM T40332 C6WR4P 44445934 Ki = 65 nM T40332 CA6E2R 44445935 Ki = 410 nM T40332 C3EBM1 44445936 Ki = 130 nM T40332 CBP7C3 44445937 Ki = 71 nM T40332 CE50KV 44452404 IC50 = 1560 nM T40332 C6M7VJ 44453668 Ki = 21000 nM T40332 C6J2PV 44453794 Ki = 6.4 nM T40332 CQT15C 44453896 Ki = 0.2 nM T40332 C2YA0P 44453914 Ki = 0.66 nM T40332 CUA0E6 44453915 Ki = 0.81 nM T40332 CN3K8S 44453963 Ki = 0.06 nM T40332 CMH91A 44454011 Ki = 0.35 nM T40332 CCP29L 44459365 Ki = 309 nM T40332 C20MDV 44459881 IC50 = 7000 nM T40332 CY34QH 44461452 Ki = 240 nM T40332 CSK2J8 44461627 Ki = 340 nM T40332 C5UHG2 44461629 Ki = 40 nM T40332 CU4O1C 44461630 Ki = 120 nM T40332 C7Y9HQ 44461644 Ki = 34 nM T40332 C82FIS 44461664 Ki = 9800 nM T40332 CG05CL 44461760 Ki = 400000 nM T40332 C23EAH 44461777 Ki = 20 nM T40332 C5RJ9A 44461780 Ki = 41000 nM T40332 C2R4ZM 44461781 Ki = 95000 nM T40332 CB0HR7 44461805 Ki = 1100 nM T40332 CZ4Q6H 44473061 IC50 = 7.6 nM T40332 C8WU0Y 44473063 IC50 = 43 nM T40332 CGA18I 44473064 IC50 = 42 nM T40332 CA8D5R 44473065 IC50 = 35 nM T40332 CCN52T 44473066 IC50 = 1000 nM T40332 CX4FB6 44473067 IC50 > 1000 nM T40332 C60FLK 44517752 IC50 = 8.1 nM T40332 CIT5G7 44561891 IC50 > 100000 nM T40332 C90BGR 44561892 IC50 > 100000 nM T40332 C9RGX4 44561893 IC50 > 100000 nM T40332 CU7NP5 44561930 IC50 > 100000 nM T40332 CV21IQ 44561931 IC50 = 33000 nM T40332 CR08WA 44561932 IC50 > 100000 nM T40332 C97JBD 44584781 IC50 > 100000 nM T40332 CBP4J9 44584783 IC50 > 100000 nM T40332 CUV18S 44584784 IC50 > 100000 nM T40332 C7ZYA5 44626812 Ki = 1.3 nM T40332 C98FOV 44626813 Ki = 33.9 nM T40332 CPG20K 44626906 Ki = 99.3 nM T40332 CJXK95 44626907 Ki = 7.6 nM T40332 CMXF01 44626997 Ki = 203 nM T40332 CR9I0Y 44626998 Ki = 0.82 nM T40332 COL76S 44626999 Ki = 0.34 nM T40332 CQS4G2 44627000 Ki = 1 nM T40332 C8KQH6 44627001 Ki = 1.1 nM T40332 C6V5XI 44627002 Ki = 0.5 nM T40332 CTP5R6 44627003 Ki = 1.8 nM T40332 CYO0Q2 44627268 IC50 = 16 nM T40332 C2PVE0 45103523 Ki > 26000 nM T40332 CGN14R 45103723 Ki > 26000 nM T40332 CJ0D8A 45267494 IC50 = 22 nM T40332 C32KHM 45267507 IC50 = 900 nM T40332 CY2VP7 45267519 IC50 = 8.6 nM T40332 CT18QR 45267524 IC50 = 28 nM T40332 CBS28A 45267536 IC50 = 850 nM T40332 CITF18 45268358 IC50 = 24 nM T40332 CKO71F 45268410 IC50 = 140 nM T40332 CL5GJ6 45268419 IC50 = 23 nM T40332 CLN7M0 45269246 IC50 = 79 nM T40332 C6K5CY 45269247 IC50 = 74 nM T40332 CKS94Q 45269257 IC50 = 5300 nM T40332 CSM9D3 45269258 IC50 = 2600 nM T40332 CIAG68 45269260 IC50 = 210 nM T40332 C90YKZ 45269266 IC50 = 15000 nM T40332 CM19HY 45269268 IC50 = 25 nM T40332 CPU0F3 45269270 IC50 = 28 nM T40332 C10DXZ 45270089 IC50 = 170 nM T40332 C6U2VN 45270092 IC50 = 160 nM T40332 COVE69 45270109 IC50 = 120 nM T40332 C6WZI7 45270119 IC50 = 27 nM T40332 CFY4G5 45270120 IC50 = 21 nM T40332 CMCK76 45270925 IC50 = 87 nM T40332 C5DC9K 45270953 IC50 = 150 nM T40332 CV1UK4 45271765 IC50 = 85 nM T40332 CAL64K 45271771 IC50 = 710 nM T40332 CLOK73 45271783 IC50 = 8.5 nM T40332 C8SM0J 45271784 IC50 = 20 nM T40332 CBW47X 45271792 IC50 = 330 nM T40332 C1BQ7N 45271797 IC50 = 34 nM T40332 C6SRB3 45272629 IC50 = 16 nM T40332 CND82I 45272646 IC50 = 28 nM T40332 C4U6MS 45272654 IC50 = 250 nM T40332 CTS68D 45272660 IC50 = 180 nM T40332 CES4L3 45273539 IC50 = 21 nM T40332 C5WYG0 45273548 IC50 = 9300 nM T40332 CYI53S 45273574 IC50 = 71 nM T40332 C5KYI2 45273582 IC50 = 140 nM T40332 CJ3MI1 45273583 IC50 = 110 nM T40332 C6T2AJ 45273590 IC50 = 1300 nM T40332 CD4T1L 46221636 Ki = 13000 nM T40332 CN7QI3 46221638 IC50 = 300 nM T40332 CF16UR 46225505 IC50 > 100000 nM T40332 C81XNC 46225794 IC50 = 33 nM T40332 C4YAJ7 46228924 IC50 > 10000 nM T40332 C46YMU 46838142 IC50 = 30.8 nM T40332 COP81J 46838143 IC50 = 30.7 nM T40332 C1PDI7 46838144 IC50 = 24.8 nM T40332 COQH23 46838145 IC50 = 48.8 nM T40332 CI19BN 46838146 IC50 = 15.4 nM T40332 CD28QR 46882316 Ki > 7500 nM T40332 C86FZA 46882318 Ki = 32 nM T40332 C3G9BA 46882319 Ki = 21 nM T40332 C8JFN6 46882328 Ki = 520 nM T40332 CUI91D 46905615 IC50 = 1900 nM T40332 CX8S3H 46933351 Ki = 7340 nM T40332 C41UEJ 49759015 IC50 = 2400 nM T40332 CJH50R 49797481 IC50 > 100000 nM T40332 CI7P2B 49797571 IC50 = 170 nM T40332 CI59MV 49797572 IC50 > 30000 nM T40332 C96CKU 49797573 IC50 = 220 nM T40332 C50QVP 53262865 IC50 = 830 nM T40332 C6AFX0 53320723 IC50 = 500 nM T40332 CCR6H5 53357861 IC50 = 89 nM T40332 CI9GP5 53357862 IC50 = 130 nM T40332 C52ZET 53357863 IC50 = 240 nM T40332 C53JUT 53357864 IC50 = 260 nM T40332 C9YK0S 53357865 IC50 = 180 nM T40332 CP7ZW2 53784885 IC50 = 0.036 nM T40332 CBJQ98 54132077 IC50 = 370 nM T40332 C0WH1K 54675757 Ki = 8128305.16 nM T40332 CNEI60 54678950 Ki = 1100000 nM T40332 CL42YZ 54685126 Ki = 93325.43 nM T40332 C29BYX 54686804 Ki = 1700000 nM T40332 CJ6BS7 54690337 Ki = 6309573.44 nM T40332 CPQ05N 54693753 IC50 = 3150000 nM T40332 CY4VG6 54693756 IC50 = 1620000 nM T40332 CQ85OF 54694046 Ki = 4897788.19 nM T40332 CV0U6E 54694048 Ki = 10000000 nM T40332 C95DEC 54694049 Ki = 645654.23 nM T40332 C9FGL4 54694052 Ki = 6025595.86 nM T40332 C01LMD 54694053 Ki = 489778.82 nM T40332 C1K4RP 54695445 IC50 = 26800 nM T40332 CL4N6C 54707146 Ki = 95499.26 nM T40332 C9FQ0U 54709932 IC50 = 35800 nM T40332 C5FPG9 54728809 IC50 = 153000 nM T40332 C28IAV 54732424 Ki = 151356.12 nM T40332 C1T9XJ 54733673 Ki = 977237.22 nM T40332 COA25T 54733674 Ki = 363078.05 nM T40332 CJ4LH1 54735926 Ki = 400000 nM T40332 CPGD29 56598201 IC50 = 9280 nM T40332 C6QCK2 56598333 IC50 > 20000 nM T40332 C8U4OD 56649692 IC50 > 1000000 nM T40332 C8QC6E 56659686 IC50 = 29000 nM T40332 CFTW24 56659687 IC50 = 5900 nM T40332 C6TDH1 56659688 IC50 = 8100 nM T40332 C4A7XT 56659690 IC50 = 36000 nM T40332 C2Y7HM 56659691 IC50 = 930 nM T40332 C3LO5F 56659692 IC50 = 1600 nM T40332 CJ0AU4 56659693 IC50 = 400 nM T40332 C0FP7U 56659694 IC50 = 780 nM T40332 CZ1RB3 56659695 IC50 = 650 nM T40332 C9C6SF 56659699 IC50 = 22000 nM T40332 C8GT6J 56663146 IC50 = 3900 nM T40332 CX8BK7 56663147 IC50 = 6100 nM T40332 CVEQ14 56663148 IC50 = 11000 nM T40332 C0A9JD 56663149 IC50 = 52000 nM T40332 CZS51B 56663151 IC50 = 310 nM T40332 CA9LH5 56663152 IC50 = 1900 nM T40332 CFL20B 56663153 IC50 = 510 nM T40332 CAXE63 56663154 IC50 = 890 nM T40332 CM7DT1 56663155 IC50 = 510 nM T40332 CS3O6Z 56663156 IC50 = 340 nM T40332 C9HUK8 56666600 IC50 = 38000 nM T40332 C1CV4T 56666601 IC50 = 25000 nM T40332 CJPL65 56666602 IC50 = 410 nM T40332 C7RWF1 56666605 IC50 = 700 nM T40332 C12FWP 56666606 IC50 = 690 nM T40332 CWH4G9 56666607 IC50 = 480 nM T40332 CVU62F 56670016 IC50 = 1800 nM T40332 C4GJH8 56670017 IC50 = 3100 nM T40332 CFMA80 56670019 IC50 = 10000 nM T40332 CL20GF 56673430 IC50 = 800 nM T40332 CDH38Y 56673525 IC50 = 33000 nM T40332 C7ET5S 56673526 IC50 = 1700 nM T40332 CY4JH2 56673529 IC50 = 550 nM T40332 C1MN5G 56673530 IC50 = 400 nM T40332 C3TUR8 56674980 Ki = 269700 nM T40332 CY5R9M 56676773 IC50 = 420 nM T40332 CSC9U1 56676774 IC50 = 34000 nM T40332 CK9YG2 56676775 IC50 = 930 nM T40332 C5P4NQ 56676842 IC50 = 1700 nM T40332 C8NC2F 56676843 IC50 = 38000 nM T40332 C74KYG 56676844 IC50 = 460 nM T40332 C0AV1L 56680166 IC50 = 3100 nM T40332 CY1TH5 56680168 IC50 = 28000 nM T40332 C4SW5X 56680170 IC50 = 1900 nM T40332 CAJN07 56683509 IC50 = 760 nM T40332 C0UIF5 57671050 IC50 > 100000 nM T40332 CY26NE 57671116 IC50 > 10000 nM T40332 C9E6CB 57671131 IC50 > 10000 nM T40332 CJO75X 57671161 IC50 > 10000 nM T40332 CTH9W2 58343687 IC50 = 2700 nM T40332 CDZ05M 59145670 IC50 = 3.5 nM T40332 C5ON3H 60195210 IC50 = 680 nM T40332 C48UHX 66561877 IC50 = 2600 nM T40332 CL93DE 66725365 IC50 = 17 nM T40332 C17JAZ 68284084 IC50 > 30000 nM T40332 CTP6M3 70681508 IC50 > 500000 nM T40332 C25DHK 70685488 IC50 >> 5000 nM T40332 CD9N4J 70687893 IC50 > 500000 nM T40332 CLW0V4 70687894 IC50 > 500000 nM T40332 C3SZ6M 70696249 IC50 > 500000 nM T40332 C8JPF6 71450320 Ki = 5000 nM T40332 C06BIJ 71452128 Ki = 4000 nM T40332 CBU34G 71452812 IC50 = 7000 nM T40332 C03DMT 71452813 IC50 = 15000 nM T40332 CKG69H 71454592 IC50 = 700 nM T40332 C0XV2L 71455698 IC50 = 14000 nM T40332 CH8C9Z 71455699 IC50 > 200000 nM T40332 C6TI5U 71455700 IC50 > 200000 nM T40332 C3A8KU 71456312 IC50 = 3000 nM T40332 CL62BK 71457475 IC50 = 300 nM T40332 CF9XP4 71457476 IC50 > 200000 nM T40332 C96SGY 71457477 IC50 = 46000 nM T40332 CU9O8L 71459588 Ki = 0.6 nM T40332 CZH4E8 71460024 IC50 = 600 nM T40332 CF5O8M 71461119 IC50 = 39000 nM T40332 CH87QX 71461740 IC50 = 300 nM T40332 C2PKD0 71462857 IC50 = 51000 nM T40332 C83ZNH 71562308 IC50 = 40 nM T40332 CL9VA2 71562455 IC50 = 121 nM T40332 CTJR81 71562563 IC50 = 28 nM T40332 C6LB5N 71659627 IC50 = 8400 nM T40332 C0DPM1 71659628 IC50 > 100000 nM T40332 CRH4J2 71659766 IC50 > 100000 nM T40332 C2BDV0 71659767 IC50 = 46600 nM T40332 C78DJQ 71711730 IC50 < 10000 nM T40332 C51TZR 71717105 IC50 = 21 nM T40332 CQIA07 71717727 IC50 = 195 nM T40332 CULQ46 71718935 IC50 = 41 nM T40332 CL23VT 71723878 IC50 > 100000 nM T40332 C5RSD4 71818404 IC50 = 20 nM T40332 CS0OQ1 71818406 IC50 = 330 nM T40332 CXO32I 71818543 IC50 = 310 nM T40332 CDH81R 71818544 IC50 = 140 nM T40332 COX58Z 71818547 IC50 = 31 nM T40332 CQ9OD7 71818548 IC50 = 40 nM T40332 CVPL10 71818549 IC50 = 7 nM T40332 C6X9AY 71818550 IC50 = 260 nM T40332 CKS7E3 71818686 IC50 = 12500 nM T40332 CY7ZS9 71818687 IC50 = 6400 nM T40332 CVCM38 71818688 IC50 = 30 nM T40332 CA56TS 71818689 IC50 = 15 nM T40332 C1S2VT 71818690 IC50 = 50 nM T40332 CFV7P5 71818691 IC50 = 50 nM T40332 CK2XH0 71818692 IC50 = 20 nM T40332 CXV8Z4 71818829 IC50 = 25 nM T40332 C7UY4N 71818830 IC50 = 30 nM T40332 C6X2FC 71818831 IC50 = 30 nM T40332 C80YBP 71818832 IC50 = 18 nM T40332 CKCP90 71818833 IC50 = 50 nM T40332 CYC57T 71818834 IC50 = 210 nM T40332 C2D1NZ 71818963 IC50 = 100 nM T40332 CXV20J 71818964 IC50 = 12 nM T40332 C2M1ZG 71818965 IC50 = 50 nM T40332 CLV3J9 71818966 IC50 = 330 nM T40332 CQI96C 71819101 IC50 = 80 nM T40332 CY82VQ 71819102 IC50 = 80 nM T40332 CL3KA5 71819103 IC50 = 210 nM T40332 CWY8D4 71819104 IC50 = 160 nM T40332 CQ1K8Y 71819105 IC50 = 80 nM T40332 C2NP3X 71819106 IC50 = 270 nM T40332 CL8I3R 71819107 IC50 = 260 nM T40332 C4QL2M 71819248 IC50 = 220 nM T40332 C7HQD3 71819249 IC50 = 150 nM T40332 CSDL97 71819250 IC50 = 100 nM T40332 CYF8I9 71819251 IC50 = 80 nM T40332 CCKZ58 71819252 IC50 = 140 nM T40332 CMXU14 71819253 IC50 = 60 nM T40332 CO72XA 71819254 IC50 = 110 nM T40332 CR43YH 71819387 IC50 = 6400 nM T40332 CW3QR2 72712049 Ki = 68700 nM T40332 CAL2W7 72712050 Ki = 11300 nM T40332 C2A4TH 72712051 Ki > 250000 nM T40332 CN73TI 72712053 Ki > 250000 nM T40332 C3J8RV 72712070 Ki > 250000 nM T40332 C8QJ2R 72793725 IC50 = 450 nM T40332 CG9R4L 72793726 IC50 = 4100 nM T40332 CHLW60 72793743 IC50 = 8900 nM T40332 C7J9MS 72793744 IC50 = 14300 nM T40332 CC28PB 72793745 IC50 > 50000 nM T40332 C60WDY 72793746 IC50 = 670 nM T40332 C1MBU7 72793747 IC50 = 110 nM T40332 CBT72J 72793748 IC50 = 1190 nM T40332 CP7XG2 72793760 IC50 = 1200 nM T40332 CETY07 72793761 IC50 = 4600 nM T40332 CNF72C 72793762 IC50 = 5190 nM T40332 C76CUL 72793763 IC50 = 960 nM T40332 C9MWN6 72793764 IC50 = 300 nM T40332 CLY96J 72793765 IC50 = 280 nM T40332 C6BY5D 72793776 IC50 = 180 nM T40332 CHL95X 72793777 IC50 = 2460 nM T40332 C1DI8A 72793778 IC50 = 80 nM T40332 CNU1I7 73051428 IC50 < 20 nM T40332 C10ITF 73345210 IC50 >> 5000 nM T40332 CR7HX5 73345258 IC50 = 2 nM T40332 C4E7TG 73345260 IC50 = 94 nM T40332 C7BKZ5 73345448 IC50 = 100 nM T40332 CR3E1A 73345466 Ki = 17 nM T40332 C14AZB 73345741 Ki = 3.9 nM T40332 C3M6NT 73345742 Ki = 15 nM T40332 CV0TP1 73345743 Ki = 150 nM T40332 C5KHS8 73347173 Ki = 1200 nM T40332 CD26JR 73347227 Ki = 7.8 nM T40332 C04QVO 73347230 IC50 = 32 nM T40332 C5AMR2 73348056 IC50 = 7800 nM T40332 CL1Z5W 73348476 Ki = 500 nM T40332 C8OMT5 73348493 Ki = 43 nM T40332 CTP68V 73348565 Ki = 200 nM T40332 CE26GR 73348743 Ki = 2 nM T40332 C4XN1F 73348744 Ki = 0.63 nM T40332 CD6HY8 73349819 IC50 >> 5000 nM T40332 C87PWL 73349864 IC50 = 31 nM T40332 C0ONC3 73350318 Ki = 2.9 nM T40332 CU0H6E 73350319 Ki = 14 nM T40332 CH4L7K 73350322 IC50 = 210 nM T40332 CO01PD 73351555 IC50 = 30 nM T40332 CRQS78 73351639 Ki = 44 nM T40332 CXL3Q6 73351830 Ki = 16 nM T40332 C8TOM4 73351831 Ki = 0.96 nM T40332 CH52ZV 73351832 Ki = 3.8 nM T40332 CVGO29 73352827 IC50 = 29 nM T40332 C7BYL1 73353012 IC50 = 120000 nM T40332 C84NFB 73353013 IC50 = 60 nM T40332 C8TC2M 73353039 Ki = 1.9 nM T40332 CKSD62 73353041 Ki = 20 nM T40332 COQ9E0 73353305 Ki = 2.6 nM T40332 CTWH20 73353306 Ki = 45 nM T40332 C2CM8U 73354616 Ki = 234.42 nM T40332 C4DVG0 73354687 Ki = 210 nM T40332 CO3A5T 73354820 Ki = 1 nM T40332 C48MTS 73354821 Ki = 11 nM T40332 C3OTL1 73355884 IC50 = 172 nM T40332 C04GZD 73355907 IC50 = 0.69 nM T40332 CY81IS 73356107 IC50 > 1000000 nM T40332 C84MDZ 73356367 Ki = 6.8 nM T40332 CS15MB 73356368 Ki = 810 nM T40332 CJ2DF3 73356369 Ki = 20 nM T40332 CX17VC 76284943 IC50 < 20 nM T40332 CALM86 76335198 Ki = 0.4 nM T40332 CP6T1S 77844774 IC50 = 22 nM T40332 CAL1Y8 77844829 IC50 < 1 nM T40332 CGM61S 77844945 IC50 < 1 nM T40332 CH7GQ9 86268083 IC50 = 74700 nM T40332 C53SOM 90310890 IC50 = 2.4 nM T40332 CM06KI 90311037 IC50 = 1.6 nM T40332 CP50TI 90643774 Ki = 38000 nM T40332 CG2Q3B 90643775 Ki = 22000 nM T40332 CJKX87 90643776 Ki = 36000 nM T40332 CU9WA6 90643777 Ki = 39000 nM T40332 CK89GM 90643778 Ki = 39000 nM T40332 CF0R9S 90643779 Ki = 39000 nM T40332 CU5N9Z 90663487 IC50 = 107 nM T40332 CH1OE8 90666510 IC50 > 100000 nM T40332 C7ZCN4 90676239 IC50 = 4400 nM T40332 C6IO0L 90676242 IC50 = 1400 nM T40332 C4S9WP 90676243 IC50 = 900 nM T40332 C8O4GH 90676244 IC50 > 10000 nM T40332 C0CTE9 90676245 IC50 = 500 nM T40332 C7GDE8 90676248 IC50 = 500 nM T40332 C25ZWA 90676249 IC50 = 1100 nM T40332 C7OX2A 90676250 IC50 = 2900 nM T40332 CMV0H1 90676258 IC50 = 1500 nM T40332 C8E4WS 102323332 IC50 > 50000 nM T40332 CR2AU7 118010068 IC50 = 320 nM T40332 COA36C 118010069 IC50 = 370 nM T40332 C5NJH1 118202505 IC50 = 680 nM T40332 C43ADS 118202506 IC50 = 110 nM T40332 C2UXT7 118202507 IC50 = 50 nM T40332 CPV27G 118202509 IC50 = 120 nM T40332 CJB3K7 118202510 IC50 = 190 nM T40332 C12BHL 118202511 IC50 = 360 nM T40332 COT6H0 118202512 IC50 = 370 nM T40332 CFS4A9 118716662 IC50 = 3.7 nM T40332 C2WNT9 118716663 EC50 < 1 nM T40332 C8ZSC2 118727248 IC50 = 2240 nM T40332 CYIX41 118727249 IC50 = 390 nM T40332 CH1T3M 118727250 IC50 = 820 nM T40332 CVG1X5 118727251 IC50 = 480 nM T40332 C9B6KX 118727252 IC50 = 1230 nM T40332 C3OUW6 118727253 IC50 > 10000 nM T40332 C10QJC 118727254 IC50 > 10000 nM T40332 CVIF56 118727255 IC50 > 10000 nM T40332 CNQ9U4 118727256 IC50 = 3690 nM T40332 CN93WU 118727257 IC50 > 10000 nM T40332 C5DR7Z 118727258 IC50 > 10000 nM T40332 CDEU05 118727259 IC50 = 130 nM T40332 CZHT12 118727260 IC50 = 290 nM T40332 C3WC9Y 121488127 IC50 > 100000 nM T40332 CKJN32 122164799 IC50 > 30000 nM T40332 CYEA84 122190691 IC50 < 1 nM T40332 C9QKI3 127020966 IC50 > 100000 nM T40332 CE26HW 131955087 IC50 > 100000 nM T40332 CES7P6 132517499 IC50 = 21000 nM T40332 CGE51P 135672692 IC50 = 2910 nM T40332 C7YVL9 135981708 IC50 = 3010 nM T40332 CZ9X0E 137634272 IC50 = 51900 nM T40332 CNL2Z9 137635679 Ki = 12000 nM T40332 C43ETF 137637257 IC50 = 47600 nM T40332 C7BQ8O 137644210 IC50 = 19100 nM T40332 C9BEA1 137644608 IC50 = 64800 nM T40332 C6BE7C 137646856 IC50 = 157000 nM T40332 C03IMN 137647139 Ki = 8900 nM T40332 CNO2T8 137647340 IC50 = 230 nM T40332 CME1B3 137649275 IC50 = 810 nM T40332 C7WRB2 137652193 IC50 = 640 nM T40332 CZ1H4R 137655362 Ki = 43000 nM T40332 C47IZA 137655464 IC50 = 1560 nM T40332 CVN59W 137656193 IC50 = 91300 nM T40332 C34UDN 137657165 IC50 = 2650 nM T40332 C0C5JK 137657334 IC50 = 320 nM T40332 CTUM82 137658421 IC50 = 690 nM T40332 CUZ35A 138115400 IC50 > 100000 nM T40332 C6OP2I 140742745 IC50 = 250 nM T40332 CZT48W 140742746 IC50 = 7000 nM T40332 C61ODQ 145952347 Ki = 3200 nM T40332 C10EWY 145953439 IC50 > 100000 nM T40332 C5WFZ3 145955487 Ki = 6300 nM T40332 C1ZYD7 145955680 Ki = 12400 nM T40332 CFOI32 145956166 Ki = 19500 nM T40332 C1MJ0P 145957172 IC50 = 2400 nM T40332 C95HXU 145958432 IC50 = 35600 nM T40332 C27FNP 145960559 Ki = 13100 nM T40332 C9OK4P 145979023 IC50 = 800 nM T40332 C0CJ8N 145979295 IC50 = 12600 nM T40332 C2KTP8 145979350 IC50 = 1500 nM T40332 CZ2S6U 145979786 IC50 = 80 nM T40332 CLYZ05 145980145 IC50 = 6700 nM T40332 CWBN57 145980442 IC50 = 490 nM T40332 CCT8O7 145980848 IC50 = 7300 nM T40332 C6B2NR 145981285 IC50 = 11900 nM T40332 CVE50X 145982102 IC50 = 44800 nM T40332 CDT82U 145982407 IC50 = 87 nM T40332 CSL8R0 145985380 IC50 = 640 nM T40332 CJW50C 145986748 IC50 = 3400 nM T40332 CS0V3Y 145987313 IC50 = 19100 nM T40332 CO1PC5 145987373 IC50 = 15 nM T40332 CI5AZ8 145987496 IC50 = 2600 nM T40332 CNHI09 145988102 IC50 = 1500 nM T40332 CCD6J8 145988308 IC50 = 28500 nM T40332 C9EJT1 145988325 IC50 = 38500 nM T40332 CW2HO0 145988348 IC50 = 42600 nM T40332 CR8V9N 145988581 IC50 = 3600 nM T40332 C8PIN1 145988987 IC50 = 1800 nM T40332 CD6ZT8 145989305 IC50 = 24 nM T40332 CM1G6B 145989653 IC50 = 6000 nM T40332 CJT4G6 145990495 IC50 = 11500 nM T40332 C0XQV5 145990804 IC50 = 620 nM T40332 CT7R5S 145990987 IC50 = 14 nM T40332 CCJF05 145991040 IC50 = 1800 nM T40332 C91SQO 145991281 IC50 = 2400 nM T40332 CDW8L7 145991384 IC50 = 770 nM T40332 CHZ5V0 145993786 IC50 = 390 nM T40332 CSBC71 146680900 IC50 = 55000 nM T40332 CH82XM 155511283 IC50 = 4710 nM T40332 CZR36C 155511554 IC50 = 12589.25 nM T40332 CSL60M 155511684 IC50 = 3230 nM T40332 CT3GQ1 155517665 IC50 = 197 nM T40332 C9HK4E 155519617 IC50 = 1540 nM T40332 C6NX4K 155519661 IC50 > 100000 nM T40332 C4MS1B 155519676 IC50 = 100000 nM T40332 C7L5RK 155520356 IC50 = 103 nM T40332 CH1Y5O 155522603 IC50 = 10100 nM T40332 C9KE6J 155524006 IC50 = 2190 nM T40332 CBU5W0 155524880 Ki = 24 nM T40332 CN3BH5 155527998 IC50 = 794.33 nM T40332 CL4RC9 155528080 IC50 = 595 nM T40332 CHYW65 155528639 IC50 = 1258.93 nM T40332 CLJI15 155529200 IC50 = 2350 nM T40332 CD7O2G 155530095 IC50 = 31622.78 nM T40332 C3W2MJ 155530593 IC50 = 35800 nM T40332 C35QWO 155531023 IC50 > 100000 nM T40332 C2X5EJ 155531124 IC50 > 10000 nM T40332 C50ZHO 155533944 IC50 = 4830 nM T40332 CJB82P 155535066 IC50 = 5850 nM T40332 C10QDI 155535871 IC50 = 2600 nM T40332 C12HON 155536142 IC50 > 100000 nM T40332 CHUF10 155537107 IC50 > 500000 nM T40332 CX6S5M 155537400 IC50 = 140 nM T40332 CZMX52 155540843 IC50 = 10000 nM T40332 CY6DK3 155540964 IC50 = 15848.93 nM T40332 CG8OY6 155543393 IC50 = 1350 nM T40332 CV9N7I 155543726 IC50 = 21700 nM T40332 C5MB9R 155547962 IC50 = 6309.57 nM T40332 CLFB25 155548371 IC50 = 25118.86 nM T40332 CS57LN 155549377 IC50 = 2340 nM T40332 CUF2J6 155550172 IC50 = 840 nM T40332 CWC8X9 155550748 IC50 > 100000 nM T40332 COM52R 155551892 IC50 = 1584.89 nM T40332 CJ3FI5 155553630 IC50 > 100000 nM T40332 C2E5GR 155554478 Ki = 3.2 nM T40332 CJL26S 155555493 IC50 = 400 nM T40332 CE3G5W 155556110 IC50 > 10000 nM T40332 C0SND3 155557259 IC50 > 10000 nM T40332 C7E2NJ 155557306 IC50 > 10000 nM T40332 CA38JF 155557625 IC50 = 360 nM T40332 CSW48V 155557718 IC50 > 100000 nM T40332 CTS63Q 155558248 IC50 > 10000 nM T40332 CFX07G 155558369 Ki = 16 nM T40332 C9X7TF 155560751 IC50 = 450 nM T40332 C6JPU5 155564831 IC50 = 6300 nM T40332 CM8XB1 155565537 IC50 = 5011.87 nM T40332 CS54OQ 155566050 IC50 = 680 nM T40332 CW96TS 155566656 IC50 > 150000 nM T40332 CU42CE 155567829 IC50 > 100000 nM T40332 CQA3R5 155569370 IC50 = 721 nM T40332 CY9GR5 10009357 IC50 = 11100 nM T40332 CAI36L 10101940 IC50 = 404 nM T40332 C4BL1N 10327685 IC50 = 69 nM T40332 C7OHD3 10350525 IC50 = 4900 nM T40332 CAUB96 10440265 IC50 = 57 nM T40332 CX6PI4 14861876 IC50 = 153 nM T40332 CF4B3J 21832914 IC50 = 65 nM T40332 C4PVG3 44372915 IC50 = 138 nM T40332 CR1T4Y 44372920 IC50 = 5100 nM T40332 CJ8ZU5 44372983 IC50 > 5000 nM T40332 C4T1XJ 44372984 IC50 = 1562 nM T40332 CNLX57 44373015 IC50 > 5000 nM T40332 CT7R5D 44373019 IC50 = 30 nM T40332 CGX5Q3 44373020 IC50 = 84 nM T40332 C6KD9P 44373025 IC50 = 73 nM T40332 C9ZSG2 44373051 IC50 = 693 nM T40332 C18WIL 44373075 IC50 = 817 nM T40332 C0W3BJ 44373137 IC50 > 5000 nM T40332 CEN6O7 44373154 IC50 = 57 nM T40332 CO1H7G 44373162 IC50 = 149 nM T40332 CQOI69 44373163 IC50 = 175 nM T40332 CE7W2Y 44373173 IC50 > 5000 nM T40332 C23GOW 44373196 IC50 > 5000 nM T40332 C3DX2N 44373204 IC50 = 110 nM T40332 CPL8V3 44373205 IC50 = 52 nM T40332 CUI13J 44373211 IC50 = 452 nM T40332 CY0Z5O 44373212 IC50 = 5000 nM T40332 C1JMP8 44373240 IC50 = 61 nM T40332 C91JLZ 44373268 IC50 = 73 nM T40332 CYK80J 44373269 IC50 = 92 nM T40332 CJP5G2 44373315 IC50 = 156 nM T40332 CK78NM 44373333 IC50 = 153 nM T40332 CEK35P 44373526 IC50 = 217 nM T40332 C8DQ4W 44373542 IC50 = 507 nM T40332 C2N0KC 44373543 IC50 = 67 nM T40332 C8CJ2N 9986046 IC50 > 5000 nM T40332 CLNZ94 9986475 IC50 = 635 nM T40332 C68QAJ 9988180 IC50 > 5000 nM T40332 D00RIX 5280443 IC50 = 46100 nM T40332 D00TYW 54678949 Ki = 15000 nM T40332 D00WFQ 674641 Ki = 65 nM T40332 D02AKP 695069 Ki = 2500 nM T40332 D02AVL 18376720 Ki > 5000 nM T40332 D02NRY 674650 Ki = 300 nM T40332 D02PAU 16731825 Ki = 10000 nM T40332 D03BNM 10053241 Ki = 3 nM T40332 D03MNO 121963 Ki = 2.2 nM T40332 D03STO 24823606 Ki = 114 nM T40332 D04KAS 44454029 Ki = 73 nM T40332 D04ODG 44626814 Ki = 3.9 nM T40332 D04SPO 44584782 IC50 = 18000 nM T40332 D05ICF 3492365 IC50 = 230 nM T40332 D05ZIP 674656 Ki = 45 nM T40332 D06GTS 76318115 IC50 = 630 nM T40332 D06JMS 44626902 Ki = 4450 nM T40332 D06LPR 674651 Ki = 34 nM T40332 D07DOW 685230 Ki = 3400 nM T40332 D07HLC 24823444 Ki = 34.4 nM T40332 D07IBU 10696098 IC50 > 10000 nM T40332 D08OCS 699665 Ki = 28 nM T40332 D08RPN 674653 Ki = 250 nM T40332 D08WQJ 700133 Ki = 46 nM T40332 D09FGQ 123985 IC50 > 300000 nM T40332 D0A5ZF 44626811 Ki = 2.2 nM T40332 D0B4WZ 44626901 Ki = 127 nM T40332 D0C1NP 66561876 IC50 = 10200 nM T40332 D0D6ZB 25205741 IC50 = 7 nM T40332 D0E0EQ 708205 Ki = 110 nM T40332 D0F2YC 10038543 IC50 = 100 nM T40332 D0F3CA 1609 IC50 = 100 nM T40332 D0H8EO 139973 Ki = 1.21 nM T40332 D0I1AC 577102 Ki = 230 nM T40332 D0IU5E 716930 Ki = 39 nM T40332 D0J1LX 24882417 IC50 = 540 nM T40332 D0L8DL 9889727 Ki = 0.27 nM T40332 D0MQ8A 20283207 Ki = 0.85 nM T40332 D0N9DP 54737457 Ki = 4600 nM T40332 D0O8PM 669334 Ki = 290 nM T40332 D0PQ8B 54736658 Ki = 7900 nM T40332 D0Q7ST 44338671 IC50 = 800 nM T40332 D0R9CH 3400921 Ki > 10000 nM T40332 D0S5RY 4784 IC50 = 52161.7 nM T40332 D0T9WZ 54613196 IC50 = 4220 nM T40332 D0X1OY 674628 Ki = 104 nM T40332 D0Z7LS 44626810 Ki = 233 nM T16691 D00KHM 16362 Ki = 71 nM T16691 D01AZG 5073 Ki = 224 nM T16691 D01XBA 5035 Ki = 750 nM T16691 D01ZII 2726 Ki = 4 nM T16691 D03WEX 9966051 Ki = 330 nM T16691 D04JEE 4946 EC50 > 5011.87 nM T16691 D04VFJ 3005573 Ki = 4125 nM T16691 D04WFD 4543 Ki = 214 nM T16691 D06YFA 31101 Ki < 50 nM T16691 D07KSG 2733526 Ki = 1041 nM T16691 D08VRO 3822 Ki = 2800 nM T16691 D0B0CP 667467 Ki = 3 nM T16691 D0CQ0Z 33630 Ki = 1000 nM T16691 D0D1AL 3559 Ki = 1083 nM T16691 D0G8NN 119570 Ki > 10000 nM T16691 D0H3HM 60795 Ki = 89 nM T16691 D0H7KF 5002 Ki > 1000 nM T16691 D0I8LU 5311507 Ki = 169 nM T16691 D0MA9N 2955 Ki = 183 nM T16691 D0P5SA 3372 Ki < 50 nM T16691 D0R1JV 60854 Ki = 20 nM T16691 D0R6RO 4184 Ki = 55 nM T16691 D0U5FS 3396 Ki = 1188 nM T16691 D0U5OE 3964 Ki = 15 nM T16691 D0V4QS 135398745 Ki = 5 nM T16691 D0W5HK 216239 Ki = 6213 nM T16691 D0Z1RV 135398737 Ki = 4 nM T16691 D0ZS8P 2801 Ki = 112 nM T16691 D08CJK 1150 Ki = 70 nM T16691 D09IRN 21071390 Ki = 0.83 nM T16691 D0N1HW 5311200 Ki = 1656.2 nM T16691 D0R9HI 11256720 Ki = 0.166 nM T16691 D0V4ZQ 16071605 Ki = 1.3 nM T16691 D00OWF 5280953 Ki = 1480 nM T16691 D02JMI 9888211 Ki = 398.11 nM T16691 D03PJW 108029 IC50 = 79 nM T16691 D06DZI 107780 Ki > 10000 nM T16691 D06ZVC 10150497 Ki = 2 nM T16691 D08AWI 11430856 Ki > 5000 nM T16691 D0B7SP 11292933 Ki > 5011.87 nM T16691 D0M7LV 5761 Ki = 6.31 nM T16691 D0OS6O 60149 Ki = 5 nM T16691 D0Q2JS 10436045 Ki = 79.43 nM T16691 D0YP7L 6604889 Ki = 6309.57 nM T16691 C36WOC 2800 Ki = 1956 nM T16691 CJ0B9F 3158 Ki = 105 nM T16691 C5H9CN 9287 Ki = 909 nM T16691 C2TYP0 31386 Ki = 1598 nM T16691 C6WDL7 49756 Ki = 60 nM T16691 CTB26S 52899 Ki = 80 nM T16691 C3PWO1 77956 Ki = 491 nM T16691 C0ALO6 152215 Ki = 98 nM T16691 CGT8R0 160510 Ki = 1450 nM T16691 CLK7P3 169713 IC50 = 16 nM T16691 CLG13W 227584 Ki = 482 nM T16691 C5BNW8 235964 Ki = 630.96 nM T16691 CYV1R3 417052 Ki = 1930 nM T16691 CN2RL6 460659 Ki = 564 nM T16691 CYZ25A 563919 Ki = 10 nM T16691 C1EY3K 616691 Ki = 33 nM T16691 CKR2N7 621659 IC50 = 370 nM T16691 CLUH96 627240 Ki = 114 nM T16691 C86DOU 640912 Ki = 866 nM T16691 C1QWJ9 675366 Ki = 198 nM T16691 CXQ6U0 735755 IC50 > 10000 nM T16691 C1RC8P 744368 Ki > 5000 nM T16691 C2VLP8 752521 Ki = 696 nM T16691 CXB86D 846090 Ki = 875 nM T16691 C6N9QC 1244725 Ki = 61 nM T16691 C9FI5L 1296368 Ki = 15610 nM T16691 C08VKR 1472656 Ki = 237 nM T16691 C6VZT7 1984087 Ki = 2700 nM T16691 CGS9R7 2133793 Ki = 7886 nM T16691 CG9N3A 2136365 Ki = 1174 nM T16691 CT8KN9 2232766 Ki = 2539 nM T16691 CA2OY6 2737389 Ki = 596 nM T16691 CBK16O 2771410 Ki = 28 nM T16691 C0QTF4 2771418 Ki = 482 nM T16691 CP8NQ2 2771419 Ki = 25 nM T16691 CP9O0G 2771422 Ki = 1512 nM T16691 CPI2C5 2775690 Ki = 1262 nM T16691 C29YXF 2816054 Ki = 5700 nM T16691 C1C4LH 2843443 Ki = 12730 nM T16691 CO4MP2 2845118 Ki = 250 nM T16691 C7UVI2 2848343 Ki = 1221 nM T16691 CRA6F5 2853434 Ki = 3104 nM T16691 CB6EK5 2854567 Ki = 80 nM T16691 C41ULI 2855326 Ki = 245 nM T16691 C6DL8S 2866185 Ki = 1490 nM T16691 C3QRD6 2867758 Ki = 5800 nM T16691 C9WY0K 2870667 Ki = 8 nM T16691 CL2G3H 2870750 Ki = 6401 nM T16691 CC74QS 2872937 Ki = 9669 nM T16691 C2G4DQ 2876391 Ki = 5 nM T16691 CRF65H 2880253 Ki = 5600 nM T16691 C54SFI 2883218 Ki = 894 nM T16691 C6L8FJ 2891368 Ki = 119 nM T16691 C7KJ4R 2894562 Ki = 290 nM T16691 CH4X1C 2906325 Ki = 12 nM T16691 CFE09S 2906372 Ki = 1267 nM T16691 CT4VY7 2906559 Ki = 61 nM T16691 CET7C8 2921525 Ki = 3700 nM T16691 C2DE6R 2927683 Ki = 1400 nM T16691 CF01YE 2928642 Ki = 2500 nM T16691 CY8R6Q 2948971 Ki = 670 nM T16691 CLXQ01 2950739 Ki = 2400 nM T16691 CO0C7J 2962174 Ki = 1900 nM T16691 C1U5AG 3028929 Ki = 6.5 nM T16691 C5F4AI 3028955 Ki = 12 nM T16691 CAM8H3 3066250 IC50 = 80 nM T16691 C6SA2G 3132842 Ki = 3400 nM T16691 C2W7DI 3142696 Ki = 163 nM T16691 CNX8I1 3245407 EC50 = 1100 nM T16691 CEG3M8 3643745 Ki = 26 nM T16691 CS8KE2 3649661 Ki = 3587 nM T16691 CKN8W0 3950432 Ki = 20 nM T16691 CRC1M5 4494260 Ki = 59 nM T16691 C6SHA4 4713248 Ki = 2600 nM T16691 CRUB15 4723431 Ki = 91 nM T16691 C9H5AV 4723679 Ki = 266 nM T16691 CSL48K 4725280 Ki = 185 nM T16691 CZ64GQ 4976400 Ki = 774 nM T16691 C7N1KM 5206725 Ki = 4489 nM T16691 C4J3HP 5640104 Ki = 5676 nM T16691 C35XAN 6484477 Ki = 316 nM T16691 C1O2PM 6625986 IC50 = 5000 nM T16691 C0QCK1 6918455 Ki = 1.259 nM T16691 CU3X9A 6918479 Ki = 0.85 nM T16691 CN5LJ4 6918531 Ki = 50 nM T16691 CW0ZE5 6918542 Ki = 2 nM T16691 CE6GX4 6918576 Ki = 25.12 nM T16691 C5V0WQ 6918577 Ki = 1.995 nM T16691 CW8OV4 6918578 Ki = 1.259 nM T16691 CEP3W2 6918579 Ki = 1.585 nM T16691 CC5PQ0 6918601 Ki = 7.2 nM T16691 C1WXY3 6918603 Ki = 1.995 nM T16691 C5GJ8Z 6918629 Ki = 1.4 nM T16691 CD0Z4I 6918648 Ki = 0.6 nM T16691 C2EJL3 6918682 Ki = 0.5 nM T16691 C8AL9V 6918689 Ki = 1 nM T16691 C0Y9VE 6918715 Ki = 0.2 nM T16691 C02GXO 6918745 Ki = 0.1259 nM T16691 CCLE83 6918748 Ki = 29 nM T16691 CI5L3H 6918751 Ki = 0.2 nM T16691 CH9GT8 6918786 Ki = 0.04 nM T16691 C2F3BY 7125890 Ki = 1574 nM T16691 CH57FQ 7183407 IC50 = 860 nM T16691 CV57DN 7184883 Ki = 2.8 nM T16691 CPX40Y 7184886 Ki = 30.2 nM T16691 CN2Z0K 7184892 IC50 = 580 nM T16691 CAV70B 7184895 IC50 = 1490 nM T16691 CG7B6O 7184976 IC50 = 1570 nM T16691 C81PDS 7185121 IC50 = 69 nM T16691 C2MGC8 7185122 IC50 = 190 nM T16691 C13EFJ 7185123 Ki = 3.2 nM T16691 CG09XB 7185124 Ki = 87.5 nM T16691 C6CDV7 7185128 IC50 = 1200 nM T16691 CD8UQ0 7246142 IC50 = 470 nM T16691 C57ZPS 7470702 IC50 = 1900 nM T16691 CUD06Z 9796627 Ki = 54 nM T16691 CFC9Y5 9799318 Ki < 1000 nM T16691 CV6PK5 9799635 Ki = 12 nM T16691 CR8GU7 9800707 Ki = 3.1 nM T16691 CL4QT6 9802776 Ki = 0.6 nM T16691 CB8Q2P 9803937 Ki = 3.162 nM T16691 CE0DI5 9804612 Ki < 6309.57 nM T16691 C89KNW 9805455 Ki = 2.512 nM T16691 CNX4F0 9805456 Ki = 1.259 nM T16691 CWOS30 9817810 Ki = 2.4 nM T16691 CPJA40 9817950 Ki = 370 nM T16691 C3BK4L 9821904 Ki = 11 nM T16691 C1JSL5 9822215 Ki = 1.5 nM T16691 CA5ID3 9822810 Ki = 0.3 nM T16691 C41ELD 9824783 Ki = 3 nM T16691 CM4I1N 9825329 Ki = 3.981 nM T16691 CR9H2E 9827562 Ki = 7.943 nM T16691 CNA93Z 9840981 Ki = 0.3 nM T16691 C4QVD7 9841077 Ki = 19 nM T16691 CTLV76 9841434 Ki = 3.8 nM T16691 C21IJU 9842551 Ki = 1 nM T16691 CI96TG 9847669 Ki = 1.995 nM T16691 CEM28L 9849116 Ki = 6.31 nM T16691 CM13ZV 9856041 Ki = 400 nM T16691 C0ZR3E 9861687 IC50 > 10000 nM T16691 CNCK78 9862256 Ki = 1.5 nM T16691 CO5YD2 9863380 Ki = 33 nM T16691 C0Q6AD 9863611 Ki = 1.995 nM T16691 C6Z9MV 9863836 Ki = 1.4 nM T16691 C9WBO2 9865474 Ki = 5.7 nM T16691 C0WBI8 9866222 Ki = 4.9 nM T16691 CG3NI8 9867263 Ki = 1.259 nM T16691 CB1F0C 9867475 Ki = 3 nM T16691 C7AB8O 9870053 Ki = 1.259 nM T16691 C2MKO6 9885426 Ki = 8.3 nM T16691 C08DBF 9885982 Ki = 4066 nM T16691 CJW1P5 9888494 Ki < 5011.87 nM T16691 C6N8UE 9889681 Ki = 0.5012 nM T16691 CM52WU 9890119 Ki = 1 nM T16691 CEG1K5 9891002 Ki = 1 nM T16691 C7QMK5 9891617 Ki = 1.259 nM T16691 CEL29O 9891618 Ki = 1 nM T16691 C3J8GU 9892409 Ki = 5.012 nM T16691 C7CD9N 9903598 Ki = 1030 nM T16691 CHFP46 9903970 Ki = 0.25 nM T16691 C9X1IV 9905247 Ki = 18 nM T16691 CUN81Q 9905249 Ki > 10000 nM T16691 C7NPZ0 9906059 Ki = 7.9 nM T16691 CYWQ50 9906447 Ki > 10000 nM T16691 CRK69H 9907512 Ki = 45 nM T16691 CAI90C 9908552 Ki = 7.9 nM T16691 CYZ5N4 9909089 Ki > 10000 nM T16691 CR52JI 9910619 Ki = 0.2 nM T16691 C9B3EA 9911844 Ki < 1000 nM T16691 C78MDV 9913554 Ki = 0.7943 nM T16691 C1IE8Y 9914461 Ki = 19.95 nM T16691 CR9KM0 9921064 IC50 = 40 nM T16691 CZQD80 9923440 Ki = 9 nM T16691 CA7RU6 9924293 Ki = 2.7 nM T16691 CMO2Y8 9924959 Ki = 2 nM T16691 C4UYZ7 9927441 Ki = 2.9 nM T16691 CV6A1D 9929294 Ki = 5 nM T16691 C9E1UB 9929665 Ki = 3.7 nM T16691 CTF52Q 9931929 Ki = 1 nM T16691 CGQ1A6 9933223 Ki = 1.7 nM T16691 CYVZ47 9934284 Ki < 1000 nM T16691 CWO45F 9935387 Ki = 0.7943 nM T16691 C6D7SX 9935750 Ki = 1.585 nM T16691 CGBP91 9945214 Ki = 58 nM T16691 CYH3R7 9947817 Ki = 1120 nM T16691 CQG0P3 9949258 Ki = 143 nM T16691 C67MTC 9950255 Ki = 0.3 nM T16691 CDKP85 9950402 Ki = 2 nM T16691 CDU68J 9952250 Ki = 8 nM T16691 CSBZ98 9953284 Ki = 1.6 nM T16691 CK8NR2 9954121 Ki = 0.631 nM T16691 CHOJ30 9956365 Ki < 1000 nM T16691 C96YVG 9956634 Ki = 0.3 nM T16691 CFR41N 9957068 Ki < 10000 nM T16691 C2CO7R 9957092 Ki = 1.995 nM T16691 CGR57X 9969402 IC50 = 7.3 nM T16691 CK9DF0 9976690 IC50 = 8.8 nM T16691 CFN50J 9978683 Ki = 1.6 nM T16691 C86FOH 9979009 Ki = 6 nM T16691 CFZ97V 9979313 Ki = 113 nM T16691 CWPT83 9979611 Ki = 0.7079 nM T16691 CRW7U6 9979748 IC50 = 12 nM T16691 C2T1WG 9983033 Ki = 27.6 nM T16691 CVOD42 9998950 IC50 = 28 nM T16691 C4BS8G 9999118 Ki = 7.3 nM T16691 CN3D2U 10019089 Ki = 0.2 nM T16691 CV7R9F 10020040 Ki > 10000 nM T16691 CU6Q5L 10020454 IC50 = 3.4 nM T16691 CK18LT 10020895 Ki > 10000 nM T16691 C8WTP3 10021389 IC50 = 70.1 nM T16691 C40IDM 10023874 Ki = 4.3 nM T16691 CB8VQ5 10024749 Ki = 15.5 nM T16691 CR9LM8 10026658 Ki = 2.13 nM T16691 CH59BP 10027190 Ki = 0.3 nM T16691 CD4J7G 10027518 Ki = 17 nM T16691 C2EUY0 10035109 Ki > 10000 nM T16691 C57TZR 10042333 Ki > 10000 nM T16691 COH3W5 10047631 Ki = 1.3 nM T16691 C8Z6MA 10067306 Ki = 2.3 nM T16691 CIK38G 10068007 Ki = 5.2 nM T16691 CD7T2M 10069527 Ki = 25.1 nM T16691 C6L3NU 10069592 Ki = 2.3 nM T16691 CV16DZ 10088284 Ki = 141 nM T16691 CZ5Y6U 10090742 IC50 = 83 nM T16691 COC0K5 10091305 IC50 = 57 nM T16691 CB0TU4 10091389 Ki = 9.6 nM T16691 C1XH8C 10091613 Ki = 8.76 nM T16691 CXF8S6 10091667 Ki = 20 nM T16691 C1SXF3 10094169 Ki = 18.3 nM T16691 CA3YF7 10094519 IC50 = 60 nM T16691 C63MGZ 10111488 Ki = 350 nM T16691 CT2X0H 10112809 Ki = 4.7 nM T16691 CJE70W 10112810 Ki = 0.4 nM T16691 CK2OR3 10112811 Ki = 4.3 nM T16691 CFO2L3 10113751 Ki = 5.3 nM T16691 C7G4BL 10113852 Ki = 163.5 nM T16691 C3NJ8W 10115005 Ki = 3 nM T16691 C8LD2B 10115854 Ki = 1 nM T16691 CXW68C 10117854 Ki = 9 nM T16691 CIB71R 10131565 Ki = 40 nM T16691 C36BMN 10134086 Ki = 0.3162 nM T16691 C0N8OY 10136185 Ki = 3 nM T16691 C2LS7U 10136837 Ki = 1 nM T16691 CQP7C9 10140915 Ki = 15 nM T16691 CAE3I7 10141477 Ki = 14 nM T16691 CET4Q9 10149997 Ki = 25.12 nM T16691 CC8RH3 10156341 Ki = 0.3981 nM T16691 CD6Y2A 10156556 Ki = 1.259 nM T16691 CCKZ54 10156876 Ki = 44 nM T16691 C7TL2R 10157412 Ki = 0.8 nM T16691 CSI1E5 10158456 Ki = 24.3 nM T16691 CT4FQ0 10159058 Ki = 4.5 nM T16691 C0GPO6 10162467 Ki = 1 nM T16691 C2J8TV 10172764 Ki = 0.34 nM T16691 CP6Q1W 10173403 Ki = 5.012 nM T16691 C2L8PI 10177503 Ki = 1.585 nM T16691 CB61DW 10177537 Ki = 7 nM T16691 CK6X9V 10178788 Ki = 0.5 nM T16691 C2AJ4U 10180527 Ki = 3.5 nM T16691 CUB5O8 10182052 Ki = 44 nM T16691 C1NLY7 10182109 Ki = 3.162 nM T16691 CQG3N5 10182228 Ki = 1 nM T16691 CFIB73 10182243 Ki = 0.1 nM T16691 CT7Q4V 10199220 Ki = 620 nM T16691 CWD43X 10199819 Ki = 3 nM T16691 CV4A2P 10201610 Ki = 1 nM T16691 C6W0YL 10202396 Ki = 5.3 nM T16691 C16DXL 10202995 Ki = 8 nM T16691 CV7S0G 10203339 Ki = 132 nM T16691 C1ET9N 10203612 Ki = 9.3 nM T16691 CW7EI0 10205655 Ki = 4 nM T16691 CFJY39 10216820 Ki = 5.012 nM T16691 CV1B7C 10217687 Ki = 10 nM T16691 CZ0TL1 10228179 Ki = 15.1 nM T16691 CI4W8Z 10246185 IC50 = 52 nM T16691 C6VO9Y 10246789 Ki = 18 nM T16691 CX85KT 10246904 IC50 = 42 nM T16691 CUHR59 10247229 IC50 = 87.6 nM T16691 CLT62K 10249280 IC50 = 68.9 nM T16691 C7MT4V 10250472 Ki = 0.6 nM T16691 CR96OK 10252130 Ki = 122 nM T16691 CSPF93 10252272 Ki = 3.981 nM T16691 CMRA02 10257042 Ki = 1995.26 nM T16691 CH31DX 10267394 Ki > 10000 nM T16691 CLG1B8 10269916 Ki = 63 nM T16691 C0T3SA 10270799 Ki = 2 nM T16691 CWV06I 10270854 Ki = 0.2512 nM T16691 CS3XW9 10272325 Ki = 5 nM T16691 CGU4I1 10272846 Ki = 10 nM T16691 C2D4BU 10273087 Ki = 1.995 nM T16691 C93SJA 10274389 Ki = 1 nM T16691 C85XYH 10275386 Ki = 6.8 nM T16691 CWQ21X 10276057 Ki = 3.3 nM T16691 C23PDE 10278839 Ki = 0.5 nM T16691 CA31LF 10286330 Ki = 1.995 nM T16691 CO2LT5 10286610 Ki = 3.981 nM T16691 C83QPR 10291754 Ki = 1 nM T16691 C7HP9C 10293741 Ki = 2.512 nM T16691 C51EXQ 10295001 Ki = 6.31 nM T16691 CAD92Z 10295665 Ki = 21.2 nM T16691 CR37BF 10296699 Ki = 163 nM T16691 CA3SK2 10297610 Ki = 3.9 nM T16691 CU89JD 10314060 Ki = 7385 nM T16691 CFQ54B 10315621 Ki = 98 nM T16691 C9U0DZ 10319296 Ki = 0.9 nM T16691 CHS1W3 10320800 Ki = 1.995 nM T16691 C04XAL 10341241 IC50 = 60 nM T16691 C8S4EN 10342674 Ki = 49 nM T16691 C9IAV3 10346043 Ki = 1 nM T16691 C4IL7N 10362440 IC50 = 79.2 nM T16691 CY8UH2 10364512 IC50 = 420 nM T16691 CR3KU9 10380133 Ki = 5.5 nM T16691 CMZA83 10383646 Ki = 1.9 nM T16691 C2P7OJ 10383682 IC50 = 0.7 nM T16691 CFAO13 10385670 IC50 = 470 nM T16691 C8L1IC 10390318 Ki = 10.3 nM T16691 CI1RB4 10405986 Ki = 3.2 nM T16691 C04WGF 10407367 Ki = 1 nM T16691 C5Y1TN 10409272 IC50 = 56 nM T16691 C4TPN1 10413595 Ki = 0.3162 nM T16691 C07AHG 10427672 IC50 = 1.3 nM T16691 CRMB96 10427673 IC50 = 41 nM T16691 C45CAU 10427896 IC50 = 22 nM T16691 CR4LS0 10430623 Ki = 1.1 nM T16691 CD7U5I 10433930 Ki = 1.995 nM T16691 CFLA92 10449488 Ki = 1 nM T16691 C3TF6V 10450930 Ki = 96 nM T16691 CN2WK7 10451504 IC50 = 11 nM T16691 C6H7GP 10452816 IC50 = 65 nM T16691 CL5J1E 10465905 Ki > 1000 nM T16691 CQD86O 10470893 IC50 = 2.4 nM T16691 COV85C 10472143 Ki = 15 nM T16691 C5LBS7 10472158 Ki = 2 nM T16691 C1UC7T 10472756 IC50 = 120 nM T16691 C26KCR 10475231 Ki > 1000 nM T16691 CEF2O6 10478367 Ki = 2410 nM T16691 C6XSG7 10480841 Ki = 200 nM T16691 CO0HE1 10498813 Ki = 10 nM T16691 CL70NJ 10499156 Ki < 10000 nM T16691 CQ4Y0V 10500364 Ki = 63.1 nM T16691 C85LRB 10505579 Ki = 1 nM T16691 CKAO03 10526615 Ki = 1.995 nM T16691 C3VLB5 10528182 Ki = 1.259 nM T16691 C75ZKM 10541285 Ki = 1258.93 nM T16691 C04EWM 10563312 Ki = 185 nM T16691 CHE80N 10573876 Ki = 3162.28 nM T16691 CN85DJ 10637020 Ki = 63.1 nM T16691 CP1UH5 10648664 Ki = 0.7943 nM T16691 CLE8P2 10658135 Ki = 24.3 nM T16691 CBRZ19 10658892 Ki = 168 nM T16691 C1Y3ON 10708918 Ki = 1000 nM T16691 C7XUR8 10713238 Ki = 20 nM T16691 C0V4PY 10757046 Ki = 200 nM T16691 C58CSG 10769116 Ki = 3.162 nM T16691 C3VTG2 10777767 Ki = 200 nM T16691 CJNM19 10800458 Ki = 240 nM T16691 CF34UD 10808841 Ki = 794.33 nM T16691 C0PE1N 10811310 Ki = 79.43 nM T16691 CD62XF 10825266 Ki = 130 nM T16691 CF3N5R 10826203 IC50 = 2 nM T16691 CNZ17B 10837078 Ki = 0.7943 nM T16691 CVT7J1 10873805 Ki = 300 nM T16691 CRI50E 10885636 IC50 = 2280 nM T16691 CX65PW 10907460 IC50 = 800 nM T16691 CNB39C 10947658 Ki = 13 nM T16691 C51NOQ 10982183 Ki ~ 0.1 nM T16691 CK6VF7 10991109 Ki = 3000 nM T16691 C4O7MD 10994400 Ki = 430 nM T16691 CM2R5C 11003533 Ki = 130 nM T16691 CJC9K4 11005810 IC50 = 427 nM T16691 C63DAE 11014674 Ki = 50.12 nM T16691 C3FIP5 11016205 Ki = 138 nM T16691 CS0Z2D 11024311 Ki = 2.291 nM T16691 CC05LI 11064294 Ki = 19.95 nM T16691 CG41BK 11071079 IC50 = 1530 nM T16691 C5AZ0I 11079889 Ki = 1700 nM T16691 C7DE0U 11113605 IC50 = 1350 nM T16691 CVE8T3 11121216 Ki = 61 nM T16691 COA02J 11154032 Ki = 9 nM T16691 CB1MG4 11154465 Ki = 1.9 nM T16691 CWS6J2 11162301 IC50 = 3580 nM T16691 CW7Y9O 11163741 Ki = 25.12 nM T16691 CX0YB7 11164580 Ki = 1 nM T16691 C8ZN3B 11166042 IC50 > 10000 nM T16691 CZ4C8S 11166043 Ki = 100.8 nM T16691 C1YA7F 11166261 Ki = 125.8 nM T16691 CV7PC9 11176859 Ki = 19.8 nM T16691 CA3Q8R 11177383 Ki = 3 nM T16691 C5U0JK 11177658 Ki = 116.2 nM T16691 C6CL1Y 11178830 Ki < 10000 nM T16691 C7YWQ1 11190151 Ki = 50.12 nM T16691 CCI40B 11190716 Ki > 1000 nM T16691 C17ZJO 11200157 EC50 = 5.2 nM T16691 C9N5QU 11200511 Ki = 1 nM T16691 C5YT1X 11200890 Ki = 0.631 nM T16691 CG7IR2 11201712 Ki > 1000 nM T16691 CPDU74 11201726 IC50 = 1.6 nM T16691 CAN97Q 11210467 EC50 = 1.4 nM T16691 C7ESF4 11210523 Ki > 1000 nM T16691 C94AIS 11211722 Ki = 1 nM T16691 C6D1MZ 11223004 EC50 = 1.3 nM T16691 CR04PZ 11232643 Ki = 4500 nM T16691 CD9XA5 11234629 EC50 = 0.8 nM T16691 C5XGC0 11234781 Ki = 57.7 nM T16691 CZE1A5 11235953 Ki = 10 nM T16691 COE13K 11236269 Ki = 9.8 nM T16691 CC4RT3 11237275 Ki > 1000 nM T16691 C1E0SQ 11245641 Ki = 4 nM T16691 CE97VF 11246907 Ki = 1 nM T16691 C90WSG 11248705 Ki < 10000 nM T16691 CBUP32 11257897 Ki = 41.2 nM T16691 CQ90VJ 11258709 Ki = 74.5 nM T16691 CZD6N4 11259180 Ki = 74.6 nM T16691 CI84OD 11259419 Ki = 90.2 nM T16691 CGJK46 11259456 Ki > 1000 nM T16691 CAU5P1 11260183 Ki = 1 nM T16691 C2VKI7 11269402 Ki = 64.7 nM T16691 CJNT47 11270131 Ki = 140.5 nM T16691 C7G8HX 11270546 Ki = 165.9 nM T16691 CQZE84 11271219 Ki = 31.4 nM T16691 CW7A0S 11280663 Ki = 1 nM T16691 C4JTQ3 11280771 Ki = 131 nM T16691 CM54IK 11282295 Ki = 194.8 nM T16691 C9HYZ8 11282389 Ki = 18.4 nM T16691 CTH8D9 11282884 IC50 = 1.1 nM T16691 CNZ23G 11283016 Ki = 224.4 nM T16691 CDRV20 11294169 Ki > 1000 nM T16691 C9BLC7 11304596 Ki = 3162.28 nM T16691 CJS9C0 11304851 IC50 > 7900 nM T16691 C30MTX 11306131 Ki = 336 nM T16691 CI79LV 11307899 Ki = 50.12 nM T16691 CZ0RP8 11314681 Ki = 1 nM T16691 C8Y7ZH 11316095 Ki = 1 nM T16691 CV6D3C 11316536 Ki = 12 nM T16691 CC9TE2 11316594 EC50 = 4.2 nM T16691 C46YHW 11316967 Ki = 9.6 nM T16691 C4Y5FE 11317551 Ki = 7.2 nM T16691 CW67JC 11326086 Ki = 0.9 nM T16691 CQ81DR 11328408 Ki > 1000 nM T16691 CL7QR0 11333554 EC50 = 130 nM T16691 CR89ME 11338273 Ki = 36 nM T16691 C42HTF 11338378 Ki = 14.9 nM T16691 CF6D5Z 11350253 Ki = 5.7 nM T16691 C1QKY2 11351089 Ki = 0.4 nM T16691 CGD42N 11361090 IC50 = 0.4 nM T16691 CWO59Z 11362134 Ki = 18.6 nM T16691 CY27GK 11363934 Ki = 0.3 nM T16691 CHB4E1 11371056 Ki = 1.2 nM T16691 C9QTU4 11372111 Ki = 16 nM T16691 CKF72Y 11383202 Ki = 4 nM T16691 C76EVG 11383990 Ki = 34 nM T16691 CBV52J 11384146 Ki = 0.4 nM T16691 CR46IF 11384675 Ki = 51.7 nM T16691 CX54VZ 11384694 Ki = 151.9 nM T16691 C1W7MS 11385064 Ki = 1 nM T16691 CJ74CP 11396708 IC50 = 0.8 nM T16691 CF4OX6 11397149 Ki = 316.23 nM T16691 C7MD9R 11406161 Ki = 4 nM T16691 CQ87XW 11407072 Ki = 0.3162 nM T16691 CM7I9Q 11407151 Ki = 85.8 nM T16691 CBV7Q8 11407544 Ki = 35 nM T16691 CK0FG2 11407867 Ki = 3 nM T16691 C1AYG7 11408932 Ki = 107.4 nM T16691 CR49LD 11408954 Ki > 1000 nM T16691 CK1A9Y 11417978 Ki = 94.2 nM T16691 C4X7AS 11418830 Ki = 3 nM T16691 CHV83P 11419238 Ki = 1 nM T16691 CB51AS 11420098 Ki = 108.8 nM T16691 C0FP4Z 11429601 Ki = 22 nM T16691 C85LYP 11430418 IC50 > 1000 nM T16691 CDWV48 11430512 Ki = 246.2 nM T16691 C6KHG1 11440676 Ki = 3 nM T16691 CY9B8H 11441064 Ki = 11 nM T16691 CV84SK 11441983 Ki = 7 nM T16691 C0L5RN 11442097 Ki = 124.5 nM T16691 C16DOF 11451904 Ki = 1 nM T16691 C6AF5E 11452988 Ki = 4 nM T16691 COH39T 11453792 Ki = 1 nM T16691 CD5FG4 11463428 EC50 = 1 nM T16691 CE7JU3 11463924 Ki = 123.6 nM T16691 CG75FW 11464995 Ki = 131.3 nM T16691 C24SNG 11474995 Ki = 1 nM T16691 CPS97N 11475760 Ki = 55.2 nM T16691 C59GHW 11476019 Ki = 24 nM T16691 CYJQ37 11476494 Ki = 97.3 nM T16691 CO6N3B 11486933 Ki = 1 nM T16691 CIWO57 11501251 Ki = 462 nM T16691 CO97GC 11501432 Ki = 346 nM T16691 CJK63T 11503175 Ki = 0.7943 nM T16691 CLU4R7 11504338 Ki > 1000 nM T16691 CIFQ02 11508173 Ki = 715 nM T16691 C7YD0A 11515129 Ki = 728 nM T16691 CD8I9H 11515192 Ki = 0.3162 nM T16691 CHK79E 11522477 Ki = 409 nM T16691 C6O9PM 11522698 Ki = 1013 nM T16691 C70RAX 11524473 IC50 = 0.8 nM T16691 CG0D5S 11532574 Ki = 4 nM T16691 CY4R9L 11545169 Ki = 3.6 nM T16691 C1V5CH 11559090 Ki = 30.1 nM T16691 CGP56Q 11559141 Ki = 164 nM T16691 CT1DE9 11560362 Ki = 304 nM T16691 C4TI1E 11566597 Ki = 0.4 nM T16691 CJ9UY6 11566775 Ki > 1000 nM T16691 CEM42D 11567716 Ki = 196.9 nM T16691 C25RSU 11567840 Ki = 77.5 nM T16691 CK3F1Y 11569025 Ki = 0.3 nM T16691 CO58PR 11573559 Ki = 156 nM T16691 CE23IV 11574113 Ki = 28.3 nM T16691 CBW12V 11574663 Ki = 9.2 nM T16691 C8NMI4 11575479 Ki = 82.4 nM T16691 C6D1MA 11584660 Ki > 1258.93 nM T16691 CN21IG 11587610 Ki = 0.3 nM T16691 C1M2CP 11589069 Ki = 580 nM T16691 CU45DK 11595209 Ki = 12.3 nM T16691 CV9B8R 11595360 Ki = 0.1585 nM T16691 CGX8F6 11596869 Ki > 1790000 nM T16691 C21XTO 11601657 Ki > 1000 nM T16691 CVQ4R6 11601955 Ki = 108 nM T16691 CN2F6O 11603453 Ki = 928 nM T16691 COY20C 11609368 Ki = 344.6 nM T16691 C4J6KG 11616729 Ki > 1000 nM T16691 C6V3OY 11624561 Ki = 0.3 nM T16691 CCK08F 11630209 Ki > 1000 nM T16691 CK6U7Q 11630824 Ki = 481 nM T16691 CHS76B 11631738 Ki = 877 nM T16691 CCY41R 11631819 Ki = 0.4 nM T16691 COH4T9 11632439 Ki = 19 nM T16691 COL12H 11638206 Ki = 27 nM T16691 C2OU7Y 11638332 Ki = 54.7 nM T16691 CD84ZC 11639865 Ki = 0.1995 nM T16691 CJ8ZS6 11640142 Ki > 1000 nM T16691 CV49QH 11652654 Ki = 0.2 nM T16691 C1HDM5 11653679 Ki = 295.9 nM T16691 C3KMW6 11653799 Ki > 1000 nM T16691 C5YC4N 11654089 Ki > 1000 nM T16691 C9X6PO 11661320 Ki = 1284 nM T16691 CE0C3N 11667340 Ki = 172 nM T16691 CRKQ54 11674694 Ki = 147 nM T16691 C8BNM7 11681803 Ki = 257 nM T16691 CRU61B 11682024 Ki = 0.3162 nM T16691 CB95CX 11683768 Ki = 952 nM T16691 CML4E8 11688736 Ki = 0.631 nM T16691 CZM75X 11689373 Ki = 1.259 nM T16691 C93ACF 11695841 Ki = 59 nM T16691 C23VNU 11697242 Ki = 0.3981 nM T16691 C2Q6TW 11703226 Ki = 73.2 nM T16691 C4G1EZ 11709684 Ki = 23 nM T16691 CG87CL 11716331 Ki = 1365 nM T16691 CV69CM 11723168 Ki = 3 nM T16691 CC37TI 11724023 IC50 = 2 nM T16691 C0NH2T 11724112 IC50 = 12 nM T16691 CP0QV2 11725253 IC50 = 250 nM T16691 CQA4Y1 11725505 Ki = 1.6 nM T16691 CY1XU6 11729763 Ki = 320 nM T16691 CLYJ75 11729823 Ki = 48.9 nM T16691 C7PVL8 11730467 IC50 = 7780 nM T16691 CMO0I9 11739679 IC50 = 0.8 nM T16691 C2GK7T 11740084 IC50 = 700 nM T16691 C57IKL 11740526 Ki < 1000 nM T16691 CKD26I 11741319 IC50 = 50 nM T16691 CC18PB 11741686 IC50 = 18 nM T16691 C5H0YJ 11743064 IC50 = 126 nM T16691 CPG15O 11743399 IC50 > 1000 nM T16691 CBA17C 11744377 Ki = 10.2 nM T16691 CYV02C 11747350 Ki = 20 nM T16691 C9WO6G 11749539 Ki = 1 nM T16691 CA61BD 11750876 Ki = 57 nM T16691 C3CN0Y 11772625 Ki = 1 nM T16691 CUD91G 11775364 Ki = 8 nM T16691 C0WB7U 11811724 Ki = 490 nM T16691 CAC74F 11820174 Ki = 300 nM T16691 CG3QJ4 11833220 Ki = 260 nM T16691 CZ7Y1I 11849203 Ki = 38 nM T16691 CI4PE1 11849204 Ki = 17 nM T16691 CR8EY5 11849745 Ki = 52 nM T16691 CO0H2M 11849787 Ki = 15 nM T16691 CXLW54 11948707 Ki > 10000 nM T16691 C8JQL7 11957735 IC50 > 10000 nM T16691 C1H2GL 11961315 Ki = 1.7 nM T16691 CSE5A4 11983287 Ki = 1.2 nM T16691 C1QY2P 12005903 Ki = 119 nM T16691 CWE19J 12017572 Ki = 7.4 nM T16691 C2L0RA 12017573 Ki = 9.5 nM T16691 C7RUD8 12017574 Ki = 45 nM T16691 C5TY3Z 12017575 Ki = 93 nM T16691 CV9PF5 12017576 Ki = 183 nM T16691 C9ED3P 12017577 Ki = 5 nM T16691 C5J2UM 12017578 Ki = 154 nM T16691 C6AJ4F 12017579 Ki = 8000 nM T16691 CG56FM 12017580 Ki = 19600 nM T16691 CK28MT 12051078 Ki = 136 nM T16691 CUW18O 12051079 Ki = 300 nM T16691 C8EDN0 12088080 Ki > 1000 nM T16691 C8RB6W 12088082 Ki > 1000 nM T16691 C1QM4J 12147013 Ki = 20 nM T16691 C9RBT8 12147017 Ki = 16 nM T16691 CMH17C 12148615 Ki = 1.8 nM T16691 CEIP49 15480742 Ki = 60 nM T16691 C30CHU 15512229 Ki < 316.23 nM T16691 COWE74 15619875 IC50 = 10 nM T16691 C5QS1J 16019286 IC50 = 1120 nM T16691 CM1EL8 16019288 IC50 = 170 nM T16691 CRM1F0 16019292 Ki = 3.5 nM T16691 C68NQM 16019303 IC50 = 730 nM T16691 CW49DH 16019305 IC50 = 1250 nM T16691 CH03IC 16019310 IC50 = 740 nM T16691 CF0VH8 16019312 IC50 = 220 nM T16691 C1RMU0 16019339 IC50 = 350 nM T16691 CWQ67Z 16019343 IC50 = 820 nM T16691 C0E2AF 16019364 IC50 = 520 nM T16691 CSB0U1 16019366 IC50 = 90 nM T16691 CQTK41 16019372 IC50 = 270 nM T16691 C0PTX8 16019394 IC50 = 960 nM T16691 CTMC92 16019397 IC50 = 650 nM T16691 C8S6VI 16019451 IC50 = 1050 nM T16691 CG5I6Q 16019453 IC50 = 1600 nM T16691 CVW2H6 16019490 IC50 = 1930 nM T16691 C7V4MI 16019508 IC50 = 28.3 nM T16691 CXZ4T7 16019510 IC50 = 1520 nM T16691 CBK40Y 16019514 IC50 = 590 nM T16691 C9IYN1 16019519 IC50 = 710 nM T16691 CD7WK0 16019546 IC50 = 59 nM T16691 CZF0S6 16019548 IC50 = 1170 nM T16691 C4A8GT 16019550 IC50 = 170 nM T16691 C7R0QS 16019553 Ki = 15.9 nM T16691 CHB62Y 16019573 Ki = 28.8 nM T16691 C8GC1T 16019574 IC50 = 690 nM T16691 CL0OT3 16019576 Ki = 1.7 nM T16691 C7T6GI 16019580 Ki = 2.3 nM T16691 C7TP3J 16019601 IC50 = 260 nM T16691 CXMY18 16019602 IC50 = 2010 nM T16691 C3WQ1G 16019604 IC50 = 960 nM T16691 CEP4U1 16019607 IC50 = 1220 nM T16691 CY1JE9 16019609 IC50 = 180 nM T16691 CX2CT6 16019610 IC50 = 140 nM T16691 CL1C5P 16023081 Ki = 88 nM T16691 C3M8GJ 16026344 Ki = 13330 nM T16691 CWY3F2 16037746 Ki = 0.8 nM T16691 CS07QC 16040768 Ki = 32 nM T16691 CX54GY 16049388 Ki = 5.44 nM T16691 CJ1T0W 16070169 Ki = 4.3 nM T16691 CXWC93 16071727 Ki = 6.7 nM T16691 C1SR0O 16071847 Ki = 1.5 nM T16691 CQS4V1 16112801 EC50 = 0.9 nM T16691 CC6Y3J 16116896 Ki = 17 nM T16691 CQ0VT5 16116897 Ki = 28 nM T16691 CA7L8M 16116898 Ki = 9.8 nM T16691 CV6G9J 16116899 Ki = 4.2 nM T16691 C2ATQ4 16116900 Ki = 9.5 nM T16691 CZ1WJ4 16117151 Ki = 1 nM T16691 C4PEY7 16117152 Ki = 2.3 nM T16691 CM32ZX 16117153 Ki = 0.6 nM T16691 CFB1T7 16117154 Ki = 6.7 nM T16691 CJ6D1M 16117278 Ki = 6.3 nM T16691 CXTB90 16117279 Ki = 1 nM T16691 CA23RS 16117280 Ki = 1.5 nM T16691 C8M5KE 16117281 Ki = 3.1 nM T16691 CU9VB2 16117282 Ki = 9.8 nM T16691 C2HI3Q 16117283 Ki = 0.8 nM T16691 C1F2LS 16118795 Ki = 0.7 nM T16691 CT0S9V 16118796 Ki = 3.5 nM T16691 C1BPY5 16118797 Ki = 1.7 nM T16691 C69VDS 16118923 Ki = 1.1 nM T16691 CA0IB2 16118924 Ki = 53 nM T16691 C5DVW2 16118925 Ki = 57 nM T16691 CK4Y1C 16118926 Ki = 44 nM T16691 C76QZH 16118927 Ki = 31 nM T16691 C0PMY8 16118928 Ki = 30 nM T16691 C8OF0W 16118929 Ki = 66 nM T16691 CJ1N3M 16222447 Ki = 15.5 nM T16691 C50ZXQ 16222448 Ki = 8.82 nM T16691 CN16GL 16222450 Ki = 8.28 nM T16691 CGPY68 16222545 Ki = 4.21 nM T16691 C46VQT 16222547 Ki = 1.92 nM T16691 CQ9YZ4 16222548 Ki = 20.4 nM T16691 CK0IB2 16222549 Ki = 1.83 nM T16691 C89XDO 16222651 Ki = 7.5 nM T16691 CSO7W8 16222652 Ki = 5.5 nM T16691 CQC5D4 16222654 Ki = 28.99 nM T16691 CBU75J 16222655 Ki = 16.1 nM T16691 C9HOC0 16222656 Ki = 12.2 nM T16691 C79ADX 16222758 Ki = 18.09 nM T16691 CHOC30 16222759 Ki = 41.1 nM T16691 C5E6MS 16222761 Ki = 15.7 nM T16691 C4HBK5 16222762 Ki = 32.4 nM T16691 CE75KN 16222763 Ki = 15.5 nM T16691 CG8Y3L 16222764 Ki = 43.5 nM T16691 C4XV1Q 16222865 Ki = 32.8 nM T16691 CA2ZJ1 16222866 Ki = 5.89 nM T16691 CQN9G1 16222867 Ki = 19.8 nM T16691 CSJ4H8 16222868 Ki = 15.1 nM T16691 CE0LY9 16222869 Ki = 3.71 nM T16691 C2LDY6 16222870 Ki = 4.57 nM T16691 C1TC5B 16222871 Ki = 13.8 nM T16691 CA6MU9 16222962 Ki = 24.9 nM T16691 CE7QA0 16222963 Ki = 8.13 nM T16691 C9PTN1 16222965 Ki = 7.95 nM T16691 CXZ41D 16223064 Ki = 6.89 nM T16691 CBT9C0 16223065 Ki = 2.68 nM T16691 CN9I4S 16223066 Ki = 24.3 nM T16691 CZ2IS9 16660294 Ki > 10000 nM T16691 C1CER8 16718822 Ki = 17 nM T16691 CD3Q2U 16718826 Ki = 216 nM T16691 C3JV0P 16718827 EC50 = 3.2 nM T16691 C8GOW7 16718869 Ki = 20 nM T16691 C0JQ5W 16718916 Ki = 276 nM T16691 C3YN5S 16718917 EC50 = 0.3 nM T16691 CJ8Y1H 16718919 Ki = 18 nM T16691 CB7G3R 16718920 EC50 = 0.3 nM T16691 C8U4LQ 16718921 Ki = 31 nM T16691 C5MT4H 16718922 Ki = 3 nM T16691 CW03YI 16750338 Ki = 3.8 nM T16691 CT9GP4 16763549 Ki = 2945 nM T16691 C81DEA 16804502 IC50 = 1150 nM T16691 C2F7IH 16956087 IC50 = 540 nM T16691 CZ97JQ 16956089 IC50 = 580 nM T16691 CC8EA5 16956204 IC50 = 930 nM T16691 CR63LE 17055181 Ki = 5100 nM T16691 C0QX5J 17374371 Ki = 11980 nM T16691 CB2J3R 17747575 IC50 > 100 nM T16691 C3BVJ4 17940055 Ki = 31.62 nM T16691 C5D0HA 17940058 Ki = 1.585 nM T16691 CLZ60J 17940080 Ki = 19.95 nM T16691 C1M5VA 17940089 Ki = 1.995 nM T16691 C3UI5Y 17940101 Ki = 0.7943 nM T16691 CBC70F 17940113 Ki = 1.259 nM T16691 CQ96ZT 17940121 Ki = 3.981 nM T16691 C0UE9W 17940125 Ki = 0.3162 nM T16691 C8KJ1Y 17940155 Ki = 1.259 nM T16691 CF46WY 17940169 Ki = 0.5012 nM T16691 CN5G0Y 17940185 Ki = 25.12 nM T16691 CELX94 17940199 Ki = 1.259 nM T16691 C2G6ID 17940212 Ki = 0.631 nM T16691 C6IK5X 17940215 Ki = 0.5012 nM T16691 CG5CO7 17940224 Ki = 1 nM T16691 C92SPR 17940228 Ki = 2.512 nM T16691 CGUS59 17940234 Ki = 7.943 nM T16691 CUS47A 17940243 Ki = 3.162 nM T16691 C6ZM7X 17940245 Ki = 1.995 nM T16691 CL2AS8 17940260 Ki = 1.585 nM T16691 CQC56I 17940268 Ki = 5.012 nM T16691 C9L0AZ 17960999 Ki = 0.3981 nM T16691 CQM7R1 17961002 Ki = 0.631 nM T16691 CR10MN 17961003 Ki = 7.943 nM T16691 CC5SW2 17978373 Ki = 0.3162 nM T16691 C0OL1J 17978376 Ki = 5.012 nM T16691 CH2X5U 17978385 Ki = 25.12 nM T16691 C54VGS 17978406 Ki = 7.943 nM T16691 C3RK0S 17978408 Ki = 0.3162 nM T16691 C6D0PK 18180040 Ki = 2.3 nM T16691 C9PV8A 18180076 IC50 = 13 nM T16691 C6S4JR 18180095 Ki = 1.6 nM T16691 CTA6O3 18180191 Ki = 0.7943 nM T16691 CIZ3C8 18354536 Ki = 0.5012 nM T16691 CXRQ53 18354548 Ki = 0.7943 nM T16691 CHP5L8 18354552 Ki = 3.981 nM T16691 CFT01Z 18354557 Ki = 3.162 nM T16691 C9U3NH 18354572 Ki = 3.981 nM T16691 C2Z9MB 18354574 Ki = 2.512 nM T16691 C37TAU 18354589 Ki = 1.259 nM T16691 CY3P0B 18354590 Ki = 3.981 nM T16691 CV0X4I 18559283 IC50 = 1110 nM T16691 CY0G5A 18559285 IC50 = 890 nM T16691 C0NV6X 18559286 IC50 = 860 nM T16691 C7PKF0 18559353 IC50 = 900 nM T16691 C5LV1E 18559939 IC50 = 5220 nM T16691 CN20SE 18559973 IC50 = 1750 nM T16691 CK74OE 18560047 IC50 > 5000 nM T16691 CC36OB 18560059 IC50 = 1100 nM T16691 CQ4N8G 18560060 IC50 = 1480 nM T16691 CRK34J 18560180 IC50 = 1160 nM T16691 CYWK26 18560181 IC50 = 32 nM T16691 CU93YN 18560182 IC50 = 290 nM T16691 CG56OA 18560184 IC50 = 790 nM T16691 CP24LD 18560186 IC50 = 300 nM T16691 CBH94P 18560202 IC50 = 1380 nM T16691 CW42ZS 18560255 IC50 = 860 nM T16691 COR6X7 18560317 IC50 = 600 nM T16691 C42VJM 18560324 IC50 = 680 nM T16691 CX8HE9 18560325 IC50 = 1330 nM T16691 CE8W5B 18560538 IC50 = 37 nM T16691 C8MWB9 18560539 IC50 = 1370 nM T16691 CP0A5C 18560541 IC50 = 1080 nM T16691 CMPY53 18560542 IC50 = 2030 nM T16691 C7YAO8 18560556 IC50 = 410 nM T16691 C49VTO 18560559 IC50 = 1150 nM T16691 C5SN1R 18560562 IC50 = 280 nM T16691 C6QOH2 18560564 IC50 = 570 nM T16691 C1OL5W 18590273 IC50 = 1190 nM T16691 CRLJ91 18590409 IC50 = 1000 nM T16691 C0J3WX 18590411 IC50 = 1620 nM T16691 C0CAW5 18590413 IC50 = 1950 nM T16691 C2OU9R 18590416 IC50 = 1350 nM T16691 C5VI2L 18590836 IC50 = 3810 nM T16691 CL5BA2 18591074 IC50 = 1430 nM T16691 CD2OR9 18591266 IC50 = 820 nM T16691 C46POT 18591267 IC50 = 780 nM T16691 C3URK4 18591268 IC50 = 29 nM T16691 C9AYF3 18591269 IC50 = 110 nM T16691 C1RCK3 18591271 IC50 = 480 nM T16691 CT01XH 18591272 IC50 = 2500 nM T16691 C7T8JC 19958494 Ki = 7109.5 nM T16691 C6LI5E 19958507 Ki = 4460.7 nM T16691 C0FAH6 20042470 Ki = 9.3 nM T16691 COBR80 20765662 Ki = 1.995 nM T16691 C9ZE0I 20765664 Ki = 0.631 nM T16691 CKNR40 20765669 Ki = 0.5012 nM T16691 CDXS17 20765678 Ki = 12.59 nM T16691 CBY03N 20846175 Ki = 54.95 nM T16691 CEV21N 20901114 IC50 = 1990 nM T16691 CEV8G2 20901115 Ki = 8.1 nM T16691 C25LZY 20901117 Ki = 5.5 nM T16691 CD7TG3 20901118 IC50 = 290 nM T16691 C3KBJ9 20901120 IC50 = 260 nM T16691 C4A1ZK 20901122 IC50 = 600 nM T16691 CK97WL 20901124 IC50 = 820 nM T16691 C13UBY 20901125 IC50 = 500 nM T16691 C1OP7Q 20901126 IC50 = 580 nM T16691 CY9W8X 20901128 IC50 = 250 nM T16691 CNG3I6 20901131 IC50 = 2210 nM T16691 CGZB95 20901132 IC50 = 2030 nM T16691 CH10OK 20901133 IC50 = 590 nM T16691 CGK3J2 20901136 IC50 = 770 nM T16691 CHCW87 20901139 IC50 = 470 nM T16691 CT0C4W 20901141 IC50 = 46 nM T16691 CIT1E8 20901142 IC50 = 750 nM T16691 C2KBV6 20901145 IC50 = 2380 nM T16691 CLF4Y5 20901160 IC50 = 480 nM T16691 CBK05L 20901163 IC50 = 2170 nM T16691 CY3BN2 20901164 IC50 > 5000 nM T16691 C2TRE0 20901169 IC50 = 800 nM T16691 C5MQ0H 20901172 IC50 = 1830 nM T16691 CVG42R 20901177 IC50 > 5000 nM T16691 C2BVW3 20901182 IC50 > 5000 nM T16691 C4MFW3 20901183 IC50 > 5000 nM T16691 CT7FU4 20901186 IC50 = 590 nM T16691 C27ZYB 20901203 IC50 > 5000 nM T16691 CVE0S9 20901207 Ki = 46 nM T16691 C1R9XF 20901210 IC50 = 670 nM T16691 CD3E7L 20901217 IC50 = 170 nM T16691 CGAH45 20901220 IC50 = 1290 nM T16691 CUV3F8 20901229 IC50 = 610 nM T16691 C0OIT1 20901240 IC50 > 5000 nM T16691 CQ4W3Y 20901253 IC50 = 690 nM T16691 CWA26O 20901254 IC50 = 190 nM T16691 CB5D8X 20901255 IC50 = 1040 nM T16691 CLU06V 20901258 IC50 = 1540 nM T16691 C12EZR 20901259 IC50 = 68 nM T16691 CE45NR 20901261 IC50 = 150 nM T16691 CX8EI0 20901263 IC50 = 540 nM T16691 CP0K5O 20901264 IC50 = 60 nM T16691 CEL9U6 20901265 IC50 = 69 nM T16691 CKE98H 20901266 IC50 = 150 nM T16691 C9Z5WA 20901267 IC50 = 2000 nM T16691 CERG41 20901268 IC50 = 150 nM T16691 C5ZRC0 20901270 IC50 = 920 nM T16691 CO0PH4 20901271 IC50 = 1210 nM T16691 C9LWB8 20901273 IC50 = 1070 nM T16691 C5DG2K 20901275 IC50 = 740 nM T16691 CS9Q4E 20901291 IC50 = 1220 nM T16691 C6H9WC 21092408 Ki = 41858718 nM T16691 C0CA1J 21254909 Ki = 16.6 nM T16691 C3T5HF 21509921 Ki = 154.88 nM T16691 CUO9Q1 21512050 IC50 = 40 nM T16691 CG21AX 21514234 Ki = 64 nM T16691 C4B0TN 21557475 Ki = 1966 nM T16691 C36XOS 22028185 Ki = 22 nM T16691 C5JL1M 22028187 Ki = 200 nM T16691 CYS15E 22028199 Ki = 368 nM T16691 CBN84K 22065997 Ki > 10000 nM T16691 C6UXL4 22330705 Ki = 11360 nM T16691 C6G7ZE 22424009 IC50 = 9.6 nM T16691 CZG9S2 22425072 Ki = 6505 nM T16691 CBL97U 22504458 IC50 = 21 nM T16691 CPD8Q7 22549784 Ki = 16550 nM T16691 CAUH46 22557214 Ki = 1.995 nM T16691 C1T4AB 22557219 Ki = 39.81 nM T16691 CAXR08 22557224 Ki = 199.53 nM T16691 CBN2M3 22557235 Ki = 0.0631 nM T16691 C5VA1T 22557241 Ki = 0.1585 nM T16691 CIRF78 22557257 Ki = 10 nM T16691 C03XCL 22557272 Ki = 0.3981 nM T16691 C9W5CD 22557286 Ki = 316.23 nM T16691 CMN2J0 22557287 Ki = 2.512 nM T16691 CH12KP 22557292 Ki = 3.162 nM T16691 C8NR3D 22662986 Ki = 64 nM T16691 CZ7J4B 22857296 Ki = 400 nM T16691 CDL7A8 23288143 Ki = 99 nM T16691 CO1NA8 23624297 Ki = 11.8 nM T16691 CPX21U 23624307 Ki = 0.5 nM T16691 CLI4F8 23624309 Ki = 3.1 nM T16691 CJ2W3A 23625763 Ki = 1 nM T16691 CA5QC2 23625764 Ki = 2.399 nM T16691 CXD3E6 23625925 Ki = 630.96 nM T16691 CJ18ET 23652557 Ki = 10.8 nM T16691 CIY3P0 23652635 Ki = 8.6 nM T16691 CCL15O 23652787 Ki = 9.2 nM T16691 C3YBE2 23652788 Ki = 10.2 nM T16691 CSIP14 23652790 Ki = 10.6 nM T16691 C76LZN 23652861 Ki = 30.1 nM T16691 C4BXD0 23652863 Ki = 82.3 nM T16691 CV74XB 23652922 Ki = 55.3 nM T16691 CKI17V 23652993 Ki = 20.3 nM T16691 CE24HU 23652994 Ki = 30.5 nM T16691 CR6PO0 23653062 Ki = 10.7 nM T16691 CF7VS8 23653130 Ki = 63.5 nM T16691 C6J3NA 23653133 Ki = 15.2 nM T16691 CKW7V5 23653135 Ki = 3.4 nM T16691 CY9TE3 23655287 Ki = 11 nM T16691 C5I8BA 23655288 Ki = 16 nM T16691 CQL1O9 23655289 Ki = 6 nM T16691 C92TKG 23655290 Ki = 21 nM T16691 C5ZH1E 23655462 Ki = 10 nM T16691 C4I2PZ 23655463 Ki = 14 nM T16691 CA29ZB 23655464 Ki = 47 nM T16691 CU6Y4G 23655465 Ki = 1 nM T16691 CEMW69 23655466 Ki = 30 nM T16691 CS1B3A 23655467 Ki = 7 nM T16691 CLD3F4 23655468 Ki = 6 nM T16691 CFRH01 23655469 Ki = 7 nM T16691 CA03MU 23655664 Ki = 31 nM T16691 CNU2X4 23725134 Ki = 1.6 nM T16691 CVLG35 23757269 Ki = 6 nM T16691 CGD1E3 23757270 Ki = 0.8 nM T16691 CN36KF 23786472 Ki = 43 nM T16691 C9KL1S 23815446 Ki = 230 nM T16691 CVE1R9 23815447 Ki = 3 nM T16691 CG6L3F 23844114 Ki = 0.6 nM T16691 C0KM6Q 23872163 Ki = 27 nM T16691 C37QMN 23872164 Ki = 0.6 nM T16691 CC9XE5 23900125 Ki = 34 nM T16691 CQE1N7 23906630 Ki = 5826 nM T16691 CEA76H 23955921 Ki = 90 nM T16691 C7Y6VG 24763349 Ki = 9.6 nM T16691 CT9HL7 24763350 Ki = 55 nM T16691 C4JZ8U 24763351 Ki = 93 nM T16691 CC1N3K 24763352 Ki = 19 nM T16691 CT8BO3 24763353 Ki = 66 nM T16691 CQ64TA 24763354 Ki = 50 nM T16691 CXI4H2 24763355 Ki = 46 nM T16691 CH1UL9 24763429 Ki = 48 nM T16691 CX7CL6 24763430 Ki = 14 nM T16691 CR89US 24768515 Ki = 10.3 nM T16691 CD7CV6 24771120 Ki = 2.3 nM T16691 CGF70N 24771124 Ki = 15 nM T16691 CC6L2F 24771185 Ki = 18 nM T16691 C89WOM 24776044 Ki = 7.92 nM T16691 C0R4EZ 24776942 Ki = 1.8 nM T16691 CV09KG 24777061 Ki = 49 nM T16691 CNWQ34 24777062 Ki = 90 nM T16691 C9E2MV 24777063 Ki = 220 nM T16691 CCEH06 24781896 IC50 > 100 nM T16691 CD86PT 24781897 IC50 > 100 nM T16691 CP7TJ3 24781898 IC50 > 100 nM T16691 CF17PW 24781899 IC50 > 100 nM T16691 C1JSY8 24781900 IC50 > 100 nM T16691 CJI2O1 24782049 IC50 > 100 nM T16691 CK9T1F 24782050 IC50 > 100 nM T16691 C2O7MV 24782051 IC50 > 100 nM T16691 C0G3RV 24782052 IC50 > 100 nM T16691 CR8DV4 24782058 IC50 > 100 nM T16691 CYR67K 24783294 Ki = 7.1 nM T16691 CW20VF 24783295 Ki = 52 nM T16691 C8B7EG 24783296 Ki = 196 nM T16691 C8UQF0 24783550 Ki = 13 nM T16691 CULV50 24783808 Ki = 13 nM T16691 C9LDH4 24783809 Ki = 9.7 nM T16691 C0VKE6 24783810 Ki = 12 nM T16691 CYAU35 24784066 Ki = 41 nM T16691 CN2W9R 24784069 Ki = 54 nM T16691 C38VPE 24784321 Ki = 64 nM T16691 C37OYB 24784323 Ki = 31 nM T16691 CX3KC0 24784325 Ki = 22 nM T16691 CJ73UQ 24784573 Ki = 22 nM T16691 CU40PB 24784575 Ki = 25 nM T16691 CI9T6E 24784577 Ki = 36 nM T16691 C69JES 24784578 Ki = 88 nM T16691 CN52JE 24784824 Ki = 72 nM T16691 C3JSR4 24794436 IC50 = 53 nM T16691 C58AMS 24829343 Ki = 186.5 nM T16691 CDC91N 24839550 Ki = 1737.8 nM T16691 CUW23K 24854106 Ki = 1800 nM T16691 C6BSX7 24855787 Ki = 27.8 nM T16691 C4LC2K 24855826 Ki > 1000 nM T16691 C7ZOP1 24855830 Ki > 1000 nM T16691 CGHZ87 24855831 Ki = 92 nM T16691 C7ZEF0 24856058 Ki = 2.56 nM T16691 CU90ZK 24861250 Ki = 434 nM T16691 C3HK0J 24865725 Ki > 10000 nM T16691 C0O6FX 24865727 Ki = 1584.89 nM T16691 CT7Z5L 24873459 Ki = 0.1995 nM T16691 C6L7KS 24887518 Ki < 3162.28 nM T16691 CI53SE 24893978 Ki = 4100 nM T16691 CJ63YQ 24894055 Ki = 19 nM T16691 CAOF91 24894071 IC50 > 10000 nM T16691 C5EIW1 24965329 Ki = 3.24 nM T16691 CVYJ09 24965330 Ki = 23.41 nM T16691 C5YX0U 24965331 Ki = 8.58 nM T16691 C5S7UA 24965678 Ki = 11.13 nM T16691 C6U2AP 24965679 Ki = 1.43 nM T16691 CY3BJ4 24965680 Ki = 9.89 nM T16691 CFM8C2 24965681 Ki = 29.15 nM T16691 C91FZJ 24966378 Ki = 30.28 nM T16691 CCGJ63 24966381 Ki = 122 nM T16691 CBK7U0 24966733 Ki = 75.3 nM T16691 CG96KI 24966734 Ki = 97.61 nM T16691 C6WD7A 24966736 Ki = 53.62 nM T16691 CJY04G 24966737 Ki = 222 nM T16691 CT47SL 24966738 Ki = 90.71 nM T16691 C1OKR6 24967096 Ki = 27.19 nM T16691 C8HE6A 24967097 Ki = 165 nM T16691 C49BMW 24967099 Ki = 4.82 nM T16691 CJQR84 24967457 Ki = 13.17 nM T16691 CERH27 24968180 Ki = 278 nM T16691 CGX13L 24968181 Ki = 99.7 nM T16691 C8LD4F 24969960 Ki = 10.72 nM T16691 CMC9J2 24970038 Ki = 7.84 nM T16691 C0YK9A 25024144 Ki = 14.6 nM T16691 C02ABD 25024146 Ki = 17.9 nM T16691 C2G8OK 25024148 Ki = 28.2 nM T16691 CEXI24 25024322 Ki = 3.21 nM T16691 CY7AC1 25024326 Ki = 12.4 nM T16691 CJI5U8 25024332 Ki = 11 nM T16691 CO2RU1 25024524 Ki = 5.52 nM T16691 C4YBW2 25024528 Ki = 11.3 nM T16691 CCQ2Y5 25024529 Ki = 8.3 nM T16691 CL83UF 25024530 Ki = 18 nM T16691 CAN16E 25024724 Ki = 3.02 nM T16691 CJX9Q5 25024725 Ki = 3.15 nM T16691 CMD35T 25024726 Ki = 9.33 nM T16691 CP6K8J 25024727 Ki = 2.97 nM T16691 CKEB12 25024729 Ki = 3.36 nM T16691 CQ3ZF4 25024731 Ki = 4.16 nM T16691 CRYA79 25024924 Ki = 2.58 nM T16691 CCF9K4 25024926 Ki = 7.77 nM T16691 C90GZM 25024928 Ki = 5.57 nM T16691 CW6QY9 25024930 Ki = 2.52 nM T16691 CSCP07 25025118 Ki = 14.9 nM T16691 CQ3P5R 25025314 Ki = 5.81 nM T16691 C1PKF0 25056080 Ki = 24.1 nM T16691 CYJ5G1 25067564 Ki = 4.46 nM T16691 CBY3O2 25070582 IC50 = 1800 nM T16691 C4GSD8 25110702 Ki = 1.585 nM T16691 CR17NY 25110703 Ki = 2.512 nM T16691 CNS84K 25117676 Ki = 0.51 nM T16691 C4WV0K 25117677 IC50 = 17.5 nM T16691 CL19XF 25117679 Ki = 21.1 nM T16691 CWFY19 25117680 Ki = 13.7 nM T16691 CSW9K6 25117681 Ki = 36.9 nM T16691 C1PG8Z 25122651 Ki = 4.27 nM T16691 CD3R5U 25122652 Ki = 3.62 nM T16691 CK58IM 25122653 Ki = 4.52 nM T16691 CA12QG 25122654 Ki = 8.04 nM T16691 C3M0EY 25123011 Ki = 18.22 nM T16691 CZX2R0 25123012 Ki = 13.09 nM T16691 CNV98C 25123013 Ki = 3.55 nM T16691 C3N6SM 25123014 Ki = 3.06 nM T16691 CDQ70A 25208878 EC50 = 14 nM T16691 CJ1Z9H 25216680 Ki > 10000 nM T16691 C1T3LR 25218143 Ki > 10000 nM T16691 CPI03N 25218397 Ki > 10000 nM T16691 CL1R3Q 25218401 Ki > 10000 nM T16691 CLIZ27 25251903 Ki = 8883 nM T16691 CM2T9Y 25263297 Ki = 7.9 nM T16691 CR5D2U 25263298 Ki = 50 nM T16691 CR5JL8 25263299 Ki = 1.2 nM T16691 C9G3TC 25263300 Ki = 1.8 nM T16691 CAF19L 25263301 Ki = 2.1 nM T16691 CFJM71 25263302 Ki = 1.3 nM T16691 C5IB8J 25263304 Ki = 10.3 nM T16691 CUBL21 25263305 Ki = 0.6 nM T16691 C8BV1Y 25263306 Ki = 15.3 nM T16691 CM2P4B 25263307 Ki = 11.6 nM T16691 CP25TS 25263308 Ki = 9.3 nM T16691 CUT3O9 25263309 Ki = 61.6 nM T16691 CK0UJ9 25263310 Ki = 126 nM T16691 CAH0F1 25263311 Ki = 45.6 nM T16691 C73QEX 25263312 Ki = 70.7 nM T16691 C18HPB 25263313 Ki = 2.5 nM T16691 C0RK3L 25263314 Ki = 3.3 nM T16691 CFK36A 25263315 Ki = 174 nM T16691 C18PIH 25263316 Ki = 92.5 nM T16691 C1DS3N 25263317 Ki = 42 nM T16691 C0W3ZY 25263318 Ki = 219 nM T16691 CZ69DU 25263319 Ki > 440 nM T16691 C15QMB 25263320 Ki = 6.9 nM T16691 CQH59C 25263321 Ki = 39.8 nM T16691 C1XZ9U 25263322 Ki = 2.8 nM T16691 C1GPQ9 25263323 Ki = 39.5 nM T16691 CP50YT 25263324 Ki = 17.9 nM T16691 C2HJ4M 25263325 Ki > 440 nM T16691 CJQ87U 25263326 Ki = 8.1 nM T16691 C8QS7R 25263327 Ki = 17.8 nM T16691 CPK94B 25263328 Ki = 19.1 nM T16691 CI4OU7 25263329 Ki > 440 nM T16691 CC89NU 25263330 Ki = 50 nM T16691 C56YFT 25263331 Ki > 440 nM T16691 CK7JV5 25263332 Ki > 440 nM T16691 C5XZ3Y 25263333 Ki = 239 nM T16691 CPV78N 25263334 Ki = 48.5 nM T16691 CFCT24 25263335 Ki > 440 nM T16691 C06CZE 25263336 Ki = 10.5 nM T16691 C52XBP 25263337 Ki = 208 nM T16691 CD9HU0 25263338 Ki = 6.4 nM T16691 CTUR83 25263339 Ki = 2.4 nM T16691 CJ69LP 25263340 Ki = 4.3 nM T16691 C5FQW4 25263341 Ki > 440 nM T16691 C0LNU7 25263342 Ki = 3.5 nM T16691 C5A1YV 25263343 Ki = 6.5 nM T16691 C8CMO5 25263344 Ki = 19.6 nM T16691 CQP58M 25263345 Ki = 26.1 nM T16691 CN4JF1 25263346 Ki = 18.4 nM T16691 C3OIN1 25263347 Ki = 5.8 nM T16691 CJ2LH8 25263348 Ki = 24.7 nM T16691 C3RQW5 25263349 Ki = 13.6 nM T16691 CX63AQ 25263350 Ki = 10.1 nM T16691 CPE2C1 25263351 Ki = 15.1 nM T16691 CLNE06 25263352 Ki = 28.9 nM T16691 CUE1X8 25263353 Ki = 11.3 nM T16691 C15JZS 25263354 Ki = 1.5 nM T16691 CFDT07 25263355 Ki = 2.7 nM T16691 CG56DF 42388639 IC50 = 2634 nM T16691 CH5QX6 42389467 IC50 > 10000 nM T16691 COBT83 42602875 Ki < 10 nM T16691 CY7W2J 42631003 Ki = 1.2 nM T16691 CV2X5B 42635027 IC50 = 2839 nM T16691 CS9Q3H 42635204 IC50 = 1956 nM T16691 CQ2M5S 42635387 IC50 = 768 nM T16691 CR3KM7 42635388 IC50 = 6925 nM T16691 CJ3NP5 42636941 IC50 > 10000 nM T16691 CJ41QV 44126269 Ki = 2.399 nM T16691 CG1VP5 44126270 IC50 = 1050 nM T16691 CN3IA4 44126272 IC50 = 974 nM T16691 CY6PC2 44126325 IC50 = 666 nM T16691 C32MRX 44126326 IC50 = 977 nM T16691 CQ28AG 44126327 IC50 = 4070 nM T16691 CNF19Z 44126328 IC50 = 2270 nM T16691 CHFE79 44126329 IC50 = 860 nM T16691 C2Q0UX 44126330 IC50 = 440 nM T16691 CV4TD7 44155107 Ki = 0.549 nM T16691 C6TND7 44155109 Ki = 0.44 nM T16691 CEZ18Q 44155871 Ki = 22.2 nM T16691 C1VF8H 44155874 Ki = 1.2 nM T16691 C1LJY7 44155875 Ki = 1.91 nM T16691 C2Z6PY 44155876 Ki = 6.761 nM T16691 CEJY41 44155992 Ki = 1.072 nM T16691 CE41VX 44155994 Ki = 0.7586 nM T16691 CA5N1Z 44156502 Ki = 14.5 nM T16691 CH68EA 44156622 Ki = 0.3981 nM T16691 C91MAJ 44156624 Ki = 0.5012 nM T16691 C97EQS 44156626 Ki = 0.1862 nM T16691 CXM4K7 44156628 Ki = 0.088 nM T16691 CY41DQ 44156752 Ki = 0.202 nM T16691 C73FZD 44156754 Ki = 0.112 nM T16691 CNXV95 44156756 Ki = 0.49 nM T16691 CPE0L5 44156863 Ki = 0.458 nM T16691 C2SYR0 44216882 Ki = 1.5 nM T16691 CPI9X4 44224259 IC50 = 5990 nM T16691 CR0W9C 44240753 Ki = 7.1 nM T16691 CC4A6H 44240802 Ki = 25 nM T16691 CN1UZ6 44240860 Ki = 11.6 nM T16691 CA8GC6 44242965 Ki = 48 nM T16691 CA9E6X 44248103 Ki = 3.83 nM T16691 C2FDB1 44250364 IC50 > 10000 nM T16691 C8MC0Q 44251387 IC50 > 10000 nM T16691 C5YEA8 44251388 IC50 > 10000 nM T16691 C0BSF6 44251389 IC50 > 10000 nM T16691 CL09IQ 44263496 Ki = 80 nM T16691 C87MXH 44263497 Ki = 64 nM T16691 CB0OX8 44263956 Ki = 510 nM T16691 CC2OD4 44278111 Ki > 10000 nM T16691 CRMA84 44278114 Ki = 6486.5 nM T16691 CF0Y4M 44278115 Ki > 10000 nM T16691 CMI97L 44292800 Ki = 4.7 nM T16691 CKQ5B7 44293023 Ki = 3.3 nM T16691 CL8GV9 44293077 Ki = 3.6 nM T16691 C7PC8W 44327453 Ki = 130 nM T16691 C6MU4R 44327527 Ki = 7.2 nM T16691 CG06CL 44327759 Ki = 0.3 nM T16691 CER86D 44327952 Ki = 180 nM T16691 CQC8S9 44327972 Ki = 33 nM T16691 C5QXL8 44327999 Ki = 6.9 nM T16691 C59TSH 44328120 Ki = 50.12 nM T16691 C6BMZ7 44328589 Ki = 79.43 nM T16691 CU89ZL 44328649 Ki = 31.62 nM T16691 CU2Z3F 44328732 Ki = 1.995 nM T16691 CNHP91 44328748 Ki = 5.012 nM T16691 C02WXU 44341344 Ki = 23 nM T16691 CUXH48 44352308 Ki = 1770 nM T16691 C3LKN1 44364048 Ki = 125.89 nM T16691 CQ07ZJ 44369364 Ki = 3.981 nM T16691 C52GZW 44369415 Ki = 0.7943 nM T16691 C4B3EU 44369594 Ki = 1.995 nM T16691 C5MF9A 44369599 Ki = 158.49 nM T16691 CPQ84Z 44369828 Ki = 3.162 nM T16691 C3LD8S 44369855 Ki = 2.512 nM T16691 CV1O8R 44369858 Ki = 2.512 nM T16691 C3YSZ1 44386408 Ki = 9.4 nM T16691 CZOG07 44386469 Ki = 47 nM T16691 CZQK94 44386665 Ki = 6000 nM T16691 CX05UV 44386717 Ki = 2 nM T16691 C6WJ7D 44386718 Ki = 14 nM T16691 C4IFL1 44386772 Ki = 29 nM T16691 CTP90D 44386815 Ki = 6000 nM T16691 CB72DR 44386821 Ki = 5.1 nM T16691 C83PMF 44386822 Ki = 7.6 nM T16691 C57ANV 44386851 Ki = 200 nM T16691 C9NS0P 44386911 Ki = 5 nM T16691 C48ZFS 44387089 Ki = 2.4 nM T16691 C7VJO9 44387804 Ki = 57.7 nM T16691 CQCJ32 44387817 Ki = 117 nM T16691 CXD1R3 44388701 Ki = 1.4 nM T16691 CX8GB0 44388943 Ki = 1 nM T16691 CCA46R 44388944 Ki = 7 nM T16691 C4FBC2 44388950 Ki = 3 nM T16691 CPW47O 44388951 Ki = 3 nM T16691 C2AS1M 44388953 Ki = 31 nM T16691 CCX5P2 44388954 Ki = 118 nM T16691 CT50YA 44388955 Ki = 20 nM T16691 CTPG47 44388956 Ki = 3 nM T16691 CVE02M 44388970 Ki = 5 nM T16691 CNAH73 44388971 Ki = 246 nM T16691 CJVF20 44388980 Ki = 50 nM T16691 C7UO3A 44388986 Ki = 54 nM T16691 C1XJR3 44388987 Ki = 29 nM T16691 C6FWJ7 44388999 Ki = 2 nM T16691 CKWI18 44389001 IC50 = 0.7 nM T16691 C6QG9Z 44389002 IC50 = 3.9 nM T16691 CQ85AW 44389003 Ki = 0.4 nM T16691 C3LRC0 44389004 Ki = 1 nM T16691 CCV4R6 44389010 Ki = 27 nM T16691 CW25QI 44389015 Ki = 1 nM T16691 C8AG7U 44389016 Ki = 1 nM T16691 C5Q2DG 44389023 IC50 = 4.1 nM T16691 C0C6AK 44389024 Ki = 77 nM T16691 CW2VL5 44389025 Ki = 2.4 nM T16691 C3TQF5 44389074 Ki = 3 nM T16691 C0Y1WT 44389075 Ki = 14 nM T16691 C9Q8HJ 44389081 IC50 = 1.3 nM T16691 CMK43D 44389086 Ki = 20 nM T16691 C6F0PN 44389091 Ki = 18 nM T16691 CI29MW 44389099 Ki = 4 nM T16691 C49POD 44389999 Ki = 63 nM T16691 CEP37C 44390011 Ki = 57 nM T16691 C8EO5M 44390023 Ki = 35 nM T16691 CCS1R5 44390045 Ki = 21 nM T16691 CD27FB 44390095 Ki = 54 nM T16691 CRE63B 44390105 Ki = 190 nM T16691 CG9S1O 44393045 Ki = 172 nM T16691 CO6EY0 44393113 Ki = 380 nM T16691 CFZ06U 44395451 Ki = 5.7 nM T16691 C2YT8F 44395458 Ki = 1011 nM T16691 CWP5C1 44395499 Ki = 27 nM T16691 CDWH09 44395500 Ki = 15.5 nM T16691 CWV3T0 44395570 Ki = 23 nM T16691 C28QOZ 44395595 Ki = 5 nM T16691 CIVS89 44395604 Ki = 57 nM T16691 CK9QF8 44395632 Ki = 46 nM T16691 CG1P9D 44395633 Ki = 42 nM T16691 CGH8T3 44395663 Ki = 44 nM T16691 CM4Q5J 44395664 IC50 = 23 nM T16691 CL70AX 44396965 Ki = 2400 nM T16691 C2CV9R 44397117 Ki = 550 nM T16691 CWH17E 44397119 Ki = 29 nM T16691 C2H4SK 44397258 Ki = 8750 nM T16691 CA2M3N 44397322 Ki = 9.9 nM T16691 C21NVO 44397392 Ki = 7.8 nM T16691 CW3D4Z 44397420 Ki = 640 nM T16691 CA0G3Y 44397550 Ki = 27.7 nM T16691 C4B0OI 44397588 Ki < 7943.28 nM T16691 C5FP0R 44397589 Ki < 1995.26 nM T16691 CD6JC7 44397650 Ki = 9.1 nM T16691 CE3G8U 44397670 Ki = 3981.07 nM T16691 C51HTB 44397689 Ki = 1.7 nM T16691 C5FG9Z 44398251 Ki = 5.012 nM T16691 CGXA61 44398325 Ki = 0.7943 nM T16691 CZT23U 44398389 Ki = 0.1995 nM T16691 CMW7N1 44398420 Ki = 79.43 nM T16691 C7FJ9V 44398455 Ki = 63.1 nM T16691 CZ86NU 44398555 Ki = 39.81 nM T16691 CSA67D 44398568 Ki = 3.162 nM T16691 CXH9F6 44398569 Ki = 251.19 nM T16691 C25PRL 44398570 Ki = 1 nM T16691 C2J7IK 44398571 Ki = 0.1259 nM T16691 CK19DL 44398577 Ki = 6.31 nM T16691 CKB7D0 44401278 Ki = 100 nM T16691 CZOP35 44401434 Ki = 57 nM T16691 C9XM1K 44401465 Ki = 50 nM T16691 C4UG8Z 44403044 IC50 = 1 nM T16691 CE10DO 44403046 Ki = 9.8 nM T16691 C6D7PC 44403047 Ki = 3 nM T16691 CV4I3H 44403048 Ki = 11 nM T16691 C53GTV 44403052 Ki = 43 nM T16691 CU42TN 44403053 Ki = 22 nM T16691 C3G0NR 44403055 Ki = 4.6 nM T16691 COC2X7 44403056 Ki = 49 nM T16691 C42TYP 44403057 Ki = 34 nM T16691 CD71OL 44403059 Ki = 9.2 nM T16691 C5NS1R 44403060 Ki = 13 nM T16691 CS6QR7 44403061 Ki = 33 nM T16691 C2VJK8 44403062 Ki = 40 nM T16691 C4SI2K 44403063 Ki = 21.7 nM T16691 C7GNI8 44403064 Ki = 8.5 nM T16691 CNV08U 44403065 Ki = 7 nM T16691 C0MDT3 44403066 Ki = 49 nM T16691 CAE0Q4 44403070 Ki = 14 nM T16691 C8FH9R 44403071 Ki = 44.7 nM T16691 CCKI37 44403072 Ki = 10.5 nM T16691 CA5HK9 44403073 Ki = 23 nM T16691 CM04HK 44403074 Ki = 25 nM T16691 C6JG7H 44403075 Ki = 22 nM T16691 C5CHG2 44403076 Ki = 16 nM T16691 C1FJK7 44403077 Ki = 20 nM T16691 CHJ21O 44403078 Ki = 283.7 nM T16691 CRGK10 44403079 Ki = 252.7 nM T16691 CT0K6J 44403080 Ki = 41.7 nM T16691 CK5B2Y 44403082 Ki = 13 nM T16691 C69KGB 44403083 Ki = 20 nM T16691 CJ3NF1 44403084 Ki = 4 nM T16691 CUF3Y7 44403085 Ki = 271.3 nM T16691 CYPN60 44403086 Ki = 116 nM T16691 CN76UV 44403087 Ki = 26 nM T16691 CB9N2C 44403088 Ki = 48 nM T16691 C2U5VA 44403089 Ki = 7 nM T16691 C1D5XJ 44403090 Ki = 22.7 nM T16691 C7DI0U 44403091 Ki = 58 nM T16691 CT5J9L 44403092 Ki = 4 nM T16691 CM52PQ 44403093 Ki = 7 nM T16691 C0MJ5E 44403094 Ki = 1.5 nM T16691 C1B4QL 44403095 Ki = 5089 nM T16691 C78XLE 44403096 Ki = 8 nM T16691 C8JVC0 44403097 Ki = 3 nM T16691 C1YL7Z 44403098 Ki > 10000 nM T16691 C2F3PA 44403099 Ki = 5 nM T16691 CJE43P 44403100 Ki = 19.3 nM T16691 CFV98A 44403101 Ki = 1429 nM T16691 C6OY9S 44403102 Ki = 2863 nM T16691 CZYP63 44403103 Ki = 3 nM T16691 CUS27C 44403104 IC50 = 7.3 nM T16691 CH4SX6 44403105 Ki > 10000 nM T16691 CK73IG 44403277 Ki = 7.943 nM T16691 CK8ZC2 44403297 Ki = 1 nM T16691 CU20KD 44403304 Ki = 0.631 nM T16691 CGV60Z 44403305 Ki = 0.3981 nM T16691 CCR38V 44403327 Ki = 0.5012 nM T16691 C93VWG 44403335 IC50 = 90 nM T16691 CDR8Y4 44403351 IC50 = 40 nM T16691 CC4X2L 44403358 IC50 = 30 nM T16691 CNE30I 44403366 IC50 = 40 nM T16691 CQ98FN 44403367 IC50 = 100 nM T16691 CMUH71 44403375 IC50 = 30 nM T16691 CQH74S 44403376 IC50 = 60 nM T16691 CGMD49 44403377 IC50 = 50 nM T16691 C6WB0T 44403384 IC50 = 70 nM T16691 CBX76M 44403386 IC50 = 600 nM T16691 C4LKC1 44404394 Ki = 469 nM T16691 C3EJ4G 44404396 Ki = 841 nM T16691 C6NEJ8 44405348 Ki = 7 nM T16691 C9T0GF 44405357 Ki = 1.9 nM T16691 CJB4D6 44405369 Ki = 26 nM T16691 CE5N7Y 44405385 Ki = 21 nM T16691 CG87PW 44409290 Ki > 720 nM T16691 CI3F8D 44413493 Ki = 210 nM T16691 COC47A 44413644 Ki = 165 nM T16691 CS01VM 44413645 Ki = 205 nM T16691 C8XO7Q 44420490 Ki = 14 nM T16691 CB7L2P 44420491 Ki = 11 nM T16691 CJIP85 44420568 Ki = 106 nM T16691 C0TC1M 44420569 Ki = 15 nM T16691 CE2V0S 44425698 Ki = 50.12 nM T16691 C2TE3S 44425699 Ki = 5.012 nM T16691 CU52GB 44425701 Ki = 1.259 nM T16691 C9F1XP 44425702 Ki = 7.943 nM T16691 CR1QN5 44425703 Ki = 25.12 nM T16691 C5UZS7 44425704 Ki = 6.31 nM T16691 CN96FA 44425705 Ki = 10 nM T16691 C1J9MY 44425706 Ki = 15.85 nM T16691 CPI52U 44425708 Ki = 12.59 nM T16691 CNZ3M7 44425711 Ki = 50.12 nM T16691 C92AZG 44425714 Ki = 50.12 nM T16691 C7LP1B 44425717 Ki = 31.62 nM T16691 CX8TR0 44425719 Ki = 7.943 nM T16691 CZ3RM2 44435219 Ki = 9900 nM T16691 C6NA0Z 44435538 IC50 = 9.6 nM T16691 CFZ43E 44435603 Ki = 1.995 nM T16691 C2NUK7 44435604 Ki = 2.692 nM T16691 C64YGX 44435607 Ki = 8.5 nM T16691 CU8MX9 44435608 Ki = 1.5 nM T16691 CEL2F1 44435609 Ki = 5.495 nM T16691 CGJX16 44435610 Ki = 1.288 nM T16691 CB0A9Z 44435612 Ki = 4.266 nM T16691 C0HBD2 44435613 Ki = 1.288 nM T16691 C4SC3H 44435614 Ki = 2.5 nM T16691 C7K9LY 44435615 Ki = 5.6 nM T16691 CR2U0J 44435616 Ki = 1.4 nM T16691 CO6YJ3 44435617 Ki = 5 nM T16691 CCK8S6 44435618 Ki = 2.188 nM T16691 CI07QG 44435619 Ki = 1.5 nM T16691 CO9S3E 44435620 Ki = 4.169 nM T16691 C5K3CJ 44435621 Ki = 0.8913 nM T16691 CN9T5I 44435622 Ki = 10.96 nM T16691 C5WQ7O 44435623 Ki = 8.3 nM T16691 CYCH81 44435624 Ki = 3.3 nM T16691 COS74A 44435625 Ki = 1 nM T16691 CB2O6F 44435626 Ki = 5.7 nM T16691 CIB4M5 44435627 Ki = 4.898 nM T16691 C8UW3X 44435628 Ki = 3.7 nM T16691 CW9SM4 44435629 Ki = 1.288 nM T16691 C2L6RY 44435630 Ki = 7.586 nM T16691 CL02YH 44435631 Ki = 11.48 nM T16691 CL2M7U 44435632 Ki = 33.11 nM T16691 CA09IP 44435633 Ki = 11.1 nM T16691 CD4M9E 44435635 Ki = 4.571 nM T16691 CEA1M2 44435637 Ki = 12 nM T16691 C8S1WD 44435638 Ki = 2.089 nM T16691 C1WX0B 44435639 Ki = 3.8 nM T16691 CSQ21Z 44435640 Ki = 1.995 nM T16691 C9JR1U 44435641 Ki = 4.677 nM T16691 CD8GO7 44435642 Ki = 4.365 nM T16691 CY27QR 44435643 Ki = 3.388 nM T16691 C8H5MA 44435644 Ki = 9.333 nM T16691 C8GY6Q 44435646 Ki = 6.1 nM T16691 CSHJ16 44435647 Ki = 3.89 nM T16691 C9P1AJ 44435649 Ki = 13.49 nM T16691 CL13NV 44435650 Ki = 1.2 nM T16691 CC1I9Y 44435652 Ki = 1.9 nM T16691 CC5G9M 44435653 Ki = 3.2 nM T16691 CS6HP4 44438689 Ki = 590 nM T16691 C6D5OV 44438708 Ki = 280 nM T16691 C3HJY2 44438709 Ki = 135 nM T16691 C0V6QX 44438711 Ki = 220 nM T16691 C54RZL 44438716 Ki = 440 nM T16691 CH0YR3 44438718 Ki = 210 nM T16691 CJ9IW7 44438720 Ki = 13 nM T16691 CI9BD3 44438722 Ki = 1.9 nM T16691 C7R1IF 44438723 Ki = 94 nM T16691 CY9B7P 44438726 Ki = 29 nM T16691 C4UCP2 44438728 Ki = 132 nM T16691 C2I9YU 44438729 Ki = 44 nM T16691 C6R3CH 44438731 Ki = 445 nM T16691 CYZ2F7 44438732 Ki = 20 nM T16691 C0YE5U 44438738 Ki = 1.5 nM T16691 C4U5VN 44438743 Ki = 6000 nM T16691 CKZF16 44439165 Ki = 7943.28 nM T16691 CA4HZ3 44439167 Ki < 10000 nM T16691 C6R7JW 44441237 Ki = 1.259 nM T16691 CE95NG 44441238 Ki = 630.96 nM T16691 CD7WK4 44441239 Ki = 3.981 nM T16691 CP3V1M 44441240 Ki = 3.981 nM T16691 C8E3UZ 44441241 Ki = 5.012 nM T16691 CMY15F 44441242 Ki = 125.89 nM T16691 C3F8TA 44443506 Ki = 402 nM T16691 CNBC07 44443511 Ki = 1888 nM T16691 CO6R9T 44446213 Ki = 293 nM T16691 C6PR5Y 44446214 Ki = 893 nM T16691 CZL97F 44455426 Ki = 3890 nM T16691 C6BFI0 44456033 Ki = 1028.4 nM T16691 C12XGE 44456400 Ki > 10000 nM T16691 CS79YN 44459048 Ki = 42.66 nM T16691 C4DL5C 44469677 IC50 > 10000 nM T16691 CM5EY8 44474470 Ki = 26 nM T16691 C8UON6 44474625 Ki = 5.2 nM T16691 C6HVU1 44474629 Ki = 1.2 nM T16691 CE2Z8S 44474631 Ki = 2.6 nM T16691 C8LA4W 44474797 Ki = 4.1 nM T16691 CMST50 44476434 Ki = 1.9 nM T16691 CXY7T9 44476436 Ki = 0.39 nM T16691 CPX32Z 44476514 Ki = 0.68 nM T16691 C6V2YR 44476607 Ki = 0.82 nM T16691 C3F8HQ 44476611 Ki = 2.1 nM T16691 C2WXT0 44476704 Ki = 60.4 nM T16691 C8QCU7 44476801 Ki = 372 nM T16691 CO5SX2 44476804 Ki = 1155 nM T16691 C1H8NX 44516817 Ki = 0.2 nM T16691 C3D4HR 44537940 Ki = 7.5 nM T16691 CJ7U3K 44554227 Ki = 2.9 nM T16691 CT67VS 44554228 Ki = 2.2 nM T16691 CM0I1P 44554393 Ki = 4.6 nM T16691 CXDZ28 44554394 Ki = 1.9 nM T16691 CNHA47 44554395 Ki = 1.6 nM T16691 CA5G3B 44567932 Ki = 193 nM T16691 C3PZE4 44567933 Ki = 33 nM T16691 CJBD54 44567981 Ki = 23 nM T16691 CRM8G3 44567982 Ki = 19 nM T16691 COB09W 44567983 Ki = 41 nM T16691 CS5X2K 44567984 Ki = 18 nM T16691 C65HIW 44567985 Ki = 68 nM T16691 CRG8E2 44568019 Ki = 89 nM T16691 CGU0L3 44568020 Ki = 46 nM T16691 CFKG06 44568021 Ki = 24 nM T16691 CU3SX6 44568022 Ki = 33 nM T16691 C8WC9P 44568061 Ki = 12 nM T16691 CV0RZ9 44568062 Ki = 19 nM T16691 CGD81I 44568063 Ki = 50 nM T16691 CPYC85 44568064 Ki = 124 nM T16691 C7LZ4X 44568065 Ki = 85 nM T16691 C20LPH 44568101 Ki = 139 nM T16691 C3RFT5 44568102 Ki = 504 nM T16691 C3UX9P 44568103 Ki = 324 nM T16691 C8M0YW 44568104 Ki = 253 nM T16691 CN8M2K 44568139 Ki = 12 nM T16691 C68JSG 44579085 Ki = 1.585 nM T16691 CVU2Z0 44579129 Ki = 7.943 nM T16691 C4PJ7T 44579130 Ki = 7.943 nM T16691 CEH1N0 44579131 Ki = 1.995 nM T16691 CW69AF 44579132 Ki = 100 nM T16691 CM1PH0 44579133 Ki = 7.943 nM T16691 CL3J1S 44579180 Ki = 3.981 nM T16691 C4N2PZ 44579181 Ki = 1.259 nM T16691 C74XJR 44579182 Ki = 1.995 nM T16691 C9PY2D 44579183 Ki = 39.81 nM T16691 C5NS6H 44581972 Ki = 489.78 nM T16691 CK8Z1P 44581973 Ki = 831.76 nM T16691 C3UQ9Z 44581974 Ki = 3388.44 nM T16691 CRCH48 44582675 Ki = 3842 nM T16691 CEJ4R8 44582676 Ki > 10000 nM T16691 CZGP86 44582677 Ki > 10000 nM T16691 C5QB4K 44582678 Ki > 10000 nM T16691 C01RCI 44582705 Ki > 10000 nM T16691 CXL25V 44582706 Ki > 10000 nM T16691 C8MR1X 44582707 Ki > 10000 nM T16691 C4IT1N 44582708 Ki > 10000 nM T16691 C18APH 44591028 Ki = 176 nM T16691 C8C2RL 44591029 Ki = 127 nM T16691 C0TGD4 44591068 Ki = 33 nM T16691 CQU75A 44591069 Ki = 79 nM T16691 C6RYT5 44591592 Ki = 4 nM T16691 C5JN4B 44591611 Ki = 3.2 nM T16691 CB0S4Z 44592109 IC50 > 10000 nM T16691 CQI0D4 45102707 Ki = 158.49 nM T16691 CSEP-69 45102708 Ki = 630.96 nM T16691 C0DLU3 45109862 IC50 = 1412 nM T16691 C1AM5U 45113275 IC50 = 26000 nM T16691 CH0BX2 45113399 IC50 = 62000 nM T16691 CGB2Z0 45113400 Ki = 2.1 nM T16691 C50CMH 45113401 IC50 = 3900 nM T16691 CWE53Z 45113403 IC50 = 85 nM T16691 CHN63A 45113404 IC50 = 3400 nM T16691 CCVA63 45113530 Ki = 5.7 nM T16691 CR52JD 45113534 IC50 = 620 nM T16691 C7I2OM 45113535 IC50 = 28000 nM T16691 CZ71RN 45278805 IC50 = 713 nM T16691 CZN6M7 45278882 IC50 = 1904 nM T16691 CPEY83 45378934 Ki = 54.3 nM T16691 CU36SC 45378935 Ki = 48.7 nM T16691 CHNI56 45378936 Ki = 75.8 nM T16691 C0CHF4 45482789 IC50 = 9580 nM T16691 CD5H2X 45483622 Ki = 2.2 nM T16691 C1BQT4 45483628 Ki = 70 nM T16691 C4IY7C 45483630 Ki <= 8 nM T16691 C5O1SN 45483634 Ki <= 8 nM T16691 CNLO32 45484297 Ki = 4.7 nM T16691 C28VBH 45484298 Ki = 11.7 nM T16691 C0VI9E 45484299 Ki = 9 nM T16691 C0C2LY 45484307 Ki = 15 nM T16691 CK1CD7 45484322 Ki = 3.3 nM T16691 CHI36F 45484332 Ki = 88 nM T16691 C3JZC6 45484333 Ki = 0.9 nM T16691 CAM93H 45484339 Ki = 45 nM T16691 CCB6J0 45484340 Ki = 0.9 nM T16691 C6YO5M 45484352 EC50 = 30 nM T16691 C0Z8VW 45484381 Ki = 4.2 nM T16691 C1IBR5 45484382 Ki = 4.7 nM T16691 CU0YM2 45484383 Ki = 2.1 nM T16691 C83ZJN 45484384 Ki = 2.1 nM T16691 CGZW45 45484398 Ki = 4.3 nM T16691 CYS1T3 45484399 Ki = 2.9 nM T16691 CKYS61 45487099 Ki = 46 nM T16691 C4M9EL 45487100 Ki = 42 nM T16691 CZ4E6T 45487112 Ki = 214 nM T16691 CI7S4B 45487113 Ki = 56 nM T16691 C8PGH3 45487128 Ki = 11.3 nM T16691 CBF24J 45487129 Ki = 3.9 nM T16691 CO81XT 45487139 Ki = 1.7 nM T16691 C7HN5G 45487140 Ki = 76 nM T16691 CL2JK1 45487150 Ki = 35 nM T16691 CH90CZ 45488126 Ki > 1000 nM T16691 CG9U2R 45488130 Ki > 1000 nM T16691 C7N4GP 45488138 Ki > 1000 nM T16691 CH29KP 45488139 Ki = 16 nM T16691 CDAJ27 45488143 Ki = 16 nM T16691 CZYC01 45488151 Ki = 13 nM T16691 C8PH0Y 45488152 Ki = 5 nM T16691 CC2OU0 45488156 Ki > 1000 nM T16691 CL4G8T 45488165 Ki = 27 nM T16691 C5NDO6 45488166 Ki = 17 nM T16691 C0GMN4 45488171 Ki > 1000 nM T16691 C3ZAL4 45488172 Ki > 1000 nM T16691 C3PYL9 45488174 Ki > 1000 nM T16691 CFT7C5 45488175 Ki > 1000 nM T16691 CX1A2N 45488179 Ki > 1000 nM T16691 CA8I7U 45488180 Ki > 1000 nM T16691 C01QBM 45488181 Ki > 1000 nM T16691 COX47A 45488183 Ki > 1000 nM T16691 C8ETO2 45488184 Ki > 1000 nM T16691 C5KOL1 46189932 Ki = 0.5248 nM T16691 CQ8I3H 46189935 Ki = 0.6457 nM T16691 CD2Y4X 46189980 Ki = 1.38 nM T16691 C1YO4C 46189984 Ki = 0.5495 nM T16691 CI30OJ 46189987 Ki = 1.413 nM T16691 CF3WR6 46190034 Ki = 0.7079 nM T16691 C71HDV 46190037 Ki = 0.4169 nM T16691 C2DF3H 46190041 Ki = 2.089 nM T16691 C5KRC3 46203710 Ki = 0.53 nM T16691 CIV92F 46214153 Ki = 47 nM T16691 C0LZ2J 46220503 Ki = 0.1995 nM T16691 CZJH90 46224877 IC50 = 5730 nM T16691 CFL32X 46224878 IC50 = 2580 nM T16691 C5FQ4S 46224879 Ki = 0.6166 nM T16691 CB0OH9 46224880 IC50 = 1680 nM T16691 C37TXV 46224881 IC50 = 910 nM T16691 CQ8P2A 46224914 IC50 = 180 nM T16691 C5DV2F 46224915 IC50 = 2810 nM T16691 CS0D4H 46224916 IC50 = 550 nM T16691 CC29VZ 46224917 IC50 = 1000 nM T16691 CH43AW 46224918 IC50 = 1750 nM T16691 C2G4FT 46224941 IC50 = 1440 nM T16691 CZX2L5 46224942 IC50 = 2950 nM T16691 C67UFY 46224943 IC50 = 5580 nM T16691 CUW7O3 46224944 IC50 = 1500 nM T16691 C4E6CK 46224945 IC50 = 1980 nM T16691 CW3R4Q 46224973 IC50 = 3720 nM T16691 CAZX21 46225000 IC50 = 692 nM T16691 CDR41P 46225001 IC50 = 1130 nM T16691 CDBP61 46225002 IC50 = 20700 nM T16691 C38OVM 46225027 IC50 = 2350 nM T16691 CFV3D0 46227395 Ki = 0.4 nM T16691 CY82LR 46227396 Ki = 3 nM T16691 C79UFN 46227404 Ki = 10 nM T16691 C42SVX 46700866 IC50 > 10000 nM T16691 CD0K6E 46700867 IC50 = 5000 nM T16691 CA4HD5 46830134 Ki = 0.68 nM T16691 C5TC2S 46830335 IC50 > 10000 nM T16691 C1K7FL 46830336 IC50 > 10000 nM T16691 C1N4KX 46842383 IC50 > 10000 nM T16691 CC62SX 46866711 IC50 = 16 nM T16691 C0HCI4 46867519 Ki = 0.499 nM T16691 C2B1NM 46867521 Ki = 0.256 nM T16691 C7K5AG 46867523 Ki = 28.8 nM T16691 CSLN36 46867524 Ki = 25.5 nM T16691 CCJ72Y 46867654 Ki = 869 nM T16691 C0HP4U 46867655 Ki = 1764 nM T16691 CRHN02 46880486 Ki = 6 nM T16691 C1T3YB 46880529 Ki = 10.7 nM T16691 CQC7S6 46880530 Ki = 68 nM T16691 CWI3U0 46880531 Ki = 16 nM T16691 C3HFU0 46880532 Ki = 4 nM T16691 CFK3A1 46880533 Ki = 21 nM T16691 CC9EQ0 46880606 Ki = 7.1 nM T16691 C6DO1B 46880607 Ki = 5.6 nM T16691 CZ4OL7 46880608 Ki = 4.7 nM T16691 CR8WY3 46880655 Ki = 3.5 nM T16691 CRZ1S3 46880656 Ki = 18 nM T16691 C47GTW 46880657 Ki = 9.6 nM T16691 C30YQL 46880658 Ki = 5 nM T16691 CCV2U9 46880659 Ki = 18 nM T16691 CFN34C 46880705 Ki = 15 nM T16691 C4RL1V 46880706 Ki = 72 nM T16691 CC8PU0 46880707 Ki = 3.2 nM T16691 CS7NP1 46880708 Ki = 1.3 nM T16691 CW5Y1T 46880709 Ki = 4.6 nM T16691 CW8DH2 46880756 Ki = 23.3 nM T16691 CM53AL 46880757 Ki = 6 nM T16691 C6FZG0 46880758 Ki = 1.5 nM T16691 C9JR7V 46880759 Ki = 2.8 nM T16691 CF8IJ2 46882520 Ki = 6.31 nM T16691 CQN87I 46882521 Ki = 125.89 nM T16691 C56ULO 46882522 Ki = 199.53 nM T16691 CX72IN 46882583 Ki = 15.85 nM T16691 C04JRH 46884709 Ki = 7.97 nM T16691 CB8GE1 46884818 IC50 > 10000 nM T16691 C4MQ0A 46884856 IC50 > 10000 nM T16691 CCNT25 46884898 IC50 > 10000 nM T16691 C3MSG2 46885027 IC50 > 10000 nM T16691 CB7XI0 46885213 IC50 = 3600 nM T16691 C8XK4D 46889325 Ki = 0.7943 nM T16691 CZK2Y7 46889326 Ki = 0.05012 nM T16691 C1NRH4 46889327 Ki = 5.012 nM T16691 CMF2K4 46889328 Ki = 0.1 nM T16691 CI0LR5 46889329 Ki = 1.259 nM T16691 CS86BA 46889349 Ki = 1 nM T16691 C8WJ7D 46889350 Ki = 0.1259 nM T16691 C6L0RO 46889351 Ki = 0.2512 nM T16691 CFCL20 46889352 Ki = 1.259 nM T16691 CI8OB1 46889353 Ki = 0.3162 nM T16691 C01JSO 46889472 Ki = 0.85 nM T16691 CUE0M9 46889856 Ki = 0.0631 nM T16691 CX7KU0 46889857 Ki = 25.12 nM T16691 CVKR52 46889858 Ki = 0.631 nM T16691 C04LNT 46889890 Ki = 0.1585 nM T16691 C2RL9U 46889891 Ki = 0.2512 nM T16691 C8AO0P 46889892 Ki = 0.3981 nM T16691 CA82ZW 46889893 Ki = 0.07943 nM T16691 CR13XZ 46889894 Ki = 3.981 nM T16691 CYU82R 46889895 Ki = 0.5012 nM T16691 CJRE76 46889915 Ki = 158.49 nM T16691 C4W2VY 46889916 Ki > 1000 nM T16691 CS8VY2 46889917 Ki = 0.3162 nM T16691 CV9ZF7 46889918 Ki = 0.1585 nM T16691 C81CYN 46889919 Ki = 7.943 nM T16691 CZY21R 46889920 Ki = 1.995 nM T16691 CC26DS 46890056 Ki = 31.62 nM T16691 C02CYN 46890057 Ki = 7.943 nM T16691 C9R5DS 46890058 Ki = 25.12 nM T16691 C63WEI 46890059 Ki = 50.12 nM T16691 C0FDW6 46890103 Ki = 158.49 nM T16691 C8BVJ4 46890104 Ki = 79.43 nM T16691 CWP20Q 46890105 Ki = 7.943 nM T16691 CGS9H6 46890106 Ki = 63.1 nM T16691 CDQS62 46890155 Ki = 0.3981 nM T16691 C3CX6A 46890156 Ki = 0.631 nM T16691 C9BUE2 46890157 Ki = 0.3981 nM T16691 CGB3Q0 46890158 Ki = 2.512 nM T16691 CO0GK6 46890188 Ki = 39.81 nM T16691 C1B8FI 46890189 Ki = 1.585 nM T16691 C5AGP8 46890190 Ki = 0.1259 nM T16691 CUC1W9 46890191 Ki = 1.585 nM T16691 C61GYF 46890192 Ki = 0.1 nM T16691 CKX3H2 46890218 Ki = 0.7943 nM T16691 C9M6BC 46890219 Ki = 3.981 nM T16691 CQE27V 46890220 Ki = 1.995 nM T16691 C6ZW7P 46890221 Ki = 0.3981 nM T16691 C1VND9 46890263 Ki = 31.62 nM T16691 CB5YT0 46890264 Ki = 0.1259 nM T16691 CE65DF 46890265 Ki = 3.981 nM T16691 C1CS6T 46890266 Ki = 1 nM T16691 CMVY84 46890267 Ki = 1.995 nM T16691 C75QXU 46890292 Ki = 31.62 nM T16691 C78KYS 46890293 Ki = 5.012 nM T16691 CO84JE 46890294 Ki = 15.85 nM T16691 CY42MI 46890295 Ki = 0.631 nM T16691 CL0Y8V 46890322 Ki = 0.1 nM T16691 CD8P6A 46890323 Ki = 6.31 nM T16691 C5QSL3 46890324 Ki = 0.1585 nM T16691 C9P5ZH 46890325 Ki = 0.1995 nM T16691 C50TPC 46890326 Ki = 0.2512 nM T16691 C4OBP5 46890884 Ki = 0.1585 nM T16691 C2Q1CG 46890885 Ki = 1.259 nM T16691 CAEV87 46890886 Ki = 19.95 nM T16691 CT71MK 46890887 Ki = 79.43 nM T16691 CHGA24 46890946 Ki = 31.62 nM T16691 CQSK68 46890947 Ki = 79.43 nM T16691 C4DMB0 46890948 Ki = 5.012 nM T16691 CRX51I 46890949 Ki = 31.62 nM T16691 C0ZN6Q 46891004 Ki = 25.12 nM T16691 CW6R3C 46891005 Ki = 31.62 nM T16691 CXRO49 46891006 Ki = 50.12 nM T16691 C72HAI 46891007 Ki = 316.23 nM T16691 CN9E0A 46891053 Ki = 125.89 nM T16691 C0JTL3 46891054 Ki = 63.1 nM T16691 CHZ25O 46891055 Ki = 316.23 nM T16691 CEH9I0 46891056 Ki = 316.23 nM T16691 C64NDL 46891111 Ki = 25.12 nM T16691 CI43LK 46891112 Ki = 19.95 nM T16691 CFC7A4 46891113 Ki = 25.12 nM T16691 CY0NP6 46891114 Ki = 100 nM T16691 C5ND3Q 46891174 Ki = 100 nM T16691 CRL43U 46891175 Ki = 125.89 nM T16691 CKB43Z 46891176 Ki = 31.62 nM T16691 CH86DQ 46933237 Ki = 23 nM T16691 CUTX67 46934428 IC50 = 3 nM T16691 CLT9W7 49780170 Ki = 447 nM T16691 CM98BZ 49780586 Ki = 27 nM T16691 CMA5Q3 49781032 Ki = 747 nM T16691 CS0EZ3 49781034 Ki = 215 nM T16691 CNR45W 49781036 Ki = 741 nM T16691 C1M7UP 49781038 Ki = 8 nM T16691 CL4R1V 49781250 Ki = 135 nM T16691 CMHL69 49781252 Ki = 175 nM T16691 CH1W6B 49781254 Ki = 554 nM T16691 C1QRV6 49781469 Ki = 194 nM T16691 C5X0JU 49781471 Ki = 523 nM T16691 CFSO43 49782361 Ki = 165 nM T16691 CQ39JR 49782362 Ki = 266 nM T16691 C2LZJ0 49783209 Ki = 489 nM T16691 C57SMG 49783415 Ki > 10000 nM T16691 C0TG6I 49783419 Ki > 10000 nM T16691 CB63SX 49798858 IC50 > 5000 nM T16691 C34YMO 49798859 IC50 = 120 nM T16691 C1RY7B 49799629 IC50 > 300 nM T16691 CHWT97 49799645 IC50 = 2260 nM T16691 CYC36S 49799656 IC50 = 580 nM T16691 CY4ZF0 49799663 IC50 = 1990 nM T16691 CPW4R7 49799664 IC50 = 1340 nM T16691 CAI82J 49799665 IC50 > 300 nM T16691 CL74MS 49799667 Ki = 14.7 nM T16691 CEJ4N3 49799678 IC50 > 300 nM T16691 COIW10 49799683 IC50 > 30 nM T16691 CG2W7R 49799684 IC50 > 30 nM T16691 C8AXI7 49799685 Ki = 26.3 nM T16691 C5AWK0 49799703 Ki = 103 nM T16691 CR40BA 49836386 IC50 = 37 nM T16691 C6N1PQ 49836504 Ki = 134 nM T16691 C1GJ9H 49836505 Ki = 125 nM T16691 CF98HT 49836507 Ki = 88 nM T16691 CSP1K6 49836508 Ki = 5.5 nM T16691 C6L8IS 49836509 Ki = 1.7 nM T16691 CU2X8O 49836615 Ki = 4 nM T16691 CI35ZA 49836616 Ki = 1 nM T16691 C2Z0KC 49836617 Ki = 8.1 nM T16691 C7F1MN 49836618 Ki = 1.1 nM T16691 CV3M8N 49836619 Ki = 12 nM T16691 C5HK3L 49836620 Ki = 0.9 nM T16691 C2SF3J 49836715 Ki = 7.8 nM T16691 C9NA6O 49836716 Ki = 2.6 nM T16691 C5T8CJ 49836717 Ki = 11 nM T16691 C6CZ9E 49836718 Ki = 110 nM T16691 CQ28NW 49836720 Ki = 124 nM T16691 CF71YC 49836721 Ki = 207 nM T16691 C7QAT9 49836823 Ki = 4.6 nM T16691 CJE9R5 49836824 Ki = 2.9 nM T16691 C8OAJ4 49836825 Ki = 1.7 nM T16691 C7G1VL 49836826 Ki = 1.7 nM T16691 CRUP23 49836827 Ki = 1.8 nM T16691 C36URZ 49836828 Ki = 1.8 nM T16691 C3DR7S 49836923 Ki = 1.4 nM T16691 C5DLH2 49836924 Ki = 2 nM T16691 C06HID 49836925 Ki = 22 nM T16691 C4R2YS 49850567 Ki = 794.33 nM T16691 C07JTU 49850570 Ki > 6309.57 nM T16691 CK68QR 49850672 Ki > 1584.89 nM T16691 CN5XR1 49850772 Ki > 10000 nM T16691 CR4EZ0 49850870 Ki > 2511.89 nM T16691 C5K4EC 49850872 Ki > 3981.07 nM T16691 C8AW0R 49850874 Ki > 1000 nM T16691 C9KIU1 49864289 IC50 = 6 nM T16691 CHO9C0 49864292 IC50 = 3 nM T16691 CU0TJ6 49864530 IC50 = 2191 nM T16691 C9FD2E 49864599 IC50 = 27 nM T16691 CVY4O3 49864600 IC50 = 422 nM T16691 CJF6T5 49864601 IC50 = 1180 nM T16691 C90MTG 49864602 IC50 = 644 nM T16691 C5BCS4 49864722 IC50 = 7 nM T16691 CKZO79 49864723 IC50 = 4 nM T16691 C74LZS 49864724 IC50 = 3 nM T16691 C2RY0J 50878551 Ki = 84 nM T16691 C1W6TV 50898777 Ki > 10000 nM T16691 CXMZ73 50898778 Ki > 10000 nM T16691 C8TA1J 51003550 IC50 = 28 nM T16691 CQ1UJ7 51003551 IC50 = 8 nM T16691 CGMI37 51003586 IC50 = 9 nM T16691 CE4KP1 51050257 Ki > 10000 nM T16691 C1DSG2 52912973 Ki = 8.2 nM T16691 CMJ5W7 52912975 Ki = 60 nM T16691 C2SCZ1 52913102 Ki = 4.1 nM T16691 C4JCT8 52913104 Ki = 1.8 nM T16691 C96RXD 52913108 Ki = 1.5 nM T16691 CPWJ93 52913218 Ki = 7.2 nM T16691 C0HSY1 52913224 Ki = 11 nM T16691 CF84CP 52913226 Ki = 35 nM T16691 C9HLS4 52913228 Ki = 6.3 nM T16691 CPFA98 52914691 Ki = 0.28 nM T16691 C1DQA4 52915868 Ki = 68.4 nM T16691 CBJS54 52915869 Ki = 2600 nM T16691 CB3UK9 52915979 Ki = 764 nM T16691 CZ2JV5 52915980 Ki = 489 nM T16691 CKA21J 52915982 Ki = 2200 nM T16691 C6G2KC 52915983 Ki = 1380 nM T16691 CL8C4Z 52915984 Ki = 2960 nM T16691 CRW65Z 52918030 Ki = 2.138 nM T16691 CP5LJ0 52918031 Ki = 7.586 nM T16691 CT8XL4 52918032 Ki = 0.2692 nM T16691 CYJM62 52940867 Ki = 1.698 nM T16691 CRI12K 52942395 Ki = 16 nM T16691 C08VZD 52945114 Ki = 90 nM T16691 C0UH4W 52945634 Ki = 1.413 nM T16691 C4PY3N 52945783 Ki = 0.7079 nM T16691 C9N6JV 52946845 Ki = 1 nM T16691 CA6H5W 52946846 Ki = 0.7943 nM T16691 CW0M1K 53259021 Ki = 2.9 nM T16691 CW2LS0 53303985 Ki = 0.75 nM T16691 CY92LZ 53310757 Ki = 10 nM T16691 C7GO1V 53316820 Ki = 3.4 nM T16691 C74VWQ 53316984 Ki = 0.5623 nM T16691 CK67HM 53317295 Ki = 30.2 nM T16691 CD1NU6 53317398 IC50 = 47 nM T16691 C02MWG 53318109 Ki = 1.4 nM T16691 C7V0JR 53318111 Ki = 12 nM T16691 CZP8O0 53318142 Ki = 24 nM T16691 C39KVU 53318267 Ki = 37.15 nM T16691 CY21CF 53318300 Ki = 114.82 nM T16691 C9ERL2 53318694 IC50 = 15 nM T16691 C2TI4Y 53319229 IC50 = 129 nM T16691 CLX9O5 53319441 Ki = 2.8 nM T16691 CI2M1K 53319443 Ki = 17 nM T16691 C5ZD7H 53319475 Ki = 44 nM T16691 C2VS1D 53319627 Ki = 7.943 nM T16691 CU6C0J 53319628 Ki = 3.89 nM T16691 CB3H8N 53319629 Ki = 9.55 nM T16691 C61DNP 53320009 IC50 = 26 nM T16691 C9ZDR5 53320010 IC50 = 61 nM T16691 CP6JY7 53320011 IC50 = 42 nM T16691 C8L9UI 53320746 Ki = 17 nM T16691 C8XA1F 53320775 Ki = 2.9 nM T16691 CKO65P 53320926 Ki = 3.236 nM T16691 CI5X2B 53320927 Ki = 15.14 nM T16691 CH5MP9 53320928 Ki = 37.15 nM T16691 C8HIW1 53320929 Ki = 1.995 nM T16691 CG98LC 53321318 IC50 = 165 nM T16691 C95JEG 53321319 IC50 = 58 nM T16691 C1EDO9 53322082 Ki = 24 nM T16691 CT34MP 53322258 Ki = 0.2818 nM T16691 CXR3D2 53322259 Ki = 3.162 nM T16691 C2Q5BC 53322547 Ki = 15.9 nM T16691 C5E6PM 53322548 Ki = 7.8 nM T16691 CME93W 53322637 IC50 = 353 nM T16691 CQLK01 53322638 IC50 = 11 nM T16691 C8FET1 53322935 Ki = 1.175 nM T16691 CG05WD 53323402 Ki = 0.24 nM T16691 CI1E4P 53323436 Ki = 12 nM T16691 CW8E9X 53323439 Ki = 4.8 nM T16691 CWP1D3 53323441 Ki = 107 nM T16691 CDV8Y5 53323599 Ki = 131.83 nM T16691 CCWQ31 53323600 Ki = 44.67 nM T16691 C1COV0 53323601 Ki = 11.75 nM T16691 C3I0AS 53323873 Ki = 25.5 nM T16691 C29PDB 53323972 IC50 = 17 nM T16691 C32YWL 53324045 Ki = 1695 nM T16691 CR4W9L 53324553 Ki > 10000 nM T16691 CG46AB 53324895 Ki = 154.88 nM T16691 C5WA0M 53324896 Ki = 1.445 nM T16691 C5BO0F 53324933 Ki = 22.91 nM T16691 CBHG43 53325160 Ki = 23.2 nM T16691 CRQF15 53325242 Ki = 1671 nM T16691 CNWH58 53325265 IC50 = 43 nM T16691 CKTW17 53325266 IC50 = 419 nM T16691 C4BM0X 53325267 IC50 = 7 nM T16691 CCE93D 53325519 Ki = 3.981 nM T16691 C0LRC8 53325577 Ki = 27 nM T16691 C87RZQ 53326022 Ki = 14 nM T16691 CMO38N 53326048 Ki = 65 nM T16691 C3G4ZS 53326175 Ki = 3.802 nM T16691 CNS74M 53326176 Ki = 0.2399 nM T16691 C5F2MI 53326177 Ki = 0.4786 nM T16691 CE6KO2 53326178 Ki = 0.6026 nM T16691 CTD50L 53326548 IC50 = 311 nM T16691 C7J8ZY 53327611 Ki = 4.4 nM T16691 C3MEG7 53327952 Ki = 8.913 nM T16691 CZL9W7 53327953 Ki = 95.5 nM T16691 CCL48Y 53327973 Ki = 20.89 nM T16691 CT5MJ8 53327974 Ki = 23.99 nM T16691 C5J8IG 53327976 Ki = 28.84 nM T16691 CGV7O2 53327979 Ki = 181.97 nM T16691 C4G7RQ 53327999 Ki = 25.7 nM T16691 CU9ON5 53328000 Ki = 23.99 nM T16691 C1HU7Y 53328001 Ki = 168 nM T16691 CD8C0G 54238415 Ki = 2039 nM T16691 C5Z1LN 54579956 IC50 = 2980 nM T16691 C8BSR5 54579957 IC50 = 8910 nM T16691 C9JZ7K 54580137 Ki = 300 nM T16691 CQKO51 54580394 Ki = 123 nM T16691 CYTC09 54580442 Ki = 5.72 nM T16691 CJO04Z 54580942 IC50 = 3240 nM T16691 CTN1V9 54580943 IC50 > 10000 nM T16691 CSK36H 54581122 Ki = 760 nM T16691 C43JTB 54581997 IC50 = 4340 nM T16691 CZ90MU 54581998 IC50 = 43200 nM T16691 CWB48T 54582158 Ki = 110 nM T16691 C5VS4M 54582159 Ki = 160 nM T16691 C8JG0O 54582465 Ki > 1000 nM T16691 CWY0J9 54582938 IC50 = 8360 nM T16691 CGZ2A0 54582939 IC50 = 1040 nM T16691 C63EMH 54582940 IC50 = 1590 nM T16691 C8QLJ2 54583109 Ki = 50 nM T16691 CE2SJ4 54583938 IC50 = 2060 nM T16691 CU2VZ8 54584108 Ki = 81 nM T16691 C2TE0Z 54584885 IC50 = 5800 nM T16691 CCN6S2 54585045 Ki = 78 nM T16691 CM56LK 54585846 IC50 = 10690 nM T16691 CNU5D7 54585847 IC50 = 6400 nM T16691 C03QMG 54585848 IC50 = 7470 nM T16691 C2SDF5 54586019 Ki = 110 nM T16691 COJ5R8 54586020 Ki = 330 nM T16691 C5QTZ6 54586316 Ki > 1000 nM T16691 C39KWS 54586812 IC50 = 15750 nM T16691 CY0G9U 54586813 IC50 > 10000 nM T16691 C4VA8X 54586997 Ki = 150 nM T16691 CD97AP 54752954 Ki = 4.8 nM T16691 CAZ5T6 54764323 Ki = 1950 nM T16691 COZ82F 55479093 Ki = 862 nM T16691 CN5M4X 56593642 Ki = 21.9 nM T16691 CIHK28 56593643 Ki = 119.4 nM T16691 C6B4VJ 56593644 Ki = 196.7 nM T16691 C1HEY6 56593645 Ki = 2.7 nM T16691 CWB5U7 56593646 Ki = 5.6 nM T16691 CL5G1M 56593647 Ki = 17.2 nM T16691 CX3Z4Q 56593797 Ki = 7.9 nM T16691 C3I1DH 56593798 Ki = 4.1 nM T16691 CE0GS3 56593799 Ki = 510.1 nM T16691 CND64S 56593800 Ki < 6 nM T16691 CXS0Y9 56593803 Ki = 49.9 nM T16691 CS7IL1 56593931 Ki = 6.4 nM T16691 C1LZQ6 56593932 Ki = 5.2 nM T16691 C1SUQ3 56593933 Ki = 71.1 nM T16691 C8WHT5 56593934 Ki = 7.2 nM T16691 CA4L8Y 56593935 Ki = 92 nM T16691 CN1QP8 56593936 Ki = 146.6 nM T16691 C4B6PY 56595280 Ki = 33.9 nM T16691 CW89BT 56595402 Ki = 2.8 nM T16691 C93KHG 56595403 Ki = 14.6 nM T16691 CK7F3O 56595404 Ki = 17.8 nM T16691 CE6YT2 56595405 Ki = 24.2 nM T16691 C9YF4L 56595406 Ki = 8 nM T16691 C3H8ED 56595407 Ki = 33.9 nM T16691 C1KA4D 56595408 Ki = 231.1 nM T16691 CDJ2H6 56595409 Ki > 1000 nM T16691 C4C3XQ 56595529 Ki = 23.9 nM T16691 C98WJL 56595531 Ki = 9.3 nM T16691 C42VXP 56595532 Ki > 1000 nM T16691 C14YAC 56595533 Ki = 321.8 nM T16691 C6KMX2 56595534 Ki = 8.2 nM T16691 CF41OI 56595535 Ki = 138.1 nM T16691 CHSO06 56595666 Ki = 18.5 nM T16691 CTXE98 56595667 Ki = 17 nM T16691 CI3V6E 56595668 Ki = 17.9 nM T16691 C6QL1G 56595669 Ki = 27.4 nM T16691 CSV45G 56595670 Ki = 26.6 nM T16691 CQ29HL 56595671 Ki = 7.9 nM T16691 CGK09C 56655504 Ki = 0.302 nM T16691 CM81NH 56655505 Ki = 0.9772 nM T16691 C3XC0S 56665086 Ki = 8.5 nM T16691 C8IE6A 56849575 Ki = 0.2188 nM T16691 C52SBY 56849576 Ki = 0.14 nM T16691 C1SH7I 56849577 Ki = 18.62 nM T16691 CO5T1U 56849578 Ki = 0.5754 nM T16691 C19QNC 56849579 Ki = 0.3467 nM T16691 C7U2DH 56849580 Ki = 69.18 nM T16691 CGDA95 56849581 Ki = 22.39 nM T16691 CN1PJ7 56849713 Ki = 112 nM T16691 CK1X6T 56849714 Ki = 16.6 nM T16691 CUF7Y5 56849715 Ki = 4.365 nM T16691 C9DX8R 56849716 Ki = 1.862 nM T16691 CN4A2H 56849717 Ki = 1.82 nM T16691 C4K3XA 56849719 Ki = 3.09 nM T16691 C16PYF 56849720 Ki = 33.88 nM T16691 C2E7OX 56849856 Ki = 4.677 nM T16691 C6QYO3 56849857 Ki = 0.8913 nM T16691 C1ZG7A 56933434 Ki = 13 nM T16691 CO0N2W 56943599 Ki = 18 nM T16691 C3DF5Z 56943600 Ki = 2.4 nM T16691 C19BDH 56943695 Ki = 25 nM T16691 CS7K3T 56943891 Ki = 71 nM T16691 CZ4L3S 56944082 Ki = 27 nM T16691 C5NI3K 56944086 Ki = 5200 nM T16691 C37BYO 56944186 Ki = 46 nM T16691 C9UOZ6 56944189 Ki = 95 nM T16691 CH7V9J 56944190 Ki = 26 nM T16691 CE49MC 56944191 Ki = 48 nM T16691 CX2RP5 56944287 Ki = 23 nM T16691 CB0P9N 56944383 Ki = 4.1 nM T16691 CEQ7I3 56944384 Ki = 3.3 nM T16691 CHWI01 56944473 Ki = 70 nM T16691 C6Y4ZQ 56944564 Ki = 5 nM T16691 C3B0MZ 56944565 Ki = 100 nM T16691 CI4KW0 56944664 Ki = 87 nM T16691 C39YHD 56944665 Ki = 8.8 nM T16691 C1W3GL 56944666 Ki = 2.4 nM T16691 C7J4UT 56944667 Ki = 140 nM T16691 CZT80U 56944668 Ki = 32 nM T16691 CTW2F5 56944763 Ki = 133 nM T16691 C50WEX 56944764 Ki = 210 nM T16691 CX0ZW2 56944859 Ki = 250 nM T16691 C1ST9U 56944860 Ki = 130 nM T16691 CQKL90 56944861 Ki = 100 nM T16691 CS5J6Y 56944862 Ki = 150 nM T16691 CFLB40 56944863 Ki = 110 nM T16691 C53OTR 56944864 Ki = 210 nM T16691 C5T3RI 56944951 Ki = 280 nM T16691 CR6H7U 56944952 Ki = 92 nM T16691 C1Y2RP 56944953 Ki = 180 nM T16691 C1BH7I 56944954 Ki = 30 nM T16691 CTK9I8 56944955 Ki = 46 nM T16691 CCF1A5 56944956 Ki = 10 nM T16691 C2YVT8 56945042 Ki = 35 nM T16691 CNI2G3 56945043 Ki = 10 nM T16691 CF9V3Q 56945045 Ki = 61 nM T16691 CE4S5M 56945046 Ki = 100 nM T16691 CHN2F6 56949640 Ki > 10000 nM T16691 CP31JY 56963265 Ki < 10 nM T16691 C1TC7Q 56963799 Ki > 10000 nM T16691 C3ZG6J 57325520 Ki = 139 nM T16691 CDK7B0 57325521 Ki = 16650 nM T16691 C3V5EM 57334669 Ki < 20 nM T16691 CSU54I 57334813 Ki < 100 nM T16691 C1PDV8 57334815 Ki < 10 nM T16691 C6VP7I 57334817 Ki < 10 nM T16691 CFNG46 57334819 Ki < 10 nM T16691 CJ23AC 57334821 Ki < 10 nM T16691 CX1AB6 57334823 Ki < 100 nM T16691 C2IY4K 57334968 Ki < 10 nM T16691 C0KP6N 57334970 Ki < 100 nM T16691 CU19GD 57334972 Ki < 10 nM T16691 CIJ0G1 57334974 Ki < 10 nM T16691 CS2O8K 57334976 Ki < 10 nM T16691 CX9W4N 57334978 Ki < 10 nM T16691 C4D6VQ 57335122 Ki < 10 nM T16691 CYS80P 57335124 Ki < 20 nM T16691 CZV73L 57335126 Ki < 100 nM T16691 CIQ08T 57335128 Ki < 100 nM T16691 CR9MZ4 57384073 Ki = 3567 nM T16691 C3HG2F 57390799 Ki = 1010 nM T16691 C83GWU 57391158 Ki = 6548 nM T16691 CS54WD 57391567 Ki = 11 nM T16691 CDL1T9 57391569 Ki = 21 nM T16691 CYD8T2 57391618 Ki = 11 nM T16691 CM8FX7 57391620 Ki = 562 nM T16691 CPE8N4 57391622 Ki = 750 nM T16691 CHG51U 57391624 Ki = 127 nM T16691 C78TOG 57391669 Ki = 49 nM T16691 CJP14X 57391729 Ki = 7.7 nM T16691 CZ28FL 57392612 Ki = 350 nM T16691 CO74HK 57392613 Ki = 4.8 nM T16691 C8OM2N 57392614 Ki = 51 nM T16691 CK89TZ 57392615 Ki = 32 nM T16691 C41ZCO 57393363 Ki = 11 nM T16691 CFI39D 57393365 Ki = 28 nM T16691 C6SO4I 57393467 Ki = 17.5 nM T16691 CJTY79 57393468 Ki = 2.1 nM T16691 CUF40C 57393877 Ki = 2652 nM T16691 CPU53I 57394331 Ki = 7.8 nM T16691 CFRN89 57394332 Ki = 192 nM T16691 CRQ16C 57394333 Ki = 0.74 nM T16691 C3S4KL 57394334 Ki = 0.28 nM T16691 C7VFQ3 57394663 Ki = 147 nM T16691 CN39YP 57395082 Ki = 48 nM T16691 CEW0O4 57395084 Ki = 155 nM T16691 CL96RC 57395086 Ki = 3765 nM T16691 CTG35L 57395190 Ki = 139 nM T16691 CJ15YT 57395598 Ki = 590 nM T16691 C6V3GB 57396088 Ki = 156 nM T16691 C51GCK 57396417 Ki = 17150 nM T16691 CZ2SJ8 57396419 Ki = 24840 nM T16691 C6HBG0 57396813 Ki = 4 nM T16691 CKQH25 57396848 Ki = 32 nM T16691 C92SIX 57396850 Ki = 15 nM T16691 CZ8KA2 57396855 Ki = 1725 nM T16691 CN7QE4 57396857 Ki = 2209 nM T16691 C3L4ED 57396970 Ki = 1.6 nM T16691 CKM78R 57397900 Ki = 54 nM T16691 CYCN81 57397901 Ki > 10000 nM T16691 C51XVB 57398613 Ki = 83 nM T16691 CV1P0K 57398615 Ki = 17 nM T16691 C7W5XA 57398619 Ki = 2757 nM T16691 CY3D5F 57398717 Ki = 22 nM T16691 C2DRP9 57398718 Ki = 5.6 nM T16691 CMA0U2 57398803 Ki = 2.7 nM T16691 CTF76G 57399090 Ki = 825 nM T16691 C0XFB2 57399091 Ki = 2159 nM T16691 CI6ET3 57399092 Ki = 1920 nM T16691 CMX4K5 57399093 Ki = 4587 nM T16691 CR5WK3 57399547 Ki = 91 nM T16691 CUQ14N 57399548 Ki = 52 nM T16691 C3PZ2J 57399549 Ki = 4.6 nM T16691 CAN0W7 57399866 Ki = 10570 nM T16691 C9BG7C 57399868 Ki = 5043 nM T16691 CH0CL2 57400234 Ki = 2 nM T16691 CAI2N9 57400275 Ki = 2.9 nM T16691 CYKA35 57400277 Ki = 385 nM T16691 C5HGO2 57400281 Ki = 397 nM T16691 CWY4G5 57400391 Ki = 18 nM T16691 CQ9KY6 57400392 Ki = 22.3 nM T16691 C4IB3E 57400477 Ki = 46 nM T16691 CT7Q3E 57400828 Ki = 1082 nM T16691 C3D1UP 57400830 Ki = 14460 nM T16691 CC6BP9 57401298 Ki = 37 nM T16691 C5GPJ0 57401515 Ki = 29070 nM T16691 CG8MF3 57401516 Ki = 20410 nM T16691 CP6JM8 57402070 Ki = 38 nM T16691 C2GMY9 57402072 Ki = 203 nM T16691 C7CG1T 57402187 Ki = 16 nM T16691 CN9J5I 57402588 Ki = 1518 nM T16691 CTD09H 57403055 Ki = 814 nM T16691 C75RIG 57403056 Ki = 131 nM T16691 C75KOS 57403057 Ki = 0.68 nM T16691 C4CD2L 57403058 Ki = 0.81 nM T16691 CD2WK3 57403833 Ki = 37 nM T16691 CO24AV 57403835 Ki = 85 nM T16691 CIL3W4 57403837 Ki = 64 nM T16691 C3A1YW 57403839 Ki = 339 nM T16691 CA10YX 57403841 Ki = 1535 nM T16691 CP4OY8 57520121 IC50 = 360 nM T16691 CFW1T3 57520122 IC50 = 440 nM T16691 CQ7GV6 58149665 Ki = 7.7 nM T16691 CC79AK 58149671 Ki > 10000 nM T16691 CUI3O8 58149672 Ki = 35.7 nM T16691 C4Y5KG 58158668 Ki = 20.6 nM T16691 C7CN4T 58158673 Ki = 399.1 nM T16691 CVI3T6 58158682 Ki = 18.5 nM T16691 CRI13V 58158707 Ki = 28.6 nM T16691 C31CYM 58158709 Ki = 31.6 nM T16691 CP9A8Q 58158717 Ki = 160.2 nM T16691 CPME36 58158719 Ki = 14.6 nM T16691 C3VF9E 58158721 Ki = 1.8 nM T16691 C8EVD4 58158738 Ki = 14.2 nM T16691 CK10XC 58158739 Ki = 5.8 nM T16691 C2JP3M 58158748 Ki = 97.2 nM T16691 CN6K3Z 58158749 Ki = 6.1 nM T16691 CBH2G3 59017478 Ki = 1 nM T16691 CZ2E6P 59339309 Ki = 205.9 nM T16691 C2RFW6 59339335 Ki = 7.2 nM T16691 C93KWC 59339383 Ki = 8.7 nM T16691 CKI6R9 60141574 IC50 = 3600 nM T16691 C6AUO2 66800823 Ki = 120 nM T16691 C34ACQ 66800909 Ki = 27 nM T16691 CGT9E6 66800910 Ki = 130 nM T16691 C0QY7D 66800916 Ki = 54 nM T16691 CM58FG 66800926 Ki > 10000 nM T16691 CQ43WD 66800934 Ki = 47 nM T16691 CK0I5J 66800939 Ki = 40 nM T16691 C0X2SF 66800942 Ki = 430 nM T16691 CN30YT 66800947 Ki = 9.2 nM T16691 CZ3MR6 66800959 Ki = 34 nM T16691 C92CMO 66800965 Ki = 320 nM T16691 CFPK92 66800991 Ki = 84 nM T16691 C13GMO 66801000 Ki = 63 nM T16691 CZ1TF9 66801018 Ki = 17 nM T16691 CBO9U3 66801028 Ki = 35 nM T16691 C3K8DC 66801052 Ki = 300 nM T16691 CA4DM3 66801062 Ki = 40 nM T16691 C2OUX9 66801107 Ki = 22 nM T16691 C4J5RZ 66801115 Ki = 110 nM T16691 C1H8BS 66801116 Ki > 10000 nM T16691 C4JGC6 66801120 Ki = 26 nM T16691 CX2GN1 66801139 Ki = 13 nM T16691 C1NG8S 66801140 Ki = 53 nM T16691 CR7OW6 66801158 Ki = 6.2 nM T16691 CJU53X 66801160 Ki = 5.1 nM T16691 CH3BJ8 66801167 Ki = 83 nM T16691 C0AV5M 66801173 Ki = 33 nM T16691 C0V9EF 66801186 Ki = 100 nM T16691 CTHY41 66801210 Ki = 1.8 nM T16691 CSD67P 66801225 Ki = 13 nM T16691 C8J3YU 66801226 Ki = 330 nM T16691 CX45OZ 66801229 Ki = 680 nM T16691 C1S0EV 66801230 Ki = 42 nM T16691 C7S1KY 66801234 Ki = 1.6 nM T16691 CB53AV 66801246 Ki = 100 nM T16691 C3F1TZ 66801251 Ki = 44 nM T16691 CF8O9U 66801259 Ki > 10000 nM T16691 C2Q9FS 66801263 Ki = 29 nM T16691 C7Y9VP 66801267 Ki = 2300 nM T16691 CED17M 66801271 Ki = 66 nM T16691 C41VYW 66801295 Ki = 200 nM T16691 C2FYL1 66801333 Ki = 1100 nM T16691 CS75LK 66801335 Ki = 56 nM T16691 CR2N0J 66801344 Ki = 220 nM T16691 CDH7S9 66801346 Ki = 7.1 nM T16691 CGC4U6 66801354 Ki = 1600 nM T16691 CY4FM5 66801379 Ki = 120 nM T16691 C3RX4C 66801425 Ki = 250 nM T16691 C7JD0I 66801429 Ki = 130 nM T16691 CN8OU1 66801430 Ki = 100 nM T16691 C93EGP 66801455 Ki = 140 nM T16691 COR1H8 66801528 Ki = 67 nM T16691 C1F3YV 66801537 Ki = 20 nM T16691 CIRW86 66801551 Ki = 3.4 nM T16691 C75WXP 66801561 Ki = 200 nM T16691 C8H5PD 66801565 Ki = 23 nM T16691 CT5SP8 66801605 Ki = 45 nM T16691 C8MH0I 66801613 Ki = 15 nM T16691 CC8JV6 66801624 Ki = 180 nM T16691 C3EI2F 66801625 Ki = 350 nM T16691 C49XBJ 66801673 Ki = 1100 nM T16691 C0XG6B 66801701 Ki = 360 nM T16691 C42EBQ 66801837 Ki = 250 nM T16691 CW3AI2 66803474 Ki = 6.4 nM T16691 CPKH06 66803497 Ki = 120 nM T16691 CNJE57 66803500 Ki = 330 nM T16691 CN6FZ1 66803595 Ki = 3.5 nM T16691 CD7Y0H 66852770 Ki = 7.5 nM T16691 CR26JV 67156504 Ki = 5 nM T16691 C1LEH8 67268994 Ki = 248 nM T16691 CLK0B7 68014784 Ki = 48.3 nM T16691 CYHG09 68014793 Ki = 153 nM T16691 CLA7F3 68281136 Ki = 140 nM T16691 C84MZH 68281137 Ki = 4800 nM T16691 CDG8X3 68544797 Ki = 2.82 nM T16691 CV54LO 68638941 Ki = 23.5 nM T16691 CD3U6K 68731121 Ki > 10000 nM T16691 C6IP8Q 69082816 Ki > 10000 nM T16691 CH3A6M 69485025 Ki = 36.3 nM T16691 C9L0TF 70245924 Ki = 0.66 nM T16691 CTE40A 70301391 Ki = 0.93 nM T16691 CC43QK 71151588 Ki = 1 nM T16691 CG5A0O 71151591 Ki = 23 nM T16691 CB4K3V 71151664 Ki = 24 nM T16691 CO8CB3 71151683 Ki = 9.9 nM T16691 C5U2BI 71151704 Ki = 2.3 nM T16691 CU74VQ 71151756 Ki = 11 nM T16691 CVMJ59 71151757 Ki = 2.8 nM T16691 C4AF8X 71151767 Ki = 45 nM T16691 CN05SR 71151870 Ki = 83 nM T16691 CG18YE 71151889 Ki = 12.6 nM T16691 CC9M3F 71151924 Ki = 20 nM T16691 CP9A6W 71151925 Ki = 16 nM T16691 C2V5SX 71151929 Ki = 6.9 nM T16691 CM4QC9 71151933 Ki = 0.4 nM T16691 CYP91I 71151953 Ki = 7.3 nM T16691 CN4AJ3 71152026 Ki = 100 nM T16691 CZM5O9 71163244 Ki = 118 nM T16691 C91SZN 71449641 Ki = 315 nM T16691 C2GCN7 71449642 Ki = 957 nM T16691 CQN93U 71449643 Ki = 327 nM T16691 CEJ3B4 71449644 Ki = 156 nM T16691 C5SAJ1 71449645 Ki = 537 nM T16691 CLM07O 71449795 Ki = 2.85 nM T16691 CM0TQ2 71449796 Ki = 10.4 nM T16691 C6LD8A 71449798 Ki = 13.1 nM T16691 C3XNC2 71450247 Ki = 6256 nM T16691 CI95UR 71450930 Ki = 49 nM T16691 CHT21G 71451454 Ki = 2759 nM T16691 C2QZL4 71451455 Ki = 147 nM T16691 CXI5Q2 71451456 Ki = 3785 nM T16691 CKJZ57 71451457 Ki = 258 nM T16691 C0F1HU 71451458 Ki = 185 nM T16691 CTZ24N 71451459 Ki = 200 nM T16691 C70JUP 71451460 Ki = 202 nM T16691 C10IGU 71451603 Ki = 5.02 nM T16691 C8VXH9 71451605 Ki = 17.12 nM T16691 CYK20Z 71452384 Ki > 10000 nM T16691 CKI58Z 71453278 Ki = 1799 nM T16691 C1QM8D 71453279 Ki = 225 nM T16691 C6O4KT 71453280 Ki = 515 nM T16691 CL49VI 71453281 Ki = 245 nM T16691 CGXT64 71453282 Ki = 551 nM T16691 C65RKA 71453361 Ki = 73.4 nM T16691 CE0R9D 71454275 IC50 > 580000 nM T16691 CGO13Q 71454997 Ki = 410 nM T16691 C0K1JV 71454998 Ki = 177 nM T16691 C3JF1D 71454999 Ki = 240 nM T16691 C2QZ1N 71455000 Ki = 199 nM T16691 C6FE5D 71455001 Ki = 951 nM T16691 C4L0JN 71455002 Ki = 102 nM T16691 CTP83A 71455149 Ki = 4.3 nM T16691 CAQF34 71455625 Ki > 10000 nM T16691 CWR40I 71456780 Ki = 831 nM T16691 CZUX67 71456781 Ki = 267 nM T16691 CZ17FC 71456782 Ki = 248 nM T16691 CKF09U 71456783 Ki = 96 nM T16691 CJKV72 71456784 Ki = 271 nM T16691 C7C2ST 71456942 Ki = 3.63 nM T16691 C35RLC 71456943 Ki = 70.6 nM T16691 CQ6WA2 71456944 Ki = 61.21 nM T16691 CMJ1O9 71457409 Ki > 10000 nM T16691 C37EBC 71458647 Ki = 313 nM T16691 CM6OP1 71458648 Ki = 2124 nM T16691 CRGE05 71458649 Ki = 1779 nM T16691 CJN4S1 71458650 Ki = 91 nM T16691 CNT5J9 71458651 Ki = 504 nM T16691 C3NAM7 71458652 Ki = 357 nM T16691 CR9I8F 71458723 Ki = 39.1 nM T16691 C3RS9W 71458811 Ki = 1.6 nM T16691 CY05VS 71458812 Ki = 4.68 nM T16691 CS83IF 71459269 Ki > 10000 nM T16691 CK5T4P 71459604 Ki > 10000 nM T16691 CG0WO9 71459954 EC50 = 0.4 nM T16691 CT17XB 71460468 Ki = 1761 nM T16691 C63YLA 71461049 Ki > 10000 nM T16691 CJD96I 71461050 Ki > 10000 nM T16691 C7AX1Q 71462178 Ki = 1335 nM T16691 C1CS0Z 71462179 Ki = 102 nM T16691 CDX7M6 71462329 Ki = 5.01 nM T16691 CF15LQ 71462330 Ki = 9.15 nM T16691 C5KJZ7 71462331 Ki = 29.01 nM T16691 C4P3JU 71462776 Ki > 10000 nM T16691 C3GUQ2 71462777 Ki > 10000 nM T16691 CP2SY9 71463515 Ki = 100 nM T16691 CJYW50 71463516 Ki = 84 nM T16691 CB4K0Y 71463517 Ki = 41 nM T16691 CI98TK 71463518 Ki = 2600 nM T16691 CC2PE0 71463519 Ki = 270 nM T16691 CJ57BD 71463520 Ki = 4900 nM T16691 CG4AF3 71463521 Ki = 2900 nM T16691 C1E9HB 71502591 Ki = 13 nM T16691 CE9ZL1 71502631 Ki = 7.6 nM T16691 CQ3EZ2 71502632 Ki = 5.4 nM T16691 CQ8FW4 71502633 Ki = 1.7 nM T16691 CBY90L 71502676 Ki = 3.8 nM T16691 CT2ME3 71574204 Ki = 220 nM T16691 C3SXR5 71574206 Ki = 901 nM T16691 C2YRI9 71574208 Ki = 326 nM T16691 C62RWV 71574210 Ki = 257 nM T16691 CKC53S 71574212 Ki = 1331 nM T16691 CNV42M 71574298 Ki = 555 nM T16691 C9PGQ1 71574300 Ki = 484 nM T16691 C2LXH5 71574302 Ki = 301 nM T16691 C2YPB8 71574304 Ki = 598 nM T16691 CK7GM0 71574306 Ki = 454 nM T16691 C0W2YA 71727193 Ki = 9363 nM T16691 C79TLS 71727194 Ki = 19100 nM T16691 CFB10W 71727195 Ki = 8836 nM T16691 C6CIB5 71727196 Ki = 13600 nM T16691 C7Z3JS 71727308 Ki = 5939 nM T16691 C2W5JT 71727892 Ki = 0.16 nM T16691 CR4Q3A 71769065 IC50 = 1800 nM T16691 CGMN49 71769066 IC50 = 7400 nM T16691 CC07ST 71769190 IC50 = 2900 nM T16691 CFPC45 71769315 IC50 = 6600 nM T16691 C17QTG 71769424 IC50 = 1400 nM T16691 CIZ98N 71770821 IC50 = 2400 nM T16691 C0K8NC 71770822 IC50 = 4740 nM T16691 C6CVD5 71770944 IC50 = 2040 nM T16691 C9PIE1 71813685 IC50 = 5220 nM T16691 CH7IG2 71813833 IC50 = 3280 nM T16691 C0P6JL 71813835 IC50 = 6770 nM T16691 C0TMX6 71813838 IC50 = 1660 nM T16691 C1R0QA 71813986 IC50 = 580 nM T16691 C0A3SV 71813988 IC50 = 7080 nM T16691 C7VP8T 71814155 IC50 = 770 nM T16691 C7I9KL 71814157 IC50 = 310 nM T16691 CL4B0J 71814318 IC50 = 310 nM T16691 C53MXL 71815503 IC50 = 740 nM T16691 C3ATN5 72197484 IC50 = 36.8 nM T16691 C20HSN 72197485 IC50 = 22.2 nM T16691 CN8A5R 72197486 IC50 = 21.8 nM T16691 CL3BF7 72197668 IC50 = 30.4 nM T16691 CUVJ59 72197845 Ki = 63 nM T16691 CIKU20 72198011 Ki = 159 nM T16691 COH95V 72198014 Ki = 264 nM T16691 C0WY2V 72198191 Ki = 1146 nM T16691 CWH6T3 72548703 IC50 = 254 nM T16691 C80VRM 72549033 Ki = 0.22 nM T16691 C8Z0NM 72550642 Ki = 1517 nM T16691 CL6W2Q 72550645 Ki = 1321 nM T16691 C78LYM 72698087 Ki > 10000 nM T16691 C63HPK 72698088 Ki > 10000 nM T16691 CC6Q5R 72771081 Ki < 100 nM T16691 CC65OA 73213195 Ki = 273 nM T16691 CW83DK 73213196 Ki > 10000 nM T16691 CXM8O2 73347306 EC50 = 5.3 nM T16691 C9X8GY 73347307 EC50 = 32 nM T16691 CE2H9S 73347593 Ki = 8.3 nM T16691 CH9M8C 73347610 IC50 = 3600 nM T16691 CR97NO 73347825 Ki > 10000 nM T16691 CY60RD 73347826 Ki > 10000 nM T16691 C9ML2B 73348100 Ki = 12.5 nM T16691 C0V3YM 73349113 Ki = 30.1 nM T16691 CIJ64B 73349123 IC50 = 3800 nM T16691 CVUT85 73350387 EC50 = 6.6 nM T16691 C8GQK9 73350823 Ki = 187 nM T16691 CC8I7X 73351903 EC50 = 32 nM T16691 C0C7PV 73351904 IC50 = 100 nM T16691 CG4M8P 73351905 IC50 = 1000 nM T16691 C1YOX0 73351911 IC50 = 80 nM T16691 C0PT9Z 73353367 IC50 = 100 nM T16691 C89NZA 73353655 Ki = 1.65 nM T16691 CAR7Z5 73354882 EC50 = 2.7 nM T16691 CFI26G 73354883 IC50 = 9 nM T16691 C5N7EC 73356442 EC50 = 21 nM T16691 CET52A 73356443 IC50 = 700 nM T16691 CUB97Z 74538690 Ki = 830 nM T16691 COB03V 74763017 Ki = 15 nM T16691 C2E7QW 75201901 Ki = 8100 nM T16691 C8IDL3 75306277 Ki = 15.85 nM T16691 C45OSP 76284193 Ki = 2518 nM T16691 CIU19B 76328541 IC50 = 330 nM T16691 C9S0XK 86288947 Ki = 10790 nM T16691 CIA2B8 86294717 Ki = 14 nM T16691 CCY5N2 86302554 Ki = 2.6 nM T16691 CHE2U4 90178632 Ki = 148 nM T16691 C86OJA 90468813 Ki = 3 nM T16691 CFDW68 90644074 Ki = 1500 nM T16691 C0T8RE 90644075 Ki = 2200 nM T16691 C2KE9G 90644076 Ki > 10000 nM T16691 C1SOF5 90644077 Ki = 35 nM T16691 CIE9Z2 90644078 Ki = 560 nM T16691 CWMU25 90644511 IC50 = 280 nM T16691 CYB8K4 90644513 Ki = 46.77 nM T16691 C3U1IQ 90645147 Ki = 2707 nM T16691 CVG2C1 90654672 Ki = 282 nM T16691 CJG31T 90654831 Ki = 4139 nM T16691 CMU45O 90654832 Ki = 3071 nM T16691 C14NPE 90654833 Ki = 9600 nM T16691 C3C4BW 90654834 Ki = 25520 nM T16691 C8QWR3 90654835 Ki = 14650 nM T16691 C6ZR9L 90654837 Ki = 4368 nM T16691 C0AC7R 90654839 Ki = 8611 nM T16691 CKLG40 90654841 Ki = 2926 nM T16691 C5JS8D 90654843 Ki = 2506 nM T16691 C4VHZ6 90654845 Ki = 1945 nM T16691 CG78PS 90654847 Ki = 7469 nM T16691 CL39WP 90654849 Ki = 8104 nM T16691 C0TVQ9 90654851 Ki = 1762 nM T16691 C4I1CU 90654853 Ki = 395 nM T16691 CZ28YC 90654855 Ki = 314 nM T16691 CRO83N 90654857 Ki = 2879 nM T16691 CTN1D3 90656153 Ki = 54 nM T16691 C1I3ZB 90656154 Ki = 100 nM T16691 CE6C9U 90656155 Ki = 650 nM T16691 C1Z3PQ 90656156 Ki = 1200 nM T16691 CC95ZU 90656157 Ki = 140 nM T16691 CZ9OD5 90656158 Ki = 70 nM T16691 CIB5P7 90656159 Ki = 84 nM T16691 C30EKW 90656160 Ki = 48 nM T16691 C5TD0H 90656161 Ki = 4100 nM T16691 C6T8KC 90656162 Ki > 30000 nM T16691 CAOR80 90656163 Ki = 55 nM T16691 CN4VR5 90656164 Ki = 4900 nM T16691 CN5TQ9 90656165 Ki = 10 nM T16691 C6S7EM 90656166 Ki = 16 nM T16691 CG7IS2 90656167 Ki = 15 nM T16691 CPQ39B 90656168 Ki = 47 nM T16691 CF8M7I 90656169 Ki = 87 nM T16691 C23VSZ 90656170 Ki = 10 nM T16691 CX24VH 90656171 Ki = 240 nM T16691 CW07FN 90656172 Ki = 140 nM T16691 C5QK6I 90656173 Ki = 1900 nM T16691 C3S9CI 90656174 Ki = 150 nM T16691 CYW04S 90656175 Ki = 330 nM T16691 CCOV98 90664359 Ki = 19460 nM T16691 C4MUI2 90664601 IC50 = 136 nM T16691 CXD5Q9 90664621 Ki = 14420 nM T16691 CWNR05 90664684 IC50 = 780 nM T16691 CHT7D5 90664962 IC50 = 1682 nM T16691 CACG19 90666899 Ki = 213.8 nM T16691 CODM50 90666903 Ki = 354.81 nM T16691 CFEO02 91971999 IC50 = 0.17 nM T16691 CUQ6V0 92042918 Ki < 1000 nM T16691 CPEM50 118456745 IC50 = 2.7 nM T16691 CEMZ15 118464420 Ki = 3031 nM T16691 CV2L6O 118464425 Ki = 4777 nM T16691 CFNG86 118464427 Ki = 5909 nM T16691 C7AMX4 118464990 IC50 = 31 nM T16691 CJ6YV9 118464995 IC50 = 0.92 nM T16691 CNS8P6 118464996 IC50 = 0.5 nM T16691 CUDR52 118464997 IC50 = 1.3 nM T16691 C46JBK 118464998 IC50 = 1 nM T16691 C5MI2D 118465009 IC50 = 2 nM T16691 CYMK37 118465011 IC50 = 0.28 nM T16691 C2D0KT 118465015 IC50 = 3.2 nM T16691 CZ1NX5 118465021 IC50 = 5.5 nM T16691 C0VGE2 118465023 IC50 = 0.46 nM T16691 CU0I6P 118465024 IC50 = 11 nM T16691 CZD43F 118465025 IC50 = 1.6 nM T16691 CR38IZ 118465026 IC50 = 2.6 nM T16691 CG6N7X 118465027 IC50 = 4.1 nM T16691 C13GUZ 118465034 IC50 = 16 nM T16691 CO3W8Q 118465035 IC50 = 1.3 nM T16691 COKX07 118465038 IC50 = 11 nM T16691 CWR0B1 118465045 IC50 = 0.31 nM T16691 CAUL06 118465046 IC50 = 5 nM T16691 C98REJ 118465048 IC50 = 1.4 nM T16691 CKZ50J 118465050 IC50 = 1.7 nM T16691 CQ4RU0 118465051 IC50 = 2.1 nM T16691 CH4E0L 118465054 IC50 = 1.1 nM T16691 C7TEA2 118465055 IC50 = 3.7 nM T16691 C3VZ5N 118465064 IC50 = 1.2 nM T16691 C0TP5K 118465065 IC50 = 2.3 nM T16691 C10IRY 118465087 IC50 = 2.1 nM T16691 CJ29GH 118465171 IC50 = 0.69 nM T16691 CK04PJ 118512792 IC50 = 1420 nM T16691 CX71LC 118512797 IC50 = 10900 nM T16691 C76UQN 118512804 IC50 = 1780 nM T16691 CNE79I 118512805 IC50 = 3300 nM T16691 C78ZFD 118512807 IC50 = 8780 nM T16691 C3AK8G 118512815 IC50 = 2430 nM T16691 CA91YU 118512827 IC50 = 5650 nM T16691 CB5I1A 118512841 IC50 = 4010 nM T16691 CMSN80 118626035 Ki = 82 nM T16691 CT3AI0 118626042 Ki = 2057 nM T16691 CKNJ72 118626045 Ki = 72 nM T16691 CGB42Y 118626088 Ki = 996 nM T16691 C0XJT5 118626089 Ki = 116 nM T16691 CIE4C7 118626101 Ki = 766 nM T16691 C1NYS5 118626120 Ki = 1483 nM T16691 CPG04R 118626121 Ki = 9 nM T16691 C3S5LJ 118626129 Ki = 13 nM T16691 CY3F0N 118626140 Ki = 60 nM T16691 CE07IQ 118626142 Ki = 11 nM T16691 C72OZY 118626161 Ki = 38 nM T16691 CY3E7S 118626169 Ki = 1263 nM T16691 CHRB75 118626208 Ki = 2533 nM T16691 CIM3W2 118712402 Ki = 10 nM T16691 C5IF4Q 118712403 Ki = 99 nM T16691 C93OIS 118712404 Ki = 118 nM T16691 CHT8B0 118712405 Ki = 1 nM T16691 CKRA34 118712406 Ki = 11 nM T16691 C1JG4L 118712407 Ki = 1.2 nM T16691 C6XZC4 118712408 Ki = 3.8 nM T16691 CVL8B4 118712409 Ki = 0.9 nM T16691 C1F9ZM 118724639 Ki = 10350 nM T16691 CE05XG 118727442 IC50 = 1830 nM T16691 C1ZH2I 118727443 IC50 = 4970 nM T16691 C0M5AR 118727444 IC50 = 6340 nM T16691 CDHS51 118727445 IC50 = 2120 nM T16691 CWZ7P0 118727447 IC50 = 1400 nM T16691 CH9V1A 118727448 IC50 = 2440 nM T16691 C6AZG2 118727449 IC50 = 2960 nM T16691 CZ1LD0 118727450 IC50 = 2530 nM T16691 CB97QH 118727451 IC50 = 3900 nM T16691 C5O2NU 118729733 Ki = 5805 nM T16691 C8GKX6 118731351 Ki = 594 nM T16691 CQ8F6C 118731354 Ki = 603 nM T16691 CU12XM 118731356 Ki = 376 nM T16691 CD5RI3 118731502 Ki = 22 nM T16691 C5UQ3P 118731503 Ki = 52 nM T16691 CB6H8O 118731504 Ki = 150 nM T16691 CLFJ64 118731505 Ki = 140 nM T16691 CFPX32 118731506 Ki = 150 nM T16691 CL35UJ 118731507 Ki = 52 nM T16691 CF3TJ0 118731508 Ki = 590 nM T16691 CRBZ61 118731509 Ki = 33 nM T16691 CRJ4A6 118731510 Ki = 490 nM T16691 CCPL16 118731511 Ki = 57 nM T16691 C2POB0 118731512 Ki = 680 nM T16691 CZRB40 118731513 Ki = 62 nM T16691 CED26B 118732439 Ki = 100 nM T16691 C75OXS 118736395 Ki > 1000 nM T16691 C74FCM 118736396 Ki = 86 nM T16691 C3F8PA 118736397 Ki = 839 nM T16691 CWU1A0 121238068 Ki = 20 nM T16691 C8I7TE 121238069 Ki = 95 nM T16691 C5X8MN 122186880 Ki = 627 nM T16691 C7ODW3 122195524 Ki < 300 nM T16691 CBHT01 122377930 Ki = 471 nM T16691 CLW53P 122483274 Ki = 879 nM T16691 C4QM2E 124247485 Ki = 416 nM T16691 CVJR26 125513586 Ki = 450 nM T16691 CX1L8T 126720370 Ki = 165 nM T16691 C8Q3HT 126720389 Ki = 337 nM T16691 CLWM12 126720394 Ki = 7 nM T16691 CH98YW 126720395 Ki = 108 nM T16691 C8Q1JB 126720403 Ki = 13 nM T16691 CB3H1C 126720406 Ki = 165 nM T16691 CU3D1V 126720407 Ki = 92 nM T16691 CHCB04 126720410 Ki = 61 nM T16691 C02ZVU 126720412 Ki = 142 nM T16691 CEQ5C2 126720417 Ki = 21 nM T16691 C1U3SZ 126720425 Ki = 20 nM T16691 CWOK84 126720426 Ki = 57 nM T16691 CQ9Y8F 126720427 Ki = 162 nM T16691 C2QSR6 126720429 Ki = 101 nM T16691 C5G8FD 126720440 Ki = 6 nM T16691 C59SNQ 126720442 Ki = 107 nM T16691 CVL36P 126720443 Ki = 56 nM T16691 C2ZFI0 126720444 Ki = 42 nM T16691 CZN9Q7 126720445 Ki = 254 nM T16691 CT13NH 126720448 Ki = 177 nM T16691 CFG95T 126720449 Ki = 829 nM T16691 CIHZ54 127025242 Ki = 539 nM T16691 CCY7P3 127025243 Ki = 559 nM T16691 CTBN56 127026052 Ki = 74.13 nM T16691 CTYP30 127026133 Ki = 325 nM T16691 C0SZI4 127026515 Ki = 595 nM T16691 CX6EI2 127026750 Ki = 281 nM T16691 C8MC1I 127028408 Ki = 111 nM T16691 C6ARO4 127031618 Ki > 1000 nM T16691 CS16FX 127031619 Ki = 251.2 nM T16691 C34QDL 127032187 Ki = 210.2 nM T16691 C4V7RY 127032188 Ki > 1000 nM T16691 C3H2LU 127032424 Ki = 47.5 nM T16691 CJF14Z 127033666 Ki = 97.1 nM T16691 CZ61LK 127034966 EC50 > 5011.87 nM T16691 CA0SN5 127034967 EC50 > 5011.87 nM T16691 CU49VE 127036186 Ki = 741.31 nM T16691 CG06BD 127036932 Ki = 69.18 nM T16691 CVW71O 127036953 Ki = 131.83 nM T16691 C7N5DF 127037679 Ki = 324 nM T16691 CTE43C 127037681 Ki = 641 nM T16691 CDAE15 127038033 Ki = 233 nM T16691 CES26L 127039755 Ki = 276 nM T16691 CX1W5M 127040442 Ki = 240 nM T16691 C83YZJ 127045665 Ki = 231 nM T16691 C9EH4D 127045870 Ki = 87 nM T16691 C9CRG7 127045871 Ki = 12 nM T16691 C06KDX 127045872 Ki = 129 nM T16691 CRYE28 127045873 Ki = 54 nM T16691 CX84AD 127045874 Ki = 6 nM T16691 C4Q6DY 127046815 Ki = 290 nM T16691 CF4X5D 127046817 Ki = 7 nM T16691 CZU72I 127046818 Ki > 2000 nM T16691 CF4E8W 127046819 Ki = 5 nM T16691 C38UBC 127046963 Ki = 36 nM T16691 CH6W2T 127046982 Ki = 4 nM T16691 C84PLD 127047536 Ki = 15 nM T16691 C17RWQ 127047537 Ki = 7 nM T16691 C7OCX9 127047538 Ki = 8 nM T16691 CJH46E 127047680 Ki = 3 nM T16691 CUC1G6 127047776 Ki = 16 nM T16691 CV1KL4 127047898 Ki = 11 nM T16691 C3BU0X 127047899 Ki = 48 nM T16691 C7W4MF 127047900 Ki = 24 nM T16691 CLK3C5 127047901 Ki = 2 nM T16691 C5M7AB 129103161 Ki = 241 nM T16691 CI4M9Y 129103313 Ki = 17.7 nM T16691 CR0GI7 129103315 Ki = 29.46 nM T16691 C3WIA6 129103318 Ki = 5.55 nM T16691 C51ZGV 129103322 Ki = 6.36 nM T16691 C50GOC 130442480 Ki = 7900 nM T16691 CM04RF 130442572 Ki = 6900 nM T16691 CCL8F6 132495282 Ki = 39.81 nM T16691 CR7TA8 132495283 Ki = 12.59 nM T16691 C4LJ2Y 132503215 Ki = 401 nM T16691 CM8B1L 132525569 Ki = 121 nM T16691 CU5L0K 132525570 Ki = 12 nM T16691 CAVB41 132584404 Ki > 10000 nM T16691 CS0MB3 132938109 Ki = 295 nM T16691 C5BEG9 134129897 Ki = 8 nM T16691 C6Z5UG 134129927 Ki = 50.12 nM T16691 CPR31M 134130034 Ki = 16 nM T16691 C0QU1J 134130058 Ki = 10 nM T16691 CG4X6D 134130069 Ki = 8 nM T16691 CO3IZ2 134130116 Ki = 10 nM T16691 CM1N3J 134130197 Ki = 8 nM T16691 CZ7GB0 134130237 Ki = 10 nM T16691 CV97TW 134130269 Ki = 13 nM T16691 CL2XT1 134130413 Ki = 6 nM T16691 CJFT74 134130472 Ki = 12 nM T16691 C6XHB4 134130475 Ki = 113 nM T16691 CB2V9D 134130529 Ki = 15 nM T16691 C87WMF 134130564 Ki = 2 nM T16691 CDYJ03 134130753 Ki = 3.8 nM T16691 CP95OK 134130920 Ki = 2 nM T16691 C7NVB0 134131115 Ki = 16 nM T16691 C5Z9WG 134131252 Ki = 2 nM T16691 C4TSE6 134131296 Ki = 39 nM T16691 CA6Z0F 134131307 Ki = 4 nM T16691 CK37GX 134131322 Ki = 11.7 nM T16691 CG5H3O 134131347 Ki = 36 nM T16691 CK57YE 134131472 Ki = 0.5 nM T16691 C2M8RI 134131482 Ki = 36 nM T16691 CLW62U 134131970 Ki = 79.43 nM T16691 C0RQC6 134131976 Ki = 927 nM T16691 C7UOA9 134132432 Ki = 25.12 nM T16691 CTS3J4 134133483 Ki = 1623 nM T16691 CC1DO8 134134456 Ki = 614 nM T16691 C2Q3JY 134135516 Ki = 1633 nM T16691 CJG3U0 134136134 Ki = 1152 nM T16691 CFOU70 134136921 Ki = 3.981 nM T16691 C87ZJW 134137152 Ki = 7.943 nM T16691 C08ZBY 134137332 Ki = 1074 nM T16691 CXF52V 134137560 Ki = 652 nM T16691 CN4LI8 134137732 Ki = 721 nM T16691 C50WSG 134137966 Ki = 1.585 nM T16691 C2DK7E 134139144 Ki = 316.23 nM T16691 CRC2V0 134139826 Ki = 1621 nM T16691 CHK39T 134141166 Ki = 745 nM T16691 C6PSI9 134142907 Ki = 3441 nM T16691 C80TGJ 134144864 Ki = 1706 nM T16691 CK5RU9 134145903 Ki = 480 nM T16691 C2E0ID 134146185 Ki = 2215 nM T16691 CZDH24 134147097 Ki = 1 nM T16691 CV0QZ5 134147124 Ki = 1039 nM T16691 CV4WJ5 134147644 Ki = 316.23 nM T16691 C41XSD 134147935 Ki = 2815 nM T16691 CH21YW 134148634 Ki = 158.49 nM T16691 CBU81N 134149168 Ki > 10000 nM T16691 CSE17M 134150535 Ki = 158.49 nM T16691 C6O8QW 134150900 Ki = 199.53 nM T16691 CE6LN3 134151118 Ki = 1506 nM T16691 C2JN8Y 134151729 Ki = 395 nM T16691 CNC39L 134151926 Ki = 158.49 nM T16691 C76BZW 134151980 Ki = 1724 nM T16691 CIV4H5 134152583 Ki = 2634 nM T16691 C42ZDI 134153624 Ki = 125.89 nM T16691 CX4W7F 134153716 Ki = 843 nM T16691 CM6D4G 134155367 Ki = 10 nM T16691 CIUZ94 134155476 Ki = 561 nM T16691 C90QNV 134155645 Ki = 434 nM T16691 C0AE1P 134156091 Ki = 1 nM T16691 CAB4K6 134156305 Ki = 700 nM T16691 C50XNE 134156520 Ki = 413 nM T16691 CUHE07 134157171 Ki = 640 nM T16691 CL6DN0 134157769 Ki = 1336 nM T16691 C6N8GM 135367405 Ki = 109 nM T16691 C6LU0C 135367816 Ki = 360 nM T16691 CD2TH9 135367820 Ki > 10000 nM T16691 C5AMD9 135367857 Ki = 492 nM T16691 C92ZLY 135437144 Ki = 1.3 nM T16691 C8WL0I 135449090 Ki = 1716 nM T16691 C9ZCL5 135458672 Ki = 3213 nM T16691 CTE23K 135464118 Ki = 742 nM T16691 CF7D9Y 135804742 Ki = 1 nM T16691 CUI8Q2 135847967 Ki = 10 nM T16691 CUKO20 136020617 Ki > 10000 nM T16691 COF0U5 136020618 Ki > 10 nM T16691 CF89JI 136030596 Ki > 10000 nM T16691 CE8GB9 136030693 Ki > 10000 nM T16691 C65VFI 136030744 Ki > 10000 nM T16691 C9G2KR 136046098 Ki = 1.259 nM T16691 COIX80 136054961 Ki > 10000 nM T16691 CS0JL5 136118616 Ki = 1409 nM T16691 CHWC38 136118619 Ki = 2306 nM T16691 CLH0V9 136118648 Ki = 3733 nM T16691 C76XEJ 136118649 Ki = 860 nM T16691 C0W1TM 136118658 Ki = 7523 nM T16691 C42FCS 136118661 Ki = 7300 nM T16691 COX1F8 136118729 Ki = 1405 nM T16691 CN3W5O 136123549 Ki = 1 nM T16691 CB12QP 136152964 Ki = 4476.2 nM T16691 CAE39V 136188797 Ki > 10000 nM T16691 CWP0V5 136216703 Ki > 10000 nM T16691 C7FW4R 136239492 Ki > 10000 nM T16691 CC6OP7 136244089 Ki > 10000 nM T16691 CLAP52 136259032 Ki > 10000 nM T16691 CA18HL 137210067 Ki = 22 nM T16691 CHM36P 137631892 Ki = 791 nM T16691 CD65BY 137632931 Ki = 158 nM T16691 CSL7O5 137633065 Ki = 29.6 nM T16691 CLWC06 137633076 Ki = 1.7 nM T16691 CYNQ85 137633569 Ki = 12 nM T16691 CE61HV 137633644 Ki = 150 nM T16691 CO2X7L 137633663 Ki = 385 nM T16691 CU01TV 137633827 Ki = 4 nM T16691 CQW9J6 137633849 Ki = 91 nM T16691 C6LA9R 137633855 Ki = 239 nM T16691 CFP4L9 137634216 Ki = 326 nM T16691 CYD64J 137634238 Ki = 90.5 nM T16691 C8N4SP 137634321 Ki = 36.1 nM T16691 C9RSC0 137634934 Ki = 29.4 nM T16691 CC51JN 137635185 Ki = 28 nM T16691 C3BOD0 137635355 Ki = 2.5 nM T16691 C94VXJ 137635884 Ki = 60 nM T16691 CYL39G 137635979 Ki = 6 nM T16691 CFM92C 137636384 Ki = 5 nM T16691 CG7T3S 137636699 Ki = 49 nM T16691 CLXP71 137636791 Ki = 17.5 nM T16691 CK6SF0 137637392 Ki = 8.8 nM T16691 C8N1EH 137637698 Ki = 64 nM T16691 CDX39B 137637994 Ki = 3802 nM T16691 CXZ5N7 137638969 Ki = 9.2 nM T16691 C17PBG 137640158 Ki = 20 nM T16691 CEA1L2 137640705 Ki = 305 nM T16691 CKL78U 137640727 Ki = 5 nM T16691 CXP45J 137640850 Ki = 289 nM T16691 C7LN2D 137640966 Ki = 28.2 nM T16691 CYB58F 137641062 Ki = 6.9 nM T16691 C3LYX9 137641832 Ki = 36 nM T16691 C5WS6Q 137642134 Ki = 1863 nM T16691 CCQ2D0 137642224 Ki = 22 nM T16691 CBW26M 137642284 Ki = 100 nM T16691 C35ZUH 137643300 Ki = 18.7 nM T16691 CLPC81 137643504 Ki = 29 nM T16691 CR59HE 137643783 Ki = 30 nM T16691 C7J0MK 137644129 Ki = 96.3 nM T16691 C0VXH9 137644304 Ki = 9.2 nM T16691 CWUM83 137644521 Ki = 20 nM T16691 CUEZ28 137644687 Ki = 133 nM T16691 CDA80E 137644790 Ki = 1041 nM T16691 CZE12U 137645373 Ki = 7.79 nM T16691 CE7G2D 137645440 Ki = 58 nM T16691 CZ8CU6 137645501 Ki = 640 nM T16691 CI4J2N 137645924 Ki = 30 nM T16691 CCP38D 137645926 Ki = 1020 nM T16691 CGC4W8 137645927 Ki = 1.3 nM T16691 CVX74E 137646045 Ki = 1 nM T16691 CLT73G 137647199 Ki = 2 nM T16691 CUDM82 137647787 Ki = 11.6 nM T16691 CVOX24 137648172 Ki = 5.7 nM T16691 CP7U1T 137648205 Ki = 277 nM T16691 CJ83AX 137648352 Ki = 398 nM T16691 CN19AD 137648438 Ki = 37.8 nM T16691 CQU92A 137649408 Ki = 11.5 nM T16691 CJCU15 137649536 Ki = 56 nM T16691 CMXI62 137649997 Ki = 6712 nM T16691 CM4YW3 137650127 Ki = 119 nM T16691 C3JKC5 137650191 Ki = 52 nM T16691 C52IRM 137650705 Ki = 445 nM T16691 CP2WU7 137650747 Ki = 4.5 nM T16691 CE0UW8 137650795 Ki = 35.7 nM T16691 CTSB07 137650870 Ki = 348 nM T16691 CKG08R 137650961 Ki = 8279 nM T16691 C24NHR 137651282 Ki = 88 nM T16691 CH96PE 137651330 Ki = 64 nM T16691 CZM2Q5 137651613 Ki = 6.7 nM T16691 CU4S1W 137651887 Ki = 36 nM T16691 CVK26R 137652044 Ki = 2412 nM T16691 CHFK13 137652210 Ki = 266 nM T16691 CZLK69 137652249 Ki = 18.4 nM T16691 C51CGJ 137652310 Ki = 1459 nM T16691 CAE1F8 137652414 Ki = 50 nM T16691 CZ5K3F 137653132 Ki = 55.6 nM T16691 CA7JP5 137653219 Ki = 7.8 nM T16691 C2E3FV 137653850 Ki = 1185 nM T16691 COLJ56 137654026 Ki = 95 nM T16691 CKN9V4 137654042 Ki = 100 nM T16691 CX82HS 137654666 Ki = 250 nM T16691 C0SKV1 137654850 Ki = 52 nM T16691 CX5YF2 137655402 Ki = 4 nM T16691 C4VG0U 137655411 Ki = 309 nM T16691 C48TXI 137655693 Ki = 1828 nM T16691 CK5L7D 137655929 Ki = 440 nM T16691 CV4XE1 137656063 Ki = 16.3 nM T16691 C5D2GX 137656602 Ki = 59.7 nM T16691 CQ3HV5 137656608 Ki = 7.8 nM T16691 CIW45A 137656837 Ki = 5.7 nM T16691 CO3L7F 137656918 Ki = 755 nM T16691 C1UZX3 137657317 Ki = 312 nM T16691 C5V6CH 137657598 Ki = 32 nM T16691 CG07QC 137657740 Ki = 193 nM T16691 CFC57K 137658350 Ki = 194 nM T16691 C72MIH 137658424 Ki = 28 nM T16691 CKVH89 137658916 Ki = 2 nM T16691 C4JO1X 137659244 Ki = 80 nM T16691 C4JVW5 137659459 Ki = 64 nM T16691 CL6Y2M 137659696 Ki = 34.9 nM T16691 CB4HN7 137660291 Ki = 19 nM T16691 CX4D7Y 137660741 Ki = 1016 nM T16691 CA4MT5 137661210 Ki = 1.63 nM T16691 CC1X5S 137661237 Ki = 14.3 nM T16691 CO9R5P 137661730 Ki = 348 nM T16691 C78CZR 137661837 Ki = 31.2 nM T16691 CNA2D1 137662033 Ki = 64 nM T16691 C8ZIY5 137662324 Ki = 365 nM T16691 C0R6XM 138691314 Ki = 1660 nM T16691 CU3Y7W 138691316 Ki = 1349 nM T16691 CH2W4P 138691317 Ki = 3020 nM T16691 CHSC40 138691321 Ki = 2455 nM T16691 C18UZA 138691329 Ki = 4169 nM T16691 C1XWV0 138691338 Ki = 6918 nM T16691 C6LE1A 138691362 Ki > 10000 nM T16691 CN9R4A 138691364 Ki = 7762 nM T16691 C8H2KR 138691366 Ki = 4898 nM T16691 C2Z9CD 139488518 Ki = 6457 nM T16691 CJK95T 139488527 Ki > 10000 nM T16691 CZ6H9M 139488539 Ki = 2951 nM T16691 CAF2H8 139488606 Ki = 2884 nM T16691 C54CIL 139488740 Ki > 10000 nM T16691 CK42UE 142592111 Ki = 2.6 nM T16691 CM03WS 142592130 Ki = 1.9 nM T16691 CL8Y2Z 145949620 Ki = 80 nM T16691 C6IFL5 145950947 Ki = 26 nM T16691 CSA0M6 145951217 Ki = 126 nM T16691 CD69JU 145951815 Ki = 1298 nM T16691 CTPH52 145952652 Ki = 139 nM T16691 CG36FD 145953693 Ki = 62 nM T16691 CF67VS 145953749 Ki = 36 nM T16691 CA2J5S 145954503 Ki = 9000 nM T16691 CRQ16N 145954675 Ki = 0.2 nM T16691 CY71FH 145955674 Ki = 320 nM T16691 C8ZXQ4 145955822 Ki = 33 nM T16691 C6A4BR 145957184 Ki = 42 nM T16691 CGU2Y4 145958161 Ki = 30 nM T16691 C5CH7K 145958329 Ki = 80 nM T16691 C2YCL8 145959790 Ki = 312 nM T16691 C9X7KL 145959871 Ki = 110 nM T16691 CQ9P6R 145960299 Ki = 1251 nM T16691 CBX8F6 145960391 Ki = 49 nM T16691 C67GQI 145961372 Ki = 1837 nM T16691 CEYW94 145961507 Ki = 137 nM T16691 CNVZ94 145961959 Ki = 61 nM T16691 C8BWY4 145962006 Ki = 427 nM T16691 C6QCV1 145962275 Ki = 269 nM T16691 CC75OQ 145962993 Ki = 365 nM T16691 CD45OW 145963033 Ki = 131 nM T16691 C5LJY2 145963274 Ki = 45 nM T16691 CW3K5O 145963649 Ki = 711 nM T16691 C7KC3T 145963830 Ki = 2200 nM T16691 C4Y2AL 145964000 Ki > 5000 nM T16691 CHDN35 145964150 Ki > 10000 nM T16691 C1KH2E 145964159 Ki = 2600 nM T16691 C95NZO 145964427 Ki = 1540 nM T16691 C6T4RY 145964846 Ki > 5000 nM T16691 C12OVL 145965034 Ki > 10000 nM T16691 C9D8IB 145965203 Ki > 5000 nM T16691 CA8KF0 145965309 Ki > 5000 nM T16691 CLP94W 145965668 Ki = 2843 nM T16691 C8TF9G 145965840 Ki = 1693 nM T16691 C5W4LM 145965940 Ki > 10000 nM T16691 C1T4DN 145966418 Ki = 2005 nM T16691 C81VUO 145967771 Ki > 10 nM T16691 CJS56K 145967795 Ki > 10000 nM T16691 CQ8EM6 145969402 Ki = 4737 nM T16691 C1T7GL 145971527 Ki = 1800 nM T16691 C8A2XG 145971561 Ki = 1131 nM T16691 CQJ5O8 145971635 Ki > 10000 nM T16691 CUZ2E9 145971739 Ki = 374 nM T16691 C56RAO 145972025 Ki = 4577 nM T16691 C79TNE 145972796 Ki > 10000 nM T16691 CB3KH0 145973178 Ki = 5 nM T16691 CEOY46 145973577 Ki = 200 nM T16691 CT5CX0 145973771 Ki = 7900 nM T16691 C6XIN0 145974114 Ki > 10000 nM T16691 CW6EX3 145974189 Ki = 268 nM T16691 CD8ZL6 145974750 Ki > 10 nM T16691 C6ZEI2 145974789 Ki = 317 nM T16691 C6PH4F 145975226 Ki > 10000 nM T16691 COY2P3 145975720 Ki = 4744 nM T16691 CL7EX5 145975776 Ki = 2155 nM T16691 C7R2MD 145975905 Ki = 6556 nM T16691 C71CYU 145975946 Ki > 10000 nM T16691 C0V4AL 145975992 Ki = 5285 nM T16691 C2TN8W 145976085 Ki > 10000 nM T16691 C8XFM7 145976120 Ki > 5000 nM T16691 CZ5XK2 145976408 Ki = 5559 nM T16691 C34XME 145976696 Ki = 2427 nM T16691 CXDR94 145977222 Ki > 5000 nM T16691 C8NW7Y 145977256 Ki = 6267 nM T16691 C6BFY7 145977338 Ki > 10000 nM T16691 C0Y6QO 145977799 Ki > 10000 nM T16691 C3BI1R 145978113 Ki > 10000 nM T16691 C8VL3Y 145978472 Ki = 7746 nM T16691 CQU8R0 145978665 Ki > 10000 nM T16691 C6AV9G 145978819 Ki > 10000 nM T16691 C87MSW 145980271 Ki = 1670 nM T16691 CEK60A 145982506 Ki = 2310 nM T16691 CI59TX 145983018 Ki = 3912 nM T16691 CYC58R 145983059 Ki = 130 nM T16691 C4F5OT 145983128 Ki = 641 nM T16691 C5ZG9M 145983139 Ki = 291 nM T16691 CV2GU9 145983144 Ki = 77 nM T16691 C4PKM2 145983390 Ki = 623 nM T16691 CIAF74 145983468 Ki = 344 nM T16691 CE7MF4 145983751 Ki = 1259 nM T16691 CDQ4U7 145983760 Ki = 176 nM T16691 CYW9B2 145983794 Ki = 221 nM T16691 C8I1WG 145983961 Ki = 40 nM T16691 CP5H4D 145984065 Ki = 23 nM T16691 CJ35DM 145984299 Ki = 313 nM T16691 CU7E4M 145984511 Ki = 348 nM T16691 C6JUY0 145984737 Ki = 360 nM T16691 CID02G 145984807 Ki = 2990 nM T16691 CM5X3V 145985050 Ki = 137 nM T16691 CG10LK 145985224 Ki = 457 nM T16691 CFJ9B3 145985233 Ki = 169 nM T16691 C5AOI6 145985289 Ki = 190 nM T16691 CW30NA 145985505 Ki = 92 nM T16691 C7ZRP1 145985527 Ki = 18 nM T16691 C2XY8Q 145985533 Ki = 311 nM T16691 C7NI4X 145985585 Ki = 497 nM T16691 C9LJ5T 145985692 Ki = 40 nM T16691 C7QIX0 145985718 Ki = 949 nM T16691 C6V5QS 145985823 Ki = 45 nM T16691 C07GKD 145985958 Ki = 1810 nM T16691 CCM18E 145986031 Ki = 337 nM T16691 CR0XQ3 145986138 Ki = 104 nM T16691 CNJH37 145986752 Ki = 1400 nM T16691 CUGO10 145988693 Ki = 1680 nM T16691 C4GV8Q 145990586 Ki = 862 nM T16691 CC2G1V 146025727 Ki = 7200 nM T16691 C5ZOJ3 146680920 Ki = 3 nM T16691 CD1CB9 151199471 Ki = 20 nM T16691 C6P3SR 153287553 Ki > 10000 nM T16691 CV9G7Z 153287572 Ki > 10000 nM T16691 CO85KL 153287574 Ki > 10000 nM T16691 CZ1K4D 155510674 Ki = 1716 nM T16691 CC3KP7 155510927 Ki = 2 nM T16691 CM4RB0 155511262 Ki = 55 nM T16691 CNE0U3 155511424 Ki = 109 nM T16691 C9KX6O 155511928 Ki = 433 nM T16691 CXF90M 155512487 Ki = 2 nM T16691 CO68LC 155512944 Ki = 550 nM T16691 CP0W8C 155513247 Ki = 132 nM T16691 C90FST 155513438 Ki = 5 nM T16691 C95QOT 155514378 Ki = 4 nM T16691 C3SQI7 155514459 Ki = 14 nM T16691 C0F8BR 155514505 Ki = 1032 nM T16691 CI4DT8 155514575 Ki = 10 nM T16691 CJUI87 155514774 Ki = 58 nM T16691 CQ9ZH8 155514839 Ki = 18 nM T16691 C4X2RG 155515318 Ki = 60 nM T16691 C3NB0D 155515324 Ki = 3574 nM T16691 CZQ32K 155515399 Ki = 475 nM T16691 C0Q8PR 155515407 Ki = 3187 nM T16691 CWO56B 155515415 Ki = 250 nM T16691 C2TN5D 155515890 Ki = 1461 nM T16691 C7KT0D 155515919 Ki = 10 nM T16691 C13LOV 155515942 Ki = 20 nM T16691 C7OF4C 155516118 Ki = 25 nM T16691 CG5M1O 155516282 Ki = 3666 nM T16691 CCS1D6 155517413 Ki = 20 nM T16691 CW0B5K 155518159 Ki = 25 nM T16691 CY7PH5 155518290 Ki = 24 nM T16691 CYB12O 155518974 Ki = 5765 nM T16691 C2E6UC 155519088 Ki = 18 nM T16691 CCEZ93 155519102 Ki = 23 nM T16691 CQD2J7 155519393 Ki = 101 nM T16691 C2SXT1 155519515 Ki = 374 nM T16691 C0KLD8 155519559 Ki = 2 nM T16691 C07BTO 155519598 Ki = 2214 nM T16691 CUSA24 155519891 Ki > 10000 nM T16691 C5FL7R 155520499 Ki = 494 nM T16691 C8OC3W 155520552 Ki = 237 nM T16691 CQ76MP 155521503 Ki = 9 nM T16691 C1OS6D 155522116 Ki = 34 nM T16691 C98RDQ 155522218 Ki = 435 nM T16691 CHA82N 155522233 Ki = 1696 nM T16691 C2TV4Y 155522487 Ki = 50 nM T16691 CK26JU 155522511 Ki = 693 nM T16691 CP6H1D 155522562 Ki = 624 nM T16691 CUG8L3 155522920 Ki = 23 nM T16691 CUG4Q8 155523121 Ki = 21 nM T16691 CN4Y6C 155523355 Ki = 11 nM T16691 CD9QU6 155523519 Ki = 157 nM T16691 C76ARL 155523771 Ki = 220 nM T16691 C5KYB4 155524228 Ki = 71 nM T16691 CK4B0R 155524491 Ki = 1030 nM T16691 CUO93F 155524808 Ki = 921 nM T16691 CQB0M8 155524884 Ki = 78 nM T16691 C65UZD 155524956 Ki = 507 nM T16691 C7FAU5 155525318 Ki = 6 nM T16691 CG2ZS4 155525596 Ki = 522 nM T16691 CZ81JA 155526026 Ki = 459 nM T16691 CN6Z4X 155526468 Ki = 44 nM T16691 C1U2XO 155526651 Ki = 999 nM T16691 CS1GY7 155527191 Ki = 199 nM T16691 CI4UY3 155527359 Ki = 145 nM T16691 C10BPO 155527391 Ki = 37 nM T16691 CW68KC 155528355 Ki = 10 nM T16691 CF29DP 155528725 Ki = 152 nM T16691 C7C1EF 155528967 Ki = 697 nM T16691 C5J7AU 155529153 Ki = 111 nM T16691 C9KS5C 155529450 Ki = 52 nM T16691 CKZ25Y 155529679 Ki = 1272 nM T16691 C7UZI1 155530285 Ki = 157 nM T16691 C3X4IA 155530328 Ki = 372 nM T16691 C9PC3D 155530350 Ki = 937 nM T16691 C57ETL 155530553 Ki = 303 nM T16691 CVLC03 155530779 Ki = 76 nM T16691 C98YQF 155531012 Ki = 132 nM T16691 C4W6VC 155531065 Ki = 7 nM T16691 C5HWP4 155531362 Ki = 9 nM T16691 CQ86CH 155531455 Ki = 16 nM T16691 CCT8V9 155531846 Ki = 507 nM T16691 C5XNT1 155532396 Ki = 105 nM T16691 CS86HA 155532544 Ki = 345 nM T16691 CX35QS 155532545 Ki = 79 nM T16691 CFI23P 155532887 Ki = 556 nM T16691 C3W6HV 155532983 Ki = 100 nM T16691 CX6DV4 155533028 Ki = 952 nM T16691 C23GDV 155533534 Ki = 1651 nM T16691 CSY06A 155533573 Ki = 15 nM T16691 C3OEH2 155533648 Ki = 1410 nM T16691 C15RYP 155533660 Ki = 10 nM T16691 CX1U4H 155533704 Ki = 596 nM T16691 CY01GZ 155533850 Ki = 1320 nM T16691 C2GIL4 155533990 Ki = 247 nM T16691 C6ACO9 155534040 Ki = 65 nM T16691 CP3J8B 155534152 Ki = 29 nM T16691 C3L0CP 155534184 Ki = 1030 nM T16691 C9BGE1 155534201 Ki = 30 nM T16691 CG85SB 155534301 Ki = 5253 nM T16691 C3VGT0 155534362 Ki = 1709 nM T16691 CW7SV9 155534575 Ki = 104 nM T16691 C5HS8N 155534670 Ki = 5 nM T16691 C75FSY 155534794 Ki = 8 nM T16691 C6KF4E 155535154 Ki = 452 nM T16691 C14JEX 155535878 Ki = 4 nM T16691 CB79ZW 155536080 Ki > 10000 nM T16691 C5I1JA 155536087 Ki = 1619 nM T16691 C72FLG 155536152 Ki = 128 nM T16691 C7FVE8 155537034 Ki = 6910 nM T16691 C36FRH 155537074 Ki = 14 nM T16691 CD75GP 155537227 Ki = 15 nM T16691 CB8IC7 155538144 Ki = 3467 nM T16691 C5F2GI 155538236 Ki = 1146 nM T16691 C9TIU2 155538367 Ki = 1622 nM T16691 CYC1P3 155538451 Ki = 246 nM T16691 CM08NT 155538716 Ki = 280 nM T16691 CQ69UA 155538814 Ki = 148 nM T16691 C0D6AQ 155538873 Ki = 10 nM T16691 CAT98F 155539483 Ki = 301 nM T16691 CC1VR4 155539573 Ki = 201 nM T16691 C6S8BA 155539600 Ki = 19 nM T16691 C2HE6C 155540062 Ki = 7 nM T16691 C42GUK 155540147 Ki = 603 nM T16691 CJD9C8 155540541 Ki = 186 nM T16691 CCFM15 155540673 Ki = 21 nM T16691 C2OWD4 155540721 Ki = 17 nM T16691 CR2K1T 155540795 Ki = 19 nM T16691 CNU92V 155540807 Ki = 81 nM T16691 COS2E7 155541072 Ki = 7271 nM T16691 CMP8Q2 155541547 Ki = 83 nM T16691 C6SU1V 155541676 Ki = 501 nM T16691 CP7UG2 155541866 Ki = 90 nM T16691 COZ46W 155541871 Ki = 480 nM T16691 C58YSH 155542160 Ki = 4.8 nM T16691 CB62ZS 155542237 Ki = 21 nM T16691 CX61OI 155542267 Ki = 219 nM T16691 CXCW81 155542321 Ki = 11 nM T16691 C9FS3Y 155542461 Ki = 14 nM T16691 CGC1P6 155543054 Ki = 334 nM T16691 CUI2G9 155543192 Ki = 556 nM T16691 CDO05U 155543223 Ki = 266 nM T16691 CT6HY4 155543250 Ki = 245 nM T16691 C68MSK 155543653 Ki = 118 nM T16691 CIEQ43 155543869 Ki = 31 nM T16691 CZ7O0A 155544139 Ki = 355 nM T16691 CD84VK 155544810 Ki = 1681 nM T16691 CP54KO 155544836 Ki = 102 nM T16691 C2XZD8 155545087 Ki = 225 nM T16691 CO9X1Z 155545526 Ki = 263 nM T16691 CI0YL8 155545625 Ki = 7079 nM T16691 CFQE48 155545832 Ki = 13 nM T16691 C86MKF 155546176 Ki = 175 nM T16691 C74GFO 155546189 Ki = 710 nM T16691 CJBP49 155546194 Ki = 128 nM T16691 CH3W9N 155546350 Ki > 10000 nM T16691 C1SVX6 155547259 Ki = 8.2 nM T16691 CD02EN 155547436 Ki = 347 nM T16691 COJ27N 155547693 Ki = 207 nM T16691 CM4XB6 155548127 Ki = 4.6 nM T16691 CJ7AL8 155548205 Ki = 71 nM T16691 CAT9X4 155548275 Ki = 107 nM T16691 C5LYE8 155548677 Ki = 21 nM T16691 C87JGN 155549153 Ki = 585 nM T16691 CGP8O5 155549315 Ki = 3270 nM T16691 C52FRY 155549978 Ki = 971 nM T16691 CU93YK 155550351 Ki = 12 nM T16691 CY34NR 155550580 Ki = 28 nM T16691 CHXB35 155551102 Ki = 21 nM T16691 C8HPN7 155551113 Ki = 1726 nM T16691 CYOW72 155551197 Ki = 418 nM T16691 CUZJ87 155551219 Ki = 12 nM T16691 C61IVC 155551353 Ki = 407 nM T16691 CHS71N 155551685 Ki = 920 nM T16691 CMCG80 155551834 Ki = 22 nM T16691 C6E9LK 155552054 Ki = 1699 nM T16691 CA1WS9 155552212 Ki = 918 nM T16691 CY94BV 155552356 Ki = 440 nM T16691 CMS62Z 155552380 Ki = 23 nM T16691 CF40VB 155552641 Ki = 69 nM T16691 CDQ7C2 155552798 Ki = 2045 nM T16691 CPV35U 155552826 Ki = 6062 nM T16691 CT23YW 155553005 Ki = 1463 nM T16691 C6STK4 155553745 Ki = 1034 nM T16691 C48LRX 155554020 Ki = 289 nM T16691 CDV6B9 155554036 Ki = 129 nM T16691 CL3FC8 155554246 Ki = 264 nM T16691 CKF75H 155554324 Ki = 689 nM T16691 C6ZSU3 155554462 Ki = 26 nM T16691 C0P6IW 155554556 Ki = 240 nM T16691 CCA21K 155554569 Ki = 2.3 nM T16691 CRY82F 155554955 Ki = 42 nM T16691 CC70RV 155555136 Ki = 8 nM T16691 CLN79H 155555200 Ki = 527 nM T16691 C1RCM0 155555224 Ki = 60 nM T16691 CWL03Q 155555238 Ki = 9 nM T16691 C5Q4UP 155555402 Ki = 2.7 nM T16691 C2E5TR 155555506 Ki = 61 nM T16691 CUNK28 155555525 Ki = 9 nM T16691 CF6R7E 155556168 Ki = 58 nM T16691 CO52HW 155556527 Ki = 794 nM T16691 C1N5VF 155556756 Ki = 50 nM T16691 C2GE4Q 155557005 Ki = 0.43 nM T16691 C5QYS0 155557134 Ki = 476 nM T16691 C59EUZ 155557143 Ki = 210 nM T16691 CD2L3K 155557443 Ki = 3802 nM T16691 CER48T 155557500 Ki = 455 nM T16691 C64EMC 155557523 Ki = 82 nM T16691 CJ0LE3 155557661 Ki = 419 nM T16691 C6END5 155557760 Ki = 7 nM T16691 CHC8S1 155557772 Ki = 11 nM T16691 CF08HV 155557890 Ki = 531 nM T16691 CJZ12T 155558380 Ki = 254 nM T16691 CF6H3V 155558408 Ki = 911 nM T16691 C06BZW 155559811 Ki = 129 nM T16691 CFU9P0 155560188 Ki = 14 nM T16691 C1Z2GD 155560272 Ki = 594 nM T16691 CL4I0D 155560922 Ki = 13 nM T16691 COG70U 155560942 Ki = 3 nM T16691 C2HF6P 155561581 Ki = 242 nM T16691 C5O8AU 155561865 Ki = 759 nM T16691 COL7N8 155561901 Ki = 3467 nM T16691 CXPT57 155561906 Ki = 112 nM T16691 CL45NV 155561914 Ki = 1128 nM T16691 CW7M1D 155561995 Ki = 728 nM T16691 CRTD49 155562063 Ki = 486 nM T16691 C93KWN 155562202 Ki = 671 nM T16691 CO3C6L 155562423 Ki = 31 nM T16691 C5AI0S 155562519 Ki = 85 nM T16691 C4ZA0Q 155562620 Ki = 13 nM T16691 C5BQ8U 155562652 Ki = 690 nM T16691 C5E6BI 155562755 Ki = 45 nM T16691 CF6B4W 155562834 Ki = 182 nM T16691 CZ6IA2 155562918 Ki = 87 nM T16691 CRCW25 155562997 Ki = 29 nM T16691 CBH14K 155563164 Ki = 83 nM T16691 CG1L8E 155563286 Ki = 5888 nM T16691 C38WXS 155563374 Ki = 9 nM T16691 C0INS4 155563826 Ki = 93 nM T16691 C2QLX9 155565138 Ki = 25 nM T16691 CIB3R0 155565292 Ki = 74 nM T16691 C2MIU5 155565813 Ki = 2 nM T16691 C7P5VG 155566191 Ki = 3 nM T16691 C7O6YP 155566439 Ki = 235 nM T16691 CU46EB 155566665 Ki = 3 nM T16691 CEV3B9 155566852 Ki = 25 nM T16691 C67LAG 155566854 Ki = 14 nM T16691 CW1TN7 155566925 Ki = 794 nM T16691 C41UWT 155567307 Ki = 1916 nM T16691 C6I5QA 155567666 Ki = 170 nM T16691 CW3Q7C 155567905 Ki = 18 nM T16691 CA68TK 155568224 Ki = 126 nM T16691 C4EX7C 155568246 Ki = 427 nM T16691 C6V5KP 155568249 Ki = 247 nM T16691 CP03VZ 155568299 Ki = 9 nM T16691 CVU42Z 155568628 Ki = 125 nM T16691 CXP3E4 155568794 Ki = 121 nM T16691 CB5IP9 155569021 Ki = 1860 nM T16691 C0CZK6 155569337 Ki = 18 nM T16691 CP9V7M 155569396 Ki = 1380 nM T16691 C3ZNX6 155569414 Ki = 2352 nM T16691 CZ8RV4 155569568 Ki = 67 nM T16691 C3N9VU 10251906 Ki = 73 nM T16691 CP9TR0 10324985 Ki = 120.3 nM T16691 D00AVR 135476741 Ki = 8768 nM T16691 D00CRA 1574 Ki = 46 nM T16691 D00DZY 11849201 Ki = 4000 nM T16691 D00GSD 25107716 Ki = 1571 nM T16691 D00OBS 44559159 Ki > 10000 nM T16691 D00OCC 9948345 Ki = 1.2 nM T16691 D00VRV 10171 Ki = 17 nM T16691 D01DCE 44401620 Ki = 4200 nM T16691 D01KAX 135453290 Ki > 10000 nM T16691 D01KVG 9843179 Ki = 524.81 nM T16691 D01TYJ 44405257 Ki = 980 nM T16691 D01WWC 16573 Ki = 306 nM T16691 D01ZMO 44401549 Ki = 11800 nM T16691 D02JFD 6918649 Ki = 0.7 nM T16691 D02SBM 49836719 Ki = 27 nM T16691 D02UWB 1809 Ki = 720 nM T16691 D02VHJ 21071574 Ki = 10 nM T16691 D02YSX 197033 Ki = 26 nM T16691 D03DET 10287730 Ki < 10000 nM T16691 D03LPH 107838 Ki > 5000 nM T16691 D03TDN 1342 Ki = 100 nM T16691 D03TSY 24825775 Ki > 1000 nM T16691 D04AQE 1833 Ki < 50 nM T16691 D05DAF 11849198 Ki = 2840 nM T16691 D05EQG 5265 Ki = 1595 nM T16691 D05GDP 599482 Ki > 10000 nM T16691 D05HJP 6476992 Ki = 640 nM T16691 D05JPG 44401277 Ki = 3 nM T16691 D05SAP 11849791 Ki = 290 nM T16691 D05XGR 6918647 Ki = 5 nM T16691 D06FXO 10042892 Ki = 13 nM T16691 D06QVB 44390054 Ki = 34 nM T16691 D06VDN 443391 IC50 = 667 nM T16691 D07DCN 11849196 Ki = 62 nM T16691 D07LIE 11849199 Ki = 50 nM T16691 D07LRJ 5312149 Ki = 0.631 nM T16691 D08BCF 5011 Ki = 3600 nM T16691 D08OFG 11177588 Ki > 10000 nM T16691 D08SMK 14571158 Ki = 8 nM T16691 D08VGJ 9904281 Ki = 1157 nM T16691 D09HJL 10331436 Ki = 2200 nM T16691 D09LVG 44401550 Ki = 4470 nM T16691 D09RPR 16737207 Ki > 10000 nM T16691 D09RXU 45488131 Ki = 31 nM T16691 D09VSK 4301799 Ki = 2530 nM T16691 D09WIL 10028436 Ki = 851.14 nM T16691 D0B1KT 15953802 Ki = 100000000 nM T16691 D0C4AE 10246639 Ki = 91 nM T16691 D0C5GF 6918515 Ki = 20 nM T16691 D0C5XQ 1832 Ki = 13 nM T16691 D0C8UV 5113605 Ki = 6.9 nM T16691 D0CK9K 6918513 Ki = 16 nM T16691 D0CY6E 44414681 Ki = 37 nM T16691 D0D2XH 44413494 Ki = 3.3 nM T16691 D0D3YN 1238 Ki < 50 nM T16691 D0D6FC 15281645 Ki = 38 nM T16691 D0E0DR 11849194 Ki = 21 nM T16691 D0F0IA 11301655 Ki > 2000 nM T16691 D0F1FN 15893127 Ki > 5000 nM T16691 D0F6CD 5202 Ki = 33 nM T16691 D0F6GP 49836621 Ki = 4.9 nM T16691 D0FF6S 16038374 IC50 > 10000 nM T16691 D0FV7K 19779451 Ki = 8200 nM T16691 D0G6NV 44413495 Ki = 1.8 nM T16691 D0G7QT 10131112 IC50 = 7.4 nM T16691 D0H0IZ 11849794 Ki = 70 nM T16691 D0H3WJ 44435193 Ki = 1200 nM T16691 D0H5EP 44388931 Ki = 12 nM T16691 D0H7PC 6918553 Ki = 2.6 nM T16691 D0H9QG 5312148 Ki < 15848.93 nM T16691 D0I9IF 56655571 Ki = 0.2089 nM T16691 D0J6JT 1355 Ki = 2300 nM T16691 D0J7EM 24776941 Ki = 90 nM T16691 D0J9MP 11849197 Ki = 230 nM T16691 D0JT3M 20722800 Ki = 32 nM T16691 D0K5NZ 68848 Ki = 776 nM T16691 D0KS0I 24894910 EC50 > 10000 nM T16691 D0L5MW 181743 Ki = 257 nM T16691 D0L7PA 3248571 Ki = 2.512 nM T16691 D0LA4I 44401621 Ki = 740 nM T16691 D0N7NK 10202564 EC50 = 0.06457 nM T16691 D0N8AO 11849789 Ki = 85 nM T16691 D0O3GF 1220 Ki > 10000 nM T16691 D0O3GQ 11849796 Ki = 115 nM T16691 D0OG0R 10337743 Ki = 4.8 nM T16691 D0P8JA 5312145 IC50 = 26.3 nM T16691 D0PQ1U 11818252 Ki = 3 nM T16691 D0Q7AF 6918836 Ki = 0.2 nM T16691 D0R3GW 10296414 Ki < 10000 nM T16691 D0R7VT 44263491 Ki = 10 nM T16691 D0S4XR 25263303 Ki = 1.3 nM T16691 D0SJ6E 44438719 Ki = 2.5 nM T16691 D0T7VZ 44397102 Ki = 6 nM T16691 D0TG0I 10154392 Ki = 0.3 nM T16691 D0TX8W 594590 Ki = 2700 nM T16691 D0V2PB 5312144 Ki = 12 nM T16691 D0V4RP 1346 Ki = 1.2 nM T16691 D0V5AN 44567986 Ki = 29 nM T16691 D0VI0S 49836506 Ki = 134 nM T16691 D0W2HW 6090 Ki = 575 nM T16691 D0W2QN 44403334 IC50 = 300 nM T16691 D0X1IU 44401390 Ki = 6100 nM T16691 D0X6MT 4106 Ki = 0.4 nM T16691 D0XJ6D 10356663 Ki = 12 nM T16691 D0Y1LJ 10017687 Ki = 25 nM T16691 D0Y4WH 9840311 Ki = 5 nM T16691 D0Y9TL 13702393 Ki > 10000 nM T16691 D0ZC9Q 44393574 Ki = 1900 nM T39921 D0A9KI 9863367 IC50 = 160 nM T39921 D0T3ME 156422 IC50 = 58 nM T39921 C61KPI 24856363 IC50 = 53 nM T39921 CH1YI6 24856364 IC50 = 27 nM T39921 C9VXN3 44578709 IC50 = 6 nM T39921 CDC2V8 44593640 IC50 = 88 nM T39921 C69HNG 56967399 IC50 = 200 nM T62974 D02XIY 448601 Ki = 66 nM T62974 D0TV0C 9941444 Ki < 100 nM T62974 D06JFI 11251755 IC50 = 1.8 nM T62974 D0J8PI 158782 IC50 > 1000 nM T62974 D09JXL 5311430 Ki < 1000 nM T62974 D0Y2HR 2247 Ki > 10000 nM T62974 C6XYL5 6918011 Ki < 1000 nM T62974 CHM63P 6918026 Ki = 158.49 nM T62974 CR0U6E 9827283 Ki = 6840 nM T62974 CA8UQ7 9848232 Ki > 10000 nM T62974 CTRI07 9852911 Ki = 1100 nM T62974 C9BJ3Q 9854636 IC50 = 0.84 nM T62974 CS2D0V 9872511 Ki = 118 nM T62974 C71BKL 9893924 Ki = 6 nM T62974 CMLP16 9918828 Ki < 100 nM T62974 CRP01W 9959684 Ki = 413 nM T62974 C3Z5YJ 9963342 Ki = 501.19 nM T62974 CIT57N 9985523 Ki = 1700 nM T62974 C64LIB 10009650 Ki = 100 nM T62974 C58EOI 10053855 Ki = 1400 nM T62974 CL6G0Z 10094509 Ki = 5010 nM T62974 C9C7RK 10096510 Ki > 10000 nM T62974 CFZN71 10166743 Ki = 3840 nM T62974 CI21CK 10179247 Ki > 10000 nM T62974 C6DRE9 10210016 Ki > 10000 nM T62974 C4M9GN 10248767 Ki > 10000 nM T62974 CSY5K2 10325243 Ki = 2000 nM T62974 C67NLY 10369961 Ki = 16 nM T62974 CL87OB 10411795 Ki > 10000 nM T62974 CP2S9D 10436888 Ki = 14 nM T62974 C0YFD4 10505242 Ki = 4200 nM T62974 CN3IV5 10528970 Ki = 7000 nM T62974 CJ40IE 10531093 Ki = 53 nM T62974 CS96ON 10534086 IC50 = 1000 nM T62974 CRZ9I3 10553122 Ki = 4000 nM T62974 CB2NK4 10554498 Ki = 70 nM T62974 CA1VI4 10554709 Ki = 1000 nM T62974 CHZ9I8 10554930 Ki = 3000 nM T62974 CY3ZE9 10577746 IC50 = 1047 nM T62974 CIY02U 10578474 Ki = 477 nM T62974 C9C0HF 10580397 Ki = 500 nM T62974 CUW4E5 10601454 Ki = 2000 nM T62974 CD8ZW7 10602230 Ki = 476 nM T62974 CVY6D0 10603005 Ki = 1200 nM T62974 CGZ6W8 10625454 Ki = 176 nM T62974 C0SXF1 10625762 Ki = 1000 nM T62974 CU3DQ6 10630127 Ki = 1000 nM T62974 C15AHJ 10650427 Ki = 1700 nM T62974 C7AX8J 10650940 Ki = 132 nM T62974 C5UOS4 10698494 Ki = 185 nM T62974 CT81RB 10698706 Ki = 15000 nM T62974 C45JIZ 10699714 Ki = 2000 nM T62974 CG2UX4 10701257 IC50 = 1000 nM T62974 C27FVZ 10720221 Ki = 7000 nM T62974 CP0F7C 10724811 IC50 = 1000 nM T62974 C3TMY5 10724880 IC50 = 1000 nM T62974 CK7R2B 10745635 Ki = 1400 nM T62974 CJM47E 10748701 IC50 = 1000 nM T62974 CWF2N5 10748831 IC50 = 943 nM T62974 CLQ07H 10768264 Ki = 803 nM T62974 C4X2CO 10769191 Ki = 514 nM T62974 CLW4V6 10770814 Ki = 1900 nM T62974 CO56HI 10772403 IC50 = 1000 nM T62974 CGN0Z5 10772578 IC50 = 1000 nM T62974 COY17C 10793795 Ki = 71000 nM T62974 C3L4DH 10796238 IC50 = 1000 nM T62974 C0WND2 10815650 Ki = 113 nM T62974 C61EOJ 10816544 Ki = 1700 nM T62974 C15QGO 10819673 IC50 = 1000 nM T62974 CJ4T3I 10841338 Ki = 520 nM T62974 CFL71O 10843862 IC50 = 1000 nM T62974 CRP17A 10865371 Ki = 1260 nM T62974 CDE2S9 10876118 Ki = 1040 nM T62974 C2PJ1O 10876898 Ki = 630.96 nM T62974 CEV12M 10887003 Ki = 680 nM T62974 CPN29H 10963480 Ki = 890 nM T62974 C6TVQ8 10964197 Ki = 316.23 nM T62974 CU70TI 10974426 Ki = 260 nM T62974 CK5XB4 10974575 Ki = 1200 nM T62974 CXDG12 10996788 Ki < 100 nM T62974 CJAH75 11050695 Ki = 570 nM T62974 C6AW0M 11112736 Ki = 9800 nM T62974 C5JX9W 11125276 Ki = 360 nM T62974 CK1RX4 11136828 Ki = 316.23 nM T62974 CR1JP9 11147505 Ki < 100 nM T62974 C1I9EX 11159133 IC50 = 3 nM T62974 C7REL4 11170698 IC50 = 1.8 nM T62974 CIEM12 11170867 IC50 = 453 nM T62974 CW2JA8 11182381 IC50 = 2.2 nM T62974 CE3GC2 11205475 IC50 = 0.7 nM T62974 CXI32T 11205496 IC50 = 0.88 nM T62974 C2RNJ5 11205515 IC50 = 1.1 nM T62974 CUT8Z0 11240205 IC50 = 1.8 nM T62974 CK78SD 11240206 IC50 = 1.3 nM T62974 C67WXD 11274767 IC50 = 0.51 nM T62974 COK06N 11320738 IC50 = 2.1 nM T62974 C5D6AM 11332138 IC50 = 0.98 nM T62974 C5PAN4 11343811 IC50 = 4.3 nM T62974 CLQ53A 11355270 IC50 = 3.5 nM T62974 CQ0UC7 11378229 IC50 = 41 nM T62974 CC09ZU 11378299 IC50 = 2 nM T62974 CG7PT9 11389178 IC50 = 1.5 nM T62974 CFJD72 11423410 IC50 = 1.1 nM T62974 C4S2HG 11434734 IC50 = 4 nM T62974 C3T6XG 11442741 Ki = 1.2 nM T62974 C6XHC3 11457491 IC50 = 1.2 nM T62974 CJ5A9B 11457521 IC50 = 1.1 nM T62974 CMA8C7 11468709 IC50 = 3.5 nM T62974 CG8A0J 11468887 IC50 = 1.3 nM T62974 CZ3N5J 11468916 IC50 = 1 nM T62974 CORY59 11480246 IC50 = 0.55 nM T62974 C63QMX 11535351 IC50 = 214 nM T62974 C0R6TS 11548587 IC50 = 440 nM T62974 CF6K7M 11563877 IC50 = 100 nM T62974 CS68YA 11642413 IC50 = 430 nM T62974 CZHN61 11678313 IC50 > 10000 nM T62974 CW65KY 11705763 Ki = 800 nM T62974 CN63YV 11787877 IC50 = 9.5 nM T62974 CR6UF9 11788180 IC50 = 3.5 nM T62974 CK7BN1 11800917 Ki = 96 nM T62974 CK4U8N 11804376 IC50 = 1000 nM T62974 C9XH7F 11815114 Ki < 100 nM T62974 CUI15C 11828523 IC50 = 53 nM T62974 CRA01O 11845058 IC50 = 494 nM T62974 C8X3CL 11845059 IC50 > 1000 nM T62974 CO3HT9 11847587 IC50 = 872 nM T62974 CAD8P9 11848624 Ki > 10000 nM T62974 CM49QW 11848625 Ki > 10000 nM T62974 CEBA46 11848626 Ki > 10000 nM T62974 CCT5G7 11848677 Ki > 10000 nM T62974 CMR10F 11848679 Ki > 10000 nM T62974 C9QDX3 11848833 Ki > 10000 nM T62974 CL6B5X 11848835 Ki > 10000 nM T62974 CW7I8U 13690207 IC50 = 3 nM T62974 C8OU7I 15429504 IC50 = 406 nM T62974 CEO3F0 15585102 IC50 = 8.2 nM T62974 CC2YJ8 16062553 Ki > 10000 nM T62974 C3H1RT 16062555 Ki > 10000 nM T62974 C1LH5T 16062816 Ki > 10000 nM T62974 C1GKF8 16130982 IC50 = 2.3 nM T62974 C2TRA5 16144717 IC50 = 605 nM T62974 CW20OC 16144977 IC50 = 1000 nM T62974 CS6A3Z 16145268 IC50 = 1000 nM T62974 CN3LS1 16145579 IC50 = 1000 nM T62974 C72MUC 16146425 IC50 = 312 nM T62974 CD91IL 16148220 IC50 = 2844 nM T62974 C59OUC 16148481 Ki < 79.43 nM T62974 CJG1X9 16148596 Ki < 1 nM T62974 CNY09C 16148922 Ki < 1000 nM T62974 CP0DC8 16149640 Ki < 0.631 nM T62974 CDPC19 16149975 Ki < 3.981 nM T62974 C0SE6V 16150676 Ki < 0.1995 nM T62974 CSP6A9 16150915 Ki < 0.1 nM T62974 C6N7SR 16151159 Ki < 1.995 nM T62974 C2B9IL 16151570 IC50 = 932 nM T62974 CQM8J1 16151781 IC50 = 1.2 nM T62974 CM8UF7 16151826 IC50 = 562 nM T62974 CJ7UT6 16151923 IC50 = 8.8 nM T62974 CIM03U 16152257 IC50 = 1.9 nM T62974 CU7X6V 16153077 IC50 = 0.9 nM T62974 CK4O1V 16153193 IC50 = 1.2 nM T62974 C16LMW 16153418 IC50 = 2.4 nM T62974 CO0LG7 16154000 IC50 = 2.1 nM T62974 CX4RM8 16154096 IC50 = 1.6 nM T62974 COYU86 16156815 Ki < 1000 nM T62974 CI3FW1 16157160 IC50 = 1000 nM T62974 C7GN0S 16157479 Ki < 0.1995 nM T62974 CQL5O0 16181427 IC50 > 1000 nM T62974 C2CUY9 16181428 IC50 > 1000 nM T62974 CUH8D7 16737812 IC50 = 129 nM T62974 C8QIT3 16737813 IC50 = 75 nM T62974 CNP36U 16737814 IC50 = 3.3 nM T62974 C7Q6JL 16738359 IC50 = 73 nM T62974 CJ9K1C 24740750 Ki > 10000 nM T62974 CS6VO9 24740751 Ki > 10000 nM T62974 CA4K0B 24740752 Ki > 10000 nM T62974 C4N3AX 24740753 Ki > 10000 nM T62974 COQU12 24740861 Ki > 10000 nM T62974 CAD4S1 24740862 Ki > 10000 nM T62974 C67YVI 24740863 Ki > 10000 nM T62974 CO0IF5 24740864 Ki > 10000 nM T62974 C6F1RZ 24777672 IC50 = 141 nM T62974 C5GZO7 24858018 IC50 = 0.9 nM T62974 CV1U7H 24858920 IC50 = 1 nM T62974 C0UB7K 24859055 IC50 = 2.6 nM T62974 CQCW58 24859056 IC50 = 1.3 nM T62974 CT6J2A 24859195 IC50 = 0.7 nM T62974 CUDV69 24859196 IC50 = 4.5 nM T62974 C45NYA 24859341 IC50 = 3.25 nM T62974 C4AB6I 24859342 IC50 = 3.1 nM T62974 CH50QU 24859494 IC50 = 1.9 nM T62974 C8L2KJ 24859495 IC50 = 6 nM T62974 CDS6W5 24859645 IC50 = 2 nM T62974 CHF20D 24859646 IC50 = 3 nM T62974 CKH2R4 24859787 IC50 = 1.5 nM T62974 CT1BM6 24859788 IC50 = 5 nM T62974 C2IKX3 24859919 IC50 = 4.4 nM T62974 C5OQ2X 24859920 IC50 = 2.7 nM T62974 CSZ73L 24860057 IC50 = 2.6 nM T62974 C36ZHQ 24860058 IC50 = 2.2 nM T62974 CVL48C 24860201 IC50 = 1.6 nM T62974 C20ZFS 24860202 IC50 = 1.4 nM T62974 C3C0KP 24894134 EC50 > 50000 nM T62974 CI8BZ6 24936235 Ki = 3200 nM T62974 CHKC79 25187396 IC50 = 7 nM T62974 C4YXJ1 25187398 IC50 = 8.1 nM T62974 CO9PI7 25187400 IC50 = 1.3 nM T62974 C8C9PL 25187679 IC50 = 2.3 nM T62974 C9ECD8 25187681 IC50 = 161 nM T62974 C43OES 25187683 IC50 = 14 nM T62974 CNTB73 25187685 IC50 = 6.9 nM T62974 C1IUQ2 25187953 IC50 = 2.1 nM T62974 CQ3F8L 25187955 IC50 = 35 nM T62974 CS2ZV1 25188218 IC50 = 14 nM T62974 CLI2U1 25188220 IC50 = 1 nM T62974 CNDU95 25188496 IC50 = 2.4 nM T62974 C7KF8N 25188776 IC50 = 56 nM T62974 CCHN50 25188780 IC50 = 7 nM T62974 C3T8DA 25189052 IC50 = 4.4 nM T62974 CI21ED 25189054 IC50 = 59 nM T62974 C97LHK 25189325 IC50 = 2.4 nM T62974 CEG4J0 25189327 IC50 = 17 nM T62974 CSQH26 42637069 IC50 = 95 nM T62974 CJ1S9K 42637136 IC50 = 525 nM T62974 C3NYM8 42637137 IC50 > 1000 nM T62974 CJ47CL 42637210 IC50 > 1000 nM T62974 CR3A8Q 42637283 IC50 > 1000 nM T62974 CENZ47 42637363 IC50 = 250 nM T62974 CX0JC7 42637503 IC50 = 27 nM T62974 C90LHS 42637563 IC50 = 266 nM T62974 C80WBK 42637632 IC50 = 270 nM T62974 CR49YE 42637984 IC50 > 1000 nM T62974 CEFO24 42638065 IC50 > 1000 nM T62974 CF5JK4 42638066 IC50 = 252 nM T62974 CHY04A 44290718 IC50 > 100 nM T62974 C16BKW 44290734 IC50 = 7 nM T62974 CW76YB 44290735 IC50 = 49.5 nM T62974 CA6IS7 44290766 IC50 > 100 nM T62974 C6BZ1J 44298104 Ki > 1000 nM T62974 CCXL10 44298113 Ki = 301 nM T62974 CB9JK1 44298131 Ki > 1000 nM T62974 CJ5WL8 44298155 Ki > 1000 nM T62974 CHL57J 44298156 Ki > 1000 nM T62974 CP61LB 44298165 Ki > 1000 nM T62974 CM0B6J 44298166 Ki > 1000 nM T62974 C8XZR7 44298169 Ki > 1000 nM T62974 C0DPX7 44298171 Ki = 1570 nM T62974 C62OEU 44298177 Ki > 1000 nM T62974 CS9JW8 44298178 Ki > 1000 nM T62974 C20MBI 44298179 Ki = 847 nM T62974 C3QBP0 44298188 Ki = 176 nM T62974 C1R3QD 44298189 Ki = 436 nM T62974 C5RJ7U 44298195 Ki > 1000 nM T62974 C8N3EJ 44298197 Ki > 1000 nM T62974 C1R2SL 44298204 IC50 = 800 nM T62974 CZU05A 44298214 Ki > 1000 nM T62974 CQUS98 44298218 Ki > 1000 nM T62974 COTK07 44298219 Ki > 1000 nM T62974 CAJO07 44298231 Ki = 728 nM T62974 C9S4IX 44298232 Ki = 672 nM T62974 CB1A3K 44298235 Ki = 1040 nM T62974 C2TQ1V 44298248 Ki > 1000 nM T62974 C3WFV5 44298250 Ki = 3310 nM T62974 CL2P9B 44298251 IC50 = 100 nM T62974 CMO1Q9 44298441 Ki > 1000 nM T62974 C8Y9ZP 44298443 Ki = 1590 nM T62974 CUSR45 44298468 Ki > 1000 nM T62974 C8EN2H 44298469 Ki > 1000 nM T62974 CWE7Q0 44298482 IC50 > 1000 nM T62974 CF69PL 44298522 Ki > 1000 nM T62974 CRQJ98 44308836 Ki = 2480 nM T62974 CRFM02 44308969 Ki = 2000 nM T62974 C40MJU 44308970 Ki = 1.76 nM T62974 C9KR7Q 44309052 Ki = 2176 nM T62974 C4YG1S 44311590 IC50 > 1000 nM T62974 CY0OV9 44311591 IC50 = 267 nM T62974 C29GQB 44311601 IC50 = 1.7 nM T62974 CC8DS0 44311602 IC50 > 1000 nM T62974 C5KST2 44311690 IC50 > 1000 nM T62974 C6N4MH 44311691 IC50 > 10000 nM T62974 CIR4G6 44311695 IC50 > 10000 nM T62974 CTG6X5 44311696 IC50 > 1000 nM T62974 C7Y8SF 44311697 IC50 > 1000 nM T62974 CK52MY 44311702 IC50 > 10000 nM T62974 CX39CV 44311703 IC50 > 1000 nM T62974 C5RM2A 44311730 IC50 > 1000 nM T62974 CBG70T 44311731 IC50 > 1000 nM T62974 CQH20F 44311765 IC50 > 10000 nM T62974 CZG4K6 44311836 IC50 = 487 nM T62974 CWNP79 44311837 IC50 > 1000 nM T62974 CEMH98 44311848 IC50 > 1000 nM T62974 CWSF38 44311868 IC50 > 1000 nM T62974 C2T0YP 44311869 IC50 > 10000 nM T62974 C1ONB3 44311870 IC50 > 1000 nM T62974 CXM6D3 44311888 IC50 > 1000 nM T62974 C1LQN0 44311889 IC50 > 1000 nM T62974 C1GY0F 44311912 IC50 > 1000 nM T62974 C14DIH 44311913 IC50 > 1000 nM T62974 C1X4TI 44311914 IC50 = 1.3 nM T62974 C74BDM 44311936 IC50 > 1000 nM T62974 C64WAE 44311958 IC50 > 1000 nM T62974 CFT90E 44311959 IC50 > 1000 nM T62974 C3PQD0 44311960 IC50 > 1000 nM T62974 C3WFS2 44311993 IC50 > 1000 nM T62974 CS7PB4 44312258 IC50 > 10000 nM T62974 C5PE1D 44325273 IC50 = 41 nM T62974 C1P0QV 44332931 Ki > 10000 nM T62974 CX1Y9V 44361984 Ki = 71000 nM T62974 C6UV4B 44362068 Ki = 50 nM T62974 CHP41F 44363816 Ki = 83 nM T62974 CH2DN4 44367916 IC50 > 1000 nM T62974 CM9YQ0 44367953 IC50 = 30 nM T62974 C5W4YL 44368019 IC50 = 14 nM T62974 CO6ZJ9 44368020 IC50 = 61 nM T62974 CQ5T1D 44368043 IC50 = 9.8 nM T62974 C1SWO5 44368044 IC50 = 21 nM T62974 C29EZK 44368080 IC50 = 1.8 nM T62974 C9ZW6U 44368093 IC50 = 11.8 nM T62974 C71URM 44368094 IC50 = 9.2 nM T62974 CC1ZP9 44368109 IC50 > 1000 nM T62974 CQ7OP1 44368112 IC50 = 8.7 nM T62974 C0EW4I 44368117 IC50 = 12 nM T62974 C6TNZ9 44368144 IC50 = 105 nM T62974 C53IAG 44368153 IC50 = 0.53 nM T62974 CKU8J7 44368156 IC50 = 0.7 nM T62974 CR12GB 44368157 IC50 = 1.8 nM T62974 C50DMO 44368226 IC50 = 6.9 nM T62974 CN31HS 44368398 IC50 = 24 nM T62974 C2RC0P 44368406 IC50 = 6.5 nM T62974 CB1HC8 44368422 IC50 = 429 nM T62974 C27DLY 44368489 IC50 = 80 nM T62974 CWHK38 44377332 Ki > 10000 nM T62974 CVH1O7 44377366 Ki > 5000 nM T62974 CRC2N1 44377555 Ki = 7200 nM T62974 CS1WT5 44377591 Ki > 10000 nM T62974 C3LUY8 44377623 Ki > 10000 nM T62974 CQD0P4 44377645 Ki > 5000 nM T62974 CWNF42 44385504 Ki = 3970 nM T62974 CAFD79 44385508 Ki > 10000 nM T62974 CHY14B 44385591 Ki > 10000 nM T62974 CJQI19 44385652 Ki = 7090 nM T62974 CG12HD 44385712 Ki = 5920 nM T62974 C8MU5C 44385757 Ki > 10000 nM T62974 C0LRT9 44386389 Ki = 6660 nM T62974 C1EVK8 44387399 Ki > 1000 nM T62974 C6U9VC 44388027 IC50 > 1000 nM T62974 C2IW5J 44388028 IC50 > 1000 nM T62974 C27ANT 44388029 IC50 = 611 nM T62974 CHQK20 44388035 IC50 > 1000 nM T62974 CI9XS1 44388036 IC50 > 1000 nM T62974 CD4BX6 44388037 IC50 = 215 nM T62974 CDS08Z 44388038 IC50 > 1000 nM T62974 CZA03Y 44388040 IC50 > 1000 nM T62974 C21WBR 44388043 IC50 > 1000 nM T62974 C7VK6B 44388052 IC50 > 1000 nM T62974 CT93BI 44388060 IC50 > 1000 nM T62974 C4E5VS 44388061 IC50 > 1000 nM T62974 C7P5RO 44388066 IC50 > 1000 nM T62974 C7T8IY 44388069 IC50 > 1000 nM T62974 C2TWO3 44388070 IC50 > 1000 nM T62974 CDBE87 44388075 IC50 > 1000 nM T62974 C25GWK 44388078 IC50 > 1000 nM T62974 CT93LV 44388079 IC50 > 1000 nM T62974 CX54SC 44388083 IC50 > 1000 nM T62974 C2C0RU 44388084 IC50 > 1000 nM T62974 C5SMA2 44388085 IC50 > 1000 nM T62974 C26OCG 44388086 IC50 > 1000 nM T62974 C8SR2O 44388087 IC50 > 1000 nM T62974 CHL5T1 44388088 IC50 > 1000 nM T62974 C4VNC2 44388089 IC50 > 1000 nM T62974 C1IH3T 44388090 IC50 > 1000 nM T62974 CNC91I 44388093 IC50 > 1000 nM T62974 CN45OF 44388095 IC50 = 700 nM T62974 C82HJL 44388104 IC50 > 1000 nM T62974 CV6T2H 44388105 IC50 > 1000 nM T62974 CLC0N2 44388106 IC50 > 1000 nM T62974 C0VO1K 44388107 IC50 > 1000 nM T62974 CM5O3B 44388108 IC50 > 1000 nM T62974 CAF02P 44388109 IC50 = 99 nM T62974 C23XBM 44388110 IC50 > 1000 nM T62974 CPX74G 44388112 IC50 > 1000 nM T62974 CG9SA3 44388114 IC50 = 772 nM T62974 C2C4MH 44388116 IC50 > 1000 nM T62974 CW1EL5 44388118 IC50 > 1000 nM T62974 CN0K3V 44388119 IC50 > 1000 nM T62974 CE8DH4 44388120 IC50 > 1000 nM T62974 C1A0OY 44388121 IC50 = 562 nM T62974 CS53NP 44388122 IC50 > 1000 nM T62974 CX67WG 44388123 IC50 = 435 nM T62974 CB50EK 44388124 IC50 = 660 nM T62974 C9SN1X 44388132 IC50 > 1000 nM T62974 C6W4YT 44388133 IC50 > 1000 nM T62974 CMTN20 44388134 IC50 > 1000 nM T62974 CAK42W 44388135 IC50 > 1000 nM T62974 CTW48B 44388136 IC50 > 1000 nM T62974 C4P1AS 44388137 IC50 > 1000 nM T62974 CEAZ82 44388138 IC50 > 1000 nM T62974 C1KMT8 44397389 Ki = 74 nM T62974 CN6Z8C 44397648 Ki = 130 nM T62974 CRW0M6 44397706 Ki = 140 nM T62974 CM1R8X 44400000 IC50 > 10000 nM T62974 CP89CS 44400135 IC50 = 300 nM T62974 C1BY2P 44444935 IC50 = 412 nM T62974 CH17TI 44560858 IC50 = 349 nM T62974 C2AZY7 44560859 IC50 = 287 nM T62974 C2I8NB 44560860 IC50 > 1000 nM T62974 C4XRT0 44560861 IC50 > 1000 nM T62974 C21TZI 44560862 IC50 > 1000 nM T62974 C2YM5N 44560863 IC50 > 1000 nM T62974 CS39FB 44560864 IC50 = 296 nM T62974 CU3FD2 44560865 IC50 = 715 nM T62974 C8IKU1 44560866 IC50 > 1000 nM T62974 CTQ83Z 44560867 IC50 = 116 nM T62974 CQC29N 44560868 IC50 = 908 nM T62974 C47MDA 44560869 IC50 = 479 nM T62974 CHAJ41 44560870 IC50 = 136 nM T62974 CT0A9U 44560871 IC50 = 831 nM T62974 CM0T9R 44560872 IC50 > 1000 nM T62974 CO2J6R 44560873 IC50 = 728 nM T62974 CKQD64 44560874 IC50 > 1000 nM T62974 CEK26Y 44560875 IC50 > 1000 nM T62974 CBL1P7 44560876 IC50 > 1000 nM T62974 CY47DM 44560877 IC50 = 800 nM T62974 C5OZD1 44560878 IC50 = 551 nM T62974 CFT47C 44560898 IC50 > 1000 nM T62974 CAO7R0 44560899 IC50 = 883 nM T62974 C80ZCF 44560900 IC50 = 813 nM T62974 CATH94 44560901 IC50 = 287 nM T62974 C2AXG6 44560902 IC50 = 905 nM T62974 COQ9W7 44560903 IC50 > 1000 nM T62974 CLZ23V 44560904 IC50 > 1000 nM T62974 C0OKG2 44560905 IC50 > 1000 nM T62974 CPIW17 44560906 IC50 > 1000 nM T62974 CFR3Y5 44560907 IC50 > 1000 nM T62974 CS85LR 44560908 IC50 = 455 nM T62974 C6K1FI 44577218 IC50 = 214 nM T62974 CAJ15T 44577219 IC50 = 115 nM T62974 CQD56E 44577220 IC50 = 296 nM T62974 CV18IC 44577221 IC50 = 174 nM T62974 C4NG5O 44820544 Ki = 690 nM T62974 CF5I4L 44820545 Ki = 160 nM T62974 CKRO61 44820563 Ki = 26 nM T62974 CTSR92 44820569 Ki = 19 nM T62974 CLJD09 45102042 IC50 > 10000 nM T62974 C63YJS 45139239 IC50 > 1000 nM T62974 C63XPN 45267999 IC50 > 1000 nM T62974 CF09UA 45268875 IC50 = 45 nM T62974 C2PNH4 45272264 IC50 > 1000 nM T62974 CFL9K7 45273129 IC50 = 296 nM T62974 C9Z4MR 45273130 IC50 > 1000 nM T62974 C4RGN0 45273131 IC50 = 71 nM T62974 CH18QA 46882131 Ki > 10000 nM T62974 CBZ3T9 46882132 Ki > 10000 nM T62974 C6KBJ2 46882133 Ki > 10000 nM T62974 CNL16U 46882180 Ki > 10000 nM T62974 CCX75M 46882181 Ki > 10000 nM T62974 C2BOJ6 46882182 Ki > 10000 nM T62974 C9ASC1 46882224 Ki > 10000 nM T62974 CB38SE 46882225 Ki > 10000 nM T62974 CP2N1U 46882226 Ki > 10000 nM T62974 CJ3Q6B 46882227 Ki > 10000 nM T62974 CRYQ47 46882445 Ki > 10000 nM T62974 CRZ1B0 46882446 Ki > 10000 nM T62974 CNEZ46 46882447 Ki > 10000 nM T62974 C8D1OR 46882448 Ki > 10000 nM T62974 CZ0G2R 46882449 Ki > 10000 nM T62974 CR37UF 46882513 Ki > 10000 nM T62974 CF3L8U 46882514 Ki > 10000 nM T62974 C91WKZ 46882515 Ki > 10000 nM T62974 CX21JH 46882516 Ki > 10000 nM T62974 CBJ92C 46882517 Ki > 10000 nM T62974 C8N3KX 46882577 Ki > 10000 nM T62974 CAH31I 46882578 Ki > 10000 nM T62974 CD2NL0 46882579 Ki > 10000 nM T62974 C9B0DF 46882620 Ki > 10000 nM T62974 CJ8I4L 46882621 Ki > 10000 nM T62974 C2YMA7 46882622 Ki > 10000 nM T62974 CD0VH7 46882664 Ki > 10000 nM T62974 C50YRJ 46882665 Ki > 10000 nM T62974 CXFV62 46882666 Ki > 10000 nM T62974 CR07WV 46882667 Ki > 10000 nM T62974 CF1HC7 46882668 Ki > 10000 nM T62974 CVIU56 46882708 Ki > 10000 nM T62974 C8S4LN 46882709 Ki > 10000 nM T62974 CJ7GM9 46882746 Ki > 10000 nM T62974 C6OM5H 46882789 Ki > 10000 nM T62974 C5MV8K 46882790 Ki > 10000 nM T62974 C6RD3V 46882791 Ki > 10000 nM T62974 C1WUF9 46882831 Ki > 10000 nM T62974 C5LM3W 46882832 Ki > 10000 nM T62974 CU1D6I 46902023 IC50 = 4000 nM T62974 CG78MV 46919128 IC50 = 180 nM T62974 C84ZTC 49865341 IC50 = 412 nM T62974 C3VZ4U 49865342 IC50 > 1000 nM T62974 CGYR09 49865343 IC50 = 346 nM T62974 C35WID 49865344 IC50 = 249 nM T62974 C0RK7G 49865345 IC50 = 1000 nM T62974 C4YLM7 49865346 IC50 > 1000 nM T62974 CZ4RI1 49865347 IC50 > 1000 nM T62974 CQJP15 51003591 Ki = 4400 nM T62974 C9SNL1 52941607 IC50 > 10000 nM T62974 CO04IG 52943613 IC50 = 660 nM T62974 CVO9X2 52947330 IC50 = 720 nM T62974 C40ZRY 52948630 IC50 > 10000 nM T62974 CED3O6 53473658 IC50 = 25 nM T62974 CE7J0U 53473659 IC50 = 16 nM T62974 CY0G2K 53473744 IC50 = 12 nM T62974 CBQG96 53473824 IC50 = 12 nM T62974 CW53YV 53473917 IC50 > 1000 nM T62974 C87SME 53474004 IC50 > 1000 nM T62974 C7EO1Z 53474005 IC50 > 1000 nM T62974 CY3M2A 53474090 IC50 = 590 nM T62974 CM58UZ 56651206 IC50 = 1200 nM T62974 COBQ28 56651207 Ki = 580 nM T62974 CGKP76 56661222 Ki = 60 nM T62974 C3RWH0 56661224 Ki = 124 nM T62974 C9JHI4 56664813 Ki = 2 nM T62974 C3M6AT 56678313 Ki < 1 nM T62974 C05RSG 56681656 Ki = 700 nM T62974 C59PKT 56681657 Ki = 3.7 nM T62974 C4MT8I 56681776 IC50 = 100 nM T62974 C8ZW3O 56927659 IC50 = 384 nM T62974 CHK8T1 56945132 EC50 = 6.8 nM T62974 C73XBL 57384077 IC50 > 1000 nM T62974 C3KC9Z 57398462 IC50 = 2.5 nM T62974 CTVI05 70683416 IC50 = 214 nM T62974 CV42WQ 70689221 IC50 = 6.9 nM T62974 C3P0AN 70689413 IC50 > 1000 nM T62974 CP58HL 70689414 IC50 > 1000 nM T62974 CB14OW 70689415 IC50 > 1000 nM T62974 CNZC97 70689723 IC50 = 63 nM T62974 C2WQM9 70691295 IC50 > 1000 nM T62974 C5E8MY 70693613 IC50 = 373 nM T62974 C3TZ9U 70695246 IC50 = 932 nM T62974 C34XGS 70695722 IC50 > 1000 nM T62974 CIPF50 70695723 IC50 > 1000 nM T62974 CF08XL 71458043 Ki = 7200 nM T62974 CU82HG 71460000 IC50 > 1000 nM T62974 CPC69G 71461645 Ki > 10000 nM T62974 CLAV92 71461684 IC50 > 1000 nM T62974 C1NZU3 71461685 IC50 > 10000 nM T62974 CI0GU8 71660496 IC50 > 48500 nM T62974 CFKH42 71717904 IC50 = 1000 nM T62974 CGDO59 72947672 Ki = 1.77 nM T62974 CW83DK 73213196 Ki > 10000 nM T62974 CIO28F 73345407 Ki = 1000 nM T62974 CMN6X8 73345525 IC50 = 5.4 nM T62974 C70XZC 73345528 IC50 = 1.2 nM T62974 CXGJ67 73345700 IC50 = 729 nM T62974 CV23JS 73345701 IC50 = 1033 nM T62974 C81UME 73345740 Ki > 1000 nM T62974 CX5VM1 73346900 IC50 > 10000 nM T62974 CA3MU5 73346903 IC50 = 3.5 nM T62974 C62NFY 73346927 Ki = 575 nM T62974 CK64MX 73346930 Ki = 1000 nM T62974 C15CAN 73346972 Ki > 1000 nM T62974 CD09FU 73347225 Ki = 2880 nM T62974 CI4L6W 73347226 Ki = 682 nM T62974 CGM61R 73348311 Ki > 10000 nM T62974 CN1FD2 73348312 Ki > 10000 nM T62974 C01GIQ 73348427 Ki = 1000 nM T62974 C7Y9ZT 73348428 Ki = 1000 nM T62974 CFLT50 73348719 IC50 = 61.8 nM T62974 C75NBQ 73348741 Ki = 145 nM T62974 C5MNX3 73348742 Ki > 1000 nM T62974 CL94MY 73350006 Ki = 1000 nM T62974 C0N6XK 73350010 Ki = 1000 nM T62974 CTV30F 73350011 Ki = 1000 nM T62974 CF2AK4 73350012 Ki = 1000 nM T62974 CK9CS4 73351516 Ki = 1000 nM T62974 CNY13O 73351517 Ki = 1000 nM T62974 CUN6L1 73351622 IC50 = 41 nM T62974 CC98JE 73351624 IC50 = 1.4 nM T62974 CWUH52 73351718 Ki = 1246 nM T62974 CS9I4W 73351829 Ki > 1000 nM T62974 CF70XH 73351873 IC50 > 1000 nM T62974 C0KJ6N 73352984 Ki = 80 nM T62974 CFB54J 73352985 Ki = 1000 nM T62974 CKFV85 73353009 Ki = 987 nM T62974 CC45AV 73353272 IC50 = 337 nM T62974 C41OCY 73353278 IC50 = 35.9 nM T62974 CW54CU 73353340 IC50 > 1000 nM T62974 CL7DT2 73354494 Ki = 1000 nM T62974 CA48EL 73354535 Ki > 1000 nM T62974 CFK7Z3 73354633 IC50 = 3.5 nM T62974 C1UYL2 73354783 IC50 = 346 nM T62974 CG1CX0 73354798 IC50 > 100 nM T62974 CIVZ67 73354818 Ki = 895 nM T62974 CGCE64 73354819 Ki = 888 nM T62974 C1Y0CI 73356066 Ki = 1000 nM T62974 C52JAS 73356068 Ki = 1000 nM T62974 CN5LG8 73356069 Ki = 1000 nM T62974 C9GKV2 73356181 IC50 = 2.3 nM T62974 C7XFB6 73356331 IC50 = 4.11 nM T62974 CI02SE 73356366 Ki = 1640 nM T62974 CW8L6C 76310862 IC50 > 1000 nM T62974 CHV6K7 76314485 IC50 = 5.4 nM T62974 C0PR3Y 76314486 IC50 > 1000 nM T62974 C94BWD 76314487 IC50 = 2.8 nM T62974 C25XKO 76314488 IC50 = 0.9 nM T62974 CS54IV 76321777 IC50 = 4 nM T62974 C94OAT 76321778 IC50 = 1.2 nM T62974 CU1IR8 76325402 IC50 = 3.7 nM T62974 CL09JQ 86279005 IC50 > 10000 nM T62974 C3JOS4 86292350 EC50 = 1.2 nM T62974 CVLE34 86293506 EC50 = 0.4 nM T62974 C15VTO 86294248 EC50 = 0.4 nM T62974 C2BAV8 90644981 Ki = 1089 nM T62974 CI58FM 90663867 IC50 = 837 nM T62974 CK62FO 90663868 IC50 > 1000 nM T62974 C7AFD4 90663869 IC50 = 482 nM T62974 C94XTF 90663872 IC50 > 1000 nM T62974 CA7W0U 90663873 IC50 = 797 nM T62974 C4EG8T 90663874 IC50 = 823 nM T62974 CW21UO 90663875 IC50 = 356 nM T62974 C7Q4PD 90665458 Ki = 20000 nM T62974 CR43ZL 90665459 Ki = 4900 nM T62974 CLK7C3 90665460 Ki = 7200 nM T62974 CZ0UC6 90665461 Ki = 10000 nM T62974 C0IBJ6 90665462 Ki = 21000 nM T62974 CPX0C9 90665463 Ki = 12000 nM T62974 C3UVC8 91936728 IC50 > 1000 nM T62974 CT3UP7 91936729 IC50 = 523 nM T62974 CD2E4L 101941290 IC50 = 1000 nM T62974 C9KB3W 117711399 EC50 = 4.3 nM T62974 CTH52C 118718416 Ki < 0.3162 nM T62974 CKQ4P6 118718462 IC50 = 1172 nM T62974 C1Z7UJ 118718463 Ki < 1000 nM T62974 CPYA80 118718465 IC50 = 1000 nM T62974 CR61UD 118718466 IC50 = 1000 nM T62974 CW64XN 118718500 IC50 = 1000 nM T62974 CB4D5T 118718501 IC50 = 632 nM T62974 CW5HG2 118718502 IC50 = 1000 nM T62974 CC36KP 118718503 IC50 = 1000 nM T62974 C7FIQ1 118718504 IC50 = 1000 nM T62974 CNBY57 118718505 IC50 = 3007 nM T62974 CPY4Q5 118718506 IC50 = 757 nM T62974 CO13JR 118718507 IC50 = 1000 nM T62974 CLFJ60 118718508 IC50 = 1000 nM T62974 C13YUH 118718509 IC50 = 1000 nM T62974 CP2O7U 118718510 IC50 = 1000 nM T62974 CLDZ63 118718511 IC50 = 1000 nM T62974 CYQ7X2 118718854 IC50 = 31 nM T62974 CA6C4T 118719101 IC50 = 2.3 nM T62974 CDZ3H4 118719196 IC50 = 2.4 nM T62974 CQRO32 118719197 IC50 = 5.6 nM T62974 CGXH91 118719198 IC50 = 3.2 nM T62974 C1QJX7 118719199 IC50 = 2.6 nM T62974 C0GLC8 118719200 IC50 = 153 nM T62974 C40NGQ 118719201 IC50 = 133 nM T62974 CK2W9T 118719202 IC50 = 5.2 nM T62974 CW4AT0 118719275 IC50 = 5.4 nM T62974 C5VWI1 118719303 IC50 = 1000 nM T62974 CS12JW 122179457 IC50 = 3200 nM T62974 CNGQ19 122179477 IC50 > 100000 nM T62974 C9B4DJ 122181226 Ki = 5400 nM T62974 CH1P7L 122181227 Ki = 1900 nM T62974 C6M3TH 127032865 Ki = 7090 nM T62974 CB5Q9D 127032866 Ki = 1170 nM T62974 CUO25F 127032867 Ki = 2020 nM T62974 CF1T6D 127033186 Ki = 2050 nM T62974 CE79SV 138377584 IC50 > 10000 nM T62974 C9CEY3 145949026 Ki = 1.34 nM T62974 CP0WF8 155510657 IC50 > 100000 nM T62974 C0I2UD 155513010 Ki > 10000 nM T62974 CV2BZ9 155516168 Ki > 10000 nM T62974 C2OG9Y 155517592 Ki > 10000 nM T62974 C59SVW 155518749 Ki > 10000 nM T62974 C1BS2T 155519582 Ki = 1426 nM T62974 CHJO90 155524485 Ki > 10000 nM T62974 CW0XC1 155526536 IC50 = 103 nM T62974 CD73TA 155526663 IC50 > 100000 nM T62974 CGXE80 155528330 Ki = 6800 nM T62974 C9QIB6 155529288 Ki = 7200 nM T62974 CI9HE4 155532172 Ki < 10000 nM T62974 CYT0Z4 155532886 Ki > 10000 nM T62974 CKZ82R 155538553 Ki > 10000 nM T62974 C9XB6L 155539840 Ki > 100000 nM T62974 CVOW56 155541238 Ki > 10000 nM T62974 CBD2Q8 155541853 Ki = 2.41 nM T62974 C5RI8K 155541897 Ki = 21000 nM T62974 CIA72K 155543246 IC50 > 100000 nM T62974 CVR3U2 155546680 Ki = 1900 nM T62974 CY68DL 155546826 Ki = 4471 nM T62974 CGZY28 155549889 Ki > 100000 nM T62974 CLJU08 155550820 Ki = 20000 nM T62974 CI6E8B 155552577 Ki > 10000 nM T62974 C89BNQ 155553012 Ki = 2100 nM T62974 CX02AJ 155555535 Ki = 4803 nM T62974 CR1AY2 155557409 Ki = 2380 nM T62974 CD58IO 155558366 Ki = 2032 nM T62974 C6T0IB 155560534 Ki > 10000 nM T62974 C5RL2K 155565048 Ki = 5400 nM T62974 CN7CQ1 155567326 Ki > 10000 nM T62974 CE76TG 42637005 IC50 = 468 nM T62974 C6ELN4 42637006 IC50 = 329 nM T62974 CS73LG 42637433 IC50 > 1000 nM T62974 C6C3YF 45270549 IC50 > 1000 nM T62974 C9Y3BS 45270550 IC50 > 1000 nM T62974 CQC51Z 45270552 IC50 > 1000 nM T62974 CXE30U 45271377 IC50 > 1000 nM T62974 D01BWV 9802572 Ki = 7100 nM T62974 D01NID 44388055 IC50 > 1000 nM T62974 D02CQW 11847438 IC50 > 1000 nM T62974 D02NJV 44388048 IC50 = 932 nM T62974 D02OJQ 44388115 IC50 = 0.5 nM T62974 D02WOX 44388129 IC50 > 1000 nM T62974 D03DRL 44388045 IC50 = 417 nM T62974 D03SXC 44388041 IC50 > 1000 nM T62974 D03VHX 44388111 IC50 > 1000 nM T62974 D04EWA 44388034 IC50 > 1000 nM T62974 D04FPW 44388024 IC50 > 1000 nM T62974 D04ORV 44388047 IC50 = 0.6 nM T62974 D04QBM 5311374 Ki = 0.7 nM T62974 D05COQ 11847588 IC50 > 1000 nM T62974 D05XZA 44388071 IC50 > 1000 nM T62974 D06JWT 44388073 IC50 > 1000 nM T62974 D07DUF 44388130 IC50 > 1000 nM T62974 D07OSF 44388044 IC50 > 1000 nM T62974 D07WRP 15965425 Ki = 81 nM T62974 D09DAC 44388046 IC50 = 1.2 nM T62974 D09LHN 44311674 IC50 = 384 nM T62974 D0A0DO 44388056 IC50 > 1000 nM T62974 D0A1XX 44388113 IC50 = 418 nM T62974 D0BE3D 44388092 IC50 > 1000 nM T62974 D0C5RH 44388125 IC50 = 1.4 nM T62974 D0CC1P 44388042 IC50 > 1000 nM T62974 D0H0DC 44388051 IC50 = 786 nM T62974 D0H4WH 44388128 IC50 = 1.7 nM T62974 D0I9ME 44388074 IC50 > 1000 nM T62974 D0J5OY 44388022 IC50 = 3.3 nM T62974 D0M5LA 44388050 IC50 > 1000 nM T62974 D0N2MA 44388103 IC50 > 1000 nM T62974 D0N4LH 44388065 IC50 > 1000 nM T62974 D0O4GU 44403230 Ki > 1000 nM T62974 D0P6ZZ 10581102 IC50 > 1000 nM T62974 D0R0OX 44388102 IC50 = 245 nM T62974 D0R4IS 44388131 IC50 > 1000 nM T62974 D0S7YR 44388059 IC50 > 1000 nM T62974 D0T5RO 16129706 Ki = 0.59 nM T62974 D0W0AF 44388072 IC50 = 226 nM T62974 D0WG0O 44388049 IC50 = 229 nM T62974 D0Z0OF 44388094 IC50 > 1000 nM T62974 D0Z1XY 44388064 IC50 > 1000 nM T62974 D0Z3LZ 44388023 IC50 = 1 nM T90818 D0V2GT 5311023 Ki = 84 nM T90818 C65NED 9573348 EC50 = 1000 nM T90818 CL57KJ 9707420 EC50 = 501.19 nM T90818 C2H5NY 9854861 Ki = 1.2 nM T90818 C3H7AS 9955930 Ki = 92 nM T90818 CH1Q6E 10008757 Ki > 3000 nM T90818 C6S2CB 25138123 IC50 = 2400 nM T90818 CMTA17 44542176 EC50 = 1258.93 nM T90818 COW17D 44542178 EC50 = 501.19 nM T90818 C7Q9PI 44542320 EC50 = 794.33 nM T90818 CY14UJ 44542322 EC50 = 398.11 nM T90818 C3ILH8 44542324 EC50 = 100 nM T90818 C8D4AT 44542326 EC50 = 199.53 nM T90818 CIRQ85 44542328 EC50 = 100 nM T90818 CB58DA 44542330 EC50 = 158.49 nM T90818 CS12HR 44542332 EC50 = 125.89 nM T90818 CY4L2G 53318788 IC50 = 0.79 nM T90818 CO72VY 60168134 EC50 = 1256 nM T90818 CW7KQ1 60168135 EC50 = 298 nM T90818 CH58GJ 71450762 Ki = 227 nM T90818 C6AV0I 71451611 EC50 = 1.7 nM T90818 C7K8BZ 71452593 Ki = 425 nM T90818 COM10Q 71454352 Ki = 142 nM T90818 CM31QR 71454353 Ki = 424 nM T90818 CL9E0V 71454357 Ki = 672 nM T90818 C8MP1A 71454358 Ki = 94 nM T90818 CHFO89 71454359 Ki = 417 nM T90818 C7ROU1 71456101 Ki = 117 nM T90818 CO07CE 71456102 Ki = 1620 nM T90818 C24UFT 71456103 Ki = 47 nM T90818 CL82IR 71456104 Ki = 9 nM T90818 C3SOE7 71457908 Ki = 136 nM T90818 CZ7C4L 71457909 Ki = 4 nM T90818 CJWQ68 71457910 Ki = 155 nM T90818 C3W7BS 71461185 Ki = 2015 nM T90818 C0VA5C 71463271 Ki = 141 nM T90818 C49KZP 71463273 Ki = 208 nM T90818 C1EGB8 71463275 Ki = 3196 nM T90818 CW9XZ8 71463276 Ki = 206 nM T90818 CA7S8C 71463277 Ki = 590 nM T90818 C75FXY 71463278 Ki = 4 nM T90818 CA7G4S 71463279 Ki = 22 nM T90818 CU9O4B 101493753 Ki = 0.53 nM T90818 CW3LH2 101882818 Ki = 1052 nM T90818 CW5H9D 101882819 Ki = 1426 nM T90818 CGQV37 101882820 Ki = 30 nM T90818 CA51CQ 118724536 Ki = 75 nM T90818 CR4MG1 118724537 Ki = 0.47 nM T90818 CBA2Z0 118724538 Ki > 5000 nM T90818 CL3T4A 118724539 Ki = 1694 nM T90818 CTHD48 118724540 Ki = 304 nM T90818 CZL32K 118724541 Ki > 5000 nM T90818 C5HNX2 118724542 Ki = 6616 nM T90818 C4AT2F 118724543 Ki = 2773 nM T90818 CE1NT2 118724544 Ki = 7579 nM T90818 CM3RN4 118724970 Ki = 2907 nM T90818 C5XD1N 118724971 Ki = 3220 nM T90818 C6M1AZ 118724972 Ki = 2682 nM T90818 CSF21L 118724973 Ki = 2223 nM T90818 CH4LB0 118724977 Ki = 405 nM T90818 C6GK5N 118724978 Ki = 1893 nM T90818 C9SN0M 118724979 Ki = 309 nM T90818 CH9GT5 118724980 Ki = 987 nM T90818 CHK0S7 118724981 Ki = 884 nM T90818 C1BVC2 118724982 Ki = 409 nM T90818 C76XZK 118724983 Ki = 3505 nM T90818 CG7SQ8 118724984 Ki = 84 nM T90818 CB3D6X 118724985 Ki = 465 nM T90818 CG04KW 118724986 Ki = 2757 nM T90818 CO69YD 118724987 Ki = 298 nM T90818 C72AKO 118724988 Ki = 330 nM T90818 C4CRS0 118724989 Ki = 129 nM T90818 CJIB02 118724990 Ki = 504 nM T90818 CD41AL 118724991 Ki = 454 nM T90818 C2DCZ3 118724992 Ki = 1513 nM T90818 C49HSM 118724993 Ki = 82 nM T90818 CE9ZS5 118724994 Ki = 205 nM T90818 CP2WY4 118724995 Ki = 910 nM T90818 C1TD6L 127030365 Ki = 41 nM T90818 C7YA8H 127030940 Ki = 27 nM T90818 C5PA2G 127041908 Ki = 1200 nM T90818 C62JIE 127042244 Ki > 3000 nM T90818 CNX9D2 136948074 Ki = 1620 nM T90818 CY35MT 136998789 Ki = 993 nM T90818 CBAP98 136998790 Ki = 2398 nM T90818 C8F9WQ 155515973 EC50 = 250 nM T90818 CF42WX 155520785 EC50 = 158.49 nM T90818 D01VSI 25240297 IC50 = 76 nM T90818 D08UWO 53320361 Ki = 43 nM T90818 D0JE3Z 16735569 IC50 = 1800 nM T17339 D0I2AN 86298439 IC50 = 2900 nM T17339 CKH70I 72705451 Ki = 150000 nM T17339 C0IJ2X 118737463 IC50 = 5700 nM T17339 CG0Z1I 137649766 Ki = 6900 nM T93283 C7GTI4 81312 IC50 > 500000 nM T93283 CFB8H3 96536 IC50 = 30000 nM T93283 CE0U1R 195023 IC50 = 142000 nM T93283 CEP2N4 242551 IC50 > 500000 nM T93283 CJR57B 4469578 IC50 = 4 nM T93283 CW9DQ2 4476325 IC50 = 6000 nM T93283 C0KAB3 9867336 IC50 = 1400 nM T93283 CIYE74 9881235 IC50 = 88000 nM T93283 CUJI84 9973036 IC50 = 9000 nM T93283 C3PB6D 10039105 IC50 = 14000 nM T93283 C2L3NF 10383023 IC50 = 21000 nM T93283 CIWE62 15341136 IC50 = 9300 nM T93283 CB9R2F 22988798 IC50 = 38000 nM T93283 C9LR1V 44296499 IC50 = 21000 nM T93283 C20DWM 44296500 IC50 = 11400 nM T93283 CFL2N8 44296527 IC50 = 6300 nM T93283 CIU45S 44296534 IC50 = 11000 nM T93283 C7N2KA 44296536 IC50 = 89000 nM T93283 C4R6WG 44309346 IC50 = 14000 nM T93283 C76YXK 44309396 IC50 = 8.6 nM T93283 C5XCT6 44336394 IC50 = 152000 nM T93283 CBM6E8 44336450 IC50 = 70000 nM T93283 C3P1KZ 44336452 IC50 = 67000 nM T93283 CBS80R 44336458 IC50 = 31000 nM T93283 C7RQ4C 44336463 IC50 = 37000 nM T93283 C58SWT 44336464 IC50 = 143000 nM T93283 CG0AV1 44336465 IC50 = 41000 nM T93283 CR32EI 44336472 IC50 = 100000 nM T93283 CAK08U 44336531 IC50 = 15000 nM T93283 CL2V8T 44336543 IC50 = 17000 nM T93283 C32ZLU 44336551 IC50 = 16000 nM T93283 CT31VP 44336553 IC50 = 36000 nM T93283 C98QZE 44336560 IC50 = 94000 nM T93283 C0VI7H 44336562 IC50 = 67000 nM T93283 CP1Z0W 49797574 IC50 = 1210 nM T93283 CK0X5J 49797575 IC50 = 25.7 nM T93283 CAJ35Z 49797576 IC50 = 1070 nM T93283 CZ7PV6 49797577 IC50 = 18 nM T93283 CI27BD 49797578 IC50 = 5 nM T93283 C3ETV8 49797579 IC50 = 198 nM T93283 D0N4XG 417214 IC50 = 34000 nM T75570 D0E6XR 3062316 IC50 = 0.5 nM T75570 D0OB0F 5328940 IC50 = 0.4 nM T75570 D03LWG 53235510 IC50 = 1100 nM T75570 D05PZB 135398495 IC50 = 1 nM T75570 D07EHV 44814409 IC50 > 10000 nM T75570 D0E0NM 25066467 IC50 = 1.5 nM T75570 D0E3TC 44259 IC50 = 2.35 nM T75570 D0G2QH 10297043 IC50 = 13.1 nM T75570 D0GP9Q 11973736 IC50 >= 2500 nM T75570 D0M0XB 10302451 IC50 = 0.7 nM T75570 D03BNU 59604787 IC50 > 10000 nM T75570 D0T3ME 156422 IC50 = 8900 nM T75570 CB1VW3 1400 IC50 = 36 nM T75570 CY13FW 644243 IC50 = 510 nM T75570 CR0DJ8 4078145 IC50 = 7700 nM T75570 CI80BK 9803350 IC50 = 20 nM T75570 CM2VB6 10100735 IC50 = 156000 nM T75570 C6DC8Q 10275163 IC50 = 10 nM T75570 C8RD3V 10301884 IC50 = 3 nM T75570 C5CBF9 10320381 IC50 = 10 nM T75570 CLAX64 10413508 IC50 = 30 nM T75570 CDQO71 10461517 IC50 = 110000 nM T75570 CJ5M1D 10482445 IC50 = 10 nM T75570 CACS26 11561968 Ki > 2000 nM T75570 CJV20L 11569758 IC50 = 4.1 nM T75570 CAJQ78 11584678 IC50 = 1.3 nM T75570 CU0E8O 11690457 Ki > 2000 nM T75570 CHL5W3 11712625 IC50 = 0.3 nM T75570 CZY05V 11719421 IC50 = 1.2 nM T75570 C73MLJ 16108977 IC50 = 8.7 nM T75570 C6TQ2O 16664354 Ki = 5.97 nM T75570 CY1E2N 16723801 IC50 = 30000 nM T75570 CG12OL 23518511 IC50 = 20 nM T75570 C6O8QY 23661616 IC50 = 4.8 nM T75570 CA3I4T 24753787 IC50 > 50000 nM T75570 CP1WR0 24795070 IC50 = 240 nM T75570 C2MUA7 24823072 IC50 = 110 nM T75570 CX94DT 24823073 IC50 = 22 nM T75570 CCFQ29 44187005 IC50 = 246 nM T75570 CH3J2E 44299176 IC50 = 40 nM T75570 C27GVO 44299203 IC50 = 160 nM T75570 CY6WC0 44299236 IC50 = 10 nM T75570 C3RG0C 44299304 IC50 = 20 nM T75570 CJM26I 44299321 IC50 = 10 nM T75570 C9UGL3 44299325 IC50 = 10 nM T75570 CJEZ96 44299338 IC50 = 40 nM T75570 C8XGN5 44299339 IC50 = 30 nM T75570 CNH34G 44299354 IC50 = 10 nM T75570 C82MSD 44299360 IC50 = 30 nM T75570 CJ3PF9 44313929 IC50 > 500000 nM T75570 CUV7K3 44313930 IC50 > 500000 nM T75570 CHK9N3 44313931 IC50 = 94500 nM T75570 CEKR19 44313990 IC50 > 500000 nM T75570 CD5PI9 44313997 IC50 = 2600 nM T75570 C0GH7J 44314372 IC50 > 500000 nM T75570 C5E4GK 44314373 IC50 > 500000 nM T75570 C3YD1G 44314380 IC50 = 303000 nM T75570 CPC68H 44314402 IC50 > 500000 nM T75570 C1L6MG 44444041 IC50 = 5.2 nM T75570 C3VRO9 44557921 IC50 > 10000 nM T75570 CYT37A 46232443 IC50 > 50000 nM T75570 C48ZVW 46232555 IC50 = 26000 nM T75570 CS9B1U 46232556 IC50 > 50000 nM T75570 CL0O4U 46911726 Ki = 24 nM T75570 CCN08S 46934144 IC50 = 38100 nM T75570 CG5IK8 52936268 IC50 > 100000 nM T75570 CEQN27 52936621 Ki > 1000 nM T75570 C2CT5J 53236670 IC50 = 7950 nM T75570 C3M6LV 53236671 IC50 > 100000 nM T75570 CZ5L6F 53239373 IC50 > 100000 nM T75570 C2WFI8 53239374 IC50 = 41800 nM T75570 C0ZHF8 53239375 IC50 = 85540 nM T75570 CD1EQ3 53239587 IC50 = 26940 nM T75570 C8NA4L 53384644 IC50 > 30000 nM T75570 CPHX64 57325478 IC50 > 50000 nM T75570 CQ9BW4 57325479 IC50 > 50000 nM T75570 C1JLW8 57332840 IC50 = 5560 nM T75570 CD01JZ 57332841 IC50 = 5110 nM T75570 CCFK37 57332844 IC50 = 5340 nM T75570 CK1SR7 57332969 IC50 = 2410 nM T75570 C5TRE2 57332970 IC50 = 2010 nM T75570 C46TJK 57332974 IC50 = 8820 nM T75570 C09ZJY 57333095 IC50 = 11100 nM T75570 CVK0G4 58056356 IC50 > 50000 nM T75570 C1MR8Q 60097495 IC50 > 1000 nM T75570 CE49GC 67098566 Ki = 79 nM T75570 CV63UL 67240318 IC50 > 10000 nM T75570 CAIO65 68796885 IC50 = 44 nM T75570 COU73Y 71226944 IC50 = 37 nM T75570 C40JOZ 71235465 IC50 = 73 nM T75570 C5ZKU7 71546969 IC50 = 284 nM T75570 C7ARI9 71547113 IC50 = 496 nM T75570 CDJY72 71568837 IC50 = 1800 nM T75570 C8CAG7 71578921 IC50 > 10000 nM T75570 C7E6YV 71720026 IC50 = 160.4 nM T75570 CGDB30 74538658 IC50 = 30 nM T75570 CPG3A5 86302574 IC50 > 30000 nM T75570 CQCX41 118737057 IC50 = 0.8 nM T75570 CKBP72 121231408 IC50 < 0.5 nM T75570 C81IFQ 122163152 IC50 > 100000 nM T75570 CCXA46 122190499 Ki = 470 nM T75570 C3PQ4W 122190505 Ki = 610 nM T75570 CN1DK0 122190507 Ki = 800 nM T75570 CD67LU 122705248 IC50 = 12 nM T75570 CX63VW 122705258 IC50 = 696 nM T75570 C76IKM 122705261 IC50 = 566 nM T75570 C8ALO2 124088839 IC50 = 344 nM T75570 C0HN2Y 127030123 IC50 = 22060 nM T75570 C7S9GI 127030124 IC50 > 31600 nM T75570 CHGN68 127030424 IC50 = 6210 nM T75570 CRV62L 127030425 IC50 > 31600 nM T75570 CF7JT8 127030426 IC50 > 31600 nM T75570 C5YCU2 127030427 IC50 > 31600 nM T75570 C0GES2 127031075 IC50 > 100000 nM T75570 CFJ32Y 127031076 IC50 > 100000 nM T75570 CC8V4J 127031368 IC50 = 27210 nM T75570 C78GYH 127031383 IC50 = 20430 nM T75570 C5WA9Z 127031384 IC50 = 31510 nM T75570 CD7LN1 127031385 IC50 = 8100 nM T75570 CI0VX4 127031386 IC50 = 12630 nM T75570 CO89TC 127031387 IC50 = 1020 nM T75570 CAM4S5 127031675 IC50 = 7070 nM T75570 C4QD0M 127031676 IC50 = 23110 nM T75570 C0LTC3 127031677 IC50 > 100000 nM T75570 CO1G2K 127032542 IC50 > 100000 nM T75570 C12IOL 127033165 IC50 > 31600 nM T75570 C5RO0L 127033758 IC50 > 100000 nM T75570 CD04YX 127034308 IC50 > 31600 nM T75570 CG8DA9 127045861 IC50 > 100000 nM T75570 CC4ND8 127046862 IC50 > 100000 nM T75570 CO25WH 127052538 IC50 = 71 nM T75570 C8F0DQ 129909860 IC50 = 4 nM T75570 CLCO61 135398510 IC50 = 1.4 nM T75570 CAW0E4 136065882 IC50 = 42900 nM T75570 CXC69T 137321158 IC50 = 384 nM T75570 CZOD53 137633880 IC50 = 189 nM T75570 C7BJY5 137636807 IC50 = 60 nM T75570 CO89DX 137649100 IC50 = 32 nM T75570 CINE03 137652514 IC50 = 266 nM T75570 C28QUP 137652864 IC50 = 57.3 nM T75570 CRWA29 139030520 IC50 > 10000 nM T75570 C2MD1Q 155513187 IC50 > 10000 nM T75570 C3NA2I 155519537 IC50 = 86 nM T75570 D03OKV 9844320 IC50 > 4.7 nM T75570 D06HVH 54613583 IC50 > 10000 nM T75570 D08RZB 11153014 IC50 = 2 nM T75570 D0C0ZC 11676786 IC50 = 51.2 nM T75570 D0CE3R 5312137 IC50 = 20 nM T75570 D0H1OK 11562302 IC50 = 10 nM T75570 D0N4LR 53469448 IC50 = 3195 nM T75570 D0O8AR 16097523 IC50 = 3 nM T75570 D0Y0BK 11524144 IC50 = 29.8 nM T79400 CGN48U 9827867 IC50 = 41 nM T79400 CW1G9B 10672666 IC50 > 10000 nM T79400 CW7Q2U 10895700 IC50 > 2500 nM T79400 CIQH43 11445130 IC50 = 3.4 nM T79400 C37MRI 16718808 IC50 = 12 nM T79400 CVO5L6 24748791 IC50 = 15 nM T79400 CS9TK6 38335241 IC50 > 200000 nM T79400 C25ELB 44143088 IC50 = 14454.4 nM T79400 CL0M7R 44143089 IC50 = 9772.37 nM T79400 C9QDC0 44143091 IC50 = 177827.94 nM T79400 C30CFX 44436704 IC50 = 40 nM T79400 CM83VP 72163524 IC50 > 10000 nM T79400 CWP85J 87360663 IC50 > 10000 nM T79400 CDCG19 122192781 Ki = 9 nM T79400 CD5SN7 122192782 Ki = 19.9 nM T79400 CJ6DA9 127028140 IC50 = 250 nM T79400 CD9KI3 127028141 IC50 = 80 nM T79400 C5MAS1 155510638 Ki = 0.13 nM T79400 CV8YT6 155516274 Ki = 1.8 nM T79400 CU80TM 155522954 Ki = 1.3 nM T79400 CU52QS 155545897 Ki = 1.6 nM T79400 CH2S6R 155546346 Ki = 0.44 nM T79400 CNZ1K5 155559920 Ki = 0.1 nM T79400 CTWE96 155561147 Ki = 0.3 nM T79400 D0Y5IQ 44255320 IC50 = 10000 nM T46937 D01BYB 5957 IC50 = 251188.64 nM T46937 D07VLY 31703 Ki > 10000 nM T46937 D09QBG 9854012 IC50 = 2 nM T46937 D0R3JB 4212 Ki > 10000 nM T46937 D0R6RC 54675777 Ki > 10000 nM T46937 D0WF7L 9871419 Ki = 1.995 nM T46937 D09VBE 16066663 IC50 < 10 nM T46937 D0KE4Z 5310954 EC50 = 1.3 nM T46937 D0UF2N 21706 IC50 < 250000 nM T46937 D0W4JI 11273179 IC50 = 16 nM T46937 D08NXX 5487281 EC50 = 20 nM T46937 D0M4LF 23649325 IC50 = 9 nM T46937 D0U7OU 3220 Ki > 10000 nM T46937 COE28J 7220 IC50 = 7430000 nM T46937 C4RT3E 10208 Ki > 10000 nM T46937 C73JPZ 10639 Ki > 10000 nM T46937 C9K3IP 78253 Ki = 17100 nM T46937 CFG7T8 80533 IC50 = 2060000 nM T46937 CZ8J9T 118348 Ki = 2390 nM T46937 CQ8JF0 131257 IC50 = 13000 nM T46937 C85EPW 167523 Ki = 2450 nM T46937 CKE6V0 196979 Ki > 10000 nM T46937 C1T2BC 442744 Ki > 10000 nM T46937 C20KPF 601138 IC50 = 1800000 nM T46937 C1VW6X 601157 IC50 = 1840000 nM T46937 C2JP7W 1149185 Ki = 4400 nM T46937 CHBV51 2741913 IC50 = 1260 nM T46937 CD68IW 2746549 IC50 = 320 nM T46937 C3KM2I 2746550 IC50 = 300 nM T46937 CX5MV4 4603056 IC50 = 1960000 nM T46937 CH8TP5 4742792 IC50 = 850 nM T46937 C7Z4OR 4742793 IC50 = 4000 nM T46937 C92LSY 4742794 IC50 = 3000 nM T46937 C7BQ1N 5492386 EC50 = 10 nM T46937 CW46EH 9823796 Ki = 2.512 nM T46937 C93YKA 9846875 Ki = 5.012 nM T46937 CPHL60 9850430 Ki = 5.012 nM T46937 CL73SJ 9866696 Ki > 10000 nM T46937 CEG2J4 9953334 Ki = 19.95 nM T46937 C5ZXR3 9969173 Ki = 660 nM T46937 C39LZS 9999105 EC50 = 40 nM T46937 CXQ0V1 10016898 EC50 = 24300 nM T46937 C4ST7G 10017729 EC50 = 66 nM T46937 C2F7DR 10098947 IC50 = 10800 nM T46937 CW2Q3B 10109037 Ki = 2990 nM T46937 CQRU04 10110666 IC50 > 2000 nM T46937 CV1I0S 10202847 Ki = 29 nM T46937 CT73IB 10260031 IC50 = 0.7 nM T46937 C61MTA 10292521 IC50 = 1800 nM T46937 CJ9W1G 10294407 IC50 = 690 nM T46937 C5COM0 10438063 IC50 = 316227.77 nM T46937 CMBN72 10480103 IC50 > 3000 nM T46937 CBQ9P2 10557443 IC50 = 0.7943 nM T46937 CI6FS2 11273178 IC50 = 16 nM T46937 C1TE6Z 11497605 IC50 = 690 nM T46937 CE6OM7 11503160 IC50 = 190 nM T46937 C2GL4P 11503687 IC50 = 190 nM T46937 C29GJZ 11504727 Ki = 19740 nM T46937 CDQ2L4 11504760 IC50 = 110 nM T46937 CHB3C7 11510273 Ki > 70000 nM T46937 C0EX1O 11519648 IC50 = 38 nM T46937 C2VW4K 11526078 IC50 = 90 nM T46937 CA7G1M 11532836 IC50 = 260 nM T46937 CT74ZJ 11560464 Ki > 70000 nM T46937 C7EWL5 11561528 IC50 = 180 nM T46937 C1V0UF 11561748 IC50 = 310 nM T46937 C2UH6Z 11569565 IC50 = 42 nM T46937 CG7D2T 11570029 IC50 = 210 nM T46937 CN62XG 11585280 Ki = 50.7 nM T46937 C03UQZ 11595497 IC50 = 40000 nM T46937 CUD1J5 11611428 Ki > 70000 nM T46937 CFZ48K 11620159 IC50 = 740 nM T46937 C0TDC2 11627317 IC50 = 560 nM T46937 CXM91P 11627571 IC50 = 250 nM T46937 CN3Z2G 11641496 IC50 = 650 nM T46937 C19DSA 11649277 Ki = 3130 nM T46937 C2IH1A 11656053 IC50 = 380 nM T46937 CI8VZ7 11663657 IC50 = 380 nM T46937 C1V2CG 11670815 Ki = 19 nM T46937 CH48LB 11677907 IC50 = 37 nM T46937 C85RIU 11684524 IC50 = 1100 nM T46937 C5IB0G 11684912 IC50 = 170 nM T46937 CPF5V6 11691323 IC50 = 370 nM T46937 CYK4J8 11697626 IC50 = 200 nM T46937 CKPR59 11699088 IC50 = 210 nM T46937 C3VW7P 11699570 IC50 = 800 nM T46937 C4P7MS 11706300 IC50 = 95 nM T46937 CA19OH 11706351 IC50 = 90 nM T46937 C15YHK 11712235 IC50 = 130 nM T46937 C9JTV2 11786496 IC50 = 11 nM T46937 CR9YO8 11950159 Ki = 8 nM T46937 C1OEX4 11950328 Ki = 172 nM T46937 CQ02OS 11950687 Ki = 3 nM T46937 C8PI6W 11955421 Ki = 35 nM T46937 C3WGI2 11955422 Ki = 397 nM T46937 CM07WK 11993787 IC50 = 250 nM T46937 CPS34X 12000684 IC50 = 97 nM T46937 CBW05G 12000767 IC50 = 142 nM T46937 CO94DG 12000848 IC50 = 266 nM T46937 CGV57W 12001028 IC50 = 428 nM T46937 CF0GO7 12001030 IC50 = 533 nM T46937 CRYI50 12001296 IC50 = 31 nM T46937 CTN8D0 12001479 IC50 = 73 nM T46937 CVLK47 12001567 IC50 = 53 nM T46937 C5UAK6 12001662 IC50 = 35 nM T46937 CWI0T3 12001755 IC50 = 21 nM T46937 C2AQN5 12002005 IC50 = 178 nM T46937 CXVM04 12002012 IC50 = 218 nM T46937 CH4S8D 14280990 EC50 = 1040 nM T46937 CD1Q4U 14280991 EC50 > 106000 nM T46937 C03ZNU 14280992 EC50 = 1910 nM T46937 CZ9WG1 14280994 EC50 > 106000 nM T46937 CL4AF3 14280995 EC50 > 100000 nM T46937 C1MK5R 14280996 EC50 = 1900 nM T46937 CCTP04 14280998 EC50 = 950 nM T46937 CXH95F 14280999 EC50 = 9110 nM T46937 CZ6N0W 14281000 EC50 = 280 nM T46937 CR1G8Y 14281001 EC50 = 20 nM T46937 C18OUM 14281003 EC50 = 420 nM T46937 CJ6VF1 14281004 EC50 = 180 nM T46937 CH1BM2 14281005 EC50 = 16 nM T46937 C9MY5X 14281006 EC50 = 0.7 nM T46937 CUCR03 14281008 EC50 = 60 nM T46937 CUFJ35 14281010 EC50 = 70 nM T46937 CQ8TE3 14281011 EC50 = 110 nM T46937 CSEC89 14281012 EC50 = 10860 nM T46937 CU0J8E 14281015 EC50 = 90 nM T46937 CDP92K 14281016 EC50 = 5 nM T46937 C6FCS9 14281018 EC50 = 50 nM T46937 CK3E1F 14281020 EC50 = 1400 nM T46937 CUDO17 14281023 EC50 = 150 nM T46937 CZ19AJ 14281024 EC50 = 140 nM T46937 CY8PC6 14281025 EC50 = 1 nM T46937 CBT8K9 14281026 EC50 = 1 nM T46937 C3F7MZ 14281027 EC50 = 250 nM T46937 C2CF9I 14281031 EC50 = 4840 nM T46937 CQ2YL0 14281033 EC50 = 770 nM T46937 CM1NW7 14281034 EC50 = 330 nM T46937 CEUF73 14281035 EC50 = 870 nM T46937 C7QJ4Y 14281036 EC50 = 50300 nM T46937 CWSR46 14281041 EC50 = 100 nM T46937 CZ1ML0 15005564 EC50 = 38 nM T46937 CTL89M 15005565 EC50 = 12 nM T46937 CRO7P1 15005566 EC50 = 360 nM T46937 CCO0S1 15005567 EC50 = 90 nM T46937 C74EYG 15005568 EC50 > 87500 nM T46937 C7RC1U 15005569 EC50 = 1660 nM T46937 CAC98D 15005570 EC50 = 9410 nM T46937 CW0UP4 15005571 EC50 = 3170 nM T46937 C6I0LA 15005572 EC50 = 520 nM T46937 CM63ZU 15005573 EC50 = 26700 nM T46937 CE0DR4 15005574 EC50 = 20 nM T46937 CAQ7J2 15005576 EC50 = 20 nM T46937 CTE39J 15005577 EC50 = 910 nM T46937 C8TQ6C 15005578 EC50 = 380 nM T46937 C5Z8QA 15005579 EC50 = 3020 nM T46937 CS17FZ 15005580 EC50 = 1330 nM T46937 CN13YK 15005581 EC50 = 190 nM T46937 CQ9Y7J 15005583 EC50 = 950 nM T46937 CJ72ZA 15005584 EC50 = 4 nM T46937 CVA9B0 15005585 EC50 = 55 nM T46937 C4PM2K 15005586 EC50 = 260 nM T46937 C95NSJ 15005588 EC50 = 180 nM T46937 CI60HD 15005590 EC50 = 6320 nM T46937 CDHV05 15005591 EC50 = 1320 nM T46937 C7VR0Q 15005592 EC50 = 5400 nM T46937 C7QZO0 15005594 EC50 = 390 nM T46937 C2V3LD 15005598 EC50 = 440 nM T46937 CPS49B 15005599 EC50 = 2690 nM T46937 CP6DI1 15005600 EC50 = 2470 nM T46937 C0Z6GL 15005601 EC50 = 2950 nM T46937 CTU06K 15005602 EC50 = 440 nM T46937 C23MUZ 15005603 EC50 = 430 nM T46937 CRA5G0 15005604 EC50 = 63100 nM T46937 C96YTU 15005605 EC50 = 210 nM T46937 CH7I9M 15005606 EC50 = 1070 nM T46937 CX9L6N 15005608 EC50 = 420 nM T46937 CYH3R2 15650856 IC50 = 41000 nM T46937 CU5TM4 15650857 IC50 = 47000 nM T46937 CZE1S0 15650858 IC50 = 44000 nM T46937 C36DUQ 15650859 IC50 = 58000 nM T46937 C43IYK 15650860 IC50 = 65000 nM T46937 C9R7HT 15650861 IC50 = 19000 nM T46937 COA37U 15650862 IC50 = 4000 nM T46937 C1TKE3 15650863 IC50 = 9000 nM T46937 CYF68T 15650864 IC50 = 43000 nM T46937 C3LJD1 15650865 IC50 = 12000 nM T46937 CCT4M2 15650866 IC50 = 2600 nM T46937 CE5J9H 15650867 IC50 = 43000 nM T46937 COA46R 15650868 IC50 = 7000 nM T46937 C9R8UL 15650869 IC50 = 14000 nM T46937 C93OLX 15650870 IC50 = 14000 nM T46937 C85VYP 15650871 IC50 = 5000 nM T46937 C7JUK0 15650872 IC50 = 4000 nM T46937 C8S5GB 15650873 IC50 = 4000 nM T46937 C07KVS 15650874 IC50 = 4300 nM T46937 C84LEG 15650875 IC50 = 3000 nM T46937 CGA45I 15650876 IC50 = 4000 nM T46937 CDF63H 15650877 IC50 = 11000 nM T46937 CIQ3E8 15650878 IC50 = 12000 nM T46937 C60ZLB 15650879 IC50 > 75000 nM T46937 CFUQ16 15650880 IC50 = 12000 nM T46937 C9KQ1O 15650881 IC50 = 2000 nM T46937 CKM82C 15650882 IC50 = 2800 nM T46937 CE2G8F 15650883 IC50 = 8000 nM T46937 CBHY29 15650884 IC50 > 75000 nM T46937 C5XCK6 15650885 IC50 > 75000 nM T46937 CAC01F 15650886 IC50 = 59000 nM T46937 C2OMY3 15650887 IC50 = 53000 nM T46937 C5ZF4J 15650888 IC50 = 41000 nM T46937 CBJ3X2 15650897 IC50 = 8900 nM T46937 CC8UZ0 15650898 IC50 = 69000 nM T46937 CLP60K 15650899 IC50 = 1400 nM T46937 CLF93J 15982392 IC50 = 88 nM T46937 C5U0ED 15982393 IC50 = 54 nM T46937 CUCB94 15983052 IC50 = 67 nM T46937 C7SN1C 15983053 IC50 = 10 nM T46937 C0KRQ7 15983055 IC50 = 290 nM T46937 CS97JR 15983175 IC50 = 12 nM T46937 CBOI12 15983301 IC50 = 79 nM T46937 C0O5BA 15983546 IC50 = 17 nM T46937 CNZ60E 15983670 IC50 = 32 nM T46937 C83NXU 15983672 IC50 = 2900 nM T46937 C8QR1T 16739091 IC50 = 210 nM T46937 CN3M1O 16739092 IC50 = 237 nM T46937 C5VMW8 16739093 IC50 = 36.2 nM T46937 CJ0B4K 16739094 IC50 = 41 nM T46937 CPXH49 16739123 IC50 = 53 nM T46937 C9YK5V 16739124 IC50 = 160 nM T46937 C3T8JD 16739125 IC50 = 211 nM T46937 CZXV43 16739157 IC50 = 13 nM T46937 C8YUX6 16739158 IC50 = 288 nM T46937 C8UT0S 18717762 Ki = 5.012 nM T46937 CIX18B 20300396 IC50 = 810000 nM T46937 C7I1XM 20638786 Ki = 79.43 nM T46937 C5R9GU 20690429 Ki = 1.585 nM T46937 CV5O1T 20690446 Ki = 0.2512 nM T46937 CFO0M2 22184796 IC50 = 890 nM T46937 C8VW6J 22184814 IC50 = 840 nM T46937 C3KYN9 22184858 IC50 = 520 nM T46937 CK39QS 22184864 IC50 > 3000 nM T46937 C2AG9D 22184925 IC50 = 1800 nM T46937 C2R1DL 22185065 IC50 = 1200 nM T46937 CP7R6Y 22185105 IC50 = 910 nM T46937 CIL9Z6 23642329 IC50 = 280 nM T46937 C7GV8K 23662455 Ki = 10000 nM T46937 C7P1SA 23662764 Ki > 10000 nM T46937 CYZK58 23664788 Ki = 12200 nM T46937 C67WBS 23672996 Ki > 10000 nM T46937 CN5OC4 23673110 Ki = 10000 nM T46937 CZ7SX0 23675739 Ki > 10000 nM T46937 C4HJO0 23718715 Ki > 10000 nM T46937 CHI5U8 24750557 IC50 = 83 nM T46937 CKSW41 24750561 IC50 = 580 nM T46937 C6ST2J 24750719 IC50 = 1900 nM T46937 CN5X0A 24750723 IC50 = 230 nM T46937 C42LRT 24750874 IC50 = 490 nM T46937 CBS78H 24750876 IC50 = 430 nM T46937 CF3TC8 24751017 IC50 = 2400 nM T46937 CH85JK 24751297 IC50 = 960 nM T46937 CWX59N 24751300 IC50 = 1100 nM T46937 C6JQ1Z 24751438 IC50 = 1200 nM T46937 CJB3P1 24751572 IC50 = 1800 nM T46937 C24TLB 24751574 IC50 = 920 nM T46937 CA8GF1 24751575 IC50 = 1100 nM T46937 CX7ZD3 24751576 IC50 = 450 nM T46937 CK9W7Z 24751577 IC50 = 700 nM T46937 CABO68 24751579 IC50 = 1600 nM T46937 C0KEY2 24751581 IC50 = 1700 nM T46937 CPJ35E 24751708 IC50 = 2000 nM T46937 C7YDT9 24751709 IC50 = 1100 nM T46937 CCO3F4 24751710 IC50 = 460 nM T46937 CY1GS7 24751711 IC50 = 960 nM T46937 C84SJB 24751712 IC50 = 380 nM T46937 CHC14Q 24751850 IC50 = 420 nM T46937 C8VPT2 24751851 IC50 = 600 nM T46937 CRZ2M3 24751995 IC50 = 2000 nM T46937 CV61HI 24751996 IC50 = 950 nM T46937 C57JFC 24751997 IC50 = 100 nM T46937 C8KLX7 24751998 IC50 = 600 nM T46937 CRO0A3 24751999 IC50 = 2600 nM T46937 CA03BZ 24752128 IC50 = 1000 nM T46937 CN82FY 24752129 IC50 = 1060 nM T46937 CSV5W3 24752130 IC50 = 180 nM T46937 C9RPZ4 24752131 IC50 = 190 nM T46937 CJ3R5H 24752269 IC50 = 1800 nM T46937 CV2HF0 24752270 IC50 = 350 nM T46937 C05FEI 24752271 IC50 = 500 nM T46937 C2O5VN 24752419 IC50 = 450 nM T46937 C10VIG 24752420 IC50 = 180 nM T46937 C96OHY 24752421 IC50 = 270 nM T46937 C2OX8U 24752422 IC50 = 320 nM T46937 C8RW1L 24752557 IC50 = 490 nM T46937 C0H7LB 24752558 IC50 = 1300 nM T46937 CZA1J9 24752559 IC50 = 950 nM T46937 C26MWN 24752560 IC50 = 1500 nM T46937 CDKW17 24752561 IC50 = 270 nM T46937 CLAN49 24752711 IC50 = 240 nM T46937 CK35PX 24786234 IC50 = 2 nM T46937 CXZ58T 24799317 IC50 = 23000 nM T46937 C4QT3E 24799834 IC50 = 45070 nM T46937 C3HA4N 24799835 IC50 = 57070 nM T46937 CMJA06 24801414 IC50 = 52 nM T46937 CZO0W8 24801416 IC50 = 11170 nM T46937 C68IKP 24801573 IC50 = 3110 nM T46937 CC86QR 24829442 Ki = 15 nM T46937 CICF42 24829780 Ki = 42 nM T46937 C5JQB6 24829943 Ki = 114 nM T46937 CLG45Z 24830601 Ki = 209 nM T46937 CHA2I6 24868313 Ki > 10000 nM T46937 CLBW37 24937181 Ki = 11 nM T46937 CAN92Q 24968874 IC50 = 16 nM T46937 C20GMW 25022501 IC50 = 243 nM T46937 CK85UZ 25165435 IC50 = 76 nM T46937 CQOU76 39073052 Ki = 2100 nM T46937 C3TS7K 44125995 Ki = 372 nM T46937 C2Z4BL 44126504 Ki > 5000 nM T46937 CHQO90 44128387 Ki = 283 nM T46937 C2GK9P 44128468 Ki = 42 nM T46937 C5X1AQ 44128900 Ki = 42 nM T46937 CTVG29 44128901 Ki = 23 nM T46937 CM3YG0 44128980 Ki = 30 nM T46937 C7DST0 44128981 Ki = 40 nM T46937 CMWY16 44128982 Ki = 193 nM T46937 C6X3YI 44128983 Ki = 82 nM T46937 CGC56I 44129058 Ki = 23 nM T46937 C85OKZ 44129060 Ki = 0.8 nM T46937 C52VAZ 44129136 Ki = 5 nM T46937 CPM7E0 44129137 Ki = 1.5 nM T46937 C8R6LJ 44129368 Ki = 105 nM T46937 COC12W 44129369 Ki = 7.7 nM T46937 C6VKN3 44129371 Ki = 71 nM T46937 C0Z4TY 44129445 Ki = 303 nM T46937 C3VR2G 44129446 Ki = 66 nM T46937 CK5SD1 44129447 Ki = 56 nM T46937 C7F2LI 44129448 Ki = 41 nM T46937 CGH08U 44129449 Ki = 33 nM T46937 CUH15M 44129451 Ki = 107 nM T46937 C5H3LE 44129522 Ki = 219 nM T46937 C47SDX 44129524 Ki = 27 nM T46937 CNM86R 44129525 Ki = 459 nM T46937 C5WP3I 44157464 Ki = 3760 nM T46937 CTZ81X 44157465 Ki = 884 nM T46937 C0LTK8 44157466 Ki = 10000 nM T46937 CJN39O 44157467 Ki > 10000 nM T46937 CJ4E6Y 44157518 Ki = 614 nM T46937 CI21HV 44157519 Ki = 63 nM T46937 CU5X8A 44157520 Ki = 541 nM T46937 CHF40V 44241562 IC50 = 8080 nM T46937 CL72TA 44295999 IC50 = 480 nM T46937 CH06ZN 44296001 IC50 = 2200 nM T46937 CJ7Z2M 44296486 IC50 = 170 nM T46937 CXZ0V1 44304081 IC50 = 35000 nM T46937 CTY4U2 44323790 EC50 = 960 nM T46937 C4D0ZF 44443917 IC50 = 100 nM T46937 CGP27V 44443919 IC50 = 0.3162 nM T46937 CLBC52 44443921 IC50 = 0.5012 nM T46937 CSN3M1 44443933 Ki = 3.162 nM T46937 CQR1P9 44443935 Ki = 1.995 nM T46937 CU3E5S 44443938 Ki = 5.012 nM T46937 C64HOJ 44443939 Ki = 0.631 nM T46937 CF7SB1 44452736 IC50 = 4730 nM T46937 CGI90J 44452737 IC50 = 1270 nM T46937 C9A8LW 44452878 IC50 = 616 nM T46937 CAT75E 44452879 IC50 = 1310 nM T46937 CR2M9J 44452898 IC50 = 40 nM T46937 C2IDA9 44452921 IC50 = 663 nM T46937 CJ08RK 44452925 IC50 = 2480 nM T46937 CK0E2B 44452926 IC50 = 2550 nM T46937 C96SQE 44452947 IC50 = 3800 nM T46937 C9LMZ4 44452951 IC50 = 2700 nM T46937 CK1AU7 44452952 IC50 = 580 nM T46937 CM60LZ 44452977 IC50 = 9900 nM T46937 C5XKP6 44452982 IC50 = 2490 nM T46937 CEW93M 44453009 IC50 = 4330 nM T46937 CM34EZ 44453032 IC50 = 495 nM T46937 C78BQV 44453107 IC50 = 201 nM T46937 CRS1M7 44453109 IC50 = 4860 nM T46937 C1DWQ9 44453110 IC50 = 2230 nM T46937 C0JN3W 44453131 IC50 = 2950 nM T46937 CJPF52 44453132 IC50 = 513 nM T46937 CEYV61 44456046 Ki = 1850 nM T46937 CA82XJ 44456077 Ki > 10000 nM T46937 C1DU4Z 44456078 Ki = 6760 nM T46937 C1W8IK 44456201 Ki = 10000 nM T46937 CL74DQ 44457247 IC50 = 8680 nM T46937 C6LWM3 44457249 IC50 = 3300 nM T46937 C56JUQ 44457251 IC50 = 522 nM T46937 CYB0H2 44457262 IC50 = 8290 nM T46937 CIP6B7 44457274 IC50 = 1820 nM T46937 C23NHF 44457276 IC50 = 16700 nM T46937 C9S6OQ 44457278 IC50 = 11710 nM T46937 C5Y2RW 44457290 IC50 = 27100 nM T46937 C0V3OU 44457292 IC50 = 4630 nM T46937 CD70CI 44457294 IC50 = 6540 nM T46937 CVT6W1 44457324 IC50 = 3060 nM T46937 C3D5SF 44457338 IC50 = 7590 nM T46937 C5ITD1 44457371 IC50 = 10690 nM T46937 CQI0O7 44457392 IC50 = 16880 nM T46937 C2UMA5 44457401 IC50 = 48 nM T46937 CTC7N5 44457411 IC50 = 12920 nM T46937 C6BAK3 44457422 IC50 = 23930 nM T46937 C78AUJ 44464779 IC50 = 3 nM T46937 C9XNT2 44554515 IC50 = 1 nM T46937 CTJQ59 44555026 IC50 = 100 nM T46937 C2OTX9 44583417 Ki > 10000 nM T46937 C2KWN7 44583454 Ki > 10000 nM T46937 C41BAQ 44583493 Ki = 25100 nM T46937 CD47MO 44583494 Ki = 10000 nM T46937 CVP5H0 44583549 Ki = 7070 nM T46937 CD5O7G 44583580 Ki = 1900 nM T46937 C9BM5G 44583581 Ki = 660 nM T46937 C4ZTQ0 44583637 Ki > 10000 nM T46937 CIA6S4 44608149 IC50 = 57 nM T46937 CW3XJ1 44610468 IC50 = 17 nM T46937 C3T6BG 44610518 IC50 = 270 nM T46937 CO7K2H 44610519 IC50 = 42 nM T46937 CG7RS8 44610522 IC50 = 130 nM T46937 CPQ09B 44610759 Ki = 5 nM T46937 C8BI6C 44610760 Ki = 4 nM T46937 CP68UD 44631970 Ki = 15 nM T46937 CIX15W 44631974 Ki = 2.1 nM T46937 C43HON 44762396 IC50 = 1540 nM T46937 C6K5ZT 45139236 Ki = 1.5 nM T46937 CYC57N 45139400 Ki = 69 nM T46937 C4TKJ3 45139401 Ki = 31 nM T46937 C9M7PY 45139402 Ki = 6.9 nM T46937 CGX5E1 45139403 Ki = 5.9 nM T46937 CR3ZA2 45139404 Ki = 10 nM T46937 CBR1T8 45139405 Ki = 1.3 nM T46937 CKJ3F7 45139406 Ki = 4.5 nM T46937 C23TQM 45139407 Ki = 12 nM T46937 CR48LE 45139408 Ki = 1.3 nM T46937 CV5Z1L 45139585 Ki = 11 nM T46937 CX0S1R 45139586 Ki = 6.9 nM T46937 CTA9Y2 45139587 Ki = 3.7 nM T46937 CN3F4K 45139588 Ki = 4.2 nM T46937 C9CB8Q 45139589 Ki = 5.3 nM T46937 C15JAY 45139590 Ki = 7.4 nM T46937 CDK5Q7 45139591 Ki = 7.5 nM T46937 CNL12Y 45139592 Ki = 10 nM T46937 CYJ3R6 45139764 Ki = 94 nM T46937 C2GTC1 45139765 Ki = 280 nM T46937 C4L8KR 45139766 Ki = 3.7 nM T46937 C6UQY5 45139767 Ki = 11 nM T46937 C96FBC 45139768 Ki = 3 nM T46937 CYF1Q0 45139769 Ki = 2.5 nM T46937 CR9T4K 45139770 Ki = 11 nM T46937 C38IDA 45139771 Ki = 2.4 nM T46937 C0Y5XP 45139772 Ki = 2.6 nM T46937 C0VN3U 45139773 Ki = 5.8 nM T46937 C5S8FZ 45139945 Ki = 18 nM T46937 CRQ05I 45139946 Ki = 79 nM T46937 CI9O6G 45139947 Ki = 47 nM T46937 CD9WJ2 45139948 Ki = 44 nM T46937 CU6V2B 45139949 Ki = 28 nM T46937 CAWB56 45139950 Ki = 3.7 nM T46937 CL09QD 45139951 Ki = 11 nM T46937 CDI3Y9 45139952 Ki = 7.9 nM T46937 CEC34T 45139953 Ki = 18 nM T46937 C96JYB 45139954 Ki = 8.8 nM T46937 C3PQS1 45139955 Ki = 13 nM T46937 CM7S2J 45139956 Ki = 7.9 nM T46937 C8BQ4F 45139957 Ki = 6.1 nM T46937 CQZ14O 45139958 Ki = 4.6 nM T46937 C9MWK0 45140154 Ki = 46 nM T46937 C6KZ5T 45140155 Ki = 15 nM T46937 C5H8ZC 45140156 Ki = 33 nM T46937 CZ5O9H 45140157 Ki = 42 nM T46937 CA3F2Q 45140158 Ki = 492 nM T46937 C7VG9C 45140159 Ki = 4.5 nM T46937 CJ5W6E 45140160 Ki = 20 nM T46937 CVY48K 45140161 Ki = 89 nM T46937 CH9ZS5 45140162 Ki = 18 nM T46937 CWL6A9 45140163 Ki = 8.6 nM T46937 C9RK4J 45140164 Ki = 11 nM T46937 C27UDM 45140165 Ki = 2.8 nM T46937 C32CMN 45140166 Ki = 4.4 nM T46937 CR2EO1 45140353 Ki = 196 nM T46937 C58XUB 45140361 Ki = 14 nM T46937 CSL0F1 45140362 Ki = 8.4 nM T46937 C1VGX4 45140363 Ki = 9.4 nM T46937 CUHA50 45140364 Ki = 4.5 nM T46937 CD4BF9 45140365 Ki = 2.6 nM T46937 CSM1K9 45140366 Ki = 3.2 nM T46937 C6PYZ9 45140367 Ki = 5.4 nM T46937 CHYK36 45140368 Ki = 5.8 nM T46937 C30VPY 45140551 Ki = 2 nM T46937 CUEF96 45140552 Ki = 1.5 nM T46937 CCPI40 45140553 Ki = 1.8 nM T46937 C0JX7Z 45140554 Ki = 1.7 nM T46937 C2PKQ0 45140555 Ki = 8.6 nM T46937 C9Z6RL 45140556 Ki = 3.8 nM T46937 CKZ19G 45140557 Ki = 3.6 nM T46937 C1A6PI 45140558 Ki = 2.8 nM T46937 C0A8CM 45140743 Ki = 45 nM T46937 CX2K5M 45140744 Ki = 45 nM T46937 CI1B0U 45140745 Ki = 112 nM T46937 C8P4YN 45140746 Ki = 39 nM T46937 CK53VS 45140748 Ki = 2.1 nM T46937 CFGH76 45140749 Ki = 5.5 nM T46937 CTH63Z 45140750 Ki = 45 nM T46937 CM32HO 45140751 Ki = 1.7 nM T46937 C45KFH 45140752 Ki = 8.4 nM T46937 CD5H9K 45140753 Ki = 8.3 nM T46937 C6WN2Z 45140754 Ki = 12 nM T46937 CA1PF4 45140927 Ki = 54 nM T46937 C8KI9O 45140928 Ki = 2.4 nM T46937 C9LEC4 45140929 Ki = 4 nM T46937 C76CDE 45140930 Ki = 3.3 nM T46937 CNB64P 45140931 Ki = 3.5 nM T46937 C9UT6B 45140932 Ki = 2.3 nM T46937 CF98ZN 45140933 Ki = 7.7 nM T46937 C7WH3A 45140934 Ki = 11 nM T46937 CL7RE6 45140935 Ki = 4.8 nM T46937 CB4A8S 45140936 Ki = 22 nM T46937 C4YBC2 45140937 Ki = 3.3 nM T46937 CN2E7I 45140938 Ki = 2.1 nM T46937 CH2AT1 45140939 Ki = 3.7 nM T46937 CPA02Z 45141128 Ki = 2.7 nM T46937 CYQM02 45141129 Ki = 5 nM T46937 CY7NU0 45141130 Ki = 64 nM T46937 C79QWL 45141131 Ki = 4 nM T46937 CF6TO0 45141133 Ki = 6 nM T46937 C7IVG1 45141134 Ki = 2.5 nM T46937 C8P3QC 45141135 Ki = 10 nM T46937 C8FN0X 45141136 Ki = 1 nM T46937 C7QN8R 45141341 Ki = 3.2 nM T46937 CSG1V2 45141342 Ki = 1.5 nM T46937 C3XIM0 45141343 Ki = 12 nM T46937 CBU59A 45141344 Ki = 5.7 nM T46937 CWQD34 45141345 Ki = 9.4 nM T46937 CC0P6E 45141347 Ki = 12 nM T46937 CK0PL3 45141578 Ki = 9.8 nM T46937 CVE0H2 45141579 Ki = 2.1 nM T46937 CQSN29 45141580 Ki = 5.5 nM T46937 CZ94QB 45141581 Ki = 15 nM T46937 C3S2PW 45141582 Ki = 20 nM T46937 C79LVU 45141583 Ki = 7.6 nM T46937 CAO1U8 45141584 Ki = 5 nM T46937 CTI7Y8 45141585 Ki = 7 nM T46937 CSCF14 45141770 Ki = 17 nM T46937 C8N6QH 45141771 Ki = 6.5 nM T46937 C2L0AO 45141772 Ki = 22 nM T46937 CP54ZM 45141773 Ki = 9 nM T46937 CZ06AP 45141774 Ki = 9.9 nM T46937 CDV5G3 45141776 Ki = 19 nM T46937 C94KUS 45141980 Ki = 10 nM T46937 CS81XD 45141981 Ki = 2.4 nM T46937 CG35EM 45141982 Ki = 22 nM T46937 C9Y8AH 45141983 Ki = 1.5 nM T46937 CK3S1X 45141984 Ki = 6.5 nM T46937 C2U6YC 45141985 Ki = 5.1 nM T46937 C5CQ9D 45141986 Ki = 2.5 nM T46937 C4IAD0 45141987 Ki = 4.5 nM T46937 CF6AD8 45142213 Ki > 5680 nM T46937 C6VG8P 45142216 Ki = 1.9 nM T46937 C47RYG 45142217 Ki = 1.1 nM T46937 CG98TA 45142218 Ki = 11 nM T46937 CAFL20 45142219 Ki = 3.3 nM T46937 C4LI9R 45142220 Ki = 5.3 nM T46937 C3TRE2 45142221 Ki = 3.9 nM T46937 CC7VE3 45142222 Ki = 10 nM T46937 CPSW54 45142223 Ki = 2.6 nM T46937 CH4N7O 45142445 Ki = 2.6 nM T46937 CM2DP3 45142446 Ki = 62 nM T46937 CYS85V 45142447 Ki = 94 nM T46937 CL5KF9 45142448 Ki = 120 nM T46937 C6E3XL 45142449 Ki = 68 nM T46937 C4STP8 45142450 Ki = 7.6 nM T46937 CFS9H3 45142451 Ki = 5.3 nM T46937 CFG74S 45142452 Ki = 5.3 nM T46937 CY43GD 45142453 Ki = 5.5 nM T46937 C6A7CG 45263658 Ki = 6.31 nM T46937 CGX80T 45267707 Ki = 1190 nM T46937 C86TKV 45267712 Ki > 5700 nM T46937 CJC9Q1 45267721 Ki = 7 nM T46937 CD1W5O 45267722 Ki = 96 nM T46937 C8GXD4 45267728 Ki = 92 nM T46937 C3AK2I 45267738 Ki = 157 nM T46937 C86BFJ 45267750 Ki = 49 nM T46937 C9NS3P 45267751 Ki = 12 nM T46937 CTK5Y2 45267776 Ki = 373 nM T46937 C2FD9O 45268593 Ki = 14 nM T46937 C5Q0YP 45268594 Ki = 28 nM T46937 CN4HX2 45268619 Ki = 26 nM T46937 C9B2IO 45268630 Ki = 31 nM T46937 C4U2CA 45268641 Ki = 93 nM T46937 CIB4K5 45268642 Ki = 15 nM T46937 CS0DF4 45268660 Ki > 5700 nM T46937 C7WJU9 45269438 Ki = 11 nM T46937 C9FA5L 45269454 Ki = 68 nM T46937 CU37SK 45269461 Ki = 23 nM T46937 CA6XK1 45269465 Ki = 270 nM T46937 CX4JK8 45269472 Ki = 20 nM T46937 CK3HU9 45269473 Ki = 95 nM T46937 CWNL09 45269482 Ki = 157 nM T46937 CV8F1O 45269483 Ki = 48 nM T46937 CS5GA3 45269484 Ki = 80 nM T46937 CR32NL 45269502 Ki > 5400 nM T46937 C2CEO3 45270266 Ki = 484 nM T46937 CI8QM6 45270267 Ki = 733 nM T46937 COWU62 45270274 Ki = 5.7 nM T46937 C41HAP 45270288 Ki = 328 nM T46937 CSEQ82 45270294 Ki = 214 nM T46937 C4A9PG 45270295 Ki = 81 nM T46937 CF0L5I 45270296 Ki = 35 nM T46937 CFZS57 45270300 Ki = 99 nM T46937 CSOT19 45270314 Ki = 39 nM T46937 CLEI08 45270318 Ki = 146 nM T46937 CPY1U9 45270321 Ki = 69 nM T46937 C34GWX 45270322 Ki = 47 nM T46937 C0HGU8 45270323 Ki = 10 nM T46937 CGBA08 45271082 Ki = 356 nM T46937 C8C4FS 45271092 Ki = 27 nM T46937 CV0P4Y 45271100 Ki = 43 nM T46937 C2SY0E 45271128 Ki = 190 nM T46937 C5Z7QD 45271145 Ki = 36 nM T46937 CK6C5N 45271154 Ki = 11 nM T46937 CPBF35 45271155 Ki = 18 nM T46937 CI0NU9 45271162 Ki = 15 nM T46937 C6XI2F 45271977 Ki = 1610 nM T46937 C7CHR1 45271978 Ki = 2440 nM T46937 CFN09J 45271984 Ki = 29 nM T46937 C41ZUD 45272035 Ki = 189 nM T46937 CYKJ35 45272036 Ki = 18 nM T46937 C3GQ2K 45272054 Ki = 40 nM T46937 CO4F1R 45272055 Ki = 34 nM T46937 CHV96U 45272074 Ki = 3640 nM T46937 C1M4YS 45272842 Ki = 455 nM T46937 C1RJ0T 45272846 Ki = 203 nM T46937 CE7WP6 45272861 Ki = 9.9 nM T46937 CM24LU 45272869 Ki = 3.5 nM T46937 C2RUJ8 45272880 Ki = 18 nM T46937 C9RUX5 45272881 Ki = 33 nM T46937 CYCS21 45272902 Ki = 209 nM T46937 CCDZ68 45273782 Ki = 76 nM T46937 CI1O0G 45273789 Ki = 64 nM T46937 CZRX73 45273798 Ki = 145 nM T46937 CZK63V 45273811 Ki = 99 nM T46937 C0HB9W 45273812 Ki = 35 nM T46937 CF92SN 45273818 Ki = 24 nM T46937 C8D0IE 45273819 Ki = 14 nM T46937 C21EFP 45273820 Ki = 7 nM T46937 C5SAO6 45485848 Ki = 12 nM T46937 CO4N6X 45485849 Ki = 1.2 nM T46937 C9A1QE 45485850 Ki = 1.2 nM T46937 CA52GP 45485851 Ki = 55 nM T46937 C7SEY6 45485852 Ki = 72 nM T46937 CW9ZK8 45485853 Ki = 27 nM T46937 CW56DP 45485854 Ki = 184 nM T46937 CVO1I8 45485855 Ki = 2.8 nM T46937 C57UAI 45485856 Ki = 11 nM T46937 C9XPS3 45485857 Ki = 19 nM T46937 CJ35NO 45485858 Ki = 16 nM T46937 CF15OM 45485859 Ki = 2.2 nM T46937 C30RBF 45485860 Ki = 31 nM T46937 C0O9SQ 45485861 Ki = 15 nM T46937 CQL67G 45485862 Ki = 5.7 nM T46937 CP1F0U 45485863 Ki = 12 nM T46937 C9F8JX 45485864 Ki = 123 nM T46937 CD4ZJ1 45485865 Ki = 42 nM T46937 CI8O1H 45485880 Ki = 4.5 nM T46937 CP0YJ1 45485881 Ki = 22 nM T46937 C3Q7DF 45485882 Ki = 17 nM T46937 CD5N2R 45485883 Ki = 70 nM T46937 CI2Y7S 45485884 Ki = 1.2 nM T46937 CX0NC7 45485885 Ki = 5.2 nM T46937 CWK64B 45485886 Ki = 1 nM T46937 C6Q5RW 45485887 Ki = 11 nM T46937 CJU65A 45485888 Ki = 2.5 nM T46937 CN0S5H 45485889 Ki = 1.2 nM T46937 C26XAU 45485890 Ki = 4.8 nM T46937 CL7EW0 45485891 Ki = 38 nM T46937 CZ2V1S 45485892 Ki = 4.1 nM T46937 CN5ZT0 45485893 Ki = 19 nM T46937 C4PE7J 45485894 Ki = 9.4 nM T46937 CXP98J 45485895 Ki = 35 nM T46937 C9D6YA 45485896 Ki = 2.7 nM T46937 C2WC1A 45485897 Ki = 11 nM T46937 CET6H3 45485898 Ki = 0.69 nM T46937 CP1NK2 45485899 Ki = 8.4 nM T46937 C4NS9G 45485900 Ki = 2 nM T46937 CL52BA 45485901 Ki = 22 nM T46937 C1AG4M 45485902 Ki = 3.7 nM T46937 CT8FO2 45485903 Ki = 29 nM T46937 CW78YS 45485904 Ki = 1.2 nM T46937 CC83HT 45485905 Ki = 5.8 nM T46937 C7K4OZ 45485906 Ki = 2.9 nM T46937 C8COX6 45485907 Ki = 14 nM T46937 CS1PN6 45485908 Ki = 2.6 nM T46937 CDLE53 45485909 Ki = 6.8 nM T46937 CG3W8L 45485910 Ki = 2.1 nM T46937 CT6ZU5 45485911 Ki = 2.3 nM T46937 CZW7Y2 45485912 Ki = 12 nM T46937 CR1YJ9 45485913 Ki = 7.5 nM T46937 CM26UH 45485914 Ki = 1.7 nM T46937 CR76LO 45485915 Ki = 1.5 nM T46937 C5NA1E 45485916 Ki = 7.4 nM T46937 C7HP0T 45485917 Ki = 1.3 nM T46937 CMO8T0 45485918 Ki = 2.9 nM T46937 CY34QO 45485919 Ki = 5.9 nM T46937 CNZ61J 45485920 Ki = 3 nM T46937 CA4RQ5 45485921 Ki = 9.4 nM T46937 C5H9DG 45485922 Ki = 1.2 nM T46937 C8IG5O 45485928 Ki = 11 nM T46937 CYM5B3 45485929 Ki = 2.2 nM T46937 CIWL84 45485930 Ki = 11 nM T46937 CEY93C 45485931 Ki = 0.61 nM T46937 C46HGC 45485932 Ki = 0.4 nM T46937 CRUQ16 45485933 Ki = 2.7 nM T46937 CK0S4N 45485934 Ki = 3 nM T46937 CH8ZV1 45485935 Ki = 2.8 nM T46937 C9H2MB 45485936 Ki = 2.1 nM T46937 C9AZ1U 45485937 Ki = 4.2 nM T46937 CT5P0G 45485938 Ki = 1.4 nM T46937 C7CP1G 45485939 Ki = 5 nM T46937 CNJP56 45485940 Ki = 7.4 nM T46937 CV9G4L 45485941 Ki = 5.3 nM T46937 CC57DL 45485942 Ki = 7.1 nM T46937 C2EQO3 45485943 Ki = 0.71 nM T46937 CPA16Y 45485944 Ki = 10 nM T46937 CME01Q 45485945 Ki = 8.4 nM T46937 CCZ16M 45485946 Ki = 12 nM T46937 COXP14 45485947 Ki = 4.3 nM T46937 C15VLC 45485948 Ki = 8.1 nM T46937 CQ17ES 45485949 Ki = 2 nM T46937 CB3C4P 45485950 Ki = 10.2 nM T46937 C1T4GP 45485951 Ki = 8.4 nM T46937 CLVB13 45485952 Ki = 0.99 nM T46937 CZ6W9U 45485953 Ki = 2 nM T46937 CRNG05 45485954 Ki = 3.5 nM T46937 C0G7VB 45485955 Ki = 1.3 nM T46937 C0H7QZ 45485956 Ki = 2.5 nM T46937 C73WXS 45485957 Ki = 0.38 nM T46937 C1MG8V 45485958 Ki = 0.6 nM T46937 C7F9WV 45485959 Ki = 0.79 nM T46937 C2DFB9 45485960 Ki = 3.6 nM T46937 CMQ15J 45485961 Ki = 0.83 nM T46937 C9IA7C 45485962 Ki = 0.7 nM T46937 CJ53NZ 45485963 Ki = 0.46 nM T46937 CF72IM 45485964 Ki = 3.6 nM T46937 CP0S1Q 45485965 Ki = 0.9 nM T46937 C5OIB6 45485966 Ki = 0.67 nM T46937 CM59YQ 45485967 Ki = 3.1 nM T46937 CU9M0E 45485968 Ki = 0.92 nM T46937 CQE2D6 45485969 Ki = 1.6 nM T46937 CQWH31 45487789 Ki = 223 nM T46937 CU12YR 45487790 Ki = 213 nM T46937 C93PEY 45487796 Ki = 130 nM T46937 CGAY47 45487800 Ki = 36 nM T46937 C6BJ1X 45487801 Ki = 539 nM T46937 C1C6BE 45487809 Ki = 37 nM T46937 CUTP63 45487813 Ki = 191 nM T46937 CA53DG 45487817 Ki = 27 nM T46937 CN17LS 45487821 Ki = 68 nM T46937 C7TO3S 45487837 Ki = 240 nM T46937 CO68ZR 45487838 Ki = 839 nM T46937 CR24MB 45487841 Ki = 37 nM T46937 CKG8Z5 45487842 Ki = 78 nM T46937 CIOH61 45487843 Ki = 295 nM T46937 C47CSK 45487844 Ki = 380 nM T46937 C19MHZ 45487850 Ki = 31 nM T46937 COCJ34 46232830 Ki = 3.8 nM T46937 CQP62R 46232879 Ki = 1.5 nM T46937 CWA82V 46232880 Ki = 7.5 nM T46937 CKN5C7 46232881 Ki = 4 nM T46937 C09PJV 46232882 Ki = 11 nM T46937 CI8Y4W 46232883 Ki = 2.8 nM T46937 CJ0W1O 46232884 Ki = 12 nM T46937 C9KY1C 46232885 Ki = 8 nM T46937 C0Z2DI 46232886 Ki = 25 nM T46937 CV9PC5 46232887 Ki = 0.79 nM T46937 CC20BA 46232888 Ki = 6.5 nM T46937 C9W8XE 46232889 Ki = 7.9 nM T46937 C6DS2Y 46232890 Ki = 0.58 nM T46937 C1SK2F 46232891 Ki = 4.3 nM T46937 C7A1BX 46232892 Ki = 6 nM T46937 CB2SN5 46232893 Ki = 2.6 nM T46937 CL21DR 46232894 Ki = 0.98 nM T46937 CKZS79 46232895 Ki = 12 nM T46937 CR5CV6 46232896 Ki = 1.1 nM T46937 CPJ41D 46232897 Ki = 4 nM T46937 CXM05D 46232898 Ki = 4.8 nM T46937 C8CMR5 46232899 Ki = 1.2 nM T46937 C8RP5H 46232900 Ki = 2.8 nM T46937 C4M9TH 46232901 Ki = 6.5 nM T46937 CT3CB2 46232902 Ki = 15 nM T46937 CM4S2A 46232903 Ki = 29 nM T46937 CVW47M 46232904 Ki = 13 nM T46937 CW5C6S 46232905 Ki = 8.3 nM T46937 CT1V2F 46232906 Ki = 6.3 nM T46937 CT0JF6 46232907 Ki = 4.5 nM T46937 CM4FR7 46232908 Ki = 8.5 nM T46937 CCA21B 46232909 Ki = 8.4 nM T46937 C2LX4J 46232910 Ki = 8.9 nM T46937 CL6KU2 46232911 Ki = 1.7 nM T46937 C9N2DT 46232912 Ki = 4.9 nM T46937 C3EWR0 46232913 Ki = 5.9 nM T46937 C4Q7ED 46232914 Ki = 5.2 nM T46937 CSX0C1 46232915 Ki = 22 nM T46937 C5V7ZC 46232916 Ki = 16 nM T46937 C5K0AF 46232917 Ki = 2.8 nM T46937 CG2Q0P 46232918 Ki = 6.3 nM T46937 C2CBX6 46232919 Ki = 5.9 nM T46937 CP4DL3 46232920 Ki = 12 nM T46937 CWE0H5 46232921 Ki = 10 nM T46937 C6OJ8N 46232922 Ki = 18 nM T46937 C2M9NJ 46232923 Ki = 16 nM T46937 C96VNX 46232924 Ki = 31 nM T46937 CR6W5O 46232925 Ki = 22 nM T46937 CT21LP 46232926 Ki = 5.5 nM T46937 C9F3OL 46232927 Ki = 11 nM T46937 CQ5IB9 46232928 Ki = 7.3 nM T46937 C9FUS3 46232929 Ki = 9.9 nM T46937 CK4T7U 46232930 Ki = 10 nM T46937 CF18EQ 46232931 Ki = 17 nM T46937 C04DRM 46232932 Ki = 26 nM T46937 CXT3Q5 46232933 Ki = 13 nM T46937 C2HJ0E 46232934 Ki = 5 nM T46937 C1O5RS 46232935 Ki = 3.5 nM T46937 CW5F1D 46232936 Ki = 21 nM T46937 CE3R8K 46232937 Ki = 31 nM T46937 CTB0W6 46232940 Ki = 1.7 nM T46937 CNV89R 46232941 Ki = 2.6 nM T46937 CS60LF 46232942 Ki = 1.7 nM T46937 CB3T7O 46232943 Ki = 1.4 nM T46937 C7DO0E 46232944 Ki = 2.5 nM T46937 CYW60D 46232945 Ki = 2 nM T46937 C3U5NH 46232946 Ki = 5.5 nM T46937 C8XGB6 46232947 Ki = 3.3 nM T46937 CO0P1Y 46232948 Ki = 7.1 nM T46937 CNOI84 46232949 Ki = 0.64 nM T46937 CX1C6B 46232950 Ki = 1.7 nM T46937 CV82XQ 46232951 Ki = 2 nM T46937 CIC1X6 46233093 Ki > 3590 nM T46937 CCA2D3 46233094 Ki > 3590 nM T46937 CNRH34 46233095 Ki = 842 nM T46937 C8H1KS 46233096 Ki = 288 nM T46937 CIX16N 46233130 Ki = 277 nM T46937 CT7IR5 46233131 Ki = 613 nM T46937 C14FKB 46233132 Ki = 55 nM T46937 CRPZ16 46233133 Ki = 54 nM T46937 CZ42KE 46233134 Ki = 842 nM T46937 CBT14W 46233174 Ki = 9 nM T46937 C2RIO9 46233175 Ki = 42 nM T46937 CM01FC 46233176 Ki = 8 nM T46937 CT56IZ 46233222 Ki = 132 nM T46937 C24DJR 46233223 Ki = 4.9 nM T46937 CQ9G7I 46233224 Ki = 6 nM T46937 C1C5YP 46233225 Ki = 6.2 nM T46937 CYG90O 46233226 Ki = 9.1 nM T46937 C3A5QP 46233227 Ki = 8.5 nM T46937 C0UVF8 46233228 Ki = 3 nM T46937 CWIN59 46233229 Ki = 2.3 nM T46937 C5Y9MB 46233230 Ki = 25 nM T46937 CVLW59 46233231 Ki = 5.7 nM T46937 C3UP9V 46233232 Ki = 4.1 nM T46937 C2VES7 46233233 Ki = 2.7 nM T46937 CH1V0B 46233234 Ki = 1.4 nM T46937 CD8K6M 46233235 Ki = 4.7 nM T46937 C2LZ8X 46233236 Ki = 5.8 nM T46937 C05LBX 46233237 Ki = 3.2 nM T46937 CYA83J 46233238 Ki = 9.2 nM T46937 C5ZGP7 46233239 Ki = 43 nM T46937 C57LNR 46233240 Ki = 11 nM T46937 CFLO71 46233241 Ki = 1.4 nM T46937 CBT2O9 46233242 Ki = 1.9 nM T46937 C26MHU 46233243 Ki = 1.7 nM T46937 C0NK3C 46233290 Ki > 5400 nM T46937 CX8Y9L 46233321 Ki > 5700 nM T46937 CJG70T 46233322 Ki = 373 nM T46937 C6IG4P 46233323 Ki = 3640 nM T46937 CXE56T 46233324 Ki = 28 nM T46937 CXEF72 46233325 Ki = 1.5 nM T46937 C2MK7D 46233326 Ki = 4.9 nM T46937 C3ZCA6 46233327 Ki = 2.8 nM T46937 C35TNK 46233328 Ki = 3.6 nM T46937 CD92SU 46233329 Ki = 2.4 nM T46937 CL5SQ7 46233330 Ki = 11 nM T46937 C8MH6O 46233354 Ki = 484 nM T46937 C0E7KD 46233355 IC50 = 64 nM T46937 C48ZWF 46233356 Ki = 1190 nM T46937 C8BG5H 46233357 Ki = 733 nM T46937 CD0JE2 46233386 Ki = 1610 nM T46937 CHR32N 46233387 Ki > 5700 nM T46937 C49FAM 46233388 Ki = 1430 nM T46937 C86YOM 46233389 Ki = 1310 nM T46937 CWO5Q7 46233451 Ki = 87 nM T46937 C0IAC3 46233532 Ki > 3800 nM T46937 CU27WP 46233553 Ki > 3800 nM T46937 C8N0DY 46233554 Ki > 3590 nM T46937 C8W6EH 46233555 Ki > 2710 nM T46937 C5C6IN 46233586 Ki > 3590 nM T46937 CVT9H3 46233587 Ki > 3590 nM T46937 C69VFP 46233588 Ki > 3590 nM T46937 CO52XP 46233589 Ki = 3100 nM T46937 CKP38S 46233630 Ki = 1430 nM T46937 CXE6J5 46233631 Ki > 3590 nM T46937 C0Q9JC 46233632 Ki > 3590 nM T46937 C6P7IQ 46233668 Ki = 1880 nM T46937 C7QIO4 46233669 Ki > 3590 nM T46937 C5BMY9 46233670 Ki > 3590 nM T46937 CQNZ48 46241018 IC50 = 1400 nM T46937 CVP5D0 46241232 IC50 = 310 nM T46937 CEB52S 51032397 IC50 = 820000 nM T46937 CD9C1M 53233471 IC50 = 110 nM T46937 CR98BF 53350233 IC50 > 20000 nM T46937 CZI4D6 54579992 IC50 > 33000 nM T46937 C37EUW 54579993 IC50 > 33000 nM T46937 COH9F8 54579994 IC50 > 33000 nM T46937 CC4H9D 54579995 IC50 = 5500 nM T46937 CA95EC 54579996 IC50 = 3000 nM T46937 CA9W6B 54579997 IC50 = 4600 nM T46937 CD6R5X 54580043 IC50 > 33000 nM T46937 C2R4NO 54580044 IC50 = 29000 nM T46937 C01JXK 54580185 IC50 = 8500 nM T46937 C97ZBQ 54580993 IC50 = 2700 nM T46937 C4XDL0 54580994 IC50 = 9600 nM T46937 CT8S3D 54580995 IC50 = 2700 nM T46937 CI3A4F 54581027 IC50 = 760 nM T46937 CE4O3T 54581187 IC50 > 33000 nM T46937 C5H8MZ 54582036 IC50 > 33000 nM T46937 CO0AU9 54582209 IC50 > 33000 nM T46937 C4WH5A 54583010 IC50 > 33000 nM T46937 CPG8J3 54583974 IC50 = 4600 nM T46937 CSW27C 54583975 IC50 = 3000 nM T46937 C0B6QV 54584163 IC50 = 3800 nM T46937 CSM50F 54584960 IC50 = 2100 nM T46937 CS0YL3 54585098 IC50 = 8600 nM T46937 CDKR61 54585884 IC50 > 33000 nM T46937 CC8WI6 54585885 IC50 = 1800 nM T46937 CMIX30 54586076 IC50 = 890 nM T46937 CAB1F6 54732982 IC50 = 35000 nM T46937 C6MGO8 59534139 IC50 = 3 nM T46937 CTJM21 59534140 IC50 = 16 nM T46937 C8Z5FQ 60150614 IC50 > 10000 nM T46937 CA1KI7 66575818 IC50 = 1800 nM T46937 CM5CX3 66575819 IC50 = 5.1 nM T46937 C9EUN4 66575821 IC50 = 275 nM T46937 CFBA98 66575899 IC50 = 17 nM T46937 CC8K0B 66576220 IC50 = 7 nM T46937 CWD98Y 66576221 IC50 = 48 nM T46937 CXF02Q 66576296 IC50 = 15 nM T46937 C3JR2F 66576297 IC50 = 20 nM T46937 CU8A4R 66576298 IC50 = 27 nM T46937 CGRD93 66576377 IC50 = 22 nM T46937 C7EHJ6 66576448 IC50 = 500 nM T46937 CM8T2U 66576450 IC50 = 26 nM T46937 CXEP01 66576451 IC50 = 48 nM T46937 CA48WV 66576530 IC50 = 11 nM T46937 CLE6I7 66576610 IC50 = 50 nM T46937 CDH3K2 66854409 Ki = 613 nM T46937 C1NXY6 66854417 Ki = 238 nM T46937 C4EZJ9 66854424 Ki = 56 nM T46937 CK0MP7 66854575 Ki = 130 nM T46937 CW08UL 66854714 Ki = 183 nM T46937 CIM37J 66854759 Ki = 6.5 nM T46937 C04PRO 66854841 Ki = 5.7 nM T46937 C3J2VK 66854919 Ki = 180 nM T46937 CJY0F5 66855084 Ki = 56 nM T46937 CL65PY 66855175 Ki = 111 nM T46937 CBRU59 66855176 Ki > 5000 nM T46937 C9BKL3 66855197 Ki = 20 nM T46937 CS8B3V 66855285 Ki = 22 nM T46937 CR6B2X 66855732 Ki = 3.1 nM T46937 CR7W0Y 66855824 Ki = 7.3 nM T46937 CF0EX4 66855902 Ki = 5 nM T46937 CEJ1Z9 66855932 Ki = 48 nM T46937 CC4FR1 66856100 Ki = 172 nM T46937 C9E5DR 66856658 Ki = 51 nM T46937 CE45CN 66856790 Ki = 54 nM T46937 C4Z5AD 66856844 Ki = 19 nM T46937 CT16XL 66856952 Ki = 202 nM T46937 CIA84K 66856999 Ki = 207 nM T46937 C5AT4J 66857005 Ki = 80 nM T46937 CON4R7 66919940 Ki = 242 nM T46937 C1MNH8 66919958 Ki = 2720 nM T46937 CG0Y7J 66919996 Ki = 249 nM T46937 C3P4ZO 66920261 Ki = 574 nM T46937 CR1J5S 67459247 IC50 = 46 nM T46937 CB29XL 67459391 IC50 = 198 nM T46937 C0UXC9 67459556 IC50 = 95.5 nM T46937 C7NWK1 67459575 IC50 = 27 nM T46937 CPKE56 67460268 IC50 = 25 nM T46937 C2PYM3 67460312 IC50 = 100 nM T46937 CSA0H7 67460401 IC50 = 169 nM T46937 C63EOD 67460624 IC50 = 11 nM T46937 C3NWK7 67460741 IC50 = 129 nM T46937 CEHN20 67460935 IC50 = 36 nM T46937 C2KJ5P 67460979 IC50 = 52 nM T46937 CFDP23 67461519 IC50 = 257 nM T46937 CL5Q6D 67461716 IC50 = 21 nM T46937 CGBJ01 67461890 IC50 = 279 nM T46937 CA4E9H 67462098 IC50 = 40 nM T46937 CIXA56 67462183 IC50 = 56 nM T46937 CBHW91 67462328 IC50 = 201 nM T46937 C8W6XY 67462688 IC50 = 177 nM T46937 CMH1P6 67462816 IC50 = 59.5 nM T46937 CU90BR 67463039 IC50 = 122 nM T46937 CJD0F6 67463112 IC50 = 162 nM T46937 C6YF1M 67463220 IC50 = 52 nM T46937 CN0C3L 67463698 IC50 = 223 nM T46937 CRU26C 67463976 IC50 = 98 nM T46937 C5E4VR 67464143 IC50 = 2780 nM T46937 C6IO7J 67464394 IC50 = 219 nM T46937 CF59TE 68529945 Ki > 70000 nM T46937 C4VFI2 68530100 Ki > 70000 nM T46937 CNR0K9 68556549 IC50 = 190 nM T46937 CE7G0I 68556579 IC50 = 11000 nM T46937 CBP40H 68842714 IC50 = 680 nM T46937 C6TUH7 68910943 IC50 = 59 nM T46937 CDAK52 68911008 IC50 = 3200 nM T46937 C4VN1H 68911027 IC50 = 240 nM T46937 CV5HD9 68911088 IC50 = 110 nM T46937 CQC63W 68911120 IC50 = 710 nM T46937 CMQS54 68911155 IC50 = 27 nM T46937 CYAK78 68911205 IC50 = 39 nM T46937 C8QND7 68911289 IC50 = 9.5 nM T46937 C1B4XM 68913141 IC50 = 86 nM T46937 C87OTJ 68913220 IC50 = 690 nM T46937 CN61KV 68913927 IC50 = 190 nM T46937 C89ZLC 68914580 IC50 = 380 nM T46937 CE6OV1 68916097 IC50 = 3800 nM T46937 C70RGD 68916926 IC50 = 22 nM T46937 CP1NH0 68918061 IC50 = 240 nM T46937 CO43WI 69223141 IC50 = 220 nM T46937 C02UFD 69224054 IC50 = 7 nM T46937 C7SQT4 69224555 IC50 = 6 nM T46937 CCV7T0 69224603 IC50 = 180 nM T46937 C7Z9LF 69224988 IC50 = 30 nM T46937 C6EUY5 70618043 IC50 = 1070000 nM T46937 CI23ZK 70683418 Ki = 24 nM T46937 CKX7O8 70687668 Ki = 26 nM T46937 C84IOJ 70922234 IC50 = 46 nM T46937 CG56TS 71449929 Ki = 536 nM T46937 CGJ70Y 71455298 Ki = 173 nM T46937 C3LB1G 71462475 Ki = 958 nM T46937 CQ1SO4 71462476 Ki > 5000 nM T46937 CU8LY5 71607553 IC50 = 1730 nM T46937 CC4Y0J 71607589 IC50 = 280 nM T46937 CAH29B 71607592 IC50 = 16300 nM T46937 CI4PG7 71607631 IC50 = 220 nM T46937 CB3ED0 71607632 IC50 = 350 nM T46937 CTJ57B 71607634 IC50 = 11280 nM T46937 C0M4ED 71607663 IC50 = 6350 nM T46937 C6SLH7 71607664 IC50 = 1670 nM T46937 CJ3O6U 71607665 IC50 = 4820 nM T46937 CI04FH 71607666 IC50 = 1970 nM T46937 C4G8TJ 71607689 IC50 = 330 nM T46937 CRD4I9 71625797 Ki > 30000 nM T46937 CR0HK1 71740352 IC50 = 3700 nM T46937 CD8HZ2 71740353 IC50 = 5300 nM T46937 C8YZ2K 71740354 IC50 > 33000 nM T46937 CD6QV9 71740705 IC50 = 9300 nM T46937 C3UA0H 71740819 IC50 = 660 nM T46937 C9A2RG 73294137 IC50 = 230 nM T46937 CWV9G3 73603967 IC50 = 7 nM T46937 CT0FK7 74220534 IC50 = 40 nM T46937 C4IC1L 85909513 IC50 = 1300000 nM T46937 CUA2D5 85909522 IC50 = 1050000 nM T46937 CES8C1 90078535 IC50 > 10000 nM T46937 CCEV76 90644279 IC50 = 270 nM T46937 C1DML0 90644280 IC50 = 11500 nM T46937 C8E0CO 90644281 IC50 = 93 nM T46937 CXZ8K5 90644282 IC50 = 20000 nM T46937 C27IDK 118710241 IC50 = 46 nM T46937 CZ1D6E 118710242 IC50 = 76 nM T46937 C6JY4L 118710243 IC50 = 291 nM T46937 C2K0BX 118710244 IC50 = 23 nM T46937 C6HN8Y 118710245 IC50 = 39 nM T46937 CSAX95 118710246 IC50 = 43 nM T46937 C3PM1C 118710247 IC50 = 9 nM T46937 C10PNU 118711064 IC50 = 15000 nM T46937 CQGB17 118711065 IC50 = 272 nM T46937 CH28LI 118711066 IC50 = 93 nM T46937 CZAC38 118711067 IC50 = 800 nM T46937 CX24WK 118711069 IC50 = 31 nM T46937 C8KD4V 118711070 IC50 = 61 nM T46937 CA9VN3 118711071 IC50 = 94 nM T46937 CWD74Q 118711072 IC50 = 92 nM T46937 CGH0Q5 118711073 IC50 = 194 nM T46937 C9BG2N 118711074 IC50 = 124 nM T46937 CB08DC 118711075 IC50 = 61 nM T46937 C0FOK2 118711076 IC50 = 88 nM T46937 CP9DZ6 118711077 IC50 = 139 nM T46937 C5QB8J 118711078 IC50 = 47 nM T46937 CQZ27P 118711079 IC50 = 71 nM T46937 CE16LZ 118711080 IC50 = 84 nM T46937 C21ZCF 118711081 IC50 = 95 nM T46937 C7EXA6 118711082 IC50 = 71 nM T46937 CV6LC1 118711083 IC50 = 115 nM T46937 CT52KG 118711084 IC50 = 94 nM T46937 C7QFM6 118711085 IC50 = 87 nM T46937 C9CPJ3 118711086 IC50 = 46 nM T46937 C4QI0G 118711087 IC50 = 65 nM T46937 CC4NM8 118711088 IC50 = 73 nM T46937 C7S5GQ 118711089 IC50 = 111 nM T46937 C9VB0Y 118711090 IC50 = 100 nM T46937 CQC05Z 118711091 IC50 = 117 nM T46937 C9BZ8T 118711092 IC50 = 89 nM T46937 CCS8T0 118711093 IC50 = 106 nM T46937 C63SGU 118711094 IC50 = 33 nM T46937 C2TRX6 118711095 IC50 = 66 nM T46937 CH5X7F 118711096 IC50 = 121 nM T46937 CH2ST8 118711097 IC50 = 41 nM T46937 C1YR4C 118711098 IC50 = 29 nM T46937 CV7S2E 118711099 IC50 = 44 nM T46937 CN2T0A 118711100 IC50 = 76 nM T46937 C4FPM5 118711101 IC50 = 82 nM T46937 C8EP3X 118711102 IC50 = 27 nM T46937 CH42SK 118711172 IC50 = 102 nM T46937 CVI36F 118711173 IC50 = 28 nM T46937 CI94EL 118711174 IC50 = 19 nM T46937 CK78YV 118711175 IC50 = 19 nM T46937 C7B0TZ 118711176 IC50 = 66 nM T46937 C28QNW 118711177 IC50 = 15 nM T46937 C41DUA 118711178 IC50 = 86 nM T46937 CHV13J 118711179 IC50 = 70 nM T46937 C93IST 118711180 IC50 = 12 nM T46937 CW0NK6 118711181 IC50 = 48 nM T46937 CV02RP 118711182 IC50 = 34 nM T46937 C9QY3L 118711183 IC50 = 76 nM T46937 C63OXP 118711184 IC50 = 118 nM T46937 C64VUZ 118711185 IC50 = 138 nM T46937 C5NW9I 118711186 IC50 = 99 nM T46937 CS6V2F 118711187 IC50 = 142 nM T46937 C4G0NR 118711190 IC50 = 11 nM T46937 C0R4SX 118711191 IC50 = 11 nM T46937 CP9U2T 118711192 IC50 = 336 nM T46937 CU0PB7 118711193 IC50 = 143 nM T46937 C7RFM3 118711194 IC50 = 574 nM T46937 CE37HG 118711247 IC50 = 480 nM T46937 CEWV27 118711248 IC50 = 75 nM T46937 C9UJH0 118711249 IC50 = 266 nM T46937 CCN04Q 118711250 IC50 = 559 nM T46937 CB1L4V 118711969 IC50 = 80 nM T46937 CD3W2I 118711970 IC50 = 17 nM T46937 CD7G9H 118711971 IC50 = 47 nM T46937 C2C6BT 118711972 IC50 = 24 nM T46937 CP32DO 118711973 IC50 = 4000 nM T46937 CU6ZG2 118711974 IC50 = 304 nM T46937 CKR2L7 127038948 IC50 = 730 nM T46937 CBXP14 127038950 IC50 = 1120 nM T46937 CN7C8A 127039315 IC50 = 220 nM T46937 C2N9XI 127039918 IC50 = 210 nM T46937 CF0M8H 127039999 IC50 = 2400 nM T46937 CV8XS2 127040346 IC50 = 140 nM T46937 CIMH26 127040665 IC50 = 1020 nM T46937 C7RQT4 127040675 IC50 = 3100 nM T46937 CNPL48 127040996 IC50 = 9300 nM T46937 CH42ZI 127040998 IC50 = 340 nM T46937 CV4AL5 127041004 IC50 = 1350 nM T46937 C9ON2A 127041006 IC50 > 200000 nM T46937 CKB30T 127041008 IC50 = 156000 nM T46937 CL7VJ2 127047545 IC50 = 8.3 nM T46937 CHIG78 132574706 IC50 = 2340 nM T46937 CMG81E 135434015 EC50 = 100 nM T46937 CE24WD 135838395 EC50 = 6910 nM T46937 C8PHX6 137631406 IC50 = 940000 nM T46937 C6ZB1D 137632198 IC50 = 60.4 nM T46937 CRO8T3 137634506 IC50 = 1260000 nM T46937 CPOU41 137635690 IC50 = 1320000 nM T46937 C7VYP0 137639442 IC50 = 1020000 nM T46937 C4GA0J 137641946 IC50 = 3590 nM T46937 CT92FG 137642967 IC50 = 940000 nM T46937 C7O3US 137643396 IC50 = 2410 nM T46937 C6G7QI 137644622 IC50 = 860000 nM T46937 CUR8V1 137648798 IC50 = 2960 nM T46937 CE5ON3 137649986 IC50 = 1620000 nM T46937 CAC0Y8 137650737 IC50 = 650000 nM T46937 CM8UT3 137651269 IC50 = 1070000 nM T46937 C3A9YO 137651373 IC50 = 930000 nM T46937 C6G8JF 137651603 IC50 = 950000 nM T46937 CK74CY 137652006 IC50 = 910000 nM T46937 CJ69KN 137652138 IC50 = 920000 nM T46937 CJ07WQ 137654461 IC50 = 1040000 nM T46937 CUAT36 137656414 IC50 = 1500000 nM T46937 CVQ2D4 145967492 IC50 = 86 nM T46937 CMCP51 145967502 IC50 = 1100 nM T46937 CTAL93 145967657 IC50 = 190 nM T46937 CYDT13 145967823 IC50 = 1700 nM T46937 CM6QO7 145967859 IC50 = 4500 nM T46937 CE89CL 145968144 IC50 = 14000 nM T46937 CM6D7Y 145968628 IC50 = 1100 nM T46937 CG7N0Z 145969318 IC50 = 22000 nM T46937 CIT74R 145969360 IC50 = 1500 nM T46937 CJ4YR6 145969559 IC50 = 7900 nM T46937 C5GVL6 145969883 IC50 = 2100 nM T46937 C8SMZ3 145970029 IC50 = 4300 nM T46937 CC0QB7 145970199 IC50 = 8600 nM T46937 CN3L2D 145970219 IC50 = 1500 nM T46937 CY5Z4X 145970444 IC50 = 200 nM T46937 CCU54P 145970653 IC50 = 18000 nM T46937 C03KDV 145970872 IC50 = 1900 nM T46937 CLPQ37 145970953 IC50 = 2500 nM T46937 C4XRG5 145971125 IC50 = 270 nM T46937 C7GI9R 145971167 IC50 = 1100 nM T46937 C54YEP 145986354 IC50 = 21000 nM T46937 CG7JW1 145986356 IC50 = 860 nM T46937 CZ3B4C 145987950 IC50 = 150 nM T46937 C6BOT2 145987961 IC50 = 26000 nM T46937 CNP81R 54719874 IC50 = 800 nM T46937 D00BSX 122635 Ki > 10000 nM T46937 D01APA 66855377 Ki = 7.7 nM T46937 D01IEX 44583582 Ki = 24.9 nM T46937 D02TXW 16681707 IC50 = 29 nM T46937 D07MTB 11510579 Ki > 70000 nM T46937 D08DXA 23675622 IC50 = 3120 nM T46937 D09BUG 10207 Ki > 10000 nM T46937 D0B0ZQ 9875920 Ki = 680 nM T46937 D0C0KJ 5280879 EC50 = 1.3 nM T46937 D0KF2P 44126037 Ki = 139 nM T46937 D0N3FL 44157521 Ki = 21 nM T46937 D0P6KN 44457307 IC50 = 34730 nM T77546 D05EAM 4735 Ki = 290 nM T77546 D0V0NL 2146 Ki = 140 nM T77546 CLRO58 127456 Ki = 1700 nM T77546 CQ85DB 6438855 Ki = 200 nM T77546 C9C6LU 10334080 IC50 > 1000000 nM T77546 CCUJ60 10445232 IC50 > 1000000 nM T77546 CY41LT 10445774 IC50 > 1000000 nM T77546 C9X2AQ 10583188 IC50 = 120 nM T77546 CBP6U9 10589155 IC50 > 1000000 nM T77546 CDY0H7 10728071 IC50 = 1000000 nM T77546 C9ILF3 11147919 IC50 = 16000 nM T77546 CUL1G2 11171749 IC50 = 16000 nM T77546 CI2ZB6 11182637 IC50 = 160 nM T77546 CV0MO3 11184629 IC50 = 19000 nM T77546 C7QW3P 11229730 IC50 = 18000 nM T77546 C25MKL 11263687 IC50 = 5000 nM T77546 C9OU4R 11321047 IC50 = 500 nM T77546 CQV28Z 11333471 IC50 = 50000 nM T77546 C3AYC4 11366979 IC50 = 300 nM T77546 COU09A 12655267 IC50 > 100000 nM T77546 CY7MI9 14049939 Ki = 2700 nM T77546 C8O4SL 14983630 Ki = 170 nM T77546 CH56AF 20668674 IC50 > 100000 nM T77546 C92KMP 44345335 Ki = 7100 nM T77546 CMBT65 44387943 IC50 > 100000 nM T77546 CO6A3U 44387955 IC50 > 1000000 nM T77546 C3ZRO0 44387981 IC50 = 61 nM T77546 C2YI1D 44387984 IC50 = 2500 nM T77546 CZJY25 44387994 IC50 = 1000 nM T77546 C2H1UN 44387996 IC50 = 10000 nM T77546 CR1LE3 135432900 Ki = 25000 nM T77546 CA07BI 135465901 Ki = 100000 nM T77546 C8V6MP 135547345 Ki = 5500 nM T77546 C5F1QX 136076500 Ki = 8000 nM T77546 D0B8TJ 2354 Ki = 13 nM T42446 D01AJY 2284 IC50 = 35 nM T42446 D01RBR 130021 IC50 = 38000 nM T42446 D0C9XA 119 IC50 = 25 nM T42446 CGV16B 14113 Ki = 177000 nM T42446 CZS7U8 44600 IC50 = 1770 nM T42446 CZY5M2 685622 Ki = 92000 nM T42446 CH8RL0 4332683 EC50 = 1900 nM T42446 C14BFY 5024764 EC50 = 5370 nM T42446 CW9MS8 6604928 EC50 = 741.31 nM T42446 C9GF0X 10130862 IC50 = 200 nM T42446 C7UK5Q 10132408 IC50 = 18 nM T42446 CLH26M 10419163 IC50 = 280 nM T42446 C9WNM3 14362811 IC50 = 920 nM T42446 C87UMH 14362819 IC50 = 780 nM T42446 CD7V6F 14362824 IC50 = 500 nM T42446 C2Z4GX 14362838 IC50 = 880 nM T42446 CAOK62 14362839 IC50 = 39 nM T42446 CW2UL1 14362840 IC50 = 360 nM T42446 C5VUL6 15603270 EC50 = 870.96 nM T42446 CR2ZU8 19889410 IC50 = 21300 nM T42446 C4ZA6P 23757305 IC50 = 4410 nM T42446 CM01WR 44433820 EC50 = 5011.87 nM T42446 C7UL4T 44433825 EC50 = 4570.88 nM T42446 CSV94A 44433826 EC50 = 2754.23 nM T42446 CZE52B 44433827 EC50 = 3467.37 nM T42446 C96QPG 44433828 EC50 = 1659.59 nM T42446 CFY27E 44433830 EC50 = 1659.59 nM T42446 C5XLV4 44433839 EC50 = 1202.26 nM T42446 CUXT14 44433840 EC50 = 2041.74 nM T42446 CH8UR6 44433842 EC50 = 1659.59 nM T42446 CJMS06 53261132 EC50 = 99300 nM T42446 CGRZ23 71532869 EC50 = 61800 nM T42446 CNC39I 71601649 EC50 > 100000 nM T42446 CN28FE 71601650 EC50 > 100000 nM T42446 CXN32Z 71716205 EC50 = 66900 nM T42446 C6QT8A 71716206 EC50 > 100000 nM T42446 C2HRA1 71717438 EC50 > 100000 nM T42446 C3FZ2O 71718024 EC50 = 40000 nM T42446 CE2H4L 71718648 EC50 = 53500 nM T42446 CHS3M1 71718649 EC50 > 100000 nM T42446 C02RHD 71719256 EC50 = 15900 nM T42446 C4B1MD 71720465 EC50 > 100000 nM T42446 C30YRP 71720467 EC50 > 100000 nM T42446 CN5I0R 122184355 EC50 = 8.6 nM T42446 D02ALQ 86279004 IC50 = 37900 nM T42446 D03KZK 5097016 IC50 = 29 nM T42446 D07BIF 6335948 IC50 = 2.4 nM T42446 D08LFC 5230 IC50 = 6.6 nM T42446 D0AK9X 125917 IC50 = 610 nM T42446 D0H5JW 44602 IC50 = 15 nM T42446 D0N4WZ 9898878 IC50 = 1350 nM T42446 D0S5YH 122150 IC50 = 33000 nM T42446 D0U4HM 5521 EC50 = 500000 nM T42446 D0V0LA 10219532 IC50 = 166 nM T86918 C9QEP1 448828 Ki = 1800000 nM T86918 C6UQJ0 448829 Ki = 25000 nM T86918 C34ELK 449164 Ki = 75 nM T86918 CV0WS2 449165 Ki = 12 nM T86918 CM6CA2 23644309 Ki = 12 nM T86918 C4ES6H 44333048 EC50 = 20 nM T86918 CG9SW2 44333049 EC50 = 3 nM T86918 CDU94X 44333078 IC50 = 0.3 nM T86918 C3XJ9W 73345199 IC50 = 8 nM T86918 CCUJ79 73346731 EC50 = 6 nM T86918 CM76NZ 73346732 EC50 = 22 nM T86918 CQ1ME6 73349806 EC50 = 4 nM T86918 CBC73K 73349808 IC50 = 1 nM T86918 C3QUR8 73351326 EC50 = 50 nM T86918 CFG96R 73351327 EC50 = 20 nM T86918 CU0ZM1 73354298 IC50 = 0.5 nM T86918 C9CW1L 78349960 Ki = 1250 nM T86918 C69QTW 122189583 Ki = 14.3 nM T86918 CTK0D4 122189584 Ki = 41.6 nM T86918 C89YLA 122191023 IC50 = 2590 nM T86918 C2LOE8 122191024 Ki = 14.7 nM T86918 CM06HN 122191026 Ki = 8 nM T86918 C9L2FX 122191027 Ki = 3600 nM T86918 C67END 122191028 Ki = 6100 nM T86918 D01FHK 3086453 EC50 = 0.05 nM T86918 D0R2BA 445248 Ki = 18000000 nM T85309 CT08EI 484751 IC50 = 5900 nM T85309 CA6W3C 1396823 IC50 = 170000 nM T85309 C6HNE1 2246840 IC50 = 187000 nM T85309 C8O4KD 5281599 IC50 = 17100 nM T85309 C3ZJ8U 5281609 IC50 = 11500 nM T85309 CQEL68 6055630 IC50 = 108000 nM T85309 C9HJE6 7032560 IC50 = 125000 nM T85309 CSJ73Q 10347674 IC50 = 5500 nM T85309 CP2D3Q 10364369 IC50 = 7400 nM T85309 C3MZ0D 14186891 IC50 = 8100 nM T85309 CJ26AL 21604873 IC50 = 83000 nM T85309 CS56LP 49822436 IC50 = 6200 nM T85309 CO87MN 118729943 IC50 = 87000 nM T85309 C09ING 118729944 IC50 = 136000 nM T85309 CD0L9T 145958807 IC50 = 7800 nM T85309 D01BTV 286 IC50 = 1000 nM T85309 D0I4NN 14056555 IC50 = 156000 nM T85309 D0T3PW 5281672 IC50 = 18800 nM T86385 D00UVA 11556711 IC50 > 30000 nM T86385 D0FT4R 107706 IC50 > 10000 nM T86385 D0SH3I 387447 IC50 = 520 nM T86385 D00LOB 9866964 Ki > 26000 nM T86385 D01YIO 10146470 Ki = 38 nM T86385 D0VO0T 24800541 EC50 = 13.5 nM T86385 D0Y6SQ 2536 IC50 > 100000 nM T86385 D0HM5J 118253852 IC50 > 20000 nM T86385 D0NJ1A 65663 IC50 = 1100 nM T86385 D0WY9H 9892148 Ki = 250 nM T86385 CKO7V4 1701 IC50 = 250000 nM T86385 CP9FG4 99625 IC50 = 24000 nM T86385 CLX4V7 130395 IC50 > 100000 nM T86385 C5Q7EX 160817 IC50 > 60000 nM T86385 CC9E0Y 232547 IC50 = 2100 nM T86385 CN0XJ3 439647 IC50 = 110000 nM T86385 CN67CR 555078 IC50 = 3700 nM T86385 CHF5A4 578663 IC50 = 433200 nM T86385 C05EGK 736344 IC50 > 1000000 nM T86385 CW9DQ2 4476325 IC50 = 4100 nM T86385 CHU41D 5013064 IC50 > 60000 nM T86385 CF9VK2 5236960 IC50 > 139000 nM T86385 CO58XD 5311161 IC50 > 100000 nM T86385 C8OE6S 6913584 IC50 > 100000 nM T86385 CANW64 9798519 IC50 = 700 nM T86385 CMUY79 9800909 IC50 = 52 nM T86385 CD8G1T 9818360 IC50 = 4500 nM T86385 C9NHA3 9821476 IC50 = 1500 nM T86385 C7UKF5 9825353 IC50 > 1000 nM T86385 C3K8PQ 9830518 IC50 = 530 nM T86385 CGNB60 9830581 IC50 = 280 nM T86385 CL61HY 9888442 IC50 > 100000 nM T86385 CG2EZ0 9889108 IC50 < 100000 nM T86385 C5T0GJ 9895523 IC50 = 64 nM T86385 C7KJP3 9908917 IC50 > 100000 nM T86385 CGL12S 9916581 Ki = 1390 nM T86385 CQ84MG 9917430 Ki > 600000 nM T86385 CGT3K4 9932145 IC50 > 100000 nM T86385 CIQX83 9938207 Ki = 379 nM T86385 C2CE1A 9962331 Ki > 2000000 nM T86385 C3HI6E 9972080 IC50 > 100000 nM T86385 C0WT4P 10024711 IC50 = 20000 nM T86385 CVHQ60 10048700 Ki = 130000 nM T86385 C7CW1P 10080504 IC50 = 740 nM T86385 CEN06H 10093642 IC50 > 100000 nM T86385 CD6KX7 10162462 IC50 > 1000 nM T86385 CRP54X 10364794 IC50 = 22000 nM T86385 C9M3VF 10366027 IC50 > 1000 nM T86385 CCQA34 10383086 IC50 > 1000000 nM T86385 C79FQG 10383359 Ki = 400000 nM T86385 CEPM12 10391460 IC50 = 8.4 nM T86385 CCL85B 10394816 IC50 = 1.4 nM T86385 C2UNX1 10407325 IC50 = 3700 nM T86385 CORP79 10431323 IC50 > 100000 nM T86385 C9M7CE 10497407 IC50 = 330 nM T86385 CYC5G6 10497621 IC50 = 220 nM T86385 CJN97A 10499538 IC50 = 1700 nM T86385 C6D3UM 10504812 IC50 = 83000 nM T86385 CA4RW1 10517868 IC50 > 60000 nM T86385 COKF15 10520443 IC50 = 4500 nM T86385 CIMX79 10524714 IC50 = 600 nM T86385 C5LR1J 10527210 IC50 = 4800 nM T86385 C3VQM6 10529952 IC50 = 200 nM T86385 CTN78E 10545533 IC50 = 4200 nM T86385 CCE5M4 10551184 IC50 = 4800 nM T86385 CZL85V 10572734 IC50 > 100000 nM T86385 CVO85L 10577862 IC50 = 440000 nM T86385 C20JKT 10593313 IC50 = 780 nM T86385 CZ8PK9 10599803 IC50 = 2300 nM T86385 C2V4IZ 10616405 IC50 = 100000 nM T86385 C9I3QE 10616695 IC50 = 1500 nM T86385 CS52KZ 10617888 IC50 = 2200 nM T86385 C38SDV 10619385 IC50 = 340 nM T86385 C83JQD 10620089 IC50 = 230 nM T86385 C4K1BD 10620298 IC50 = 6500 nM T86385 C5X0QT 10625780 IC50 = 77 nM T86385 C6V4NJ 10642042 IC50 = 75000 nM T86385 CBHW74 10653967 Ki > 15000 nM T86385 CMXS14 10653995 Ki > 15000 nM T86385 CM57UY 10666214 IC50 = 1900 nM T86385 C8QB4K 10689926 IC50 = 6500 nM T86385 CZ57RO 10697572 IC50 = 6600 nM T86385 C6S2JY 10712874 IC50 = 2500 nM T86385 CFCP28 10714430 IC50 = 640 nM T86385 CP7Y9Z 10714544 IC50 = 4100 nM T86385 CPT0M6 10715096 IC50 = 3900 nM T86385 CE7CB3 10715299 IC50 = 5400 nM T86385 CD0I2U 10736348 IC50 = 8000 nM T86385 CX9JY3 10737216 IC50 = 1000 nM T86385 C06EQF 10739429 IC50 > 100000 nM T86385 CVX58I 10740202 IC50 = 3700 nM T86385 C1TB8N 10764081 IC50 > 100000 nM T86385 C3MH6G 10765640 IC50 = 16000 nM T86385 C4J2AM 10782637 IC50 = 1800 nM T86385 CSO9H0 10811389 IC50 > 100000 nM T86385 CG9B1J 10819798 Ki > 15000 nM T86385 CL85VD 10835279 IC50 = 3300 nM T86385 CX3E7A 10838826 IC50 = 1500 nM T86385 C39NQW 11235804 Ki = 9500 nM T86385 C92PMV 11253808 IC50 = 55000 nM T86385 CLAK97 11540629 IC50 = 16000 nM T86385 C93USP 11626693 IC50 = 2900 nM T86385 C07MTY 11634767 IC50 = 28000 nM T86385 C1ZK9V 11684537 IC50 = 8000 nM T86385 C6RY7J 11725023 IC50 = 80000 nM T86385 CC53TD 12043588 IC50 = 63000 nM T86385 C10ALY 13339657 IC50 = 32000 nM T86385 C2DGN3 14046022 IC50 = 3100 nM T86385 CDP91C 15743471 IC50 > 60000 nM T86385 CJ41CN 15743472 IC50 = 25000 nM T86385 C9OSM6 16144480 Ki > 15000 nM T86385 CDR0G7 16145606 Ki > 15000 nM T86385 CY20PW 16147332 Ki > 15000 nM T86385 CF5Y3L 16147570 Ki > 15000 nM T86385 C7S6IT 16148231 Ki = 1500 nM T86385 C63HAE 18572952 IC50 > 134000 nM T86385 CZPF48 23648277 IC50 > 50000 nM T86385 C1Z9SX 24776379 Ki = 0.15 nM T86385 CN0VA7 24822701 IC50 > 50000 nM T86385 CCG0Z2 25124204 IC50 = 22 nM T86385 CUC8N5 25141405 IC50 > 100000 nM T86385 C3GS6F 33009902 IC50 > 10000 nM T86385 CL0M7R 44143089 IC50 = 147910.84 nM T86385 C8Y9JZ 44284991 Ki = 44.1 nM T86385 CMZ71H 44284992 Ki = 3.74 nM T86385 C5NU9L 44285118 Ki = 14.3 nM T86385 CU9G2F 44285211 Ki = 0.916 nM T86385 C0FPN1 44285253 Ki = 25.3 nM T86385 C9N1ZL 44285281 Ki = 0.187 nM T86385 C5PX3O 44285312 Ki = 0.174 nM T86385 C9LRW8 44285352 Ki = 3.85 nM T86385 CN7SA3 44287645 IC50 = 33000 nM T86385 C1GU7P 44287670 IC50 = 56000 nM T86385 CB8L9Q 44287782 IC50 = 37000 nM T86385 CR6QO0 44287881 IC50 > 60000 nM T86385 CT98XO 44287910 IC50 = 55000 nM T86385 C4KWZ8 44287967 IC50 = 24000 nM T86385 C6KJ4D 44288060 IC50 > 60000 nM T86385 CMO3X2 44288136 IC50 = 28000 nM T86385 C65TOU 44303193 IC50 = 17000 nM T86385 C2DM3E 44303204 IC50 = 12000 nM T86385 C9N4KA 44303215 IC50 = 11000 nM T86385 CE3NJ0 44303216 IC50 = 210000 nM T86385 C3E6HC 44303217 IC50 = 9300 nM T86385 CR68VO 44303218 IC50 = 65000 nM T86385 CR6GO9 44303240 IC50 = 91000 nM T86385 C6YB7J 44303242 IC50 = 25000 nM T86385 CWOM61 44303259 IC50 = 8100 nM T86385 C0C8FX 44303260 IC50 = 23000 nM T86385 CWUI78 44303375 IC50 = 18000 nM T86385 CJ15HX 44303391 IC50 = 58000 nM T86385 CH6TE7 44303392 IC50 = 24000 nM T86385 CVJS18 44303415 IC50 = 25000 nM T86385 C1W6MX 44303477 IC50 = 42000 nM T86385 CSB6M5 44303496 IC50 = 12000 nM T86385 CGNR45 44303533 IC50 = 890000 nM T86385 CTRX10 44303534 IC50 = 130000 nM T86385 C20OYT 44303535 IC50 = 36000 nM T86385 C1Y2QB 44303536 IC50 = 140000 nM T86385 CGP52Y 44303588 IC50 = 35000 nM T86385 CH13CK 44303589 IC50 = 32000 nM T86385 CQ82JC 44303644 IC50 = 30000 nM T86385 CO3V6E 44303657 IC50 = 44000 nM T86385 C5L1DC 44308976 IC50 > 100000 nM T86385 CKN8C1 44316486 IC50 = 230 nM T86385 C2AT7J 44342409 Ki > 15000 nM T86385 CD8AL2 44351097 IC50 = 3600 nM T86385 CHGE39 44351104 IC50 = 67000 nM T86385 CQH2K6 44353359 Ki = 200 nM T86385 C14NKU 44353376 Ki = 1600 nM T86385 CK13HZ 44353387 Ki = 1100 nM T86385 C4OQZ5 44353439 Ki = 200 nM T86385 CDLQ89 44354931 IC50 = 75 nM T86385 CZG9E2 44354934 IC50 = 170 nM T86385 C7NWU8 44354935 IC50 = 1600 nM T86385 C5UJB8 44354936 IC50 = 6.4 nM T86385 CRL78E 44354968 IC50 = 520 nM T86385 CM73HF 44354971 IC50 = 160 nM T86385 CVYF38 44354984 IC50 = 140 nM T86385 CZDW93 44355000 IC50 = 15 nM T86385 CG1VN6 44355001 IC50 = 190 nM T86385 CL04TR 44355071 IC50 = 69 nM T86385 C9U4BR 44355072 IC50 = 48 nM T86385 CI4R1U 44355083 IC50 = 80 nM T86385 CDON50 44355100 IC50 = 21000 nM T86385 C34UGZ 44366594 Ki = 1700 nM T86385 CFL1J0 44366665 Ki > 1000000 nM T86385 C27VSQ 44366666 Ki = 2200 nM T86385 CNE14G 44378491 IC50 = 500 nM T86385 CSV48N 44378519 IC50 = 380 nM T86385 CL9HZ0 44378543 IC50 = 800 nM T86385 CDA68B 44378603 IC50 = 1300 nM T86385 C34YAJ 44378694 IC50 = 1000 nM T86385 C3BX5Y 44412781 Ki > 150000 nM T86385 CIT5G7 44561891 IC50 > 100000 nM T86385 C90BGR 44561892 IC50 > 100000 nM T86385 C9RGX4 44561893 IC50 > 100000 nM T86385 CU7NP5 44561930 IC50 > 100000 nM T86385 CV21IQ 44561931 IC50 > 100000 nM T86385 CR08WA 44561932 IC50 > 100000 nM T86385 C2PVE0 45103523 Ki > 26000 nM T86385 CGN14R 45103723 Ki > 26000 nM T86385 CD4T1L 46221636 IC50 = 120000 nM T86385 CUI91D 46905615 IC50 = 1200 nM T86385 CJH50R 49797481 IC50 > 100000 nM T86385 CI7P2B 49797571 IC50 = 90 nM T86385 CI59MV 49797572 IC50 > 50000 nM T86385 C96CKU 49797573 IC50 = 150 nM T86385 CEC3R4 52943167 IC50 = 100 nM T86385 C5H3GD 52943168 IC50 = 200 nM T86385 C4WVX9 52943169 IC50 = 200 nM T86385 C8AR2B 52946468 IC50 = 100 nM T86385 CZ3FS0 52949270 IC50 = 150 nM T86385 CO6F3U 53249965 IC50 = 1400 nM T86385 CBJQ98 54132077 IC50 = 53000 nM T86385 CY3IO1 56659828 IC50 > 10 nM T86385 CI2AB4 56663296 IC50 > 10 nM T86385 CT2G3R 56666720 IC50 = 2.1 nM T86385 CQH46K 56666721 IC50 > 10 nM T86385 C3V0AU 56666722 IC50 > 10 nM T86385 CZ3O2H 56670144 IC50 > 10 nM T86385 CNL70Y 56670149 IC50 = 7 nM T86385 C0HJL7 56673658 IC50 = 4.8 nM T86385 CP5B7A 56673659 IC50 = 8.8 nM T86385 CE58OY 56673664 IC50 > 10 nM T86385 C9F5UR 56676983 IC50 > 10 nM T86385 CL9XA8 56680306 IC50 > 10 nM T86385 CHNX69 56680307 IC50 > 10 nM T86385 CP3IV1 56680314 IC50 > 10 nM T86385 CSF9P8 56683631 IC50 > 10 nM T86385 CD57KP 56683632 IC50 > 10 nM T86385 CP1MR2 56683633 IC50 > 10 nM T86385 CG7O3N 56683634 IC50 = 9.5 nM T86385 CL16UQ 56949326 IC50 < 10000 nM T86385 C0UIF5 57671050 IC50 = 7800 nM T86385 CY26NE 57671116 IC50 > 10000 nM T86385 C9E6CB 57671131 IC50 > 10000 nM T86385 CJO75X 57671161 IC50 = 8500 nM T86385 CF2Q3E 59497392 IC50 > 10000 nM T86385 C2W3AK 59497404 IC50 > 10000 nM T86385 C0E1KN 59497528 IC50 = 5400 nM T86385 CAWN80 59497611 IC50 > 10000 nM T86385 CSQY41 59497643 IC50 > 10000 nM T86385 C31NTK 59497690 IC50 > 10000 nM T86385 C48UHX 66561877 IC50 = 369000 nM T86385 C50MEH 71682307 IC50 > 10000 nM T86385 CO8PQ5 71682308 IC50 = 3800 nM T86385 C78DJQ 71711730 IC50 < 10000 nM T86385 CL23VT 71723878 IC50 = 16000 nM T86385 C1MBU7 72793747 IC50 > 100000 nM T86385 C6BY5D 72793776 IC50 > 100000 nM T86385 C1DI8A 72793778 IC50 = 19000 nM T86385 C5U9CI 73355715 Ki = 0.437 nM T86385 CFPT98 90655054 IC50 > 30000 nM T86385 C5JZ8R 90655055 IC50 > 30000 nM T86385 C8E4WS 102323332 IC50 > 50000 nM T86385 CR2AU7 118010068 IC50 > 10000 nM T86385 COA36C 118010069 IC50 > 10000 nM T86385 C5NJH1 118202505 IC50 > 10000 nM T86385 C43ADS 118202506 IC50 > 10000 nM T86385 C2UXT7 118202507 IC50 > 10000 nM T86385 CPV27G 118202509 IC50 > 10000 nM T86385 CJB3K7 118202510 IC50 > 10000 nM T86385 C12BHL 118202511 IC50 > 10000 nM T86385 COT6H0 118202512 IC50 > 10000 nM T86385 C0GRU4 118718129 Ki = 3.9 nM T86385 C8ZSC2 118727248 IC50 > 10000 nM T86385 CYIX41 118727249 IC50 > 10000 nM T86385 CH1T3M 118727250 IC50 > 10000 nM T86385 CVG1X5 118727251 IC50 > 10000 nM T86385 C9B6KX 118727252 IC50 > 10000 nM T86385 C3OUW6 118727253 IC50 > 10000 nM T86385 C10QJC 118727254 IC50 > 10000 nM T86385 CVIF56 118727255 IC50 > 10000 nM T86385 CNQ9U4 118727256 IC50 > 10000 nM T86385 CN93WU 118727257 IC50 > 10000 nM T86385 C5DR7Z 118727258 IC50 > 10000 nM T86385 CDEU05 118727259 IC50 > 10000 nM T86385 CZHT12 118727260 IC50 > 10000 nM T86385 CD21PC 118731187 IC50 = 6000 nM T86385 CGV2Y0 122192762 Ki = 12 nM T86385 C6RDX4 122192767 Ki = 490 nM T86385 C9QKI3 127020966 IC50 > 100000 nM T86385 CNL2Z9 137635679 Ki = 0.89 nM T86385 CDQ62V 137637214 Ki > 50000 nM T86385 C2K8JV 137639385 Ki > 50000 nM T86385 CNO8Y2 137639848 Ki = 3.4 nM T86385 CCF5A0 137640149 Ki = 4.8 nM T86385 CZ95CD 137642316 Ki = 62 nM T86385 CF0TK8 137642520 Ki = 7.3 nM T86385 C8WS7U 137646736 Ki = 390 nM T86385 CCQ4H7 137647098 Ki = 1200 nM T86385 C03IMN 137647139 Ki = 1.7 nM T86385 C71MRD 137649122 Ki = 160 nM T86385 C2D6KY 137650380 Ki = 410 nM T86385 CYGV01 137650976 Ki = 1.1 nM T86385 COR29F 137652632 Ki = 480 nM T86385 CNX46H 137654508 Ki > 50000 nM T86385 CZ1H4R 137655362 Ki = 1.6 nM T86385 CQAV71 137657536 Ki = 12 nM T86385 CD25CQ 137657864 Ki = 530 nM T86385 CTUM82 137658421 IC50 = 1100 nM T86385 CIGV31 137660044 Ki = 630 nM T86385 C1S2LC 137660418 Ki = 3000 nM T86385 CX5S3Y 137661570 Ki = 4.9 nM T86385 CE7GI1 137662261 Ki = 2.9 nM T86385 CYT20V 155514020 Ki = 29000 nM T86385 CW1B5Z 155521967 Ki < 0.1 nM T86385 CBU5W0 155524880 IC50 > 10000 nM T86385 C4QT3M 155526246 Ki = 54 nM T86385 C2X5EJ 155531124 Ki = 160 nM T86385 CPC60R 155533917 Ki = 7.4 nM T86385 CM06WG 155535720 Ki = 38 nM T86385 CU9FL4 155551858 Ki = 13000 nM T86385 C2E5GR 155554478 IC50 > 10000 nM T86385 CE3G5W 155556110 Ki = 1200 nM T86385 C0SND3 155557259 Ki = 5200 nM T86385 CTS63Q 155558248 Ki = 150 nM T86385 CFX07G 155558369 IC50 > 5000 nM T86385 C5R4VY 155566937 Ki = 8.2 nM T86385 CP4F1U 155567613 Ki = 7800 nM T86385 CU42CE 155567829 IC50 > 100000 nM T86385 CO8GJ3 155568502 Ki = 14 nM T86385 CU62EW 155568945 Ki = 0.26 nM T86385 D02AVL 18376720 Ki > 5000 nM T86385 D02PAU 16731825 Ki > 10000 nM T86385 D05ICF 3492365 IC50 = 2.3 nM T86385 D08QZD 9829503 Ki = 720 nM T86385 D0C1NP 66561876 IC50 = 14200 nM T86385 D0E9EH 44353386 Ki > 800000 nM T86385 D0F2YC 10038543 IC50 = 0.39 nM T86385 D0F3CA 1609 IC50 = 93000 nM T86385 D0R9CH 3400921 Ki > 10000 nM T09185 D00STL 644241 IC50 < 100 nM T09185 D0AZ3C 5291 IC50 = 43 nM T09185 D0E6XR 3062316 IC50 = 0.5 nM T09185 D0E3TC 44259 IC50 = 4.28 nM T09185 D0D5PL 71577234 IC50 = 164 nM T09185 D0LL1P 71768628 IC50 = 97 nM T09185 CL14BG 4426513 IC50 > 100000 nM T09185 CA3I4T 24753787 IC50 > 50000 nM T09185 CJ0CU5 24825841 IC50 = 2.4 nM T09185 C4FZ8E 24875320 IC50 = 4.799 nM T09185 C3VRO9 44557921 IC50 > 10000 nM T09185 CF57GK 46215462 IC50 = 20 nM T09185 C2VAX9 51035420 IC50 = 68 nM T09185 CPHX64 57325478 IC50 > 50000 nM T09185 CQ9BW4 57325479 IC50 > 50000 nM T09185 CVK0G4 58056356 IC50 > 50000 nM T09185 C7SGT6 60202316 IC50 = 39 nM T09185 CV63UL 67240318 IC50 > 10000 nM T09185 CB61ZO 67347910 IC50 = 9 nM T09185 CRH2Y9 68639605 IC50 = 8.93 nM T09185 C1IT5U 71550931 IC50 = 6.8 nM T09185 CG1I5B 71550932 IC50 = 7.02 nM T09185 C1F5NV 71624671 IC50 = 39.63 nM T09185 CQE01I 71624672 IC50 = 65.14 nM T09185 CV8XI0 71624673 IC50 > 1000 nM T09185 CY82NR 71624674 IC50 = 29.15 nM T09185 C0IM7Z 71624675 IC50 = 39.82 nM T09185 C6JS8P 71624676 IC50 = 38.9 nM T09185 C2F0QN 71624677 IC50 > 1000 nM T09185 CQ75IY 71624788 IC50 = 5.96 nM T09185 C6GT1Q 71624789 IC50 = 47.75 nM T09185 C6ZYR9 71624790 IC50 > 1000 nM T09185 CCSI30 71624792 IC50 > 1000 nM T09185 C4JD7I 71624793 IC50 = 470 nM T09185 CS0AQ6 71624904 IC50 = 4.04 nM T09185 C23XIU 71624905 IC50 = 22.36 nM T09185 C4KTH9 71624906 IC50 = 16.64 nM T09185 C7BG9F 71624907 IC50 = 19.75 nM T09185 CC61DF 71624908 IC50 = 6.14 nM T09185 CRLN56 71624909 IC50 > 1000 nM T09185 CLO8V2 71625035 IC50 = 35.02 nM T09185 CQI0N1 71625036 IC50 = 9.72 nM T09185 CO41GB 71625037 IC50 = 19.03 nM T09185 CC68IJ 71625038 IC50 = 386.5 nM T09185 C4SV3X 71625039 IC50 = 324.1 nM T09185 CT2K6M 71625040 IC50 = 6.34 nM T09185 C6JZ2E 71625161 IC50 = 29.81 nM T09185 CRGQ64 71625290 IC50 = 6.71 nM T09185 CP83JY 71625291 IC50 = 13.94 nM T09185 CGJ8H4 71625292 IC50 = 13.3 nM T09185 C0D4LN 71625406 IC50 = 17.49 nM T09185 C9B1RV 71625407 IC50 = 37.58 nM T09185 CKOL80 71625408 IC50 = 12.47 nM T09185 CQY4U2 71625409 IC50 = 10.05 nM T09185 C42VJY 71764060 IC50 = 235 nM T09185 CEH2B7 72836888 IC50 = 86 nM T09185 C9IZF3 86763814 IC50 = 1500 nM T09185 CR9V4A 86763924 IC50 = 6 nM T09185 C6F5PQ 119081684 IC50 = 309 nM T09185 CN4X0C 121231414 IC50 = 9.4 nM T09185 C81IFQ 122163152 IC50 = 2110 nM T09185 C49UGP 122187122 IC50 = 150 nM T09185 CQL0W7 122197565 IC50 = 75.7 nM T09185 C6UY2L 122633880 IC50 = 212 nM T09185 CC7P2W 122633900 IC50 = 265 nM T09185 CN41IF 122634050 IC50 = 292 nM T09185 CBYC49 126617676 IC50 = 22.2 nM T09185 CC58IQ 127043948 IC50 = 126 nM T09185 CVF8Z9 127045862 IC50 = 4.7 nM T09185 CH68NT 127046076 IC50 = 137 nM T09185 CF5D2Y 129318936 IC50 = 2462 nM T09185 C6RPF1 130364436 IC50 = 191 nM T09185 CSY34O 130364443 IC50 = 254 nM T09185 CI9H2W 130364450 IC50 = 24.3 nM T09185 CM4TO5 130364451 IC50 = 38.3 nM T09185 C28CLN 130364457 IC50 = 328 nM T09185 CV4DH7 130364460 IC50 = 80.7 nM T09185 CW91ZV 130364461 IC50 = 223 nM T09185 CQIZ43 130364463 IC50 = 89 nM T09185 C4IKC6 130364464 IC50 = 123 nM T09185 C0X6JS 130364465 IC50 = 79.9 nM T09185 C0ZGC1 130364467 IC50 = 71.1 nM T09185 CO9C5Q 130364468 IC50 = 442 nM T09185 CQW3P1 130364471 IC50 = 50.5 nM T09185 CHWX05 130364473 IC50 = 49.9 nM T09185 CLB65Y 130364478 IC50 = 66.6 nM T09185 CUZG19 130364481 IC50 = 614 nM T09185 C34OMJ 130364482 IC50 = 209 nM T09185 C6TWR3 130364484 IC50 = 132 nM T09185 C8SF5Q 130364488 IC50 = 19.9 nM T09185 CS5C4E 130364494 IC50 = 222 nM T09185 CVQ32Y 130364503 IC50 = 25.6 nM T09185 CV8B0Y 130364506 IC50 = 545 nM T09185 CHX23J 130364524 IC50 = 44.6 nM T09185 CHYL89 130364535 IC50 = 167 nM T09185 C6OMB1 132204257 IC50 = 63 nM T09185 C6ROQ3 132546210 IC50 = 116 nM T09185 CQR94G 134198433 IC50 = 193 nM T09185 C1X6FJ 134693894 IC50 = 9.4 nM T09185 CXC69T 137321158 IC50 = 35 nM T09185 CWC49K 137321210 IC50 = 5.6 nM T09185 CI1E8V 137634241 IC50 > 10000 nM T09185 C5VE4K 137636547 IC50 = 167 nM T09185 CZ05TY 137637593 IC50 = 10000 nM T09185 CU9YQ3 137637635 IC50 = 5020 nM T09185 C6PKY7 137645383 IC50 > 10000 nM T09185 CHR9E0 137651685 IC50 = 13.1 nM T09185 CY53VO 137651787 IC50 > 10000 nM T09185 CE8DW7 137658399 IC50 > 10000 nM T09185 CU61WM 137658936 IC50 > 10000 nM T09185 CY9N8Q 137662234 IC50 = 6.6 nM T09185 C3K5LU 137796291 IC50 = 326 nM T09185 CM3A8O 139030333 IC50 = 3000 nM T09185 C6AK0N 139030518 IC50 = 135 nM T09185 CB69CL 145925694 IC50 = 0.7078 nM T09185 C7SH9V 145949579 IC50 = 3.2 nM T09185 CQCV54 145950906 IC50 = 151 nM T09185 CKWZ34 145950923 IC50 = 6.2 nM T09185 CGOE73 145951398 IC50 = 11.4 nM T09185 CZF70O 145951916 IC50 = 5 nM T09185 CNK12Z 145952731 IC50 = 12.5 nM T09185 CGV16H 145954003 IC50 = 1200 nM T09185 CUIT87 145955254 IC50 = 7.9 nM T09185 CX2U6N 145956375 IC50 = 16 nM T09185 CC0RU9 145956925 IC50 = 614 nM T09185 CA2F0O 145958559 IC50 = 3.9 nM T09185 C12VOP 145959821 IC50 = 380 nM T09185 C5PZ9J 145959874 IC50 = 8.4 nM T09185 CF0C6K 145960274 IC50 = 3.9 nM T09185 CQE9M5 145966810 IC50 = 100 nM T09185 CWJ12M 145969155 IC50 = 35 nM T09185 C8NDS6 145971939 IC50 = 12.6 nM T09185 CP9NB6 145974090 IC50 = 695 nM T09185 CI85EU 145998085 IC50 = 14.9 nM T09185 CD49VM 155295006 IC50 = 23.8 nM T09185 CSHC63 155510467 IC50 = 359.5 nM T09185 C5MP1Q 155510890 IC50 = 36.4 nM T09185 CG09WO 155512858 IC50 = 55.6 nM T09185 C6H8ZU 155513172 IC50 = 10.4 nM T09185 CZDH58 155514096 IC50 = 36.5 nM T09185 CDU75B 155514157 IC50 = 3.97 nM T09185 CB5T9G 155515436 IC50 = 15.5 nM T09185 CUHZ87 155516883 IC50 = 723.1 nM T09185 C84GJO 155517474 IC50 = 21.3 nM T09185 C63PZX 155518871 IC50 = 42.3 nM T09185 CT0V6H 155519724 IC50 = 10.5 nM T09185 CNP8T7 155530083 IC50 = 9.2 nM T09185 CK10UA 155531677 IC50 = 16.5 nM T09185 CS69CA 155532132 IC50 = 3 nM T09185 CURO30 155532620 IC50 = 5.89 nM T09185 C3PWI1 155534046 IC50 > 1000 nM T09185 CWLZ25 155535008 IC50 = 107.8 nM T09185 CTXK93 155535665 IC50 = 14.4 nM T09185 C14SEB 155535950 IC50 = 42.5 nM T09185 C8NA6L 155536370 IC50 = 8.7 nM T09185 CPG5T4 155538560 IC50 > 3000 nM T09185 C3O6WX 155540330 IC50 > 1000 nM T09185 CXG71B 155540768 IC50 = 36.4 nM T09185 C3Q9UA 155541932 IC50 = 1260 nM T09185 C76NKG 155543431 IC50 = 68.7 nM T09185 CC9LQ2 155546287 IC50 = 13000 nM T09185 CI27QV 155546853 IC50 = 4879 nM T09185 CYP2O5 155547984 IC50 = 63.7 nM T09185 C9MJL5 155551408 IC50 = 14.7 nM T09185 C14QWH 155551649 IC50 > 3000 nM T09185 CL8KR2 155552517 IC50 = 357.1 nM T09185 CA9Y3J 155552522 IC50 = 8.53 nM T09185 C1TA9J 155553503 IC50 = 73.8 nM T09185 C8BAU3 155554243 IC50 = 92 nM T09185 CCQF25 155555943 IC50 = 22.5 nM T09185 C7N1AT 155560186 IC50 > 2000 nM T09185 CYD1C7 155560599 IC50 > 1000 nM T09185 C2EDK1 155562180 IC50 = 15.2 nM T09185 C2QC5F 155562643 IC50 > 1000 nM T09185 CHLY93 155562871 IC50 = 30.3 nM T09185 CBG9Z1 155562952 IC50 = 150.5 nM T09185 C0WZ9S 155563842 IC50 > 1000 nM T09185 C60KLJ 155564326 IC50 = 1296 nM T09185 C4BS6J 155565938 IC50 = 15.6 nM T09185 CINX89 155566065 IC50 = 4850 nM T09185 C7Q4RY 155566792 IC50 = 30.1 nM T09185 C0V7SM 155567015 IC50 = 638.9 nM T09185 CP69SU 155567937 IC50 = 66.9 nM T09185 D0BL0O 71624791 IC50 = 2.29 nM T30803 D00ENY 33032 Ki = 42700 nM T30803 D01OXI 2578 IC50 = 8100 nM T30803 D03GET 4055 Ki = 12100 nM T30803 D04OSE 4485 Ki = 17400 nM T30803 D0K8KX 5280343 IC50 = 218000 nM T30803 D0V4GY 9552079 Ki = 192000 nM T30803 C52MFS 1756 IC50 > 50000 nM T30803 CBF49Z 7416 Ki = 274100 nM T30803 CT48KR 21025 IC50 = 79300 nM T30803 CRT9K5 128254 IC50 < 1000 nM T30803 CCZ04P 214232 IC50 = 105000 nM T30803 C8MEI0 223143 IC50 = 20300 nM T30803 CB1K8N 363243 IC50 = 5000 nM T30803 CUF5O9 390735 IC50 > 50000 nM T30803 CJKN12 432139 IC50 = 64800 nM T30803 CN1TR3 580286 IC50 > 173000 nM T30803 C39UQA 723918 IC50 > 212000 nM T30803 CTX3F0 831028 IC50 > 157000 nM T30803 C2ZL6W 877340 IC50 = 86300 nM T30803 CV0S1M 877450 IC50 = 58000 nM T30803 C4L7CX 1550330 IC50 > 100000 nM T30803 C39ODA 1550696 IC50 > 100000 nM T30803 CD4IA9 1712537 IC50 > 155000 nM T30803 CK1N3W 2223018 IC50 > 135000 nM T30803 C2O8ZG 2288440 IC50 = 24900 nM T30803 C4VJW9 2724179 Ki = 211 nM T30803 C1ESQ4 2862129 IC50 > 100000 nM T30803 C49TLS 2881754 IC50 > 100000 nM T30803 C07WHI 4362773 IC50 > 100000 nM T30803 CSZU71 4448737 IC50 = 20400 nM T30803 CHW3L7 5291033 IC50 > 100000 nM T30803 C9ZG4E 5325382 IC50 > 50000 nM T30803 C8VZ9T 5325386 IC50 > 50000 nM T30803 C1BM9S 5377539 IC50 > 100000 nM T30803 C0MPR9 5387357 IC50 > 100000 nM T30803 CZT90E 5802828 IC50 > 100000 nM T30803 CW0E3Y 5925463 IC50 > 100000 nM T30803 C4VK5N 6382486 IC50 > 100000 nM T30803 CC92GK 6445552 IC50 > 100000 nM T30803 C3MX1J 9979274 IC50 = 20000 nM T30803 C6XJT3 10026610 IC50 = 40000 nM T30803 CR95VY 10072380 IC50 = 44700 nM T30803 C35RWB 10253825 IC50 = 55800 nM T30803 CKJO89 10317614 IC50 = 3500 nM T30803 CB2D6A 10319412 IC50 = 18000 nM T30803 C4US6F 10387232 IC50 = 14000 nM T30803 CRYV80 10429818 IC50 = 2500 nM T30803 C8T6XZ 10475024 IC50 = 12000 nM T30803 CI2B1P 10489510 IC50 = 12300 nM T30803 CAJ5W4 10791392 Ki = 2000000 nM T30803 CD8WK2 10847727 IC50 = 18900 nM T30803 C9NC5T 10964817 IC50 = 21000 nM T30803 CI2T6R 11595259 IC50 = 4.1 nM T30803 CK2Y6S 11798906 Ki = 2200000 nM T30803 CG1CU7 12219475 IC50 > 50000 nM T30803 C4EUP9 12247627 IC50 = 2000 nM T30803 CLK87P 13989170 IC50 = 2000 nM T30803 C62BRX 14016406 IC50 < 1000 nM T30803 CJ4OE6 14860354 IC50 = 1000 nM T30803 CROS94 15192338 IC50 = 1000 nM T30803 CY32OJ 15192339 IC50 = 3500 nM T30803 CGH65T 15192340 IC50 = 7000 nM T30803 CY3HI1 15192341 IC50 = 8000 nM T30803 CUHY70 15192342 IC50 = 100000 nM T30803 CHX2S0 15192343 IC50 = 25000 nM T30803 CL21QK 15192344 IC50 = 3000 nM T30803 C3F6KS 15192393 IC50 = 8000 nM T30803 C1TS7N 15192395 IC50 = 1000 nM T30803 CD0CS6 15605637 IC50 > 100000 nM T30803 C1V6AR 16047174 IC50 > 100000 nM T30803 C1NQ6R 16047175 IC50 > 100000 nM T30803 C5FS1M 16047278 IC50 > 100000 nM T30803 CYT94W 16047279 IC50 > 100000 nM T30803 CB78XP 16047280 IC50 > 100000 nM T30803 CPF60C 16047281 IC50 > 100000 nM T30803 CRW35E 16047388 IC50 > 100000 nM T30803 CK8J4C 16047389 IC50 > 100000 nM T30803 C4G2DK 16048003 IC50 > 100000 nM T30803 CTLC91 16193441 IC50 > 100000 nM T30803 CZ0QS6 25269037 IC50 > 50000 nM T30803 CKM60R 25269039 IC50 > 50000 nM T30803 C1X6ZW 25269388 IC50 = 35700 nM T30803 C7ST8I 25269389 IC50 > 50000 nM T30803 C2R4CZ 25269392 IC50 > 50000 nM T30803 C97JED 25269394 IC50 > 50000 nM T30803 CH2G5I 25269395 IC50 > 50000 nM T30803 CSV31T 25269732 IC50 = 45300 nM T30803 CAO45X 25269733 IC50 > 50000 nM T30803 C6XZ7O 25269736 IC50 > 50000 nM T30803 CQ5HC3 25269737 IC50 > 50000 nM T30803 C0NL9Y 25269738 IC50 > 50000 nM T30803 C6GAR8 25269740 IC50 > 50000 nM T30803 C57MBW 25270069 IC50 > 50000 nM T30803 CN72TR 40727263 Ki = 4570 nM T30803 CCBD40 44285823 IC50 = 4000 nM T30803 CI1AD7 44286066 IC50 < 1000 nM T30803 C4U5AV 44315802 Ki > 10000000 nM T30803 CK6F2H 44322851 IC50 = 17100 nM T30803 CF9YK8 44322860 IC50 = 27200 nM T30803 CMDE38 44323177 IC50 = 13900 nM T30803 CGO0X7 44323190 IC50 = 27200 nM T30803 C2B6VO 44323235 IC50 = 9900 nM T30803 C0E4HP 44411997 IC50 > 100000 nM T30803 C7V0IZ 44412016 IC50 > 100000 nM T30803 CZ50GV 44412091 IC50 > 100000 nM T30803 CCY74J 44412123 IC50 > 100000 nM T30803 CUER27 44511333 IC50 = 6810 nM T30803 CUQB41 45266944 IC50 = 29000 nM T30803 CLGA48 45267883 IC50 = 8710 nM T30803 C3VB9U 45268767 IC50 = 23000 nM T30803 CZ3J1P 45269616 IC50 = 8100 nM T30803 CPN74S 45272169 IC50 = 10300 nM T30803 C65XIU 45273032 IC50 = 7170 nM T30803 CZ7DW4 45484008 IC50 > 50000 nM T30803 C5MB8F 46845029 IC50 = 7130 nM T30803 C60IQZ 46888469 IC50 = 11000 nM T30803 CR3Z7V 56678909 Ki = 4160 nM T30803 C83FRX 76313868 IC50 > 100000 nM T30803 C38MOW 76313869 IC50 > 100000 nM T30803 C8KR6Q 76317389 IC50 = 228000 nM T30803 C27QEH 76321111 IC50 > 100000 nM T30803 C6FC4Q 76328308 IC50 > 100000 nM T30803 C7FVU3 76331990 IC50 > 100000 nM T30803 CCX4Q3 76335573 IC50 > 100000 nM T30803 CL73RB 76335574 IC50 > 100000 nM T30803 C3B4VU 135426515 IC50 = 26700 nM T30803 C2APM1 135453064 IC50 = 7600 nM T30803 C0DGX1 135921472 IC50 > 50000 nM T30803 D03MJM 45273020 IC50 = 16000 nM T30803 D03YVX 6018993 IC50 > 100000 nM T30803 D05ABT 10352496 IC50 = 35200 nM T30803 D05CCT 4139 IC50 = 16000 nM T30803 D07TMZ 5962 Ki = 54600 nM T30803 D0A1CM 5281855 IC50 = 22800 nM T30803 D0I8HK 11665560 IC50 = 5000 nM T30803 D0L1AV 45273021 IC50 = 14200 nM T30803 D0O2DQ 237 IC50 > 1000000 nM T84703 D03ZBT 11626560 IC50 = 2 nM T84703 D04LVK 57379345 IC50 = 1829 nM T84703 D07TOK 46188928 IC50 = 5.21 nM T84703 D0AF6O 71731823 Ki = 23 nM T84703 D0OB0F 5328940 IC50 = 27 nM T84703 D00DRL 44137946 IC50 = 61 nM T84703 D01HKZ 57345941 IC50 < 3 nM T84703 D02QWY 24785538 IC50 = 4 nM T84703 D03LWG 53235510 IC50 = 3139 nM T84703 D0E3TC 44259 IC50 = 0.96 nM T84703 D0FA6S 54576299 IC50 = 4.6 nM T84703 D0FD6D 11751922 IC50 = 5 nM T84703 D0O0LS 25141092 IC50 = 3 nM T84703 D0O6WV 24794418 IC50 = 190 nM T84703 D0WS1V 448991 IC50 = 11 nM T84703 D0T3ME 156422 IC50 = 50 nM T84703 CU9J0H 2125863 IC50 = 20000 nM T84703 CY9D7W 2517470 IC50 = 20000 nM T84703 CVL95J 2535914 IC50 = 20000 nM T84703 CJ59NC 2541025 IC50 = 20000 nM T84703 C7UN1Z 2597009 IC50 = 20000 nM T84703 CF89XO 2597103 IC50 = 20000 nM T84703 CXVB08 3399504 IC50 = 20000 nM T84703 CJ3Q5R 3666186 IC50 > 10000 nM T84703 CJM9Q8 4410298 IC50 = 20000 nM T84703 CV1PK6 4798875 IC50 = 20000 nM T84703 CJU3B9 4798877 IC50 = 10461.4 nM T84703 C5AW4U 4802531 IC50 = 20000 nM T84703 CR1HA0 4802711 IC50 = 20000 nM T84703 C1DW3F 5019229 IC50 = 20000 nM T84703 CPZY43 5121984 IC50 > 50000 nM T84703 C7WO8K 7190453 IC50 = 20000 nM T84703 CDB7F4 10321590 IC50 = 646 nM T84703 CBOP58 11293798 Ki > 10000 nM T84703 C26BZX 11362471 Ki > 10000 nM T84703 CWXB93 11397177 Ki > 10000 nM T84703 CTG83F 11539329 Ki > 4500 nM T84703 CMIL86 11590363 Ki > 4500 nM T84703 C4U7HM 11621097 IC50 = 14 nM T84703 C9T6SC 11640926 Ki > 4500 nM T84703 C0AVC3 12751666 EC50 = 87.2 nM T84703 CFPW41 16007116 Ki > 4500 nM T84703 CC5J0U 16112865 IC50 = 1 nM T84703 C5VPH9 16129448 IC50 = 126 nM T84703 CFC39H 16265338 IC50 = 20000 nM T84703 C9NV2A 16272977 IC50 = 20000 nM T84703 C81LCV 16276659 IC50 = 47.1 nM T84703 C1ATH6 16322912 IC50 = 20000 nM T84703 C2HVS1 16739794 IC50 < 1 nM T84703 C03EXR 16739855 IC50 = 1 nM T84703 CW64AB 16739883 IC50 = 1 nM T84703 CD7B6L 17561456 IC50 = 20000 nM T84703 CE1TZ9 20971557 IC50 = 20000 nM T84703 CQHK69 23646624 IC50 = 160 nM T84703 CJ0CU5 24825841 IC50 = 9.37 nM T84703 CY8L7E 24896769 IC50 > 10000 nM T84703 C0KMW8 24937716 IC50 = 13 nM T84703 C5WG1H 24937847 IC50 = 11 nM T84703 C8CO4B 24971342 IC50 = 1100 nM T84703 C3DI7Y 24995523 IC50 = 5 nM T84703 C76PSW 44518384 IC50 = 50 nM T84703 C6LP9V 44518674 IC50 = 47 nM T84703 C36KYB 44520611 IC50 = 29 nM T84703 CZH80Q 44520612 IC50 = 1970 nM T84703 CY3HW5 46224684 IC50 > 10000 nM T84703 CBI7V6 46382265 IC50 = 20000 nM T84703 CMP5T4 46382269 IC50 = 20000 nM T84703 CRP7H0 46382271 IC50 = 5460.3 nM T84703 CT5ZD0 46382272 IC50 = 9064.5 nM T84703 COB29T 46382277 IC50 = 20000 nM T84703 C7TY0M 46382278 IC50 = 20000 nM T84703 CUCX57 46382281 IC50 = 20000 nM T84703 CGR3T6 46382286 IC50 = 20000 nM T84703 CPZ81K 46382288 IC50 = 20000 nM T84703 CU9IK7 46382290 IC50 = 20000 nM T84703 C61WCT 46382295 IC50 = 20000 nM T84703 C4P1AT 46382302 IC50 = 3224.9 nM T84703 CMDC48 46382303 IC50 = 20000 nM T84703 C2ZA3E 46382304 IC50 = 1196.8 nM T84703 CN5R0P 46382305 IC50 = 20000 nM T84703 CH53ZD 46382308 IC50 = 20000 nM T84703 CT3UO5 46382309 IC50 = 20000 nM T84703 C3R5DF 46382310 IC50 = 20000 nM T84703 CVP36M 46382311 IC50 = 20000 nM T84703 CEP0C1 46382312 IC50 = 20000 nM T84703 CUG2W7 46382314 IC50 = 423.2 nM T84703 CDOR02 46382315 IC50 = 2594.4 nM T84703 CG6D4E 46382317 IC50 = 2843.4 nM T84703 C2L3WY 46382318 IC50 = 20000 nM T84703 CPA41J 46382319 IC50 = 20000 nM T84703 C54EDX 46382322 IC50 = 20000 nM T84703 C9J1CQ 46382323 IC50 = 20000 nM T84703 C37VDC 46382324 IC50 = 778 nM T84703 CG13SB 46382326 IC50 = 20000 nM T84703 CD3QY0 46382327 IC50 = 20000 nM T84703 C6ZNO1 46382331 IC50 = 20000 nM T84703 CE6N3J 46382332 IC50 = 20000 nM T84703 COD4I0 46382336 IC50 = 20000 nM T84703 CGD5Q0 46382338 IC50 = 20000 nM T84703 C40NSR 46382339 IC50 = 20000 nM T84703 C8H2CR 46382341 IC50 = 20000 nM T84703 C64RBV 46382343 IC50 = 20000 nM T84703 C6NS1L 46382344 IC50 = 20000 nM T84703 CP23VF 46382346 IC50 = 20000 nM T84703 CP9W3T 46382349 IC50 = 20000 nM T84703 CZNH36 46382354 IC50 = 3886.6 nM T84703 CYH93R 46382355 IC50 = 3575.6 nM T84703 CV51XI 46382356 IC50 = 20000 nM T84703 C7SKH2 46382366 IC50 = 20000 nM T84703 CJD49N 46382375 IC50 = 20000 nM T84703 CJ8E1N 46382394 IC50 = 20000 nM T84703 CW4EI1 46390524 IC50 = 20000 nM T84703 CQG51S 46390527 IC50 = 20000 nM T84703 CZ49OG 46390528 IC50 = 20000 nM T84703 CSJ20W 46390529 IC50 = 10000 nM T84703 CRAK47 46390532 IC50 = 20000 nM T84703 CLS29B 46872626 IC50 > 10000 nM T84703 C2O8RZ 46886323 IC50 > 1000 nM T84703 C1NKE3 46905987 IC50 > 3000 nM T84703 C8KT1S 50802118 IC50 = 20000 nM T84703 C2X9OA 50802180 IC50 = 20000 nM T84703 CF57GW 50802181 IC50 = 2138.5 nM T84703 C1ED3N 50802184 IC50 = 10000 nM T84703 C6G1LV 50802187 IC50 = 20000 nM T84703 CC3YE6 50802196 IC50 = 10000 nM T84703 CBF28N 50802197 IC50 = 20000 nM T84703 CK6G9M 50802198 IC50 = 771 nM T84703 CIC1B4 50802201 IC50 = 9280 nM T84703 CWCP03 50802214 IC50 = 10000 nM T84703 CQP98F 50802215 IC50 = 2497.3 nM T84703 CVT2O0 50802216 IC50 = 10000 nM T84703 C2G4HZ 50802217 IC50 = 10000 nM T84703 CB1AM0 50802226 IC50 = 20000 nM T84703 CNRX75 50802227 IC50 = 10000 nM T84703 COJ6T7 50802228 IC50 = 20000 nM T84703 CH4K8I 50802229 IC50 = 10000 nM T84703 CST50B 50802232 IC50 = 10000 nM T84703 CI9H3K 50802245 IC50 = 20000 nM T84703 C1LHW9 50802246 IC50 = 20000 nM T84703 C7IQV2 50802247 IC50 = 20000 nM T84703 CY61RH 50802250 IC50 = 10000 nM T84703 CEA48B 50802259 IC50 = 20000 nM T84703 CRT9S8 50802262 IC50 = 4615.5 nM T84703 C23SQR 50802263 IC50 = 20000 nM T84703 C5IZR7 50802274 IC50 = 9792.4 nM T84703 CVR8K4 50802276 IC50 = 10000 nM T84703 C4WMI1 50802277 IC50 = 20000 nM T84703 CG52PC 50802293 IC50 = 20000 nM T84703 CQ3R5U 50802295 IC50 = 20000 nM T84703 CB3CE4 50802298 IC50 = 2027.5 nM T84703 C3FYU7 50802299 IC50 = 20000 nM T84703 C8A6MI 50802307 IC50 = 20000 nM T84703 C94SOF 50802309 IC50 = 63.7 nM T84703 C4Y6SN 50802310 IC50 = 358.6 nM T84703 CCKR79 50802312 IC50 = 10000 nM T84703 CFA79B 50802314 IC50 = 20000 nM T84703 CB8PD0 50802328 IC50 = 10000 nM T84703 C17YAG 50802329 IC50 = 6706 nM T84703 CSL61K 50802332 IC50 = 20000 nM T84703 CGBH51 50802345 IC50 = 10000 nM T84703 C13KBR 50802348 IC50 = 10000 nM T84703 C5SZE1 50802358 IC50 = 10000 nM T84703 C0F1XK 50802359 IC50 = 20000 nM T84703 CE4HR6 50802360 IC50 = 20000 nM T84703 CU5B4V 50802364 IC50 = 20000 nM T84703 CV9PN1 50802374 IC50 = 1340.8 nM T84703 C17PKR 50802391 IC50 = 20000 nM T84703 CJ7G2O 50802392 IC50 = 10000 nM T84703 C5V3JC 50802393 IC50 = 10000 nM T84703 C8JKA9 50802404 IC50 = 20000 nM T84703 C16UZW 50802409 IC50 = 20000 nM T84703 C7KC5M 50802410 IC50 = 20000 nM T84703 CX7BU6 50802411 IC50 = 10000 nM T84703 C5RI6H 50802419 IC50 = 10000 nM T84703 CR6GC8 50802420 IC50 = 10000 nM T84703 C6R1VG 50802424 IC50 = 10000 nM T84703 C6O9GD 50802433 IC50 = 20000 nM T84703 C9UR2X 50825254 IC50 = 20000 nM T84703 CWR12L 50825338 IC50 = 20000 nM T84703 CH6OS5 50825345 IC50 = 20000 nM T84703 CVYM85 50825346 IC50 = 20000 nM T84703 CM24LF 52938983 IC50 < 1 nM T84703 C8NA4L 53384644 IC50 = 8700 nM T84703 C6U0SG 57629460 IC50 = 1 nM T84703 C1EVX0 58063117 IC50 = 5380 nM T84703 CSG5T1 58335664 IC50 = 4 nM T84703 C0HR7L 59804298 IC50 = 27 nM T84703 CZM10S 59804305 IC50 = 15 nM T84703 CJ1BN7 59804319 IC50 = 7 nM T84703 CUQ6Y0 59804322 IC50 = 60 nM T84703 C8ZF3L 59804374 IC50 = 35 nM T84703 C37NKO 67129970 IC50 = 5240 nM T84703 CK80LJ 67130050 IC50 > 10000 nM T84703 CV63UL 67240318 IC50 > 10000 nM T84703 C0VJW8 68545858 IC50 = 21 nM T84703 C7GRV2 68755406 IC50 = 8340 nM T84703 C7VJ6A 70647728 IC50 = 100 nM T84703 C3PX5C 70692373 IC50 = 17 nM T84703 CXZ40O 70696497 IC50 = 19 nM T84703 CKT60L 71455860 Ki > 4500 nM T84703 CRI51K 73819548 Ki = 0.4 nM T84703 CGDB30 74538658 IC50 = 190 nM T84703 CIQ5D8 74627727 IC50 = 132.2 nM T84703 CRSY98 89808125 Ki = 77 nM T84703 C40VNJ 89816720 Ki = 65 nM T84703 CM64AB 90644193 Ki = 0.5 nM T84703 CI4N8P 91801232 IC50 = 0.3 nM T84703 CLZ74S 91826737 IC50 = 94000 nM T84703 CJQ5N6 91936970 IC50 = 1190000 nM T84703 C3PAN1 117967296 IC50 > 81000 nM T84703 CE86QC 118128728 IC50 = 1303.7 nM T84703 C0TMZ8 118167692 IC50 = 2.6 nM T84703 CLH8X7 118189551 IC50 = 6.1 nM T84703 CU3K0B 118456253 IC50 = 14000 nM T84703 C60TWO 118665627 IC50 = 15 nM T84703 CPK47S 118868365 IC50 = 6.2 nM T84703 CN4X0C 121231414 IC50 = 36.8 nM T84703 C08KEM 122179540 IC50 = 270 nM T84703 CQ43XF 122179541 IC50 = 200 nM T84703 C2TXZ9 122179542 IC50 = 120 nM T84703 CXS1Y6 122179543 IC50 = 27 nM T84703 CPF2L7 122179544 IC50 = 7 nM T84703 C3NJ6T 122179545 IC50 = 130 nM T84703 C3AJ4C 122179546 IC50 = 1 nM T84703 CG0RP7 122179547 IC50 = 1 nM T84703 C1A0SQ 122179548 IC50 = 4 nM T84703 C4X7SD 122192466 IC50 > 10000 nM T84703 CC83HO 123131777 IC50 = 27000 nM T84703 C93UNX 132041675 IC50 = 4.2 nM T84703 C1X6FJ 134693894 IC50 = 40 nM T84703 CXC69T 137321158 IC50 = 8 nM T84703 CWC49K 137321210 IC50 > 1000 nM T84703 CI1E8V 137634241 IC50 = 379 nM T84703 CNRT47 139434032 EC50 = 790 nM T84703 CIN6L7 139434035 EC50 = 370 nM T84703 CTFE03 139434036 EC50 = 230 nM T84703 CX9H4W 139434047 EC50 = 750 nM T84703 CU10QZ 139434077 EC50 = 370 nM T84703 CLRW84 139434103 EC50 = 950 nM T84703 CB6F5R 139434105 EC50 = 1400 nM T84703 C7FBY1 139434107 EC50 = 390 nM T84703 C08MUD 139434127 EC50 = 250 nM T84703 C2MZ4L 139434198 EC50 = 610 nM T84703 CJIH42 139434200 EC50 = 270 nM T84703 C7W5MH 139434224 EC50 = 110 nM T84703 CXIT16 139434239 EC50 = 460 nM T84703 C2B8OV 139442846 EC50 = 120 nM T84703 C4ID6F 139442949 EC50 = 450 nM T84703 CX4E3H 142736778 IC50 = 4.42 nM T84703 CAJQ14 145964002 IC50 = 6.6 nM T84703 CVF4M6 145965985 IC50 = 2.7 nM T84703 C5MHK6 145967970 IC50 = 900 nM T84703 CK9C0H 145970062 IC50 = 29 nM T84703 CI85EU 145998085 IC50 > 1000 nM T84703 CA10CQ 155512867 IC50 > 1000 nM T84703 C2MD1Q 155513187 IC50 > 10000 nM T84703 C5B2AX 155513312 IC50 = 24.19 nM T84703 CZMD64 155514443 IC50 > 1000 nM T84703 CB5T9G 155515436 IC50 = 145.4 nM T84703 CUHZ87 155516883 IC50 > 1000 nM T84703 COR4M0 155517181 IC50 = 20000 nM T84703 CIU1T6 155518465 IC50 = 41.34 nM T84703 C86HPW 155518524 IC50 = 6300 nM T84703 CO63MP 155519543 IC50 = 10.47 nM T84703 C9TU2A 155520832 IC50 = 5000 nM T84703 CBG4P0 155524103 IC50 = 43.47 nM T84703 CN6C2T 155528463 IC50 = 13.11 nM T84703 C0HW7F 155530527 IC50 > 1000 nM T84703 CP5IW9 155530600 IC50 > 1000 nM T84703 C3MC2P 155532434 IC50 = 178.45 nM T84703 CNE6A3 155532801 IC50 = 38.35 nM T84703 C2KAU0 155533663 IC50 = 22.73 nM T84703 C75AKY 155533695 IC50 < 10 nM T84703 C3PWI1 155534046 IC50 > 1000 nM T84703 CTXK93 155535665 IC50 = 270.7 nM T84703 C14SEB 155535950 IC50 = 343.9 nM T84703 CV9D5J 155536164 IC50 = 315.13 nM T84703 C3O6WX 155540330 IC50 > 1000 nM T84703 C76NKG 155543431 IC50 > 1000 nM T84703 CRV40J 155546026 IC50 = 253.65 nM T84703 C8AG4U 155550655 IC50 = 15.59 nM T84703 C2RQT8 155550913 IC50 < 10 nM T84703 C9MJL5 155551408 IC50 > 1000 nM T84703 CM7Q3F 155556300 IC50 = 1500 nM T84703 C9OLA3 155557330 IC50 = 0.2 nM T84703 CYD1C7 155560599 IC50 > 1000 nM T84703 C40IYS 155562258 IC50 = 58.8 nM T84703 CBG9Z1 155562952 IC50 = 569 nM T84703 C0WZ9S 155563842 IC50 > 1000 nM T84703 CWR4O5 155565233 IC50 = 9.3 nM T84703 CRFW02 155566430 IC50 = 43.92 nM T84703 C0V7SM 155567015 IC50 > 1000 nM T84703 D00ERW 44444843 Ki > 4536 nM T84703 D00HVA 11624601 Ki > 4500 nM T84703 D02RWC 59397065 IC50 = 12 nM T84703 D07ADX 54764565 IC50 = 217 nM T84703 D0E7VO 59627005 IC50 < 100 nM T84703 D0K5UF 72710568 IC50 = 4 nM T84703 D0L3JR 25212148 IC50 = 9 nM T84703 D0N4LR 53469448 IC50 = 2962 nM T84703 D0O8AR 16097523 IC50 = 0.93 nM T84703 D0Q3NG 11715520 Ki > 4500 nM T84703 D0R2WK 16038120 IC50 = 2018 nM T84703 D0S7IE 11658882 Ki > 4500 nM T89697 D00AXJ 4189 IC50 = 1400 nM T89697 D03GET 4055 IC50 = 370 nM T89697 D04GYO 5353853 IC50 = 28000 nM T89697 D05EJG 6305 IC50 = 498700 nM T89697 D0AA2D 2378 IC50 = 23000 nM T89697 D0EV8E 3198 IC50 = 1100 nM T89697 D0O6UZ 65863 IC50 = 8400 nM T89697 D0P9AC 3675 IC50 = 14000 nM T89697 D0X8XA 5318 IC50 = 6400 nM T89697 D0Y0GH 5746 Ki = 25000 nM T89697 D06MHZ 66558287 Ki = 7 nM T89697 D08CJK 1150 Ki = 156000 nM T89697 D0B1FE 3194 Ki = 94 nM T89697 D0B5HS 405012 EC50 = 110000 nM T89697 D0C0NH 3806 IC50 = 1000 nM T89697 D0DA5M 75202656 IC50 = 23 nM T89697 D0DP5I 121328278 IC50 = 0.5 nM T89697 D0J1HB 23063810 IC50 = 410 nM T89697 D0PM5U 135564890 IC50 = 7 nM T89697 D0W0VD 3885 Ki = 100 nM T89697 D09HVV 118898844 IC50 = 3 nM T89697 D0MQ3X 5316743 IC50 = 1300 nM T89697 D0QZ8K 70874141 EC50 = 330 nM T89697 D0S7BW 78426054 IC50 < 1000 nM T89697 D0WR7B 122650373 IC50 = 9.7 nM T89697 D0YY4R 121339537 IC50 = 3 nM T89697 D0R7MJ 135403797 IC50 = 60000 nM T89697 C6A3UH 3037 IC50 = 70000 nM T89697 C0RFA2 3102 IC50 = 1000000 nM T89697 C9LCD8 3823 IC50 = 25000 nM T89697 CP62OB 5138 IC50 = 61000 nM T89697 CXHL15 6755 IC50 = 675000 nM T89697 C2JK3W 7104 IC50 = 1000000 nM T89697 COE28J 7220 IC50 = 2570000 nM T89697 CEUJ71 7400 IC50 > 20000 nM T89697 CV9D7A 7516 IC50 = 230 nM T89697 C9KP5F 7518 IC50 = 9200 nM T89697 CV79ZO 7564 IC50 = 400000 nM T89697 CJ19CF 7812 IC50 = 1319000 nM T89697 C45VRP 7815 IC50 = 1900 nM T89697 CM75BH 8447 IC50 > 500000 nM T89697 CG47UK 10241 IC50 > 200000 nM T89697 CBIR94 10313 IC50 = 16000 nM T89697 COI9A4 10852 IC50 = 61000 nM T89697 C25MFK 11157 IC50 = 71000 nM T89697 COZB91 11988 IC50 = 8000 nM T89697 C08ZTB 13397 IC50 > 20000 nM T89697 CGC0N1 13886 IC50 = 161000 nM T89697 CE4X3M 21095 IC50 = 3970 nM T89697 CUP89L 22244 IC50 = 15000 nM T89697 C0HZ4G 22641 IC50 = 1000000 nM T89697 CC0BW7 22704 IC50 > 500000 nM T89697 CA90DS 23116 IC50 = 800 nM T89697 COY1P0 32238 IC50 = 130000 nM T89697 CL1A5R 37175 IC50 = 23000 nM T89697 C51XBL 40302 IC50 = 1000000 nM T89697 C2HMI7 66036 IC50 > 20000 nM T89697 C0F5BM 67430 IC50 > 20000 nM T89697 C1B9ZO 68094 IC50 = 2000000 nM T89697 C3AVU2 72732 IC50 = 4340 nM T89697 CW95YM 73468 IC50 = 22600 nM T89697 C1BI4N 74318 IC50 > 1000000 nM T89697 CYH1I4 74787 IC50 = 870 nM T89697 CHO9A0 74967 IC50 = 2700 nM T89697 CDL20X 75899 IC50 > 1000000 nM T89697 CRY89S 83050 IC50 = 500000 nM T89697 CSMK07 98112 IC50 = 14690 nM T89697 CB4VI8 99128 IC50 = 114000 nM T89697 C3CKU4 102313 IC50 < 10000 nM T89697 CD68XC 104251 IC50 = 400000 nM T89697 CD24AO 114918 Ki = 326 nM T89697 CBZX05 120425 IC50 = 24000 nM T89697 CS53VH 128994 IC50 = 4680 nM T89697 C5LQN0 199162 IC50 = 10000 nM T89697 CTDZ45 201863 EC50 = 2000 nM T89697 CUG38M 203812 IC50 = 410 nM T89697 CH0ZD7 207299 IC50 = 134 nM T89697 CN6O1K 217573 IC50 = 1300 nM T89697 CNQE70 224502 IC50 = 21000 nM T89697 CCQ3W7 233294 IC50 = 35600 nM T89697 C8PEY0 234811 IC50 = 400 nM T89697 CR36LZ 235240 Ki > 100000 nM T89697 CFPL09 236715 IC50 = 1780 nM T89697 CR48HG 239465 IC50 = 750 nM T89697 C37KML 244989 IC50 = 15700 nM T89697 CVO36F 248768 IC50 = 6300 nM T89697 C4MLK5 255448 IC50 = 1600 nM T89697 CRJ5W7 259418 IC50 = 1500 nM T89697 CU3D0T 261066 IC50 = 42500 nM T89697 CR1C6K 261602 IC50 = 714 nM T89697 CE7M6K 269624 Ki = 4300 nM T89697 CLC05O 272989 IC50 = 1950 nM T89697 CRF3E1 273059 IC50 = 8200 nM T89697 CR9VJ4 273769 IC50 = 332 nM T89697 CS46CV 276137 IC50 = 35600 nM T89697 CY3BT7 291128 IC50 = 31600 nM T89697 CV57WU 291217 IC50 = 266000 nM T89697 C9TU7X 291363 IC50 = 32600 nM T89697 C8GDA3 302654 IC50 = 44900 nM T89697 C1OA7G 313613 IC50 = 3300 nM T89697 C0UAT7 313614 IC50 = 660 nM T89697 C8RHI3 313619 IC50 = 24000 nM T89697 CJ1V4S 325901 IC50 = 42500 nM T89697 CC2M9A 332650 IC50 = 4100 nM T89697 C4HP3I 332972 IC50 = 4900 nM T89697 COK78A 333769 IC50 = 6080 nM T89697 C3RMI4 333770 IC50 = 34960 nM T89697 C8BS0X 334304 IC50 = 464000 nM T89697 CA1H8B 336270 IC50 = 183 nM T89697 CL2JH7 336699 IC50 = 930 nM T89697 CD3RI9 356301 IC50 = 76000 nM T89697 CDK1S3 356303 IC50 = 96000 nM T89697 CM49EY 362360 IC50 = 460 nM T89697 CVD5W0 363326 IC50 = 3000 nM T89697 C7EZ4T 369539 IC50 = 1000000 nM T89697 CNS32X 371271 IC50 = 35600 nM T89697 CUR85O 378581 IC50 = 46700 nM T89697 CB9RU8 421540 IC50 > 10000 nM T89697 CQ7P3K 432556 IC50 = 890 nM T89697 C46VHU 478572 IC50 = 53.9 nM T89697 C72ZLN 478574 IC50 = 23 nM T89697 CC7IW3 478577 IC50 = 121200 nM T89697 C2ZR8M 478643 IC50 = 466 nM T89697 CY38AJ 478645 IC50 = 864400 nM T89697 CZT01E 478647 IC50 = 27.1 nM T89697 CD1AO0 487082 IC50 = 4400 nM T89697 C74FPR 497025 Ki = 35 nM T89697 C03NZX 523214 IC50 = 156 nM T89697 C4ONK2 555630 IC50 = 490 nM T89697 CR2L7A 600260 IC50 = 6000000 nM T89697 CZI5R2 601577 IC50 = 817000 nM T89697 CN7WA6 615185 IC50 = 4800 nM T89697 CD3V5T 651817 IC50 > 100000 nM T89697 C8K5LQ 657876 IC50 = 123000 nM T89697 C6C9AZ 658687 IC50 = 50000 nM T89697 CEM8K0 685364 IC50 = 195000 nM T89697 C6NX0C 689063 IC50 = 90490 nM T89697 CKMP38 697993 IC50 = 126000 nM T89697 C7M4VB 698285 IC50 = 1800 nM T89697 CO46LB 706988 IC50 > 50000 nM T89697 CNV69W 707050 IC50 = 15000 nM T89697 C5W2PB 717704 IC50 > 50000 nM T89697 CV53ZJ 725906 IC50 = 1690 nM T89697 C6WQ0V 735843 IC50 > 20000 nM T89697 CM7C6Y 737132 IC50 > 50000 nM T89697 C3WG8U 737138 IC50 > 50000 nM T89697 C5LN3R 737149 IC50 = 1800 nM T89697 CUMJ16 737276 IC50 > 50000 nM T89697 CO5F6Z 737504 IC50 = 41000 nM T89697 CAG2B4 763555 IC50 = 522000 nM T89697 CK89WR 781705 IC50 = 112000 nM T89697 CY02AP 795453 IC50 = 71 nM T89697 CI43WJ 802727 IC50 = 1800 nM T89697 CG54RM 802728 IC50 = 83000 nM T89697 C64NSF 819511 IC50 = 35000 nM T89697 CDEF92 820765 IC50 = 5888.44 nM T89697 CXYV26 849731 IC50 = 767 nM T89697 C47XAO 849732 IC50 > 10000 nM T89697 CB27WS 849733 IC50 = 808.9 nM T89697 C5S9DF 849734 IC50 = 4612 nM T89697 C34QEU 849735 IC50 = 1770 nM T89697 CC10TB 852498 IC50 = 65000 nM T89697 CFD05W 992980 IC50 = 20100 nM T89697 C85BIS 992984 IC50 = 3200 nM T89697 CXWM34 993112 IC50 = 5600 nM T89697 CEQ35N 1016842 IC50 = 18000 nM T89697 CSC0B6 1041635 IC50 = 2587 nM T89697 CY6C8D 1085103 IC50 = 1190 nM T89697 CK4G6F 1167203 IC50 = 12400 nM T89697 CT2F4J 1479909 IC50 = 2600 nM T89697 CTE7D4 1484508 IC50 > 20000 nM T89697 C7NOW6 1712812 IC50 = 82000 nM T89697 C5D0MU 1810299 IC50 > 50000 nM T89697 C25ERJ 1810302 IC50 = 17000 nM T89697 C4QW9C 2728703 IC50 = 1000 nM T89697 CI85YE 2731263 IC50 > 50000 nM T89697 C0FH4G 2732070 IC50 > 20000 nM T89697 CY78SE 2735617 IC50 = 1600 nM T89697 CN35FD 2737499 IC50 = 3700 nM T89697 C7I1HC 2744597 IC50 = 38610 nM T89697 C94BMC 2757941 IC50 > 50000 nM T89697 C3IRL6 2758211 IC50 = 18000 nM T89697 CQ6Z8A 2759372 IC50 = 3500 nM T89697 CYD7A1 2764014 IC50 = 630 nM T89697 CHS3B0 2794173 IC50 = 6000 nM T89697 C84XTS 2803091 IC50 = 11700 nM T89697 CHJQ46 2806436 IC50 = 6300 nM T89697 CXM75A 2807416 IC50 = 3100 nM T89697 CCEN29 2810177 IC50 = 13000 nM T89697 C59BGS 2818222 IC50 > 100000 nM T89697 C1H3JC 2821620 IC50 = 97000 nM T89697 CN7MC6 2821621 IC50 = 15000 nM T89697 CHB3S4 2821626 IC50 = 4600 nM T89697 CK2FZ7 2821627 IC50 = 18000 nM T89697 CG8L6W 2824871 IC50 = 710 nM T89697 CM9J0C 2825091 IC50 = 2000000 nM T89697 C7X5WE 2828334 IC50 = 110 nM T89697 CU6Z9O 2917429 Ki = 342300 nM T89697 C3KZ0U 3028808 IC50 = 2000 nM T89697 CHRQ07 3032509 Ki = 72410 nM T89697 C09JXD 3032646 Ki = 62360 nM T89697 C37ABE 3035211 Ki = 12000 nM T89697 C6ZP2C 3106159 IC50 = 1000 nM T89697 C7D6IH 3161266 IC50 = 310000 nM T89697 C53LIN 3325609 EC50 = 128 nM T89697 C61GRB 3443692 IC50 = 2400 nM T89697 CZ9IS6 3529520 IC50 = 120 nM T89697 CB0D8U 3595344 EC50 = 3118 nM T89697 C7O9DU 3720080 IC50 = 2600 nM T89697 CIO57N 3761458 IC50 > 20000 nM T89697 C12IDC 3901929 IC50 = 1510 nM T89697 C7DM2Y 4099901 IC50 = 108000 nM T89697 CV10YZ 4190125 EC50 = 420 nM T89697 CA3PO5 4240303 EC50 > 10 nM T89697 CH6K0A 4310362 IC50 = 68000 nM T89697 C87WUF 4381769 IC50 = 15000 nM T89697 CNUQ02 4456830 IC50 = 1580 nM T89697 CB5P9D 4574587 IC50 = 379.5 nM T89697 C45WVE 4638522 EC50 = 640 nM T89697 CZNE04 4794706 IC50 = 49 nM T89697 CU6XY2 5068606 IC50 = 26000 nM T89697 C0VGT3 5170924 IC50 > 50000 nM T89697 CAW37X 5240714 IC50 = 3740 nM T89697 C8KM3N 5371761 IC50 = 110 nM T89697 CS67OL 5712754 IC50 = 20000 nM T89697 C9C5OF 5937842 IC50 = 50000 nM T89697 CFGA74 6198019 Ki = 3000 nM T89697 C1RPA8 6223130 EC50 = 13260 nM T89697 CL82TX 6400901 IC50 = 940 nM T89697 CGP9S8 6409664 IC50 = 620 nM T89697 C3AV5I 6419227 IC50 = 22000 nM T89697 CIQ4X3 6419341 IC50 = 1256000 nM T89697 C5KX9O 6494204 Ki = 35 nM T89697 CXE93M 6494205 Ki = 35 nM T89697 CP1O4X 7064051 IC50 = 2700 nM T89697 CR0P9A 7463552 IC50 = 17910 nM T89697 CN16IB 8005342 EC50 = 609 nM T89697 CP61HD 8070877 IC50 = 9750 nM T89697 CZ06FE 8071109 IC50 = 30800 nM T89697 CN9Y1O 8106455 IC50 > 100000 nM T89697 CP43WG 8106458 IC50 > 20000 nM T89697 CNW5G7 9573924 Ki = 1500 nM T89697 C0PE9C 9584160 IC50 = 60000 nM T89697 C7HIG1 9584719 IC50 = 31000 nM T89697 C8VKT5 9685191 IC50 = 2780 nM T89697 CAVT12 9812842 IC50 = 39000 nM T89697 C4UYP5 9815283 IC50 > 100000 nM T89697 CQ25OP 9833992 IC50 = 680000 nM T89697 C4QZ1I 9877471 IC50 = 190000 nM T89697 C7N9PW 9877511 IC50 = 1028000 nM T89697 C71STY 9899224 IC50 = 2300000 nM T89697 C6NS2U 9899225 IC50 = 6000 nM T89697 CU3RN8 9920462 IC50 = 70000 nM T89697 C69CDF 9920916 IC50 = 2600 nM T89697 C2PCN3 9964175 IC50 = 1500000 nM T89697 CUP4N1 9964258 Ki = 14500 nM T89697 CE64VW 10101379 IC50 = 440 nM T89697 CQC7N5 10332864 IC50 = 80.3 nM T89697 C4XB1O 10355804 IC50 = 140000 nM T89697 CH8N5K 10374898 IC50 = 190000 nM T89697 CYO69B 10511388 IC50 = 825000 nM T89697 C9JU5L 10559053 IC50 = 41000 nM T89697 CL21AV 10583021 IC50 = 5700 nM T89697 C8GMF7 10890197 IC50 > 100000 nM T89697 C7Q6NX 10909696 IC50 = 1800000 nM T89697 CI3T6M 11086357 IC50 = 4950 nM T89697 CYKR73 11175492 Ki = 35 nM T89697 CFD24O 11209246 Ki = 35 nM T89697 C4RKW2 11255489 Ki = 35 nM T89697 C32WXK 11275256 IC50 = 2900 nM T89697 CB50ZE 11423685 IC50 = 422000 nM T89697 C2P0LW 11482022 Ki = 47570 nM T89697 CJ3AO4 11528610 Ki = 1292000 nM T89697 C9A3BN 11528678 Ki = 42060 nM T89697 C5AI2W 11536281 Ki = 33970 nM T89697 CGT35V 11543253 Ki = 179600 nM T89697 CF5C4D 11580169 IC50 = 420 nM T89697 C5H7ZN 11629967 Ki = 1267000 nM T89697 CL48GN 11651542 Ki = 149350 nM T89697 CZS94C 11673059 Ki = 328700 nM T89697 CZS6U0 11694196 IC50 = 650000 nM T89697 CXKY79 11701328 Ki = 202000 nM T89697 CEM3R0 11708775 Ki = 40950 nM T89697 CT7KH0 11757335 IC50 = 15000 nM T89697 C4Q1MV 12014591 Ki = 35 nM T89697 CD6L1H 12239941 IC50 = 2920 nM T89697 CQ9ZI8 12239942 IC50 = 121 nM T89697 C53LFZ 12240982 IC50 = 533000 nM T89697 CQN15E 12243104 IC50 = 22000 nM T89697 C1MS3C 12244898 IC50 = 61000 nM T89697 CT0AG4 12398786 IC50 > 20000 nM T89697 CW0OD3 12398789 IC50 > 100000 nM T89697 CSM6Z7 12457713 IC50 > 50000 nM T89697 C3NTB9 12463137 IC50 = 1200000 nM T89697 CYO6J1 12471537 IC50 = 460000 nM T89697 C1FL0I 12474093 IC50 = 3400 nM T89697 CRX8P7 12674978 IC50 = 1970 nM T89697 C9BJU0 12722498 IC50 > 50000 nM T89697 C5PD2B 12760607 IC50 = 200000 nM T89697 C29LGR 12800721 IC50 = 980 nM T89697 C39AWQ 13393248 IC50 = 3390 nM T89697 CQ21YE 13762869 IC50 = 779 nM T89697 C3Y2XJ 14034883 IC50 = 190 nM T89697 CC94WU 14171303 IC50 = 29 nM T89697 CYE1A6 14171304 IC50 = 26.2 nM T89697 CW53FC 14269350 IC50 = 24920 nM T89697 C19VME 14269353 IC50 = 50810 nM T89697 C7G0ME 14269354 IC50 = 62660 nM T89697 CO2TC8 14694516 IC50 = 18000 nM T89697 C96HAY 14736077 IC50 > 20000 nM T89697 C7XD2T 15118768 Ki = 635000 nM T89697 C9MNU7 15326268 IC50 = 370 nM T89697 CTF31B 15326270 IC50 = 53000 nM T89697 C83DSK 15754003 IC50 = 13000 nM T89697 CXW9D2 15946462 Ki = 210 nM T89697 C0W9ID 16059788 Ki = 120 nM T89697 CMJV13 16069892 IC50 > 30000 nM T89697 C07KDO 16069930 IC50 > 30000 nM T89697 C3J1EB 16069933 IC50 = 20600 nM T89697 CM74CV 16069934 IC50 > 30000 nM T89697 CKH6M4 16090079 IC50 = 977 nM T89697 CQ7B2J 16118954 Ki = 82540 nM T89697 CGDT43 16228806 IC50 = 1500 nM T89697 C91JFG 17750145 IC50 = 320 nM T89697 CNR81H 17995458 IC50 = 1000000 nM T89697 CB21MY 18314043 IC50 > 20000 nM T89697 CNS59Y 18506325 IC50 = 1028000 nM T89697 CTS6O0 18525978 IC50 = 1600 nM T89697 C2IQL8 18525980 IC50 = 450 nM T89697 C68SNL 18525982 IC50 = 2500 nM T89697 CAF4Q6 18525983 IC50 = 5400 nM T89697 C3C7JL 18525997 IC50 = 9500 nM T89697 CZ84SF 18526040 IC50 = 8900 nM T89697 CS84LJ 19702149 IC50 = 60000 nM T89697 CEL18N 19974989 IC50 = 630 nM T89697 CQIY45 20373984 IC50 = 209000 nM T89697 C2ID7K 20525178 IC50 = 830000 nM T89697 C2B0PJ 21125239 IC50 = 340 nM T89697 C4EOJ3 21155916 IC50 = 880 nM T89697 CP37KN 21192890 IC50 = 1400 nM T89697 C0VLB8 21683122 IC50 = 2100 nM T89697 C08CBI 21723626 IC50 = 24000 nM T89697 C50TDQ 21798789 IC50 = 820000 nM T89697 CGM9O7 22009901 IC50 > 100000 nM T89697 C4J1QN 22989754 IC50 = 7100 nM T89697 C1BI5L 22989786 IC50 = 1680 nM T89697 C07TJG 22989894 IC50 = 12000 nM T89697 CEM41C 23063802 IC50 = 830 nM T89697 C0TJ5U 23084904 IC50 = 179000 nM T89697 C0CIY4 23084917 IC50 = 60000 nM T89697 CPC8I6 23206139 IC50 = 1000 nM T89697 CQ93UJ 23332019 IC50 = 1300000 nM T89697 C3P4TR 23766450 Ki = 35 nM T89697 C3BVO4 24264313 IC50 > 100000 nM T89697 CBXC05 24424330 IC50 = 37000 nM T89697 C0Z3PM 24741909 IC50 = 2310 nM T89697 CP4I3W 24742062 IC50 = 94000 nM T89697 CSK1I0 24788785 Ki = 260 nM T89697 CQ16CP 24822271 IC50 = 247 nM T89697 CZ5PI3 24822272 IC50 = 5520 nM T89697 C4BOC3 24822273 IC50 = 2050 nM T89697 C40EMQ 24824456 IC50 = 2130 nM T89697 CAL06M 24824607 IC50 = 3020 nM T89697 C1JN8S 24824608 IC50 = 933 nM T89697 CPFN24 24824612 IC50 = 130 nM T89697 CWO6G7 24825243 Ki = 41 nM T89697 CO29PG 24825244 Ki = 1490 nM T89697 CF65SE 24825245 Ki = 10900 nM T89697 C4HY5W 24825246 Ki = 420 nM T89697 C3PE8G 24825247 Ki = 200 nM T89697 CJ5O3I 24825249 Ki = 260 nM T89697 C9TH2J 24971328 Ki = 4800 nM T89697 C4OA9Q 24971329 IC50 = 25000 nM T89697 C7FWD4 24971330 IC50 = 38000 nM T89697 CV1IW8 24971331 IC50 = 73000 nM T89697 CF8G3E 24971332 IC50 = 365000 nM T89697 CPR02N 24971333 IC50 = 734000 nM T89697 C10SAI 24971370 IC50 = 4950 nM T89697 CV6L8H 25141140 Ki = 76300 nM T89697 C1XU4T 25141142 Ki = 87100 nM T89697 CQJ8F1 25211983 IC50 = 127 nM T89697 C0ZJY1 25211984 IC50 = 188 nM T89697 CO2GF9 25241857 IC50 = 5400 nM T89697 C0DT1U 25241896 IC50 = 2200 nM T89697 CPC12H 25241897 IC50 = 900 nM T89697 C9OWU5 26921488 IC50 > 30000 nM T89697 CX8T3C 28934713 IC50 > 50000 nM T89697 CUGD12 28934715 IC50 = 34000 nM T89697 CJ9S5L 28934757 IC50 > 50000 nM T89697 CJU84V 28934769 IC50 > 50000 nM T89697 CZ98CD 28934783 IC50 = 1200 nM T89697 CF8CJ7 30762236 IC50 > 30000 nM T89697 CH0DU1 35353466 IC50 = 99350 nM T89697 C8JMZ6 35354409 IC50 = 99830 nM T89697 CE8F0K 36688758 IC50 = 54100 nM T89697 CN19VO 40418972 IC50 = 3800 nM T89697 C4S7PI 43348154 IC50 = 34000 nM T89697 CL04IU 44156271 IC50 = 14000 nM T89697 CPN0X1 44251142 Ki = 11550 nM T89697 C4G3PD 44406794 Ki = 28380 nM T89697 CX5Y4V 44406795 Ki = 20480 nM T89697 C7Q8JF 44406806 Ki = 36950 nM T89697 CR57ND 44406812 Ki = 363600 nM T89697 CVH98E 44457253 IC50 = 82 nM T89697 CVRQ27 44457255 IC50 = 186 nM T89697 CS17JV 44457280 IC50 = 55 nM T89697 C24PTC 44457418 IC50 = 1500 nM T89697 CS7I1E 44457419 IC50 = 512 nM T89697 CT0YX5 44457436 IC50 = 2120 nM T89697 CT8K3L 44457437 IC50 = 1090 nM T89697 CI2VN4 44457447 IC50 = 3960 nM T89697 C87CKB 44457448 IC50 = 360 nM T89697 C7W8KH 44465701 IC50 = 450 nM T89697 CO15EU 44465944 IC50 > 1000000 nM T89697 C97EPW 44465950 IC50 = 400000 nM T89697 C1SF4O 44465951 IC50 = 90000 nM T89697 C04XGN 44465952 IC50 = 60000 nM T89697 C0JPM6 44466194 IC50 = 105000 nM T89697 C3BVF5 44466197 IC50 = 5000 nM T89697 CT1KO3 44466198 IC50 = 200000 nM T89697 C15FTG 44467660 IC50 = 9100 nM T89697 CEQ9F7 44467799 IC50 = 18000 nM T89697 C8C4GX 44468002 IC50 = 23000 nM T89697 CA60ES 44597169 IC50 > 20000 nM T89697 CWC4K1 44597274 IC50 = 1400 nM T89697 CM7T5C 44597275 IC50 = 1400 nM T89697 C2QT3S 44597276 IC50 > 2000 nM T89697 CF8DA5 44597277 IC50 > 2000 nM T89697 C2AP6Q 44819148 IC50 = 22400 nM T89697 CA0KJ8 44819149 IC50 = 12600 nM T89697 CZ3M0U 45158558 IC50 = 570 nM T89697 CW9B1I 45248340 IC50 = 18600 nM T89697 CPLJ59 45482936 IC50 = 11900 nM T89697 C4GO2W 45482946 IC50 = 4200 nM T89697 C24MGQ 45482949 IC50 = 7100 nM T89697 CU3F6W 45487175 IC50 = 50000 nM T89697 CL93SV 45487181 IC50 = 200 nM T89697 C6U2HB 45487187 IC50 = 50000 nM T89697 C7O5EN 45487189 IC50 = 44000 nM T89697 C2ASP5 45487202 IC50 = 40000 nM T89697 CYD0A1 45487207 IC50 = 50000 nM T89697 C2D3ZL 45487229 IC50 = 25000 nM T89697 CLWY27 46180669 IC50 = 520 nM T89697 C6HTU7 46834223 IC50 = 1371000 nM T89697 CQL2S9 46913822 IC50 = 24600 nM T89697 C96QOX 47827438 IC50 = 90 nM T89697 C7T2OH 47827446 IC50 = 961 nM T89697 C9BM5X 49866156 IC50 > 20000 nM T89697 CWOF35 49866158 IC50 > 20000 nM T89697 C2NJ3B 51003508 IC50 = 14000 nM T89697 CMF2O6 52912227 IC50 < 1000 nM T89697 CQP52L 52918052 IC50 = 36000 nM T89697 C06VWA 52932742 IC50 < 1000 nM T89697 C58PSL 52935731 IC50 = 1700 nM T89697 C7P1KN 52936167 IC50 = 1700 nM T89697 CEQN27 52936621 Ki > 1000 nM T89697 CZ0CG8 52942238 IC50 = 880 nM T89697 CFR5M9 53316976 IC50 = 37000 nM T89697 CO2KF5 53317021 IC50 = 96000 nM T89697 CW6Q5U 53317048 IC50 = 37000 nM T89697 CD1J7C 53318255 IC50 = 45000 nM T89697 CKF1H7 53318256 IC50 = 141000 nM T89697 CFB26Q 53318297 IC50 = 83000 nM T89697 C2ZLA8 53318331 IC50 = 43000 nM T89697 CW9T8K 53319620 IC50 = 34000 nM T89697 CS3Y6N 53319657 IC50 = 18000 nM T89697 CS5T9R 53319675 IC50 = 82000 nM T89697 CF6EU4 53320957 IC50 = 87000 nM T89697 CD0IC5 53322284 IC50 = 153000 nM T89697 CSO21L 53323252 IC50 = 29000 nM T89697 CG1R0E 53323675 IC50 = 13100 nM T89697 C7RKN6 53324267 IC50 = 26200 nM T89697 C7BA9R 53324928 IC50 = 58000 nM T89697 CP2AK1 53324929 IC50 = 49000 nM T89697 CK4LN0 53324956 IC50 = 63000 nM T89697 CAB8U0 53326252 IC50 = 139000 nM T89697 CQ4PM6 55254080 IC50 = 490 nM T89697 CT5M9H 56659238 Ki = 40000 nM T89697 CKG5F8 56666431 IC50 = 92000 nM T89697 CP6V9F 57408307 IC50 = 21000 nM T89697 CA19IT 57611775 EC50 = 1260 nM T89697 CA3XG9 58294074 IC50 = 6600 nM T89697 CR57BA 58294080 EC50 = 2400 nM T89697 CGQ3X8 58294086 EC50 = 110000 nM T89697 CPAV97 58294088 IC50 = 3800 nM T89697 C8EYR1 58294092 IC50 > 1000000 nM T89697 C26VNU 58294099 IC50 = 187000 nM T89697 C4LD1V 58294110 IC50 = 312000 nM T89697 COXA92 58294117 IC50 = 300 nM T89697 CZXO68 58294132 IC50 = 5100 nM T89697 CJL85W 58294141 IC50 = 7200 nM T89697 C01SLN 58294147 IC50 = 960 nM T89697 CRL75F 58294169 IC50 = 7800 nM T89697 CU0V3W 58294216 EC50 = 1700 nM T89697 C63ZDL 58294226 IC50 = 44000 nM T89697 CLI6P9 58294227 IC50 > 1000000 nM T89697 CO05DE 58693509 IC50 = 1000 nM T89697 CVJ0N6 60154724 IC50 = 4300 nM T89697 CA1TW8 60154725 IC50 = 6400 nM T89697 CA8W4D 60154726 IC50 = 23000 nM T89697 C6AMR4 60154727 IC50 = 72000 nM T89697 C0ZP8T 60154728 IC50 = 1200000 nM T89697 CU12TW 60154729 IC50 = 3000000 nM T89697 CRKM01 60154730 IC50 = 3200000 nM T89697 CW0FS2 60156091 IC50 = 1100 nM T89697 CDM64W 60156092 IC50 = 2800 nM T89697 CS31CB 60156093 IC50 = 3300 nM T89697 C2LSA3 60156094 IC50 = 7400 nM T89697 CA34YM 60156095 IC50 = 56000 nM T89697 CP34LY 60156096 IC50 = 1800000 nM T89697 CK9JV7 60623327 IC50 = 53130 nM T89697 CQ0G4K 60623350 IC50 = 49250 nM T89697 CSVT86 66553577 IC50 = 10000 nM T89697 CP59KG 66553578 IC50 = 11000 nM T89697 CD2H5Z 66553579 IC50 = 53000 nM T89697 C3C2VH 66553580 IC50 = 29000 nM T89697 C1LB6D 66558197 IC50 = 610 nM T89697 CHX38T 66558199 EC50 = 5900 nM T89697 CU4E2L 66558294 IC50 = 1100 nM T89697 CN91RJ 66558377 EC50 = 5400 nM T89697 C7UKS4 66558379 EC50 = 1100 nM T89697 C9ML2G 66558380 EC50 = 15000 nM T89697 CA4B9P 66558554 IC50 = 1000 nM T89697 CCK6E5 66558639 IC50 = 45 nM T89697 C35NBR 66558640 IC50 = 2400 nM T89697 CK2ZH4 66558723 IC50 = 2900 nM T89697 C8PJ5X 66558811 IC50 = 370 nM T89697 CZ1R2N 66558888 IC50 = 8800 nM T89697 CFM1C3 66760716 IC50 = 3400 nM T89697 C9XC3P 66761410 IC50 = 1400 nM T89697 CBZT64 66761654 IC50 = 2700 nM T89697 CQO09P 67036471 IC50 = 53000 nM T89697 CBH06U 67131986 IC50 = 340 nM T89697 CL0ZD8 67132094 IC50 = 2400 nM T89697 CIC2O5 67132131 IC50 = 1600 nM T89697 C9XRU4 67132184 IC50 = 900 nM T89697 CJ6YI2 67207384 IC50 = 47000 nM T89697 C69FWP 67222089 IC50 > 1000000 nM T89697 C27GIY 68348080 EC50 = 7900 nM T89697 C46KPQ 68348135 IC50 = 32000 nM T89697 CC42EQ 68348137 IC50 = 154000 nM T89697 CX4Y2I 69476274 IC50 = 15000 nM T89697 CA92SK 70874201 IC50 = 3400 nM T89697 CUCQ24 70874317 EC50 = 93 nM T89697 CSO9W5 70874322 EC50 = 490 nM T89697 C1IJ0W 70874391 EC50 = 780 nM T89697 CO3Y9B 70874393 EC50 = 510 nM T89697 C8LCK6 70874412 EC50 = 2200 nM T89697 C1H7VK 70874453 IC50 = 19 nM T89697 CJF91M 70874544 IC50 = 46 nM T89697 C9EWB8 70874603 EC50 = 200 nM T89697 C8CMD0 70874604 IC50 < 1000 nM T89697 C82PUD 70874605 EC50 = 78 nM T89697 CMW8S2 70874703 EC50 = 2700 nM T89697 CIW3M7 70874768 EC50 = 725 nM T89697 CQC35B 70874783 IC50 = 110 nM T89697 C8Q4LJ 70874786 EC50 = 130 nM T89697 CKQ5U7 70874818 IC50 = 1000 nM T89697 CA45OH 70874831 EC50 = 240 nM T89697 C83RQG 70874868 EC50 = 820 nM T89697 CCW4B5 70874889 EC50 = 6700 nM T89697 C2TZ8D 70874895 EC50 = 760 nM T89697 CF1G3K 70874916 IC50 = 200 nM T89697 CPLT90 70874941 EC50 = 230 nM T89697 CJ24YM 70914178 IC50 = 468 nM T89697 CJ80SV 70914181 IC50 = 127000 nM T89697 C30AJI 70914208 IC50 = 50 nM T89697 C7BDH0 70914212 IC50 = 1500 nM T89697 C71AZM 70914219 EC50 = 1300 nM T89697 C2TC8W 70914230 Ki = 5.8 nM T89697 C8V5NF 70914234 EC50 = 220 nM T89697 CP8HI7 70914358 IC50 = 700 nM T89697 CJN0M5 70925897 EC50 = 6100 nM T89697 CNUF17 71458329 IC50 = 47000 nM T89697 CN8Q3X 74221589 IC50 < 100 nM T89697 CTL8X2 75202661 IC50 = 100 nM T89697 C5YFU8 75202920 IC50 = 1000 nM T89697 C6HPF7 75202926 IC50 = 1000 nM T89697 C2D6KV 75203053 IC50 < 100 nM T89697 CVLP16 75203175 IC50 = 100 nM T89697 CQ5LH4 75405939 IC50 = 64 nM T89697 C56YXL 76320783 IC50 = 24.3 nM T89697 C40EJG 76324723 IC50 = 6000 nM T89697 CRT2C5 76327994 IC50 = 451000 nM T89697 C1HXJ9 76327995 IC50 = 185 nM T89697 CFT9L1 76334268 IC50 = 1600 nM T89697 C2JYL9 77050772 IC50 = 240 nM T89697 CF9X8G 77050773 IC50 = 240 nM T89697 CXC63V 77952883 EC50 = 1100 nM T89697 CZL45X 78425875 IC50 = 0.5 nM T89697 CT7VC8 84374905 IC50 = 3109.3 nM T89697 CGT4O9 85469240 IC50 = 1870 nM T89697 C8T0MJ 85469241 IC50 = 1800 nM T89697 C5SWD9 85469242 IC50 = 590 nM T89697 CA5CG1 85469243 IC50 = 760 nM T89697 C5R6WS 85469292 IC50 = 2960 nM T89697 CWN56M 85626388 IC50 = 4730 nM T89697 C8T0CH 86240712 IC50 > 50000 nM T89697 C1Z2TQ 86240717 IC50 = 1800 nM T89697 CO82UY 86240725 IC50 = 2100 nM T89697 CSGQ82 86240731 IC50 = 54000 nM T89697 CT8SW0 86764097 IC50 = 2400 nM T89697 C1WBQ3 86764098 IC50 = 70 nM T89697 CRL9C7 86764205 IC50 = 120 nM T89697 CI05RT 89052784 IC50 = 20370 nM T89697 CH8JT1 89052953 IC50 = 120000 nM T89697 C7VB9Z 89999091 EC50 = 220 nM T89697 CC32EF 90423425 IC50 < 200 nM T89697 C39EMN 90644514 IC50 > 50000 nM T89697 CPV54D 90644515 IC50 > 50000 nM T89697 C0FH2K 90644516 IC50 > 50000 nM T89697 C7Z5NK 90718185 IC50 = 4 nM T89697 C3Z8YX 91758737 IC50 = 20 nM T89697 C3BXV4 101894468 IC50 = 110 nM T89697 CBF1P2 101894469 IC50 = 4000 nM T89697 CJ19AQ 102128193 Ki = 35 nM T89697 C6AFB0 102128195 Ki = 35 nM T89697 C9VZ4F 117620853 EC50 > 10000 nM T89697 C46AOF 117704863 IC50 < 200 nM T89697 CI0Y8F 117779240 IC50 = 350 nM T89697 CJH1Z4 117800109 IC50 = 5 nM T89697 CP75IE 117927565 IC50 = 661 nM T89697 C7L6SF 117927575 IC50 = 76 nM T89697 CQZI27 117927580 IC50 = 13 nM T89697 C4YE0X 118511968 IC50 = 13000 nM T89697 CUAP64 118511969 IC50 > 50000 nM T89697 CS74VJ 118511985 IC50 = 620 nM T89697 CDP71A 118511986 IC50 = 290 nM T89697 C37OSM 118511993 IC50 > 50000 nM T89697 CKG90Q 118512005 IC50 > 50000 nM T89697 C4SWU1 118512015 IC50 = 1200 nM T89697 CN98IG 118512017 IC50 = 120 nM T89697 C50AFG 118512030 IC50 = 1700 nM T89697 C0MEC2 118512032 IC50 = 46000 nM T89697 C4J7UP 118512042 IC50 = 580 nM T89697 C41XHC 118512043 IC50 = 490 nM T89697 C4Z8QL 118512052 IC50 = 8000 nM T89697 CJ6B7A 118512054 IC50 = 2200 nM T89697 CM1DS2 118512060 IC50 > 50000 nM T89697 CPT8K5 118512063 IC50 = 4600 nM T89697 CPFQ23 118512079 IC50 = 3400 nM T89697 CEK8O4 118512091 IC50 = 1700 nM T89697 C8IUD4 118569598 IC50 < 1000 nM T89697 CMRV56 118706416 IC50 = 80 nM T89697 CK9GQ7 118706833 IC50 = 43 nM T89697 CG1A3O 118706834 IC50 = 59 nM T89697 C32BDE 118706835 EC50 = 296 nM T89697 C4Z8XI 118706836 EC50 = 1171 nM T89697 C0IHA8 118706837 IC50 = 254 nM T89697 C2T8ZF 118706838 EC50 = 1393 nM T89697 CHE7P0 118706839 EC50 = 181 nM T89697 CFU73S 118706840 EC50 = 142 nM T89697 CD5YM8 118706841 EC50 = 85 nM T89697 C9KME7 118706842 IC50 = 122 nM T89697 C5O2BI 118706843 IC50 = 255 nM T89697 CT6L3M 118706844 EC50 = 2494 nM T89697 CNMZ08 118706845 EC50 = 2588 nM T89697 C2FN6H 118706846 EC50 = 187 nM T89697 COU9T3 118706847 EC50 = 130 nM T89697 CU40NV 118706848 EC50 = 84 nM T89697 CG9B5A 118706849 EC50 = 2229 nM T89697 C5Q3DP 118706850 IC50 = 608 nM T89697 C2GLY9 118706851 IC50 = 247 nM T89697 C9G8WM 118706944 EC50 = 508 nM T89697 CHQV01 118706945 EC50 = 374 nM T89697 CW2HM0 118706946 EC50 = 134 nM T89697 CTB7D6 118706947 EC50 = 465 nM T89697 COZV69 118706948 EC50 = 187 nM T89697 CTF8K6 118706949 EC50 = 183 nM T89697 CK5W7Z 118706950 IC50 = 125 nM T89697 CT87ZE 118706951 EC50 = 172 nM T89697 C1REB5 118706952 IC50 = 4055 nM T89697 C26LNH 118708818 IC50 = 84000 nM T89697 CV8M5E 118716422 IC50 = 18000 nM T89697 CD08UQ 118716423 IC50 > 100000 nM T89697 C0NHP3 118716424 IC50 > 100000 nM T89697 C0LN8P 118716425 IC50 > 100000 nM T89697 CYI8E6 118716426 IC50 > 100000 nM T89697 CMX5F2 118716427 IC50 = 24000 nM T89697 CT9HZ8 118716428 IC50 = 56000 nM T89697 CIOK68 118716429 IC50 = 8100 nM T89697 C1OMC9 118716430 IC50 = 5500 nM T89697 C0TA6G 118716431 IC50 > 100000 nM T89697 CHOC51 118716432 IC50 = 3500 nM T89697 CA6NH1 118716433 IC50 = 1900 nM T89697 C0M2FU 118716434 IC50 = 3600 nM T89697 CV7DW6 118716435 IC50 = 220 nM T89697 C41QXJ 118716436 IC50 = 750 nM T89697 CF16UH 118716437 IC50 = 1800 nM T89697 CDK5J0 118716438 IC50 = 120 nM T89697 CW3HZ6 118716439 IC50 = 160 nM T89697 C6AI5J 118716440 IC50 = 190 nM T89697 C8YUR0 118716441 IC50 = 77 nM T89697 CI0CN3 118720652 IC50 = 1300 nM T89697 CRH1D8 121332565 IC50 > 1000 nM T89697 C3BMW5 121332569 IC50 = 50 nM T89697 CK82EH 121332589 IC50 = 830 nM T89697 CU6JL0 121332595 IC50 = 690 nM T89697 C65ZYO 121332604 IC50 = 22 nM T89697 CK4W2N 121332617 IC50 = 250 nM T89697 C6CTF1 121332626 IC50 = 540 nM T89697 C5YS9V 121332627 IC50 = 160 nM T89697 CZ2TG3 121332650 IC50 = 1800 nM T89697 CNMK19 121332652 IC50 = 330 nM T89697 C92NOH 121332654 IC50 = 100 nM T89697 CF2Y4A 121332661 IC50 = 790 nM T89697 C5CH7A 121332672 IC50 = 2900 nM T89697 C2Z9YC 121332674 IC50 = 280 nM T89697 CF1C2J 121332677 IC50 = 340 nM T89697 CDL5N6 121332679 IC50 = 1000 nM T89697 C0O2WL 121332691 IC50 = 62 nM T89697 CN0UL6 121332697 IC50 = 2100 nM T89697 CB5LH6 121332700 IC50 = 570 nM T89697 C96RZJ 121332707 IC50 = 1800 nM T89697 CRG82W 121332712 IC50 = 840 nM T89697 CLD6W9 121332721 IC50 = 2600 nM T89697 CNBH32 121332727 IC50 = 49 nM T89697 C0M1TY 121332731 IC50 = 1500 nM T89697 C2EQP8 121332773 IC50 = 50 nM T89697 CMP01Q 121354659 IC50 = 5 nM T89697 C8GXR1 121469000 IC50 = 42 nM T89697 CFQ9P6 121469056 IC50 = 159 nM T89697 C7J0RI 121469136 IC50 = 348 nM T89697 C7OQU1 121469151 IC50 = 14 nM T89697 CW7N8S 121469162 IC50 = 504 nM T89697 CND02B 121469183 IC50 = 45 nM T89697 CJ85LD 121469184 IC50 = 23 nM T89697 C9Q0TD 121469223 IC50 > 1000 nM T89697 CX3Q8C 121469247 IC50 = 600 nM T89697 CS6PA4 121469296 IC50 > 1000 nM T89697 CUP95H 121474590 IC50 > 1000 nM T89697 CSF24O 122193552 IC50 = 3163 nM T89697 C25XGV 122193553 IC50 > 10000 nM T89697 CV30GB 122193590 IC50 = 1242 nM T89697 C4RSB3 122193591 IC50 = 2323 nM T89697 C4N9HG 122193592 IC50 = 977 nM T89697 C8A0DL 122193593 IC50 = 1928 nM T89697 CR27QH 122193594 IC50 = 602 nM T89697 CXY02W 122193595 IC50 = 936 nM T89697 CJ6RO8 122193596 IC50 = 640 nM T89697 CL7S4T 122193597 IC50 = 1097 nM T89697 CCL63T 122193598 IC50 = 982 nM T89697 CP93QC 122193599 IC50 = 2069 nM T89697 CIDM29 122193600 IC50 = 1593 nM T89697 C2U6VA 122193601 IC50 = 921.8 nM T89697 CPG6T0 122368191 IC50 = 48 nM T89697 CC6VJ5 122525709 IC50 = 180 nM T89697 CY0X9D 122525711 IC50 = 20 nM T89697 CZE79W 122525712 IC50 = 680 nM T89697 C51WNS 122606362 IC50 = 20 nM T89697 CGO29F 122608329 IC50 = 130 nM T89697 CXS30F 122650362 IC50 > 10000 nM T89697 CF9Q1R 122650368 IC50 > 10000 nM T89697 CU2K4P 122650372 IC50 = 26 nM T89697 C3RCU4 122650378 IC50 = 21 nM T89697 C3LY8T 122650476 IC50 = 81 nM T89697 CP9EY1 122650500 IC50 = 167 nM T89697 CN6MK9 122650505 IC50 = 87 nM T89697 CHZY51 122650508 IC50 = 79 nM T89697 CS47AD 122650581 IC50 = 8 nM T89697 C3YM4T 124927661 IC50 = 289.5 nM T89697 CWN4D0 125315466 IC50 = 217000 nM T89697 CGP91U 127026194 IC50 = 77 nM T89697 C1XVD6 127026502 IC50 = 68.1 nM T89697 C86NVH 127026503 EC50 = 231.4 nM T89697 CJL27E 127027129 EC50 = 30.6 nM T89697 CY7SM8 127027130 EC50 = 36.4 nM T89697 CDV03C 127027131 EC50 = 67 nM T89697 C36HFU 127027132 EC50 = 211.5 nM T89697 C9A4RT 127027138 EC50 = 63.1 nM T89697 CY6M9H 127027139 EC50 = 68.4 nM T89697 C8YKZ6 127027140 EC50 = 134.9 nM T89697 CEU96I 127027427 IC50 = 111.8 nM T89697 CG08KV 127028367 IC50 = 10000 nM T89697 CW7A2Q 127028368 IC50 = 10000 nM T89697 C51QDO 127028910 IC50 > 10000 nM T89697 C9QVB4 127036449 EC50 > 10000 nM T89697 CK6SC5 127036625 IC50 = 48000 nM T89697 C1HUY5 127036630 IC50 > 10000 nM T89697 C23XQU 127036787 IC50 = 1139 nM T89697 CQ8U6F 127037839 IC50 = 1100 nM T89697 C7ZC9Q 127037878 EC50 = 67.6 nM T89697 CIA42L 127038189 IC50 = 20000 nM T89697 CIQ15P 127038190 IC50 = 730 nM T89697 C46ISV 127038222 IC50 = 82 nM T89697 CV7FO1 127038232 IC50 = 4600 nM T89697 CX0JH6 127038891 IC50 = 5200 nM T89697 C3YQJ0 127039199 IC50 = 4200 nM T89697 C2S6BH 127039223 IC50 = 1700 nM T89697 C9RB4I 127039229 IC50 = 19000 nM T89697 C9MK6V 127039238 IC50 = 61000 nM T89697 C79HKG 127039239 IC50 = 490 nM T89697 CSG51N 127039240 IC50 = 570 nM T89697 C7T0HM 127039543 IC50 = 55000 nM T89697 CGL2K6 127039550 IC50 = 26000 nM T89697 CV5I4T 127039862 IC50 = 75.8 nM T89697 CS1X3N 127040995 IC50 = 7700 nM T89697 CT4RU6 127041800 IC50 > 10000 nM T89697 CB2S4P 127042503 IC50 < 1000 nM T89697 C3SXY7 127046261 IC50 > 30000 nM T89697 CM4R5A 127046282 IC50 > 30000 nM T89697 C75UNV 127046283 IC50 > 30000 nM T89697 CAHF82 127046284 IC50 > 30000 nM T89697 C6XZ7M 127046780 IC50 > 30000 nM T89697 C6J3PV 127046921 IC50 > 30000 nM T89697 C57UIH 127047228 IC50 = 3500 nM T89697 CDKF67 127047240 IC50 > 30000 nM T89697 CZ4SV2 127047241 IC50 = 3400 nM T89697 C2JTQ3 127047242 IC50 > 30000 nM T89697 C5P4JH 127047325 IC50 = 1500 nM T89697 CHZA26 127047364 IC50 > 30000 nM T89697 CGE49W 127047365 IC50 > 30000 nM T89697 CIX95S 127047490 IC50 > 30000 nM T89697 CE94JR 127047748 IC50 = 6300 nM T89697 CV1X0F 127047886 IC50 = 1700 nM T89697 CM2NL5 127048012 IC50 = 4700 nM T89697 CI38DX 127048013 IC50 = 4900 nM T89697 C7XW2S 127048014 IC50 > 30000 nM T89697 C9L7ZW 127048015 IC50 > 30000 nM T89697 C7F3TB 127048016 IC50 = 2800 nM T89697 C6JZ9N 127048017 IC50 = 3800 nM T89697 CK5C8N 127048018 IC50 = 5400 nM T89697 CJ43QC 127048019 IC50 = 7200 nM T89697 C60WCP 127048119 IC50 = 2100 nM T89697 CY7G4D 129282405 EC50 = 720 nM T89697 CQ97RT 129282436 EC50 = 1400 nM T89697 CL9J8N 129282617 EC50 = 2200 nM T89697 CP09TF 129282671 EC50 = 2900 nM T89697 C42ZDX 129282689 EC50 = 1600 nM T89697 C3GA7K 129282703 EC50 = 4500 nM T89697 CV28YE 129282706 EC50 = 1300 nM T89697 C7LG2X 129282851 EC50 = 20000 nM T89697 C3SGN0 129282870 EC50 = 1400 nM T89697 CU70NI 129282903 EC50 > 25000 nM T89697 C3CH6E 129283030 EC50 = 13000 nM T89697 C7FXS8 129283166 EC50 = 880 nM T89697 C32WDC 129283174 EC50 = 240 nM T89697 C9HZ2S 129283211 EC50 = 4600 nM T89697 C5L7MR 129283737 EC50 = 970 nM T89697 CE19JM 129296385 EC50 = 800 nM T89697 C56BAE 129296459 EC50 > 25000 nM T89697 COU73Q 132528948 IC50 = 5300 nM T89697 CDMH46 132606955 IC50 = 560 nM T89697 CNX3D4 134130983 Ki = 35 nM T89697 CCX46W 134131669 Ki = 35 nM T89697 C0KX5B 134132343 Ki = 35 nM T89697 C95RJQ 134132658 Ki = 35 nM T89697 CC47DZ 134132888 Ki = 35 nM T89697 CCS0M6 134133190 Ki = 35 nM T89697 C5UM0A 134135015 Ki = 35 nM T89697 CPR5A4 134136354 Ki = 35 nM T89697 C46MUG 134136717 Ki = 35 nM T89697 CQZB67 134137635 Ki = 35 nM T89697 C8QOD7 134138847 Ki = 35 nM T89697 CNE10R 134139474 Ki = 35 nM T89697 CVB51Y 134141021 Ki = 35 nM T89697 C2QL6D 134142610 Ki = 35 nM T89697 CQD8V6 134142830 Ki = 35 nM T89697 C0HKW5 134143335 Ki = 35 nM T89697 CV5XQ0 134143523 Ki = 35 nM T89697 C4KDS5 134145910 Ki = 35 nM T89697 C2HJ8Z 134146158 Ki = 35 nM T89697 C8D9KR 134146460 Ki = 35 nM T89697 CZ73SH 134147587 Ki = 35 nM T89697 CSUE71 134149657 Ki = 35 nM T89697 CH3C9P 134150058 Ki = 35 nM T89697 CI69YJ 134150572 Ki = 35 nM T89697 CB87LJ 134152033 Ki = 35 nM T89697 CS8W4E 134153755 Ki = 35 nM T89697 CM62BZ 134154095 Ki = 35 nM T89697 C15WLQ 134154247 Ki = 35 nM T89697 C9WQ6T 134155013 Ki = 35 nM T89697 CH7CX3 134155058 Ki = 35 nM T89697 CIV1X4 134156014 Ki = 35 nM T89697 CCP20Z 134156288 Ki = 35 nM T89697 CA6C5U 134157947 Ki = 35 nM T89697 C9ZEJ4 134462563 IC50 = 568 nM T89697 CO1YD8 135401349 IC50 > 30000 nM T89697 CCJ85U 135412567 IC50 = 1240 nM T89697 CPK9A8 135420064 IC50 = 8600 nM T89697 CFWY62 135424939 IC50 = 1500 nM T89697 CG81PH 135424940 IC50 = 270 nM T89697 CDC15J 135424941 IC50 = 19 nM T89697 CUK07Z 135424945 IC50 = 6800 nM T89697 C3P7VU 135424946 IC50 = 970 nM T89697 CB9Q2N 135424953 IC50 = 14 nM T89697 CY20NS 135424981 IC50 = 14 nM T89697 CIT4U8 135437626 IC50 > 30000 nM T89697 CVQ6I5 135442567 IC50 = 2850 nM T89697 C9L3NY 135465938 IC50 = 21100 nM T89697 CHI9L5 135472487 IC50 > 30000 nM T89697 CWV63H 135478380 IC50 = 10300 nM T89697 CXE5S3 135482065 IC50 = 1700 nM T89697 CRYK71 135491081 IC50 = 11300 nM T89697 C0A5WI 135510775 IC50 = 73 nM T89697 CNY13I 135510784 IC50 = 54 nM T89697 CEU6N4 135533698 IC50 > 30000 nM T89697 CW5LN1 135533790 IC50 = 2100 nM T89697 CKT9M6 135567420 IC50 = 2.8 nM T89697 CI2GV6 135588554 IC50 > 30000 nM T89697 CZJ24D 135588681 IC50 = 4800 nM T89697 CXD4W7 135611181 IC50 = 6000 nM T89697 CS0DA5 135741412 IC50 = 10 nM T89697 CASN86 135743630 IC50 > 100000 nM T89697 CK7RW0 135821912 IC50 > 30000 nM T89697 CF95ES 135895369 IC50 = 100 nM T89697 CO56EF 135895372 IC50 = 120 nM T89697 CA2M7V 135899518 Ki = 367000 nM T89697 C7H3IM 135905429 IC50 = 100 nM T89697 C7Y0PK 135936842 IC50 = 2100 nM T89697 C9KHP8 135981331 IC50 = 53 nM T89697 CDH36U 136036203 Ki = 197000 nM T89697 C2L6CP 136099973 IC50 = 280 nM T89697 CU13NF 136123535 IC50 = 7000 nM T89697 C98DMB 136898218 IC50 = 98 nM T89697 C9V1YI 137223162 IC50 = 12 nM T89697 CW2RC3 137245067 IC50 = 35 nM T89697 CNGL30 137250365 IC50 = 17.9 nM T89697 C7EJZ4 137297236 IC50 = 16 nM T89697 CO32JA 137297260 IC50 = 52 nM T89697 C15UNK 137297264 IC50 = 373 nM T89697 CU34ZO 137297270 IC50 = 23070 nM T89697 C8VQ9X 137297286 IC50 > 10000 nM T89697 CVDH54 137297313 IC50 = 2748 nM T89697 CX7L0Y 137297324 IC50 = 2094 nM T89697 CWCD40 137297341 IC50 = 26 nM T89697 C1ARX6 137297350 IC50 = 26 nM T89697 C31AZO 137297358 IC50 = 20 nM T89697 C4SM2V 137297442 IC50 = 853 nM T89697 CZ7MF4 137297447 IC50 = 18 nM T89697 CQM4I6 137297497 IC50 = 1235 nM T89697 CL5Q1S 137386090 IC50 = 151.5 nM T89697 C5LPK1 137386135 IC50 = 55.7 nM T89697 CX8ZD9 137386139 IC50 = 14.4 nM T89697 CY73OP 137386143 IC50 = 17.1 nM T89697 CO5SY2 137386223 IC50 = 18.8 nM T89697 CKHW29 137386229 IC50 = 35.6 nM T89697 C2A3WV 137386236 IC50 = 251 nM T89697 CJ73IG 137390209 EC50 = 420 nM T89697 CA5OY1 137628667 EC50 = 410 nM T89697 C4HJU2 137631563 IC50 = 23000 nM T89697 CB3RA0 137632598 IC50 = 366000 nM T89697 CK5TL4 137634430 EC50 = 15310 nM T89697 CMU1O6 137634654 IC50 > 5000 nM T89697 CK8A9L 137637814 IC50 = 5255 nM T89697 C85QBH 137639169 IC50 = 47000 nM T89697 C4JM6K 137639484 IC50 = 9784 nM T89697 C2B3NF 137640065 IC50 = 22 nM T89697 CXJH24 137640336 IC50 = 6000 nM T89697 C8RVQ3 137641068 IC50 = 9700 nM T89697 CGL56P 137643600 IC50 = 41000 nM T89697 CY6R3Q 137647941 IC50 = 210 nM T89697 CQ5G4T 137650989 IC50 = 100 nM T89697 C0K9MI 137651594 EC50 = 17540 nM T89697 CFQ2V0 137655049 IC50 = 4500 nM T89697 CI8A1Y 137655874 IC50 = 2400 nM T89697 C46BDF 137657792 IC50 = 172000 nM T89697 COED37 137661429 IC50 = 27600 nM T89697 C96QPV 137662004 IC50 = 87 nM T89697 CQ89OP 138737778 IC50 = 230 nM T89697 CZHY27 138737927 IC50 = 15 nM T89697 C1WFB4 138737941 IC50 = 9.3 nM T89697 C39POY 139507046 IC50 = 14 nM T89697 CD29IP 139507088 IC50 = 21 nM T89697 CEFG75 141483091 IC50 = 14560 nM T89697 C5L2QN 141483093 IC50 = 99940 nM T89697 C3GQC2 141483094 IC50 = 31820 nM T89697 CKY6N8 141483096 IC50 = 6400 nM T89697 CRT49I 141483097 IC50 = 80780 nM T89697 C7LPO8 141483098 IC50 > 100000 nM T89697 CB0GA4 141483099 IC50 = 28490 nM T89697 CHA20C 141483100 IC50 > 100000 nM T89697 CH60KW 141501915 IC50 = 50900 nM T89697 CV91LK 141501916 IC50 = 74390 nM T89697 CBE81C 141501917 IC50 = 39040 nM T89697 CCJV28 141501918 IC50 = 14980 nM T89697 C69RFM 141501919 IC50 = 64470 nM T89697 C81KPZ 141501920 IC50 = 22720 nM T89697 CCN50V 141501921 IC50 = 25930 nM T89697 CA1YE4 141501922 IC50 = 95070 nM T89697 CS9OX0 141501923 IC50 = 53930 nM T89697 C5HW7N 141501924 IC50 = 69440 nM T89697 CNL6A2 141501925 IC50 = 840 nM T89697 CF41KS 141501926 IC50 = 33100 nM T89697 C8BVO4 141501927 IC50 = 21930 nM T89697 CI90SH 141501931 IC50 = 77540 nM T89697 CZ6E1A 141501932 IC50 = 60560 nM T89697 CX7K2H 141514151 IC50 = 260.3 nM T89697 C7XGA5 141744794 IC50 > 10000 nM T89697 C5W6QL 141744795 IC50 = 250 nM T89697 CS0VF4 141744796 IC50 = 6780 nM T89697 CEF7Q9 141744797 IC50 > 10000 nM T89697 CS1N8K 141744798 IC50 > 10000 nM T89697 CRK06D 141744799 IC50 = 4840 nM T89697 C78ELY 141744800 IC50 = 9600 nM T89697 C03BNS 141744801 IC50 = 78 nM T89697 CDV98B 141744802 IC50 = 160 nM T89697 CY1CJ9 141744803 IC50 > 10000 nM T89697 CX37LU 141744804 IC50 > 10000 nM T89697 C3A8DH 141744805 IC50 > 10000 nM T89697 CDAP21 141744806 IC50 = 6110 nM T89697 C8VTK2 141744807 IC50 = 630 nM T89697 CJB0H5 141744808 IC50 = 240 nM T89697 C4LW7Q 141744809 IC50 = 2090 nM T89697 C7LA5F 141744810 IC50 = 8190 nM T89697 CLUM57 141744811 IC50 > 10000 nM T89697 CAM31S 141744813 IC50 > 10000 nM T89697 CMKN19 141744814 IC50 > 10000 nM T89697 CU2Q6E 141744815 IC50 > 10000 nM T89697 C9YT2N 141744816 IC50 > 10000 nM T89697 C9KVZ4 141744817 IC50 = 74 nM T89697 C78GZL 141744818 IC50 = 97 nM T89697 C7JYI3 141744820 IC50 = 82 nM T89697 C0EDU6 141744821 IC50 = 8270 nM T89697 CGO28U 141744823 IC50 = 3210 nM T89697 CE5O2V 141744824 IC50 > 10000 nM T89697 CB8X5H 141744825 IC50 = 1510 nM T89697 C7Q2WE 141744826 IC50 = 3540 nM T89697 C37XEL 141744827 IC50 > 10000 nM T89697 CVOP58 141744828 IC50 = 450 nM T89697 CC17LW 141744829 IC50 > 10000 nM T89697 CWNS62 141744830 IC50 > 10000 nM T89697 CR5B2L 141744831 IC50 = 950 nM T89697 C8V9BA 141744832 IC50 > 10000 nM T89697 CVK4X8 141744833 IC50 > 10000 nM T89697 CU7VO6 141744834 IC50 = 69 nM T89697 CVF1I5 141744835 IC50 = 680 nM T89697 CYKD76 141744836 IC50 = 90 nM T89697 CEC19U 141744837 IC50 > 10000 nM T89697 C2AT5E 141744838 IC50 > 10000 nM T89697 C9INH5 141744839 IC50 > 10000 nM T89697 CEBS63 141744841 IC50 > 10000 nM T89697 CQMU70 141744842 IC50 > 10000 nM T89697 CW1JR2 141744843 IC50 = 46 nM T89697 C0VD7G 141744844 IC50 > 10000 nM T89697 CL8XN3 141744845 IC50 = 2530 nM T89697 CFP60C 141744846 IC50 > 10000 nM T89697 C96KQW 141744848 IC50 > 10000 nM T89697 CRJ3S0 141744849 IC50 = 530 nM T89697 C0EYH1 142341866 IC50 = 13 nM T89697 C6UAR5 142341947 IC50 = 8.1 nM T89697 CKRU13 142341971 IC50 = 16 nM T89697 CKDT74 142341993 IC50 = 84 nM T89697 CF9N0H 142342024 IC50 = 17 nM T89697 C1JQ0Z 142342046 IC50 = 8.4 nM T89697 CB59EZ 142509480 IC50 = 5.6 nM T89697 C47ERW 142509516 IC50 = 4.3 nM T89697 CTH94V 142509574 IC50 = 21 nM T89697 CZFT65 142509579 IC50 = 66.1 nM T89697 CE9WC7 142509586 IC50 = 16.9 nM T89697 CNQ50X 142509588 IC50 = 4.8 nM T89697 C0S9PQ 142619907 EC50 = 1450 nM T89697 C7JKA2 142619908 EC50 = 10800 nM T89697 CL2AV8 142619909 EC50 = 320 nM T89697 CP1UF7 142619910 EC50 = 6260 nM T89697 CQ8OU6 142619912 EC50 = 4190 nM T89697 C12KDR 142619913 EC50 = 6400 nM T89697 C5H7FG 142619916 EC50 = 6920 nM T89697 CI31ZV 142619918 EC50 = 10700 nM T89697 CM8P4F 142619919 EC50 = 260 nM T89697 CEY1X4 142619920 EC50 = 11000 nM T89697 CH2E7P 142619921 EC50 = 1040 nM T89697 C1CEU5 142619922 EC50 = 18700 nM T89697 CZ9IW2 142619923 IC50 = 1600 nM T89697 CYB27V 142619924 EC50 = 890 nM T89697 C67QGT 142619926 EC50 = 4590 nM T89697 C3LOW2 142619927 EC50 = 5550 nM T89697 CWEC07 142619928 EC50 = 12000 nM T89697 CLU62H 142619929 EC50 = 4560 nM T89697 C5GJ8V 142619931 EC50 = 480 nM T89697 C16SVH 142619932 EC50 = 9120 nM T89697 C9U3KI 142619933 EC50 = 9470 nM T89697 C6NQ9I 145720956 IC50 = 14000 nM T89697 CO40MZ 145951275 EC50 = 5010 nM T89697 C8XCW4 145953593 EC50 = 4290 nM T89697 C5H4UJ 145954041 IC50 = 18 nM T89697 C09ZQS 145954548 IC50 = 1.8 nM T89697 CV6HZ0 145959475 EC50 = 3090 nM T89697 C96GIW 145964069 IC50 = 450 nM T89697 CA7B3R 145964241 IC50 = 200 nM T89697 C9HKR1 145964500 IC50 = 76580 nM T89697 CUA2K5 145964731 IC50 = 580 nM T89697 CT20SR 145965635 IC50 = 60880 nM T89697 CN6SK2 145965768 IC50 = 80580 nM T89697 CK23NR 145966752 IC50 = 5030 nM T89697 CAP6W8 145966837 IC50 = 28 nM T89697 CE5I7C 145967008 IC50 = 65920 nM T89697 CSQJ42 145967348 IC50 = 97 nM T89697 CYN5V8 145967463 IC50 = 58110 nM T89697 CBJ3P1 145967730 IC50 = 2200 nM T89697 C65NHX 145968756 IC50 = 1200 nM T89697 CQ21PR 145968804 IC50 = 4200 nM T89697 C4EZN1 145969081 IC50 = 2200 nM T89697 CPNZ97 145969599 IC50 = 810 nM T89697 CCG1P0 145969967 IC50 = 5700 nM T89697 CLY2T3 145970519 IC50 = 690 nM T89697 C6K9GW 145971318 IC50 = 66730 nM T89697 C2VBX5 145972107 IC50 = 10200 nM T89697 CS5TW7 145973304 IC50 = 82120 nM T89697 CAK60H 145973431 IC50 = 630 nM T89697 CU6KO4 145973699 IC50 = 405 nM T89697 CNV36S 145974038 IC50 = 22730 nM T89697 C0W2XY 145974378 IC50 = 730 nM T89697 CV6Y2O 145976341 IC50 = 20680 nM T89697 CS1O9L 145976459 IC50 = 49340 nM T89697 CSV9N2 145976739 IC50 = 870 nM T89697 CLI94M 145978059 IC50 = 71700 nM T89697 CHWK59 145978347 IC50 = 340 nM T89697 CZW46Y 145978425 IC50 > 1000 nM T89697 CG4M5X 145979054 IC50 = 27 nM T89697 C5SK4O 145979193 IC50 = 209.6 nM T89697 C8CXN2 145979858 EC50 = 480 nM T89697 CRYW71 145980148 IC50 = 2200 nM T89697 C3UG5E 145980172 IC50 = 207.9 nM T89697 CX35HL 145980717 IC50 = 8330 nM T89697 C1IGW2 145980819 IC50 > 100000 nM T89697 CS4MI8 145981708 IC50 = 9500 nM T89697 CW8B6A 145981750 IC50 = 22 nM T89697 C3X8OD 145981785 IC50 = 151.8 nM T89697 CV1RQ9 145981894 EC50 = 330 nM T89697 C7S9MG 145982245 IC50 = 233.7 nM T89697 C2YO8R 145982459 IC50 = 4100 nM T89697 CHT8M1 145982739 IC50 = 87 nM T89697 C9VS3X 145982780 IC50 = 7 nM T89697 CC7ZF9 145982970 IC50 = 394 nM T89697 CHN2M6 145982993 IC50 = 390 nM T89697 CCLP04 145983079 IC50 = 23 nM T89697 C4AKU1 145983122 IC50 = 119 nM T89697 CG02AM 145983180 IC50 = 597.8 nM T89697 C2NH0Y 145983235 IC50 = 39 nM T89697 CPR1W2 145983299 IC50 = 148 nM T89697 CQF57C 145983500 IC50 = 288 nM T89697 C50ZIQ 145984327 IC50 = 448 nM T89697 CH1X5E 145984494 IC50 = 361 nM T89697 C5U2QK 145984896 IC50 = 122.5 nM T89697 CJC34M 145984936 IC50 = 134 nM T89697 C69OSL 145985132 IC50 = 299 nM T89697 C2O7XA 145985324 IC50 = 1192 nM T89697 C4TBS0 145985331 IC50 = 438 nM T89697 CF3ME9 145985603 IC50 = 427 nM T89697 CP09AH 145985633 IC50 > 100000 nM T89697 CKJ8O3 145985919 IC50 = 420 nM T89697 CK0MI7 145985929 IC50 = 50 nM T89697 CM81NX 145986030 IC50 = 117 nM T89697 C3QCS5 145986385 IC50 = 133 nM T89697 CT71UQ 145986568 IC50 = 890 nM T89697 CEJR90 145986692 IC50 = 11000 nM T89697 CJ3TE7 145986756 IC50 = 119.6 nM T89697 C3P0BK 145986889 IC50 = 1100 nM T89697 C05UPF 145987627 IC50 = 18 nM T89697 CGT41S 145987994 EC50 = 460 nM T89697 CH8S9C 145988339 IC50 = 50300 nM T89697 C02ART 145988358 IC50 = 18 nM T89697 CFRN35 145988434 IC50 = 167.9 nM T89697 CDGV74 145988791 IC50 = 1500 nM T89697 CL05NY 145989048 IC50 = 2800 nM T89697 CHJD48 145989519 IC50 = 1580 nM T89697 C29ITB 145989650 IC50 = 338 nM T89697 CI8WB3 145989715 IC50 = 4000 nM T89697 CQ7JU8 145989915 IC50 = 7800 nM T89697 CLK52R 145990092 IC50 = 113.4 nM T89697 CB15WE 145990300 IC50 = 42200 nM T89697 C13KCJ 145990635 IC50 = 2250 nM T89697 CVN6T9 145990888 IC50 = 13590 nM T89697 CKU2L4 145991209 IC50 = 139.8 nM T89697 CX7J2S 145991557 IC50 = 134 nM T89697 CV9DX7 145991568 IC50 = 684 nM T89697 CV61QH 145991788 IC50 = 577.2 nM T89697 CB0ZR4 145992186 IC50 = 3300 nM T89697 C2L0NS 145992195 IC50 = 2700 nM T89697 CJC82P 145993052 IC50 = 61 nM T89697 CYQ79U 145993068 IC50 = 11000 nM T89697 CNWY78 145993645 IC50 = 1950 nM T89697 CR6XN8 145994164 IC50 = 590 nM T89697 CD4WA8 145994224 IC50 = 450 nM T89697 C3SY9B 146018670 IC50 = 16.4 nM T89697 C31MCG 146018671 IC50 = 102.1 nM T89697 C6EF3U 146633829 IC50 = 6.4 nM T89697 C9CH8X 146634682 IC50 = 12.4 nM T89697 C8J3TV 146669430 IC50 = 740 nM T89697 CHE6V5 148026225 IC50 = 12 nM T89697 C1I7JK 148270333 IC50 = 12 nM T89697 C20YQK 153434844 IC50 = 19 nM T89697 CJM43I 153434859 IC50 = 13 nM T89697 C36ISR 153434865 IC50 = 10 nM T89697 CZ7JQ2 153434882 IC50 = 12 nM T89697 C63FMQ 154601093 IC50 = 21 nM T89697 C59HOL 155510561 IC50 > 200 nM T89697 C4JB1R 155511259 IC50 = 70 nM T89697 CF3V7Y 155511297 IC50 = 150 nM T89697 CZT0W5 155511328 IC50 > 1000 nM T89697 CLWA53 155511337 IC50 = 358 nM T89697 C7PTI6 155511361 IC50 = 23000 nM T89697 C6ED7O 155511708 IC50 = 27.6 nM T89697 CX5QS1 155511756 IC50 = 7.6 nM T89697 CWDH25 155511770 IC50 = 18.9 nM T89697 CX04BL 155512330 IC50 = 7200 nM T89697 CHD3C4 155512917 IC50 > 10000 nM T89697 CAG5F0 155513388 IC50 = 1760 nM T89697 CRYM58 155513720 IC50 = 43800 nM T89697 C8VD2I 155513747 IC50 = 781 nM T89697 CHP5L0 155514083 IC50 = 2890 nM T89697 C16XWD 155514212 IC50 = 45.7 nM T89697 CV32TF 155514242 IC50 = 126 nM T89697 CYFW59 155514258 IC50 = 1090 nM T89697 C3CD4X 155514316 IC50 = 3350 nM T89697 CNUW02 155514339 IC50 = 37.2 nM T89697 CX4JQ3 155514783 IC50 = 132 nM T89697 C0G6CR 155515087 IC50 = 14 nM T89697 CES90B 155515098 IC50 = 571 nM T89697 C7LFA0 155515243 IC50 = 457 nM T89697 C1FTN9 155515411 IC50 > 1000 nM T89697 C0H6ZE 155515556 IC50 = 36.9 nM T89697 CCJ14L 155516448 IC50 = 14 nM T89697 CVP8Q5 155516616 IC50 = 16.8 nM T89697 CI4LE2 155516619 IC50 = 28.7 nM T89697 CWJS36 155516630 IC50 = 4.5 nM T89697 CNJ47R 155516651 IC50 = 636 nM T89697 CJ0FH7 155516689 IC50 = 6740 nM T89697 C7IBH0 155516857 IC50 = 657 nM T89697 C4NC7Q 155517508 IC50 = 19.1 nM T89697 CN46XW 155517655 IC50 = 2220 nM T89697 C34RQN 155518507 IC50 = 1094 nM T89697 CJA45U 155518566 IC50 = 1260 nM T89697 CGCO97 155518865 IC50 = 22.2 nM T89697 C9T7MC 155519004 IC50 = 17.9 nM T89697 C8W6QP 155519650 IC50 > 10000 nM T89697 CIW3F0 155519816 IC50 = 72 nM T89697 CO1DT2 155520102 IC50 = 822.5 nM T89697 CH9XP5 155520130 IC50 = 341 nM T89697 C2F6OX 155520170 IC50 = 7150 nM T89697 CZ57XQ 155520612 IC50 = 767 nM T89697 C3ZP5H 155521897 IC50 = 17000 nM T89697 CZ8FN1 155522016 IC50 = 21.4 nM T89697 C4BLS9 155522057 IC50 = 99.4 nM T89697 CTL2I9 155522175 IC50 = 477 nM T89697 C8FS1P 155523075 IC50 = 259 nM T89697 C6B4EL 155523872 IC50 = 24 nM T89697 CRJ9O3 155524304 IC50 = 24 nM T89697 CMDH32 155524514 IC50 = 119 nM T89697 C4PW8J 155524534 IC50 = 14500 nM T89697 CLY12I 155525014 IC50 = 14700 nM T89697 CZK57D 155525299 IC50 = 21 nM T89697 CA01HU 155525338 IC50 = 74.5 nM T89697 CHZD38 155525566 IC50 = 14.4 nM T89697 CY1I6V 155525573 IC50 = 284 nM T89697 CLY5M4 155525580 IC50 = 501.6 nM T89697 CQ3W2E 155525624 IC50 = 3195.3 nM T89697 CC1R5A 155525641 IC50 = 72.9 nM T89697 C3EJR0 155525993 IC50 = 36 nM T89697 C27HXG 155526119 IC50 = 696 nM T89697 C8E5PM 155526671 IC50 = 73.9 nM T89697 CH4KS8 155526712 IC50 = 42 nM T89697 C8TWV7 155527273 IC50 = 338.8 nM T89697 C6VK2Q 155527721 IC50 = 107.4 nM T89697 CCH6I4 155528124 IC50 = 104 nM T89697 C5FW7I 155528311 IC50 = 461 nM T89697 C4LCP3 155528885 IC50 = 44 nM T89697 CA30OB 155529610 IC50 = 44 nM T89697 CZ39JY 155529671 IC50 = 96870 nM T89697 CU3K9S 155529868 IC50 = 94 nM T89697 C13JBA 155530161 IC50 = 148 nM T89697 CYX4D6 155530375 IC50 > 1000 nM T89697 C5X7DV 155530398 IC50 = 35 nM T89697 CYBZ42 155530883 IC50 = 100000 nM T89697 C58PHY 155531191 IC50 = 33 nM T89697 CF5N2S 155531195 IC50 = 3870 nM T89697 CCWU58 155531250 IC50 = 150 nM T89697 CHQ8N5 155531385 IC50 = 2830 nM T89697 CCR71O 155531812 IC50 = 134 nM T89697 C3CVZ1 155532036 IC50 = 73 nM T89697 C5A8MO 155532280 IC50 = 96870 nM T89697 CAQ2Y8 155532641 IC50 = 105000 nM T89697 C3F6ZI 155532803 IC50 = 1281.3 nM T89697 CXS20Z 155532816 IC50 = 418 nM T89697 C70XJB 155533149 IC50 = 21000 nM T89697 CG1K4V 155533289 IC50 = 8000 nM T89697 C7OEH8 155533973 IC50 > 1000 nM T89697 C86BTK 155536043 IC50 = 407 nM T89697 C4H8XB 155536067 IC50 = 20.8 nM T89697 CJVZ35 155536135 IC50 = 10100 nM T89697 C9X7LC 155536325 IC50 = 23 nM T89697 C0O4AQ 155536365 IC50 = 870 nM T89697 CC80FB 155536449 IC50 = 27300 nM T89697 C6RJ2I 155537896 IC50 = 19.2 nM T89697 CXC91A 155538594 IC50 = 817 nM T89697 C0HXA8 155538715 IC50 = 764 nM T89697 CR6EJ3 155539196 IC50 = 25 nM T89697 CFKI70 155539267 IC50 = 10.1 nM T89697 CJ5FY6 155539290 IC50 = 52.7 nM T89697 CR8EP5 155539904 IC50 = 45 nM T89697 CQT17I 155540569 IC50 = 36.3 nM T89697 CJYR81 155540830 IC50 = 29.5 nM T89697 C58KYQ 155540941 IC50 = 2.5 nM T89697 CD3Y5U 155540952 IC50 = 590 nM T89697 CPKO04 155541165 IC50 = 7.4 nM T89697 C4C6RX 155541201 IC50 = 113 nM T89697 CFOQ59 155541414 IC50 = 218.8 nM T89697 CK01YF 155541436 IC50 = 24 nM T89697 C9TJ2I 155541446 IC50 = 112 nM T89697 CP5R8Z 155541668 IC50 = 850 nM T89697 CF3AW0 155541799 IC50 = 1730 nM T89697 CP25JB 155542022 IC50 = 151 nM T89697 CLC81R 155542366 IC50 = 8.7 nM T89697 C02NAK 155542721 IC50 = 691 nM T89697 C94KJF 155543368 IC50 = 217 nM T89697 CKN39Q 155544466 IC50 = 399 nM T89697 CIUK86 155544692 IC50 = 26 nM T89697 CI9O0P 155544755 IC50 = 143 nM T89697 CZAL46 155545224 IC50 = 9 nM T89697 C1Z5EA 155545364 IC50 = 44.9 nM T89697 CHN82B 155546259 IC50 > 1000 nM T89697 CNPU01 155546283 IC50 = 2741 nM T89697 CE04JU 155546342 IC50 = 327 nM T89697 C0OC8M 155547213 IC50 = 322 nM T89697 C0C8FP 155547279 IC50 = 9.6 nM T89697 CN03BT 155547734 IC50 = 7.1 nM T89697 CMH35W 155547809 IC50 = 3.3 nM T89697 CWX19H 155548140 IC50 = 6.6 nM T89697 C9J2RI 155548653 IC50 = 306 nM T89697 C8C3SW 155548933 IC50 = 180 nM T89697 CYD57L 155549229 IC50 > 1000 nM T89697 CGZ2A8 155549756 IC50 = 539 nM T89697 C3NX1M 155549772 IC50 > 200 nM T89697 CH96DK 155550037 IC50 = 2480 nM T89697 C6O7LQ 155550877 IC50 > 10000 nM T89697 C2GSR8 155550907 IC50 = 969 nM T89697 C6JV3E 155551216 EC50 = 690 nM T89697 CSU75P 155551311 IC50 = 22 nM T89697 CNU93S 155551336 IC50 = 7.8 nM T89697 C20NJG 155551633 IC50 = 73.2 nM T89697 C3YG1T 155551998 EC50 = 4200 nM T89697 CX5NG6 155552179 IC50 = 51.7 nM T89697 CN46IF 155552796 IC50 = 35.7 nM T89697 CE95UF 155552938 IC50 = 3360 nM T89697 C8M1QG 155553198 IC50 = 939 nM T89697 C0ASJ7 155553201 EC50 = 2600 nM T89697 C12IJV 155553541 EC50 = 24000 nM T89697 C20SOV 155554077 IC50 > 10000 nM T89697 CQ7BU3 155554221 IC50 = 5.7 nM T89697 C6U9KC 155555102 IC50 = 7153.3 nM T89697 CQ6D7M 155555581 IC50 = 19 nM T89697 C6HNU8 155555675 IC50 = 102 nM T89697 C6DKG1 155555719 IC50 = 75 nM T89697 C86QJW 155556390 IC50 = 10.5 nM T89697 CA3KH1 155556529 IC50 = 4.6 nM T89697 C63AHT 155557140 IC50 > 1000 nM T89697 C0XC9H 155557271 IC50 = 223 nM T89697 CO7P3Z 155557740 IC50 = 933 nM T89697 CI0V8G 155558434 IC50 = 1072.1 nM T89697 C4RWF1 155558731 IC50 = 27 nM T89697 C1TIH7 155558824 IC50 = 33 nM T89697 C5QB1Y 155558872 IC50 = 304 nM T89697 CBYL12 155559016 IC50 = 1910 nM T89697 CU8L5V 155559057 IC50 = 4 nM T89697 CJ82RN 155559113 IC50 = 55.8 nM T89697 CZ14NM 155559275 EC50 = 340 nM T89697 CNJ4C7 155559429 IC50 > 1000 nM T89697 CQY4A1 155560339 IC50 = 743.9 nM T89697 CA48WP 155560350 IC50 = 24000 nM T89697 C6R2SJ 155560411 IC50 = 58350 nM T89697 C7ZPV4 155560705 IC50 = 354 nM T89697 CQIT48 155560791 IC50 = 3814 nM T89697 CQT16B 155561274 IC50 = 14.6 nM T89697 CEK9J1 155561942 IC50 = 10.1 nM T89697 C25KBO 155562131 IC50 = 357 nM T89697 CFX43K 155562566 IC50 = 19 nM T89697 C3NDJ2 155562711 IC50 = 1090 nM T89697 CSQ8U0 155562797 IC50 = 2734 nM T89697 CF5G4Y 155563108 IC50 > 200 nM T89697 CB4E0U 155563312 IC50 = 38.1 nM T89697 CC7P0V 155563603 IC50 = 20.3 nM T89697 CXMP83 155564029 IC50 > 1000 nM T89697 C4MJ7U 155564599 IC50 = 19.5 nM T89697 CG02FV 155564613 IC50 = 1990 nM T89697 C2C7EU 155564852 IC50 = 255.5 nM T89697 CP19JR 155564990 IC50 = 8.5 nM T89697 CXM8P9 155565017 IC50 = 1020 nM T89697 C83WCP 155565053 IC50 > 1000 nM T89697 CG43BS 155565222 IC50 = 2200 nM T89697 CFP34M 155565482 IC50 = 5623 nM T89697 CP5Y9H 155566146 IC50 = 110000 nM T89697 CNX9T1 155566545 IC50 = 138 nM T89697 CY5LV8 155566655 IC50 = 7.5 nM T89697 CEA02R 155566797 IC50 = 37.1 nM T89697 C61SEH 155567075 IC50 = 1210 nM T89697 CFN2U7 155567243 IC50 = 413 nM T89697 CN91VH 155567244 IC50 = 221 nM T89697 CI0D1N 155567338 IC50 = 855 nM T89697 C07ASO 155567542 IC50 = 3563 nM T89697 CO58ME 155567694 EC50 = 10000 nM T89697 CB19FR 155567818 IC50 = 62.5 nM T89697 C2O8RC 155568012 IC50 = 1430 nM T89697 CW45BT 155568279 IC50 = 4.2 nM T89697 CAH57R 155569047 IC50 > 10000 nM T89697 C6OA1Z 155569140 IC50 = 258 nM T89697 CU3Y0S 155569235 IC50 = 5.1 nM T89697 CSB45Q 155569293 EC50 = 670 nM T89697 D00BGN 24971326 IC50 = 5300 nM T89697 D00GYX 7509 IC50 = 1700 nM T89697 D00UIK 17937479 IC50 = 2500 nM T89697 D00XOT 45487214 IC50 = 12500 nM T89697 D01CSZ 44466195 IC50 = 15000 nM T89697 D01HST 1085108 IC50 = 3000 nM T89697 D02ADV 594397 IC50 = 1000000 nM T89697 D02DRL 199161 IC50 = 4800 nM T89697 D02IVJ 2803022 IC50 = 2000 nM T89697 D02SRL 3000729 IC50 = 4000 nM T89697 D02XRG 45487209 IC50 = 50000 nM T89697 D03ETX 44406807 Ki = 13220 nM T89697 D03JAE 12465608 IC50 = 800 nM T89697 D03JMD 49866094 IC50 = 2600 nM T89697 D04OXY 16871 IC50 = 720 nM T89697 D05AFW 49866090 IC50 = 16000 nM T89697 D05LFV 12526770 IC50 = 6800 nM T89697 D06MUL 44406804 Ki = 17150 nM T89697 D06OUR 44466196 IC50 = 3000 nM T89697 D06YFT 676159 IC50 = 78 nM T89697 D07NSZ 13266247 IC50 = 1400 nM T89697 D07NYX 7222 IC50 = 652000 nM T89697 D08GZK 24856337 Ki = 80 nM T89697 D08MOG 45487171 IC50 = 3500 nM T89697 D08MRL 45487219 IC50 = 4500 nM T89697 D08PIF 80407 IC50 = 1400 nM T89697 D08XXD 17815 IC50 = 6000 nM T89697 D08YGW 10444038 IC50 = 32000 nM T89697 D08YHA 72734 IC50 = 214 nM T89697 D09BVH 11305 IC50 = 10000 nM T89697 D09DSZ 3266369 IC50 = 7000 nM T89697 D09JOM 15945669 IC50 = 400 nM T89697 D09ZJW 80409 IC50 = 1100 nM T89697 D0A7NH 45487176 IC50 = 15000 nM T89697 D0B9IA 16091658 Ki = 140 nM T89697 D0DB2N 16059787 Ki = 690 nM T89697 D0DQ6Z 8530 IC50 = 460 nM T89697 D0FO2B 1923 IC50 = 750000 nM T89697 D0G0EE 24971327 Ki = 5300 nM T89697 D0G8IH 20029042 IC50 = 12500 nM T89697 D0GJ7J 3760 IC50 = 23000 nM T89697 D0H0HM 135411931 IC50 = 2560 nM T89697 D0I2RW 8342 IC50 = 280 nM T89697 D0I9AT 73549 IC50 = 53.7 nM T89697 D0J9DD 69590 Ki = 4400 nM T89697 D0K3SZ 78252 IC50 = 1300 nM T89697 D0K4MG 21609882 Ki = 2300 nM T89697 D0MC4U 16066751 Ki = 41 nM T89697 D0N1ZJ 44465947 IC50 = 4000 nM T89697 D0NI8W 10307884 IC50 = 1200 nM T89697 D0O3IE 137153 IC50 = 8900 nM T89697 D0O9QG 68342 IC50 = 2200 nM T89697 D0P1CO 2830968 IC50 = 7300 nM T89697 D0P3XW 580759 IC50 = 1200 nM T89697 D0PR7L 85171 IC50 = 1800 nM T89697 D0Q9JG 13885856 IC50 = 10000 nM T89697 D0R6FJ 64961 Ki = 120 nM T89697 D0S1FF 44465702 IC50 = 2500 nM T89697 D0SZ9F 95756 IC50 = 3500 nM T89697 D0TM0Z 152300 Ki = 190 nM T89697 D0UV8T 9942176 IC50 = 5000 nM T89697 D0V8FG 81062 IC50 = 320000 nM T89697 D0W3ON 416002 IC50 = 3000 nM T89697 D0W3OY 78062 IC50 = 2200 nM T89697 D0W3XP 356405 Ki = 1200 nM T89697 D0W9VA 10667 IC50 = 7100 nM T89697 D0Z0BB 118986 IC50 = 100 nM T89697 D0Z3NE 478573 IC50 = 0.018 nM T89697 D0Z4JG 11074644 IC50 = 5500 nM T22977 CSTX48 12029908 IC50 = 381100 nM T22977 CFCQ32 24823795 IC50 = 365800 nM T22977 CCM1W9 24823796 IC50 = 67900 nM T22977 C78RBD 24823798 IC50 = 786900 nM T22977 CV75UN 24823942 IC50 = 129300 nM T22977 CFG3S8 24970402 IC50 = 56600 nM T22977 CU16PV 34363640 EC50 = 1930 nM T22977 CGCZ64 45102767 EC50 = 67 nM T22977 C0ZCI8 46196578 EC50 = 790 nM T22977 C1S4FQ 46215250 EC50 > 32000 nM T22977 C10GXV 46215251 EC50 = 1470 nM T22977 C2P4ZD 46215255 EC50 = 4700 nM T22977 CUMR17 50993705 EC50 = 170 nM T22977 CD49KF 51003102 IC50 = 96600 nM T22977 CB50PY 51003103 IC50 = 103300 nM T22977 CUQ4H3 53324606 EC50 = 710 nM T22977 C9V4XG 56945435 EC50 = 2880 nM T22977 CPDZ84 56945436 EC50 = 1410 nM T22977 C0Y8TI 56945437 EC50 = 1960 nM T22977 C4YE3U 56945438 EC50 = 720 nM T22977 CBLU36 56945439 EC50 = 870 nM T22977 CM40FZ 56945440 EC50 = 580 nM T22977 C0ZL2B 56945548 EC50 = 1070 nM T22977 CMRJ61 56945549 EC50 = 510 nM T22977 CTGZ70 56945550 EC50 = 1020 nM T22977 C4TK9D 56945551 EC50 = 2840 nM T22977 C0XJU1 56945552 EC50 = 3700 nM T22977 CPB16S 62140981 IC50 = 83120 nM T22977 CS43AO 71459115 IC50 = 71460 nM T22977 CTWB85 71460923 IC50 = 125320 nM T22977 COD7K9 71462627 IC50 = 65980 nM T22977 C2DM8H 71652393 IC50 = 408000 nM T22977 CL7I0C 71652552 IC50 = 178500 nM T22977 C81MVZ 71652554 IC50 = 641000 nM T22977 C47ETO 101519736 IC50 = 58900 nM T22977 CKI9V6 145960712 IC50 > 100000 nM T22977 CQ2D5R 145961082 IC50 = 100000 nM T22977 C6AX9C 145963675 IC50 = 145800 nM T22977 CW2LP6 155518910 IC50 > 100000 nM T22977 C5D3QO 155521025 IC50 > 100000 nM T22977 CQM2B3 155521222 IC50 > 100000 nM T22977 CABH43 155522156 IC50 > 100000 nM T22977 CNH43F 155533839 IC50 > 50000 nM T22977 C8H4CG 155537441 IC50 > 50000 nM T10756 C06BAM 219561 IC50 = 8900 nM T10756 CV5HI2 219565 IC50 = 11000 nM T10756 C8ZR3J 256755 IC50 = 8800 nM T10756 CFWY79 10099159 IC50 = 7000 nM T10756 C3YE9J 10393519 IC50 = 7000 nM T10756 C0QT1V 11758430 IC50 = 14000 nM T10756 CLG8I5 44178850 IC50 > 100 ug.mL-1 T10756 C94LUQ 44178851 IC50 = 38 ug.mL-1 T10756 CN84ZR 45270893 IC50 = 9 ug.mL-1 T10756 C3Z4TA 45271732 IC50 = 4.2 ug.mL-1 T10756 C2W3DX 127038789 IC50 = 5000 nM T10756 CP3W5G 127038790 IC50 = 4200 nM T10756 C6UQ9T 127038791 IC50 = 5300 nM T10756 CX2U4F 127039115 IC50 = 3900 nM T10756 C04WTC 127039117 IC50 = 5400 nM T10756 C08HWM 127040772 IC50 = 14000 nM T10756 CCE90R 127040773 IC50 = 9800 nM T10756 CUST62 127041091 IC50 = 16000 nM T10756 CJ2U3N 127041092 IC50 = 7100 nM T10756 CREI95 127041093 IC50 = 6700 nM T10756 C7UI6S 127041094 IC50 = 8200 nM T10756 CK1Q6H 127041986 IC50 = 38000 nM T10756 C93YZB 127042064 IC50 = 9400 nM T10756 C0AR9E 127042065 IC50 = 3800 nM T10756 C62BOX 127042391 IC50 = 4900 nM T10756 D0F3TM 219564 IC50 = 6900 nM T41702 D0E3TC 44259 IC50 = 7440 nM T41702 CEC30Q 3674 IC50 > 40000 nM T41702 CN64JR 8323 IC50 = 26200 nM T41702 C3YRU7 15295578 IC50 = 250 nM T41702 C2UOE0 24766030 IC50 > 50000 nM T41702 CY8L7E 24896769 IC50 > 10000 nM T41702 CLFM35 25206064 IC50 = 520 nM T41702 CK73NR 44219749 IC50 > 50000 nM T41702 C3VRO9 44557921 IC50 = 9549.93 nM T41702 CCL85F 44575073 IC50 > 50000 nM T41702 CJX06P 44575126 IC50 = 4900 nM T41702 CE8FC7 44575127 IC50 = 11600 nM T41702 C28QLM 44605035 IC50 = 17900 nM T41702 C75XHS 44605037 IC50 > 50000 nM T41702 CC95PQ 45375865 IC50 > 50000 nM T41702 CEOQ27 45375866 IC50 > 50000 nM T41702 C96BNW 46179972 IC50 > 50000 nM T41702 CO3P0J 46866604 IC50 < 50000 nM T41702 CLS29B 46872626 IC50 > 10000 nM T41702 CJOM49 46880136 IC50 = 9510 nM T41702 CV63UL 67240318 IC50 > 10000 nM T41702 C2MD1Q 155513187 IC50 > 10000 nM T41702 D01YWE 25207521 IC50 = 160 nM T41702 D0L4WN 31420 IC50 = 34000 nM T41702 D0Y6OK 6688 IC50 > 40000 nM T89041 D00AXJ 4189 Ki = 243 nM T89041 D02STN 132971 IC50 ~ 1 nM T89041 D06CNP 9821849 IC50 = 18 nM T89041 D07ABV 468595 IC50 = 42 nM T89041 D09GOS 2812 Ki = 81.5 nM T89041 D09LNI 3365 IC50 > 200000 nM T89041 D0AA2D 2378 Ki = 56.5 nM T89041 D0B4IF 456201 IC50 = 1800 nM T89041 D0CA6J 5482 Ki = 505 nM T89041 D0EV8E 3198 Ki = 325 nM T89041 D0M6DO 2145 IC50 = 60000 nM T89041 D0Q9JT 4174 IC50 > 10000 nM T89041 D0ZX1P 59693 IC50 > 5000 nM T89041 D03AJU 44139752 IC50 = 3981.07 nM T89041 D0U0BU 11188409 IC50 = 28.1 nM T89041 D0X3OI 9883029 IC50 = 38 nM T89041 D0SX7F 60876 Ki = 447 nM T89041 C9LCD8 3823 IC50 = 26 nM T89041 CWMQ17 92747 IC50 = 1430 nM T89041 C8EQ1Z 92855 IC50 = 1710 nM T89041 C2GRN7 94199 IC50 = 440 nM T89041 C7VP8E 101966 IC50 = 800 nM T89041 CHWM72 125921 IC50 > 34000 nM T89041 CYSE03 196941 IC50 = 6.13 nM T89041 CUP91R 245872 IC50 = 66 nM T89041 CPE17Q 320374 IC50 = 43900 nM T89041 C7TYH9 585624 IC50 = 18000 nM T89041 CUL8N9 709713 IC50 > 31622.78 nM T89041 C3H1DE 2998104 IC50 = 1600 nM T89041 C1WIR4 4499193 IC50 > 31622.78 nM T89041 CA15IT 9796590 IC50 = 19 nM T89041 CC3QF5 9797875 Ki = 1.9 nM T89041 C9QVL1 9816909 IC50 = 130 nM T89041 C9D4MI 9819290 Ki = 1.4 nM T89041 CRQA29 9830290 IC50 = 28 nM T89041 CKJ1I6 9838340 IC50 = 18 nM T89041 CBZQ79 9840765 Ki = 41 nM T89041 CN9U6I 9840821 Ki = 1.2 nM T89041 CAQ52K 9861918 IC50 = 15 nM T89041 CL2W9Z 9862746 Ki = 1.4 nM T89041 CUK64X 9880846 IC50 = 400 nM T89041 CQHE82 9883170 IC50 = 19 nM T89041 C8YQ6V 9883171 IC50 = 27 nM T89041 C5VA7T 9884336 Ki = 23 nM T89041 CJ56EL 9904146 IC50 = 18 nM T89041 CG0I7C 9905837 IC50 = 39 nM T89041 CUZT98 9906455 IC50 = 75 nM T89041 C4PF5A 9923132 IC50 = 190 nM T89041 CWL3O1 9926844 IC50 = 75 nM T89041 C3TH4Q 9927224 IC50 = 16 nM T89041 C7LSP1 9927786 Ki = 8 nM T89041 C8RPF6 9949067 IC50 = 130 nM T89041 C3IQV6 9965885 IC50 = 29 nM T89041 CO1Z0A 9971194 IC50 = 1.8 nM T89041 CE3L8V 10061454 IC50 = 1100 nM T89041 CG24IZ 10247264 IC50 = 270 nM T89041 CEMU16 10335364 IC50 = 48 nM T89041 C1OA8L 10337109 IC50 = 50 nM T89041 CB7RI8 10358293 IC50 = 490 nM T89041 C5IZ0X 10380012 IC50 = 13 nM T89041 CR0O6C 10447478 IC50 = 2.7 nM T89041 CQWX01 10450499 IC50 = 1000 nM T89041 C3YI0N 10467502 IC50 = 110 nM T89041 C1JC9V 10521065 IC50 = 108 nM T89041 C86HTI 10522113 IC50 = 400 nM T89041 CFK2N9 10543224 IC50 = 970 nM T89041 C4L8OX 10566080 IC50 = 92 nM T89041 CB90LV 10593280 IC50 = 62 nM T89041 C72XUK 10594248 IC50 = 74 nM T89041 C38SOM 10595962 IC50 = 75 nM T89041 C3OY0Q 10636825 IC50 = 820 nM T89041 C3WZ7D 10638951 Ki = 3 nM T89041 C38WKE 10642746 IC50 = 260 nM T89041 C9QN4J 10660816 IC50 = 150 nM T89041 C82HFM 10663232 IC50 = 1250 nM T89041 C0N2BV 10684551 IC50 = 35 nM T89041 C01ZPW 10684552 IC50 = 320 nM T89041 CPS30O 10689427 IC50 = 5 nM T89041 C7U3ZR 10755577 IC50 = 230 nM T89041 CH8T4Y 10758923 IC50 = 2500 nM T89041 C45HMW 10758924 IC50 > 2500 nM T89041 C3AJ4U 10759395 Ki = 8 nM T89041 CIKB07 10806964 IC50 = 21 nM T89041 C94PCN 10826001 IC50 = 460 nM T89041 CN7I8H 10827014 IC50 = 74 nM T89041 CZW6V4 10828130 IC50 = 220 nM T89041 CE23TU 10831118 IC50 = 219 nM T89041 CY34VS 10854385 Ki = 1.9 nM T89041 C58ETU 11002256 Ki = 1.2 nM T89041 CCFU47 11440648 IC50 = 300 nM T89041 CN4T0K 11544009 IC50 = 233 nM T89041 CZ50DQ 11708478 IC50 = 721 nM T89041 CZH43C 11725276 IC50 = 3 nM T89041 C3N4FE 11792279 IC50 = 27 nM T89041 CHLB06 11855878 IC50 = 1250 nM T89041 C96DPL 11855879 IC50 = 915 nM T89041 C7EF1B 11855880 IC50 = 5817.4 nM T89041 C0EPD3 12039019 IC50 = 220 nM T89041 C13GAW 12043371 IC50 = 54 nM T89041 CZJ0B5 12043372 IC50 = 33 nM T89041 C85ZFQ 12043374 IC50 = 28 nM T89041 CF28CA 12074093 IC50 = 22 nM T89041 CJY17R 12074102 IC50 = 36 nM T89041 CJV5G1 12074103 IC50 = 19 nM T89041 CXQI20 12310542 IC50 = 8000 nM T89041 CLSM38 14872624 IC50 = 140000 nM T89041 C39MVQ 15462429 Ki = 23 nM T89041 CC9BE5 17963726 IC50 = 39 nM T89041 CRL9N5 18395624 IC50 = 42 nM T89041 CX6L9A 18395626 IC50 = 24 nM T89041 CK2AJ8 18668528 IC50 = 49 nM T89041 CI3HL4 18668538 IC50 = 40 nM T89041 CCWH59 18668580 IC50 = 36 nM T89041 CW8PF5 18668583 IC50 = 120 nM T89041 C6ADH5 18668593 IC50 = 24 nM T89041 C4-JAN-02 18668607 IC50 = 45 nM T89041 C9V4BO 18668614 IC50 = 44 nM T89041 CY1HK4 18668617 IC50 = 38 nM T89041 CTA76E 18769059 IC50 = 39 nM T89041 C7UKI6 18769065 IC50 = 200 nM T89041 C0LCW3 18769074 IC50 = 160 nM T89041 C8QA0F 18769127 IC50 = 30 nM T89041 CM9NU7 21852976 IC50 = 3950 nM T89041 CKV94G 21879620 IC50 = 13 nM T89041 C2KMV5 21879624 IC50 = 290 nM T89041 C3DT1N 22018410 IC50 = 28 nM T89041 CXMA20 22018425 IC50 = 36 nM T89041 CT24BF 22664964 IC50 = 24 nM T89041 C0F4YM 22737877 IC50 = 46 nM T89041 CZ2BC5 23288050 IC50 = 40 nM T89041 C59VCE 23424811 IC50 = 2880 nM T89041 C5BVZ6 25022443 IC50 = 345 nM T89041 C29WQM 25033651 IC50 > 10000 nM T89041 C1VPF8 25033652 IC50 = 423 nM T89041 CDR34P 25033653 IC50 = 2346 nM T89041 CE0L8C 25033655 IC50 > 5000 nM T89041 C9Q8ZK 25033657 IC50 > 5000 nM T89041 CWIC10 25033659 IC50 = 307 nM T89041 C32QBZ 25033661 IC50 > 20000 nM T89041 CAI47X 25033725 IC50 = 163 nM T89041 C1XW6O 25033727 IC50 = 144 nM T89041 C23EWR 25033729 IC50 > 20000 nM T89041 CW5A1U 25033730 IC50 = 587 nM T89041 CV49HP 25033731 IC50 > 5000 nM T89041 CJHY97 25033732 IC50 > 20000 nM T89041 C86AIT 25033734 IC50 > 5000 nM T89041 CEJ89P 25033804 IC50 = 188 nM T89041 C3UF1V 25033806 IC50 = 233 nM T89041 CF46OB 25033808 IC50 = 1222 nM T89041 CBI59C 25033810 IC50 = 64 nM T89041 CZPW03 25034656 IC50 > 20000 nM T89041 C7KAR1 25034657 IC50 = 333 nM T89041 CZX08M 25142015 Ki = 54 nM T89041 C0XHA2 25180109 IC50 = 316.23 nM T89041 C1HYO5 40513267 IC50 = 430 nM T89041 CV3Y2B 42642720 IC50 = 90 nM T89041 C9AQ7N 42642721 IC50 = 52 nM T89041 C6GR3F 42642761 IC50 = 379 nM T89041 CQ5M2Z 42642929 IC50 = 261 nM T89041 C2D1MN 42642930 IC50 = 217 nM T89041 CD4OQ8 42643273 IC50 > 5000 nM T89041 CO7YV0 42643327 IC50 = 188 nM T89041 C6UR8G 44315168 IC50 = 3810 nM T89041 C4F5JS 44315175 IC50 = 562 nM T89041 C0B2KL 44315318 IC50 = 1400 nM T89041 C9OPM6 44315319 IC50 = 2600 nM T89041 CO1N3V 44315442 IC50 = 3700 nM T89041 CYKB02 44315468 IC50 = 660.25 nM T89041 C0A4LF 44315469 IC50 = 178.2 nM T89041 CD4VR0 44315540 IC50 = 616.5 nM T89041 CM0ZU4 44315606 IC50 = 225 nM T89041 CY76KC 44315613 IC50 = 500 nM T89041 C5SN0H 44340248 IC50 = 59 nM T89041 CC2E3X 44340275 IC50 = 400 nM T89041 C4PJ1H 44340350 IC50 = 58 nM T89041 CA6B2U 44340378 IC50 = 400 nM T89041 CRW68V 44340379 IC50 = 1113 nM T89041 C5HZX0 44340405 IC50 = 150 nM T89041 CN2DW3 44340421 IC50 = 150 nM T89041 CEGT92 44340434 IC50 > 30000 nM T89041 CECD15 44340462 IC50 = 400 nM T89041 CX9HV5 44340476 IC50 = 1200 nM T89041 CM6PF7 44340585 IC50 = 400 nM T89041 CJ0DG8 44340586 IC50 = 150 nM T89041 C03ATJ 44340924 IC50 = 150 nM T89041 C03EXH 44340925 IC50 = 150 nM T89041 CO8XJ3 44354706 IC50 = 5 nM T89041 C7YDP6 44354757 IC50 = 6 nM T89041 C1W6IR 44354758 IC50 = 9 nM T89041 C4AXM5 44354773 IC50 = 270 nM T89041 CZN1X8 44354907 IC50 = 15 nM T89041 CN8M5U 44354930 IC50 = 88 nM T89041 CCA28Y 44354942 IC50 = 35 nM T89041 CNRO38 44354943 IC50 = 10 nM T89041 CQIP34 44354944 IC50 = 670 nM T89041 CO1W4F 44355172 IC50 = 14 nM T89041 CX2R3P 44355187 IC50 > 1000 nM T89041 CCF7G1 44355188 IC50 = 38 nM T89041 CD4S9E 44357420 IC50 = 1770 nM T89041 CKO6B3 44357421 IC50 = 240 nM T89041 CL2I0F 44357429 IC50 = 510 nM T89041 CZ5VG2 44357431 IC50 = 6480 nM T89041 CU1BG7 44357482 IC50 = 35000 nM T89041 C2WAV8 44357582 IC50 = 720 nM T89041 CJ06LT 44357609 IC50 = 230 nM T89041 C6EY7I 44357615 IC50 = 750 nM T89041 CCN6B1 44357617 IC50 = 890 nM T89041 CO1F8W 44357623 IC50 = 190 nM T89041 CJE4I1 44357624 IC50 = 750 nM T89041 CLZM23 44358638 IC50 > 2500 nM T89041 C64IWU 44358640 Ki = 6 nM T89041 C0SX7B 44358689 IC50 > 25000 nM T89041 CJM80V 44358932 IC50 = 1800 nM T89041 CV5HF6 44367009 IC50 = 27 nM T89041 C4D7ZY 44456181 IC50 = 263 nM T89041 C8VI7P 44456221 IC50 = 236 nM T89041 C6JHB5 44456224 IC50 = 584 nM T89041 C1E8RI 44461114 IC50 = 2.9 nM T89041 CIM9D1 44461115 IC50 > 10000 nM T89041 CQ8MP7 44461136 IC50 = 5.6 nM T89041 C5VF2C 44461174 IC50 = 23 nM T89041 C6RV0L 44461240 IC50 = 160 nM T89041 CY7OD4 44461241 IC50 = 3 nM T89041 CECX12 44461375 IC50 > 10000 nM T89041 CAW3I8 44461376 IC50 = 1.8 nM T89041 CK58SI 44461377 IC50 = 2.5 nM T89041 C2QVD9 44586763 IC50 = 2200 nM T89041 C31AFB 44586764 IC50 = 1700 nM T89041 C1A6IL 44586765 IC50 > 5000 nM T89041 C1TFP5 44586766 IC50 = 3800 nM T89041 CB30QW 44586793 IC50 = 1300 nM T89041 CT38XH 44586824 IC50 > 5000 nM T89041 C4VU2E 44586825 IC50 = 756 nM T89041 CYR4O7 44586826 IC50 > 5000 nM T89041 CH0Y5Z 44586865 IC50 = 168 nM T89041 C7W9EK 44586866 IC50 = 118 nM T89041 CUCM51 44587269 IC50 = 460 nM T89041 CIU9Z3 44587270 IC50 = 1050 nM T89041 C1M6TX 44587293 IC50 > 5000 nM T89041 CH28TE 44587294 IC50 > 5000 nM T89041 CNOG06 44587313 IC50 = 670 nM T89041 C6JSU2 44587318 IC50 = 3100 nM T89041 C7Q6UK 44587319 IC50 > 5000 nM T89041 COM7P5 44587320 IC50 > 5000 nM T89041 C24XTP 44587322 IC50 > 5000 nM T89041 CWF4V8 44587323 IC50 > 5000 nM T89041 CUV83E 46854605 IC50 = 56 nM T89041 CIA08B 46854608 IC50 = 37 nM T89041 C3NO7G 46854609 IC50 = 1458 nM T89041 C0NIH6 46854610 IC50 = 493 nM T89041 C78THB 46854611 IC50 = 852 nM T89041 COVL29 46854757 IC50 > 10000 nM T89041 CWJ3F1 46854758 IC50 = 38 nM T89041 CKRQ67 46854759 IC50 = 75 nM T89041 CZ1YJ0 46854760 IC50 = 62 nM T89041 C9UO5G 46901439 IC50 > 5000 nM T89041 C8LQX7 46901612 IC50 > 5000 nM T89041 CN5G2X 46901617 IC50 = 3340 nM T89041 CC25UL 46901778 IC50 = 1370 nM T89041 C7Y0PC 46901779 IC50 > 10000 nM T89041 CHNF30 46901780 IC50 > 10000 nM T89041 CIC9S5 49799473 IC50 = 75 nM T89041 C9W8HK 49863993 IC50 > 10000 nM T89041 CYMO96 49864179 IC50 > 5000 nM T89041 CNBU93 50994740 IC50 = 19 nM T89041 C6RD7G 53249084 IC50 = 26 nM T89041 CP31IL 53319749 IC50 = 38 nM T89041 C6HPO5 53323744 IC50 = 270 nM T89041 CAE25J 53763992 IC50 = 15 nM T89041 C60LIJ 54580449 IC50 = 22 nM T89041 C8V9GW 54582428 IC50 = 150 nM T89041 C7LHV1 54583409 IC50 = 21 nM T89041 CAO9B4 54584364 IC50 = 77 nM T89041 CAK7Z9 54585325 IC50 = 160 nM T89041 CS51ZD 54585326 IC50 = 340 nM T89041 CSV1M4 54586281 IC50 = 26 nM T89041 C01JOU 54586320 IC50 = 92 nM T89041 C9FBH0 54586321 IC50 = 240 nM T89041 C4N0WL 56645363 IC50 > 10000 nM T89041 C57NSZ 56645568 IC50 > 10000 nM T89041 C6PUX9 56645570 IC50 > 10000 nM T89041 CTW6K2 56645571 IC50 > 10000 nM T89041 CA3VO0 56949328 IC50 = 19 nM T89041 CBMY17 56952125 IC50 = 8 nM T89041 C4EPA7 56952126 IC50 = 37 nM T89041 CDL64H 56952128 IC50 = 396 nM T89041 CX1TL3 56952129 IC50 = 361 nM T89041 C7ND1A 56952239 IC50 = 674 nM T89041 CD94CU 56952242 IC50 = 797 nM T89041 C4R3KU 56952244 IC50 = 135 nM T89041 CNXD75 56952346 IC50 = 330 nM T89041 CQ0IA7 56952348 IC50 = 405 nM T89041 CIO9C5 56953325 IC50 = 8 nM T89041 CEW8L6 56953509 IC50 = 656 nM T89041 C4B1EA 56953512 IC50 = 758 nM T89041 CZG03U 56953601 IC50 = 11 nM T89041 CB1FO5 56953605 IC50 = 40 nM T89041 CONW20 56953606 IC50 = 5.8 nM T89041 C1K2YU 56968076 IC50 = 180 nM T89041 C6ATQ0 57390715 IC50 = 88 nM T89041 CD7M5V 57397795 IC50 = 410 nM T89041 CY97BO 57402969 IC50 = 5.5 nM T89041 C2TUJ7 58255382 IC50 = 2880 nM T89041 C3DPC0 58255407 IC50 > 5000 nM T89041 C9DK1X 58255415 IC50 > 10000 nM T89041 CRQ70M 58255438 IC50 = 1550 nM T89041 CP6RA9 58255482 IC50 > 10000 nM T89041 CW71EO 58255581 IC50 > 10000 nM T89041 CB7N8A 60195126 IC50 > 5000 nM T89041 CX4N0I 62707515 IC50 > 10000 nM T89041 C0G3LA 66559847 IC50 > 10000 nM T89041 C4RSI6 66559935 IC50 > 10000 nM T89041 CDX7I8 66559936 IC50 > 10000 nM T89041 CF9EQ5 66559939 IC50 > 10000 nM T89041 CQN6D3 66559940 IC50 > 10000 nM T89041 CN4H8G 66559941 IC50 > 10000 nM T89041 CTP6Q4 66559942 IC50 > 10000 nM T89041 C9EGW2 66575742 IC50 > 10000 nM T89041 CMXA10 66575743 IC50 > 10000 nM T89041 CKWB91 66575744 IC50 > 10000 nM T89041 C7I3MW 66575745 IC50 > 10000 nM T89041 CPN17S 66575746 IC50 > 10000 nM T89041 CG0ZA7 66575747 IC50 > 10000 nM T89041 C6HF0U 66575748 IC50 > 10000 nM T89041 CDI93T 66575817 IC50 > 10000 nM T89041 CBP6I7 66576773 IC50 > 10000 nM T89041 C4NYB0 66576930 IC50 > 10000 nM T89041 C3LP5H 66576931 IC50 > 10000 nM T89041 CE03WG 66576932 IC50 > 10000 nM T89041 C9DP3R 66850314 IC50 = 25900 nM T89041 C97BGW 69093249 IC50 = 940 nM T89041 CZC4E1 69093450 IC50 = 170 nM T89041 C7ZX9P 69281312 IC50 = 570 nM T89041 C7PY1Q 69281314 IC50 = 74 nM T89041 C1VMF2 70977969 IC50 > 10000 nM T89041 CLR3Q2 71452704 IC50 = 280 nM T89041 CI6B9U 71454429 Ki = 8 nM T89041 CC01FB 71454470 IC50 = 199 nM T89041 CG1CQ6 71454483 IC50 > 2500 nM T89041 C70TUP 71455138 IC50 > 10000 nM T89041 C70ARH 71456230 IC50 = 970 nM T89041 CFG4L5 71456934 IC50 > 10000 nM T89041 CX4U8V 71459926 IC50 = 1520 nM T89041 C0SU7M 71461598 IC50 = 1520 nM T89041 C7XIS4 71461624 IC50 = 430 nM T89041 C58SMB 71574941 IC50 = 260 nM T89041 CC09FQ 71574942 IC50 = 1346 nM T89041 CA2T5L 71574943 IC50 = 1886 nM T89041 C9MFZ7 71574944 IC50 = 610 nM T89041 CW73OE 71574945 IC50 > 5000 nM T89041 C70NHJ 71574946 IC50 = 1250 nM T89041 CLH83S 71574947 IC50 > 5000 nM T89041 CF71AB 71575030 IC50 > 5000 nM T89041 CCG1S5 71575031 IC50 > 5000 nM T89041 CH9WE7 71575032 IC50 > 5000 nM T89041 CO4ZQ7 71575033 IC50 = 493 nM T89041 CT86GV 71575034 IC50 = 1737 nM T89041 CKPV51 71621803 IC50 = 38000 nM T89041 C56LUJ 71716957 IC50 > 10000 nM T89041 CRP1G5 71733625 IC50 = 122000 nM T89041 C7V2LS 71733626 IC50 = 93700 nM T89041 C3J8DZ 71734667 IC50 = 130000 nM T89041 C48JAU 71735007 IC50 = 132000 nM T89041 CJE01S 71745100 IC50 > 10000 nM T89041 CX0WV5 71817943 IC50 = 64 nM T89041 CN1LU6 71817944 IC50 = 106 nM T89041 CGV4U3 71817945 IC50 = 523 nM T89041 CJ4L5G 71818086 IC50 = 147 nM T89041 COXA51 71818087 IC50 = 375 nM T89041 CP1A3M 71818088 IC50 = 454 nM T89041 CPJ42T 71818089 IC50 = 525 nM T89041 CAP03I 71818090 IC50 = 94 nM T89041 CO23PK 71818091 IC50 = 185 nM T89041 CL4X6A 71818092 IC50 = 11 nM T89041 CL8GK5 71818093 IC50 = 16 nM T89041 C4ZVG0 71818094 IC50 = 294 nM T89041 CH2GR0 71818232 IC50 = 1028 nM T89041 C0VGQ9 71818233 IC50 = 632 nM T89041 C5QRF2 71818234 IC50 = 1520 nM T89041 CCG7R3 72703685 IC50 = 480 nM T89041 CAU4Z0 72703889 IC50 = 2160 nM T89041 C56KEC 72703890 IC50 > 5000 nM T89041 CZB6E9 73345904 IC50 = 206 nM T89041 C5TD1Y 76335179 IC50 = 1800 nM T89041 C1YJW0 77846787 IC50 = 67 nM T89041 CV73PD 77846790 IC50 = 9 nM T89041 C0DIH7 77846872 IC50 = 15 nM T89041 COI25M 77846873 IC50 = 7 nM T89041 CJI8R0 77846875 IC50 = 8 nM T89041 CZK4J1 77846962 IC50 = 9 nM T89041 CEK89G 77846963 IC50 = 19 nM T89041 C5BA8Z 77846964 IC50 = 11 nM T89041 C4D6XJ 77847803 IC50 = 0.73 nM T89041 CF7O4Q 77847804 IC50 = 12 nM T89041 C3RHG9 85468997 IC50 = 480 nM T89041 CZH2O5 87178837 IC50 = 258000 nM T89041 CL30TR 89471870 IC50 > 10000 nM T89041 C3BUS8 89471889 IC50 > 10000 nM T89041 CI7HY8 89471890 IC50 = 5700 nM T89041 CX0M7B 89961716 IC50 = 84 nM T89041 CR5D6Y 89961785 IC50 > 10000 nM T89041 C89TEU 89968659 IC50 > 10000 nM T89041 CY5IC7 90252834 IC50 > 10000 nM T89041 C84NVA 90252850 IC50 > 10000 nM T89041 CBY46O 90252851 IC50 > 10000 nM T89041 CNVA50 90252852 IC50 > 10000 nM T89041 C89BFG 90333640 IC50 = 3.7 nM T89041 C0YK1U 90656806 IC50 = 310 nM T89041 CWE0X5 90656807 IC50 > 4000 nM T89041 CQS8C9 91664365 IC50 = 2 nM T89041 CLB2E7 91827654 IC50 > 10000 nM T89041 CN5ZQ2 117629963 IC50 > 15000 nM T89041 CJ9Z0S 118496546 IC50 > 10000 nM T89041 CJ54UQ 118618017 IC50 = 21 nM T89041 C7FT2M 118691578 IC50 = 22.8 nM T89041 CZD9X8 118691599 IC50 = 15.5 nM T89041 CDHI10 118733086 IC50 > 10000 nM T89041 C18PWB 118733087 IC50 > 10000 nM T89041 C8WJ2Y 118733088 IC50 > 10000 nM T89041 C31ZXP 118733089 IC50 > 10000 nM T89041 CHR84E 118733090 IC50 > 10000 nM T89041 CAQ72M 118733091 IC50 > 10000 nM T89041 CIV1Z5 118733092 IC50 > 10000 nM T89041 CU3Y9W 118733093 IC50 > 10000 nM T89041 CF49NU 118733094 IC50 > 10000 nM T89041 CK73VU 118733095 IC50 > 10000 nM T89041 CR1WU5 118733096 IC50 > 10000 nM T89041 CK7Y2L 118858329 IC50 = 230 nM T89041 CK09QT 118858331 IC50 = 12.4 nM T89041 C4CB3G 118867913 IC50 = 39000 nM T89041 CFND03 121481824 IC50 = 1 nM T89041 CO48UI 121481829 IC50 = 5 nM T89041 CM71FR 121481838 IC50 = 1 nM T89041 C48QHN 121481842 IC50 = 6.2 nM T89041 CMJB40 121481843 IC50 = 5 nM T89041 CMP69L 121481849 IC50 = 5 nM T89041 C02XEN 121481855 IC50 = 5 nM T89041 CRP3W8 121481856 IC50 = 5 nM T89041 CTE53N 121481871 IC50 = 17 nM T89041 C1GI5N 121481873 IC50 = 86 nM T89041 CYD80P 121481874 IC50 = 100 nM T89041 CX1FE7 121481875 IC50 = 39 nM T89041 C4XF6C 121481880 IC50 = 117 nM T89041 CBGY79 121481882 IC50 = 1200 nM T89041 CGA71F 121481885 IC50 = 42 nM T89041 C29AKG 121481886 IC50 = 5 nM T89041 C2NWZ7 121481888 IC50 = 180 nM T89041 C8IZ9B 121481891 IC50 = 2500 nM T89041 C8XO3C 121481900 IC50 = 58 nM T89041 C7SOX9 122439257 IC50 = 24 nM T89041 C15NCI 122439267 IC50 = 4.6 nM T89041 CP3K5Z 122439268 IC50 = 21 nM T89041 CX4T7L 122439274 IC50 = 5 nM T89041 CT9E7N 122439276 IC50 = 17 nM T89041 CSI91Y 122439277 IC50 = 18 nM T89041 C8EG3B 122439285 IC50 = 5 nM T89041 C80OLS 122462854 IC50 > 31622.78 nM T89041 C15JTL 122462980 IC50 > 31622.78 nM T89041 CUF8C5 126761305 IC50 = 7.83 nM T89041 C2ZFR8 127027572 IC50 > 10000 nM T89041 CV1BD6 127027573 IC50 > 10000 nM T89041 CQO36B 127028499 IC50 = 6600 nM T89041 CN42BR 127028817 IC50 > 10000 nM T89041 C49IME 127031799 IC50 = 4800 nM T89041 C6U0PW 127031978 IC50 = 5 nM T89041 C7EV5P 127031979 IC50 = 2 nM T89041 C6T5VG 127031980 IC50 = 5 nM T89041 CD1NK7 127031981 IC50 = 4 nM T89041 CX05HP 127032282 IC50 = 5 nM T89041 CP4WZ3 127033243 IC50 = 4 nM T89041 CNJW13 127034300 IC50 = 3 nM T89041 C2EO9D 129811602 IC50 > 20000 nM T89041 C74WZM 131748940 IC50 = 42 nM T89041 CH3V9Q 134139925 IC50 > 10000 nM T89041 C4DLP3 136029154 IC50 = 5900 nM T89041 CAV9U3 136219390 IC50 = 910 nM T89041 CC7LY3 136239517 IC50 = 550 nM T89041 C2V0IM 136244612 IC50 > 5000 nM T89041 CYIF59 136245971 IC50 > 5000 nM T89041 CG91VC 137633656 IC50 = 24.3 nM T89041 C4ALG0 137635843 IC50 = 20.1 nM T89041 C6Y8VD 137636260 IC50 = 45 nM T89041 CH2SR6 137636922 IC50 = 23.7 nM T89041 C6MJU7 137653906 IC50 = 45.4 nM T89041 CL45EH 137658689 IC50 = 29 nM T89041 C0ROV3 145961601 IC50 = 5 nM T89041 C63WHT 145961979 IC50 = 6 nM T89041 CVR84G 145962556 IC50 = 5 nM T89041 COPL56 145962564 IC50 = 5 nM T89041 CGP0Z7 145963339 IC50 = 34 nM T89041 CK71RV 145963932 IC50 > 31622.78 nM T89041 C74HIS 145965339 IC50 = 7.2 nM T89041 C9G2OD 145974857 IC50 = 16.5 nM T89041 CMW1H3 155544953 IC50 > 15000 nM T89041 D00DSE 49864196 IC50 = 386 nM T89041 D00IUN 25099145 IC50 = 953 nM T89041 D00YHD 46854449 IC50 = 783 nM T89041 D00ZME 9861000 IC50 = 4 nM T89041 D01REI 46901610 IC50 = 52 nM T89041 D01SZX 46867545 IC50 = 880 nM T89041 D02BXS 46901445 IC50 = 337 nM T89041 D03EDD 10593052 Ki = 41 nM T89041 D03EXD 49864181 IC50 = 248 nM T89041 D04CFP 46901927 IC50 = 760 nM T89041 D04ISG 11680597 IC50 = 27 nM T89041 D04SHY 42642719 IC50 = 195 nM T89041 D05LXA 44587266 IC50 = 310 nM T89041 D05PKT 46901928 IC50 = 2000 nM T89041 D06AKB 49864180 IC50 = 4040 nM T89041 D07CTI 10853186 IC50 = 130 nM T89041 D07IQG 10473365 IC50 = 42 nM T89041 D07VGT 46901929 IC50 = 438 nM T89041 D08FAB 11845485 IC50 = 3000 nM T89041 D08YCD 10354661 IC50 = 910 nM T89041 D09GEH 44587233 IC50 = 450 nM T89041 D09GJI 44586828 IC50 = 99 nM T89041 D09VQZ 46901616 IC50 = 598 nM T89041 D0B9XL 25099144 IC50 = 373 nM T89041 D0E0ZS 46901613 IC50 = 876 nM T89041 D0GJ7J 3760 Ki = 610 nM T89041 D0I1YH 46901446 IC50 = 97 nM T89041 D0J4VA 46854606 IC50 = 343 nM T89041 D0JE1I 9815923 IC50 > 19952.62 nM T89041 D0K5KG 6540050 IC50 = 1085 nM T89041 D0L6HY 20298212 IC50 = 2300 nM T89041 D0LJ9D 46901783 IC50 = 647 nM T89041 D0M8JE 13416469 IC50 = 780 nM T89041 D0MM7G 18976090 IC50 = 388 nM T89041 D0N1GH 11601068 IC50 = 686 nM T89041 D0N1PQ 11506923 IC50 = 667 nM T89041 D0N7CQ 42642718 IC50 = 152 nM T89041 D0P5CT 46901614 IC50 = 1790 nM T89041 D0Q0BK 46901611 IC50 = 186 nM T89041 D0Q1FX 42642717 IC50 = 164 nM T89041 D0Q1LG 44587267 IC50 = 300 nM T89041 D0RD3C 44587268 IC50 = 2100 nM T89041 D0RI7T 44586827 IC50 = 1400 nM T89041 D0SM4F 42642716 IC50 = 231 nM T89041 D0SP7S 5995 IC50 = 56 nM T89041 D0SU0Y 44587265 IC50 = 580 nM T89041 D0T1CH 46901440 IC50 = 1610 nM T89041 D0U5GF 18976091 IC50 = 282 nM T89041 D0U6JI 46854448 IC50 = 189 nM T89041 D0WN9P 46901444 IC50 = 226 nM T89041 D0X1DV 44587321 IC50 = 2000 nM T89041 D0Y5KX 46901443 IC50 = 408 nM T89041 D0Z3GX 46901784 IC50 = 577 nM T76522 CCYB38 206441 Ki = 22500 nM T76522 C4MRT6 16193817 IC50 > 10000 nM T76522 CKXV20 53434646 Ki = 125000 nM T76522 CM0CB3 71385905 Ki = 24000 nM T76522 CI5PJ9 71400937 Ki = 68100 nM T76522 CV7YP6 90655688 Ki = 105000 nM T76522 CKV18N 134146743 IC50 > 10000 nM T74307 D09KTS 24821094 IC50 = 0.23 nM T74307 D02TUL 118115473 IC50 = 19000 nM T74307 D08AOZ 86582336 IC50 = 23 nM T74307 D08UUL 46700756 IC50 = 4409 nM T74307 D0E3TC 44259 IC50 = 1.07 nM T74307 D0G5XV 135565884 IC50 = 1.13 nM T74307 D0H9FR 118295624 IC50 = 371 nM T74307 D0O6WV 24794418 IC50 > 500 nM T74307 D0YB3W 156414 IC50 = 29 nM T74307 D03BNU 59604787 IC50 > 10000 nM T74307 D09HEV 6539952 IC50 = 46 nM T74307 D0T3ME 156422 IC50 > 30000 nM T74307 CB7WK3 5938113 IC50 = 8800 nM T74307 CBOP58 11293798 Ki > 10000 nM T74307 C26BZX 11362471 Ki > 10000 nM T74307 CWXB93 11397177 Ki > 10000 nM T74307 C0APW4 11422034 IC50 = 10000 nM T74307 CTG83F 11539329 Ki > 1500 nM T74307 CMIL86 11590363 Ki > 1500 nM T74307 C9T6SC 11640926 Ki > 1500 nM T74307 CU0E8O 11690457 Ki > 10000 nM T74307 CB0AP2 11705863 Ki > 10000 nM T74307 CZY05V 11719421 IC50 = 1320 nM T74307 CP7AH3 11755812 IC50 = 50000 nM T74307 CFPW41 16007116 Ki > 1400 nM T74307 C9TU1O 16046126 IC50 > 1000 nM T74307 CQNP54 24764449 IC50 = 519 nM T74307 C3VRO9 44557921 IC50 > 10000 nM T74307 CY3HW5 46224684 IC50 = 8300 nM T74307 CLS29B 46872626 IC50 > 10000 nM T74307 C2O8RZ 46886323 IC50 = 320 nM T74307 C8NA4L 53384644 IC50 > 30000 nM T74307 CE1A9V 57394653 IC50 = 16 nM T74307 CI50KU 58167984 IC50 = 959 nM T74307 C1MR8Q 60097495 IC50 > 10000 nM T74307 CV63UL 67240318 IC50 > 10000 nM T74307 C7VJ6A 70647728 IC50 = 20 nM T74307 COU73Y 71226944 IC50 = 9 nM T74307 C40JOZ 71235465 IC50 = 78 nM T74307 CKT60L 71455860 Ki > 1400 nM T74307 CEV53L 71548006 IC50 = 32 nM T74307 C1SR5V 71576693 IC50 = 377 nM T74307 C4X1CP 71748056 IC50 = 366 nM T74307 CZM1K4 71765510 IC50 = 36 nM T74307 CKO8S6 71815907 IC50 = 339 nM T74307 CF6QG1 73602845 IC50 = 191 nM T74307 CDN83F 73707530 IC50 = 30.2 nM T74307 CCQN01 73775788 IC50 = 250 nM T74307 CHF08G 73775789 IC50 = 1130 nM T74307 COL37D 73775921 IC50 = 83.6 nM T74307 CVQW20 73775923 IC50 = 2060 nM T74307 C5U4AF 73776059 IC50 = 160 nM T74307 CXW54V 73776061 IC50 = 177 nM T74307 CD83FL 73776204 IC50 = 342 nM T74307 CG84BR 73776205 IC50 = 2090 nM T74307 C1P3DO 73776206 IC50 = 1950 nM T74307 CN5D1R 73776207 IC50 = 300 nM T74307 CO1C8Y 73776208 IC50 = 246 nM T74307 CGC46K 73776360 IC50 = 295 nM T74307 CN39OQ 78341183 IC50 = 22 nM T74307 C64SIO 92042864 IC50 = 157 nM T74307 CAKD54 102594000 IC50 > 10000 nM T74307 CJGT03 118346182 IC50 = 607 nM T74307 C02DGP 118346184 IC50 > 10000 nM T74307 CU6NE2 118346192 IC50 = 336 nM T74307 CW25VP 118346194 IC50 = 293 nM T74307 CQCX41 118737057 IC50 = 19 nM T74307 CDSV38 121316062 Ki = 190 nM T74307 C81IFQ 122163152 IC50 > 100000 nM T74307 C76IKM 122705261 IC50 > 100000 nM T74307 CG8DA9 127045861 IC50 > 100000 nM T74307 CC4ND8 127046862 IC50 > 100000 nM T74307 CIU72D 127264586 IC50 = 8.1 nM T74307 C6ROQ3 132546210 IC50 = 81 nM T74307 CXC69T 137321158 IC50 = 138 nM T74307 C3Z4AT 137321159 IC50 > 10000 nM T74307 CZOD53 137633880 IC50 = 53 nM T74307 C7BJY5 137636807 IC50 = 50 nM T74307 C4DRX1 137643187 IC50 = 3050 nM T74307 CO89DX 137649100 IC50 = 29 nM T74307 CINE03 137652514 IC50 = 280 nM T74307 C28QUP 137652864 IC50 = 76.4 nM T74307 CGW9I0 137656387 IC50 = 5260 nM T74307 C4OD9Q 145967187 IC50 = 0.2 nM T74307 CE31VG 145979714 IC50 > 10000 nM T74307 C9BX4U 145988956 IC50 > 10000 nM T74307 C2MD1Q 155513187 IC50 > 10000 nM T74307 CI23DH 155516489 IC50 = 198 nM T74307 C3NA2I 155519537 IC50 = 10 nM T74307 CY5MR2 155522337 Ki = 170 nM T74307 CL0US4 155530459 IC50 = 0.7 nM T74307 C78MZC 155536330 IC50 = 8 nM T74307 CZQM57 155554194 IC50 = 2713.75 nM T74307 D00ERW 44444843 Ki > 1453 nM T74307 D00HVA 11624601 Ki > 1500 nM T74307 D01RHR 71519693 IC50 = 2.7 nM T74307 D01VFR 4708 IC50 = 5470 nM T74307 D06BJG 71556703 IC50 = 4.2 nM T74307 D0GN5Z 5281295 IC50 = 2880 nM T74307 D0Q3NG 11715520 Ki > 1500 nM T74307 D0S7IE 11658882 Ki > 1500 nM T21865 D02AUB 9811353 IC50 = 70000 nM T21865 D0Z0AM 12004316 IC50 = 150000 nM T21865 C96KNY 643990 IC50 = 15000000 nM T21865 CM8YN2 11348172 IC50 = 413000 nM T21865 CTDH45 14498151 IC50 = 4000000 nM T21865 CZ13DK 14498163 IC50 = 1000000 nM T21865 CJE6Y0 16099896 IC50 = 1500000 nM T21865 CGK0T7 16099901 IC50 = 1500000 nM T21865 C8CUQ4 16099902 IC50 = 3000000 nM T21865 C8D0KF 16099905 IC50 = 450000 nM T21865 CM8CL1 16099913 IC50 = 400000 nM T21865 C3UK7A 16099914 IC50 = 250000 nM T21865 C3V2KY 16099916 IC50 = 700000 nM T21865 C31XCS 16099919 IC50 = 225000 nM T21865 C0U9ZL 16099921 IC50 = 1500000 nM T21865 C2FXW0 16099923 IC50 = 200000 nM T21865 C3W7YQ 16099925 IC50 = 2000000 nM T21865 CFY05L 16099926 IC50 = 375000 nM T21865 CO5SY7 16099929 IC50 = 625000 nM T21865 CR6W3S 16099936 IC50 = 1500000 nM T21865 C7E3WD 16099940 IC50 = 1000000 nM T21865 CI0GX1 16099943 IC50 = 1000000 nM T21865 C0L5FE 16099944 IC50 = 200000 nM T21865 C0T6OC 16099945 IC50 = 400000 nM T21865 CZS67I 16099962 IC50 = 2000000 nM T21865 C51NZE 16099968 IC50 = 75000 nM T21865 C2NH3G 16099971 IC50 = 125000 nM T21865 C0IBF1 16099978 IC50 = 300000 nM T21865 CK4IH9 16099980 IC50 = 240000 nM T21865 CZ2FH9 16099985 IC50 = 1000000 nM T21865 CUM26S 16100003 IC50 = 600000 nM T21865 C4ZVE0 16100004 IC50 = 550000 nM T21865 CUMK61 16100005 IC50 = 1600000 nM T21865 CDG5U9 16100006 IC50 = 625000 nM T21865 CN6EC7 16100010 IC50 = 300000 nM T21865 C4B7JV 16100012 IC50 = 525000 nM T21865 CBK6Z3 16100014 IC50 = 175000 nM T21865 C7VE4W 16100015 IC50 = 500000 nM T21865 C9BKC2 16100016 IC50 = 225000 nM T21865 C2FHQ1 16100024 IC50 = 250000 nM T21865 C80LWT 16100025 IC50 = 250000 nM T21865 CT7HP1 25103104 IC50 = 250000 nM T21865 CD9KM7 44287084 IC50 = 2500000 nM T21865 CUS84P 46915502 IC50 = 175000 nM T21865 C19MAV 135547550 IC50 = 3500000 nM T21865 D00YPH 10239 IC50 = 6000000 nM T22302 CL3K7I 5310497 IC50 = 1200 nM T22302 CGMN97 25067404 IC50 = 537 nM T22302 C9B6XI 70686297 IC50 = 385 nM T22302 C6TNB2 70690451 IC50 = 6900 nM T22302 C4GXP2 70690453 IC50 = 61 nM T22302 CRGC43 70694654 IC50 = 2900 nM T22302 C2QHP7 70694655 IC50 = 177 nM T22302 CORP75 70696691 IC50 = 570 nM T22302 CRY1E6 70696692 IC50 = 1057 nM T22302 C24ACH 70696693 IC50 = 640 nM T22302 D0M2PP 7211972 IC50 = 568 nM T18477 D01BYB 5957 IC50 = 861330 nM T18477 D0E7PQ 5311 IC50 > 1000 nM T18477 D01FYA 9549213 IC50 = 43 nM T18477 D02TTL 44156921 IC50 = 33 nM T18477 D05BYA 135539077 IC50 < 0.4 nM T18477 D05HWN 16736529 Ki = 1.7 nM T18477 D06YSP 11955716 IC50 = 13.6 nM T18477 D07MPL 44195571 IC50 = 38 nM T18477 D0F3NF 67501411 Ki = 34.7 nM T18477 D0I1QI 135564985 IC50 = 5 nM T18477 D0K5BP 46216556 IC50 = 13 nM T18477 D00OCB 984170 IC50 = 280 nM T18477 D00GOM 71453910 IC50 = 90 nM T18477 D09BVL 4552 IC50 = 3320 nM T18477 CG47UK 10241 IC50 > 1000 nM T18477 CTV6F8 107935 IC50 = 1630 nM T18477 CUM2L9 145989 IC50 > 1250000 nM T18477 CA23LP 448972 EC50 = 170 nM T18477 C07TEG 764764 IC50 = 4400 nM T18477 CXK79E 767613 IC50 = 4730 nM T18477 C4L6KE 2766290 IC50 = 9600 nM T18477 CB6OK2 5287464 IC50 = 15200 nM T18477 CI7MW0 9852185 IC50 = 21980 nM T18477 C7E9KA 10177135 EC50 = 160 nM T18477 CU9SK6 10183346 EC50 = 30 nM T18477 CB7D8O 11187955 EC50 = 310 nM T18477 CO3HN2 11189279 EC50 = 130 nM T18477 CYQP95 11198704 IC50 > 100000 nM T18477 CO3F6K 11221466 IC50 > 100000 nM T18477 CH4B2Z 11223683 IC50 > 200000 nM T18477 C9ZS0N 11247073 EC50 = 2000 nM T18477 CA45FP 11266813 IC50 = 28030 nM T18477 CBZS48 11302159 IC50 > 300000 nM T18477 C0L2WJ 11314518 IC50 = 23930 nM T18477 CDJX31 11326407 IC50 = 60400 nM T18477 C2ZCY3 11336657 IC50 > 300000 nM T18477 CIRH67 11349446 IC50 > 300000 nM T18477 CUO6Q7 11393625 IC50 > 100000 nM T18477 CXN76P 11406285 IC50 > 500000 nM T18477 CP3Z4O 11407267 IC50 > 100000 nM T18477 CZKO68 11407809 EC50 = 20 nM T18477 CIG8V3 11415875 EC50 = 98 nM T18477 CP90LC 11427896 IC50 > 100000 nM T18477 CR9IQ7 11450570 IC50 > 300000 nM T18477 C8VZQ6 11463506 IC50 > 100000 nM T18477 CI53RD 11473241 IC50 > 100000 nM T18477 CQL4M5 11475629 EC50 = 4300 nM T18477 C6S3TY 11488262 EC50 = 470 nM T18477 C9IY1M 11517212 Ki = 0.2 nM T18477 CKSG91 11751343 EC50 = 90 nM T18477 C79VTC 11773074 IC50 > 50000 nM T18477 CPB49N 11855206 Ki = 235 nM T18477 CR1X7L 11950337 IC50 = 0.7 nM T18477 CAGU13 11950510 EC50 = 9 nM T18477 C8WAX9 11957092 Ki = 700 nM T18477 CE8M7K 12318923 IC50 = 31000 nM T18477 C8M6SA 12331235 IC50 = 13300 nM T18477 C82YHV 12331237 IC50 = 14900 nM T18477 CG07VM 12331240 IC50 = 49600 nM T18477 C4G8MJ 12571204 IC50 = 750 nM T18477 C9C4WH 15856427 IC50 = 24000 nM T18477 C7RCT2 15856428 IC50 = 16000 nM T18477 CDFK08 16061445 IC50 = 54 nM T18477 CI14ZN 16225982 IC50 = 19 nM T18477 C6JY5F 16226184 IC50 = 10 nM T18477 CTRL63 16667105 EC50 = 250 nM T18477 C1EXG6 16727212 IC50 = 220 nM T18477 C3BXP9 17545684 IC50 = 13300 nM T18477 CPYW42 21179452 IC50 = 42200 nM T18477 CRA65J 21846414 IC50 = 6900 nM T18477 CAS5G3 23958192 IC50 = 16.82 nM T18477 C7RTS1 24768274 IC50 > 20000 nM T18477 C7P4RL 24768277 IC50 > 20000 nM T18477 C1T4WH 25003030 Ki = 11 nM T18477 COBM26 25073055 IC50 = 28 nM T18477 C8F1MA 44323467 IC50 = 33000 nM T18477 CM5XT0 44376308 EC50 = 3600 nM T18477 C8WJ9S 44376565 EC50 = 1400 nM T18477 CAKW20 44376753 EC50 = 3500 nM T18477 CSHJ14 44383813 EC50 > 50000 nM T18477 C45XQM 44400015 EC50 = 330 nM T18477 C0L5XP 44400119 EC50 = 2800 nM T18477 C2UWT8 45162180 IC50 = 308500 nM T18477 C3BJ9O 45788206 Ki = 8300 nM T18477 CS6J7Q 46861552 Ki = 1200 nM T18477 CSD39K 46912795 IC50 = 94 nM T18477 CRIB76 46913258 IC50 = 365 nM T18477 C8U9LT 46919029 IC50 = 490 nM T18477 C15CFW 46919030 IC50 = 510 nM T18477 CUP92O 49842657 IC50 = 585 nM T18477 C54HZQ 49863672 IC50 = 1400 nM T18477 CE4AN1 49863673 IC50 = 650 nM T18477 C0U8MW 49863674 IC50 = 5100 nM T18477 C6T9HE 49863675 IC50 = 790 nM T18477 C19VJH 49863676 IC50 = 3400 nM T18477 CX74OK 49863677 IC50 = 1100 nM T18477 C0Q8ZV 49863678 IC50 = 3100 nM T18477 C21JZL 49870746 IC50 = 9524 nM T18477 CBA6D2 49871894 IC50 = 470 nM T18477 CR0U5H 49871895 IC50 = 58 nM T18477 C2ERZ4 49871985 IC50 = 183 nM T18477 CMA10L 49871988 IC50 = 750 nM T18477 C7GRS3 50925477 EC50 = 60 nM T18477 C2OVL4 51049656 Ki = 130 nM T18477 C4MZ7N 52916002 IC50 = 15530 nM T18477 CK98TP 52918129 IC50 = 90 nM T18477 CB1JE7 52918144 IC50 = 110 nM T18477 CHZP24 53236116 Ki = 190 nM T18477 C3MA7Q 53236117 Ki = 120 nM T18477 C3RCQ9 53236118 Ki = 16 nM T18477 CLPO19 53236119 Ki = 250 nM T18477 C2BYJ6 53236120 Ki = 7 nM T18477 C7OSD2 53236121 Ki = 35 nM T18477 C8G5TM 53236346 Ki = 20 nM T18477 CL60TN 53236347 Ki = 13 nM T18477 CU1BE9 53236348 Ki = 12 nM T18477 CFL65I 53236349 Ki = 9 nM T18477 CV7BK2 53236350 Ki = 6 nM T18477 CH8LV9 53236351 Ki = 9 nM T18477 CQM95X 53236589 Ki = 7 nM T18477 CFI32H 53239287 Ki = 50 nM T18477 C35TQX 53239288 Ki = 26 nM T18477 CJ68VG 53239289 Ki = 38 nM T18477 CGMZ76 53239290 Ki = 21 nM T18477 CG26RE 53239291 Ki = 18 nM T18477 C1VJ0T 53239502 Ki = 7 nM T18477 C80QGZ 53239503 Ki = 110 nM T18477 CYC7B4 53239504 Ki = 7 nM T18477 C4S8QK 53239505 Ki = 27 nM T18477 CTJB43 53239506 Ki = 40 nM T18477 C13XHA 53239507 Ki = 300 nM T18477 CKNJ47 53245660 IC50 = 83 nM T18477 CW9IQ0 53248730 IC50 = 82 nM T18477 CVHW83 53259029 IC50 = 110 nM T18477 C1KYR9 53326941 IC50 = 96 nM T18477 CI0R4B 54580554 IC50 = 96 nM T18477 CRV6M8 54580555 IC50 = 126 nM T18477 CYC3K8 54580556 IC50 = 3324 nM T18477 CYC3V7 54580557 IC50 = 153 nM T18477 C34EOA 54580558 IC50 = 301 nM T18477 CRF0G6 54581044 IC50 = 830 nM T18477 CA3CX5 54581045 IC50 = 320 nM T18477 CHFD41 54581046 IC50 = 150 nM T18477 C4EH1F 54581551 IC50 = 201 nM T18477 CYAI91 54581552 IC50 = 634 nM T18477 CA73VM 54581553 IC50 = 496 nM T18477 CIHT85 54582089 IC50 > 5000 nM T18477 CZG19I 54582090 IC50 = 1240 nM T18477 CBI7N9 54582551 IC50 > 5000 nM T18477 C15SZU 54582552 IC50 = 188 nM T18477 CONG87 54582553 IC50 = 982 nM T18477 CF87RH 54583025 IC50 = 210 nM T18477 CEOZ15 54583522 IC50 = 96 nM T18477 CW2AF0 54584037 IC50 = 400 nM T18477 CQ65AR 54584038 IC50 = 570 nM T18477 C96JOM 54584500 IC50 = 883 nM T18477 CJV94T 54584501 IC50 = 78 nM T18477 C1T5NF 54584983 IC50 = 12440 nM T18477 CNJO03 54584984 IC50 > 5000 nM T18477 C96JXE 54585939 IC50 = 430 nM T18477 CSC0H3 54586414 IC50 = 61 nM T18477 C7HD0U 54586415 IC50 = 170 nM T18477 CFI5J2 54586912 IC50 = 290 nM T18477 C7G6IP 54586913 IC50 = 140 nM T18477 CZK7F1 54586914 IC50 = 920 nM T18477 CZ54WE 54586915 IC50 = 360 nM T18477 CD06RB 54587434 IC50 = 106 nM T18477 CR1I6J 54587584 IC50 = 145 nM T18477 CM01DQ 54764333 IC50 = 5600 nM T18477 C2QK8U 56659496 IC50 = 24800 nM T18477 CA9T4B 56659497 IC50 = 25200 nM T18477 CC8AZ2 56659584 IC50 = 80 nM T18477 C6QSI8 56659760 IC50 = 84 nM T18477 C71GNP 56659879 IC50 > 200000 nM T18477 CWKH97 56659880 IC50 > 200000 nM T18477 C01XAG 56662951 IC50 = 15400 nM T18477 COEU61 56662986 IC50 = 34900 nM T18477 C1RPG4 56662987 IC50 = 200000 nM T18477 CL8J5E 56663234 IC50 = 82 nM T18477 CS0OL3 56663235 IC50 = 88 nM T18477 CK81DA 56663236 IC50 = 74 nM T18477 CASK95 56663304 IC50 = 116 nM T18477 CF3DM2 56663339 IC50 > 200000 nM T18477 C28OQJ 56666428 IC50 = 72 nM T18477 CW51JK 56666664 IC50 = 116 nM T18477 C5XGS1 56666665 IC50 = 142 nM T18477 CFI5R6 56666666 IC50 = 66 nM T18477 C3D4TK 56666731 IC50 = 83 nM T18477 CYQE09 56666732 IC50 = 65 nM T18477 CEU56I 56666733 IC50 = 68 nM T18477 CA3HM7 56666734 IC50 = 228 nM T18477 CCR76H 56670085 IC50 = 64 nM T18477 C6EFP7 56670086 IC50 = 85 nM T18477 C0ABN1 56670087 IC50 = 77 nM T18477 CX92TP 56670157 IC50 = 83 nM T18477 CU6CS9 56670202 IC50 > 200000 nM T18477 C24YWF 56670203 IC50 > 200000 nM T18477 CXUI30 56673328 IC50 = 47 nM T18477 CD65HO 56673605 IC50 = 58 nM T18477 CFOE91 56673671 IC50 = 60 nM T18477 C3KZM9 56673672 IC50 = 91 nM T18477 CEN4H5 56676988 IC50 = 70 nM T18477 CI0Y5Z 56677032 IC50 > 200000 nM T18477 C10YJZ 56679993 IC50 = 33 nM T18477 C4AOI1 56679994 IC50 = 27 nM T18477 C1BPY4 56680021 IC50 = 127000 nM T18477 CW4JM5 56680236 IC50 = 81 nM T18477 CG34TX 56680322 IC50 = 183 nM T18477 CG51ZV 56681935 IC50 = 570 nM T18477 COL34U 56683638 IC50 = 131 nM T18477 CPMG31 56683692 IC50 > 200000 nM T18477 C73AOX 57404605 IC50 = 23 nM T18477 CM89YZ 57404775 IC50 = 27 nM T18477 CTQ1N2 57404776 IC50 = 95 nM T18477 CT65MO 57404777 IC50 = 270 nM T18477 CN0B1D 57405452 IC50 = 17 nM T18477 CT87RM 57406669 IC50 = 37 nM T18477 CD5C0Y 57406670 IC50 = 27 nM T18477 CO4W8R 57406671 IC50 = 36 nM T18477 C0RKH7 57406855 IC50 < 5 nM T18477 C8N1XS 57406856 IC50 = 23 nM T18477 CW1LY5 57406857 IC50 < 5 nM T18477 CI4C2X 57406859 IC50 = 21 nM T18477 CEH2P1 57406860 IC50 = 25 nM T18477 C3WPF1 57407047 IC50 < 5 nM T18477 CWH2N3 57407048 IC50 < 5 nM T18477 C3UN0J 57407049 IC50 < 5 nM T18477 C6I1SA 57407050 IC50 = 14.8 nM T18477 CA6Q1L 57407243 IC50 = 6.8 nM T18477 CP8AF0 57407244 IC50 = 15 nM T18477 CIJE49 57407246 IC50 = 32 nM T18477 CX9H1U 57407247 IC50 = 13 nM T18477 CTXS05 57407248 IC50 < 5 nM T18477 CH3OR8 57424824 IC50 = 300 nM T18477 CD56FL 57424831 IC50 = 56 nM T18477 C1L5UN 57424851 IC50 = 24 nM T18477 C70OWD 57424917 IC50 = 16 nM T18477 CI2WK1 57424929 IC50 > 10000 nM T18477 C3WLV1 57450675 IC50 = 37 nM T18477 CA4Y5Q 57450676 IC50 = 12 nM T18477 CU62HN 57450694 IC50 = 9800 nM T18477 C4G9FJ 57462510 IC50 = 27 nM T18477 CZVS05 57462516 IC50 = 140 nM T18477 CY87RC 57713841 IC50 = 3.9 nM T18477 C2FY4H 57748464 IC50 = 641 nM T18477 CSA3O2 57748552 IC50 = 479 nM T18477 C3HW6F 58762794 IC50 = 97 nM T18477 CZ7XQ5 60165612 Ki = 1800 nM T18477 CAU06M 66576834 IC50 = 100 nM T18477 C60LFE 66612138 IC50 = 27340 nM T18477 CV8B0R 67495834 Ki = 3 nM T18477 C2S9CE 67500027 IC50 = 73 nM T18477 C7IXO4 67500163 IC50 = 131 nM T18477 CZ2L9M 67500276 IC50 = 789 nM T18477 C0A6OX 67500939 IC50 = 52 nM T18477 C6VE3A 67500997 IC50 = 132 nM T18477 CD75KX 67501021 IC50 = 98 nM T18477 CPZA60 67501051 IC50 > 10000 nM T18477 CAX0I7 67501291 IC50 = 166 nM T18477 C32UVO 67502140 IC50 = 1168 nM T18477 CN26RP 67502287 IC50 = 1620 nM T18477 CX7G8L 67502777 IC50 = 72 nM T18477 C80ODY 67932020 Ki = 1380 nM T18477 C9TN8Q 67984974 IC50 = 35 nM T18477 CW4EM0 67985170 IC50 = 23 nM T18477 C4VT3I 67985199 IC50 = 30 nM T18477 C7WH6F 67985284 IC50 = 10 nM T18477 CQI6F7 67985727 IC50 < 5 nM T18477 CNC49F 71463004 IC50 = 1 nM T18477 CIG6P3 71660550 IC50 > 500000 nM T18477 C79AGJ 71660551 IC50 = 27300 nM T18477 CELO13 72376512 IC50 = 47000 nM T18477 CR3K1V 72547522 Ki = 2800 nM T18477 C9CW5M 73437615 Ki = 20 nM T18477 CUD54E 73437616 Ki = 5 nM T18477 CAW01J 74027120 IC50 = 22400 nM T18477 CUOW40 74222622 IC50 = 890 nM T18477 CRA86Z 76311786 IC50 = 48500 nM T18477 CJ2PU1 76315352 IC50 = 7600 nM T18477 CS97VJ 76315353 IC50 = 13200 nM T18477 CH0AP5 76319024 IC50 = 7400 nM T18477 CU3G6Q 76322418 IC50 = 12700 nM T18477 C68TOV 76322671 IC50 = 17300 nM T18477 C9BCH0 76322676 IC50 = 12700 nM T18477 CS0PB2 76324772 Ki = 125 nM T18477 CPX91U 76329863 IC50 = 26600 nM T18477 C2I4XM 76333294 IC50 = 12000 nM T18477 C49ZCD 76333509 IC50 = 16400 nM T18477 C6LV9H 76899944 IC50 = 410 nM T18477 CYZN80 76899957 IC50 = 470 nM T18477 C6WE9Y 77107768 IC50 = 1840 nM T18477 CAGX72 78106056 IC50 = 14330 nM T18477 C2N3CM 78106057 IC50 = 35240 nM T18477 CV2C8Q 78106150 IC50 = 8520 nM T18477 C47XUW 86280454 Ki > 100000 nM T18477 CT80DA 86294728 IC50 = 38 nM T18477 C2N7AP 86294734 IC50 = 70 nM T18477 C1ZKP7 86294735 IC50 = 38 nM T18477 CK98UO 86294736 IC50 = 21 nM T18477 C2MC0R 86294737 IC50 = 39 nM T18477 C40LNZ 86294738 IC50 = 190 nM T18477 CC3I7E 86302592 IC50 = 110 nM T18477 CVL4I0 86302593 IC50 = 29 nM T18477 C06YBD 86302594 IC50 = 33 nM T18477 CJ3Q4H 90654630 Ki = 6 nM T18477 CG8S1L 90654631 Ki = 3 nM T18477 CDIY85 90654632 Ki = 34 nM T18477 CV9YA4 90654633 Ki = 56 nM T18477 CRH14E 90654634 Ki = 180 nM T18477 C26WSJ 90654635 Ki = 94 nM T18477 CXLQ38 90654636 Ki = 14 nM T18477 C9F5UB 90654637 Ki = 10 nM T18477 CZ2MP4 90654638 Ki = 20 nM T18477 C17RWB 90654639 Ki = 40 nM T18477 C7X8WK 90654640 Ki = 32 nM T18477 CJ2ZM3 90654641 Ki = 42 nM T18477 C21FPZ 90654642 Ki = 14 nM T18477 C9ZTU1 90654643 Ki = 17 nM T18477 CTB60Y 90654644 Ki = 62 nM T18477 C81JGB 90654645 Ki = 28 nM T18477 CKM2W0 90654646 Ki = 22 nM T18477 CS8U1X 90654647 Ki = 46 nM T18477 CUE4I6 90654648 Ki = 28 nM T18477 CM5JP8 90654649 Ki = 28 nM T18477 CH8FD0 90654650 Ki = 25 nM T18477 C5DP2C 90654651 Ki = 22 nM T18477 CU87TN 90654652 Ki = 37 nM T18477 C4PJ1V 90654653 Ki > 10000 nM T18477 C2TYR0 90654654 Ki = 680 nM T18477 C6SI7L 90654655 Ki > 10000 nM T18477 CG2JK7 90654656 Ki = 390 nM T18477 CBWT05 90654657 Ki = 42 nM T18477 C6SK1Z 90654658 Ki = 36 nM T18477 C2TLY1 90654659 Ki > 10000 nM T18477 C3R1DJ 90654660 Ki = 1900 nM T18477 CT1QI5 90654661 Ki > 10000 nM T18477 CU8Q1V 90654662 Ki > 10000 nM T18477 CS42OM 90654663 Ki = 2500 nM T18477 C7M8TA 90654664 Ki = 3200 nM T18477 C1H5WC 90654665 Ki = 690 nM T18477 C9NO7L 90655134 IC50 = 34 nM T18477 C4SR1G 90655135 IC50 = 54 nM T18477 C18XMN 90655136 IC50 = 68 nM T18477 C82SQK 90655137 IC50 = 100 nM T18477 CEU4P7 90655138 IC50 = 160 nM T18477 C80KYO 90655139 IC50 = 1200 nM T18477 C29HUJ 90655140 IC50 = 1400 nM T18477 C6C7ST 90655141 IC50 = 3900 nM T18477 CGA47I 90655142 IC50 > 100000 nM T18477 C68KOR 90655143 IC50 > 100000 nM T18477 C3XL9Q 90655144 IC50 > 100000 nM T18477 CSR56C 90655296 IC50 = 31 nM T18477 C5WZ0F 90655297 IC50 = 12 nM T18477 C9HF1A 90655298 IC50 = 33 nM T18477 CW1UR6 90655299 IC50 = 181 nM T18477 CQ0JR2 90655300 IC50 > 1000 nM T18477 C76DSY 90655301 IC50 = 320 nM T18477 CZV1W0 90655302 IC50 = 295 nM T18477 C0UP3C 90656478 IC50 = 630 nM T18477 CQU83E 90656479 IC50 = 130 nM T18477 CW7L0S 90656480 IC50 = 330 nM T18477 CJY51L 90656481 IC50 = 130 nM T18477 CZ1I8E 90656482 IC50 = 250 nM T18477 CUD9J1 90656483 IC50 = 1500 nM T18477 CK94EB 90656484 IC50 = 130 nM T18477 C8R9JB 90656485 IC50 = 620 nM T18477 CWC3J9 90656486 IC50 = 78 nM T18477 CGL40M 90656487 IC50 = 71 nM T18477 CD6Z7W 90657117 Ki = 86 nM T18477 CI90DU 117736689 IC50 = 55 nM T18477 CVDP67 117736692 IC50 = 48 nM T18477 C60TAF 117736697 IC50 = 96 nM T18477 CX31TW 117736731 IC50 = 54 nM T18477 C2W9GO 117736733 IC50 = 91 nM T18477 CUVD12 117889758 IC50 > 25000 nM T18477 CUTV54 117889766 IC50 > 50000 nM T18477 CIBF07 117889785 IC50 > 100000 nM T18477 CW8J2A 117889863 IC50 > 100000 nM T18477 CP0VL5 117889908 IC50 = 24900 nM T18477 C0GZD8 117889984 IC50 > 100000 nM T18477 CGM51T 117890044 IC50 > 50000 nM T18477 C37QWO 117890084 IC50 > 50000 nM T18477 C1APC8 117890111 IC50 = 15970 nM T18477 CZ4EN5 117890133 IC50 > 50000 nM T18477 CO2R1E 117890146 IC50 > 100000 nM T18477 CE69YR 117890174 IC50 > 100000 nM T18477 C3C6KX 117890187 IC50 = 8300 nM T18477 CX6V7Q 117890195 IC50 > 50000 nM T18477 C4MQ8T 117890212 IC50 > 50000 nM T18477 CG53QV 117890216 IC50 = 20300 nM T18477 CZ45SB 117890250 IC50 > 100000 nM T18477 CLH49C 117890268 IC50 > 50000 nM T18477 CLHP30 117890308 IC50 > 100000 nM T18477 CQK30X 117890321 IC50 > 50000 nM T18477 CPWS97 117890346 IC50 > 50000 nM T18477 C1HK7L 117890351 IC50 > 50000 nM T18477 CO25TC 117890352 IC50 > 100000 nM T18477 CA15DJ 117890354 IC50 > 50000 nM T18477 CTV53C 117890368 IC50 = 1960 nM T18477 CQCT02 117890387 IC50 > 50000 nM T18477 CQ20HF 117890473 IC50 > 50000 nM T18477 C3R9DT 117890494 IC50 > 100000 nM T18477 CRYX09 117890515 IC50 > 50000 nM T18477 CK15CW 117967655 Ki = 9150 nM T18477 CQ4FL0 117968039 Ki = 3480 nM T18477 CYG8C4 117970892 Ki = 1980 nM T18477 CZ2AI8 117972517 Ki = 1020 nM T18477 CFI2P0 117972524 Ki = 6550 nM T18477 C5TFJ0 117972658 Ki = 3210 nM T18477 CN08WT 118712080 IC50 = 1040 nM T18477 CVK84L 118712081 IC50 = 430 nM T18477 C9A2OU 118719939 IC50 = 970 nM T18477 C6BGJ8 118720311 IC50 = 290 nM T18477 CXB34W 118724182 IC50 = 16 nM T18477 CG0R3L 118728263 Ki = 150 nM T18477 C3A8PL 118728264 Ki = 64 nM T18477 CKXV89 118728265 Ki = 213 nM T18477 COV7S8 118728266 Ki = 110 nM T18477 C3F7KR 118728267 Ki = 33 nM T18477 CX1DZ2 118728268 Ki = 54 nM T18477 C5TP4Q 118728269 Ki = 86 nM T18477 CX6U2K 118728270 Ki = 190 nM T18477 CRY17Z 118728271 Ki = 41 nM T18477 CTC60M 118728272 Ki = 50 nM T18477 CJT25I 118728273 Ki = 370 nM T18477 C9AT5X 118729959 Ki = 115 nM T18477 CDZ98W 118729960 Ki = 60 nM T18477 C5C8GB 118729961 Ki = 111 nM T18477 CKE49U 118737375 IC50 > 50000 nM T18477 C84YNW 118737376 IC50 > 50000 nM T18477 CKB9N5 118737377 IC50 > 50000 nM T18477 C1ZSK4 118737378 IC50 > 50000 nM T18477 CO6N4H 118796335 IC50 = 5 nM T18477 CBK28I 124081275 IC50 > 100000 nM T18477 CQ82GU 124201644 Ki = 10600 nM T18477 CCD60J 126962311 IC50 > 1000 nM T18477 CAQL68 126962384 IC50 > 1000 nM T18477 C59DWI 126962385 IC50 > 1000 nM T18477 CBXH95 127024111 Ki > 50000 nM T18477 CS1ZO6 127024161 Ki = 2510 nM T18477 CHQ12D 127024491 Ki > 50000 nM T18477 CBS1R8 127024554 Ki = 1780 nM T18477 CR6A9C 127024644 Ki > 50000 nM T18477 CGO8S5 129900226 IC50 = 698 nM T18477 CQ4S3Z 130277442 IC50 = 362 nM T18477 CX0QS8 130277744 IC50 = 611.5 nM T18477 C15ECZ 130277802 IC50 = 6.5 nM T18477 CW0D2F 131704417 IC50 = 36 nM T18477 CI47VP 131704472 IC50 = 39200 nM T18477 C0IQ4V 132601722 IC50 = 3680 nM T18477 CE3X8V 132992912 Ki > 13000 nM T18477 C4FPW8 132992920 Ki = 840 nM T18477 CUF85A 134132715 IC50 = 51 nM T18477 C1P5TE 134135478 IC50 = 94 nM T18477 CDC41Q 134138735 IC50 = 58 nM T18477 CH8G2J 134139194 IC50 = 79 nM T18477 CAB93T 134139543 IC50 = 750 nM T18477 C1PZ6L 134140295 IC50 = 480.8 nM T18477 CRDK20 134142142 IC50 = 183.3 nM T18477 CB7A0W 134145703 IC50 = 48 nM T18477 C0C4JZ 134147224 IC50 = 135.9 nM T18477 CC43OQ 134149366 IC50 = 50.3 nM T18477 CZEO76 134150482 IC50 = 8700 nM T18477 CZ68GA 134154630 IC50 > 1000 nM T18477 CT87WB 134156050 IC50 = 650 nM T18477 C0ZVI9 134157119 IC50 > 1000 nM T18477 CA0MT1 134480068 IC50 = 8932 nM T18477 CBRN70 135400938 IC50 = 60 nM T18477 CWHX62 135423284 IC50 = 62 nM T18477 CHZD50 135425202 IC50 = 210 nM T18477 CA1MC6 135433906 IC50 = 190 nM T18477 CS8JP3 135481178 IC50 = 150 nM T18477 C9NH7L 135499841 IC50 = 53 nM T18477 CVZ37K 135507483 IC50 = 120 nM T18477 C9EIC5 135507502 IC50 = 70 nM T18477 CK7PL9 135519368 IC50 = 510 nM T18477 C23HTX 135524913 IC50 = 39 nM T18477 CEK31P 135566415 IC50 = 30 nM T18477 CVJ05Z 135566858 IC50 = 70 nM T18477 CDIR12 135566860 IC50 = 27 nM T18477 CHE38I 135566861 IC50 = 23 nM T18477 C39USJ 135567370 IC50 = 37 nM T18477 CW54FS 135567371 IC50 = 38 nM T18477 C0QF7Z 135567372 IC50 = 42 nM T18477 CL59TN 135567373 IC50 = 44 nM T18477 C9KGT3 135567374 IC50 = 53 nM T18477 C1UEK8 135581701 IC50 = 40 nM T18477 CN97EY 135581702 IC50 = 800 nM T18477 CI85ZN 135981701 IC50 = 14500 nM T18477 C5J3KX 135981702 IC50 = 22100 nM T18477 CYV84F 136000662 Ki = 1400 nM T18477 C3ZBM8 136110909 IC50 = 66 nM T18477 CG06VA 136110910 IC50 = 121 nM T18477 C63FBA 136110911 IC50 = 57 nM T18477 CX27KJ 136110912 IC50 = 69 nM T18477 C5GD7K 136110913 IC50 = 295 nM T18477 CHQ05G 136110914 IC50 = 40 nM T18477 C3Y8LO 136110915 IC50 = 1660 nM T18477 CU8T5Q 136110916 IC50 = 546 nM T18477 CG2PO0 136110917 IC50 = 108 nM T18477 CUQ0B5 136110919 IC50 = 471 nM T18477 C1Y5HJ 136110920 IC50 = 307 nM T18477 CFPA47 136110921 IC50 = 99 nM T18477 CU6F1X 136110922 IC50 = 183 nM T18477 C8N1QK 136167232 Ki = 32 nM T18477 C2SRX9 136198647 IC50 > 100000 nM T18477 CEX34H 136198648 IC50 > 100000 nM T18477 CN0XY9 136198649 IC50 > 100000 nM T18477 CP79HX 136198650 IC50 > 100000 nM T18477 CR3LD9 136198651 IC50 > 100000 nM T18477 CN83ZX 136198652 IC50 > 100000 nM T18477 CEWC75 136198653 IC50 > 100000 nM T18477 C2NOH9 136236968 IC50 > 250000 nM T18477 CNM6L0 136266479 IC50 = 17 nM T18477 C0D6OT 136266481 IC50 = 35 nM T18477 C5SZ6I 136266482 IC50 = 46 nM T18477 CV7YO5 136266483 IC50 = 29 nM T18477 C8K5DR 136266484 IC50 = 57 nM T18477 C37HLR 136266485 IC50 = 36 nM T18477 C6XHU2 136266487 IC50 = 35 nM T18477 C4FLS0 136266488 IC50 = 27 nM T18477 C8G1CX 136266497 IC50 = 58 nM T18477 C0H9TJ 136266498 IC50 = 55 nM T18477 CDC53A 136266499 IC50 = 140 nM T18477 CKP7A9 136266500 IC50 = 30 nM T18477 CAPE16 136266501 IC50 = 44 nM T18477 C5XW9N 136266513 IC50 = 53 nM T18477 C7PCL8 136266514 IC50 = 44 nM T18477 C9NOM4 136266515 IC50 = 60 nM T18477 CO1U4Q 136266516 IC50 = 43 nM T18477 CL8MY2 136266517 IC50 = 35 nM T18477 C5LB9C 136266518 IC50 = 88 nM T18477 C5I3SJ 136266519 IC50 = 180 nM T18477 C05RDT 136266522 IC50 = 59 nM T18477 CJ3FE1 136266530 IC50 = 140 nM T18477 C1RP5H 136266531 IC50 = 42 nM T18477 CD9O8U 136266533 IC50 = 300 nM T18477 C2N5HF 136266558 IC50 = 70 nM T18477 C01ZXH 136266559 IC50 = 21 nM T18477 CTCO28 136934953 IC50 > 100000 nM T18477 CMZ90X 136934954 IC50 > 100000 nM T18477 CW40ER 136934955 IC50 > 100000 nM T18477 CKS79P 136934956 IC50 > 100000 nM T18477 CA4OC9 136934957 IC50 > 500000 nM T18477 CI8FR0 136934958 IC50 > 250000 nM T18477 C5VIG4 136934959 IC50 > 100000 nM T18477 C2YZ6E 136934960 IC50 > 100000 nM T18477 C6B4DY 136934961 IC50 > 100000 nM T18477 C01EUC 137069409 IC50 = 127 nM T18477 C0KZD3 137069410 IC50 = 50 nM T18477 COZ20T 137069411 IC50 = 78 nM T18477 C81TKF 137069412 IC50 = 120 nM T18477 C9PDL7 137069413 IC50 = 1660 nM T18477 CKH8P9 137069414 IC50 = 546 nM T18477 CB3P2W 137069415 IC50 = 66 nM T18477 CE35LW 137069416 IC50 = 207 nM T18477 CEL0H2 137069417 IC50 = 45 nM T18477 C7PGC2 137069418 IC50 = 144 nM T18477 CGWX25 137069419 IC50 = 114 nM T18477 CZX7K1 137069420 IC50 = 28 nM T18477 CFOU34 137069421 IC50 = 91 nM T18477 C18RKL 137069422 IC50 = 48 nM T18477 CG05CN 137069423 IC50 = 66 nM T18477 C2GB4N 137069424 IC50 = 33 nM T18477 CYF42G 137069425 IC50 = 54 nM T18477 CTG86A 137069426 IC50 = 152 nM T18477 C4ZM0V 137069427 IC50 = 125 nM T18477 CQEZ48 137069428 IC50 = 347 nM T18477 CZ8IH9 137069429 IC50 = 45 nM T18477 CTI86X 137069430 IC50 = 108 nM T18477 C5GKE7 137069431 IC50 = 66 nM T18477 CRL7Z3 137287446 IC50 > 1000 nM T18477 C8ZP0L 137440573 IC50 > 1000 nM T18477 C8V9ER 137440575 IC50 = 5.3 nM T18477 CD5H0E 137440576 IC50 = 413 nM T18477 CR60OH 137440582 IC50 = 995 nM T18477 CK0S4Q 137440583 IC50 = 429 nM T18477 CZW8E2 137440584 IC50 = 11.4 nM T18477 C9J2MH 137440585 IC50 = 830 nM T18477 C3O9BW 137440587 IC50 = 585 nM T18477 CRS03O 137440588 IC50 = 496 nM T18477 CAT74Q 137440592 IC50 = 558 nM T18477 C5QYW2 137440596 IC50 = 454 nM T18477 CZ54WU 137440598 IC50 > 1000 nM T18477 C3IT5C 137440602 IC50 = 528 nM T18477 CN26IS 137440610 IC50 = 135 nM T18477 CXF50C 137632543 IC50 > 1000 nM T18477 C9BX6Y 137635266 IC50 = 374 nM T18477 C39AGH 137635456 IC50 = 852 nM T18477 CC1DT5 137636870 IC50 = 307 nM T18477 CQ02SA 137637101 IC50 = 528 nM T18477 CKEW37 137638689 IC50 = 112 nM T18477 CI1G9X 137638702 IC50 = 14 nM T18477 CU4ZQ2 137638985 IC50 = 514 nM T18477 C4Q9JZ 137640085 IC50 = 749 nM T18477 C21FBO 137640720 IC50 = 28 nM T18477 CV0E9Z 137641466 IC50 = 473 nM T18477 CS3KF0 137642154 Ki = 1230 nM T18477 C12MZJ 137645122 IC50 = 260 nM T18477 C5CQ9Z 137645320 IC50 = 154 nM T18477 CPT60O 137645600 IC50 = 189 nM T18477 CHR4Z3 137648200 IC50 = 752 nM T18477 CJ16QN 137649039 IC50 = 151 nM T18477 CX4QS7 137649776 IC50 = 368 nM T18477 CF3L0U 137649852 IC50 = 836 nM T18477 CNXW27 137650729 IC50 = 285 nM T18477 CJ39SV 137650769 IC50 = 429 nM T18477 CL5J0D 137651203 IC50 = 206 nM T18477 CBTS61 137651332 IC50 > 10000 nM T18477 CQA9I8 137651592 IC50 = 98 nM T18477 CU9X3H 137651850 IC50 = 72 nM T18477 C7NG3S 137653255 IC50 = 21 nM T18477 C56PSW 137653748 IC50 = 397 nM T18477 CCEA75 137654206 IC50 = 122 nM T18477 C06UCI 137654541 IC50 = 106 nM T18477 C9YPV6 137657005 IC50 = 206 nM T18477 CBUZ81 137657937 IC50 = 79 nM T18477 C2A8IQ 137657990 IC50 > 10000 nM T18477 CA7G0C 137658950 IC50 = 39 nM T18477 COR37X 137659330 IC50 > 1000 nM T18477 CPH71E 137659954 IC50 = 407 nM T18477 CO6XK1 137660391 Ki = 184 nM T18477 C9SC4G 137660536 IC50 = 259 nM T18477 C43OWV 145953418 IC50 = 40 nM T18477 CNE6Q7 145953506 IC50 > 1000 nM T18477 CU9J0X 145954267 IC50 > 1000 nM T18477 CROY34 145956057 IC50 = 260 nM T18477 C9CBZ7 145956245 IC50 = 84.8 nM T18477 C14ICP 145956607 IC50 = 100 nM T18477 CG5IT7 145956784 IC50 > 1000 nM T18477 C20VAD 145957128 IC50 = 370 nM T18477 CR26HS 145959950 IC50 = 123 nM T18477 CWU27Z 145969804 IC50 > 100000 nM T18477 C63KEL 145970838 IC50 = 20200 nM T18477 C7UG3O 145971121 IC50 > 100000 nM T18477 CGSA67 145971928 IC50 = 47 nM T18477 CDVM26 145971994 IC50 > 1000 nM T18477 C9VDE5 145982499 IC50 = 40.2 nM T18477 C6OL1K 145983267 IC50 = 55.9 nM T18477 C8O1GU 145983616 IC50 = 49.3 nM T18477 C17UTC 145983813 IC50 = 85.7 nM T18477 CIWO70 145984314 IC50 = 52.1 nM T18477 C9ZKC1 145984665 IC50 = 58.6 nM T18477 CN6KB9 145985243 IC50 = 46.3 nM T18477 C0DR4V 146034184 IC50 = 21 nM T18477 CKO79M 155511775 IC50 = 70 nM T18477 CQ5L3O 155515228 IC50 = 52670 nM T18477 C0ZY8Q 155516833 IC50 > 100000 nM T18477 CEG67W 155518415 IC50 = 54680 nM T18477 C9AC7B 155518571 IC50 = 164 nM T18477 CDY5H6 155519645 IC50 = 77210 nM T18477 C83HYP 155521152 IC50 = 430 nM T18477 C6Q4LC 155521952 IC50 = 15290 nM T18477 CJ34YH 155524691 IC50 = 643 nM T18477 C68ZRJ 155524949 IC50 = 97.11 nM T18477 CQ3AI0 155525851 IC50 = 302290 nM T18477 CX2D6L 155525906 IC50 = 1702 nM T18477 CH52FD 155526273 IC50 > 1000000 nM T18477 CU4X5I 155527383 IC50 > 10000 nM T18477 C9O0EU 155528011 IC50 = 72 nM T18477 CLVW69 155528303 IC50 > 1000000 nM T18477 C5F1IZ 155528743 IC50 > 1000000 nM T18477 C9TIO5 155528896 IC50 = 169340 nM T18477 C1B2FN 155530610 IC50 = 145800 nM T18477 C0VZ9J 155532068 IC50 > 1000000 nM T18477 CVL8J4 155532571 IC50 = 280 nM T18477 C6LTV0 155536018 IC50 = 42980 nM T18477 C45YWP 155537090 IC50 = 52.97 nM T18477 C8WNG3 155539047 IC50 = 60 nM T18477 CLD19W 155539311 IC50 = 153070 nM T18477 C9PFH1 155539933 IC50 = 13620 nM T18477 CNC1O0 155543432 IC50 = 89830 nM T18477 CFM68U 155545469 IC50 > 1000 nM T18477 CWZ82Y 155546946 IC50 = 1258 nM T18477 CE9R1Q 155549076 IC50 = 76810 nM T18477 C02YXA 155550058 IC50 = 186070 nM T18477 CUN7G5 155554476 IC50 = 8.319 nM T18477 CTC6O0 155554826 IC50 > 10000 nM T18477 CVH3K6 155555734 IC50 = 630 nM T18477 CG7OQ2 155556818 IC50 > 1000 nM T18477 CE1Q6X 155558343 IC50 = 58 nM T18477 CMPA40 155559139 IC50 = 204 nM T18477 CG0HE7 155559221 IC50 = 6200 nM T18477 C3QA1U 155561308 IC50 = 150 nM T18477 C8R0WI 155561564 IC50 = 67060 nM T18477 C8JD0L 155561717 IC50 = 36620 nM T18477 C7L2RV 155562486 IC50 = 67 nM T18477 C1JQG6 155563956 IC50 = 1506 nM T18477 C0XJ5Q 155564241 IC50 = 22630 nM T18477 C40KVW 155565004 IC50 = 42410 nM T18477 C3J4AQ 155567472 IC50 > 10000 nM T18477 C3IU9Q 155567695 IC50 = 87 nM T18477 D05NWF 6022 EC50 = 120000 nM T18477 D07APP 131255 EC50 > 50000 nM T18477 D07TYL 1130 IC50 = 12500 nM T18477 D08OLB 49784944 IC50 = 3000 nM T18477 D0C2UJ 8974 IC50 <= 1250000 nM T18477 D0K0TJ 24772860 Ki = 4 nM T18477 D0T4MS 4369536 IC50 = 25 nM T18477 D0ZA6G 6323491 IC50 = 150 nM T72835 D02AUB 9811353 IC50 > 500000 nM T72835 CKM1X8 128677 IC50 = 50 nM T72835 C1GDY7 587790 IC50 = 31700 nM T72835 C96KNY 643990 IC50 = 300000 nM T72835 CXI3Y4 645569 IC50 > 100000 nM T72835 C5Q0FP 745480 IC50 = 49000 nM T72835 CYBV18 916176 IC50 = 27000 nM T72835 C16YNJ 962611 IC50 = 95000 nM T72835 COB6U4 2807642 IC50 = 3000 nM T72835 CYBK67 5481003 IC50 = 6600 nM T72835 CT3BF9 9797597 IC50 = 88 nM T72835 C74QCT 9798233 IC50 = 60 nM T72835 CCI90K 9799728 IC50 = 620 nM T72835 C18UGE 9818339 IC50 = 8400 nM T72835 CJQ2W6 9835897 IC50 > 1000 nM T72835 C6G5RT 9836507 IC50 > 4000 nM T72835 CUGN49 9836683 IC50 = 70 nM T72835 CJ5SU0 9839311 IC50 = 20 nM T72835 CSK6P4 9841875 IC50 = 500 nM T72835 C5DRX6 9856682 IC50 = 60 nM T72835 C9MA3Z 9858009 IC50 = 16 nM T72835 C0ZQV7 9858022 IC50 = 43 nM T72835 C3MG0X 9860649 IC50 = 690 nM T72835 C8IO4M 9878726 IC50 = 42000 nM T72835 C91VCO 9878930 IC50 = 20 nM T72835 CP34JF 9879093 IC50 = 600 nM T72835 C5S6CZ 9879529 IC50 = 6 nM T72835 CBKH73 9880710 IC50 = 100 nM T72835 C1L5WE 9880711 IC50 = 31 nM T72835 C0O5BM 9881984 IC50 = 2200 nM T72835 C0W1SB 9882382 IC50 = 660 nM T72835 CY7KG3 9883504 IC50 = 8 nM T72835 CL1FR4 9900816 IC50 = 1 nM T72835 C3D1XN 9900943 IC50 = 150 nM T72835 C9DHR2 9901085 IC50 = 800 nM T72835 CRND31 9901574 IC50 = 170 nM T72835 CBM7Y3 9903965 IC50 = 1800 nM T72835 CKJ7T0 9903998 IC50 = 22000 nM T72835 C1JI7S 9904207 IC50 = 4000 nM T72835 C3VJ9K 9904395 IC50 = 140 nM T72835 C62JUP 9904430 IC50 > 4000 nM T72835 CYN51E 9905179 IC50 = 12 nM T72835 CDML85 9906347 IC50 = 4 nM T72835 CO63ID 9921367 IC50 = 1700 nM T72835 CQ4WG3 9921987 IC50 = 100 nM T72835 C9T3ME 9922373 IC50 = 45 nM T72835 CO5L2R 9922793 IC50 = 76 nM T72835 C36KVQ 9922943 IC50 = 150 nM T72835 CW5P9J 9924766 IC50 = 100 nM T72835 C7QP1H 9944101 IC50 = 30 nM T72835 C2JZW5 9944163 IC50 = 55 nM T72835 C9AJP0 9944774 IC50 = 130 nM T72835 CL9I6U 9945784 IC50 = 19 nM T72835 CB3P7T 9946091 IC50 > 1000 nM T72835 CYJ59B 9946991 IC50 = 9 nM T72835 CAFK13 9947244 IC50 = 5 nM T72835 CR4LP3 9948282 IC50 = 16000 nM T72835 CNH47D 9948311 IC50 = 3200 nM T72835 C0YEQ7 9952465 IC50 = 120 nM T72835 C2TYQ1 9953413 IC50 > 100000 nM T72835 CWH3L0 9965679 IC50 = 20 nM T72835 CI4DU5 9966679 IC50 = 32 nM T72835 CFEI36 9967126 IC50 = 79 nM T72835 CA5W9Z 9967290 IC50 = 670 nM T72835 CS9DM3 9967511 IC50 = 340 nM T72835 CYXW91 9968489 IC50 = 44 nM T72835 CZ98HT 9977686 IC50 > 500000 nM T72835 CX30HT 10089338 IC50 = 0.7 nM T72835 C8TZ5Q 10101726 IC50 = 30000 nM T72835 C4E8NU 10106199 IC50 = 3300 nM T72835 COIF97 10107659 IC50 = 1400 nM T72835 CY23GM 10108997 IC50 = 200 nM T72835 C2P4UO 10110987 IC50 > 4000 nM T72835 CTW3P9 10116693 IC50 = 110 nM T72835 C07COW 10132518 IC50 = 80 nM T72835 C6N1FU 10134148 IC50 > 4000 nM T72835 CH49BD 10154440 IC50 = 630 nM T72835 COF2S9 10154441 IC50 = 20 nM T72835 CL7H2B 10154801 IC50 = 210 nM T72835 C0CP1T 10155661 IC50 = 300 nM T72835 CSB5F9 10156828 IC50 = 110 nM T72835 CF4DP2 10177047 IC50 = 60 nM T72835 C6RN4F 10178848 IC50 = 6 nM T72835 CHN3X1 10202790 IC50 > 4000 nM T72835 CD95KA 10221525 IC50 = 520 nM T72835 CJZU30 10267771 IC50 = 13 nM T72835 C2OQ0K 10267925 IC50 = 370 nM T72835 C9C0UG 10291112 IC50 > 4000 nM T72835 CWZU32 10291698 IC50 = 31 nM T72835 CTUP45 10291904 IC50 > 4000 nM T72835 CM05NG 10298900 IC50 = 120 nM T72835 C7KO6U 10361323 IC50 = 7 nM T72835 C1NX9Z 10469899 IC50 < 30000 nM T72835 CZ3DK8 10566084 IC50 = 17000 nM T72835 C5Q8EF 10566766 IC50 = 15000 nM T72835 CN3H5M 10632359 IC50 = 250 nM T72835 C6QZG3 10686899 IC50 > 4000 nM T72835 CZF1H3 10708446 IC50 = 200 nM T72835 CAPG02 10732433 IC50 > 1000 nM T72835 C6K5GC 10860379 IC50 = 21 nM T72835 CSO95L 10862219 IC50 = 864 nM T72835 C7OFZ9 10863087 IC50 = 120 nM T72835 C6PRJ8 10880644 IC50 = 35 nM T72835 C2VX3P 10886395 IC50 > 100000 nM T72835 CV9I3D 10891751 IC50 = 3 nM T72835 C9X6VP 10892285 IC50 = 940 nM T72835 C9DUB8 10892642 IC50 = 8 nM T72835 CS1T3C 10896625 IC50 = 115 nM T72835 CARC06 10904579 IC50 = 150 nM T72835 CHWL69 10905666 IC50 = 25 nM T72835 CLPA31 10906508 IC50 = 34 nM T72835 C7YG6L 10924566 IC50 = 28 nM T72835 CR51AV 10970154 IC50 = 4 nM T72835 CQ6E7Y 10970207 IC50 > 1000 nM T72835 CB31OE 10980658 IC50 = 870 nM T72835 C94UAC 10982608 IC50 = 4 nM T72835 CVR4Y3 11001541 IC50 = 25 nM T72835 CCP7K5 11013542 IC50 = 5 nM T72835 C1ZRL6 11014018 IC50 = 5 nM T72835 CIW6J5 11023935 IC50 = 13 nM T72835 C7NCE4 11036406 IC50 = 2 nM T72835 CM5HI8 11045962 IC50 = 6 nM T72835 C7U2JK 11048059 IC50 = 28 nM T72835 C7E6GN 11048585 IC50 = 600 nM T72835 CNHY70 11057712 IC50 = 35 nM T72835 COE6W0 11068095 IC50 = 2 nM T72835 C9Q0MP 11070710 IC50 = 650 nM T72835 CZSV01 11078679 IC50 = 470 nM T72835 C1KE2T 11079237 IC50 = 7 nM T72835 C8SRX4 11080157 IC50 > 715 nM T72835 C5T1BO 11089640 IC50 = 5 nM T72835 CQYV18 11091464 IC50 = 770 nM T72835 CSF94U 11102008 IC50 = 830 nM T72835 C51PTF 11109642 IC50 = 18 nM T72835 C8RF0J 11111846 IC50 > 1000 nM T72835 C8WI4X 11120977 IC50 = 380 nM T72835 CUGV75 11122788 IC50 > 1000 nM T72835 CHIT70 11134430 IC50 = 43 nM T72835 CRPC48 11134652 IC50 = 680 nM T72835 C4Z0FP 11258464 IC50 = 41900 nM T72835 CKHO40 11558561 IC50 > 50000000 nM T72835 CN5M7E 11680708 IC50 > 50000000 nM T72835 C5DUF4 11760748 IC50 = 110 nM T72835 CF7GU9 11777631 IC50 < 30000 nM T72835 C8BJ0L 11783098 IC50 = 180 nM T72835 C43LZD 11783922 IC50 = 870 nM T72835 CKRM28 11793014 IC50 > 1000 nM T72835 CLX8Z9 11825588 IC50 = 5 nM T72835 C7SG8X 11828434 IC50 = 2.8 nM T72835 C62DAO 16114614 IC50 = 800 nM T72835 C1ET3V 16114615 IC50 = 1000 nM T72835 CQ90BS 16114616 IC50 = 3300 nM T72835 CA4MJ7 16114618 IC50 = 8400 nM T72835 CWGO19 16114619 IC50 = 1300 nM T72835 CTC76N 16114620 IC50 = 8400 nM T72835 CM7Z2R 16115893 IC50 > 500000 nM T72835 C41WNZ 16116039 IC50 = 4900 nM T72835 CUE4D8 16116040 IC50 = 85400 nM T72835 C2EHS8 16116042 IC50 = 18700 nM T72835 CTG1J6 16116159 IC50 = 2300 nM T72835 CZH0G1 16116162 IC50 = 8700 nM T72835 C5GZB3 16116163 IC50 > 500000 nM T72835 CKI2E4 16116165 IC50 = 52400 nM T72835 C5Q4GR 16116166 IC50 > 500000 nM T72835 C7F1DY 16116286 IC50 = 48600 nM T72835 CU4OF0 16116421 IC50 > 500000 nM T72835 C89WXF 16116422 IC50 > 500000 nM T72835 C82KGR 16116555 IC50 > 500000 nM T72835 C9DME7 16116556 IC50 = 57200 nM T72835 CU2IB8 16116557 IC50 = 132000 nM T72835 CTXB17 16116558 IC50 > 500000 nM T72835 CFU0D9 16116559 IC50 = 113700 nM T72835 C7WJ0Y 16725848 IC50 = 9700 nM T72835 C5WSK1 23669281 IC50 = 3100 nM T72835 CC12EZ 23709469 IC50 = 280000 nM T72835 C36WMA 44264201 IC50 > 4000 nM T72835 CU30LF 44285871 IC50 = 10000000 nM T72835 C94VZY 44285873 IC50 = 8000000 nM T72835 C4J3NI 44285918 IC50 > 10000000 nM T72835 C7Y2QI 44285932 IC50 > 10000000 nM T72835 CXDS56 44285933 IC50 = 3000000 nM T72835 C4LNK6 44286072 IC50 = 1600000 nM T72835 CPW18X 44286163 IC50 = 6700000 nM T72835 C3KEI4 44286164 IC50 = 6000000 nM T72835 CU6T4G 44286241 IC50 = 7000000 nM T72835 C57VYM 44286390 IC50 = 6000000 nM T72835 CHF78N 44286451 IC50 = 7000000 nM T72835 CQP9G7 44304820 IC50 > 1000000 nM T72835 C5PC9B 44314807 IC50 = 2800000 nM T72835 C8V5HM 44314808 IC50 = 600000 nM T72835 C9YI8T 44314810 IC50 = 360000 nM T72835 C9FOU7 44314839 IC50 = 300000 nM T72835 C4FE2A 44314950 IC50 = 3000000 nM T72835 CMR6V4 44314968 IC50 = 3000000 nM T72835 C7S8PZ 44314993 IC50 > 2500000 nM T72835 CG2R9Y 44314996 IC50 > 2500000 nM T72835 CH5N4J 44315249 IC50 > 4000000 nM T72835 CZ06IY 44315261 IC50 = 3000000 nM T72835 C6JB5F 44315289 IC50 = 840000 nM T72835 CJN5S6 44315290 IC50 = 530000 nM T72835 CE18QO 44315291 IC50 = 950000 nM T72835 C7J8LN 44315330 IC50 = 350000 nM T72835 CECK48 44315332 IC50 > 10000000 nM T72835 CH40ER 44325713 IC50 = 500000 nM T72835 CB14NL 44325784 IC50 = 50000 nM T72835 CO3WB1 44325797 IC50 = 500000 nM T72835 CWCI90 44325812 IC50 = 1000000 nM T72835 CI6W5K 44325824 IC50 = 100000 nM T72835 C5ZGP4 44325830 IC50 = 100000 nM T72835 CX1PZ3 44325844 IC50 = 300000 nM T72835 C5FP7T 44325913 IC50 = 3000000 nM T72835 CH0YQ4 44325932 IC50 = 5000000 nM T72835 CC0DP9 44325956 IC50 = 900000 nM T72835 C4EQ5L 44325958 IC50 = 500000 nM T72835 CD1Y6W 44340382 IC50 > 1000000 nM T72835 CC7G9J 44340394 IC50 > 1000000 nM T72835 C2Q7LW 44340567 IC50 > 1000000 nM T72835 CZG4T2 44340638 IC50 > 1000000 nM T72835 CK1GA0 44340639 IC50 > 1000000 nM T72835 CM7P9U 44344139 IC50 = 13 nM T72835 CICW90 44356343 IC50 = 160000 nM T72835 C1VH5G 44356439 IC50 > 500000 nM T72835 CK7WE9 44356515 IC50 > 500000 nM T72835 CPM04F 44356616 IC50 > 500000 nM T72835 C8CR4F 44356617 IC50 > 500000 nM T72835 CL8M6C 44360868 IC50 > 10000000 nM T72835 C02ULA 44360870 IC50 > 10000000 nM T72835 CXK84H 44360912 IC50 > 10000000 nM T72835 CXL0S8 44387278 IC50 > 1000000 nM T72835 CIAL79 44387290 IC50 > 1000000 nM T72835 CHIF62 44387291 IC50 > 1000000 nM T72835 C6FK5A 44387293 IC50 = 240000 nM T72835 C7WPK9 44387294 IC50 = 360000 nM T72835 CPQ09T 44387295 IC50 > 1000000 nM T72835 CPT5K3 44387297 IC50 > 1000000 nM T72835 CS0M3D 44399068 IC50 > 50000000 nM T72835 C67QAL 44399069 IC50 > 50000000 nM T72835 C3TJ5S 44399147 IC50 > 50000000 nM T72835 CB74WV 44399232 IC50 > 50000000 nM T72835 CVDP57 44399253 IC50 > 50000000 nM T72835 C0ZIP8 44420653 IC50 = 3000 nM T72835 C5QXG3 44420654 IC50 = 3100 nM T72835 C2S9CH 44420657 IC50 = 61400 nM T72835 C8Y1HG 44420659 IC50 = 48000 nM T72835 CQ08EK 44420661 IC50 = 15700 nM T72835 CA9T5O 44420662 IC50 > 500000 nM T72835 C7F6HB 44456838 IC50 = 600000 nM T72835 CZG86H 44456859 IC50 = 1000000 nM T72835 CW8KR3 46845959 IC50 = 2500000 nM T72835 C8MUB4 46881482 IC50 = 11000000 nM T72835 CM2TE6 46881483 IC50 = 5000000 nM T72835 CE7OJ4 46881484 IC50 = 3000000 nM T72835 CS68ZT 46881485 IC50 = 5000000 nM T72835 COJ35S 46881517 IC50 = 15000000 nM T72835 C8Q0YB 46881518 IC50 = 6000000 nM T72835 C1RN8P 53323826 IC50 > 10000000 nM T72835 CK9Q2E 56675135 IC50 = 32000 nM T72835 C0BAV1 70687644 IC50 = 41000 nM T72835 C0MZH5 70687646 IC50 = 49000 nM T72835 CVM5H6 70689898 IC50 = 24000 nM T72835 CJA84B 70696227 IC50 = 1125000 nM T72835 CS1FC2 71450419 IC50 = 5460000 nM T72835 CEPH60 71452644 IC50 > 1000000 nM T72835 CN0ZI6 71458017 IC50 > 1000000 nM T72835 CGE8R2 71715994 IC50 = 16000 nM T72835 C7E0WX 71715999 IC50 = 2100000 nM T72835 C0FR3U 71716010 IC50 = 3500 nM T72835 C3S7VA 71716029 IC50 = 1000000 nM T72835 C3JQ6N 71716030 IC50 = 500000 nM T72835 CEO6H7 71716031 IC50 = 3200000 nM T72835 C6C0ZR 71716033 IC50 = 2000000 nM T72835 CHJ5U3 71716622 IC50 > 6600000 nM T72835 CJ2Q9U 71716626 IC50 = 1500000 nM T72835 C2RAX0 71716634 IC50 = 20000000 nM T72835 C1B3SM 71717205 IC50 > 10000000 nM T72835 C6IM8H 71717206 IC50 = 500000 nM T72835 CO9E1I 71717225 IC50 = 80000 nM T72835 CK27AE 71717234 IC50 = 1000000 nM T72835 CGQB06 71717239 IC50 = 20000000 nM T72835 CY37OD 71717829 IC50 = 1000000 nM T72835 CWQ63V 71717841 IC50 = 1400000 nM T72835 C8P0KB 71717843 IC50 = 2000000 nM T72835 C7NA8Z 71717847 IC50 = 20200000 nM T72835 C9BQW5 71717848 IC50 = 4600000 nM T72835 C1N3RG 71718477 IC50 > 6600000 nM T72835 C8KT6Z 71718487 IC50 = 36000000 nM T72835 CL25WA 71718488 IC50 = 6100000 nM T72835 CCO93Y 71719057 IC50 = 330000 nM T72835 CH42FQ 71719059 IC50 = 300000 nM T72835 CBLP16 71719067 IC50 = 4900000 nM T72835 C8MHG7 71719069 IC50 = 34400000 nM T72835 CQR6H7 71719671 IC50 = 500000 nM T72835 C2XBN3 71719672 IC50 = 400000 nM T72835 CF85XK 71719677 IC50 = 32000000 nM T72835 CPK9T0 71719678 IC50 = 11500000 nM T72835 C97AXO 71719679 IC50 = 14600000 nM T72835 CXZA30 71720268 IC50 = 2000000 nM T72835 C32CAX 71720271 IC50 = 4000000 nM T72835 CSMU14 71720272 IC50 = 5000000 nM T72835 C7XR6V 71720274 IC50 = 2500000 nM T72835 C23OXT 71720283 IC50 = 14000000 nM T72835 CTHW87 71720284 IC50 = 8000000 nM T72835 CCNR81 71720285 IC50 = 20000000 nM T72835 CGYI26 71720286 IC50 = 9500000 nM T72835 C53BRY 71720287 IC50 = 2600000 nM T72835 CP71RD 71720288 IC50 = 7000000 nM T72835 CL50FA 73351434 IC50 = 300000 nM T72835 CEH94N 73352890 IC50 = 80000 nM T72835 C3FIJ8 73354415 IC50 = 300000 nM T72835 CBCN75 73355970 IC50 = 2900000 nM T72835 C6MGQ0 73355972 IC50 = 1000000 nM T72835 C8TE5P 76335199 IC50 = 280000 nM T72835 CQ1W3X 90663369 IC50 = 16000000 nM T72835 C6CYV1 90664029 IC50 = 500000 nM T72835 CIU4H8 90664107 IC50 = 5000000 nM T72835 CO2DA9 90664124 IC50 = 600000 nM T72835 CKZP37 90664125 IC50 > 1000000 nM T72835 C1TG5J 90664143 IC50 = 350000 nM T72835 CJ63KL 90664145 IC50 > 10000000 nM T72835 C2QW4L 90664147 IC50 > 10000000 nM T72835 CM4V1J 90664149 IC50 > 10000000 nM T72835 CNQZ02 90664151 IC50 = 80000 nM T72835 CV8B6I 90664153 IC50 = 15800000 nM T72835 CL37TX 90664156 IC50 = 3800000 nM T72835 CXN0Q3 90664160 IC50 = 280000 nM T72835 C86TFW 90664161 IC50 = 650000 nM T72835 C7V9EN 90664162 IC50 = 590000 nM T72835 C5ZKM2 90664163 IC50 > 1000000 nM T72835 CMZK65 90664164 IC50 = 5000000 nM T72835 C2J7FQ 90664165 IC50 = 1000000 nM T72835 C49RXN 90664166 IC50 = 1150000 nM T72835 CUWF73 90664170 IC50 = 700000 nM T72835 CE1DY2 90664171 IC50 = 900000 nM T72835 C13WQJ 90664172 IC50 = 270000 nM T72835 C6VS3D 90664191 IC50 = 10000 nM T72835 CO85IQ 90664193 IC50 = 30000 nM T72835 C90MHO 90664197 IC50 = 60000 nM T72835 C84CFR 90664199 IC50 = 37000 nM T72835 C1NKI3 90664201 IC50 = 1500 ug.mL-1 T72835 C9XAE4 90664202 IC50 = 100 ug.mL-1 T72835 CBI07N 90664204 IC50 = 30000 nM T72835 CKIU49 90664206 IC50 = 200000 nM T72835 CDVW23 90664222 IC50 = 700000 nM T72835 CJ4FT2 90664262 IC50 = 700000 nM T72835 CJ3O0E 90664264 IC50 = 3500 nM T72835 C6KN7R 90664265 IC50 > 100000 nM T72835 CF9XM7 118714544 IC50 = 2080000 nM T72835 CZU9S3 118714545 IC50 = 140000 nM T72835 C6G1LI 118714546 IC50 = 220000 nM T72835 CIF1K3 118714547 IC50 = 76000 nM T72835 CDYU78 118718895 IC50 = 4300 nM T72835 C1A5QG 118718900 IC50 = 13000 nM T72835 CK6Q9M 118718901 IC50 = 1500 nM T72835 C15YGB 118719302 IC50 > 1000000 nM T72835 CI3VJ0 118719304 IC50 > 100000 nM T72835 CZH6T3 118719305 IC50 > 1000000 nM T72835 C4BGF1 118719306 IC50 > 100000 nM T72835 C2FX6G 135506443 IC50 = 20000 nM T72835 D0E9NT 11874 IC50 > 500000 nM T72835 D0Y3TZ 370 IC50 > 500000 nM T32973 CI0DG1 764318 IC50 = 180 nM T32973 CPA63I 3107941 Ki = 105 nM T32973 C6SO2K 3708081 IC50 = 170 nM T32973 CRT04P 44298904 IC50 = 31 nM T32973 CCLG83 44298942 IC50 = 55 nM T32973 CVE6Z8 44299051 IC50 = 1000 nM T32973 CLC74A 44299052 IC50 = 38 nM T32973 C3DRB6 45496892 IC50 = 160 nM T32973 CU3WO1 90656770 IC50 = 140 nM T32973 CUZ5D8 90656771 IC50 = 192 nM T32973 CA0I4Q 90656772 IC50 = 108 nM T32973 CHD13U 90656773 IC50 = 282 nM T32973 C7CZK1 90656774 IC50 = 138 nM T32973 CMBD94 90656775 IC50 = 18 nM T32973 CH1LG5 90656776 IC50 = 49 nM T32973 C9YW4M 90656777 IC50 = 28 nM T32973 C0YFV2 90656778 IC50 = 169 nM T32973 C4BNV6 90656779 IC50 = 49 nM T32973 C8GMB3 90656780 IC50 = 97 nM T32973 C6ZT9S 90656781 IC50 = 83 nM T32973 C4LC5K 90656782 IC50 = 348 nM T32973 CV0ZW9 90656783 IC50 = 60 nM T32973 CS83DE 90656784 IC50 = 5 nM T32973 CC0HQ5 90656785 IC50 = 79 nM T32973 C6RU7O 90656786 IC50 = 29 nM T32973 CIY4S9 90656787 IC50 = 11 nM T32973 C01DTE 90656788 IC50 = 41 nM T32973 CV98QR 90656789 IC50 = 9 nM T32973 C5UV6T 90656790 IC50 = 124 nM T32973 C9O6FJ 90656791 IC50 = 1640 nM T32973 CN7BQ9 90656792 IC50 = 65 nM T32973 C2O9IM 90656793 IC50 = 15 nM T32973 C0U3KA 90656794 IC50 = 41 nM T32973 C0AZ6Q 90656795 IC50 = 3.2 nM T32973 C89FRT 90656797 IC50 = 7.8 nM T32973 CFB02X 90656798 IC50 = 343 nM T32973 C6E0RT 90656799 IC50 = 9 nM T32973 CV04JO 127037715 IC50 = 71 nM T32973 C6MQI3 127038634 IC50 > 10000 nM T32973 CM1CO8 127038635 IC50 = 356 nM T32973 C3WYE0 127038636 IC50 > 10000 nM T32973 CW6F1G 127038637 IC50 = 128 nM T32973 C09UKF 127038638 IC50 = 2259 nM T32973 C8JGW4 127038639 IC50 = 1035 nM T32973 CO7I3Q 127038645 IC50 > 10000 nM T32973 CBIQ30 127038646 IC50 = 323 nM T32973 CDO09Y 127038719 IC50 = 73 nM T32973 C38JYQ 127038989 IC50 = 1459 nM T32973 CC2O5W 127038990 IC50 = 252 nM T32973 C5VE8N 127038991 IC50 = 6296 nM T32973 CW89HP 127038992 IC50 = 1359 nM T32973 C8Z3HL 127039269 IC50 = 882 nM T32973 CU57WL 127039270 IC50 = 5050 nM T32973 C4JR2O 127039271 IC50 = 5854 nM T32973 C3FYV7 127039330 IC50 = 9249 nM T32973 CA9I0O 127039395 IC50 = 269 nM T32973 C2EX1W 127039396 IC50 > 10000 nM T32973 CH7P9N 127039594 IC50 = 4384 nM T32973 CGY9L1 127039595 IC50 = 7749 nM T32973 C7QP0E 127039715 IC50 = 282 nM T32973 C1MN6H 127039716 IC50 > 10000 nM T32973 C65YMT 127039717 IC50 = 332 nM T32973 CV3DF7 127039734 IC50 = 67 nM T32973 CQ69EI 127039735 IC50 = 23 nM T32973 CUQ5H2 127039930 IC50 > 10000 nM T32973 C4B3JS 127039931 IC50 > 10000 nM T32973 CN73ZO 127039932 IC50 = 3889 nM T32973 CJ9IQ8 127040049 IC50 > 10000 nM T32973 C8RPF9 127040057 IC50 = 49 nM T32973 C63WGY 127040119 IC50 = 6 nM T32973 C5Y8BK 127040330 IC50 = 1086 nM T32973 C1PR6T 127040663 IC50 > 10000 nM T32973 CKS4F0 127040664 IC50 = 6745 nM T32973 C9P4CX 127040726 IC50 = 33 nM T32973 C5G2EC 127040909 IC50 > 10000 nM T32973 CH1FG6 127040984 IC50 = 2272 nM T32973 CL9DB6 127040985 IC50 = 1818 nM T32973 C8Y3RC 127040986 IC50 > 10000 nM T32973 CF23HM 127040987 IC50 > 10000 nM T32973 CSF23D 127041612 IC50 = 425 nM T32973 CE5N9Z 127041613 IC50 = 601 nM T32973 CD8BP0 127041614 IC50 > 10000 nM T32973 CD2XR0 127041615 IC50 = 378 nM T32973 CO0NJ1 127041616 IC50 = 5854 nM T32973 C5DKU9 127041617 IC50 = 586 nM T32973 CEHK53 127041618 IC50 > 10000 nM T32973 CEL1O2 127041744 IC50 = 169 nM T32973 C9Q8DT 127041745 IC50 = 93 nM T32973 C9JOV0 127041985 IC50 = 593 nM T32973 CH19UD 127042050 IC50 = 121 nM T32973 CJ27CG 127042051 IC50 = 6 nM T32973 CVE08P 127042052 IC50 = 73 nM T32973 CIE83Y 127042053 IC50 = 969 nM T32973 CAT46D 127042341 IC50 = 12 nM T32973 CN1M5T 127042410 IC50 > 10000 nM T32973 CO2IY7 127042411 IC50 = 33 nM T32973 CW2F7T 127042682 IC50 = 47 nM T32973 CZ3BE8 127042683 IC50 = 35 nM T32973 CD42KE 127042684 IC50 = 45 nM T32973 C2C9DK 127042738 IC50 = 32 nM T32973 C36SAQ 127042739 IC50 = 71 nM T32973 CNTF18 127042740 IC50 = 5 nM T32973 C1F2AW 155512129 IC50 = 34 nM T32973 CPJK82 155512819 IC50 = 82 nM T32973 C5OGP9 155513654 IC50 = 0.26 nM T32973 CBGY41 155515971 IC50 = 59 nM T32973 C64OMX 155518715 IC50 = 18 nM T32973 C5KH2Y 155523364 IC50 = 7.1 nM T32973 CGI0C3 155529023 IC50 = 15 nM T32973 C6F1JL 155532513 IC50 = 280 nM T32973 CETH73 155533920 IC50 = 9.8 nM T32973 C03EVD 155535966 IC50 = 5.5 nM T32973 C67DMO 155536395 IC50 = 15 nM T32973 C3BWI8 155537675 IC50 = 3.6 nM T32973 CKR9O0 155540299 IC50 = 10 nM T32973 CTG0X5 155540609 IC50 = 12 nM T32973 CZT36F 155541834 IC50 = 290 nM T32973 CW5IN2 155542032 IC50 = 33 nM T32973 CMV89O 155544241 IC50 = 160 nM T32973 CKZI03 155549215 IC50 = 78 nM T32973 C6IQO0 155550525 IC50 = 26 nM T32973 CS35NF 155550740 IC50 = 1.3 nM T32973 C2B7KY 155552502 IC50 = 1.4 nM T32973 CL40SZ 155553142 IC50 = 0.12 nM T32973 C3ZO7Y 155556864 IC50 = 870 nM T32973 CF5HV2 155557380 IC50 = 0.47 nM T32973 C2IUT6 155558910 IC50 > 10000 nM T32973 CQ08FY 155562629 IC50 = 110 nM T32973 C54SNK 155567233 IC50 = 96 nM T32973 D0W6HI 90656796 IC50 = 0.9 nM T92689 D01BYB 5957 EC50 = 3300 nM T92689 D06ACW 6083 EC50 = 17250 nM T92689 D0H2UB 5361 Ki = 112.2 nM T92689 D0KE4Z 5310954 EC50 = 1500 nM T92689 D0Z7FU 6133 EC50 > 100000 nM T92689 CPQ81V 171069 EC50 = 4500 nM T92689 CCJ8P0 440317 EC50 = 63.1 nM T92689 C18IQO 10080003 Ki = 7585.78 nM T92689 C04CWB 10080210 Ki = 1000 nM T92689 CA8GR7 10080218 Ki = 446.68 nM T92689 C3L6KW 10994891 EC50 = 17250 nM T92689 CHB3C7 11510273 Ki > 15000 nM T92689 CT74ZJ 11560464 Ki > 15000 nM T92689 CGQV15 11564436 Ki = 107.15 nM T92689 CUD1J5 11611428 Ki > 15000 nM T92689 CX7J8F 11636756 Ki = 44.67 nM T92689 C10PSW 11679780 Ki = 2398.83 nM T92689 CQ40BH 14753886 EC50 = 900 nM T92689 CCZ8N0 16155349 Ki = 75.86 nM T92689 CN4BT9 16163319 Ki = 302 nM T92689 C56DVM 23656757 EC50 = 478.63 nM T92689 CM45HO 23656759 EC50 = 1288.25 nM T92689 CQ46IG 44353592 EC50 = 7000 nM T92689 C30CIT 49856886 EC50 = 13000 nM T92689 CJ2RM6 56673378 EC50 >= 40000 nM T92689 C4VFI2 68530100 Ki > 15000 nM T92689 CJK95G 71450314 EC50 = 2900 nM T92689 CL0X8W 73347374 EC50 = 1400 nM T92689 CLXM46 73351984 EC50 = 1000 nM T92689 C9CWV3 73353445 EC50 = 130 nM T92689 C1AJ6L 73354953 EC50 = 1500 nM T92689 CAS84P 76324375 EC50 > 100000 nM T92689 C78INB 118725181 EC50 = 3680 nM T92689 CM8N4I 122195891 EC50 = 1000 nM T92689 CULF46 122195892 EC50 = 500 nM T92689 CC2JO4 122195893 EC50 = 1100 nM T92689 C9HK0N 122195894 EC50 = 900 nM T92689 CZ1XL2 122195895 EC50 = 1000 nM T92689 D05MXI 42611190 IC50 > 10000 nM T92689 D05NWF 6022 EC50 = 1700 nM T92689 D07MTB 11510579 Ki > 15000 nM T92689 D0B0ZQ 9875920 EC50 > 100000 nM T92689 D0D8CZ 15993 EC50 = 9000 nM T92689 D0U1OJ 5310983 EC50 = 50000 nM T92689 D0V4GQ 5310996 EC50 = 30000 nM T28484 D0X5SI 193653 IC50 > 63000 nM T28484 D02AAO 10368812 IC50 = 429 nM T28484 D04VWJ 44224257 IC50 = 6 nM T28484 D0L4VI 5862 IC50 > 63000 nM T28484 D0PW4N 6851740 IC50 = 1.2 nM T28484 D0Q5QC 23634407 IC50 = 8 nM T28484 D0W9SL 25167017 IC50 = 7 nM T28484 D0Z0HH 3503 IC50 = 25000 nM T28484 D02CXZ 57094730 Ki = 203 nM T28484 C8V5EI 9720 IC50 = 3200 nM T28484 CG9LF7 21261 IC50 > 63000 nM T28484 C6UFG1 23011 IC50 = 23000 nM T28484 C2AJZ0 37323 Ki = 200 nM T28484 CI5X0C 76044 Ki = 26 nM T28484 C8U9DP 83278 IC50 > 20000 nM T28484 C43JDE 99558 IC50 > 63000 nM T28484 CLN9B4 128239 IC50 = 55000 nM T28484 C19ZNI 207753 IC50 > 50000 nM T28484 CD54OR 215628 Ki = 1750 nM T28484 CB09MQ 246378 IC50 = 5600 nM T28484 CCLD38 262764 Ki = 150 nM T28484 CNVZ38 277164 Ki = 5230 nM T28484 CQ20WF 282773 IC50 = 25000 nM T28484 CT9MH5 283741 Ki = 2536.3 nM T28484 CON03C 303820 IC50 = 1000 nM T28484 C9WSY2 391237 EC50 < 30000 nM T28484 C31NSG 541056 IC50 = 2500 nM T28484 CCL43Q 613965 IC50 = 10000 nM T28484 C15QBR 675901 EC50 < 30000 nM T28484 C9CBS4 686905 IC50 = 493 nM T28484 CUR7M6 692940 EC50 = 20000 nM T28484 C2B9ZV 703864 EC50 < 30000 nM T28484 CI6N1Q 806204 EC50 = 3600 nM T28484 CJ4G8Y 806211 EC50 = 2200 nM T28484 CY3A5N 1049743 EC50 = 34000 nM T28484 CX7H0T 1190622 EC50 = 540 nM T28484 C48ADI 1190625 EC50 = 480 nM T28484 CU4PQ6 1204119 EC50 = 1800 nM T28484 C72ACT 1350845 EC50 = 5800 nM T28484 C5V1EH 2729933 IC50 = 20000 nM T28484 CTM84I 2782719 IC50 > 20000 nM T28484 CGQC14 2794294 Ki = 2659.4 nM T28484 CI6JW8 2828030 IC50 = 4300 nM T28484 C8TD6I 2849314 IC50 = 14000 nM T28484 C8J4WG 2854045 EC50 = 2600 nM T28484 CT85GW 2916332 IC50 = 1700 nM T28484 CW9O2K 2930014 IC50 = 740 nM T28484 C0T8FE 3149846 IC50 = 37200 nM T28484 CVC13H 3152075 IC50 = 5100 nM T28484 CZ02NA 3158674 IC50 = 6300 nM T28484 CK53GC 3250498 IC50 = 8500 nM T28484 C01HNZ 3333657 IC50 = 6900 nM T28484 CZ0Y4W 4252653 IC50 = 950 nM T28484 C8M6EO 4368463 IC50 = 5490 nM T28484 C0L8TM 4595895 IC50 = 15600 nM T28484 CO17EG 5015306 IC50 = 37600 nM T28484 CQ8U7S 5205832 IC50 = 40180 nM T28484 COFC26 5546231 IC50 = 134 nM T28484 CR54XC 5777336 IC50 = 4600 nM T28484 CPV72R 6102824 IC50 = 2 nM T28484 CC8W0A 6857690 IC50 = 104 nM T28484 CJZ03U 6951058 IC50 > 63000 nM T28484 CQE2S4 7009563 IC50 > 63000 nM T28484 CWV64N 7019695 IC50 > 63000 nM T28484 CQM5F8 7271796 Ki = 98.6 nM T28484 C9ZP2B 7408363 IC50 > 63000 nM T28484 CZAN92 7472794 Ki = 9.1 nM T28484 C2R8BH 9541651 IC50 = 79100 nM T28484 CSI60M 9826132 IC50 = 16 nM T28484 CLV23Q 9860103 IC50 = 9700 nM T28484 CZ2AS9 9872853 IC50 = 80 nM T28484 C5WNF7 9883349 IC50 = 450 nM T28484 COP96L 9936388 Ki = 0.5 nM T28484 CDCM57 10094631 IC50 = 23000 nM T28484 C6IVA1 10149544 IC50 = 94 nM T28484 CG1UO8 10171750 IC50 = 9800 nM T28484 CYQ3O8 10172040 IC50 = 1200 nM T28484 CH5FK7 10172108 IC50 = 1800 nM T28484 C89RTM 10193550 IC50 = 903 nM T28484 C0HA8L 10195027 IC50 = 585 nM T28484 C4X6CV 10195768 IC50 = 100 nM T28484 CFVG49 10215371 IC50 = 1100 nM T28484 CG32IU 10220615 IC50 = 18400 nM T28484 CAI34D 10236493 IC50 = 3600 nM T28484 C5LI3A 10236645 IC50 = 51 nM T28484 COM49U 10238126 IC50 = 122 nM T28484 CHGS73 10286584 IC50 = 84 nM T28484 C2L7MH 10308676 IC50 = 284 nM T28484 C61ZHJ 10309476 IC50 = 44 nM T28484 C92FJO 10309662 IC50 = 55 nM T28484 CG42HR 10310151 IC50 = 103 nM T28484 CIUH41 10357373 IC50 = 4000 nM T28484 CYA1F4 10390836 IC50 = 51 nM T28484 CIE20X 10429690 Ki = 120 nM T28484 CY9F6J 10665491 EC50 = 294 nM T28484 C1D7CQ 10968573 IC50 = 720 nM T28484 CAI5X4 10989172 IC50 > 10000 nM T28484 C80FNI 11151953 IC50 = 170 nM T28484 CYW48K 11163025 IC50 = 120 nM T28484 CN3VF5 11163393 IC50 = 110 nM T28484 C7PQ1X 11163979 IC50 = 502 nM T28484 C9NJ1E 11167161 IC50 > 63000 nM T28484 C1JZX8 11175005 IC50 = 685 nM T28484 CC60IS 11176379 IC50 = 319 nM T28484 CZD62W 11185891 IC50 = 130 nM T28484 C7D0RG 11189426 IC50 = 860 nM T28484 C8KO4G 11232296 IC50 = 6000 nM T28484 CHL4C9 11232827 IC50 = 349 nM T28484 CT18DU 11244423 IC50 = 167 nM T28484 CUS5X6 11244531 IC50 = 15 nM T28484 CJL85B 11261882 IC50 = 49 nM T28484 CAY58Q 11278857 IC50 = 120 nM T28484 C76WDK 11280370 IC50 = 67 nM T28484 C4KOJ2 11290427 IC50 = 1422 nM T28484 CE65DY 11300450 IC50 = 420 nM T28484 CSX9R5 11325207 IC50 = 40 nM T28484 C0W9YB 11336022 Ki = 110 nM T28484 CVIO67 11337670 IC50 = 39 nM T28484 C61VAJ 11348021 IC50 = 31 nM T28484 CDVR87 11348100 IC50 = 792 nM T28484 CEI5U8 11351844 IC50 = 120 nM T28484 C63JHU 11359430 IC50 = 141 nM T28484 CC3VS1 11359945 IC50 = 66 nM T28484 CX1Q6E 11382921 IC50 = 86 nM T28484 CHR14M 11392225 IC50 = 130 nM T28484 CY32TM 11393385 IC50 = 24 nM T28484 CUB4A2 11405234 IC50 = 1448 nM T28484 CH4O8V 11417613 IC50 = 176 nM T28484 CS48KQ 11427185 IC50 = 482 nM T28484 CU5XJ8 11428074 IC50 = 67 nM T28484 CKY2G7 11439836 IC50 = 28 nM T28484 CH6J7A 11450574 IC50 = 34 nM T28484 C64QZF 11461630 IC50 = 2518 nM T28484 CXR6L7 11472221 IC50 = 500 nM T28484 C58GVP 11473294 IC50 = 196 nM T28484 CU5Q4D 11473399 IC50 = 1795 nM T28484 C41CXQ 11484241 IC50 = 25 nM T28484 C5ZR9B 11492539 IC50 = 270 nM T28484 C4D6GJ 11493466 Ki = 330 nM T28484 CV41ER 11494867 IC50 = 1.8 nM T28484 C4ZLJ2 11496836 IC50 = 5 nM T28484 C1W8SH 11497413 IC50 = 4.7 nM T28484 C18KEB 11507070 IC50 = 550 nM T28484 CV4IZ7 11509189 EC50 = 3.2 nM T28484 CQEZ41 11514833 IC50 = 85 nM T28484 CTA7M3 11517739 IC50 = 4.3 nM T28484 CC19SE 11518697 IC50 = 3.9 nM T28484 C78DKQ 11539390 IC50 = 1 nM T28484 CF52ZB 11545686 IC50 = 1.6 nM T28484 CHT8D7 11547260 IC50 = 2.8 nM T28484 CL9OM0 11552755 IC50 = 2.1 nM T28484 CJ0U7Q 11577209 EC50 = 208 nM T28484 CVIP95 11582321 IC50 = 1 nM T28484 C42QMA 11590877 IC50 = 3.8 nM T28484 CM4Q2B 11597510 IC50 = 4 nM T28484 C6KVY0 11598137 IC50 = 0.9 nM T28484 C1WI4H 11611859 IC50 = 0.4 nM T28484 CD2H3T 11624832 IC50 = 5.2 nM T28484 C3M2LO 11626574 EC50 = 368 nM T28484 CV7F1O 11626838 EC50 = 27 nM T28484 CJBR83 11634073 IC50 = 1.5 nM T28484 C98YKB 11653811 IC50 = 0.2 nM T28484 CGU87J 11654962 IC50 = 1 nM T28484 CKP76R 11662966 IC50 = 1.6 nM T28484 CV62EQ 11666731 IC50 = 155 nM T28484 CMW4Y3 11668820 IC50 = 1.8 nM T28484 C29PWK 11675645 IC50 = 2.6 nM T28484 CT92YC 11680877 IC50 = 120 nM T28484 CKH1U0 11687592 IC50 > 20000 nM T28484 CWX2F0 11696319 IC50 = 0.5 nM T28484 CD0V1M 11709173 Ki = 6.8 nM T28484 CC74PN 11718862 IC50 = 1.8 nM T28484 C3FP8J 11720191 IC50 = 1 nM T28484 C70FVG 11738796 IC50 = 1100 nM T28484 CVYG50 11739086 IC50 = 2780 nM T28484 CG4Z7P 11771970 Ki = 3.5 nM T28484 CS5XA3 11772457 IC50 = 20 nM T28484 C4MJS7 11840968 IC50 = 38 nM T28484 CRSJ15 11848366 IC50 = 0.82 nM T28484 CGA83V 11853779 IC50 = 100 nM T28484 CJO8L1 11858360 IC50 = 64 nM T28484 C74LXB 11858424 IC50 = 110 nM T28484 C9YX7P 12000936 Ki = 1.4 nM T28484 CZ38QX 12984537 IC50 > 20000 nM T28484 CI30WH 13008994 Ki = 21.5 nM T28484 C0PXW1 13830550 Ki = 2157.6 nM T28484 C0YBV3 13943580 Ki = 750 nM T28484 CZ6O1D 14081820 IC50 > 63000 nM T28484 C3KP6Q 14741508 IC50 > 50000 nM T28484 C0TLA5 14855134 IC50 > 6300 nM T28484 C9ZO7G 15604796 IC50 = 1.9 nM T28484 CVKB58 15942673 IC50 = 110 nM T28484 CLD0M2 15949839 IC50 = 7 nM T28484 CUS3W4 15950258 IC50 = 7.4 nM T28484 CY09XF 15984121 IC50 = 60 nM T28484 C8F9HI 16122639 EC50 = 1700 nM T28484 C1V0YD 18686366 IC50 = 6800 nM T28484 C1QTG3 19589351 IC50 = 1900 nM T28484 CFIY91 20100158 IC50 = 1470 nM T28484 C1AFL3 21117270 Ki = 1500 nM T28484 C7FT6V 21140145 Ki < 50 nM T28484 CVZ7G3 21140146 Ki = 2000 nM T28484 CBA68L 21144445 Ki = 4.2 nM T28484 CYJ46Z 21144451 Ki = 600 nM T28484 CLJ56D 21144473 Ki = 14000 nM T28484 COXV07 22179981 IC50 = 70 nM T28484 C8X0MA 22179983 IC50 = 330 nM T28484 CXH2R9 22179996 IC50 = 60 nM T28484 CU9M1H 22180000 IC50 > 25000 nM T28484 C41IWK 22180008 IC50 = 3720 nM T28484 C0E6HG 22180029 IC50 = 100 nM T28484 CBV96L 22180034 IC50 = 1920 nM T28484 CPK6E5 22180046 IC50 = 290 nM T28484 CK7A3G 22180056 IC50 = 650 nM T28484 CM5A6D 22180071 IC50 = 60 nM T28484 C8EO1I 22185227 IC50 = 52 nM T28484 CTE52X 22577556 IC50 = 41500 nM T28484 C0RA2X 23625977 IC50 > 20000 nM T28484 C73MLP 23625981 IC50 > 20000 nM T28484 CHD2W4 23625982 IC50 = 840 nM T28484 C82PAY 23625983 IC50 > 20000 nM T28484 C3FQI4 23625984 IC50 > 20000 nM T28484 CGHE36 23626137 IC50 = 118 nM T28484 CA9JV8 23626138 IC50 > 20000 nM T28484 C8OF6I 23626140 IC50 > 20000 nM T28484 C5E7MR 23626141 IC50 > 20000 nM T28484 C32QNZ 23626142 IC50 > 20000 nM T28484 C4HC0U 23626448 IC50 = 2470 nM T28484 CY1QW4 23628220 EC50 = 100 nM T28484 C87DFY 24806224 Ki = 450 nM T28484 C80ABE 24806225 Ki < 50 nM T28484 CF9B4Q 24806226 Ki = 150 nM T28484 C25EDC 24806227 Ki = 175 nM T28484 CK8NI7 24860487 Ki = 2500 nM T28484 C1IJZ4 24860488 Ki = 4000 nM T28484 CURN19 24860489 Ki = 7000 nM T28484 CU0ZL5 24860490 Ki = 600 nM T28484 C0ADM2 24860491 Ki = 1500 nM T28484 CM52YG 24860492 Ki = 6750 nM T28484 C53JWM 24860493 Ki = 150 nM T28484 CRVG54 24860494 IC50 = 26.8 nM T28484 CEVI14 24860495 Ki = 13.6 nM T28484 CX83YD 24860496 Ki = 23000 nM T28484 CKX7A6 24860497 Ki = 35000 nM T28484 CW4SJ6 24860498 Ki = 23000 nM T28484 CAY0Z3 24860499 Ki = 1000 nM T28484 C3UT1C 24860500 Ki = 1500 nM T28484 CBA6Q2 24860501 Ki = 13000 nM T28484 C73OHZ 24860502 Ki = 6000 nM T28484 C61VPR 24860504 Ki = 900 nM T28484 CP63DU 24901489 IC50 = 85 nM T28484 C9E0OD 24901490 IC50 = 113 nM T28484 CT8GA0 24901491 IC50 = 50 nM T28484 CY3C1U 24901492 IC50 = 16 nM T28484 CC2GE7 24901493 IC50 = 5.2 nM T28484 CFM1P2 24901494 IC50 = 3.6 nM T28484 CIN21Y 24901495 IC50 = 3100 nM T28484 CF24OR 24901496 IC50 = 2.7 nM T28484 CAUZ61 24901497 IC50 = 11 nM T28484 C7IQO2 24901498 IC50 = 24.7 nM T28484 C8QOY5 24901499 IC50 = 3140 nM T28484 C93PNA 24901500 IC50 = 606 nM T28484 CBG32M 24901501 IC50 = 745 nM T28484 C2E1YR 24901502 IC50 = 697 nM T28484 CC54GX 24901503 IC50 = 390 nM T28484 CA0R5M 24901504 IC50 = 67 nM T28484 C07IFO 24901505 IC50 = 119 nM T28484 CANF39 24901506 IC50 = 892 nM T28484 CY38XS 24901507 IC50 = 391 nM T28484 CMC52T 24901508 IC50 = 552 nM T28484 C0XHP1 24901509 IC50 = 686 nM T28484 CS3W4I 24901510 IC50 = 8 nM T28484 CBV2S9 24901511 IC50 = 26 nM T28484 CN2K8P 24901512 IC50 = 85 nM T28484 CX5TH2 24901513 IC50 = 4 nM T28484 C6YGU7 24901514 IC50 = 16.5 nM T28484 CY3EB5 24901515 EC50 = 53 nM T28484 CTHL35 24901516 IC50 = 5.2 nM T28484 C1V3QA 24901517 IC50 = 3.8 nM T28484 COCN23 24901519 IC50 = 8230 nM T28484 CJ8LU2 24901520 IC50 = 25200 nM T28484 CBGF57 24901521 IC50 = 11000 nM T28484 CY1CW5 24901522 IC50 > 25000 nM T28484 CML92E 24901523 IC50 = 2270 nM T28484 CAM5I2 24901524 IC50 = 3060 nM T28484 CK1UJ2 24901525 IC50 = 4650 nM T28484 CO1Z9X 24901526 IC50 > 25000 nM T28484 C3QHP5 24901527 IC50 = 8880 nM T28484 CDYR21 24901528 IC50 = 5360 nM T28484 CQXW01 24901529 IC50 = 17900 nM T28484 CJK3F0 24901530 IC50 = 16400 nM T28484 CCHV96 24901531 IC50 > 25000 nM T28484 CV59OA 24901532 IC50 = 14400 nM T28484 CH0J7C 24901533 IC50 > 25000 nM T28484 C7J3LO 24901534 IC50 > 25000 nM T28484 CY05BM 24901535 IC50 > 25000 nM T28484 C3KUV2 24901536 IC50 = 2750 nM T28484 CZ04WL 24901537 IC50 = 22300 nM T28484 CTY2R8 24901538 IC50 = 12800 nM T28484 C5V6ZS 24901539 IC50 = 5440 nM T28484 C7QOX2 24901540 IC50 = 306 nM T28484 C3EDI4 24901541 IC50 > 25000 nM T28484 CT6N0Z 24901542 IC50 = 13200 nM T28484 C4D2NY 24901543 IC50 = 3480 nM T28484 CY0P8H 24901544 IC50 > 25000 nM T28484 C5WQ9S 24901545 IC50 > 25000 nM T28484 C3RY1T 24901546 IC50 = 2490 nM T28484 CE56RM 24901547 IC50 = 808 nM T28484 C9AL2E 24901548 IC50 = 317 nM T28484 C79OHQ 24901549 IC50 = 595 nM T28484 CF14PC 24901550 IC50 = 617 nM T28484 C7N0YQ 24901551 IC50 > 25000 nM T28484 CT4G9C 24901552 IC50 > 25000 nM T28484 C97OEW 24901553 IC50 > 25000 nM T28484 C58DLP 24901554 IC50 = 4710 nM T28484 CY5TL9 24901555 IC50 = 344 nM T28484 CCBU08 24901556 IC50 = 1780 nM T28484 C5R6AJ 24901557 IC50 = 12800 nM T28484 CR61YE 24901558 IC50 = 1270 nM T28484 C1FPG9 24901560 IC50 = 639 nM T28484 C8T5CB 24901561 EC50 < 30000 nM T28484 CT1H2D 24901562 EC50 = 29000 nM T28484 C1D4VU 24901563 EC50 = 4300 nM T28484 C1C8HQ 24901564 IC50 = 76000 nM T28484 CG0O1W 24901565 IC50 = 17000 nM T28484 C7SFY5 24901567 EC50 = 1100 nM T28484 C15JND 24901568 EC50 = 37000 nM T28484 CSGI87 24901569 EC50 = 7600 nM T28484 CE43VJ 24901570 EC50 = 4700 nM T28484 COPT12 24901571 EC50 = 5400 nM T28484 C13QJL 24901572 EC50 = 1500 nM T28484 CP7C8W 24901573 IC50 = 12000 nM T28484 CBN3V7 24901574 EC50 = 1900 nM T28484 C8IC1E 24901575 IC50 = 69000 nM T28484 C10ZYD 24901576 EC50 = 17000 nM T28484 C9QA1U 24901577 IC50 = 3300 nM T28484 CH4T2K 24901578 EC50 < 30000 nM T28484 CXO6N4 24901579 EC50 < 30000 nM T28484 C5BL4Q 25014675 IC50 = 14800 nM T28484 C69ZRO 25014747 Ki < 50 nM T28484 COX3F5 25014748 IC50 = 514.2 nM T28484 CCI29G 25014750 IC50 = 680 nM T28484 CAW3B7 25014751 IC50 > 63000 nM T28484 C53QJP 25015247 IC50 = 230 nM T28484 CPLY38 25164463 IC50 > 20000 nM T28484 CAXQ03 25164661 IC50 = 7400 nM T28484 CRU76E 25164662 IC50 > 20000 nM T28484 C3NVW5 25165471 IC50 = 2500 nM T28484 CV6Y1Z 25165472 IC50 = 5000 nM T28484 CVMZ57 25165473 IC50 = 6900 nM T28484 CF9KY4 25165474 IC50 = 4800 nM T28484 CIWL28 25165475 IC50 = 1400 nM T28484 CPV3O6 25165666 IC50 = 458.8 nM T28484 C56QHJ 25165854 IC50 = 1300 nM T28484 C37LFS 25166248 IC50 = 7900 nM T28484 C25CJK 25184242 IC50 = 420 nM T28484 CB9H1A 25184517 IC50 = 1400 nM T28484 CCA5X7 25184518 IC50 = 7140 nM T28484 CQG3B5 25184521 IC50 = 1470 nM T28484 CT17QC 25184589 IC50 = 3630 nM T28484 C76VQM 25184659 IC50 = 3700 nM T28484 C3U5KV 25229667 EC50 = 139 nM T28484 CK1DA7 26367385 IC50 > 10000 nM T28484 CL60OC 26367815 IC50 > 10000 nM T28484 CWI2E1 29066543 IC50 > 6300 nM T28484 C1IGM6 42633262 EC50 = 3313 nM T28484 CT9V6K 42633458 EC50 = 246 nM T28484 CURL76 42633808 EC50 > 1000 nM T28484 CFUL48 42633810 EC50 > 1000 nM T28484 CW53FJ 42634875 EC50 > 1000 nM T28484 CE1VH8 42634877 EC50 > 500 nM T28484 CFY4X2 42634878 EC50 = 338 nM T28484 CSYR62 42635606 EC50 = 452 nM T28484 C83DTG 42635776 EC50 = 665 nM T28484 CD86FT 43132780 IC50 > 6300 nM T28484 C2TA6X 44130714 IC50 = 20 nM T28484 C5HA7I 44130820 IC50 = 40 nM T28484 CSVI35 44130821 IC50 = 60 nM T28484 CH58RQ 44187469 IC50 = 40 nM T28484 CY8UD3 44238920 IC50 = 46200 nM T28484 C0R8XE 44401424 IC50 > 5000 nM T28484 CK19QO 44401630 IC50 = 460 nM T28484 C8AE7V 44401700 IC50 = 23300 nM T28484 CH5NI0 44401702 IC50 = 10900 nM T28484 CD5GA9 44401759 IC50 = 13500 nM T28484 CA3Z6Q 44401762 IC50 = 250 nM T28484 CEM2V4 44401802 IC50 = 1800 nM T28484 CYZ40J 44401803 IC50 = 3600 nM T28484 CO8U3T 44401822 IC50 = 12700 nM T28484 CXN82K 44401861 IC50 = 6000 nM T28484 CLR2J1 44401864 IC50 > 50000 nM T28484 C53MQP 44401865 IC50 > 50000 nM T28484 COL4M1 44401990 IC50 > 50000 nM T28484 C6TZW3 44401991 IC50 > 50000 nM T28484 CH9L1R 44409515 IC50 = 50000 nM T28484 CB91NT 44409718 IC50 = 13 nM T28484 C5YP1R 44409879 IC50 = 1.3 nM T28484 CKI20Y 44409884 IC50 = 4 nM T28484 C39MWE 44409885 IC50 = 5.5 nM T28484 CF8A0Z 44409903 IC50 = 1.2 nM T28484 CYO7B5 44409904 IC50 = 0.5 nM T28484 C7BM2G 44409905 IC50 = 2.9 nM T28484 C2W8UD 44414670 IC50 = 980 nM T28484 CZX6L4 44414697 IC50 = 190 nM T28484 CET0G6 44414850 IC50 = 6880 nM T28484 CS76CV 44414851 IC50 = 6060 nM T28484 CK16MO 44426727 IC50 = 20000 nM T28484 CZ6RH3 44426731 IC50 = 26 nM T28484 CON04H 44430571 IC50 = 2.2 nM T28484 C7L0PH 44430573 IC50 = 10.2 nM T28484 CDA0X6 44430574 IC50 = 10.2 nM T28484 CT6HC8 44430575 IC50 = 12.1 nM T28484 C7LQ2E 44430576 IC50 = 110 nM T28484 CCBR69 44430578 IC50 = 5.2 nM T28484 CFW02R 44432703 IC50 = 3100 nM T28484 CG78BW 44435327 IC50 = 5000 nM T28484 CSY1J0 44435339 IC50 = 3800 nM T28484 CVS9Y7 44435350 IC50 = 0.9 nM T28484 C74VGT 44435351 IC50 = 1.4 nM T28484 C1FK4E 44435373 IC50 = 1 nM T28484 CXW8Q9 44435374 IC50 = 1.3 nM T28484 CPMN93 44435375 IC50 = 1 nM T28484 CD4EI7 44435376 IC50 = 2 nM T28484 CEX75D 44435377 IC50 = 5.2 nM T28484 COX3Q2 44442283 IC50 = 1.8 nM T28484 C2DZI3 44442301 IC50 = 3 nM T28484 C53HAL 44442302 IC50 = 800 nM T28484 CKJ0Y7 44442887 IC50 = 1.2 nM T28484 CDR7O2 44444939 IC50 = 6600 nM T28484 C4X5PE 44444940 IC50 = 15000 nM T28484 CCL96S 44444941 IC50 = 27000 nM T28484 C6LVI5 44445386 IC50 = 12 nM T28484 CL6YR4 44445387 IC50 = 280 nM T28484 CA82IF 44576259 IC50 = 150 nM T28484 C0JO7X 44590391 IC50 > 20000 nM T28484 CR68ES 44590392 IC50 = 2140 nM T28484 C79YFQ 44590435 IC50 > 20000 nM T28484 CXQE68 44590436 IC50 > 20000 nM T28484 C8O9MZ 44590437 IC50 = 120 nM T28484 CH1S4F 44590510 IC50 = 4610 nM T28484 CMDR03 44590511 IC50 > 20000 nM T28484 CA37FS 44590512 IC50 = 860 nM T28484 CQ1SU4 44590513 IC50 > 20000 nM T28484 COK1F0 44590548 IC50 = 3060 nM T28484 CAG9D7 44590549 IC50 = 700 nM T28484 C1FCO0 45266928 IC50 = 6000 nM T28484 C1Y4KO 45267020 IC50 > 20000 nM T28484 CLK10E 45267851 IC50 = 19000 nM T28484 C53DIE 45267853 IC50 = 520 nM T28484 CO5BT3 45267860 IC50 = 5200 nM T28484 C93RCK 45267863 IC50 > 20000 nM T28484 CAWS46 45267869 IC50 > 20000 nM T28484 C0C7UM 45267870 IC50 > 20000 nM T28484 CK60GY 45267896 IC50 > 20000 nM T28484 C71NGE 45268737 IC50 = 9200 nM T28484 C2ZN5S 45268741 IC50 > 20000 nM T28484 CP4M3X 45268781 IC50 = 20000 nM T28484 C9GJA6 45269595 IC50 = 16300 nM T28484 CTW13H 45269596 IC50 > 20000 nM T28484 C96UFG 45270431 IC50 = 13400 nM T28484 CZ5ID2 45271261 IC50 = 2400 nM T28484 C0X5FN 45271263 IC50 > 20000 nM T28484 CER7W9 45271267 IC50 > 50000 nM T28484 C32JIV 45271285 IC50 > 20000 nM T28484 CN32MP 45272152 IC50 = 33400 nM T28484 CATM09 45272155 IC50 > 20000 nM T28484 C8SB6M 45272157 IC50 > 20000 nM T28484 C70MZU 45272180 IC50 > 20000 nM T28484 C3SRC5 45272183 IC50 > 20000 nM T28484 CRT26A 45272991 IC50 = 2100 nM T28484 CG9XA3 45272994 IC50 = 2200 nM T28484 C3P2WK 45272999 IC50 > 20000 nM T28484 CRUZ63 45789422 IC50 = 20 nM T28484 CRK61L 46224756 IC50 = 155 nM T28484 C7U0NT 46224757 IC50 = 760 nM T28484 CR09DX 46224758 IC50 = 8100 nM T28484 C9DA2G 46224759 IC50 = 175 nM T28484 CC1K2T 46224798 IC50 = 11000 nM T28484 C1SW2H 46224799 IC50 > 25000 nM T28484 C5R3XW 46224800 IC50 > 25000 nM T28484 CBE70W 46224801 IC50 > 25000 nM T28484 C0F6LC 46224802 IC50 = 6600 nM T28484 CI0EG3 46224838 IC50 = 230 nM T28484 CA87WH 46224839 IC50 = 100 nM T28484 CD2ZR7 46224840 IC50 = 200 nM T28484 CGN91R 46225130 IC50 = 630 nM T28484 C59QCL 46225171 IC50 = 760 nM T28484 CVM2D6 46225172 IC50 = 11 nM T28484 C5ZTB8 46225173 IC50 > 25000 nM T28484 C1G8XD 46225174 IC50 = 1700 nM T28484 CF87SZ 46225213 IC50 = 27 nM T28484 C8RSW5 46225214 IC50 = 4500 nM T28484 CWR71G 46225215 IC50 = 200 nM T28484 CW8E2J 46225216 IC50 = 460 nM T28484 CLHF47 46225271 IC50 = 49 nM T28484 CW7H9X 46225272 IC50 = 186 nM T28484 CBC20V 46225273 IC50 = 100 nM T28484 CB3L9I 46225274 IC50 = 900 nM T28484 C3AXM5 46244083 IC50 > 6300 nM T28484 CZ93BW 46244085 IC50 = 95 nM T28484 CWLZ72 46244164 IC50 = 31 nM T28484 C9BGT3 46244165 IC50 = 84 nM T28484 CRZ2Y8 46881445 IC50 = 300 nM T28484 CPZH92 46881446 IC50 > 10000 nM T28484 C38PRQ 46881447 IC50 = 530 nM T28484 CXUQ18 46881495 IC50 > 10000 nM T28484 CFH1G2 46881496 IC50 > 10000 nM T28484 C87UKL 46881497 IC50 = 11 nM T28484 C4SN5I 46881539 IC50 = 14 nM T28484 CGRJ18 46881540 IC50 = 4 nM T28484 C0K3ZJ 46881541 IC50 = 7 nM T28484 CG4W0M 46881581 IC50 = 19 nM T28484 C5SR9E 46881582 IC50 = 65 nM T28484 CL37QK 46881583 IC50 = 6 nM T28484 CVG3U7 46881584 IC50 = 4 nM T28484 C5BLY4 46881627 IC50 = 58 nM T28484 C0T2QG 46881628 IC50 = 4 nM T28484 CIOR36 46881629 IC50 = 19 nM T28484 CK69QD 46881630 IC50 = 5 nM T28484 CWH96P 46881663 IC50 = 11 nM T28484 CDXM14 46881664 IC50 = 2 nM T28484 C3N7QJ 46881665 IC50 = 3 nM T28484 COJ2Z3 46881666 IC50 = 6 nM T28484 CV51NZ 46881710 IC50 = 5 nM T28484 C10HXD 46881711 IC50 = 7 nM T28484 CZ0BX5 46881712 IC50 = 2 nM T28484 CH70VR 46881713 IC50 > 10000 nM T28484 CRZ4S6 46881714 IC50 = 300 nM T28484 C38SKH 46881763 IC50 = 870 nM T28484 CS0QT5 46881764 IC50 = 10000 nM T28484 C5WA2J 46881841 IC50 = 360 nM T28484 CL25ZI 46881873 IC50 = 910 nM T28484 CAX5T3 46881905 IC50 = 3700 nM T28484 CA2S0Z 46881906 IC50 > 10000 nM T28484 C7TS6M 46881907 IC50 = 5300 nM T28484 C9AB2L 46881943 IC50 = 10000 nM T28484 CP4K8C 46881944 IC50 > 10000 nM T28484 CR2J7M 46881945 IC50 = 90 nM T28484 C4QPY2 46881946 IC50 = 540 nM T28484 C8ZJ0N 46881947 IC50 = 1250 nM T28484 CJ3QP9 46881992 IC50 > 10000 nM T28484 C5O7KT 46881993 IC50 = 95 nM T28484 CKY96D 46882035 IC50 = 17 nM T28484 C7OZ6P 46882036 IC50 > 10000 nM T28484 C40WET 46882037 IC50 > 10000 nM T28484 CAI32G 46882038 IC50 = 2300 nM T28484 CKA9Z2 46882039 IC50 > 10000 nM T28484 CA56YD 46882089 IC50 = 270 nM T28484 CUN64R 46882090 IC50 = 350 nM T28484 C3Y7CF 46882091 IC50 = 6800 nM T28484 CN74LO 46906141 IC50 = 724 nM T28484 CYE46T 46906142 IC50 = 75 nM T28484 C3DP7L 46906178 IC50 = 224 nM T28484 CU0LO3 46906179 IC50 = 380 nM T28484 CW75MT 46906180 IC50 = 118 nM T28484 C6W0RZ 46906181 IC50 = 3453 nM T28484 CTD9Y2 46906182 IC50 = 290 nM T28484 CN35PL 46906232 IC50 = 65 nM T28484 CEC3U2 46906234 IC50 = 483 nM T28484 C1DE9K 46906236 IC50 = 40 nM T28484 CI31VX 46906237 IC50 = 76 nM T28484 CK0X7D 46906238 IC50 = 50 nM T28484 C45BIP 46906260 IC50 = 664 nM T28484 C52VRS 46906261 IC50 = 169 nM T28484 CVWR15 46906262 IC50 = 710 nM T28484 C1CW4B 46906263 IC50 = 462 nM T28484 CG75KB 46906264 IC50 = 12378 nM T28484 CKI5A6 46906288 IC50 = 237 nM T28484 CFM5E4 46906290 IC50 = 83 nM T28484 C5RJ2A 46906292 IC50 = 454 nM T28484 CYT0O2 46906294 IC50 = 7 nM T28484 C3WFU8 46906296 IC50 = 204 nM T28484 C42KOP 46906327 IC50 = 347 nM T28484 CKLA96 46906328 IC50 = 51 nM T28484 CEI4X2 46906329 IC50 = 216 nM T28484 CV95BH 46906358 IC50 < 1 nM T28484 CW1H5I 46906359 IC50 = 337 nM T28484 C7OJD1 46906360 IC50 = 1703 nM T28484 CB47DW 46906361 IC50 = 163 nM T28484 C0QEB1 46906363 IC50 = 43 nM T28484 CX87SF 49772558 IC50 = 800 nM T28484 CW3A2L 50901410 EC50 = 1 nM T28484 CY89XM 51356550 IC50 = 1578 nM T28484 C1I7YM 51356551 Ki = 1349.7 nM T28484 C9G6RQ 51356552 Ki = 428.6 nM T28484 C46KAO 51356553 Ki = 84.2 nM T28484 C5AFN6 51356813 Ki < 50 nM T28484 C6N2LD 51356814 Ki < 50 nM T28484 CO6Y8P 51356815 Ki < 50 nM T28484 CU3V9I 51356816 IC50 = 21.8 nM T28484 CR23LH 51356817 IC50 = 19.3 nM T28484 CMCX63 51356818 Ki = 76.2 nM T28484 C1SB5L 51356819 Ki = 302.1 nM T28484 CJU3O1 53326599 IC50 = 41700 nM T28484 C0XG9J 53363371 IC50 = 37 nM T28484 C7HB2V 53363372 IC50 = 45 nM T28484 CQ0S7J 53363455 IC50 = 170 nM T28484 C5BDJ3 53363538 IC50 = 330 nM T28484 CO8AN7 53363539 IC50 = 40 nM T28484 CQ70WO 53363540 IC50 = 180 nM T28484 C45PEV 53363541 IC50 = 58 nM T28484 CN65FT 53363542 IC50 = 45 nM T28484 CTZ1V6 53494967 IC50 = 11 nM T28484 CDI45K 53494981 EC50 = 190 nM T28484 CUQ57S 54757107 IC50 = 10 nM T28484 CMU2H3 54757108 IC50 = 140 nM T28484 C4HTS9 54757109 IC50 = 20 nM T28484 CYMF79 54757209 IC50 = 210 nM T28484 C5LK6A 54757210 IC50 = 130 nM T28484 C6ATD7 54757211 IC50 = 160 nM T28484 CWF67S 54757212 IC50 = 760 nM T28484 CZTJ96 54757416 IC50 = 3500 nM T28484 CDF4W5 54757520 IC50 = 3800 nM T28484 C7MY9B 54757521 IC50 = 5310 nM T28484 CVLZ09 54757522 IC50 = 630 nM T28484 CSX2J4 54757523 IC50 = 9090 nM T28484 C0JZP8 54757524 IC50 = 9000 nM T28484 CSH5W0 54757525 IC50 = 390 nM T28484 CSXE03 54757628 IC50 = 310 nM T28484 CP05UA 54757629 IC50 = 1070 nM T28484 C4JNP8 54757630 IC50 = 1440 nM T28484 CI4K2Y 54757631 IC50 = 2920 nM T28484 CGA3F2 54757632 IC50 = 5990 nM T28484 C4ANQ9 54757740 IC50 = 10000 nM T28484 C76OHM 54757741 IC50 = 5520 nM T28484 CU67QC 54757742 IC50 = 4540 nM T28484 CAY9J2 54757743 IC50 = 6700 nM T28484 C6MG0Y 54757744 IC50 = 4220 nM T28484 CXG51Q 54757745 IC50 = 9000 nM T28484 C9YSJ5 54757838 IC50 = 200 nM T28484 CG41NO 54757839 IC50 = 610 nM T28484 CDE51C 54757840 IC50 = 50 nM T28484 C16YBT 54757841 IC50 = 150 nM T28484 CJV92T 54757842 IC50 = 30 nM T28484 CSQ18G 54757932 IC50 = 210 nM T28484 C1OPZ7 54757933 IC50 = 310 nM T28484 C1UGW3 54757934 IC50 = 2460 nM T28484 C9VO5E 54757935 IC50 = 90 nM T28484 CP39EO 54757936 IC50 = 1060 nM T28484 CGPF63 54758031 IC50 = 20 nM T28484 CL81AQ 54758032 IC50 = 90 nM T28484 CHK86M 54758034 IC50 = 940 nM T28484 C2G6FN 54758035 IC50 = 210 nM T28484 C50VBJ 54758036 IC50 = 140 nM T28484 CE7UF4 54758123 IC50 = 2700 nM T28484 C5KXB9 54758124 IC50 = 5960 nM T28484 CZV8K4 54758125 IC50 = 500 nM T28484 C43ZMD 54758126 IC50 = 1390 nM T28484 CKTN03 54758127 IC50 = 410 nM T28484 C8S0LO 54758216 IC50 = 980 nM T28484 CN4HU9 54758217 IC50 = 2310 nM T28484 CUW4I9 54758219 IC50 = 40 nM T28484 CGZ87Q 54758220 IC50 = 3210 nM T28484 CLF81J 54758305 IC50 = 30 nM T28484 C1RL6Q 54758306 IC50 = 150 nM T28484 C1I7AT 54758307 IC50 = 13 nM T28484 CJZ7W0 54758308 IC50 = 21 nM T28484 CI30OS 54758309 IC50 = 1900 nM T28484 CZHK43 54758400 IC50 = 141 nM T28484 C80NZC 54758401 IC50 = 85 nM T28484 C78BQR 54758402 IC50 = 161 nM T28484 CB1WF5 54758404 IC50 = 323 nM T28484 CSEO14 54758405 IC50 = 5460 nM T28484 CDCG23 54763606 IC50 = 40 nM T28484 C2A5YK 56659866 IC50 = 3959 nM T28484 CVOE09 56659867 IC50 = 1047 nM T28484 CT3U4V 56659868 IC50 = 33 nM T28484 CJ64NA 56659895 IC50 = 334 nM T28484 CG05CX 56662634 EC50 = 160 nM T28484 C3QSP7 56663328 IC50 = 146 nM T28484 CQV76H 56663329 IC50 = 169 nM T28484 COQ9D7 56663330 IC50 = 73 nM T28484 C5UMQ0 56666752 IC50 = 2345 nM T28484 C3G5ZI 56666753 IC50 = 1307 nM T28484 C0VMD1 56670186 IC50 = 232 nM T28484 CYI76G 56670187 IC50 = 1485 nM T28484 CWY2M5 56670188 IC50 = 20 nM T28484 CNTE86 56670189 IC50 = 42 nM T28484 CFH4K0 56670190 IC50 = 9925 nM T28484 CCN9I5 56670191 IC50 = 92 nM T28484 CBU09F 56673708 IC50 = 3409 nM T28484 CBOA18 56673709 IC50 = 49 nM T28484 CON3Y6 56673710 IC50 = 25 nM T28484 C4YLM0 56673740 IC50 = 360 nM T28484 CRJ3T6 56677019 IC50 = 1443 nM T28484 CV34UO 56677053 IC50 = 51 nM T28484 CDXF18 56680345 IC50 = 162 nM T28484 CO72KD 56680346 IC50 = 37130 nM T28484 C1NG8Y 56680347 IC50 = 2942 nM T28484 C0QYH3 56683673 IC50 = 1943 nM T28484 CO8VL4 56683674 IC50 = 828 nM T28484 C08HWQ 56683675 IC50 = 23 nM T28484 C37TXD 56683676 IC50 = 170 nM T28484 C02AUW 56683677 IC50 = 149 nM T28484 CY4KM5 56683678 IC50 = 2767 nM T28484 CTHB21 56683713 IC50 = 1178 nM T28484 CIL79O 56931000 Ki = 5.1 nM T28484 CKN0Z8 56964577 Ki = 6.4 nM T28484 CVC4F5 57325586 Ki = 173.5 nM T28484 C3LVB8 57325587 Ki = 384.4 nM T28484 CZ97DS 57325588 Ki = 3.4 nM T28484 CT67IO 57325589 Ki = 11.1 nM T28484 CO65CE 57325590 Ki = 16.7 nM T28484 C2G9UJ 57326381 Ki = 3018.5 nM T28484 CHM19P 57326382 Ki = 235.4 nM T28484 C43JBM 57326383 Ki = 1783.9 nM T28484 CC0K7O 57326384 Ki = 377.4 nM T28484 CVL16W 57326474 Ki = 89.9 nM T28484 C1K8UN 57326475 Ki = 297.8 nM T28484 C5KRE2 57326476 Ki = 293.9 nM T28484 CJF94R 57326477 Ki = 80 nM T28484 CA2C3V 57326478 Ki = 5.9 nM T28484 CG7Q0Z 57326479 Ki = 10.3 nM T28484 C6O2VB 57326480 Ki = 29.6 nM T28484 C79WOY 57326575 Ki = 352.7 nM T28484 CY04HP 57326576 Ki = 149.8 nM T28484 CAMQ75 57326577 Ki = 520.4 nM T28484 C26DYS 57326578 Ki = 27.8 nM T28484 CY5M7J 57326579 Ki = 519.8 nM T28484 CJ1XC9 57326580 Ki = 185.8 nM T28484 CA35GO 57326581 Ki = 271.7 nM T28484 CN2Q7U 57326676 Ki = 51 nM T28484 CPZG76 57326677 Ki = 120.6 nM T28484 CV5CP4 57326678 Ki = 8.8 nM T28484 CJW83U 57326679 Ki = 10.7 nM T28484 CRGX38 57326680 Ki = 7.5 nM T28484 C1O9PY 57326681 Ki = 9.7 nM T28484 C9UAK0 57326682 Ki = 1978.5 nM T28484 C6OVF0 57326778 Ki = 48.8 nM T28484 C3QI6O 57326779 Ki = 200.3 nM T28484 C93LBU 57326780 Ki = 450.6 nM T28484 C82GXC 57326781 Ki = 838.2 nM T28484 CLIY16 57326782 Ki = 829.2 nM T28484 CVG8I7 57326783 Ki = 990.6 nM T28484 C5PE0A 57326784 Ki = 329.9 nM T28484 CFER23 57326878 Ki = 419.7 nM T28484 C4QGS0 57326879 Ki = 887.8 nM T28484 C1W5BJ 57326880 Ki = 6055.6 nM T28484 CSHD25 57326881 Ki = 2089.6 nM T28484 CQ5IL7 57326882 Ki = 432.4 nM T28484 CDZ41W 57326883 Ki = 311.2 nM T28484 CI6X8L 57326884 Ki = 2942.4 nM T28484 CO12LV 57326973 Ki = 1721.3 nM T28484 CC6LV4 57326974 Ki = 3228.6 nM T28484 CSC21A 57326975 Ki = 2030.8 nM T28484 C5NSW2 57326976 Ki = 1526.7 nM T28484 CD2I1C 57326977 Ki = 1212.1 nM T28484 CVX8P7 57380650 Ki = 57.5 nM T28484 C36MNJ 57380880 Ki = 27.4 nM T28484 C9R5IA 57401215 IC50 = 1520 nM T28484 C1SYP6 57770895 IC50 = 43 nM T28484 C30GOZ 58274571 EC50 > 1000 nM T28484 CP5W0V 58274609 EC50 = 17 nM T28484 C7QN5G 58274649 EC50 = 367 nM T28484 CC9E2T 58274650 EC50 = 2 nM T28484 C0I8ZH 58274695 EC50 = 3 nM T28484 C2MVQ1 58274709 EC50 = 263 nM T28484 CEG26H 58274714 EC50 = 205 nM T28484 CRS37Y 58274722 EC50 > 1000 nM T28484 C7KF5J 58274841 EC50 = 11 nM T28484 C2CG0V 58274853 EC50 = 5 nM T28484 CM90LF 58274857 EC50 = 5 nM T28484 C8ABU3 58274876 EC50 = 179 nM T28484 CCV19B 58274954 EC50 = 615 nM T28484 CCD3W8 58274960 EC50 > 1000 nM T28484 C5C6DO 58274962 EC50 > 500 nM T28484 CC8O4I 66572223 IC50 = 15836 nM T28484 CL2F4E 66572224 IC50 > 150000 nM T28484 CA51QV 66572225 IC50 = 942.2 nM T28484 C30DFU 66572226 IC50 > 50000 nM T28484 CTU1R0 66572322 IC50 = 138 nM T28484 CM94VH 66572323 IC50 = 216.8 nM T28484 CHL76C 66572324 IC50 = 128.9 nM T28484 CCKA14 66572325 IC50 = 67.6 nM T28484 CV8W5P 66572326 IC50 = 150.5 nM T28484 CCY59V 66572327 IC50 = 58.6 nM T28484 C01MQK 66572328 IC50 = 167.6 nM T28484 CN52JC 66572329 IC50 = 159.4 nM T28484 C9KR7P 66572330 IC50 = 191.2 nM T28484 CEA8H0 66572331 IC50 = 567.5 nM T28484 CJS1P6 66572332 IC50 = 178.2 nM T28484 CO02JB 66572333 IC50 = 251.8 nM T28484 CSY2M1 66572334 IC50 = 106.5 nM T28484 CD1K4R 66572336 IC50 = 684.5 nM T28484 CA0T1V 66572337 IC50 = 789.5 nM T28484 CMDK30 66572339 IC50 = 519 nM T28484 CY4GT7 66572340 IC50 = 256.1 nM T28484 C5P8YR 66572341 IC50 = 577.9 nM T28484 CB79JX 66572342 IC50 = 140.9 nM T28484 C3PI0K 66572343 IC50 = 171.9 nM T28484 CMLZ63 66572344 IC50 = 665.6 nM T28484 C5V4JE 66572345 IC50 = 229.3 nM T28484 CZ0P4L 66572346 IC50 = 436.7 nM T28484 CP2V9F 66572347 IC50 = 587.8 nM T28484 CX2HN0 66572348 IC50 = 403.7 nM T28484 CEB16H 66572349 IC50 = 261 nM T28484 CAE28S 66572426 IC50 = 237.5 nM T28484 CX0RP9 66572427 IC50 = 455.8 nM T28484 CO0WK1 66572428 IC50 = 5278 nM T28484 CON57P 70052856 IC50 = 209 nM T28484 C02WNA 70053909 IC50 = 14 nM T28484 C37EFB 71582936 Ki = 17.3 nM T28484 C83PHC 71582937 Ki = 6.4 nM T28484 CLK98I 71582938 Ki = 6.7 nM T28484 CJ93HQ 71582939 Ki = 9.7 nM T28484 C3VKE2 71583032 Ki = 9 nM T28484 CHEZ52 71583033 Ki = 10.1 nM T28484 C5OZ9A 71583034 Ki = 128.6 nM T28484 CNUV80 71583035 Ki = 1.2 nM T28484 CJ87LP 71583036 Ki = 25.7 nM T28484 CD0K5I 71583037 Ki = 4.6 nM T28484 CKT07A 71583038 Ki = 7.8 nM T28484 CTU98Z 71583147 Ki = 2.1 nM T28484 CWO2B0 71583148 Ki = 10.6 nM T28484 CAQR82 71583149 Ki = 9.9 nM T28484 CS3W2I 71716295 Ki = 6.8 nM T28484 C8I6YH 71716296 Ki = 2268 nM T28484 C17ZJR 71716894 Ki = 4.8 nM T28484 CO3JW5 71716895 Ki = 7.8 nM T28484 CM5OR8 71716896 Ki = 27.3 nM T28484 CWGK81 71717524 Ki = 55.6 nM T28484 C1Q8JS 71718135 Ki = 201.3 nM T28484 C5F4AH 71718730 Ki = 33.6 nM T28484 CKV3Q0 71719339 Ki = 293.6 nM T28484 CHO97G 71719340 Ki = 10.1 nM T28484 CN9HI3 71719341 Ki = 162.2 nM T28484 C7CSF4 71719342 Ki = 29.7 nM T28484 C7EBW0 71719940 Ki = 11.6 nM T28484 CD3H0E 71719941 Ki = 35.2 nM T28484 C52WMG 71719942 Ki = 31.4 nM T28484 C1SHK7 71719943 Ki = 56 nM T28484 C46ATF 71720565 Ki = 37.9 nM T28484 C7OV0J 71720566 Ki = 200.3 nM T28484 C8T4SO 71720567 Ki = 64.2 nM T28484 CR5P1H 71720568 Ki = 88.4 nM T28484 C3WQ9R 71726419 IC50 = 7800 nM T28484 C1T3XH 71748071 IC50 = 75 nM T28484 CTA0Q7 71748279 IC50 = 11 nM T28484 CAU9T7 71748280 IC50 = 21 nM T28484 CT97BV 71748288 IC50 = 9.3 nM T28484 CI46YR 71748289 IC50 = 14 nM T28484 CJY8M1 71748290 IC50 = 301 nM T28484 CMSK27 71748293 IC50 = 61 nM T28484 CK6UI7 76309865 IC50 = 78 nM T28484 C7JPK0 76313576 IC50 = 123 nM T28484 C9Y6OA 76313577 IC50 = 98 nM T28484 C5DQI1 76313578 IC50 = 59 nM T28484 C9BGM3 76320800 IC50 = 67 nM T28484 CX1M2W 76320801 IC50 = 63 nM T28484 CEPO93 76324458 IC50 = 122 nM T28484 C0P1JY 76324459 IC50 = 23 nM T28484 C13EZQ 76324460 IC50 = 91 nM T28484 C6N8DX 76324461 IC50 = 168 nM T28484 CLH7P8 76324462 IC50 = 157 nM T28484 C9U0BW 76328015 IC50 = 52 nM T28484 CJ98YI 76331674 IC50 = 38 nM T28484 C2TP4I 76331675 IC50 = 170 nM T28484 CVWS93 76331676 IC50 = 76 nM T28484 C27RMF 76335284 IC50 = 27 nM T28484 CF7U1J 76335285 IC50 = 149 nM T28484 CCQ8W2 76751913 EC50 = 5 nM T28484 CZ5K3S 78319352 IC50 = 16500 nM T28484 CJAM82 82537489 IC50 = 7000 nM T28484 CMY36J 86291007 IC50 = 50 nM T28484 CP1K4E 86298441 IC50 = 35 nM T28484 C7HZS1 86342357 IC50 = 2000 nM T28484 CBGD01 86342358 IC50 = 330 nM T28484 CQ98RK 86342359 IC50 = 810 nM T28484 CQPS98 86342360 IC50 = 430 nM T28484 CUI63O 86342362 IC50 = 1200 nM T28484 CKX3I5 86342363 IC50 = 440 nM T28484 C7BDZ0 86342395 IC50 = 290 nM T28484 CM7DQ4 86342396 IC50 = 810 nM T28484 CWB36G 86342397 IC50 = 190 nM T28484 CXBK16 86342398 IC50 > 6300 nM T28484 CHQ4L6 86342400 IC50 = 68 nM T28484 CJG9W1 86342431 IC50 = 3600 nM T28484 C9ZJ3Q 86342432 IC50 = 430 nM T28484 CC23YM 86342433 IC50 = 920 nM T28484 C3NIL0 86342434 IC50 = 50 nM T28484 CYZR27 86342435 IC50 = 51 nM T28484 C1W2BQ 90643994 IC50 = 85 nM T28484 CO03VM 90643995 IC50 > 6300 nM T28484 CE9ZK4 90643996 IC50 > 6300 nM T28484 CJWF68 90643997 IC50 = 390 nM T28484 CSFQ95 90643998 IC50 > 6300 nM T28484 CE3M0Q 90643999 IC50 > 6300 nM T28484 C5SBF7 90644000 IC50 > 6300 nM T28484 CI42NO 90644001 IC50 > 6300 nM T28484 C8QDX2 90644002 IC50 > 6300 nM T28484 CU6VR0 90644003 IC50 = 160 nM T28484 C9BUJ7 90644004 IC50 > 6300 nM T28484 C2S4RL 90644005 IC50 > 6300 nM T28484 C7Q6DK 90644006 IC50 > 6300 nM T28484 CQF0A2 90644007 IC50 > 6300 nM T28484 C8YC9V 90644008 IC50 > 6300 nM T28484 C8SXG7 90644009 IC50 > 6300 nM T28484 CB70HL 90644010 IC50 > 6300 nM T28484 CJC67A 90644011 IC50 > 6300 nM T28484 CAQF46 90644012 IC50 > 6300 nM T28484 C75EMH 90644013 IC50 = 4600 nM T28484 C28MTR 90644014 IC50 > 6300 nM T28484 CUN3W4 90644015 IC50 > 6300 nM T28484 C3JW6B 90644016 IC50 > 6300 nM T28484 CGM90T 118709485 IC50 = 44 nM T28484 CT6R9O 118721856 IC50 = 520 nM T28484 CWUL90 122195342 IC50 = 1060 nM T28484 CXSO48 122195343 IC50 = 306 nM T28484 C2BWQ7 122195344 IC50 = 238 nM T28484 CI24TL 122195345 IC50 = 160 nM T28484 CSN3F9 122195346 IC50 = 36 nM T28484 CI7MK5 122195347 IC50 = 8.6 nM T28484 CW81CB 122195348 IC50 = 12 nM T28484 CN69PC 122195349 IC50 = 1400 nM T28484 C3N2JL 122195350 IC50 > 20000 nM T28484 CSB5A6 122195351 IC50 > 20000 nM T28484 CYRN15 122195352 IC50 > 20000 nM T28484 CASH54 127035330 IC50 = 1460 nM T28484 C7I6KC 127037279 IC50 = 840 nM T28484 C9Z2CL 134133387 IC50 = 6800 nM T28484 C9GR4X 134141351 IC50 > 20000 nM T28484 C8HX3F 135981700 IC50 = 9000 nM T28484 C6KW0R 145954973 IC50 = 11390 nM T28484 C6HT9G 145962931 IC50 = 9030 nM T28484 C1ST4D 145978176 IC50 = 4860 nM T28484 CWAK78 145979859 IC50 = 41100 nM T28484 C15VPI 145982524 IC50 = 120000 nM T28484 C1QTO7 145982560 IC50 = 60000 nM T28484 CJ3CB4 145983009 IC50 = 20200 nM T28484 CA26IM 145983110 IC50 = 70000 nM T28484 C2AS3H 145983171 IC50 = 120000 nM T28484 CNHW71 145983379 IC50 = 71900 nM T28484 CV6O9Y 145983398 IC50 = 47800 nM T28484 C3XWO4 145983532 IC50 = 51000 nM T28484 CGYI36 145983831 IC50 = 133500 nM T28484 C5D7ZK 145984469 IC50 = 106200 nM T28484 C0V1ZO 145984507 IC50 = 42700 nM T28484 CJ5Z0S 145984542 IC50 = 13200 nM T28484 CP17GR 145984551 IC50 = 90000 nM T28484 CS62PR 145984570 IC50 = 39200 nM T28484 CGA0M2 145984674 IC50 = 17200 nM T28484 CVO4X7 145984986 IC50 = 27500 nM T28484 CL0X1V 145985314 IC50 = 62100 nM T28484 C2QZN6 145985512 IC50 = 128700 nM T28484 CH5V4P 145985905 IC50 = 90000 nM T28484 CWL1Z4 145985964 IC50 = 75000 nM T28484 C3QL0R 145985999 IC50 = 63300 nM T28484 CCTS70 145987224 IC50 = 59900 nM T28484 CTN4Q2 145990080 IC50 = 2200 nM T28484 CKSM25 145991640 IC50 = 53900 nM T28484 C3WQ7O 145992319 IC50 = 7500 nM T28484 CM5N9C 145993225 IC50 = 46900 nM T28484 D00HFV 11652296 IC50 = 11 nM T28484 D00OZN 23626453 IC50 = 7200 nM T28484 D00PRE 23625979 IC50 = 345 nM T28484 D00WOE 11254540 IC50 = 2002 nM T28484 D01ESV 23626139 IC50 = 716 nM T28484 D02HMN 46855212 IC50 = 870 nM T28484 D02LDY 11737887 IC50 = 7682 nM T28484 D02SGH 46244082 IC50 = 390 nM T28484 D05MQU 11695867 IC50 = 58 nM T28484 D05OMR 11299083 IC50 = 11000 nM T28484 D06HLH 46855216 IC50 = 1400 nM T28484 D08FXD 20228010 IC50 = 1500 nM T28484 D08RMK 11593788 IC50 = 1382 nM T28484 D09DGA 9196 IC50 = 4600 nM T28484 D09FZW 46855213 IC50 = 510 nM T28484 D09MSF 12462654 IC50 = 300 nM T28484 D09MXK 42611896 IC50 = 950 nM T28484 D09PLT 12117342 IC50 = 240 nM T28484 D0A9IB 23625978 IC50 = 3726 nM T28484 D0AV3M 11630239 IC50 = 57 nM T28484 D0CU4Q 24417 IC50 > 63000 nM T28484 D0D3FV 18504802 IC50 = 14000 nM T28484 D0E2KC 15541181 IC50 = 64 nM T28484 D0EC0B 44191658 IC50 = 7500 nM T28484 D0G1DW 11232325 Ki = 6.2 nM T28484 D0H3OP 138537 IC50 = 2800 nM T28484 D0H7ZS 23626454 IC50 = 10904 nM T28484 D0J9UC 11623295 IC50 = 140 nM T28484 D0JN0N 11695302 IC50 = 240 nM T28484 D0K7HV 11659042 IC50 = 54 nM T28484 D0M3VA 16034829 Ki < 1 nM T28484 D0M3ZV 504067 IC50 = 17000 nM T28484 D0M7KF 44191653 IC50 = 1600 nM T28484 D0MW5Z 24741169 IC50 = 11000 nM T28484 D0N5OD 9877863 IC50 = 5320 nM T28484 D0N8FU 46855214 IC50 = 3200 nM T28484 D0NJ8L 11595053 IC50 = 262 nM T28484 D0O5SA 10010225 IC50 = 3500 nM T28484 D0OF6C 12169809 IC50 = 210 nM T28484 D0OS3L 42611736 IC50 = 3300 nM T28484 D0P9ZN 46855064 IC50 = 8800 nM T28484 D0RO7K 19290 IC50 = 22000 nM T28484 D0S0JL 193613 IC50 > 63000 nM T28484 D0S7AY 276707 IC50 = 145000 nM T28484 D0T6MF 46855215 IC50 = 11000 nM T28484 D0TN1F 2782709 IC50 = 1649 nM T28484 D0TR0R 12169810 IC50 = 13000 nM T28484 D0V6CM 11593764 IC50 = 1600 nM T28484 D0W4GY 15541180 IC50 = 700 nM T28484 D0Y6IQ 49799223 IC50 = 5600 nM T28484 D0Z3KV 430297 IC50 = 22000 nM T73863 D0T5WK 4506 IC50 > 200000 nM T73863 D00SUC 74766595 IC50 = 35 nM T73863 D01WHH 90216982 IC50 = 1000 nM T73863 D03TKM 76901247 IC50 = 1100 nM T73863 D04KUD 56589666 IC50 < 500 nM T73863 D05CCY 77106319 IC50 < 100 nM T73863 D09NCT 53392492 IC50 = 4300 nM T73863 D0BK5N 56589667 IC50 < 500 nM T73863 D0G8QR 76282772 IC50 = 100 nM T73863 D0GH8J 90204862 IC50 = 54 nM T73863 D0HT9Q 77106317 IC50 = 199.53 nM T73863 D0K4LW 90205053 IC50 = 1000 nM T73863 CIC2K0 1048 Ki > 200000 nM T73863 CTXS46 70914 IC50 = 2070000 nM T73863 C0PU3Z 76559 Ki > 200000 nM T73863 CE73ZQ 78046 Ki > 200000 nM T73863 CT7CW5 144086 Ki > 200000 nM T73863 CF1MG5 338352 Ki > 200000 nM T73863 C1P0WX 344114 IC50 = 2810000 nM T73863 C76AMR 439391 IC50 = 79000 nM T73863 CT0H6S 439939 IC50 = 97000 nM T73863 C5K3ZJ 459531 IC50 = 630.96 nM T73863 C8B1QV 542717 Ki > 200000 nM T73863 CKJ28Z 555194 Ki > 200000 nM T73863 CX34DR 562549 Ki > 200000 nM T73863 C7MOV3 576286 Ki > 200000 nM T73863 CV4ZC0 584578 IC50 > 100000 nM T73863 CS4P5Z 688417 IC50 = 18600 nM T73863 C8M5EK 688418 IC50 = 54700 nM T73863 CMKP07 736587 IC50 < 1000 nM T73863 CHV9I2 762277 Ki > 200000 nM T73863 CZ8IW1 817743 IC50 > 100000 nM T73863 C89WXM 1273303 Ki > 200000 nM T73863 CP53HR 1398473 Ki > 200000 nM T73863 CEQ4V8 2723716 IC50 > 100000 nM T73863 CTSO67 2755894 Ki > 200000 nM T73863 CY3V0G 2784459 IC50 = 30000 nM T73863 CTH86O 2801750 Ki > 200000 nM T73863 CBMG93 4763332 IC50 = 165000 nM T73863 CIUB05 5513694 IC50 = 176000 nM T73863 CTC90M 6519698 IC50 = 1000 nM T73863 CCYF63 9942424 IC50 = 199.53 nM T73863 CF95UP 10909714 IC50 > 100000 nM T73863 CU1Y9B 11251979 Ki > 200000 nM T73863 CD6JS2 13047427 Ki > 200000 nM T73863 C84NIM 13413393 IC50 = 100000 nM T73863 C8NG1A 13973357 Ki > 200000 nM T73863 C1PSK2 13973362 Ki > 200000 nM T73863 C0N6VT 14536434 Ki > 200000 nM T73863 CR52CA 14638329 Ki > 200000 nM T73863 C6RG4X 15179913 Ki > 200000 nM T73863 CTVD27 16773856 IC50 = 98000 nM T73863 C5R0VE 16790848 IC50 = 126000 nM T73863 CA2K7C 19623349 IC50 = 387000 nM T73863 CB1ZF9 19624675 IC50 = 58000 nM T73863 CMT92U 21766412 Ki > 200000 nM T73863 C8VQ2R 22042185 Ki > 200000 nM T73863 CCAM68 22959876 IC50 = 34000 nM T73863 CKQ14T 23610474 Ki > 200000 nM T73863 CF47JU 25138011 IC50 = 3500 nM T73863 C5O1XD 26967300 IC50 = 676000 nM T73863 C7X3WA 28330466 IC50 > 100000 nM T73863 C7OJ5E 46899602 IC50 = 2700 nM T73863 CUMF70 46899605 IC50 = 1500 nM T73863 C2DBN5 46899607 IC50 = 1000 nM T73863 C3G4QK 46899609 IC50 = 1600 nM T73863 C24GUR 46899759 IC50 = 5200 nM T73863 C6ZR3Y 46899761 IC50 = 8800 nM T73863 CLK96Z 46899763 IC50 = 2000 nM T73863 CBOM64 46899765 IC50 = 15000 nM T73863 C9ENX8 46899767 IC50 = 1300 nM T73863 CF2QL4 46899769 IC50 = 1700 nM T73863 CW10BJ 46901089 IC50 = 10000 nM T73863 C6Z1NU 46901246 IC50 = 74000 nM T73863 CUN94R 50999408 IC50 = 507000 nM T73863 CM07QJ 53380011 IC50 = 51000 nM T73863 C2HXA1 53380104 IC50 = 61000 nM T73863 C8CMI9 56766349 IC50 = 2320000 nM T73863 C6QTC3 64393791 IC50 = 316.23 nM T73863 CM9Y5X 64394359 IC50 = 1258.93 nM T73863 CELF46 64394751 IC50 = 398.11 nM T73863 C8K7LG 64395323 IC50 = 316.23 nM T73863 CVYI52 70682586 Ki > 200000 nM T73863 C0HM6A 70682588 Ki > 200000 nM T73863 C6BXR0 70684674 Ki > 200000 nM T73863 CZM97K 70684675 Ki > 200000 nM T73863 C6KM4Y 70684676 Ki > 200000 nM T73863 C81APE 70686821 Ki > 200000 nM T73863 C7SI8G 70688900 Ki > 200000 nM T73863 CAYC62 70688901 Ki > 200000 nM T73863 C5BA6D 70688902 Ki > 200000 nM T73863 C9HTX1 70690990 Ki > 200000 nM T73863 C0DO2G 70690991 Ki > 200000 nM T73863 CDQ5H7 70693123 Ki > 200000 nM T73863 CI1M5B 70695173 Ki > 200000 nM T73863 CB3VJ9 70695181 Ki > 200000 nM T73863 CB80OC 70695182 Ki > 200000 nM T73863 CM4J9D 70695183 Ki > 200000 nM T73863 CJK98Q 70695184 Ki > 200000 nM T73863 CB46OW 70697226 Ki > 200000 nM T73863 CI19FA 70697227 Ki > 200000 nM T73863 C14GIV 71735687 IC50 = 81000 nM T73863 CM02VN 71735839 IC50 = 32000 nM T73863 C4WS1H 71735840 IC50 = 22000 nM T73863 CT4YO5 71735841 IC50 = 78000 nM T73863 C2ZFM8 71735842 IC50 > 120000 nM T73863 CI5W0K 71735843 IC50 = 83000 nM T73863 C6GDP2 71765680 IC50 = 199.53 nM T73863 CN53LH 71765996 IC50 = 6309.57 nM T73863 C2RT5O 71765999 IC50 = 63095.73 nM T73863 C6DXR4 71766146 IC50 = 6309.57 nM T73863 CDT16O 71766431 IC50 = 125.89 nM T73863 CO5TU3 71766576 IC50 = 1995.26 nM T73863 COCF38 71767872 IC50 = 31622.78 nM T73863 CYF8O7 71767874 IC50 = 40000 nM T73863 CFY18G 73333510 IC50 = 110000 nM T73863 CN5B4O 73352277 IC50 = 55000 nM T73863 C68RKH 76310231 IC50 = 1200 nM T73863 CO1EN3 76317452 IC50 = 70 nM T73863 CT5FZ8 76321184 IC50 = 4500 nM T73863 C6XRT0 76321186 IC50 = 2700 nM T73863 CKB5O9 76328366 IC50 = 2500 nM T73863 CUNK03 76335652 IC50 = 3100 nM T73863 C4HXD2 76901248 IC50 = 1100 nM T73863 C4VGX7 76901615 IC50 = 380 nM T73863 CZC7E1 76901616 IC50 = 660 nM T73863 CC5WE1 76901618 IC50 = 2700 nM T73863 CA79XV 76901619 IC50 = 1800 nM T73863 CM2L1V 76901620 IC50 = 410 nM T73863 CLM1B2 77107119 IC50 = 12 nM T73863 CYOA89 77107120 IC50 > 2000 nM T73863 C16PNL 77107121 IC50 = 8 nM T73863 C6IJN1 78426128 IC50 = 1000 nM T73863 CX23ZP 78426670 IC50 > 2500 nM T73863 CMR52S 78426698 IC50 = 2000 nM T73863 CKXW73 78427224 IC50 > 2500 nM T73863 CFPV20 78972837 IC50 = 1210000 nM T73863 C9IMX6 81750118 IC50 = 316.23 nM T73863 C63ATV 81750201 IC50 = 79.43 nM T73863 CHY73I 81750365 IC50 = 158.49 nM T73863 CE6OT2 81750629 IC50 = 31622.78 nM T73863 C21MQV 81750712 IC50 = 630.96 nM T73863 CQG60A 81750714 IC50 <= 100 nM T73863 CM9P8V 81750970 IC50 = 199.53 nM T73863 C69YUM 81751142 IC50 = 125.89 nM T73863 CW47ZA 83454396 IC50 = 5200 nM T73863 C17WNZ 83698744 IC50 = 501.19 nM T73863 CYG63D 86222684 Ki > 200000 nM T73863 CS4Q1F 86268882 IC50 < 100 nM T73863 CRQ51Z 86346639 IC50 < 100 nM T73863 CZ9DC6 86725498 IC50 = 6200 nM T73863 C8WA4M 86725535 IC50 = 5 nM T73863 C8MGN0 86725568 IC50 = 14 nM T73863 CW9F0K 89564218 IC50 < 1000 nM T73863 CCI08H 89825587 IC50 <= 100 nM T73863 C83TUW 89825693 IC50 <= 100 nM T73863 CT46KN 90094283 IC50 = 100 nM T73863 CG4BZ9 90094442 IC50 < 100 nM T73863 C9IYE0 90204662 IC50 = 38 nM T73863 CHV05N 90204861 IC50 = 68 nM T73863 C6PI4M 90204893 IC50 = 2900 nM T73863 CIY20E 90204966 IC50 = 280 nM T73863 CK6L5M 90205111 IC50 = 560 nM T73863 C5ST7H 90205231 IC50 = 1100 nM T73863 CQV07L 90205291 IC50 = 3600 nM T73863 CJ5E4U 90205326 IC50 = 78 nM T73863 C5W7FL 90205353 IC50 = 19 nM T73863 CR21SC 90205356 IC50 = 2900 nM T73863 CM2NA1 90205425 IC50 = 24 nM T73863 CB7Z0A 90205426 IC50 = 74 nM T73863 CN9I0J 90205512 IC50 = 490 nM T73863 C2T4RD 90205719 IC50 = 260 nM T73863 C9H8PV 90211058 IC50 = 310 nM T73863 C1GBT5 90225370 IC50 = 100 nM T73863 CFP3G4 90253472 IC50 = 100 nM T73863 CPUK85 90253505 IC50 = 6 nM T73863 CFX8E0 90407594 IC50 > 10000 nM T73863 CJ9OZ4 90407809 IC50 = 1000 nM T73863 C5LDR2 90407841 IC50 = 100 nM T73863 C2NA5I 91801131 IC50 = 6309.57 nM T73863 CQY0K3 91938043 IC50 < 250 nM T73863 C10RDJ 101882871 IC50 = 15848.93 nM T73863 C86LNW 101882872 IC50 > 100000 nM T73863 C2S1AO 110264830 IC50 = 13300 nM T73863 C4FPD3 112726150 IC50 > 100000 nM T73863 C5OUS0 114286469 IC50 <= 100 nM T73863 C12QPH 114288702 IC50 = 31622.78 nM T73863 CT04PB 118420691 IC50 < 250 nM T73863 CPSD31 118420829 IC50 < 250 nM T73863 CU94QR 118421047 IC50 > 2500 nM T73863 CH6FX3 118421371 IC50 < 250 nM T73863 C6YT2Q 118598059 EC50 = 1.3 nM T73863 C7TBE9 118908379 IC50 = 1900 nM T73863 CJVK69 119081409 IC50 = 4100 nM T73863 C5IZD1 122181577 IC50 = 55000 nM T73863 CY3CG7 122181578 IC50 > 100000 nM T73863 CSR0K5 122181579 IC50 = 63000 nM T73863 CQ57MD 122181580 IC50 = 6500 nM T73863 CQ83MR 122181581 IC50 = 62000 nM T73863 C4GU9P 122181582 IC50 = 76000 nM T73863 CRM93S 122181583 IC50 = 37000 nM T73863 CU57QX 122181584 IC50 = 43000 nM T73863 CIM8C2 122181585 IC50 = 65000 nM T73863 CQA0H7 122181586 IC50 > 100000 nM T73863 C9QVZ5 122181587 IC50 > 100000 nM T73863 CJQ91K 122181588 IC50 = 83000 nM T73863 C8E2KI 122191450 IC50 = 3162.28 nM T73863 C75JVN 122191451 IC50 = 10000 nM T73863 C3YX7W 122191453 IC50 = 6309.57 nM T73863 C3IBR8 122191455 IC50 = 5011.87 nM T73863 C59KNQ 122191457 IC50 = 39810.72 nM T73863 CM5X8J 122191459 IC50 = 39810.72 nM T73863 C7ASR0 122191460 IC50 > 100000 nM T73863 CRI6J4 122191461 IC50 > 100000 nM T73863 CAS4H6 122191462 IC50 = 15848.93 nM T73863 C9J6LX 122191463 IC50 = 15848.93 nM T73863 C75NJO 122191464 IC50 = 10000 nM T73863 C50VYK 122191465 IC50 = 31622.78 nM T73863 CSKY20 122191466 IC50 = 79432.82 nM T73863 CS3L8H 122191467 IC50 = 1584.89 nM T73863 CZ2NV1 122191468 IC50 = 12589.25 nM T73863 CYTW93 122191469 IC50 = 7943.28 nM T73863 CZV45H 122191470 IC50 = 19952.62 nM T73863 CF6I2N 122191471 IC50 = 39810.72 nM T73863 CZU02B 122191472 IC50 = 7943.28 nM T73863 CE27AS 122191473 IC50 = 19952.62 nM T73863 CAJ28B 122191475 IC50 = 31622.78 nM T73863 C36PDK 122191476 IC50 = 39810.72 nM T73863 CQ04FW 122191477 IC50 = 15848.93 nM T73863 C12OHA 122191478 IC50 = 15848.93 nM T73863 CL2K0J 122191479 IC50 = 19952.62 nM T73863 CT6HG3 122191480 IC50 = 19952.62 nM T73863 CK7LD6 122191481 IC50 = 19952.62 nM T73863 CMJ72N 122191482 IC50 = 25118.86 nM T73863 C6H2YQ 122383780 IC50 = 5000 nM T73863 CT2UZ4 125377518 IC50 = 3900 nM T73863 CV6H7C 127028789 IC50 >= 100000 nM T73863 CB8GP9 127029091 IC50 = 25118.86 nM T73863 CIJ0G6 127030272 IC50 < 250 nM T73863 C6KT5A 127030498 IC50 = 310000 nM T73863 C63NWD 127030711 IC50 < 1000 nM T73863 CXF0U5 127030712 IC50 < 1000 nM T73863 CZ2M7U 127030808 IC50 = 125.89 nM T73863 CN16WB 127030937 IC50 < 100 nM T73863 CO4UE5 127031137 IC50 = 15000 nM T73863 CBC7G1 127032036 IC50 = 1258.93 nM T73863 CHO3V7 127032343 IC50 = 1584.89 nM T73863 CB6LF9 127032423 IC50 = 600 nM T73863 C8U9DH 127032712 IC50 = 8500 nM T73863 CDC17F 127032730 IC50 < 100 nM T73863 C5SKT0 127032945 IC50 = 15848.93 nM T73863 CW14UR 127032962 IC50 = 630.96 nM T73863 CL38FP 127033048 IC50 < 100 nM T73863 C2EY1K 127033166 IC50 < 250 nM T73863 CID1E9 127034046 IC50 < 250 nM T73863 C4L1PZ 135567036 IC50 = 6000 nM T73863 CT4O5U 135567037 Ki = 682.9 nM T73863 CC4H1N 135567038 IC50 = 5000 nM T73863 C3LG4V 135567039 IC50 = 8300 nM T73863 CQBH95 135567040 IC50 = 1200 nM T73863 CP6IH9 135567041 Ki = 43.2 nM T73863 C8HMG2 135567042 IC50 = 140 nM T73863 CIW61V 135567106 IC50 = 1995.26 nM T73863 CH2D8B 135567124 IC50 = 398.11 nM T73863 CO1F4A 135567128 IC50 = 501.19 nM T73863 CT0DW5 136048747 IC50 < 100 nM T73863 CXW0S7 136048748 IC50 < 100 nM T73863 CJ91RY 136048749 IC50 < 100 nM T73863 CI4X6R 136053672 IC50 = 1995.26 nM T73863 CO6A0C 136053673 IC50 = 2511.89 nM T73863 CD9F1K 136053674 IC50 = 630.96 nM T73863 CE9R0F 136053675 IC50 = 630.96 nM T73863 CIZV97 136053676 IC50 = 398.11 nM T73863 CE1SW8 136053677 IC50 = 630.96 nM T73863 C8S7CR 136053678 IC50 = 501.19 nM T73863 C3V1SD 136053679 IC50 = 398.11 nM T73863 CMW30T 136053680 IC50 = 630.96 nM T73863 C97FZE 136053681 IC50 = 501.19 nM T73863 CQND25 136053682 IC50 = 7943.28 nM T73863 C6IJ5M 136053683 IC50 = 2000 nM T73863 CNY5T7 136053684 IC50 = 398.11 nM T73863 CV57DW 136053685 IC50 = 199.53 nM T73863 CBGO86 136053686 IC50 = 501.19 nM T73863 C3K1OC 136053687 IC50 = 501.19 nM T73863 CZ80GB 136053688 IC50 = 3162.28 nM T73863 CN56RV 136053689 IC50 = 3162.28 nM T73863 C8HOP7 136053690 IC50 = 1995.26 nM T73863 CN4L7Q 136053691 IC50 = 630.96 nM T73863 CO17WM 136053692 IC50 = 1000 nM T73863 C6OJ3M 136053693 IC50 = 794.33 nM T73863 C5ANQ0 136053694 IC50 = 3162.28 nM T73863 CG13YI 136053695 IC50 = 12589.25 nM T73863 C4EW6T 136053696 IC50 = 1995.26 nM T73863 C5Q9HO 136053697 IC50 = 7943.28 nM T73863 CL3DH6 136053700 IC50 = 4600 nM T73863 C8BAQ6 136053701 IC50 = 460 nM T73863 C3I0DN 136053702 IC50 = 430 nM T73863 CHYC17 136053703 IC50 = 170 nM T73863 CW5FY8 136053704 IC50 = 69 nM T73863 C0DB1S 136053705 IC50 = 1020 nM T73863 C63EQY 136053706 IC50 = 770 nM T73863 C7ALO8 136053707 IC50 = 560 nM T73863 C86NDI 136053708 IC50 = 2500 nM T73863 CR6QH4 136164086 IC50 = 19952.62 nM T73863 CM2VE8 136165229 IC50 = 1900 nM T73863 CU10SL 136258480 IC50 = 450 nM T73863 C2V6MX 136644692 IC50 > 100000 nM T73863 C1H9NK 136959977 IC50 = 100 nM T73863 C1ANF3 138518187 IC50 > 25000 nM T73863 C6LWR4 145963760 IC50 = 151 nM T73863 C0RPS4 145964567 IC50 = 55 nM T73863 C3U8OD 145966600 IC50 = 466 nM T73863 CM9X8H 145967298 IC50 = 12 nM T73863 C9U5TQ 145967792 IC50 = 23 nM T73863 CB97SG 145968018 IC50 = 53 nM T73863 CT5MO6 145971004 IC50 = 154 nM T73863 CK9V5O 145972063 IC50 = 27 nM T73863 CS5FM7 145974200 EC50 = 19 nM T73863 CC8KI6 145976146 IC50 = 23 nM T73863 C1AUN0 145976182 IC50 = 17 nM T73863 CKU0D3 145976400 IC50 = 173 nM T73863 CQ4E0O 145977225 IC50 = 65 nM T73863 CIQ6Y7 145977327 IC50 = 2.2 nM T73863 C5TBS2 145977546 IC50 = 46 nM T73863 CL2FR4 145978064 IC50 = 22 nM T73863 C8OL2Q 145978411 IC50 = 164 nM T73863 CA8UD0 145978535 IC50 = 38 nM T73863 D07IOY 10365 Ki = 2.2 nM T73863 D08IZY 3080614 IC50 = 430000 nM T73863 D0B2WZ 15331 IC50 = 2500000 nM T73863 D0M7DC 574310 Ki > 200000 nM T73863 D0X5US 459617 IC50 = 600 nM T65483 CMU34O 9813856 IC50 > 50000 nM T65483 CF5A3T 9837547 IC50 > 50000 nM T65483 CQ6HP2 9857137 IC50 > 50000 nM T65483 CHI95J 9926432 IC50 > 50000 nM T65483 C9WT3L 9942902 IC50 > 50000 nM T65483 CM1A0D 9943447 IC50 > 50000 nM T65483 CW28EQ 9966944 IC50 > 50000 nM T65483 C6FQ0R 10465893 IC50 > 50000 nM T65483 D06LNX 3858 IC50 > 50000 nM T33754 D03VPC 2754 IC50 = 190 nM T33754 D05MQK 110635 IC50 > 10000 nM T33754 D0C4HG 3033825 IC50 = 8 nM T33754 D0C9SY 135400189 IC50 = 2100 nM T33754 D0D1HW 135409400 IC50 = 50 nM T33754 D0E0SW 53708 IC50 = 14000 nM T33754 D0F8RA 2153 IC50 = 240000 nM T33754 D0F9GE 3108 IC50 = 43000 nM T33754 D0L0ZF 5663 IC50 = 6200 nM T33754 D0Y9ZE 4197 Ki = 150 nM T33754 D0Z7ZM 135398744 IC50 = 7000 nM T33754 D01LCC 17754438 IC50 = 1300 nM T33754 D08HKT 5362399 IC50 = 300 nM T33754 D0LI1C 44469321 IC50 > 10000 nM T33754 D0O1IM 58298318 IC50 = 630 nM T33754 D0SM0W 44591583 IC50 = 6400 nM T33754 D0T5PO 5092 IC50 > 10000 nM T33754 D0X0PP 59351313 IC50 > 30000 nM T33754 D07EUB 46200734 IC50 = 1820 nM T33754 D00DBE 9865514 IC50 = 35800 nM T33754 D00SPK 23665864 IC50 > 100000 nM T33754 D00YPW 135399235 IC50 = 133000 nM T33754 D01QUF 9842576 Ki > 100000 nM T33754 D02EMR 151170 IC50 > 3162.28 nM T33754 D05VLN 55690 IC50 = 31622.78 nM T33754 D07FHZ 5087 IC50 > 300000 nM T33754 D08FOX 55263 IC50 = 8600 nM T33754 D08NXX 5487281 IC50 = 10 nM T33754 D09SFV 3973 IC50 = 100000 nM T33754 D09UMA 55918 IC50 = 3400 nM T33754 D0BK6B 3021729 IC50 = 260 nM T33754 D0F0CS 5723 IC50 = 110 nM T33754 D0Y6HV 187079 IC50 = 50 nM T33754 CVQ0G5 1348 Ki = 16000 nM T33754 CO2Y3R 3698 IC50 = 16000 nM T33754 CX43RE 4823 IC50 = 19000 nM T33754 CH8J2B 4977 Ki = 1000000 nM T33754 CCJ8F0 5353 IC50 = 500000 nM T33754 C3B8VG 5369 IC50 > 10000 nM T33754 CJ02EG 41946 Ki = 1400 nM T33754 CA5Q8Y 58575 IC50 = 17000 nM T33754 CJ5R9Z 60867 IC50 = 1500 nM T33754 C1OJE8 65934 IC50 = 1600 nM T33754 CZ39NL 127770 IC50 = 37000 nM T33754 CGA17S 127779 Ki = 35000 nM T33754 C54IRL 129517 IC50 = 1500 nM T33754 CB9XD5 129826 IC50 = 100 nM T33754 C3B1GP 130152 IC50 = 47 nM T33754 C3FRX9 131989 IC50 = 380000 nM T33754 COK69D 156890 IC50 = 390000 nM T33754 CH2P8A 158961 Ki = 1200000 nM T33754 CVN23X 158962 Ki = 1100000 nM T33754 CGO1D9 184661 IC50 = 125.89 nM T33754 C4IEB6 205981 Ki = 217000 nM T33754 C8FWD2 317789 IC50 = 2511.89 nM T33754 C8EFH4 349956 IC50 = 101000 nM T33754 CG7Q1D 589674 IC50 = 18800 nM T33754 C6FCR1 3015712 IC50 = 138000 nM T33754 C1UNV3 4197712 IC50 = 14000 nM T33754 CBS67I 5271722 IC50 = 61000 nM T33754 CR5GH1 5284402 IC50 = 80 nM T33754 CE5VJ9 5362132 IC50 = 550 nM T33754 CO8NK7 5487388 IC50 = 18 nM T33754 CYO52K 5487415 IC50 = 0.4 nM T33754 COPL36 5492199 IC50 = 24 nM T33754 CSQ14B 5492217 IC50 = 20 nM T33754 C7BQ1N 5492386 IC50 = 1 nM T33754 CXDJ97 5746185 IC50 = 300 nM T33754 C8ZFX6 6624932 IC50 = 160000 nM T33754 CAYS61 6918354 IC50 = 290 nM T33754 CB40PM 6918356 IC50 = 1800 nM T33754 CR0NJ7 6918510 IC50 = 27000 nM T33754 CFJ62Y 9799389 IC50 > 10000 nM T33754 C3EOU7 9799418 IC50 > 3162.28 nM T33754 C87ERL 9806003 IC50 = 251.19 nM T33754 CHK3Z5 9806981 IC50 = 199.53 nM T33754 C0F5WH 9816616 IC50 = 2000 nM T33754 CXF0J7 9818343 IC50 = 12000 nM T33754 C1CXA5 9818702 IC50 = 380000 nM T33754 CSOX21 9819114 IC50 > 3000 nM T33754 C1MN3A 9821924 IC50 = 2220 nM T33754 C0K3SA 9825739 IC50 > 100000 nM T33754 C7B1PO 9826435 IC50 = 51600 nM T33754 CKG34S 9828282 IC50 = 501.19 nM T33754 CKOT49 9829555 IC50 = 100 nM T33754 C3ZNU4 9850384 IC50 = 79.43 nM T33754 CFV1Q4 9852021 IC50 > 3162.28 nM T33754 C8QJ4D 9859958 IC50 > 100000 nM T33754 C3HJB5 9867688 IC50 > 3162.28 nM T33754 CDW03H 9867844 IC50 > 3162.28 nM T33754 CVP6S0 9869611 IC50 = 79.43 nM T33754 CF18MC 9874535 IC50 > 100000 nM T33754 C7XYK6 9881656 IC50 > 100000 nM T33754 CQJ71T 9887909 IC50 > 3162.28 nM T33754 CY65BZ 9894329 IC50 = 199.53 nM T33754 CD6IG8 9894586 IC50 > 100000 nM T33754 CET1I4 9906369 IC50 > 20000 nM T33754 CMBO89 9912467 IC50 = 330 nM T33754 C81LSK 9928390 IC50 > 100000 nM T33754 CRT85B 9953239 IC50 = 80 nM T33754 COS23J 9956462 IC50 = 199.53 nM T33754 C19FKZ 9958988 IC50 > 3162.28 nM T33754 C4P8WX 9959207 IC50 = 31.62 nM T33754 CQ40MX 9981320 IC50 = 2400 nM T33754 C39LZS 9999105 IC50 = 30 nM T33754 CFPR64 9999276 IC50 > 10000 nM T33754 CKP7I8 10014043 IC50 = 350 nM T33754 C34ZPX 10014479 IC50 = 560 nM T33754 CXQ0V1 10016898 IC50 = 2000 nM T33754 C4ST7G 10017729 IC50 = 400 nM T33754 C3R8DT 10036672 IC50 = 4200 nM T33754 CHL52O 10037253 IC50 = 230 nM T33754 CMAT67 10038096 IC50 = 78 nM T33754 CJ1Q7Z 10040540 IC50 = 15000 nM T33754 CGXS34 10043016 IC50 = 5900 nM T33754 CH0YG4 10043540 IC50 = 37 nM T33754 CGX7W1 10064431 IC50 = 18000 nM T33754 C12KAB 10065195 IC50 = 850 nM T33754 C2L8MI 10068486 IC50 > 3162.28 nM T33754 CJA37O 10082617 IC50 = 22 nM T33754 CQMC42 10083083 IC50 = 180 nM T33754 C2N4IZ 10084561 IC50 = 12.59 nM T33754 C6QVN7 10104952 IC50 = 1400 nM T33754 COB5N2 10105100 IC50 = 2800 nM T33754 C8SNV1 10105196 IC50 = 160 nM T33754 CT0A4J 10113055 IC50 = 299 nM T33754 CPWL59 10113972 IC50 = 1060 nM T33754 C2MGJ7 10117650 IC50 = 580 nM T33754 CG8RW2 10142576 IC50 = 2970 nM T33754 C89DXP 10181676 IC50 = 2710 nM T33754 C8V6FE 10225063 IC50 = 42 nM T33754 CAS6F9 10228849 IC50 = 23300 nM T33754 CZ1Y8D 10232923 IC50 > 100000 nM T33754 C1TZ0Y 10242216 IC50 = 5300 nM T33754 CNF1Z7 10243366 IC50 = 1600 nM T33754 C41REA 10243444 IC50 = 23 nM T33754 C1XL2R 10247726 IC50 = 24000 nM T33754 CK23EJ 10261617 IC50 = 960 nM T33754 C7GTC0 10264205 IC50 > 10000 nM T33754 CJQ89G 10266192 IC50 > 200000 nM T33754 CUE72P 10314633 IC50 = 2000 nM T33754 CB71WD 10322207 IC50 = 16 nM T33754 C86USM 10326035 IC50 > 3162.28 nM T33754 CF6YU1 10329832 IC50 = 3100 nM T33754 CP1M5H 10342086 IC50 > 100000 nM T33754 C1Z6TS 10352208 IC50 = 3700 nM T33754 CC14IS 10354139 IC50 = 230 nM T33754 CU45BF 10354140 IC50 = 69 nM T33754 CZ6X9Y 10391444 IC50 = 290 nM T33754 CMR4H3 10398747 IC50 = 100 nM T33754 CU32AZ 10411395 IC50 > 3162.28 nM T33754 C94CHO 10421765 IC50 = 1400 nM T33754 CY6B3J 10422444 IC50 = 28000 nM T33754 C43YLO 10422686 IC50 = 330 nM T33754 CEOK50 10428730 IC50 < 10000 nM T33754 C3WG2D 10432384 IC50 > 3162.28 nM T33754 C1OG0Y 10443570 IC50 = 2200 nM T33754 C60KSF 10444558 IC50 = 67 nM T33754 CF5O8D 10446136 IC50 = 1850 nM T33754 C23HSK 10451184 IC50 > 100000 nM T33754 CHQ38X 10455790 IC50 > 100000 nM T33754 CH2B6U 10455813 IC50 = 2400 nM T33754 C5WAM6 10465078 IC50 = 1420 nM T33754 CN40VQ 10465933 IC50 = 62 nM T33754 C0XW2I 10469627 IC50 > 3000000 nM T33754 C5CI3G 10479468 IC50 = 90 nM T33754 CZ92DR 10481735 IC50 = 6030 nM T33754 CA24TW 10491646 IC50 > 100000 nM T33754 C68VBD 10492653 IC50 > 100000 nM T33754 C3PKX6 10492654 IC50 > 100000 nM T33754 C5JPK7 10494678 IC50 > 200000 nM T33754 C2OP8L 10497499 IC50 = 8500 nM T33754 CTUW75 10503944 IC50 = 320 nM T33754 CMR6A4 10504383 IC50 = 80000 nM T33754 C6GS9R 10506218 IC50 > 100000 nM T33754 C4CN0V 10508072 IC50 > 100000 nM T33754 CW7T6I 10515565 IC50 > 100000 nM T33754 CPWU60 10524067 IC50 = 20000 nM T33754 CH4LZ1 10525677 IC50 = 86800 nM T33754 CR8SN9 10526455 IC50 > 100000 nM T33754 C9WSE6 10528313 IC50 = 2900 nM T33754 CZ6T2C 10536740 IC50 > 100000 nM T33754 CCG53Q 10541661 IC50 = 77000 nM T33754 CLI1R7 10543311 IC50 > 200000 nM T33754 C6M0ZQ 10545256 IC50 = 3500 nM T33754 CP63QK 10547069 IC50 = 18000 nM T33754 C7G1BH 10547592 IC50 > 100000 nM T33754 CP0JT2 10550927 IC50 > 100000 nM T33754 C7ID5Q 10552011 IC50 = 82000 nM T33754 CQW79N 10554042 IC50 = 50000 nM T33754 C4V8OI 10563356 IC50 > 100000 nM T33754 C5WMZ0 10563923 IC50 = 30000 nM T33754 CYUJ54 10564633 IC50 > 200000 nM T33754 C1R0HE 10567025 IC50 > 200000 nM T33754 CKUS20 10567758 IC50 > 200000 nM T33754 C7K1QW 10571952 IC50 > 100000 nM T33754 CY9P5W 10575733 IC50 = 60 nM T33754 C8V2KW 10576728 IC50 = 46000 nM T33754 C20EPT 10577926 IC50 = 4500 nM T33754 C7Z9YF 10579873 IC50 > 100000 nM T33754 C3Y8JH 10590134 IC50 = 97000 nM T33754 CW0LN4 10593644 IC50 > 200000 nM T33754 C57HYA 10600864 IC50 = 16000 nM T33754 CMNU92 10602385 IC50 = 10600 nM T33754 CS2Q1U 10602534 IC50 > 100000 nM T33754 CSPY93 10603533 IC50 > 100000 nM T33754 CJ7CU4 10603606 IC50 = 34 nM T33754 CUTK97 10610142 IC50 = 68000 nM T33754 C5LVM2 10613420 IC50 > 100000 nM T33754 CK3GR5 10624131 IC50 = 400 nM T33754 CZIQ04 10625498 IC50 = 77000 nM T33754 CN4T7O 10625920 IC50 > 100000 nM T33754 C21CUM 10626417 IC50 > 100000 nM T33754 C1O4KV 10626842 IC50 > 100000 nM T33754 C25WRZ 10627119 IC50 = 170 nM T33754 CCB7D3 10639948 IC50 = 6000 nM T33754 CF1UR8 10640268 IC50 = 5000 nM T33754 CB3R6M 10644497 IC50 = 90000 nM T33754 CUZN30 10646721 IC50 = 70000 nM T33754 CNK65G 10646809 IC50 = 2000 nM T33754 CKNA14 10648008 IC50 = 250 nM T33754 C0I4FA 10648358 IC50 = 10300 nM T33754 CP8UX9 10649414 IC50 = 58200 nM T33754 C3XAK7 10650055 IC50 > 100000 nM T33754 CE65JO 10650764 IC50 > 100000 nM T33754 CNP1D9 10651107 IC50 > 100000 nM T33754 CJ5XI4 10651803 IC50 > 100000 nM T33754 CP2B0V 10660654 IC50 = 42000 nM T33754 CY25HA 10661817 IC50 = 58000 nM T33754 CP1CJ3 10663161 IC50 > 200000 nM T33754 CR47SU 10665209 IC50 = 4.9 nM T33754 C09ROH 10668502 IC50 > 100000 nM T33754 CB9Y7A 10669693 IC50 = 2000 nM T33754 CFM5N1 10673963 IC50 > 100000 nM T33754 C9FR7P 10674875 IC50 > 100000 nM T33754 C2Y5HF 10675032 IC50 = 490 nM T33754 C6T4ZW 10687037 IC50 = 14000 nM T33754 C5KXY7 10688351 IC50 > 200000 nM T33754 CHB93E 10690761 IC50 = 200000 nM T33754 CV6WT3 10692240 IC50 > 100000 nM T33754 C6LR4V 10694878 IC50 > 100000 nM T33754 CV0H5I 10696630 IC50 = 54700 nM T33754 C1B3WP 10696971 IC50 = 3200 nM T33754 CI6ON5 10698519 IC50 = 100 nM T33754 C40GRD 10704663 IC50 = 331000 nM T33754 C23WGX 10706416 IC50 > 100000 nM T33754 C59SWD 10709216 IC50 = 43000 nM T33754 C8CM0J 10711062 IC50 = 44000 nM T33754 C8UHE3 10717022 IC50 = 9000 nM T33754 CDMP96 10717370 IC50 = 20000 nM T33754 CEW0L8 10718244 IC50 > 100000 nM T33754 CU53RA 10718426 IC50 = 18000 nM T33754 CCI8R7 10729204 IC50 > 100000 nM T33754 CF7L2E 10732847 IC50 = 29000 nM T33754 CS2ZA3 10734331 IC50 > 200000 nM T33754 C5IKL9 10734997 IC50 = 20000 nM T33754 C7JN8X 10739699 IC50 = 3500 nM T33754 CO39UQ 10744528 IC50 = 22200 nM T33754 C3X8UM 10754735 IC50 = 80000 nM T33754 CDPZ05 10758281 IC50 > 200000 nM T33754 C28FLE 10762239 IC50 = 18000 nM T33754 CINX82 10763354 IC50 = 80000 nM T33754 C3R8TI 10764856 IC50 = 28800 nM T33754 CFJL61 10768238 IC50 = 41 nM T33754 C51XRM 10776762 IC50 > 300000 nM T33754 C35YPM 10779997 IC50 > 200000 nM T33754 CO08EH 10780064 IC50 = 45000 nM T33754 CSN64H 10783300 IC50 > 200000 nM T33754 CEV60G 10783489 IC50 = 18000 nM T33754 COF0E3 10783717 IC50 > 1000 nM T33754 CKEV02 10786459 IC50 > 200000 nM T33754 CQMF39 10787820 IC50 > 100000 nM T33754 CLM42P 10788651 IC50 = 8000 nM T33754 C92SMD 10789583 IC50 = 53900 nM T33754 C19EHR 10791038 IC50 > 100000 nM T33754 CXWY95 10792119 IC50 > 100000 nM T33754 C6C5AD 10792156 IC50 > 100000 nM T33754 C2KUF1 10792829 IC50 > 100000 nM T33754 C1K4AN 10792853 IC50 > 100000 nM T33754 C9YFH4 10805458 IC50 > 200000 nM T33754 C24LPM 10810360 IC50 = 12000 nM T33754 CDL73U 10810934 IC50 > 100000 nM T33754 CAF1X8 10812634 IC50 > 100000 nM T33754 CW07PN 10814053 IC50 = 48600 nM T33754 CA9UW6 10816539 IC50 = 81 nM T33754 C4T8PS 10816641 IC50 > 100000 nM T33754 CX1B4U 10817302 IC50 = 60000 nM T33754 C49GKH 10826458 IC50 > 200000 nM T33754 CG5M7O 10827879 IC50 = 58000 nM T33754 CT8AK4 10830480 IC50 = 64000 nM T33754 COHP57 10833764 IC50 > 100000 nM T33754 CT2F6P 10835916 IC50 = 8000 nM T33754 C0QY8J 10837144 IC50 = 48500 nM T33754 CZMB59 10840332 IC50 > 100000 nM T33754 C5MTK7 10840471 IC50 > 100000 nM T33754 C2IWD7 10840815 IC50 > 100000 nM T33754 CR50XV 10841036 IC50 = 80000 nM T33754 CQWL18 10852535 IC50 > 200000 nM T33754 CCM2Y6 10853678 IC50 = 39000 nM T33754 CE3H7M 10861002 IC50 > 3162.28 nM T33754 CPI5E6 10861494 IC50 < 10000 nM T33754 C8T5KN 10864434 IC50 > 10000 nM T33754 CCV4L0 10873945 IC50 > 3162.28 nM T33754 C3T4WD 10874925 IC50 = 1258.93 nM T33754 C17SLU 10875758 IC50 > 10000 nM T33754 C2DMI8 10885725 IC50 > 10000 nM T33754 CHV5Q1 10885756 IC50 > 10000 nM T33754 CNG12D 10893436 IC50 > 3162.28 nM T33754 CR2I7H 10895319 IC50 > 3162.28 nM T33754 CE4O8T 10896876 IC50 > 3162.28 nM T33754 CRJ5T9 10897006 IC50 > 3162.28 nM T33754 C0RTU9 10897531 IC50 > 10000 nM T33754 CW5EQ0 10903429 IC50 < 10000 nM T33754 C42XNF 10917977 IC50 > 3162.28 nM T33754 C8TJ5Z 10929587 IC50 > 10000 nM T33754 C5UY2I 10940665 IC50 = 794.33 nM T33754 C7W9ZV 10940912 IC50 > 10000 nM T33754 C78BLJ 10962385 IC50 > 10000 nM T33754 CKI1O9 10971811 IC50 > 3162.28 nM T33754 CE1MC0 10980260 IC50 = 5011.87 nM T33754 C58LJN 10981074 IC50 > 3162.28 nM T33754 CR1Y2H 10989584 IC50 = 430 nM T33754 C64POJ 10993740 IC50 > 3162.28 nM T33754 C1R4NH 11004936 IC50 > 3162.28 nM T33754 CE5B8M 11006448 IC50 > 10000 nM T33754 C3AC7X 11015442 IC50 > 3162.28 nM T33754 C3L7EA 11017154 IC50 > 10000 nM T33754 CR7C1N 11017676 IC50 > 10000 nM T33754 CBMN25 11028101 IC50 = 4400 nM T33754 CKBT82 11038706 IC50 > 10000 nM T33754 CIOS65 11038955 IC50 > 10000 nM T33754 CCY7A3 11048935 IC50 > 3162.28 nM T33754 CAD3C4 11050210 IC50 > 10000 nM T33754 C54VZQ 11064194 IC50 = 540 nM T33754 CQI5O1 11067303 IC50 < 10000 nM T33754 CE28QV 11071990 IC50 > 3162.28 nM T33754 CL0VC4 11072016 IC50 > 3162.28 nM T33754 CGW6K3 11072194 IC50 > 10000 nM T33754 CA34RC 11075802 IC50 = 251.19 nM T33754 CX68HJ 11078960 IC50 > 3162.28 nM T33754 C0T1DG 11079584 IC50 > 3162.28 nM T33754 CI2TS9 11079673 IC50 < 10000 nM T33754 CGX54C 11093107 IC50 > 10000 nM T33754 CG74CI 11093245 IC50 > 10000 nM T33754 CT8GE9 11100924 IC50 > 3162.28 nM T33754 C4VJR8 11109680 IC50 < 10000 nM T33754 CG7FV9 11113983 IC50 > 3162.28 nM T33754 CAHJ81 11114030 IC50 > 10000 nM T33754 CR1IZ3 11122701 IC50 > 3162.28 nM T33754 C4C0NX 11122848 IC50 > 10000 nM T33754 CU56SF 11124260 IC50 > 10000 nM T33754 CQ4D5W 11124276 IC50 = 1584.89 nM T33754 C4AET8 11124334 IC50 > 10000 nM T33754 COB72U 11124582 IC50 > 10000 nM T33754 C24VFA 11125005 IC50 > 10000 nM T33754 CU7J6M 11128507 IC50 = 8600 nM T33754 C6KC5Y 11135635 IC50 > 10000 nM T33754 C50SRF 11145589 IC50 > 10000 nM T33754 CR6SE0 11146532 IC50 > 10000 nM T33754 CREQ98 11373312 IC50 = 31000 nM T33754 CU9IY2 11414494 IC50 = 2000 nM T33754 C45VZC 11438405 IC50 > 16000 nM T33754 CV2E4Z 11476710 IC50 = 13000 nM T33754 C4ZYH9 11547485 IC50 > 10000 nM T33754 CKJP43 11723241 IC50 = 35000 nM T33754 CNL0G1 11725859 IC50 > 3000 nM T33754 C1A0KG 11726102 IC50 = 100000 nM T33754 CLR4X2 11729202 IC50 > 3162.28 nM T33754 C2BQ9K 11729404 IC50 < 10000 nM T33754 CX3FQ5 11730938 IC50 > 10000 nM T33754 CB60VT 11733770 IC50 > 10000 nM T33754 C0AKJ4 11742456 IC50 = 12000 nM T33754 CX8J5U 11742876 IC50 > 100000 nM T33754 CFE7S1 11762426 IC50 > 3162.28 nM T33754 CJQ0N8 11775824 IC50 = 170 nM T33754 CK9C5E 11777068 IC50 = 6100 nM T33754 CY0M4H 11777232 IC50 = 140 nM T33754 CQ8Y6L 11793138 IC50 = 30000 nM T33754 CGA1F8 11794425 IC50 = 1000 nM T33754 CYX91E 11795941 IC50 = 40800 nM T33754 C7E8QN 11796403 IC50 = 11000 nM T33754 CYZS05 11798266 IC50 = 19400 nM T33754 C2SXZ1 11798380 IC50 = 19500 nM T33754 C30UGZ 11800567 IC50 > 100000 nM T33754 CBDF71 11812295 IC50 = 8500 nM T33754 CT94GH 11826581 IC50 = 3981.07 nM T33754 C1PM0R 11827787 IC50 > 10000 nM T33754 C29HOL 11828590 IC50 = 8400 nM T33754 CK2J5S 11834125 IC50 > 3162.28 nM T33754 CO9I0H 12016984 IC50 = 48000 nM T33754 CZAV59 12016985 IC50 = 67000 nM T33754 CZ4QA8 12016986 IC50 = 10000 nM T33754 C08RSO 12016987 IC50 = 86000 nM T33754 C4YOB9 12016988 IC50 = 31000 nM T33754 C0VW2U 12016989 IC50 > 100000 nM T33754 C9ZWE6 12016990 IC50 = 120000 nM T33754 C8UL5M 12016991 IC50 = 25000 nM T33754 C28HJD 12016992 IC50 > 100000 nM T33754 CCL4W3 12016993 IC50 = 26000 nM T33754 CAB5E1 12016994 IC50 > 200000 nM T33754 CYF3K5 12016995 IC50 = 102000 nM T33754 CPZ7M4 12726304 IC50 = 100000 nM T33754 C08YKT 12774626 IC50 = 630 nM T33754 CX1CN7 12789009 IC50 = 38000 nM T33754 CP4C7R 12799333 IC50 = 31000 nM T33754 C5RDG7 12850742 IC50 = 1300 nM T33754 COE42X 12851329 IC50 = 2500 nM T33754 CBA94E 12873360 IC50 = 12000 nM T33754 CA5K9I 13037186 IC50 = 16000 nM T33754 CN0UA5 13037188 IC50 = 7300 nM T33754 CE41YR 13059432 IC50 = 7200 nM T33754 CEY1B7 13066339 Ki = 270000 nM T33754 CV79BW 13195776 IC50 = 3400 nM T33754 CNW9B8 13200334 IC50 = 1350 nM T33754 CN9KG3 13232050 IC50 = 40 nM T33754 C7SPV8 13233881 IC50 = 110000 nM T33754 C75JTV 13233882 IC50 = 43000 nM T33754 C9NR8P 13233885 IC50 = 74000 nM T33754 C4AK6E 13233889 IC50 = 2300 nM T33754 CBG9R7 13365079 IC50 = 100000 nM T33754 C15QXF 13365081 IC50 = 43000 nM T33754 CD9SX6 13365089 IC50 = 22000 nM T33754 CJZ8O6 13457698 IC50 = 48 nM T33754 C89SUK 13475879 IC50 = 12100 nM T33754 C1DY8H 13475880 IC50 = 38000 nM T33754 CLU3V4 13475882 IC50 = 160000 nM T33754 C4RK3T 13518856 IC50 = 52000 nM T33754 CRD08J 13518862 IC50 = 22000 nM T33754 CA18FX 13518865 IC50 = 3200 nM T33754 C6G1RO 13535424 IC50 = 400 nM T33754 CPO2I4 13553473 IC50 = 128000 nM T33754 C58VQR 13553476 IC50 = 75000 nM T33754 CN7D9Q 13560740 IC50 = 140 nM T33754 CUT8O7 13560741 IC50 = 140 nM T33754 CN5HR4 13563538 IC50 = 300000 nM T33754 C4LJK9 13563540 IC50 = 38000 nM T33754 C3OHW1 13656051 IC50 = 1800 nM T33754 C6OG1D 13656060 IC50 = 1200 nM T33754 CZRM51 13656069 IC50 = 1600 nM T33754 CH60ZY 13724739 IC50 = 35000 nM T33754 CA35BS 13745706 IC50 = 21000 nM T33754 CL14GZ 13756656 IC50 = 1150 nM T33754 CTZU64 13756657 IC50 = 4400 nM T33754 CU5Z7B 13756658 IC50 = 3600 nM T33754 CRL4Q3 13756663 IC50 = 1300 nM T33754 CL2DO6 13756665 IC50 = 1150 nM T33754 CFKW29 13756666 IC50 = 190 nM T33754 CJXW08 13756670 IC50 = 1800 nM T33754 C6EHB3 13756788 IC50 = 15000 nM T33754 C83QIN 13756791 IC50 = 27000 nM T33754 CD7P5R 13756811 IC50 = 500 nM T33754 C8I5PH 13756813 IC50 = 76000 nM T33754 CX5RB2 13756814 IC50 = 9600 nM T33754 C8SC6J 13813706 IC50 = 129000 nM T33754 C38OTH 13813707 IC50 = 190000 nM T33754 CLO0R8 13813708 IC50 = 25000 nM T33754 CB01QR 13813709 IC50 = 18000 nM T33754 CM25BT 13813714 IC50 = 13000 nM T33754 C1HCW0 13813715 IC50 = 14000 nM T33754 CH4R1T 13854249 IC50 = 870 nM T33754 CZ50CU 13887375 IC50 = 12000 nM T33754 CJWO46 13936973 IC50 = 80 nM T33754 C2W4ML 13936978 IC50 = 20 nM T33754 CI35CU 13936979 IC50 = 35 nM T33754 CT25ZJ 13936981 IC50 = 5 nM T33754 C5M2SC 13936982 IC50 = 8 nM T33754 C0ML2S 13936983 IC50 = 2000 nM T33754 CL9KE4 13936986 IC50 = 3000 nM T33754 CB28RL 13936987 IC50 = 3000 nM T33754 C70FKI 13946679 IC50 = 140000 nM T33754 C6FY4D 13946680 IC50 = 270000 nM T33754 CXE30O 13946684 IC50 = 120000 nM T33754 C9YAU8 13946685 IC50 = 54000 nM T33754 CF49KS 13946687 IC50 = 220000 nM T33754 CF03CE 13946690 IC50 = 590000 nM T33754 CZIR61 13987616 IC50 = 30 nM T33754 CB6DA7 13987617 IC50 = 50 nM T33754 CI9Z6F 13987618 IC50 = 70 nM T33754 C8UVR7 13987619 IC50 = 20 nM T33754 CWYX95 13987620 IC50 = 300 nM T33754 CT05NR 13987621 IC50 = 20 nM T33754 CD6C1Y 13987622 IC50 = 700 nM T33754 CZ7P2Q 13987623 IC50 = 600 nM T33754 CXMG34 13987624 IC50 = 300 nM T33754 CZ6H9F 13987625 IC50 = 5000 nM T33754 C9I1NU 13987626 IC50 = 300 nM T33754 C0HDT3 14067773 IC50 = 7000 nM T33754 CB21VK 14067774 IC50 = 62000 nM T33754 CH4LJ0 14067800 IC50 = 80000 nM T33754 CTK34P 14067801 IC50 = 37000 nM T33754 CV46DH 14067807 IC50 = 5000 nM T33754 CB3N8M 14067808 IC50 = 2000 nM T33754 CJF0S2 14067809 IC50 = 10000 nM T33754 CKI45Q 14067812 IC50 = 128000 nM T33754 C5RJ9F 14067813 IC50 = 2000 nM T33754 CYZ85N 14067814 IC50 = 35000 nM T33754 CASB70 14099426 IC50 = 4100 nM T33754 CI3J7R 14099427 IC50 = 1200 nM T33754 CQ1LY8 14099432 IC50 = 1100 nM T33754 CUS17I 14099444 IC50 = 40000 nM T33754 CP5JU9 14099446 IC50 = 50000 nM T33754 C17HNR 14099449 IC50 = 22000 nM T33754 CZ0YA7 14116989 IC50 = 10000 nM T33754 C8P9XB 14177142 IC50 = 250000 nM T33754 CMF30H 14208192 IC50 > 100000 nM T33754 C85PQM 14230055 IC50 = 9500 nM T33754 C6K8HM 14230056 IC50 = 100000 nM T33754 CCP14U 14230060 IC50 = 100 nM T33754 C0KBQ4 14230061 IC50 = 1000 nM T33754 CH4S8D 14280990 IC50 = 5 nM T33754 CD1Q4U 14280991 IC50 = 600 nM T33754 C03ZNU 14280992 IC50 = 70 nM T33754 CZ9WG1 14280994 IC50 = 5 nM T33754 CL4AF3 14280995 IC50 = 80 nM T33754 C1MK5R 14280996 IC50 = 7000 nM T33754 CCTP04 14280998 IC50 = 30 nM T33754 CXH95F 14280999 IC50 = 5000 nM T33754 CZ6N0W 14281000 IC50 = 40 nM T33754 CR1G8Y 14281001 IC50 = 1 nM T33754 C18OUM 14281003 IC50 = 20 nM T33754 CJ6VF1 14281004 IC50 = 700 nM T33754 CH1BM2 14281005 IC50 = 10 nM T33754 C9MY5X 14281006 IC50 = 0.5 nM T33754 CUCR03 14281008 IC50 = 30 nM T33754 CUFJ35 14281010 IC50 = 100 nM T33754 CQ8TE3 14281011 IC50 = 20 nM T33754 CSEC89 14281012 IC50 = 2000 nM T33754 C85BRF 14281014 IC50 = 2 nM T33754 CU0J8E 14281015 IC50 = 5 nM T33754 CDP92K 14281016 IC50 = 2 nM T33754 C6FCS9 14281018 IC50 = 200 nM T33754 CK3E1F 14281020 IC50 = 80 nM T33754 CUDO17 14281023 IC50 = 500 nM T33754 CZ19AJ 14281024 IC50 = 600 nM T33754 CY8PC6 14281025 IC50 = 2 nM T33754 CBT8K9 14281026 IC50 = 0.4 nM T33754 C3F7MZ 14281027 IC50 = 4 nM T33754 C2CF9I 14281031 IC50 = 50 nM T33754 CQ2YL0 14281033 IC50 = 9 nM T33754 CM1NW7 14281034 IC50 = 100 nM T33754 CEUF73 14281035 IC50 = 30 nM T33754 C7QJ4Y 14281036 IC50 = 300 nM T33754 CWSR46 14281041 IC50 = 100 nM T33754 C69RCW 14373260 IC50 = 40000 nM T33754 CE7L8R 14373269 IC50 = 6400 nM T33754 CB41NR 14373278 IC50 = 14000 nM T33754 C2ZX8H 14756622 IC50 = 300 nM T33754 CIK71M 14836119 IC50 = 15800 nM T33754 CU4B0C 14875705 IC50 = 4000 nM T33754 C0HM4P 14875707 IC50 = 6000 nM T33754 CQE6R7 14978533 IC50 = 9800 nM T33754 CZRD06 14978534 IC50 = 2000 nM T33754 CZ1ML0 15005564 IC50 = 20 nM T33754 CTL89M 15005565 IC50 = 300 nM T33754 CRO7P1 15005566 IC50 = 2000 nM T33754 CCO0S1 15005567 IC50 = 60 nM T33754 C74EYG 15005568 IC50 = 40000 nM T33754 C7RC1U 15005569 IC50 = 1000 nM T33754 CAC98D 15005570 IC50 = 4000 nM T33754 CW0UP4 15005571 IC50 = 4 nM T33754 C6I0LA 15005572 IC50 = 100 nM T33754 CM63ZU 15005573 IC50 = 5000 nM T33754 CE0DR4 15005574 IC50 = 3 nM T33754 CAQ7J2 15005576 IC50 = 2 nM T33754 CTE39J 15005577 IC50 = 0.3 nM T33754 C8TQ6C 15005578 IC50 = 20 nM T33754 C5Z8QA 15005579 IC50 = 8 nM T33754 CS17FZ 15005580 IC50 = 7 nM T33754 CN13YK 15005581 IC50 = 40 nM T33754 CQ9Y7J 15005583 IC50 = 40 nM T33754 CJ72ZA 15005584 IC50 = 20 nM T33754 CVA9B0 15005585 IC50 = 6 nM T33754 C4PM2K 15005586 IC50 = 20 nM T33754 C95NSJ 15005588 IC50 = 6 nM T33754 CI60HD 15005590 IC50 = 3 nM T33754 CDHV05 15005591 IC50 = 100 nM T33754 C7VR0Q 15005592 IC50 = 10 nM T33754 C7QZO0 15005594 IC50 = 2 nM T33754 CP6DI1 15005600 IC50 = 60 nM T33754 C0Z6GL 15005601 IC50 = 100 nM T33754 CTU06K 15005602 IC50 = 600 nM T33754 C23MUZ 15005603 IC50 = 900 nM T33754 CRA5G0 15005604 IC50 = 20 nM T33754 C96YTU 15005605 IC50 = 40 nM T33754 CH7I9M 15005606 IC50 = 300 nM T33754 CX9L6N 15005608 IC50 = 60 nM T33754 C2WC6S 15005610 IC50 = 0.3 nM T33754 C1TUZ8 15005611 IC50 = 7 nM T33754 CK2XC5 15005612 IC50 = 1 nM T33754 CC38GH 15005613 IC50 = 1 nM T33754 C1BWP3 15005614 IC50 = 0.4 nM T33754 C8UXF9 15005615 IC50 = 0.5 nM T33754 CU3OZ1 15005616 IC50 = 0.2 nM T33754 C6FG5L 15005617 IC50 = 0.7 nM T33754 CT7S5U 15005618 IC50 = 0.9 nM T33754 CSB54R 15005619 IC50 = 0.2 nM T33754 CL0GK4 15005620 IC50 = 7 nM T33754 CI9JG7 15005621 IC50 = 0.7 nM T33754 C2PG6E 15005622 IC50 = 2 nM T33754 COXV89 15005623 IC50 = 2 nM T33754 C0RXK5 15005624 IC50 = 9 nM T33754 CLOD12 15005625 IC50 = 0.4 nM T33754 C0NL5Y 15005626 IC50 = 3 nM T33754 CS3BZ0 15005627 IC50 = 0.9 nM T33754 C8RW7L 15005628 IC50 = 2 nM T33754 C5Z1VO 15005629 IC50 = 0.3 nM T33754 C6YWR9 15005630 IC50 = 0.7 nM T33754 C43TXQ 15005631 IC50 = 0.7 nM T33754 CWS8B1 15005632 IC50 = 3 nM T33754 C6MJL0 15005633 IC50 = 0.3 nM T33754 CX2V6D 15005634 IC50 = 0.03 nM T33754 C9PB2Q 15005635 IC50 = 0.6 nM T33754 C3XVH7 15005636 IC50 = 0.08 nM T33754 C5VFK8 15005637 IC50 = 7 nM T33754 C4BJ8X 15005638 IC50 = 5 nM T33754 CU6D4I 15005639 IC50 = 2 nM T33754 CIX0K1 15005640 IC50 = 6 nM T33754 COD9P3 15005641 IC50 = 0.6 nM T33754 CEY94T 15005642 IC50 = 40 nM T33754 CK7IF9 15005643 IC50 = 80 nM T33754 C2FJA7 15005644 IC50 = 30 nM T33754 CAL8G6 15005645 IC50 = 5 nM T33754 CV4N2T 15005646 IC50 = 0.7 nM T33754 CR02FE 15005648 IC50 = 40 nM T33754 C7XTH5 15005649 IC50 = 4 nM T33754 C71XNS 15005650 IC50 = 20 nM T33754 C2FN1U 15005651 IC50 = 40 nM T33754 C4AOZ5 15005652 IC50 = 4.5 nM T33754 C29CGS 15065141 IC50 = 200 nM T33754 CU8Q4O 15065142 IC50 = 300 nM T33754 C6GL1N 15065144 IC50 = 2000 nM T33754 C7FSN1 15065145 IC50 = 50 nM T33754 CI0BC3 15065146 IC50 = 5 nM T33754 CJ9G4E 15065157 IC50 = 150 nM T33754 CJI8S1 15065158 IC50 = 40 nM T33754 C0X4QW 15065159 IC50 = 20000 nM T33754 CDS3L9 15065160 IC50 = 7000 nM T33754 CJAW97 15065161 IC50 = 1500 nM T33754 C6R9QK 15065162 IC50 = 3000 nM T33754 CF2P5L 15065163 IC50 = 3000 nM T33754 C4C9LX 15065166 IC50 = 70000 nM T33754 C1YO3J 15294417 IC50 = 24000 nM T33754 CZ3P9I 15384033 IC50 > 3500 nM T33754 CBI7C9 15599405 IC50 = 50000 nM T33754 C79SKJ 15599407 IC50 = 50000 nM T33754 COIQ39 15599408 IC50 = 100000 nM T33754 C2JFW3 15599410 IC50 = 6000 nM T33754 C9UZY4 15599411 IC50 = 30000 nM T33754 CK85LM 15599412 IC50 = 4000 nM T33754 CL25OI 15599415 IC50 = 630000 nM T33754 CB8AD5 15599416 IC50 = 18000 nM T33754 CKG0I7 15599419 IC50 = 5000 nM T33754 C0FIW4 15599420 IC50 = 6000 nM T33754 CI6PO7 15599423 IC50 = 20000 nM T33754 C9SZV1 15599429 IC50 = 5000 nM T33754 CC7B9I 15599430 IC50 = 8000 nM T33754 CO1B9U 15599431 IC50 = 23000 nM T33754 CZR79K 15599432 IC50 = 36000 nM T33754 CAV9T1 15599433 IC50 = 31000 nM T33754 C7QLW4 15599434 IC50 = 26000 nM T33754 C08RKB 15599435 IC50 = 28000 nM T33754 CF1AI9 15599436 IC50 = 7500 nM T33754 CS62TE 15599439 IC50 = 300 nM T33754 CAC5H0 15606258 IC50 > 100000 nM T33754 C8E9XA 15696722 IC50 = 300 nM T33754 C4ZQ1O 15696723 IC50 = 940 nM T33754 C0ZY9U 15696724 IC50 = 3200 nM T33754 CE50XZ 15717870 IC50 = 2000 nM T33754 CQK95D 15717874 IC50 = 30000 nM T33754 CX4BD2 15717877 IC50 = 7000 nM T33754 CZ4LV6 15717878 IC50 = 45000 nM T33754 C40CME 15717879 IC50 = 40000 nM T33754 CW6MV8 15981426 IC50 = 1300 nM T33754 CL2Y9X 16735134 IC50 = 78 nM T33754 C1PZ8C 18734933 IC50 > 16000 nM T33754 CJ95TM 20146320 IC50 = 3500 nM T33754 CDC76R 20299686 IC50 > 50000 nM T33754 CV74MN 23275981 IC50 = 39810.72 nM T33754 C20VHK 24871823 IC50 = 170 nM T33754 CJ4V0W 44178556 IC50 = 125100 nM T33754 C5X9AD 44209387 IC50 > 100000 nM T33754 C0ZKN1 44209388 IC50 > 100000 nM T33754 CW3O0T 44272155 IC50 = 65000 nM T33754 CNFR26 44272157 IC50 = 10000 nM T33754 CYP61N 44272162 IC50 = 80000 nM T33754 C5ZQN0 44272176 IC50 = 38000 nM T33754 C24ZCG 44272215 IC50 = 40000 nM T33754 CXHP96 44272313 IC50 = 150000 nM T33754 C78OJW 44272327 IC50 = 28000 nM T33754 CSR6M9 44272328 IC50 = 20000 nM T33754 CJ19DZ 44272333 IC50 = 7000 nM T33754 CRO63G 44272338 IC50 = 15000 nM T33754 C1VGQ0 44272341 IC50 = 150000 nM T33754 CRO37P 44274658 IC50 > 100000 nM T33754 C35KNC 44274717 IC50 > 100000 nM T33754 CU36PK 44274868 IC50 > 100000 nM T33754 CDN62V 44274869 IC50 = 840 nM T33754 CA6J8T 44274920 IC50 = 880 nM T33754 CX89AE 44279648 IC50 = 68000 nM T33754 C7NHE8 44279839 IC50 = 220000 nM T33754 CK8Y4F 44286951 IC50 > 50000 nM T33754 CIC45P 44294818 IC50 > 200000 nM T33754 CWTK85 44295026 IC50 > 200000 nM T33754 CEH82G 44295178 IC50 = 250000 nM T33754 CNK73O 44295200 IC50 = 339000 nM T33754 COBW92 44301890 IC50 = 1900 nM T33754 CW75QH 44312546 IC50 = 8 nM T33754 CL80RT 44314758 IC50 = 5300 nM T33754 C3ID9H 44314916 IC50 > 25000 nM T33754 CC6F4N 44315110 IC50 > 100000 nM T33754 C0KT9E 44318468 IC50 < 10000 nM T33754 C4RWG3 44318473 IC50 < 10000 nM T33754 C3L6AF 44319378 IC50 > 3162.28 nM T33754 CLBV45 44320831 IC50 > 10000 nM T33754 CVS5D1 44320863 IC50 > 10000 nM T33754 C0GM7F 44320900 IC50 > 10000 nM T33754 C4VFQ5 44321253 IC50 = 5570 nM T33754 CUQ3R1 44321255 IC50 > 10000 nM T33754 C7BM6I 44321261 IC50 > 10000 nM T33754 CR41FC 44323256 IC50 = 111000 nM T33754 C05VLD 44323257 IC50 = 68000 nM T33754 C2-JAN-01 44323270 IC50 > 200000 nM T33754 CBP5I9 44323409 IC50 > 20000 nM T33754 C0XZ6H 44323410 IC50 > 20000 nM T33754 CK5ZG3 44323424 IC50 > 20000 nM T33754 CFUB24 44323425 IC50 > 20000 nM T33754 CP5N9V 44323427 IC50 > 200000 nM T33754 C5IJQ8 44323428 IC50 > 20000 nM T33754 CMFX02 44323504 IC50 > 20000 nM T33754 C21UJZ 44323510 IC50 = 136000 nM T33754 CAH1Q0 44323556 IC50 > 20000 nM T33754 CTY4U2 44323790 IC50 = 6 nM T33754 CZ16IY 44324251 IC50 = 30000 nM T33754 CCX9Z3 44324252 IC50 = 7000 nM T33754 CG6UT1 44324296 IC50 = 20000 nM T33754 C8M4WJ 44324373 IC50 = 14000 nM T33754 CY5HZ7 44324390 IC50 = 50000 nM T33754 C5KYV6 44324391 IC50 = 50000 nM T33754 C5C4QX 44324507 IC50 = 57000 nM T33754 CXUC09 44329640 IC50 = 430 nM T33754 CA5MY8 44329642 IC50 = 720 nM T33754 CSD45M 44329651 IC50 = 430 nM T33754 CUA7P5 44329666 IC50 = 390 nM T33754 C2M3QE 44329683 IC50 = 310 nM T33754 C9R0OI 44329684 IC50 = 7800 nM T33754 CWM23U 44329685 IC50 = 700 nM T33754 CQ2WU3 44329686 IC50 = 340 nM T33754 CNK2F8 44331802 IC50 = 580 nM T33754 CZ89AS 44333023 IC50 = 10000 nM T33754 CX7E4M 44333357 IC50 = 53000 nM T33754 C5JN7O 44333375 IC50 = 13000 nM T33754 C5ZLT1 44333376 IC50 = 100000 nM T33754 CCOZ32 44339609 IC50 > 300000 nM T33754 C2G4BD 44344410 IC50 = 87000 nM T33754 CA3RE9 44344568 IC50 = 18 nM T33754 CH9P3C 44348937 IC50 = 62000 nM T33754 CVA3O4 44348938 IC50 = 27000 nM T33754 CVW1P2 44348994 IC50 > 100000 nM T33754 C5T6BV 44348995 IC50 = 7850 nM T33754 C2Q9XZ 44349115 IC50 = 17500 nM T33754 C5DKS3 44349135 IC50 = 43700 nM T33754 CS4QH0 44349295 IC50 > 100000 nM T33754 C8L4GH 44350226 IC50 = 200000 nM T33754 CNM4Y5 44350243 IC50 = 4000 nM T33754 C4GDB0 44352576 IC50 > 200000 nM T33754 C0WH4X 44352624 IC50 > 200000 nM T33754 CC3P1L 44352733 IC50 > 200000 nM T33754 C2G1JL 44363503 IC50 = 570 nM T33754 CZX3H7 44364909 IC50 = 5800 nM T33754 C8HWG0 44364924 IC50 = 5400 nM T33754 C9YDX5 44364932 IC50 = 16000 nM T33754 C2WGA3 44365034 IC50 = 11000 nM T33754 CAM5B4 44365046 IC50 = 4800 nM T33754 C9FME0 44365068 IC50 = 125000 nM T33754 CA26VF 44365094 IC50 = 7000 nM T33754 CE0MT4 44365229 IC50 = 6800 nM T33754 C6EBY9 44367306 IC50 > 500000 nM T33754 C7MI2E 44367386 IC50 = 73 nM T33754 CT8NH9 44383851 IC50 > 10000 nM T33754 C19CRH 44383901 IC50 = 3900 nM T33754 CR9O3I 44383902 IC50 = 1100 nM T33754 CW47HV 44383906 IC50 = 2500 nM T33754 CL86MY 44383907 IC50 > 1000 nM T33754 CW63HQ 44383912 IC50 > 1000 nM T33754 CF98LG 44384286 IC50 = 6400 nM T33754 CN1WS7 44384345 IC50 > 10000 nM T33754 C01XPL 44384404 IC50 = 2100 nM T33754 CWPR87 44384405 IC50 = 2100 nM T33754 C59SDR 44384406 IC50 = 3500 nM T33754 C7WT4G 44384540 IC50 = 4500 nM T33754 C4RQB0 44384541 IC50 = 2300 nM T33754 CRZ5G8 44384546 IC50 = 14400 nM T33754 C6W4GY 44384713 IC50 = 8500 nM T33754 CKH7M8 44384714 IC50 = 3600 nM T33754 C0ZGU6 44385109 IC50 = 1500 nM T33754 CE80VB 44385244 IC50 = 840 nM T33754 CH5GU8 44385282 IC50 = 1200 nM T33754 CL50UE 44385283 IC50 = 4400 nM T33754 CZF29N 44397816 IC50 > 10000 nM T33754 C7RV5Q 44438554 IC50 = 1640 nM T33754 C50ZMB 44438560 IC50 = 3130 nM T33754 CJH70L 44438564 IC50 = 1850 nM T33754 C8F3UO 44562338 IC50 = 31.62 nM T33754 C45ZVC 45258276 IC50 = 1500 nM T33754 C2N9HA 45259270 IC50 = 29000 nM T33754 C10TQI 45259276 IC50 = 700 nM T33754 CBKJ47 45259284 IC50 > 100000 nM T33754 CSX9O6 45259293 IC50 = 690 nM T33754 C31FMT 45260180 IC50 > 200000 nM T33754 CCQ35I 45260248 IC50 > 200000 nM T33754 C4BDC7 45261609 IC50 = 77 nM T33754 CSJZ49 45263853 IC50 = 3500 nM T33754 CVSY51 45263858 IC50 = 16000 nM T33754 C1Y9CW 45263914 IC50 = 5600 nM T33754 C0D2MN 46186792 IC50 = 1240 nM T33754 C0WRO9 46198713 IC50 = 7260 nM T33754 CXG34R 46199487 IC50 > 5000 nM T33754 CAL85J 46199794 IC50 > 10000 nM T33754 CI9EA4 46199799 IC50 > 10000 nM T33754 C26RJV 46200090 IC50 > 10000 nM T33754 C5WND9 46200233 IC50 > 10000 nM T33754 CKIC45 46200238 IC50 > 10000 nM T33754 CS46AE 46200399 IC50 > 10000 nM T33754 C1S3BK 46200706 IC50 > 10000 nM T33754 C4P5QJ 46200709 IC50 > 10000 nM T33754 CV8Y6W 46200711 IC50 > 10000 nM T33754 CK1N4X 46200728 IC50 > 1000 nM T33754 CH9FU8 46200877 IC50 > 1000 nM T33754 CEZ3V4 46200878 IC50 = 2250 nM T33754 CI1F5C 46239840 Ki >= 770 nM T33754 C26XVS 46240044 Ki >= 4793 nM T33754 CE4JU7 46842025 IC50 > 10000 nM T33754 CR8JC2 46842169 IC50 > 10000 nM T33754 CIU98Y 49860585 IC50 = 1.13 nM T33754 CV2B7D 49860590 IC50 = 1.13 nM T33754 C7H8OY 49860597 IC50 = 0.84 nM T33754 CS5T3A 49860598 IC50 = 0.63 nM T33754 CSPT34 49860600 IC50 = 1.03 nM T33754 C9Z2SB 49860605 IC50 = 0.81 nM T33754 C0WIU6 49860618 IC50 = 0.81 nM T33754 CBW18A 49860622 IC50 = 2.78 nM T33754 C4U6IX 49860628 IC50 = 1.25 nM T33754 C4D7IC 49860633 IC50 = 5.14 nM T33754 C4KIL0 49860634 IC50 = 2.56 nM T33754 CKD7N1 49860647 IC50 = 1.11 nM T33754 C3EX0U 49860648 IC50 > 10 nM T33754 CP29YZ 49860650 IC50 = 1.13 nM T33754 CN2K8B 49860655 IC50 = 4.96 nM T33754 CBG3J8 49860656 IC50 = 5.42 nM T33754 CURB28 54587645 IC50 = 10000 nM T33754 C0ZF1L 57328385 IC50 > 25000 nM T33754 C2PJ4N 59271992 IC50 = 1000 nM T33754 C7PB1U 59321218 IC50 = 750 nM T33754 CS32XI 59321284 IC50 > 10000 nM T33754 C23WQA 59321310 IC50 > 10000 nM T33754 CZ6C9L 59321318 IC50 > 10000 nM T33754 C1OHZ0 59321339 IC50 > 5000 nM T33754 C0AFM6 60150358 IC50 > 5000 nM T33754 C6C8RD 66802145 IC50 = 1030 nM T33754 CTJ46X 68594477 IC50 > 1000 nM T33754 C8E0XY 68596001 IC50 > 10000 nM T33754 CJ80VI 68596013 IC50 > 10000 nM T33754 CL2H4T 68596452 IC50 > 10000 nM T33754 C93IHS 68596628 IC50 > 10000 nM T33754 CDZ01B 68596639 IC50 > 1000 nM T33754 C1CD9S 68596902 IC50 > 10000 nM T33754 C7PCW0 68597211 IC50 > 1000 nM T33754 CGJB21 68597401 IC50 > 10000 nM T33754 CHK4S0 68597804 IC50 > 10000 nM T33754 C10TGO 68598825 IC50 > 10000 nM T33754 CCN10Q 70662473 IC50 > 1000 nM T33754 CUA5C6 70682518 IC50 = 1680 nM T33754 CPX6Q3 70684576 IC50 = 7490 nM T33754 C2F1WD 70684577 IC50 = 7300 nM T33754 C6DU3W 70686742 IC50 = 312400 nM T33754 C8F2IH 70686743 IC50 = 128300 nM T33754 CM3OP8 70686796 IC50 > 10000 nM T33754 CHBT91 70686797 IC50 > 1000 nM T33754 CJCW26 70688819 IC50 = 38500 nM T33754 C8RHV0 70688820 IC50 = 2660 nM T33754 CYM94A 70688823 IC50 = 8470 nM T33754 CU4I5V 70690900 IC50 = 172500 nM T33754 CR0BM7 70690901 IC50 = 163500 nM T33754 C4YI0P 70695095 IC50 = 423200 nM T33754 CA01QU 70695096 IC50 = 280700 nM T33754 CQR40F 70697129 IC50 = 172130 nM T33754 CF03DW 90168772 IC50 > 20000 nM T33754 CM6J9K 90168778 IC50 > 20000 nM T33754 CVYK24 118556943 IC50 > 50000 nM T33754 C1QMI8 135401477 IC50 > 500 nM T33754 C17YXR 135406983 IC50 > 500 nM T33754 CMHA51 135407168 IC50 = 240 nM T33754 CP3CL2 135410273 IC50 = 150 nM T33754 CXET38 135418296 IC50 = 240 nM T33754 CNP87H 135433645 IC50 > 100000 nM T33754 CMG81E 135434015 IC50 = 3 nM T33754 C94RVJ 135438569 IC50 > 500 nM T33754 CZJY69 135442775 IC50 > 100000 nM T33754 C0DBS7 135452901 IC50 = 62000 nM T33754 CFKO84 135455980 IC50 > 100000 nM T33754 CR6B9J 135456675 IC50 > 100000 nM T33754 C3MWQ9 135474380 IC50 = 83 nM T33754 CGF5P1 135485711 IC50 = 8800 nM T33754 C7SYV0 135506388 IC50 = 2600 nM T33754 CK6CQ7 135515478 IC50 = 72 nM T33754 CB1QD5 135516730 IC50 = 70 nM T33754 CP71WA 135528334 IC50 > 100000 nM T33754 C8E3OA 135531470 IC50 > 100000 nM T33754 C4ASW0 135544141 IC50 > 500 nM T33754 CK8PF5 135583531 IC50 = 520 nM T33754 C7TM3P 135626217 IC50 = 2.7 nM T33754 CZ06BM 135626238 IC50 = 9.2 nM T33754 C58IVM 135626472 IC50 = 48 nM T33754 COJQ24 135626489 IC50 = 5.9 nM T33754 C1XTH2 135626495 IC50 = 1.3 nM T33754 C7WOJ4 135626500 IC50 = 4.6 nM T33754 CQX8E7 135626515 IC50 = 16 nM T33754 CIE79C 135626519 IC50 > 100000 nM T33754 CX06PV 135626541 IC50 = 26 nM T33754 CA8VZ4 135626546 IC50 = 26 nM T33754 C32DLX 135626547 IC50 = 150 nM T33754 C5MDK4 135626551 IC50 = 1.5 nM T33754 CBMT84 135626563 IC50 = 820 nM T33754 CI3PO1 135626568 IC50 = 690 nM T33754 CH8G2M 135626614 IC50 = 3.6 nM T33754 CP81SR 135626617 IC50 = 2000 nM T33754 CJ10HE 135626618 IC50 = 15 nM T33754 C18BJR 135626635 IC50 = 1600 nM T33754 C62SAO 135626651 IC50 = 12 nM T33754 CFS3I4 135626691 IC50 = 2.2 nM T33754 C9MI0X 135626744 IC50 = 5400 nM T33754 C29FKY 135626784 IC50 = 1.45 nM T33754 C5M9KO 135626813 IC50 = 14 nM T33754 C9WI1F 135626836 IC50 = 3.2 nM T33754 C13OYK 135626842 IC50 = 1 nM T33754 CC5Z2N 135666682 IC50 = 600 nM T33754 C3KUC8 135667658 IC50 = 2000 nM T33754 C9OKL0 135668094 IC50 = 700 nM T33754 C7VBI4 135740146 IC50 > 100 nM T33754 CA5NJ0 135823924 IC50 = 1500 nM T33754 C31VFB 135832642 IC50 > 100000 nM T33754 C76RFB 135838394 IC50 = 3300 nM T33754 CE24WD 135838395 IC50 = 40 nM T33754 CRC0Z9 135838396 IC50 = 240 nM T33754 CZOT04 136000670 IC50 = 18000 nM T33754 C8YU1M 136023817 IC50 = 12.5 nM T33754 CR90MI 136026575 IC50 = 8 nM T33754 CTBR86 136026576 IC50 = 6 nM T33754 C6OU3Z 136034782 IC50 > 500 nM T33754 CO9FA3 136035288 IC50 = 300 nM T33754 C5ZIU7 136056125 IC50 > 100000 nM T33754 C70DJG 136056126 IC50 = 34000 nM T33754 C9Q3BW 136056127 IC50 = 63000 nM T33754 C4U1SF 136056128 IC50 = 47000 nM T33754 CI8E5F 136056129 IC50 = 83000 nM T33754 CH92FZ 136058101 IC50 = 290 nM T33754 CI3Z5D 136058102 IC50 = 560 nM T33754 C8PD0K 136058103 IC50 = 600 nM T33754 C13XWR 136058104 IC50 = 26000 nM T33754 CDKT63 136058105 IC50 = 30000 nM T33754 CK8AO5 136058106 IC50 = 18000 nM T33754 CXYS73 136058107 IC50 = 330000 nM T33754 CL42GB 136058108 IC50 = 1500 nM T33754 C6WH2S 136078534 IC50 > 500 nM T33754 C3H7CG 136142433 IC50 = 10000 nM T33754 C4HDJ6 136142434 IC50 > 10000 nM T33754 CUAJ91 136142435 IC50 = 370 nM T33754 CI2K9X 136142436 IC50 = 5.4 nM T33754 C6GH2D 136142437 IC50 = 3300 nM T33754 CU7KY1 136142438 IC50 = 25000 nM T33754 CD2XA8 136142439 IC50 = 17 nM T33754 CLUH17 136142440 IC50 = 1200 nM T33754 CL6CQ7 136142441 IC50 = 27.5 nM T33754 C4O7AN 136142442 IC50 = 4400 nM T33754 CGV71R 136142443 IC50 = 200 nM T33754 CU5OW3 136142444 IC50 = 3800 nM T33754 C45RMB 136142445 IC50 = 1000 nM T33754 CSMY91 136142446 IC50 > 10000 nM T33754 CI5W0G 136142447 IC50 = 6.4 nM T33754 CR7V3M 136142448 IC50 > 10000 nM T33754 C9KH1P 136142449 IC50 = 6 nM T33754 C4Y1QU 136142450 IC50 = 580 nM T33754 C5NPS9 136142451 IC50 = 26 nM T33754 CIN5D2 136142452 IC50 = 340 nM T33754 C7WPY3 136142453 IC50 = 4.1 nM T33754 CEW57J 136142454 IC50 = 1 nM T33754 CIH0D9 136142455 IC50 = 1600 nM T33754 CID97M 136142456 IC50 = 4.9 nM T33754 CH2U9V 136142457 IC50 = 260 nM T33754 CTM6W3 136142458 IC50 = 1600 nM T33754 C8TGF9 136142459 IC50 = 18.5 nM T33754 CMNO98 136142460 IC50 = 1.85 nM T33754 CO34ZP 136142461 IC50 = 76 nM T33754 C7VJX6 136142462 IC50 = 5 nM T33754 C7HG8U 136142463 IC50 = 5.6 nM T33754 CMO62W 136142464 IC50 = 13.5 nM T33754 CTZR90 136142465 IC50 = 180 nM T33754 CYR1K6 136142466 IC50 = 11 nM T33754 COS9I7 136142467 IC50 = 2 nM T33754 C4VW9B 136142468 IC50 = 120 nM T33754 CND42L 136142469 IC50 = 12 nM T33754 CXZM43 136142470 IC50 = 1.1 nM T33754 C9S8RE 136142471 IC50 = 1.45 nM T33754 C8EVA1 136142472 IC50 = 18 nM T33754 CY49SD 136142473 IC50 = 10 nM T33754 C0J9IZ 136142474 IC50 = 0.94 nM T33754 C1QHS2 136142476 IC50 = 760 nM T33754 C0EV7C 136142477 IC50 = 4.5 nM T33754 CIP98Q 136142478 IC50 = 3100 nM T33754 CY9EB3 136142479 IC50 = 1700 nM T33754 C2VI5E 136142480 IC50 = 470 nM T33754 CD9IK1 136142481 IC50 = 130 nM T33754 CA6BF0 136142482 IC50 = 140 nM T33754 C6CZW9 136144096 IC50 = 13 nM T33754 CQW7T0 136197286 IC50 > 10000 nM T33754 D00YPO 14032753 IC50 = 110 nM T33754 D01RUN 448055 IC50 > 3162.28 nM T33754 D01TOR 667555 IC50 > 100000 nM T33754 D02NWF 2573787 IC50 > 100000 nM T33754 D03GAQ 15065156 IC50 = 10 nM T33754 D04KDB 13885278 IC50 = 16000 nM T33754 D05HFD 13936971 IC50 = 50 nM T33754 D08XKO 15065155 IC50 = 300 nM T33754 D09AUL 10266864 IC50 = 50000 nM T33754 D09CPC 13728862 IC50 = 4400 nM T33754 D09GTN 13936969 IC50 = 300 nM T33754 D09LAQ 135398570 IC50 = 2400 nM T33754 D0DL6J 9843744 IC50 > 100000 nM T33754 D0DX3V 13936989 IC50 = 20 nM T33754 D0I6XA 149784 Ki > 200000 nM T33754 D0J0CB 2753 Ki = 5 nM T33754 D0J7GF 780643 IC50 > 100000 nM T33754 D0J7NR 15065143 IC50 = 90 nM T33754 D0LZ5R 5368 IC50 > 100000 nM T33754 D0N6MR 10867033 IC50 = 500 nM T33754 D0NI4Z 13936972 IC50 = 50 nM T33754 D0O3BL 19700663 IC50 = 5100 nM T33754 D0S4JI 20262 IC50 > 200000 nM T33754 D0T3UP 13724742 IC50 = 7000 nM T33754 D0TZ8C 14373279 IC50 = 4000 nM T33754 D0U8YQ 921562 IC50 > 100000 nM T33754 D0V4WB 149790 IC50 > 16000 nM T33754 D0V5BX 68765 IC50 > 200000 nM T95947 D0I0RJ 16231 IC50 = 4400 nM T95947 CV9U4J 237074 IC50 = 97000 nM T95947 C98HYW 350414 IC50 = 363000 nM T95947 CWQ6T8 598430 IC50 = 763000 nM T95947 CF8D7P 817383 IC50 = 130000 nM T95947 C2L8DB 910176 IC50 = 430000 nM T95947 C5DZ4S 2762833 IC50 = 6900 nM T95947 C1FXO2 3010990 IC50 = 6300 nM T95947 CJ79MR 11160454 IC50 = 9000 nM T95947 C4HR0W 11413259 IC50 = 190000 nM T95947 C0OKV6 15885183 IC50 = 701000 nM T95947 C9JO6S 21473659 IC50 = 3300 nM T95947 CEG0S4 25210286 IC50 = 133000 nM T95947 CL8F3J 25254508 IC50 = 95000 nM T95947 CN1A2U 25254510 IC50 = 374000 nM T95947 CVJ09D 25254512 IC50 = 77000 nM T95947 CGP5U4 29949062 IC50 = 160000 nM T95947 CQG62F 42630453 IC50 = 490 nM T95947 CNB07T 44276630 IC50 = 2765000 nM T95947 CIRV37 44574852 IC50 = 510 nM T95947 C3UZ1O 44575053 IC50 = 640 nM T95947 CA13UC 45268405 IC50 = 135000 nM T95947 CUD7O4 45268406 IC50 = 278000 nM T95947 CBY5A2 45270104 IC50 = 291000 nM T95947 C2UM9J 45270105 IC50 = 59000 nM T95947 CGVY53 45270945 IC50 = 114000 nM T95947 CK36FD 45272657 IC50 = 272000 nM T95947 CRT7U8 45272658 IC50 = 59000 nM T95947 CH4P7Z 45273577 IC50 = 51000 nM T95947 CT3F0N 53235532 IC50 = 3800 nM T95947 CG69CQ 53327817 IC50 = 3100 nM T95947 CC5JU4 53357591 IC50 = 220 nM T95947 CV8O9S 54580851 IC50 = 10900 nM T95947 C8DU2L 54580852 IC50 = 1700 nM T95947 CL2VD1 54581911 IC50 = 27600 nM T95947 C6JNA1 54581912 IC50 = 7100 nM T95947 C7FXW8 54581913 IC50 = 103000 nM T95947 CMR50V 54582827 IC50 = 17000 nM T95947 C2CWP3 54582828 IC50 = 9600 nM T95947 CM2N0V 54583845 IC50 = 14400 nM T95947 CVH03X 54585747 IC50 = 5800 nM T95947 CF93ML 54586726 IC50 = 19400 nM T95947 C5J3IG 54587763 IC50 = 2600 nM T95947 C8I7BE 54587764 IC50 = 1200 nM T95947 CXD10Y 56659437 IC50 > 50000 nM T95947 CZE85N 56659438 IC50 > 50000 nM T95947 CG0D5O 56659439 IC50 = 2500 nM T95947 C4PVI5 56662841 IC50 = 17100 nM T95947 C3VU5T 56662880 IC50 = 460 nM T95947 C8S0UA 56662881 IC50 = 4800 nM T95947 C5PC6Y 56662884 IC50 = 510 nM T95947 CK18MS 56666368 IC50 = 230 nM T95947 CDTA43 56666369 IC50 = 10200 nM T95947 C7UCQ9 56669778 IC50 = 310 nM T95947 C4Y2VS 56669779 IC50 = 230 nM T95947 C29ZIH 56669780 IC50 = 190 nM T95947 CX65FU 56673271 IC50 = 2800 nM T95947 COB8C7 56676588 IC50 = 270 nM T95947 CLT4K0 56679936 IC50 = 680 nM T95947 C5JMB3 56683256 IC50 = 3400 nM T95947 CSG38B 56683258 IC50 = 4300 nM T25315 D00XBC 46861584 IC50 > 10000 nM T25315 CLK7P3 169713 IC50 > 10000 nM T25315 C8TI6Z 197750 IC50 = 4570 nM T25315 CQX4M9 265219 IC50 > 60000 nM T25315 CEV5K8 384454 IC50 > 100000 nM T25315 CXQE10 384455 IC50 = 8000 nM T25315 C80QFG 384457 IC50 = 3000 nM T25315 CK20TD 594995 IC50 = 800 nM T25315 C3KCR4 703047 IC50 = 800 nM T25315 CB3Y5H 703050 IC50 = 3500 nM T25315 CLC86X 742729 IC50 = 4000 nM T25315 CX3FU4 871434 IC50 = 1100 nM T25315 CCAR78 1378429 Ki = 3981.07 nM T25315 CX6VK4 1448380 IC50 > 12589.25 nM T25315 CK6BI3 2396278 IC50 = 2940 nM T25315 COT07B 3453336 IC50 > 60000 nM T25315 C85BVJ 4239764 Ki = 3981.07 nM T25315 CG2MN3 4324393 IC50 = 250 nM T25315 CJB37A 6143230 Ki = 211 nM T25315 C86QRZ 9871365 IC50 = 3300 nM T25315 C1ZF0K 9886775 Ki = 110 nM T25315 C2PM8U 9913494 IC50 = 15000 nM T25315 CUB3G7 9938326 IC50 = 6 nM T25315 CMUB67 9938965 IC50 = 14 nM T25315 C81TFE 11296495 IC50 = 20 nM T25315 C97LDW 11386761 IC50 = 930 nM T25315 CVGK31 11497512 Ki = 140 nM T25315 C8TX6O 11498089 IC50 = 11 nM T25315 C1Y6EO 11526863 Ki = 160 nM T25315 CMGN54 11569938 IC50 = 0.2 nM T25315 CR0Q7V 11599725 IC50 = 35 nM T25315 CLQ14F 11635543 Ki = 320 nM T25315 CMZ08A 11707105 Ki = 85 nM T25315 C39SQF 11713886 Ki = 70 nM T25315 CWA39Z 11725848 IC50 = 2000 nM T25315 CNPX34 11757854 IC50 = 4.1 nM T25315 C91ZWK 11854699 IC50 = 6.8 nM T25315 C5EN9M 11856829 IC50 = 1.3 nM T25315 CE5AL8 11856830 IC50 = 1.4 nM T25315 CB8X2P 11964007 IC50 = 8 nM T25315 CJ1V6Z 11995700 IC50 = 1 nM T25315 C0P3HV 11995702 IC50 = 1.2 nM T25315 C7ZXA5 11995703 IC50 = 1.3 nM T25315 CYP1D7 11995772 IC50 = 9 nM T25315 CM71UD 11995774 Ki = 0.4 nM T25315 C2SR7I 11995974 IC50 = 2 nM T25315 C6B2LT 11995976 IC50 = 2.2 nM T25315 C8YLS5 11996050 IC50 = 1.5 nM T25315 C2VO4N 11996051 IC50 = 1.9 nM T25315 C1OM3A 11996344 IC50 = 1.9 nM T25315 C96NUB 11996409 IC50 = 3.9 nM T25315 C3J1YV 11996560 IC50 = 4.2 nM T25315 CZQ47C 11996722 IC50 = 5.2 nM T25315 C9PY6Q 11996726 IC50 = 6 nM T25315 C3FV2N 11997121 IC50 = 5.4 nM T25315 CD8P4G 11997270 IC50 = 18 nM T25315 CH6S5Q 11997334 IC50 = 1.8 nM T25315 CWR74C 11997336 IC50 = 6.4 nM T25315 CXSV02 11997474 IC50 = 3.6 nM T25315 CX0BJ7 11997620 IC50 = 1.5 nM T25315 CFQE74 11997623 IC50 = 3.4 nM T25315 CW6DT4 11997695 IC50 = 0.3 nM T25315 CD2WH3 11997761 IC50 = 0.4 nM T25315 CH21MR 11997845 IC50 = 0.4 nM T25315 CW0OT8 11997912 IC50 = 0.8 nM T25315 CRF9W1 11997994 IC50 = 0.8 nM T25315 C56KLN 11997995 IC50 = 0.3 nM T25315 C3DAP8 14479861 IC50 = 830 nM T25315 C19BYU 14479864 IC50 = 330 nM T25315 CNOH94 15560447 IC50 = 2400 nM T25315 C4C1BL 15604604 IC50 = 60 nM T25315 CY8QA1 15604606 IC50 = 120 nM T25315 CD4XZ9 15604607 IC50 = 170 nM T25315 C8AYG5 15604608 IC50 = 1250 nM T25315 CA3F2D 15604688 IC50 = 700 nM T25315 CJWO23 15604689 IC50 = 130 nM T25315 C80SEI 15604690 IC50 = 800 nM T25315 C9X7KF 15604773 IC50 = 80 nM T25315 CQD8K4 15604774 IC50 = 300 nM T25315 C65NQZ 15604776 IC50 = 2160 nM T25315 CYB49S 15604856 IC50 = 60 nM T25315 CZC28M 15604859 IC50 = 340 nM T25315 CF37DQ 15604934 IC50 = 320 nM T25315 C5GCE0 15604935 IC50 = 60 nM T25315 CL5ZI0 15604937 IC50 = 420 nM T25315 CT0B6H 15604938 IC50 = 240 nM T25315 CD3U7V 15605007 IC50 = 590 nM T25315 CSM0E4 15605012 IC50 = 490 nM T25315 CI4F5R 15605071 IC50 = 340 nM T25315 CF2RE4 15605073 IC50 = 250 nM T25315 CPIL45 15605074 IC50 = 50 nM T25315 C2O6LA 15605075 IC50 = 510 nM T25315 CUC1O6 15605137 IC50 = 290 nM T25315 CE29DR 15605197 IC50 = 70 nM T25315 CC1FM8 15605618 IC50 = 640 nM T25315 CV3NQ0 16040696 IC50 = 11 nM T25315 C2ARS4 16214851 IC50 = 3162.28 nM T25315 CX32OZ 17754430 IC50 = 2200 nM T25315 C97IHN 17754488 IC50 = 30 nM T25315 C8NYG4 17754713 IC50 = 800 nM T25315 C6C4QK 17754758 IC50 = 400 nM T25315 CX18AK 17754794 IC50 = 8000 nM T25315 CJI3V4 17754798 IC50 = 800 nM T25315 CAQ7S0 17754836 IC50 = 1000 nM T25315 C1CG7D 23593653 IC50 = 3100 nM T25315 CETZ25 23790139 IC50 = 40000 nM T25315 C7N4BG 24739386 IC50 = 150 nM T25315 C8KTP0 24739387 IC50 = 2310 nM T25315 CN9SZ0 24739388 IC50 = 210 nM T25315 C70CVK 24739554 IC50 = 30 nM T25315 C7K5DU 24739555 IC50 = 320 nM T25315 CSDA50 24739886 IC50 = 80 nM T25315 C12LWD 24739888 IC50 = 290 nM T25315 CY09OP 24739889 IC50 = 250 nM T25315 CMPR25 24774715 IC50 = 340 nM T25315 CUY89J 24936155 Ki = 7 nM T25315 CYLZ53 24947459 IC50 = 794.33 nM T25315 C0V8YL 24957182 IC50 = 8 nM T25315 C7D6KF 25008271 IC50 = 80 nM T25315 COH9V1 25032696 IC50 = 12 nM T25315 C9E6YT 25032697 IC50 = 7.8 nM T25315 C5NE1L 25032779 IC50 = 2 nM T25315 CJ32HC 25265835 IC50 = 31.62 nM T25315 C5NZI8 27307547 IC50 = 251.19 nM T25315 CAE5J4 34747495 IC50 = 2275 nM T25315 C5O1MR 44137674 IC50 = 7 nM T25315 C5ZJG2 44138054 Ki = 158.49 nM T25315 CYN7W6 44182602 IC50 = 7 nM T25315 C4E0DK 44237762 IC50 = 25 nM T25315 C5YFB9 44252324 IC50 > 10000 nM T25315 C31VGY 44253167 IC50 = 1295 nM T25315 C4H6BG 44253168 IC50 = 200 nM T25315 CV17CB 44253169 IC50 = 1985 nM T25315 C6P4LJ 44253170 IC50 = 2450 nM T25315 C42OMV 44253446 IC50 = 496 nM T25315 CYU6I9 44253447 IC50 = 697 nM T25315 C8C0YJ 44253448 IC50 = 673 nM T25315 CX3H2E 44253449 IC50 = 695 nM T25315 CC1IH2 44253450 IC50 = 470 nM T25315 CZ1OH8 44253589 IC50 = 1295 nM T25315 CM5F3V 44253590 IC50 = 2560 nM T25315 C1P2EV 44253591 IC50 = 1460 nM T25315 C0CQV9 44253592 IC50 = 885 nM T25315 CZ5Y7Q 44253594 IC50 = 5580 nM T25315 C4R6FA 44253725 IC50 = 940 nM T25315 CR6AY7 44253726 IC50 = 510 nM T25315 C28BEU 44253727 IC50 = 347 nM T25315 CWO8B6 44402370 IC50 = 10000 nM T25315 CPRD27 44402504 IC50 > 100000 nM T25315 C13SIY 44402582 IC50 = 5800 nM T25315 C8QL3D 44402658 IC50 > 100000 nM T25315 CTE82I 44406196 IC50 = 200 nM T25315 C8S4YD 44406244 IC50 = 890 nM T25315 C1CND2 44406261 IC50 = 3100 nM T25315 CVHX75 44406274 IC50 = 250 nM T25315 C7M4TS 44406319 IC50 = 190 nM T25315 CEK68R 44406343 IC50 = 9800 nM T25315 CC7P8K 44406348 IC50 = 13000 nM T25315 CQDI02 44406362 IC50 = 2150 nM T25315 CYWF12 44426595 IC50 = 146 nM T25315 C8E7FG 44426596 IC50 > 10000 nM T25315 C8VG5B 44426676 IC50 = 154 nM T25315 CE25ZP 44426677 IC50 = 375 nM T25315 CJM9Y8 44426678 IC50 > 10000 nM T25315 CU1QV3 44426679 IC50 = 710 nM T25315 CG9F8V 44426680 IC50 = 790 nM T25315 C3USK7 44426681 IC50 = 587 nM T25315 CQF50T 44426682 IC50 = 1400 nM T25315 CNQK92 44426684 IC50 = 75 nM T25315 CA4WI1 44426685 IC50 > 10000 nM T25315 CQ59ES 44426687 IC50 > 10000 nM T25315 CE8KT6 44426689 IC50 > 10000 nM T25315 C10DNL 44426690 IC50 = 88 nM T25315 CU2I9R 44426691 IC50 = 156 nM T25315 CD02AO 44426693 IC50 = 300 nM T25315 CQPA38 44426694 IC50 = 40 nM T25315 CW7QO3 44426696 IC50 > 10000 nM T25315 C39YWG 44426697 IC50 = 100 nM T25315 C1IB7A 44426698 IC50 = 230 nM T25315 CC3HX1 44426700 IC50 = 650 nM T25315 CHX5L4 44426702 IC50 = 240 nM T25315 CAYN63 44426704 IC50 = 73 nM T25315 CX59SN 44426705 IC50 = 12 nM T25315 CZP36J 44426707 IC50 = 299 nM T25315 C2XM8V 44426709 IC50 = 22 nM T25315 C8MTK3 44426710 IC50 = 25 nM T25315 CS26WG 44426711 IC50 = 14 nM T25315 C3JGN9 44426712 IC50 = 4 nM T25315 CI9VE2 44426713 IC50 = 7 nM T25315 C1IVP3 44426714 IC50 = 11 nM T25315 CAN3Z0 44426715 IC50 = 10000 nM T25315 CM36CB 44426716 IC50 = 1370 nM T25315 CWG81F 44426717 IC50 = 25000 nM T25315 CF8TQ5 44426718 IC50 = 2300 nM T25315 C9PC4S 44426719 IC50 = 75 nM T25315 CP1W5K 44426720 IC50 > 10000 nM T25315 C1VS2L 44426721 IC50 = 9 nM T25315 C7CAD8 44426722 IC50 = 4000 nM T25315 C2PW9U 44426723 IC50 = 6 nM T25315 CMD9W8 44426724 IC50 = 144 nM T25315 CQN23M 44426725 IC50 = 1400 nM T25315 C3YVD8 44426726 IC50 = 480 nM T25315 CZ1HM8 44426909 Ki = 88 nM T25315 CX6JZ7 44426911 Ki = 201 nM T25315 CCR8I3 44426912 Ki = 104 nM T25315 C1YA3J 44426913 Ki = 637 nM T25315 CF5T6J 44426914 Ki = 36 nM T25315 CYG30D 44426915 Ki = 47 nM T25315 C7B5KO 44426917 Ki = 41 nM T25315 CY0QL7 44426920 Ki = 306 nM T25315 CSQ39F 44426931 Ki = 1040 nM T25315 C92KYE 44426932 Ki = 3400 nM T25315 C8HXV6 44426934 Ki = 660 nM T25315 C6EPQ5 44426935 Ki = 108 nM T25315 C10HDQ 44426990 Ki = 290 nM T25315 C9NPB6 44426992 Ki = 1300 nM T25315 C56CNU 44426993 Ki = 2200 nM T25315 C9HBE6 44426994 Ki = 2000 nM T25315 C7G6VX 44426995 Ki = 26 nM T25315 C5TCJ4 44426996 Ki = 258 nM T25315 CJ52DF 44426998 Ki = 171 nM T25315 C62OEC 44426999 Ki = 429 nM T25315 C8FME2 44427000 Ki = 31 nM T25315 CZG57H 44427001 Ki = 175 nM T25315 CH41ZJ 44427002 Ki = 191 nM T25315 C6PA3B 44427003 Ki = 39 nM T25315 CWLV83 44427004 Ki = 29 nM T25315 C8QVY7 44427005 Ki = 46 nM T25315 CPGI84 44427006 Ki = 171 nM T25315 C2NPL3 44427007 Ki = 70 nM T25315 CE4U2C 44427008 Ki = 107 nM T25315 CB57WJ 44427009 Ki = 141 nM T25315 C1DQ9J 44427010 Ki = 83 nM T25315 CXE68Z 44427011 Ki = 191 nM T25315 CKCI49 44427013 Ki = 229 nM T25315 CQM6I9 44427014 Ki = 16 nM T25315 CG58XD 44427015 Ki = 81 nM T25315 C26PAQ 44427016 Ki = 376 nM T25315 CRK03J 44427019 Ki = 28 nM T25315 COI4D1 44443757 Ki = 180 nM T25315 CJ2X4L 44443759 Ki = 3600 nM T25315 CY1CM8 44443799 Ki = 3500 nM T25315 CT3AG0 44443812 Ki = 170 nM T25315 C06FOM 44443813 Ki = 200 nM T25315 CCI0V1 44443814 Ki = 680 nM T25315 CC0BL6 44443816 Ki = 720 nM T25315 CDG70K 44443818 Ki = 350 nM T25315 CUKG03 44443820 Ki = 126 nM T25315 C7N8FP 44443821 Ki = 950 nM T25315 C8M6OE 44443822 Ki = 460 nM T25315 CC5BH3 44443823 Ki = 290 nM T25315 CG06SI 44443825 Ki = 170 nM T25315 C7QU8A 44443827 Ki = 620 nM T25315 CR16SG 44443828 Ki = 150 nM T25315 CF58ZA 44443830 Ki = 130 nM T25315 C5GN2J 44443831 Ki = 880 nM T25315 CFR4S3 44443833 Ki = 460 nM T25315 CMZ3F8 44443834 Ki = 260 nM T25315 C8VTC4 44443835 Ki = 270 nM T25315 CXFA79 44446421 Ki = 1100 nM T25315 CKEW28 44446422 Ki = 180 nM T25315 C19WRK 44446423 Ki = 60 nM T25315 C6PR0N 44446438 Ki = 190 nM T25315 C41QLD 44446439 Ki = 27 nM T25315 CPH8N9 44446441 Ki = 28 nM T25315 C2JBE3 44446443 Ki = 20 nM T25315 C0HWP6 44446445 Ki = 18 nM T25315 C8C4IX 44446450 Ki = 9 nM T25315 CK6DR1 44446451 Ki = 10 nM T25315 CRG6O5 44446452 Ki = 280 nM T25315 C5CZ1N 44446453 Ki = 11 nM T25315 CTPF78 44446454 Ki = 3 nM T25315 CV4Q3Z 44446457 Ki = 120 nM T25315 CT27ON 44447090 IC50 = 21 nM T25315 CMS98X 44447091 IC50 = 27 nM T25315 CU5TN2 44447092 IC50 = 9 nM T25315 CCV03Y 44447093 IC50 = 5 nM T25315 CCZ7G4 44447094 IC50 = 4 nM T25315 CZ41CV 44447095 IC50 = 35 nM T25315 C45PYZ 44447096 Ki = 3 nM T25315 CV13QK 44447097 IC50 = 10 nM T25315 CY9ZH4 44447098 IC50 = 523 nM T25315 C2CM7R 44453168 IC50 = 15 nM T25315 CHC2Z8 44453201 IC50 = 400 nM T25315 CJ9MS5 44453232 IC50 = 100 nM T25315 CP2K3T 44453266 IC50 = 400 nM T25315 C67XKC 44453267 IC50 = 300 nM T25315 C74BMH 44453295 IC50 = 2300 nM T25315 C6OT8Y 44453296 IC50 = 800 nM T25315 CURJ65 44453322 IC50 = 500 nM T25315 CHP8R7 44453362 IC50 = 3400 nM T25315 CI8KQ3 44453364 IC50 = 200 nM T25315 CFNV87 44453439 IC50 = 1200 nM T25315 CP59RA 44453468 IC50 = 20 nM T25315 C4G1XC 44453470 IC50 = 20 nM T25315 C7VRC2 44453530 IC50 = 16 nM T25315 CCN36G 44453558 IC50 = 15 nM T25315 C3HLJ5 44453583 IC50 = 15 nM T25315 CW6M5E 44453585 IC50 = 20 nM T25315 CGC18I 44453616 IC50 = 20 nM T25315 CX24TY 44453640 IC50 = 20 nM T25315 C43LJW 44453643 IC50 = 20 nM T25315 CVAR89 44454490 IC50 = 11000 nM T25315 CD39AJ 44454491 IC50 = 22000 nM T25315 C68PRZ 44454492 IC50 = 3000 nM T25315 CQ15UF 44454527 IC50 = 16000 nM T25315 CR02BQ 44454588 IC50 = 20000 nM T25315 CLV09T 44454589 IC50 = 50000 nM T25315 CW28RB 44454591 IC50 = 11000 nM T25315 CR36OC 44454616 IC50 > 50000 nM T25315 CR7S1T 44454617 IC50 > 50000 nM T25315 CL6X9V 44454618 IC50 > 50000 nM T25315 CI06HS 44454619 IC50 > 50000 nM T25315 C8MYB0 44454644 IC50 = 3000 nM T25315 CD7HP9 44454645 IC50 > 100000 nM T25315 CS2RV7 44454796 IC50 = 700 nM T25315 CF0HE2 44454824 IC50 = 400 nM T25315 CRZ0S7 44454826 IC50 = 300 nM T25315 C9AM2E 44454895 IC50 = 5000 nM T25315 CTDO37 44454934 IC50 = 6000 nM T25315 CHMX10 44455463 IC50 = 10 nM T25315 CS07AT 44455464 IC50 = 8 nM T25315 C4B8RZ 44455480 Ki = 6 nM T25315 CDP34N 44455488 IC50 = 3.8 nM T25315 CAMQ81 44455489 IC50 = 3.2 nM T25315 CN63DX 44455507 Ki = 5 nM T25315 C0WGY8 44455508 Ki = 4 nM T25315 CLO97I 44455517 IC50 = 2.5 nM T25315 CQ2U0J 44455536 Ki = 3 nM T25315 C63XVT 44455537 Ki = 6 nM T25315 C9SHN8 44455538 Ki = 24 nM T25315 CQO4A5 44455542 IC50 = 2.6 nM T25315 C4AUD2 44455558 Ki = 25 nM T25315 CJL93M 44455559 Ki = 20 nM T25315 CGN9O2 44455561 Ki = 7 nM T25315 CO9M7F 44455565 IC50 = 6.6 nM T25315 C3LA2F 44455568 IC50 = 29 nM T25315 C7LH6V 44455569 IC50 = 43 nM T25315 C8FNQ3 44455591 Ki = 18 nM T25315 C6L5HC 44455592 Ki = 21 nM T25315 C85IXV 44455593 Ki = 26 nM T25315 CD9JS4 44455603 IC50 = 40 nM T25315 C4RM3X 44455604 IC50 = 0.7 nM T25315 C3Z8RN 44455621 Ki = 624 nM T25315 C1JY6K 44455623 Ki = 15 nM T25315 C0AT4Q 44455624 Ki = 143 nM T25315 C7AF4M 44455634 IC50 = 44 nM T25315 CK9CF3 44455640 IC50 = 2.1 nM T25315 CD7R2O 44455656 Ki = 95 nM T25315 CGA1N7 44455657 Ki = 135 nM T25315 CK3P0E 44455668 IC50 = 9.4 nM T25315 CF1MA0 44455669 IC50 = 5 nM T25315 CYK1C0 44455693 IC50 = 5.6 nM T25315 C8SJ1R 44455722 IC50 = 7.1 nM T25315 CT5LU2 44455723 IC50 = 4.8 nM T25315 CM83TF 44455751 IC50 = 0.4 nM T25315 C6YB5X 44455752 IC50 = 2.4 nM T25315 C3ER7Q 44455773 IC50 = 6.4 nM T25315 CJ85LG 44455774 IC50 = 11 nM T25315 C07RWG 44455799 IC50 = 36 nM T25315 CD7A6G 44455800 IC50 = 11 nM T25315 CE8IV9 44455801 IC50 = 81 nM T25315 CR0PD3 44455823 IC50 = 129 nM T25315 CTKJ17 44455824 IC50 = 1179 nM T25315 C4U8KC 44455825 IC50 = 752 nM T25315 CVMQ03 44455843 IC50 = 1.8 nM T25315 CY5X1B 44455852 IC50 = 72 nM T25315 CC73TZ 44455870 IC50 = 3 nM T25315 CE0J4D 44455873 IC50 = 19 nM T25315 C67ECQ 44569941 IC50 = 1584.89 nM T25315 C50RXU 44569942 IC50 = 158.49 nM T25315 CIF8H1 44569943 IC50 = 794.33 nM T25315 C7O6MC 44569944 IC50 = 199.53 nM T25315 CA9FG7 44570029 IC50 = 199.53 nM T25315 CPG92E 44570140 IC50 = 794.33 nM T25315 C9JL0W 44570141 IC50 = 1995.26 nM T25315 CPY61G 44570142 IC50 = 630.96 nM T25315 CFI5O3 44570178 IC50 = 794.33 nM T25315 CB52AH 44570179 IC50 = 7943.28 nM T25315 CWLT20 44570180 IC50 = 79.43 nM T25315 C8MJK1 44570181 IC50 = 501.19 nM T25315 CGCZ05 44570218 IC50 = 316.23 nM T25315 C5Y0GJ 44570219 IC50 = 158.49 nM T25315 C9NED2 44570220 IC50 = 31.62 nM T25315 CA6W4U 44570221 IC50 = 316.23 nM T25315 CZJ2Y0 44570272 IC50 = 50.12 nM T25315 C6P5BJ 44570273 IC50 = 63.1 nM T25315 C12LRN 44570274 IC50 = 39.81 nM T25315 C1JI8N 44570310 IC50 > 31622.78 nM T25315 CH41VM 44570311 IC50 = 25118.86 nM T25315 C6JL8T 44570312 IC50 = 125.89 nM T25315 CE3D5K 44570340 IC50 = 25118.86 nM T25315 CG3L8N 44570341 IC50 = 1584.89 nM T25315 C3R9CO 44570342 IC50 > 31622.78 nM T25315 CV1K2L 44570343 IC50 > 31622.78 nM T25315 CKMS98 44570344 IC50 > 31622.78 nM T25315 CK2I7F 44570383 IC50 > 31622.78 nM T25315 CJ1Y4O 44570384 IC50 > 31622.78 nM T25315 C06TEU 44570385 IC50 = 158.49 nM T25315 CGI97J 44570430 IC50 = 398.11 nM T25315 CT59OX 44570431 IC50 = 251.19 nM T25315 C7Q4LA 44570432 IC50 = 316.23 nM T25315 CQL02F 44570433 IC50 > 31622.78 nM T25315 CA1JV3 44570470 IC50 = 1995.26 nM T25315 CSZN78 44570471 IC50 = 316.23 nM T25315 CXC47F 44570472 IC50 = 630.96 nM T25315 C2SBW1 44570473 IC50 = 5011.87 nM T25315 CSZ10Q 44570515 IC50 = 15848.93 nM T25315 CK7MT9 44570516 IC50 = 316.23 nM T25315 C9YJ5C 44570517 IC50 = 630.96 nM T25315 C6EM9O 44570547 IC50 = 6309.57 nM T25315 CT92VI 44570548 IC50 > 31622.78 nM T25315 CSA37U 44570549 IC50 = 158.49 nM T25315 CBK73R 44570550 IC50 = 501.19 nM T25315 CXH83L 44570595 IC50 = 398.11 nM T25315 CQ47MB 44570596 IC50 = 630.96 nM T25315 CGH57K 44570597 IC50 > 31622.78 nM T25315 C3WNP8 44570598 IC50 > 31622.78 nM T25315 CHEF64 44570627 IC50 = 6309.57 nM T25315 CZY82W 44570628 IC50 = 31622.78 nM T25315 CD81NC 44570629 IC50 = 15848.93 nM T25315 CR1EN7 44570630 IC50 > 31622.78 nM T25315 CFMI18 44580796 IC50 = 790 nM T25315 CW7C5I 44580797 IC50 = 1260 nM T25315 C80DQT 44580798 IC50 = 320 nM T25315 C0KC9I 44580799 IC50 = 1000 nM T25315 CH2NB1 44580823 IC50 = 2510 nM T25315 CFRD71 44580857 IC50 = 2510 nM T25315 CW8DX0 44580858 IC50 = 5010 nM T25315 CA7T9E 44580859 IC50 = 5010 nM T25315 CQ64PE 44580860 IC50 = 2000 nM T25315 CEI7X4 44580878 IC50 = 1000 nM T25315 C6VZX1 44580902 IC50 = 690 nM T25315 CAD63V 44580903 IC50 = 180 nM T25315 CTS8M1 44580939 IC50 = 500 nM T25315 C7ZI2N 44580959 IC50 > 10000 nM T25315 C7JDB3 44580960 IC50 = 1580 nM T25315 CM5FR3 44581069 IC50 = 4270 nM T25315 CX6ZC8 44581070 IC50 = 3160 nM T25315 C27TFX 44581087 IC50 = 1260 nM T25315 CM08HC 44581088 IC50 = 2510 nM T25315 CBDG70 44581089 IC50 = 500 nM T25315 CSGK97 44581090 IC50 = 1000 nM T25315 CJP27F 44581108 IC50 = 630 nM T25315 C0PRS3 44581109 IC50 = 1260 nM T25315 CF13RW 44581110 IC50 = 3630 nM T25315 CS92ZI 44581134 IC50 = 1550 nM T25315 C2YCI0 44581135 IC50 = 170 nM T25315 COXU45 44581136 IC50 = 1450 nM T25315 C3S7LY 44581137 IC50 = 5010 nM T25315 CO7CH6 44581159 IC50 = 630 nM T25315 CR04AU 44581160 IC50 = 3160 nM T25315 CTQG38 44581161 IC50 = 3160 nM T25315 C52KSR 44581162 IC50 = 1260 nM T25315 CK68GB 44591872 Ki = 501.19 nM T25315 CH83XO 44591873 Ki = 501.19 nM T25315 C3BZ1U 44591874 Ki = 6309.57 nM T25315 CQ68TX 44591875 Ki > 10000 nM T25315 CM3CL2 44591885 Ki = 6309.57 nM T25315 CWBE05 44591886 Ki = 3981.07 nM T25315 CFI43D 44591887 Ki = 1584.89 nM T25315 CJ4CW7 44591918 Ki = 794.33 nM T25315 CYLA46 44591928 Ki = 1258.93 nM T25315 C63BCT 44592137 IC50 = 0.3 nM T25315 C8ZGH3 44592138 Ki > 100000 nM T25315 CSX5I3 44592139 Ki = 5011.87 nM T25315 CHEZ19 44592140 Ki > 10000 nM T25315 C0P3TB 44592174 Ki = 2511.89 nM T25315 C8I0QU 44592175 Ki = 5011.87 nM T25315 CL43NG 44592176 Ki = 3981.07 nM T25315 C0V1OK 44592177 Ki = 3981.07 nM T25315 CNQY29 44592178 Ki > 10000 nM T25315 CXB0Y1 44592220 Ki = 398.11 nM T25315 C6ET4R 44592221 Ki = 1000 nM T25315 CM5P7L 44592222 Ki = 1000 nM T25315 C5A1PQ 44592264 Ki = 501.19 nM T25315 CS7H3P 44592265 Ki = 1258.93 nM T25315 C3RS7M 44592266 Ki = 2511.89 nM T25315 CTXG85 44592267 Ki = 501.19 nM T25315 C0YIB3 44592268 Ki = 7943.28 nM T25315 CY8V9H 44592304 Ki = 5011.87 nM T25315 CNS17G 44592305 Ki = 3981.07 nM T25315 C0CKI4 44592306 Ki = 5011.87 nM T25315 CG5FQ2 44592341 Ki = 3981.07 nM T25315 CYS8Z3 44592342 Ki = 1995.26 nM T25315 C8P4HM 44592343 Ki = 1584.89 nM T25315 C80SLH 44592344 Ki > 10000 nM T25315 CUYP04 44592403 Ki = 3162.28 nM T25315 CI6CP5 44592404 Ki = 794.33 nM T25315 CXM01D 44592405 Ki = 10000 nM T25315 C1TO8P 44592406 Ki = 7943.28 nM T25315 CL9F5P 44592407 Ki = 1995.26 nM T25315 C1G6UJ 44592471 Ki = 1584.89 nM T25315 CGH7F5 44592472 Ki = 1995.26 nM T25315 C1OBI0 44592473 Ki = 398.11 nM T25315 CV0NE9 44592474 Ki = 2511.89 nM T25315 CO9U6M 44592475 Ki = 7943.28 nM T25315 CNCT24 44592527 Ki > 10000 nM T25315 CV4ZX1 44592528 Ki = 6309.57 nM T25315 C0T6OI 44592529 Ki = 2511.89 nM T25315 CT0B1I 44592530 Ki = 3981.07 nM T25315 CIR39K 44592531 Ki = 1995.26 nM T25315 CNZ1U7 44593651 IC50 = 60 nM T25315 C7DK9G 44593733 Ki = 398.11 nM T25315 C5JGD4 44593735 Ki = 3981.07 nM T25315 CSHE04 45101497 IC50 = 16 nM T25315 C3P5FJ 45101498 IC50 = 32 nM T25315 CM6C9Q 45101529 IC50 = 0.4 nM T25315 C9HZ2R 45379650 IC50 = 0.9 nM T25315 C8A1FM 45482784 IC50 = 179 nM T25315 C0CHF4 45482789 IC50 = 18 nM T25315 CG09IA 45482794 IC50 > 10000 nM T25315 CA7MT2 45482795 IC50 = 231 nM T25315 CU07RG 45482796 IC50 = 803 nM T25315 CS7H4A 45482800 IC50 = 2000 nM T25315 CTO70Z 45482803 IC50 > 10000 nM T25315 CK0NU7 45482807 IC50 = 100 nM T25315 C07UTP 45482808 IC50 = 564 nM T25315 CNK31C 45482813 IC50 > 10000 nM T25315 CEP68M 45482814 IC50 = 1930 nM T25315 C82CZS 45482819 IC50 = 62 nM T25315 C92SGJ 45482823 IC50 = 67 nM T25315 CUH5N1 45482836 IC50 = 60 nM T25315 CCN71E 45482843 IC50 = 510 nM T25315 CVT85J 45482849 IC50 = 28 nM T25315 C1E7BH 45484653 Ki = 870 nM T25315 C6GUW2 45484655 Ki = 1900 nM T25315 CZ19CS 45484656 IC50 = 560 nM T25315 CCV7W8 45484657 Ki = 3700 nM T25315 C95ONL 45484658 Ki = 90 nM T25315 C1EZ5R 45484671 Ki = 370 nM T25315 CX1Q9P 45484678 Ki = 4100 nM T25315 CPR4Y6 45484679 Ki = 470 nM T25315 CEK34W 45484680 Ki = 3800 nM T25315 CTX6G2 45484691 Ki = 510 nM T25315 C2WA8F 45484692 Ki = 330 nM T25315 CNEQ82 45484705 Ki = 410 nM T25315 CT1NL4 45484716 Ki = 8900 nM T25315 CXB16P 45484733 Ki = 1900 nM T25315 CR6Y2Q 45484739 IC50 = 20 nM T25315 CBMG60 45484740 Ki > 50000 nM T25315 CZ4YW9 45484748 Ki = 120 nM T25315 CA95WT 45484749 Ki = 2900 nM T25315 CBH0R2 45485420 IC50 = 4500 nM T25315 CRFG06 45485423 Ki = 7200 nM T25315 C27GJB 45485429 Ki = 86 nM T25315 CER5O9 45485434 Ki = 16 nM T25315 CB6C0G 45485437 Ki = 32 nM T25315 CO45AX 45485438 Ki = 2000 nM T25315 CH4LC2 45485451 Ki = 2700 nM T25315 CHUM15 45485458 Ki = 23000 nM T25315 CUON70 45486493 IC50 = 2 nM T25315 CGN04B 45486520 IC50 = 60 nM T25315 CCPR31 45486521 IC50 = 3 nM T25315 CM1GD4 45486522 IC50 = 18 nM T25315 CAN49B 45486523 IC50 = 0.9 nM T25315 C5CG6H 45486524 IC50 = 1.6 nM T25315 CVB49D 45486525 IC50 = 1.1 nM T25315 CL49VY 45486526 IC50 = 0.9 nM T25315 CSW98R 45486528 IC50 = 1.4 nM T25315 CSB01J 45486529 IC50 = 44 nM T25315 CEHV82 45486530 IC50 = 1.1 nM T25315 CX8JN5 45486531 IC50 = 21 nM T25315 C6DVW7 45486532 IC50 = 29 nM T25315 C1YZT7 45486533 IC50 = 1.3 nM T25315 C9SDX2 45486534 IC50 = 1.1 nM T25315 CVD09X 45486555 IC50 = 4 nM T25315 C0B1JF 45486556 IC50 = 4 nM T25315 C4A5KL 45486557 IC50 = 457 nM T25315 C9UZS8 45486558 IC50 > 1000 nM T25315 C93HDC 45486559 IC50 = 29 nM T25315 C69LTY 45486560 IC50 = 10 nM T25315 CT3V4F 45486561 IC50 = 3 nM T25315 CK8QW4 46225413 IC50 > 60000 nM T25315 C92GWM 46700871 IC50 = 192 nM T25315 CP57KH 46883287 IC50 = 690 nM T25315 C5UM7W 46883288 IC50 = 210 nM T25315 CLS3E6 46883289 IC50 = 7 nM T25315 CB2M8T 46883290 IC50 = 13 nM T25315 C9IL1T 46883291 IC50 = 2090 nM T25315 CKWP14 46883292 IC50 = 11 nM T25315 CRK72O 46883293 IC50 = 21 nM T25315 CRX7I9 46883294 IC50 = 770 nM T25315 CA2L3W 46883295 IC50 = 40 nM T25315 CT56QR 46883296 IC50 = 8 nM T25315 CT1XY7 46883297 IC50 = 7 nM T25315 C0P2ZK 46883298 IC50 = 9 nM T25315 C3JU1T 46883299 IC50 = 2 nM T25315 CYF17Z 46883300 IC50 = 23 nM T25315 CBJI21 46883301 IC50 = 110 nM T25315 CF29SM 46883302 IC50 = 42 nM T25315 C12RTY 46883303 IC50 = 2 nM T25315 CNU64B 46883304 IC50 = 10 nM T25315 CPH4U2 46883305 IC50 = 5 nM T25315 C6Y5AE 46883306 IC50 = 2 nM T25315 CBAR75 46883307 IC50 = 2 nM T25315 C61ADL 46883308 IC50 = 1 nM T25315 C8WH2O 46883309 IC50 = 131 nM T25315 C32OKX 46883310 IC50 = 5 nM T25315 C1U2JO 46883311 IC50 = 1 nM T25315 CF1WQ6 46890724 IC50 = 183 nM T25315 CNBY78 46890725 IC50 = 339 nM T25315 C7PRW5 46890726 IC50 = 216 nM T25315 CC80EV 46890727 IC50 = 207 nM T25315 CL9RS8 46891078 IC50 = 192 nM T25315 C8HMI6 46891145 IC50 = 238 nM T25315 C05ZXW 46891183 IC50 = 85 nM T25315 CG4IZ3 46891223 IC50 = 1152 nM T25315 C0RJ7G 46891224 IC50 = 360 nM T25315 C49ELR 46891272 IC50 = 13 nM T25315 C17TKX 46891273 IC50 = 6440 nM T25315 CZ6KG3 46891327 IC50 = 1132 nM T25315 CHXZ61 46891328 IC50 = 513 nM T25315 CYL9S8 46891329 IC50 = 1080 nM T25315 C5WA4D 46891371 IC50 = 882 nM T25315 C70PAG 46891424 IC50 = 233 nM T25315 C8X6IK 46891425 IC50 = 540 nM T25315 CPU40W 46891476 IC50 = 911 nM T25315 C4LNX0 46891477 IC50 = 254 nM T25315 CE7R5I 46891478 IC50 = 440 nM T25315 CM6JR5 46891536 IC50 = 158 nM T25315 COJS83 46891537 IC50 = 157 nM T25315 C2W6HF 46891538 IC50 = 236 nM T25315 C5VHE3 46893277 Ki = 199.53 nM T25315 CQAT71 53317216 IC50 = 8100 nM T25315 CIH6U1 53317274 IC50 = 31 nM T25315 CQ8RT1 53317275 IC50 = 520 nM T25315 C4M8QS 53317276 IC50 = 2.4 nM T25315 C84QKU 53317277 IC50 = 22 nM T25315 CNA91W 53317663 IC50 = 83 nM T25315 CBX25C 53318510 IC50 = 17 nM T25315 CG5R8E 53318511 IC50 > 10000 nM T25315 C0LNA3 53318512 IC50 = 1980 nM T25315 CSN30W 53318513 IC50 = 58 nM T25315 C06OAZ 53318514 IC50 = 210 nM T25315 CDCA26 53318560 IC50 = 6 nM T25315 CYS7N6 53318561 IC50 = 7000 nM T25315 CUM62K 53318562 IC50 = 280 nM T25315 CCF2J7 53318563 IC50 = 8900 nM T25315 C1M5SJ 53318914 IC50 = 830 nM T25315 CV3AR4 53319879 IC50 = 39 nM T25315 CT7KC2 53319880 IC50 = 64 nM T25315 CYP2B1 53319881 IC50 = 20 nM T25315 C68LPB 53319882 IC50 = 32 nM T25315 C6M5QK 53321134 IC50 > 10000 nM T25315 C0OG1S 53321184 IC50 = 39 nM T25315 CO0VP5 53321185 IC50 = 5 nM T25315 C3W9GC 53321186 IC50 = 3100 nM T25315 C5AZ9K 53321187 IC50 = 23 nM T25315 CRAG94 53322459 IC50 = 5 nM T25315 C4F2WR 53322460 IC50 = 63 nM T25315 C17FLG 53322461 IC50 = 8060 nM T25315 CXL54M 53322503 IC50 > 10000 nM T25315 CS37NB 53322504 IC50 = 40 nM T25315 C64WRQ 53322505 IC50 = 2700 nM T25315 CZSY87 53322506 IC50 = 27 nM T25315 C04FJG 53322507 IC50 = 7350 nM T25315 C3VGE4 53322508 IC50 = 8 nM T25315 CHJ16M 53322509 IC50 = 2.3 nM T25315 C13HWL 53322510 IC50 = 900 nM T25315 CPY5A1 53322511 IC50 = 630 nM T25315 CGK9M0 53322974 IC50 = 7990 nM T25315 C7EG5Q 53323853 IC50 = 140 nM T25315 CY2QU7 53323854 IC50 = 910 nM T25315 CF85ZO 53324231 IC50 = 3 nM T25315 C7TL6S 53324328 IC50 > 50000 nM T25315 CZ7B8C 53325131 IC50 = 1400 nM T25315 CYFL35 53325132 IC50 = 12500 nM T25315 CB0ZI6 53325133 IC50 = 80 nM T25315 CST63J 53325134 IC50 = 260 nM T25315 CI90MS 53326388 IC50 = 18 nM T25315 CXFS62 53326389 IC50 = 87 nM T25315 CIWZ65 53326434 IC50 = 220 nM T25315 CI2F1D 53326850 IC50 = 29 nM T25315 CVP7O2 54764847 IC50 = 1.3 nM T25315 C2TF8D 56660098 IC50 = 305 nM T25315 C4IB1X 56660099 IC50 = 12 nM T25315 CXJ5Q0 56660100 IC50 = 81 nM T25315 C3Y4MP 56660101 IC50 = 16 nM T25315 CK7CU3 56660102 IC50 = 5 nM T25315 CXGA53 56663557 IC50 = 17 nM T25315 CE6OU8 56663558 IC50 = 67 nM T25315 CA1MK4 56663559 IC50 = 22 nM T25315 CNM6R8 56663560 IC50 = 3 nM T25315 C9Y7XJ 56663561 IC50 = 53 nM T25315 CGZ58A 56663562 IC50 = 5 nM T25315 C3TF1C 56663563 IC50 = 8 nM T25315 C4EH6A 56667005 IC50 = 457 nM T25315 C7WH3Y 56667006 IC50 = 200 nM T25315 C90ZSJ 56667007 IC50 = 20 nM T25315 C7ZS8I 56667008 IC50 > 10000 nM T25315 C6TX1V 56667009 IC50 = 14 nM T25315 CE5B0W 56670448 IC50 = 14 nM T25315 CZI80K 56670449 IC50 = 12 nM T25315 CHPD72 56670450 IC50 = 523 nM T25315 CRX87E 56670451 IC50 = 27 nM T25315 C6KFM1 56670452 IC50 = 6200 nM T25315 CINM64 56670453 IC50 > 10000 nM T25315 C6NP4T 56670454 IC50 = 2200 nM T25315 CM9QG4 56670455 IC50 = 2600 nM T25315 CU1I9Y 56670456 IC50 = 170 nM T25315 C04IPB 56670465 IC50 = 28 nM T25315 C53OLI 56673431 IC50 = 4 nM T25315 CG7AL2 56673937 IC50 = 9 nM T25315 CSD20W 56673938 IC50 = 83 nM T25315 C68OUR 56673939 IC50 = 216 nM T25315 C13WYF 56673940 IC50 = 7 nM T25315 C7R3CU 56673941 IC50 = 160 nM T25315 C4TA3N 56673942 IC50 = 11 nM T25315 CCZ98M 56673943 IC50 = 9475 nM T25315 CW4J1Y 56673944 IC50 = 2 nM T25315 CKW4Z0 56673945 IC50 = 3 nM T25315 CB0MR9 56673953 IC50 > 10000 nM T25315 CH7NA4 56677270 IC50 = 825 nM T25315 CN58TZ 56677271 IC50 = 4 nM T25315 CDC12H 56677272 IC50 = 89 nM T25315 C4SB5Y 56677273 IC50 = 8 nM T25315 CLW35V 56677274 IC50 = 6120 nM T25315 CYA6W7 56680570 IC50 = 12 nM T25315 CNE8Q0 56680571 IC50 = 74 nM T25315 CM4H9X 56680572 IC50 = 5400 nM T25315 CJ2B3H 56680573 IC50 > 10000 nM T25315 CFU4D9 56680574 IC50 = 5 nM T25315 CWV06G 56680588 IC50 = 379 nM T25315 C7V9WR 56683907 IC50 > 10000 nM T25315 CPN57V 56834986 IC50 = 12 nM T25315 C9B3IZ 57390182 IC50 = 29 nM T25315 C0G9RK 57390209 IC50 = 7 nM T25315 C5NRS1 57390764 IC50 = 2.5 nM T25315 CB5GH2 57390765 IC50 = 0.9 nM T25315 CJ9E8I 57392573 IC50 = 3.7 nM T25315 C2W4QX 57392574 IC50 = 0.9 nM T25315 CVY53H 57392575 IC50 = 2.9 nM T25315 C71AYV 57392576 IC50 > 1000 nM T25315 CXP8A9 57393685 IC50 = 21 nM T25315 C2ZXG7 57394143 IC50 = 8 nM T25315 CA4L9P 57394299 IC50 = 1.5 nM T25315 CFCI01 57394300 IC50 = 1.8 nM T25315 CJ06XR 57394301 IC50 = 1.1 nM T25315 C0CU3Q 57396053 IC50 = 8.4 nM T25315 CZ47JD 57396054 IC50 = 4.4 nM T25315 CIE8P1 57396055 IC50 = 1.9 nM T25315 CIU06Z 57397852 IC50 = 8.5 nM T25315 C4L2BA 57397853 IC50 = 6.4 nM T25315 C80THO 57397854 IC50 = 3.4 nM T25315 CV1T4M 57397855 IC50 = 1.5 nM T25315 C0SMP4 57397856 IC50 = 1.9 nM T25315 C3WMN4 57399515 IC50 = 4 nM T25315 C15KWV 57399516 IC50 = 2.4 nM T25315 C6FIN0 57399517 IC50 = 2 nM T25315 CXNA63 57399518 IC50 = 235 nM T25315 C6WJU5 57400628 IC50 = 47 nM T25315 CRL27H 57400629 IC50 = 6 nM T25315 CB7UI1 57400677 IC50 = 50 nM T25315 CJ6T7Z 57401268 IC50 = 4.1 nM T25315 CVJ60W 57401269 IC50 = 1.2 nM T25315 C1TQ0D 57401270 IC50 = 3.6 nM T25315 CT7HP6 57402420 IC50 = 7 nM T25315 CF74AH 57402421 IC50 = 6 nM T25315 C4Y6LX 57403018 IC50 = 76 nM T25315 C2MOF3 57403019 IC50 = 2.9 nM T25315 CMCR69 57403020 IC50 = 4.2 nM T25315 CFD1H9 58186816 IC50 = 23.6 nM T25315 C0YWT1 58509213 IC50 > 10000 nM T25315 CW9QE3 58767992 IC50 = 33.8 nM T25315 CO9A1X 58768002 IC50 = 24.5 nM T25315 CV4WM6 58768027 IC50 = 1.8 nM T25315 C5AS8M 58768044 IC50 = 3.8 nM T25315 CZ35PK 58768048 IC50 = 1.2 nM T25315 CP8LT7 58768061 IC50 = 1.6 nM T25315 CN8MZ0 58768069 IC50 = 6.2 nM T25315 C2UDL3 59772540 IC50 = 286 nM T25315 CZS67E 59772541 IC50 = 0.3 nM T25315 C7R1OE 59772590 IC50 = 1376 nM T25315 C9TZ1U 68102990 IC50 = 50.5 nM T25315 CF3IV1 71450265 Ki = 50.12 nM T25315 C7H1TE 71450267 Ki = 2511.89 nM T25315 C8JQ5C 71450269 Ki = 158.49 nM T25315 CB6NI2 71450271 Ki = 1000 nM T25315 CN9E6V 71450472 Ki = 251.19 nM T25315 C2MDO0 71450474 Ki = 501.19 nM T25315 C08PIB 71450476 Ki > 316.23 nM T25315 CV94LS 71450477 Ki > 316.23 nM T25315 CYKW92 71450478 Ki > 316.23 nM T25315 C3QDS2 71450479 Ki > 316.23 nM T25315 CMS83A 71450527 Ki > 316.23 nM T25315 CQU7C0 71450528 Ki = 1584.89 nM T25315 CZD30U 71450530 Ki = 1000 nM T25315 C9SEQ1 71450532 Ki = 630.96 nM T25315 CKE64U 71450534 Ki = 630.96 nM T25315 C76YQS 71450536 Ki = 15848.93 nM T25315 CU6F5I 71450537 Ki = 2511.89 nM T25315 C64OBF 71450539 Ki = 3981.07 nM T25315 C20ATU 71450540 Ki = 794.33 nM T25315 CS8D3F 71452091 Ki = 501.19 nM T25315 CZ2LN6 71452093 Ki = 100 nM T25315 C7ASV4 71452310 Ki = 199.53 nM T25315 CF3Z1I 71452312 Ki = 316.23 nM T25315 CWOG46 71452314 Ki = 3981.07 nM T25315 CQ2MD5 71452315 Ki = 1000 nM T25315 CQ3IJ8 71452374 Ki = 3162.28 nM T25315 CC1JU7 71452375 Ki = 1995.26 nM T25315 C4Y5XB 71452377 Ki = 398.11 nM T25315 CFNK04 71452379 Ki = 7943.28 nM T25315 C07AYL 71452380 Ki = 3162.28 nM T25315 C5N6XV 71452381 Ki = 7943.28 nM T25315 CIS53Z 71453923 Ki = 398.11 nM T25315 C4Q3FX 71453925 Ki = 398.11 nM T25315 CBV1L9 71454100 Ki = 199.53 nM T25315 C25LRG 71454102 Ki = 1584.89 nM T25315 C8DQT6 71454104 Ki = 3162.28 nM T25315 C8H6RA 71454154 Ki > 316.23 nM T25315 C2LM8W 71454155 Ki = 2511.89 nM T25315 CCSO26 71454157 Ki = 7943.28 nM T25315 CYM0Z5 71455652 Ki = 158.49 nM T25315 CGLO60 71455654 Ki = 501.19 nM T25315 C5ZY7U 71455656 Ki = 100 nM T25315 CIC9O6 71455658 Ki = 398.11 nM T25315 CY93MX 71455837 Ki = 501.19 nM T25315 CHN98F 71455839 Ki = 3162.28 nM T25315 CV6B5G 71455841 Ki = 2511.89 nM T25315 CBQ85T 71455884 Ki = 1995.26 nM T25315 C3JD5K 71455885 Ki = 251.19 nM T25315 CPL57Q 71455887 Ki = 5011.87 nM T25315 CQK5Y0 71455888 Ki = 12589.25 nM T25315 C4UZH2 71455889 Ki = 3162.28 nM T25315 CNG1V3 71457435 Ki = 199.53 nM T25315 CAG4P3 71457437 Ki = 501.19 nM T25315 CHCE02 71457439 Ki = 39.81 nM T25315 CX58ZE 71457631 Ki = 398.11 nM T25315 CN36SQ 71457633 Ki = 1258.93 nM T25315 C13TZU 71457635 Ki = 6309.57 nM T25315 CP4WI9 71457636 Ki = 6309.57 nM T25315 CKJ27M 71457637 Ki > 316.23 nM T25315 C9GQO8 71457681 Ki = 1258.93 nM T25315 CW8G7L 71457683 Ki > 316.23 nM T25315 C4U0ZV 71457684 Ki = 2511.89 nM T25315 CC6QB3 71457685 Ki = 3162.28 nM T25315 CX1QO7 71459294 Ki = 63.1 nM T25315 CV7H9J 71459296 Ki = 501.19 nM T25315 CESM84 71459298 Ki = 630.96 nM T25315 C9TU4O 71459300 Ki = 199.53 nM T25315 CKM67R 71459302 Ki = 1995.26 nM T25315 CUYV29 71459523 Ki = 501.19 nM T25315 CXFU13 71459525 Ki > 316.23 nM T25315 CF4YM2 71459526 Ki > 316.23 nM T25315 CJ76KX 71459589 Ki = 316.23 nM T25315 C51UFM 71459591 Ki = 1995.26 nM T25315 C1T7DQ 71459593 Ki = 5011.87 nM T25315 C8B5LH 71459594 Ki = 5011.87 nM T25315 CK4AL7 71461073 Ki = 63.1 nM T25315 C5Y6DG 71461075 Ki = 125.89 nM T25315 C86CVJ 71461268 Ki = 630.96 nM T25315 C2ZJN0 71461270 Ki = 501.19 nM T25315 CSE9N6 71461272 Ki > 316.23 nM T25315 CGT2E1 71461273 Ki = 1995.26 nM T25315 CM5U7K 71461327 Ki > 316.23 nM T25315 CERW83 71461328 Ki = 1000 nM T25315 CQ2AS1 71461330 Ki = 1584.89 nM T25315 C3TGQ2 71461332 Ki = 6309.57 nM T25315 CF9K4W 71462809 Ki = 199.53 nM T25315 CM94FX 71462811 Ki = 316.23 nM T25315 CE63CT 71462813 Ki = 316.23 nM T25315 CP35IU 71462815 Ki = 251.19 nM T25315 C3U2YV 71462992 Ki = 1000 nM T25315 CT07HI 71462994 Ki = 398.11 nM T25315 C23LZH 71462996 Ki > 316.23 nM T25315 C6LDC4 71462997 Ki > 316.23 nM T25315 CS5F0N 71462998 Ki = 3981.07 nM T25315 C2ZF9P 71463056 Ki > 316.23 nM T25315 CFZ76K 71463057 Ki = 7943.28 nM T25315 C92XFW 71572192 IC50 = 13 nM T25315 C5D4UG 71585199 IC50 = 76 nM T25315 CT9FC8 71585298 IC50 = 99 nM T25315 CS2F9Z 71585504 IC50 = 1000 nM T25315 CN4TC7 71586201 IC50 = 60 nM T25315 C5J1QB 71586204 IC50 = 19 nM T25315 CG9Q0A 71586301 IC50 = 38 nM T25315 CY07QP 71586303 IC50 = 24 nM T25315 C27AGH 71586392 IC50 = 200 nM T25315 CV41FJ 71586393 IC50 = 37 nM T25315 C01KZL 71586394 IC50 = 35 nM T25315 C7DAX6 71586395 IC50 = 44 nM T25315 C4LZA0 71586485 IC50 = 55 nM T25315 CTIM92 71586679 IC50 = 53 nM T25315 C98ABQ 72188563 IC50 = 11 nM T25315 CNR52H 72547710 IC50 = 424 nM T25315 CEA80B 72547711 IC50 = 74 nM T25315 C5KND0 72547938 IC50 = 71 nM T25315 C5NXI9 72547939 IC50 = 81 nM T25315 C3NMQ1 72548178 IC50 = 81 nM T25315 CZC5F9 72549346 IC50 = 41 nM T25315 C0I7GV 72549347 IC50 = 34 nM T25315 CU49SV 72549349 IC50 = 44 nM T25315 C51ZCM 72549350 IC50 = 23 nM T25315 CP1WC8 72549588 IC50 = 108 nM T25315 CB40JU 72549589 IC50 = 95 nM T25315 C9XVJ7 72549590 IC50 = 677 nM T25315 C6J3EX 72549591 IC50 = 130 nM T25315 CNV52I 72549592 IC50 = 42 nM T25315 CIOM39 72549594 IC50 = 428 nM T25315 CWO36A 72549595 IC50 = 123 nM T25315 CTR8J1 72549596 IC50 = 440 nM T25315 CE4Y9I 72549821 IC50 = 31 nM T25315 CU5CS1 72550475 IC50 = 70 nM T25315 C0UP9J 72550699 IC50 = 143 nM T25315 CS74JL 76317929 IC50 = 437 nM T25315 CL4YU8 76325253 IC50 = 2295 nM T25315 C0EHJ3 76332481 IC50 = 1.6 nM T25315 CYWE71 89610442 IC50 = 1060 nM T25315 C0WE2I 89610499 IC50 = 176 nM T25315 C9QGW5 89610658 IC50 = 23 nM T25315 C7JG5M 89610683 IC50 = 25 nM T25315 CB59GM 89610699 IC50 = 607 nM T25315 CYCF45 89610786 IC50 = 26 nM T25315 CA0Z4U 90014266 IC50 = 61 nM T25315 CZ4L0V 90014377 IC50 = 152 nM T25315 CZ6Y5V 90014385 IC50 = 69 nM T25315 C5JC7Z 90014472 IC50 = 110 nM T25315 CMP3K2 90014508 IC50 = 73 nM T25315 CNB2Y5 90014551 IC50 = 256 nM T25315 CH0I5G 90014572 IC50 = 21 nM T25315 CE8FK0 90014593 IC50 = 263 nM T25315 C7J0VY 90014675 IC50 = 154 nM T25315 C85BYS 90014688 IC50 = 96 nM T25315 C74FIX 90014694 IC50 = 122 nM T25315 C76PCB 90014714 IC50 = 47 nM T25315 CNDX82 90014722 IC50 = 80 nM T25315 CEX71F 90014726 IC50 = 132 nM T25315 C9PD3S 90014869 IC50 = 146 nM T25315 CUV32W 90014874 IC50 = 91 nM T25315 C2YD5H 90015039 IC50 = 118 nM T25315 C24OKV 90015194 IC50 = 650 nM T25315 CA87ZB 90015254 IC50 = 1350 nM T25315 CAK7Q1 90066098 IC50 = 54 nM T25315 CF5L9K 90066144 IC50 = 91 nM T25315 C6ENV5 100951623 EC50 > 10000 nM T25315 C5S3FA 121292609 IC50 = 58 nM T25315 CV02LK 121292615 IC50 = 97 nM T25315 C9FH4Y 121292620 IC50 = 78 nM T25315 C1PK5J 121292622 IC50 = 32 nM T25315 CNM0Z1 121292625 IC50 = 19 nM T25315 CJV62Q 122471809 IC50 = 52 nM T25315 C1X6AT 127030692 EC50 = 600 nM T25315 CRHW82 127030693 EC50 = 758.58 nM T25315 C0J8LG 127030984 EC50 = 194.98 nM T25315 C4G6LB 127030985 EC50 = 229.09 nM T25315 CBA4V3 127030990 EC50 = 165.96 nM T25315 CVX0W5 127030991 EC50 = 512.86 nM T25315 C6JZY5 127031312 EC50 = 6025.6 nM T25315 C6WLS8 127031313 EC50 = 1230.27 nM T25315 C06IOQ 127031899 EC50 = 112.2 nM T25315 CC64XZ 127031900 EC50 = 9.772 nM T25315 C93HLB 127032163 EC50 = 158.49 nM T25315 CKE67A 127032165 EC50 = 125.89 nM T25315 CN38ZL 127032168 EC50 = 158.49 nM T25315 CKV42D 127032453 EC50 = 50.12 nM T25315 C1XSW6 127032454 EC50 = 8511.38 nM T25315 CMO31X 127032455 EC50 = 61.66 nM T25315 C0BZ6S 127032486 EC50 = 58.88 nM T25315 CL8Q5K 127032747 EC50 = 1318.26 nM T25315 CS1JN2 127032750 EC50 = 144.54 nM T25315 CUMG10 134131691 IC50 = 38 nM T25315 CEV3H8 134131840 IC50 = 202 nM T25315 CPC09W 134132003 IC50 = 1300 nM T25315 CKR13E 134132613 IC50 = 70 nM T25315 CQ2C9B 134132726 IC50 = 6600 nM T25315 CU78OH 134134300 IC50 = 340 nM T25315 CO71EK 134134604 IC50 = 4200 nM T25315 CNJ36D 134134840 IC50 = 290 nM T25315 CB9T4J 134134906 IC50 = 40 nM T25315 CC08FB 134135177 IC50 = 330 nM T25315 CAZ6K3 134136033 IC50 = 130 nM T25315 C1SA5H 134136200 IC50 = 225 nM T25315 CPQ65D 134137191 IC50 = 154 nM T25315 CNV52M 134137815 IC50 = 840 nM T25315 CZ4LV2 134137862 IC50 = 2200 nM T25315 CZC36F 134137981 IC50 = 190 nM T25315 C1GP4F 134138894 IC50 = 97 nM T25315 C46FKA 134139917 IC50 = 202 nM T25315 CND4Z9 134140161 IC50 = 82 nM T25315 C1L8KV 134140355 IC50 = 77 nM T25315 CQU74A 134140422 IC50 = 60 nM T25315 CD8HT5 134140497 IC50 = 110 nM T25315 CCPM57 134140635 IC50 = 138 nM T25315 CF41GA 134142277 IC50 = 36 nM T25315 C4DSH2 134143368 IC50 = 403 nM T25315 C9NW5Z 134145083 IC50 = 345 nM T25315 CKJ7I5 134145500 IC50 = 160 nM T25315 C2TYL4 134146441 IC50 = 121 nM T25315 CWJA75 134146842 IC50 = 120 nM T25315 C8RNK1 134147361 IC50 = 790 nM T25315 CJ0BG7 134147406 IC50 = 443 nM T25315 C7EUC1 134147547 IC50 = 3260 nM T25315 CWO0M7 134148525 IC50 = 1200 nM T25315 C6H7FC 134149982 IC50 = 110 nM T25315 CBJ4F7 134150725 IC50 = 1800 nM T25315 CCN4V5 134150746 IC50 = 187 nM T25315 CL7X9S 134150776 IC50 = 780 nM T25315 C68HZQ 134151426 IC50 = 230 nM T25315 CGMB02 134151603 IC50 = 382 nM T25315 C4CA8F 134153150 IC50 = 120 nM T25315 CBL28D 134153156 IC50 = 55 nM T25315 C2RI7V 134153689 IC50 = 65 nM T25315 CX5HE7 134155138 IC50 = 240 nM T25315 COE60H 134156130 IC50 = 105 nM T25315 CHG9K2 134156221 IC50 = 210 nM T25315 C3UM0P 134156632 IC50 = 126 nM T25315 C4C1BX 134157695 IC50 = 39 nM T25315 C6HAX2 136037880 IC50 = 760 nM T25315 D05EML 21847 IC50 > 10000 nM T25315 D0A8PV 45784923 IC50 = 5 nM T25315 D0EK9K 11997335 IC50 = 2.8 nM T89988 D0L5RW 65015 IC50 = 0.04 nM T89988 D00XBC 46861584 IC50 > 10000 nM T89988 D01UBY 46208367 IC50 = 30 nM T89988 D03KKR 3547 IC50 = 35000 nM T89988 D06EPO 11192346 IC50 = 0.5 nM T89988 D06IME 25134303 IC50 = 5 nM T89988 D0O2XQ 11256587 IC50 > 10000 nM T89988 D0TG9Q 11180808 Ki = 0.55 nM T89988 D0YQ7U 11285792 IC50 = 5.9 nM T89988 D0X4SI 9953769 Ki = 58.88 nM T89988 D07KIJ 10008367 IC50 = 3.8 nM T89988 D0Q2JS 10436045 Ki = 16.6 nM T89988 D0W0LS 183789 IC50 = 0.08 nM T89988 C9KT7Q 163751 IC50 = 35000 nM T89988 CJ8NY6 261407 IC50 = 1700 nM T89988 CQ3KO7 483339 IC50 > 1000 nM T89988 C7AP9W 483340 IC50 > 1000 nM T89988 CAB79M 483341 IC50 > 1000 nM T89988 C7XW2D 483342 IC50 > 1000 nM T89988 C7PMT6 483343 IC50 > 1000 nM T89988 CP25RI 483344 IC50 > 1000 nM T89988 CA5BZ8 491773 IC50 > 10000 nM T89988 C0KB6Y 508727 IC50 = 4330 nM T89988 C9J5OC 508729 IC50 = 832 nM T89988 CI96OK 508741 IC50 = 3170 nM T89988 C5P1IN 508742 IC50 = 121 nM T89988 C6B5MG 508744 IC50 = 66000 nM T89988 CRN41P 508749 IC50 = 5500 nM T89988 CEF6L0 508750 EC50 = 40 nM T89988 CUJ2K6 508869 IC50 = 3.9 nM T89988 CAZC09 508870 IC50 = 96 nM T89988 CT83OL 508877 IC50 = 39 nM T89988 CUK86N 3013430 Ki = 23.99 nM T89988 C1TX2Y 3794409 Ki = 199.53 nM T89988 CPZ6S1 3796276 Ki = 213.8 nM T89988 CMT8K7 5481702 IC50 = 10000 nM T89988 CHCY06 6918496 IC50 > 1000 nM T89988 C02HZB 9825735 IC50 = 1500 nM T89988 C9C8EY 9836178 IC50 = 30000 nM T89988 CHP4O1 9840006 IC50 = 1000 nM T89988 CBVJ87 9842404 IC50 = 42000 nM T89988 CH57DZ 9850318 IC50 = 2 nM T89988 C0RB2U 9851741 IC50 = 59 nM T89988 CV58QE 9852285 IC50 = 460 nM T89988 C5XMP4 9857714 IC50 = 2000 nM T89988 CC9U3T 9857981 Ki = 79.43 nM T89988 C56GPV 9858433 IC50 = 4000 nM T89988 C4JEY6 9870980 Ki = 125.89 nM T89988 C9FO1Q 9873546 IC50 = 150 nM T89988 C0PW6L 9885442 IC50 = 390 nM T89988 CZ1OG4 9885683 IC50 = 1020 nM T89988 C8LX2W 9889422 IC50 = 370 nM T89988 C1Q2IG 9890559 IC50 = 13000 nM T89988 C0T6NW 9900683 IC50 = 10000 nM T89988 CC1J0A 9900997 IC50 > 100000 nM T89988 C2R6KA 9902204 Ki = 18.62 nM T89988 C0RH2D 9902578 Ki = 138.04 nM T89988 C9Q6NK 9923015 IC50 = 1600 nM T89988 CY4B8U 9924108 Ki = 162.18 nM T89988 C3Y0QF 9924357 IC50 > 10000 nM T89988 CWG28E 9934977 IC50 = 200 nM T89988 CSH40U 9936494 IC50 > 10000 nM T89988 C7LY1M 9945265 Ki = 95.5 nM T89988 C2KXZ6 9945514 IC50 > 10000 nM T89988 C3PU5K 9946967 IC50 > 10000 nM T89988 CM28YJ 9949615 Ki = 29 nM T89988 CR1Z2G 9952114 IC50 = 6900 nM T89988 C91RTG 9956238 IC50 = 80 nM T89988 C0MGT8 9956260 IC50 = 970 nM T89988 CL3KT8 9967166 Ki = 64.57 nM T89988 CTFZ89 9967349 Ki = 36.31 nM T89988 CBVP31 9967465 Ki = 239 nM T89988 CY89AV 9967878 IC50 = 1000 nM T89988 CA74YF 9974356 IC50 = 11000 nM T89988 CT1FH0 9986630 IC50 = 2.3 nM T89988 CE7IB5 10007642 IC50 = 2.3 nM T89988 C9POK8 10025168 IC50 = 7400 nM T89988 CI3Q9B 10030247 IC50 = 44 nM T89988 C1X6HO 10041590 IC50 = 14000 nM T89988 C5GPK2 10052388 IC50 = 7.798 nM T89988 CQ7N3R 10064487 IC50 = 15000 nM T89988 CMSQ48 10065796 IC50 = 10000 nM T89988 CC03WA 10111333 Ki = 5.623 nM T89988 CM4P8A 10115566 IC50 = 540 nM T89988 C49DEF 10117347 IC50 > 30000 nM T89988 CIDS73 10117480 IC50 = 32 nM T89988 C2ICH4 10119551 IC50 = 28 nM T89988 CC5H0K 10120067 IC50 = 33 nM T89988 C7I9OB 10120907 IC50 = 2.1 nM T89988 CHFP31 10129107 IC50 = 153 nM T89988 CY4AK3 10129192 IC50 = 0.7 nM T89988 CU96TE 10129343 IC50 = 6.5 nM T89988 CM48CP 10132885 Ki = 154.88 nM T89988 CFH9U0 10133557 Ki = 91.2 nM T89988 CF25OU 10137967 IC50 = 320 nM T89988 C47VWF 10138789 IC50 = 630 nM T89988 CAP8K0 10139782 IC50 = 390 nM T89988 CO65TA 10141379 IC50 = 350 nM T89988 C4SHX2 10142792 IC50 = 8 nM T89988 CH83KL 10143025 IC50 = 1200 nM T89988 C09XVI 10144709 IC50 = 1.3 nM T89988 CP6NQ5 10152864 IC50 = 7.5 nM T89988 CF2ZP9 10153373 IC50 = 199.5 nM T89988 CK0CY4 10153431 IC50 = 46 nM T89988 C0Q5AE 10154434 IC50 = 1000 nM T89988 CXI9T2 10154979 IC50 = 1500 nM T89988 C2U4WP 10159217 IC50 > 30000 nM T89988 C93BOF 10161975 IC50 = 1000 nM T89988 CLS30W 10162782 IC50 = 240 nM T89988 CFLN89 10162844 IC50 = 17 nM T89988 CY4OA2 10164316 IC50 = 48 nM T89988 CFKN38 10164641 IC50 > 1000 nM T89988 C50XKS 10165042 IC50 = 190 nM T89988 CKAH17 10165625 IC50 = 5.3 nM T89988 C4V5KG 10165716 IC50 = 150 nM T89988 COMN76 10167417 IC50 = 5.2 nM T89988 CI45NC 10175423 IC50 = 21 nM T89988 C10HSL 10175425 IC50 = 1.4 nM T89988 CBTG57 10182382 IC50 = 66 nM T89988 C1BGH8 10182763 IC50 > 30000 nM T89988 CH5AC1 10183362 IC50 = 64 nM T89988 CGP07U 10184007 IC50 = 1190 nM T89988 C2ED3X 10184169 IC50 > 10000 nM T89988 C5A2QV 10184250 IC50 = 100 nM T89988 CM80RH 10186010 IC50 = 100 nM T89988 C5Z8RT 10187492 IC50 = 84 nM T89988 C89VMQ 10195882 IC50 = 37 nM T89988 CSM35L 10196988 IC50 = 38 nM T89988 C9SX8I 10203447 IC50 = 2200 nM T89988 CXK43P 10204589 IC50 > 30000 nM T89988 C4OM2Z 10205915 IC50 > 10000 nM T89988 CNI37B 10205937 IC50 = 110 nM T89988 CWZY76 10206007 IC50 = 65 nM T89988 CV5WX9 10206776 IC50 = 170 nM T89988 CS0RU7 10207542 IC50 = 87 nM T89988 CM0UY9 10207590 IC50 = 19 nM T89988 CH04CE 10207591 IC50 = 600 nM T89988 CS98YN 10207639 IC50 = 11 nM T89988 CWC7X1 10208080 IC50 > 10000 nM T89988 CHDE08 10208555 IC50 = 6400 nM T89988 C4NMH6 10208946 IC50 = 27 nM T89988 C6YL0V 10209102 IC50 = 7000 nM T89988 C91ZMU 10209478 IC50 = 5 nM T89988 CE4I6T 10218403 IC50 = 1.5 nM T89988 CO48MN 10218812 IC50 = 41.3 nM T89988 CHP92E 10218843 IC50 = 8.4 nM T89988 C4EBQ9 10225909 IC50 = 5500 nM T89988 CF3WZ0 10227556 IC50 = 250 nM T89988 C84HKV 10227655 IC50 = 160 nM T89988 CK9AQ7 10228205 IC50 = 88 nM T89988 CYV95X 10228435 IC50 = 7 nM T89988 C72HMR 10228761 IC50 > 30000 nM T89988 C02UNG 10232019 IC50 = 9.3 nM T89988 CV7G6W 10239671 IC50 = 172 nM T89988 CMF6D0 10239991 IC50 = 2.05 nM T89988 C1AK9C 10240064 IC50 = 0.2 nM T89988 CU53XR 10240278 IC50 = 44.5 nM T89988 C3H4ST 10245340 IC50 = 30000 nM T89988 CNEW23 10256127 IC50 = 1230 nM T89988 CMRA02 10257042 Ki = 39.81 nM T89988 CPX15I 10268598 IC50 = 3900 nM T89988 CR6SA7 10269886 IC50 > 10000 nM T89988 CK49NQ 10272003 IC50 = 700 nM T89988 CPOD91 10276594 IC50 = 230 nM T89988 CIHB65 10277182 IC50 = 3010 nM T89988 C3CZ7H 10277466 IC50 > 10000 nM T89988 CO2HE6 10278257 IC50 = 19 nM T89988 CWGJ31 10278862 IC50 = 97 nM T89988 CW0H9D 10279078 IC50 = 41 nM T89988 CXZ08C 10279914 IC50 = 2400 nM T89988 CE9ID0 10280944 IC50 > 10000 nM T89988 CD4YG9 10281316 IC50 = 3.6 nM T89988 CWGK21 10281715 IC50 = 4.7 nM T89988 C7ODM2 10289827 IC50 = 0.3 nM T89988 CH97RC 10291634 IC50 = 1500 nM T89988 CDU26C 10293022 Ki = 15.85 nM T89988 CJ06NI 10299408 IC50 = 31 nM T89988 C6E1CB 10299952 IC50 = 400 nM T89988 C06FDK 10300282 IC50 = 110 nM T89988 CFX3M7 10300284 IC50 = 6.7 nM T89988 C6LP8U 10300705 IC50 = 7860 nM T89988 CO0P4F 10301330 IC50 > 10000 nM T89988 CDRW29 10302973 IC50 = 65 nM T89988 CF01AR 10304021 IC50 = 4 nM T89988 CY7P9S 10312346 IC50 = 8.1 nM T89988 C2QM0N 10315045 IC50 = 17000 nM T89988 CWFB30 10323427 IC50 = 30 nM T89988 CCDY38 10323468 IC50 = 28 nM T89988 CBA2C6 10325032 IC50 = 6 nM T89988 C1N0CE 10346048 IC50 = 173.78 nM T89988 CT40XZ 10348168 IC50 = 165 nM T89988 C62PXQ 10360623 IC50 = 23000 nM T89988 CC0YO3 10371682 IC50 = 1040 nM T89988 C7PUE4 10392559 IC50 = 64 nM T89988 CCZ17H 10392978 IC50 = 2 nM T89988 CU81IS 10409097 IC50 = 30000 nM T89988 CKYF72 10414966 IC50 = 144 nM T89988 CZ65IG 10427217 IC50 = 14000 nM T89988 C6GQ5E 10427222 IC50 = 56 nM T89988 CYVI63 10436083 IC50 = 400 nM T89988 C8SPW7 10458152 IC50 = 218.78 nM T89988 CI10WZ 10459336 IC50 = 900 nM T89988 C9NZT2 10471319 IC50 = 22000 nM T89988 CJL0P6 10482463 IC50 = 50 nM T89988 C95LRC 10940216 Ki = 590 nM T89988 CQ6S7M 10957890 IC50 = 2000 nM T89988 CR52KG 11155781 IC50 = 49 nM T89988 C8BF7M 11179439 IC50 = 3.8 nM T89988 CAEB68 11180383 IC50 = 7.9 nM T89988 CZ80GK 11180885 IC50 = 240 nM T89988 C1KHV0 11192300 IC50 = 40 nM T89988 C16MCS 11192943 IC50 = 0.9 nM T89988 CG9OA2 11214277 IC50 = 305 nM T89988 CTN5C2 11215504 IC50 = 340 nM T89988 CK21LX 11223594 IC50 > 10000 nM T89988 C62UXT 11226430 IC50 = 20 nM T89988 CU75LJ 11227168 IC50 = 4.3 nM T89988 C5AYG7 11227368 IC50 = 102 nM T89988 CO3M2S 11227383 IC50 = 125 nM T89988 CA39QR 11227406 IC50 > 10000 nM T89988 C3G5PZ 11237168 IC50 = 65 nM T89988 C1LWU2 11237256 IC50 = 43 nM T89988 CQ6KW0 11272103 IC50 = 10000 nM T89988 CZ8DU0 11273379 IC50 = 8.8 nM T89988 CTRB13 11273475 IC50 = 131.5 nM T89988 CSG19P 11283842 IC50 = 4.5 nM T89988 C06TUD 11285791 IC50 = 5.9 nM T89988 C7N1ZH 11296325 IC50 = 53 nM T89988 C0P9IM 11296618 IC50 = 51.5 nM T89988 CA63BF 11306757 IC50 = 7.1 nM T89988 CW47VZ 11318368 IC50 = 95 nM T89988 C4FS8T 11319072 IC50 = 10 nM T89988 C1A5ET 11329244 IC50 = 10000 nM T89988 CGE2P7 11329328 IC50 = 126 nM T89988 CQ1CG9 11330529 IC50 = 5.4 nM T89988 CIT2Y7 11330837 IC50 = 10 nM T89988 CX3PY4 11340816 IC50 = 66 nM T89988 C95SAU 11341950 IC50 = 710 nM T89988 CF98IO 11342351 IC50 = 38 nM T89988 CKZ20A 11353843 IC50 = 3.6 nM T89988 CX6C2M 11353855 IC50 = 1.9 nM T89988 C0JT3P 11364218 IC50 = 217 nM T89988 CZ82WH 11365166 IC50 = 1.8 nM T89988 CE2M9F 11387511 IC50 = 2.6 nM T89988 CE5ZK6 11409228 IC50 = 11 nM T89988 C2N0AG 11421712 IC50 = 3.8 nM T89988 CWV9L6 11421840 IC50 = 2.8 nM T89988 C9Z0TH 11433008 IC50 = 2.4 nM T89988 C1K6PE 11456448 IC50 = 45.5 nM T89988 CH7E4M 11466237 IC50 = 51 nM T89988 C25XGJ 11467577 IC50 = 136.5 nM T89988 C3S7DQ 11478362 IC50 = 690 nM T89988 C78GWT 11489078 IC50 = 23 nM T89988 C70LYJ 11497533 IC50 = 15 nM T89988 C7I8FQ 11502188 IC50 = 1184 nM T89988 C40IMW 11502371 IC50 = 20 nM T89988 CB7UX1 11504634 IC50 = 17 nM T89988 C1LCD7 11510932 IC50 = 244 nM T89988 CWVX78 11512375 IC50 = 16.7 nM T89988 C54PDI 11526729 IC50 = 50 nM T89988 C0BF5R 11527661 IC50 = 2.6 nM T89988 C0F7SR 11534473 IC50 = 6 nM T89988 CG29EI 11540494 IC50 = 0.6 nM T89988 C4AH1P 11541149 IC50 = 15 nM T89988 C0HYO4 11548199 IC50 = 2 nM T89988 CKGI84 11553070 IC50 = 37 nM T89988 C26UCI 11553489 IC50 = 15 nM T89988 CK5DE0 11555541 IC50 = 40 nM T89988 CCJ4G1 11555827 IC50 = 2.5 nM T89988 C9HK2R 11562947 IC50 = 10 nM T89988 C4E7NT 11563451 IC50 = 178 nM T89988 C5AL9R 11563597 IC50 = 633.87 nM T89988 CCQ8O9 11567495 IC50 = 123 nM T89988 CQ0TD1 11570045 IC50 = 441.57 nM T89988 CLY5O2 11570431 IC50 = 209 nM T89988 C7RKT1 11577400 IC50 = 213 nM T89988 C2DG4A 11582651 IC50 = 161 nM T89988 C41DRT 11584094 IC50 = 6 nM T89988 C6KL3Q 11585168 IC50 = 43.95 nM T89988 CBN18P 11590644 IC50 = 567 nM T89988 CYG74X 11591595 IC50 = 7 nM T89988 CF50KQ 11591776 IC50 = 5 nM T89988 CN5OV9 11591956 IC50 = 4 nM T89988 CH0OD8 11598084 IC50 = 42 nM T89988 C1DKF4 11598797 IC50 > 10000 nM T89988 C1FH6B 11599317 IC50 = 7 nM T89988 C9FK3O 11605635 IC50 = 6 nM T89988 C6BET5 11605867 IC50 = 20 nM T89988 CYP0L5 11605985 IC50 = 522.4 nM T89988 CS8HR5 11606147 IC50 = 10 nM T89988 CZQ78X 11606167 IC50 = 2391 nM T89988 C84YPR 11606411 IC50 = 1.3 nM T89988 C6V9WA 11606702 IC50 = 8.995 nM T89988 CTQ6D9 11613399 IC50 = 6 nM T89988 C1N4CJ 11620726 IC50 = 167.88 nM T89988 CS9R1X 11621035 IC50 = 7.7 nM T89988 C8NKD4 11627639 IC50 = 2.4 nM T89988 C05TNG 11627840 IC50 = 0.2 nM T89988 CNS5P7 11632418 IC50 = 170 nM T89988 C40GEC 11633080 IC50 = 90 nM T89988 CU7B6I 11634118 IC50 = 904 nM T89988 C3EAG5 11634928 IC50 = 9 nM T89988 C57RHQ 11634966 IC50 > 10000 nM T89988 C2OD0U 11635092 IC50 = 120 nM T89988 CQ65EJ 11640044 IC50 = 30 nM T89988 CP21CA 11641253 IC50 = 46 nM T89988 C0B9YV 11643006 IC50 = 0.6 nM T89988 C9IOM8 11647276 IC50 = 16 nM T89988 C3IFQ9 11662833 IC50 = 80 nM T89988 CU7RT2 11663882 IC50 = 10 nM T89988 CNJE21 11663995 IC50 = 1225 nM T89988 CU7OG2 11669935 IC50 = 18 nM T89988 CPI1S3 11670910 IC50 = 1800 nM T89988 CC2LB1 11670968 IC50 = 25 nM T89988 CVX87R 11671120 IC50 = 50 nM T89988 C6BY1A 11678573 IC50 = 66 nM T89988 CR91QA 11690139 IC50 = 856 nM T89988 CS1W5I 11690536 IC50 = 337 nM T89988 CJL2T5 11692057 IC50 = 210 nM T89988 CS31YE 11699149 IC50 = 4 nM T89988 C4QLY1 11699524 IC50 = 6 nM T89988 CI5G6C 11699541 IC50 = 20 nM T89988 CU8L6Q 11700079 IC50 = 6.3 nM T89988 CCB51S 11706775 IC50 = 207.01 nM T89988 C6CM7S 11711078 IC50 = 277 nM T89988 CJ03AX 11712754 IC50 = 40 nM T89988 C9IQK5 11713221 IC50 = 10 nM T89988 CDN6X8 11718088 IC50 = 40 nM T89988 CKF6U5 11721085 IC50 = 30 nM T89988 C38IBK 11721374 IC50 = 1 nM T89988 CZR39O 11723420 IC50 = 20000 nM T89988 CPG15O 11743399 IC50 > 10000 nM T89988 C4L9EC 11752457 IC50 = 6.9 nM T89988 C7A4YV 11753466 IC50 = 1.9 nM T89988 CU5P8D 11753664 IC50 = 11 nM T89988 CKW9D4 11756884 IC50 = 2.3 nM T89988 C1S3JD 11843812 IC50 = 822 nM T89988 C2X7GJ 11843813 IC50 = 930 nM T89988 CS6JC4 11843945 IC50 = 1000 nM T89988 CBV2X9 11843946 IC50 = 1100 nM T89988 C1HV9G 11844079 IC50 = 1100 nM T89988 CR7MI5 11844083 IC50 = 780 nM T89988 CEM02F 11844209 IC50 = 160 nM T89988 C2J8RH 11844212 IC50 = 80 nM T89988 C02CKY 11844329 IC50 = 320 nM T89988 C9RE0B 11844467 IC50 = 1500 nM T89988 C63QMF 11844468 IC50 = 700 nM T89988 C0DRU3 11844469 IC50 = 140 nM T89988 CGHL19 11844470 IC50 = 45 nM T89988 C5PL9R 11844471 IC50 = 440 nM T89988 CMT8N9 11844595 IC50 = 120 nM T89988 CRY83B 12093162 Ki = 213.8 nM T89988 C2QWR3 12093163 Ki = 263.03 nM T89988 C79CBJ 12093167 Ki = 10 nM T89988 CJX31Q 12093170 IC50 = 170 nM T89988 CH5QK9 15290299 IC50 = 230 nM T89988 C1T0SU 15518124 IC50 = 13400 nM T89988 C7X3CQ 15604497 Ki = 25.12 nM T89988 CQJ7Y2 15985912 Ki = 10 nM T89988 C0G1SC 15985914 Ki = 31.62 nM T89988 CKE0U5 15985981 Ki = 501.19 nM T89988 CYA3K5 16064151 IC50 = 0.4 nM T89988 CX04NO 16066354 IC50 = 1.7 nM T89988 C9G8TZ 16124598 Ki = 1.259 nM T89988 CH90BN 16216716 IC50 = 1.8 nM T89988 C6D5FS 16720313 IC50 = 36 nM T89988 C9XH8N 17756652 Ki = 10 nM T89988 CMEZ85 17838131 IC50 > 100000 nM T89988 CGFW16 17838175 IC50 > 100000 nM T89988 CZT35Q 17838190 IC50 > 100000 nM T89988 CCR8J4 17838276 IC50 > 100000 nM T89988 C5CH8K 17866152 IC50 = 5000 nM T89988 CMD76W 18426157 IC50 = 17000 nM T89988 C0EB8U 18426192 IC50 = 11000 nM T89988 CRM90U 19430534 Ki = 794.33 nM T89988 C6K9RC 21098468 IC50 = 8000 nM T89988 CMF27K 21098469 IC50 = 7000 nM T89988 C7WBX4 21098475 IC50 > 30000 nM T89988 CFB3T6 21098478 IC50 = 8000 nM T89988 C9T8FA 21098480 IC50 = 5000 nM T89988 CMA42E 21098488 IC50 = 1000 nM T89988 C9JI3T 21098490 IC50 = 1000 nM T89988 CK51MC 21098512 IC50 = 19000 nM T89988 CN8F1W 21098519 IC50 = 1000 nM T89988 CW0BP6 21098523 IC50 = 1000 nM T89988 C1WM8S 21098530 IC50 = 19000 nM T89988 CYX26M 22143104 IC50 = 19 nM T89988 CF9I5G 22143112 IC50 = 3.8 nM T89988 C10IVJ 22143146 IC50 = 5.5 nM T89988 C8ESY2 22143155 IC50 = 5.4 nM T89988 C53NIP 22143196 IC50 = 28 nM T89988 C5G7CR 22143200 IC50 = 510 nM T89988 CZ3BU6 22143225 IC50 = 167.5 nM T89988 C17DEU 22143241 IC50 = 7 nM T89988 CDB86Q 22143255 IC50 = 2 nM T89988 C8LDZ2 22143258 IC50 = 22.5 nM T89988 CX1L8K 22143293 IC50 = 6.1 nM T89988 CH85XV 22143294 IC50 = 7.9 nM T89988 C89IFO 22143305 IC50 = 12.5 nM T89988 CY4GU1 22143308 IC50 = 123 nM T89988 CVZ64R 22143309 IC50 = 26 nM T89988 CV8F9U 22143314 IC50 = 463 nM T89988 C42ZHE 22143334 IC50 = 0.95 nM T89988 CP6X1V 22143346 IC50 = 4.8 nM T89988 C3POB6 22143349 IC50 = 155 nM T89988 C2CPY8 22268768 IC50 = 8700 nM T89988 C1TS9Z 22310839 IC50 = 2200 nM T89988 CT36VS 22310850 IC50 = 8600 nM T89988 CT4C1M 22310869 IC50 = 2300 nM T89988 CRX1D6 22310876 IC50 = 6090 nM T89988 CM2S9I 22310877 IC50 = 1130 nM T89988 C7ZJ3B 22310883 IC50 = 230 nM T89988 CI1C9R 22310896 IC50 = 170 nM T89988 C7GH1P 22310899 IC50 = 1360 nM T89988 C59BIA 22310903 IC50 = 1210 nM T89988 CG25OW 22310914 IC50 = 90 nM T89988 CDY16V 22310924 IC50 = 340 nM T89988 CG8L6I 22310929 IC50 = 125 nM T89988 C9E4LG 22310939 IC50 = 1050 nM T89988 C6R0DG 22310943 IC50 = 1640 nM T89988 CKY2B0 22310945 IC50 = 410 nM T89988 CFQ7P1 22310946 IC50 = 1310 nM T89988 C64QRB 22310953 IC50 = 1270 nM T89988 C3P8YN 22310954 IC50 = 110 nM T89988 C6D4KC 22310965 IC50 = 99 nM T89988 CW37TA 22310971 IC50 = 1190 nM T89988 C0CZL1 22310972 IC50 = 640 nM T89988 CUG43R 22310976 IC50 = 150 nM T89988 C38PHN 22310991 IC50 = 280 nM T89988 CJ2H7Q 22310992 IC50 = 96 nM T89988 C8RPO2 22310995 IC50 = 500 nM T89988 CE32SQ 22311000 IC50 = 340 nM T89988 CTV2K4 22311005 IC50 = 4780 nM T89988 CC9YA1 22335665 Ki = 57 nM T89988 CTO2A8 22335694 Ki = 17.78 nM T89988 C2NK9E 22394337 IC50 = 3010 nM T89988 CKO01W 22725647 Ki = 8.128 nM T89988 CT7Q3X 23405932 IC50 = 55 nM T89988 CB28YR 23441036 IC50 = 21000 nM T89988 CZA0F3 23441058 IC50 = 19000 nM T89988 CUI9H4 23630215 IC50 = 7.3 nM T89988 CEP68R 23655673 IC50 = 3300 nM T89988 C4BZ9J 23655877 IC50 = 1100 nM T89988 C6BDU5 23656067 IC50 = 470 nM T89988 C53TJN 23656260 IC50 = 660 nM T89988 CL0GR2 23656261 IC50 = 115 nM T89988 CZ05MF 23656430 IC50 = 4 nM T89988 C2LOI1 23656431 IC50 = 4 nM T89988 C5JNY2 23656432 IC50 = 3400 nM T89988 C0WBE1 23656433 IC50 = 6800 nM T89988 C98MGF 23656434 IC50 = 720 nM T89988 CM5SO9 23656584 IC50 = 320 nM T89988 CN9GW5 23656585 IC50 = 210 nM T89988 C7JV4W 23725177 IC50 = 0.67 nM T89988 C25HKJ 24758044 IC50 > 20000 nM T89988 C4QO9W 24801178 IC50 = 12000 nM T89988 C9P3YJ 24801179 IC50 = 2170 nM T89988 CT05NH 24801180 IC50 = 2117.2 nM T89988 C8Q4KT 24801342 IC50 = 530 nM T89988 CV28RW 24801343 IC50 = 400 nM T89988 C9NT2S 24801344 IC50 = 360 nM T89988 C5RV7A 24801345 IC50 = 4130 nM T89988 CI1EC7 24801346 IC50 = 550 nM T89988 CM81GS 24801522 IC50 = 37 nM T89988 CXYQ23 24801523 IC50 = 64 nM T89988 C64WPY 24801524 IC50 = 87 nM T89988 C9EB2J 24801525 IC50 = 130 nM T89988 C4C2LP 24801526 IC50 = 4.8 nM T89988 CKW46B 24801689 IC50 = 9 nM T89988 CA15KP 24801690 IC50 = 5.1 nM T89988 C3K1DA 25007995 IC50 = 80 nM T89988 CB45YS 25007996 IC50 = 160 nM T89988 CM17BE 25008678 IC50 = 6450 nM T89988 CU69WN 25008679 IC50 = 12000 nM T89988 C4OH9R 25008849 IC50 = 8400 nM T89988 C0HIK4 25010616 IC50 = 160 nM T89988 C9W6LE 25022597 IC50 = 3.2 nM T89988 CDKJ78 25033361 IC50 = 300 nM T89988 CLM02V 25110564 Ki = 5300 nM T89988 CGO4J0 25110660 Ki = 79 nM T89988 C9XI0Q 25110678 Ki = 7100 nM T89988 CKA50N 25110679 Ki = 5100 nM T89988 C3SHW4 25110716 IC50 = 2.5 nM T89988 C6U3YK 25110788 IC50 = 3 nM T89988 C67QXP 25154827 IC50 = 4 nM T89988 C54LQF 25230828 IC50 > 50000 nM T89988 CK5HZ8 25256791 IC50 = 1200 nM T89988 C8IHN4 25267730 IC50 = 1020 nM T89988 C50IVN 25267738 IC50 = 4750 nM T89988 C0ZVT1 25268077 IC50 > 10000 nM T89988 CJD3B9 25268081 IC50 = 200 nM T89988 CR9M5T 25268085 IC50 = 250 nM T89988 CZ3BX9 25268434 IC50 > 10000 nM T89988 CT5XC3 25268436 IC50 = 390 nM T89988 CKA42N 25268440 IC50 = 230 nM T89988 CC3Y9N 25268442 IC50 = 9550 nM T89988 C0O3DW 25268795 IC50 = 8950 nM T89988 CK03BL 25268803 IC50 = 1810 nM T89988 C41GLE 25269516 IC50 = 4250 nM T89988 CLZ9P0 25270182 IC50 = 3440 nM T89988 C2FZ9P 42606792 IC50 = 1.8 nM T89988 C1VQ0H 42632811 IC50 = 11350 nM T89988 C2L3AW 42632830 IC50 = 7800 nM T89988 COGL90 42632836 IC50 = 710 nM T89988 CTDE24 42632840 IC50 = 3250 nM T89988 CYLQ82 42632863 IC50 = 2000 nM T89988 CB95UT 42632867 IC50 > 10000 nM T89988 CLCX87 42632888 IC50 = 2550 nM T89988 CU2PO5 44180522 Ki = 6 nM T89988 C5YFB9 44252324 IC50 > 10000 nM T89988 C13YRA 44296077 Ki = 5900 nM T89988 CTN90Y 44296087 Ki = 420 nM T89988 CTNF31 44296137 Ki = 79 nM T89988 CR1WU3 44296138 Ki > 10000 nM T89988 C9D4HM 44296154 Ki = 660 nM T89988 CKU4Y6 44296155 Ki = 2500 nM T89988 CSTN01 44296156 Ki > 10000 nM T89988 CD53WG 44296219 IC50 = 32 nM T89988 CL5VC0 44296240 Ki > 10000 nM T89988 CJGP84 44296264 Ki = 1700 nM T89988 C0IT6Z 44296265 Ki = 1450 nM T89988 CUG58H 44296266 Ki = 790 nM T89988 C1ZT7N 44296268 Ki = 234 nM T89988 C4M5CB 44296269 Ki = 2800 nM T89988 CX2U4R 44296287 Ki = 2900 nM T89988 CKD7I3 44296309 Ki = 6300 nM T89988 CVG7F2 44296310 Ki = 1200 nM T89988 CG0YU3 44296344 Ki = 4200 nM T89988 C52TFI 44296366 Ki = 360 nM T89988 C9VQ3K 44296384 Ki = 360 nM T89988 CAK80S 44296398 Ki = 550 nM T89988 CW5M1B 44296409 Ki = 4400 nM T89988 C02RMO 44296410 Ki = 560 nM T89988 CUY1A6 44296428 Ki = 520 nM T89988 C1FOD9 44296429 Ki = 870 nM T89988 C4H7XD 44296469 Ki = 4400 nM T89988 CL47OS 44296501 Ki = 1600 nM T89988 C6AR0I 44296628 Ki = 790 nM T89988 CYTQ98 44296629 Ki = 460 nM T89988 C74OLQ 44296630 Ki = 350 nM T89988 C67OGJ 44309012 Ki = 251 nM T89988 CUH16K 44353170 IC50 = 12700 nM T89988 CJ51CI 44353190 IC50 = 770 nM T89988 C4SWE0 44353196 IC50 = 1030 nM T89988 C03UXF 44353197 IC50 = 370 nM T89988 CU4ZX3 44353205 IC50 > 50000 nM T89988 C8X6VI 44353223 IC50 = 27000 nM T89988 CF6SK1 44353334 IC50 = 1480 nM T89988 CQK9U6 44353356 IC50 = 12300 nM T89988 CN7MI9 44353367 IC50 = 300 nM T89988 C2LA3C 44353369 IC50 = 5770 nM T89988 CYMD40 44353370 IC50 = 650 nM T89988 CM1OG0 44353377 IC50 = 3880 nM T89988 C9XGW6 44353380 IC50 > 50000 nM T89988 C4EG3U 44353395 IC50 = 120 nM T89988 CBYQ54 44353396 IC50 = 220 nM T89988 CV54UG 44353408 IC50 > 50000 nM T89988 C5Q3VF 44353418 IC50 = 10840 nM T89988 C2PIM0 44353464 IC50 = 260 nM T89988 CRVF39 44353617 IC50 = 12600 nM T89988 CZE90S 44395028 IC50 = 1500 nM T89988 CYJC04 44395029 IC50 = 2300 nM T89988 CIHC30 44395036 IC50 = 74000 nM T89988 CUFP61 44395048 IC50 = 1500 nM T89988 CGN58X 44395055 EC50 = 610 nM T89988 C1N9IW 44395058 IC50 = 11000 nM T89988 C20DZS 44395061 IC50 = 1500 nM T89988 CJ47HB 44395062 IC50 = 1500 nM T89988 CW78VC 44395066 IC50 = 87000 nM T89988 C2HY0B 44395079 IC50 = 9300 nM T89988 CZ7EM1 44395088 IC50 = 7000 nM T89988 C7HL3J 44395092 IC50 = 6400 nM T89988 CXN1E3 44395093 IC50 = 11000 nM T89988 C1G8LN 44395094 IC50 = 4500 nM T89988 C78EIY 44395097 IC50 = 22000 nM T89988 CC0VD9 44395104 IC50 = 17000 nM T89988 C0EZ1N 44395113 IC50 = 11000 nM T89988 C4P3YI 44395114 IC50 > 100000 nM T89988 CVR3C4 44395125 IC50 = 43000 nM T89988 C17BVS 44395126 IC50 = 710 nM T89988 C98JAY 44395129 IC50 = 40000 nM T89988 CJVK23 44395136 IC50 = 4200 nM T89988 CL9B7U 44395137 IC50 = 34000 nM T89988 C2JKO7 44395138 IC50 = 28000 nM T89988 CI74MR 44395143 IC50 = 41000 nM T89988 C8W7QA 44395144 IC50 = 14000 nM T89988 CQVF83 44395160 IC50 = 19000 nM T89988 C6PO5T 44395165 IC50 = 4000 nM T89988 C0UT4Q 44395169 IC50 = 33000 nM T89988 C58SKQ 44395186 IC50 = 4100 nM T89988 CP4WI3 44395194 IC50 = 12000 nM T89988 CQG0T2 44395195 IC50 = 26000 nM T89988 CC39VA 44395201 IC50 = 64000 nM T89988 CK4RW1 44395222 IC50 = 2400 nM T89988 C2O0XM 44395232 IC50 = 7900 nM T89988 CX81WJ 44395238 IC50 = 7800 nM T89988 C1KR3H 44395239 IC50 = 50000 nM T89988 CBT0O9 44395254 IC50 = 45000 nM T89988 CQC21H 44395256 IC50 = 16000 nM T89988 C72LSP 44413076 IC50 = 8 nM T89988 CG8VJ4 44413089 IC50 = 10 nM T89988 C6R8TI 44413137 IC50 = 865 nM T89988 C2FRX1 44413144 IC50 = 720 nM T89988 C5PA2Q 44413147 IC50 = 424 nM T89988 C03JIF 44413158 IC50 = 592 nM T89988 CXB7S3 44413167 IC50 = 1000 nM T89988 CA35QW 44413214 IC50 = 32 nM T89988 C0LT7X 44413230 IC50 = 1477 nM T89988 CV26LN 44413257 IC50 = 25 nM T89988 C0UL2N 44413258 IC50 = 13 nM T89988 C5J2IA 44413310 IC50 = 678 nM T89988 C39VOA 44413311 IC50 = 521 nM T89988 COD13L 44413328 IC50 = 342 nM T89988 C9EVF0 44413344 IC50 = 575 nM T89988 C07HRT 44413399 IC50 = 831.76 nM T89988 C7W8LI 44413411 IC50 = 756 nM T89988 C71QPH 44414578 IC50 = 1070 nM T89988 CW3V9I 44415864 IC50 = 48 nM T89988 CXQ4E0 44415880 IC50 = 4 nM T89988 CJYB82 44415898 IC50 = 38 nM T89988 CDV84J 44415899 IC50 = 13 nM T89988 C79IPU 44415900 IC50 = 244 nM T89988 CS51WY 44415903 IC50 = 129 nM T89988 CLHX29 44415904 IC50 = 42 nM T89988 CGX2M9 44415922 IC50 = 15 nM T89988 C8KU5F 44415927 IC50 = 216 nM T89988 CVF2X9 44415939 IC50 = 37 nM T89988 C4RCE6 44415942 IC50 = 462 nM T89988 C0FMC7 44415945 IC50 = 437 nM T89988 CYTL74 44415957 IC50 = 86 nM T89988 CYQE71 44415958 IC50 = 73 nM T89988 CKX2L3 44415973 IC50 = 37 nM T89988 CJ51SX 44415992 IC50 = 47 nM T89988 CI38AS 44415995 IC50 = 80 nM T89988 CP4DF0 44415996 IC50 = 298 nM T89988 CF4SD2 44416015 IC50 = 72 nM T89988 COX2Z8 44416041 IC50 = 72 nM T89988 CGKV54 44416066 IC50 = 125 nM T89988 CN8V6W 44416070 IC50 = 525 nM T89988 C5D9UT 44416125 IC50 = 805 nM T89988 C7P5KX 44416138 IC50 = 11 nM T89988 CVTL23 44416156 IC50 = 783 nM T89988 CVMS82 44416157 IC50 = 3 nM T89988 CYR56S 44416273 IC50 = 570 nM T89988 CE7K0V 44416274 IC50 = 213.8 nM T89988 C9OBD5 44421855 IC50 = 20000 nM T89988 CFKZ21 44421856 IC50 > 30000 nM T89988 C7N8YR 44421860 IC50 = 10000 nM T89988 CQW39E 44421862 IC50 = 6000 nM T89988 CQ07XN 44421867 IC50 = 1000 nM T89988 C7SL3R 44421868 IC50 = 5000 nM T89988 C7L2UB 44421888 IC50 = 6000 nM T89988 CUD80R 44421889 IC50 = 1000 nM T89988 C3K7NQ 44421913 IC50 = 1000 nM T89988 C7PCB4 44421917 IC50 = 1000 nM T89988 C5T6WC 44421922 IC50 = 3000 nM T89988 C87DBT 44421923 IC50 = 2000 nM T89988 CZ6DH9 44423281 IC50 = 65 nM T89988 CWJ3C4 44423282 IC50 = 7.5 nM T89988 CKX2F3 44423283 IC50 = 1.4 nM T89988 CJH60R 44423284 IC50 > 1000 nM T89988 CQ80SV 44423285 IC50 = 47 nM T89988 CNR96O 44425241 IC50 = 20 nM T89988 C1DO8P 44425242 IC50 = 9.1 nM T89988 CZ49XH 44425243 IC50 = 28.6 nM T89988 C9POR6 44425244 IC50 = 7.3 nM T89988 CW5B2T 44425245 IC50 = 1.3 nM T89988 CNPT74 44425247 IC50 = 182.7 nM T89988 C9VET7 44425249 IC50 = 5.2 nM T89988 CIK35U 44425250 IC50 = 1.8 nM T89988 C04TAL 44425252 IC50 = 3 nM T89988 CA64XV 44425254 IC50 = 0.7 nM T89988 C0L2CH 44425255 IC50 = 0.6 nM T89988 CK1QL4 44425256 IC50 = 32.7 nM T89988 CJS6E3 44425258 IC50 = 14.5 nM T89988 CHC0X9 44425271 IC50 = 4 nM T89988 CCB89O 44425272 IC50 = 3.5 nM T89988 C46TAL 44425273 IC50 = 3.9 nM T89988 C4N9YV 44425274 IC50 = 7.4 nM T89988 CZWS87 44425276 IC50 = 18 nM T89988 C49VPJ 44425277 IC50 = 16 nM T89988 CR0W5Q 44425279 IC50 = 2.6 nM T89988 CYA4L7 44425281 IC50 = 1.3 nM T89988 C4IE0H 44425283 IC50 = 36 nM T89988 CTH31J 44425286 IC50 = 14.3 nM T89988 CM4D6U 44425288 IC50 = 13.18 nM T89988 CHD4K8 44425290 IC50 = 3.5 nM T89988 C8EXT0 44425292 IC50 = 0.43 nM T89988 CW7E4Z 44425293 IC50 = 1.4 nM T89988 CAF01W 44425294 IC50 = 0.8 nM T89988 C9HNI1 44425304 IC50 = 13.18 nM T89988 CQ7W8I 44425305 IC50 = 229 nM T89988 CPY5O8 44425306 IC50 = 41.69 nM T89988 C59CGR 44425308 IC50 = 30 nM T89988 C7XI6U 44425309 IC50 = 6.5 nM T89988 CG7Z2F 44425310 IC50 = 5.8 nM T89988 C9H1OJ 44425315 IC50 = 13 nM T89988 CT75JS 44425316 IC50 = 17 nM T89988 C4JPK2 44425317 IC50 = 19 nM T89988 CJY1R8 44425318 IC50 = 23 nM T89988 C9DHM6 44425319 IC50 = 13 nM T89988 CG1J9N 44425320 IC50 = 14 nM T89988 CB1IP4 44425321 IC50 = 74 nM T89988 CTQ3W1 44425322 IC50 = 36 nM T89988 C54TVY 44425629 IC50 = 20 nM T89988 CET0P3 44425630 IC50 = 8.913 nM T89988 C2P8SI 44425631 IC50 = 10 nM T89988 CBI1A0 44425633 IC50 = 7.586 nM T89988 CQP64B 44425634 IC50 = 15.85 nM T89988 CQ4H3S 44425635 IC50 = 8 nM T89988 C3KSH7 44425636 IC50 = 20 nM T89988 CJI4T7 44425637 IC50 = 19 nM T89988 CH13ZK 44425638 IC50 = 231 nM T89988 CNY18R 44425639 IC50 = 15.5 nM T89988 C10GTR 44425640 IC50 = 6.5 nM T89988 C6GVI5 44425641 IC50 = 13 nM T89988 CM0SY9 44425642 IC50 = 28 nM T89988 C3T7DE 44425643 IC50 = 3.981 nM T89988 CQL1F7 44425644 IC50 = 3.3 nM T89988 C9PR2I 44425645 IC50 = 0.15 nM T89988 C1IGE8 44425646 IC50 = 5 nM T89988 C3W2SM 44425647 IC50 = 0.32 nM T89988 CXI0Y9 44425648 IC50 = 5.5 nM T89988 CDKA32 44425649 IC50 = 6.3 nM T89988 CQK4M8 44425650 IC50 = 27 nM T89988 CIH7T2 44425651 IC50 = 8.5 nM T89988 C8WXN5 44425652 IC50 = 0.23 nM T89988 CIKD64 44425653 IC50 = 3.5 nM T89988 CVW1F0 44425654 IC50 = 67 nM T89988 CT93GC 44439155 IC50 = 185 nM T89988 C58AVC 44439156 IC50 = 2840 nM T89988 CNW2K9 44439157 IC50 = 9332 nM T89988 CS5YO0 44439158 IC50 = 1123 nM T89988 C8GKW0 44439159 IC50 = 1803 nM T89988 CF6KR3 44439160 IC50 = 4741 nM T89988 CN7KQ2 44439163 IC50 = 118 nM T89988 C8QRF1 44439164 IC50 = 7601 nM T89988 CXNE20 44439166 IC50 = 43 nM T89988 C01KCX 44439169 IC50 = 106.91 nM T89988 C6PS5Z 44439170 IC50 = 52 nM T89988 CGYJ76 44439173 IC50 = 6475 nM T89988 CUT9L0 44441347 IC50 = 10 nM T89988 CAG6R0 44441352 IC50 = 10 nM T89988 CBY68G 44441356 IC50 = 180 nM T89988 CB28GP 44441358 IC50 = 120 nM T89988 CDI1Z6 44441359 IC50 = 170 nM T89988 CT4L3X 44441382 IC50 = 2050 nM T89988 CJTZ15 44441396 IC50 = 290 nM T89988 C4Z6BD 44442531 IC50 = 560 nM T89988 C2AY8H 44442532 IC50 = 110 nM T89988 C4D7BR 44442540 IC50 = 15000 nM T89988 CN3AK1 44442541 IC50 = 22000 nM T89988 CR5UZ7 44442542 IC50 = 3000 nM T89988 CAIO38 44442543 IC50 = 410 nM T89988 CA37EK 44442544 IC50 = 770 nM T89988 CB8UD0 44442547 IC50 = 150 nM T89988 CPH7V8 44442553 IC50 = 130 nM T89988 CSN9R7 44442554 IC50 = 120 nM T89988 C6Z4LR 44442555 IC50 = 120 nM T89988 C45LKM 44442556 IC50 = 190 nM T89988 CGI4O8 44442557 IC50 = 100 nM T89988 CW2Q1E 44442558 IC50 = 99 nM T89988 CWR41K 44442559 IC50 = 150 nM T89988 C6JA2N 44442560 IC50 = 200 nM T89988 C7CZI3 44442561 IC50 = 60 nM T89988 C1ASE4 44442562 IC50 = 260 nM T89988 CDNB78 44442563 IC50 = 490 nM T89988 CUNH60 44442564 IC50 = 750 nM T89988 CSK0B1 44442565 IC50 = 400 nM T89988 CDX9K1 44442566 IC50 = 380 nM T89988 CSRO45 44442569 IC50 = 7200 nM T89988 C3R4SV 44442570 IC50 = 1700 nM T89988 C1AK7V 44442571 IC50 = 1100 nM T89988 C98JQT 44442572 IC50 = 530 nM T89988 C3E8MO 44442573 IC50 = 430 nM T89988 CM62RJ 44442574 IC50 = 900 nM T89988 CB1D2L 44442575 IC50 = 160 nM T89988 CZ1Q3R 44442576 IC50 = 47 nM T89988 C23KHI 44442577 IC50 = 36 nM T89988 CX2U4T 44442578 IC50 = 36 nM T89988 CHA6Z3 44442580 IC50 = 670 nM T89988 CTE0Y1 44442581 IC50 = 120 nM T89988 CVC6E9 44442582 IC50 = 690 nM T89988 CHD74R 44442583 IC50 = 1300 nM T89988 C6F9PC 44442584 IC50 = 5600 nM T89988 CWCY76 44442586 IC50 = 720 nM T89988 C89VZB 44442587 IC50 = 39 nM T89988 C6W0XY 44442588 IC50 = 23 nM T89988 CD50ZB 44442589 IC50 = 65 nM T89988 C6M2TZ 44442590 IC50 = 240 nM T89988 C5Q7BK 44442591 IC50 = 90 nM T89988 C0GN4C 44442592 IC50 = 16 nM T89988 C93GZU 44442593 IC50 = 19 nM T89988 CRB1M8 44442594 IC50 = 110 nM T89988 C2B8QU 44442595 IC50 = 130 nM T89988 CO1F2A 44442596 IC50 = 310 nM T89988 CU43VX 44442598 IC50 = 37 nM T89988 C84AZN 44442599 IC50 = 20 nM T89988 CG8MC4 44443989 IC50 = 3100 nM T89988 C8TB1M 44443996 IC50 = 2900 nM T89988 CW9ML2 44444000 IC50 = 4500 nM T89988 CGN73S 44444001 IC50 = 1900 nM T89988 COJ91E 44444002 IC50 = 2300 nM T89988 CLW9O7 44444003 IC50 = 2600 nM T89988 C3G4RP 44444005 IC50 = 3800 nM T89988 CC50LS 44444006 IC50 = 3400 nM T89988 C8P6IQ 44444007 IC50 = 1800 nM T89988 C94CZJ 44444008 IC50 = 1200 nM T89988 C18RYD 44444009 IC50 = 2100 nM T89988 C3UJV4 44444032 IC50 = 1500 nM T89988 CI7ZK4 44444035 IC50 = 12600 nM T89988 C2NU7P 44444096 IC50 = 11100 nM T89988 CWB08Z 44444098 IC50 = 4000 nM T89988 CD82NB 44444099 IC50 = 320 nM T89988 CB9HW7 44444100 IC50 = 950 nM T89988 C2N9YB 44444102 IC50 = 510 nM T89988 CQ2U7T 44444103 IC50 = 2200 nM T89988 CJY6E1 44444104 IC50 = 2000 nM T89988 C9WUP6 44444105 IC50 = 5900 nM T89988 C27YJV 44444106 IC50 = 1400 nM T89988 C7I1MY 44444107 IC50 = 5200 nM T89988 C9R3XK 44444109 IC50 = 2900 nM T89988 CLV8O7 44444110 IC50 = 140 nM T89988 C2O0GB 44444111 IC50 = 180 nM T89988 CU7I5F 44444112 IC50 = 240 nM T89988 C8T6RW 44444113 IC50 = 130 nM T89988 C3VNH1 44444114 IC50 = 790 nM T89988 C98NMR 44446951 Ki = 1700 nM T89988 COP46Z 44447424 IC50 = 229.09 nM T89988 CW1Q8I 44447426 IC50 = 193 nM T89988 C4Y9JZ 44447427 IC50 = 204.17 nM T89988 COPZ27 44447429 IC50 = 14 nM T89988 CY5CA3 44447431 IC50 = 28.18 nM T89988 C0YB3Q 44447432 IC50 = 25.12 nM T89988 C0F8BO 44447433 IC50 = 281.84 nM T89988 C93BDA 44447434 IC50 = 285 nM T89988 CQ1PG4 44447435 IC50 = 125.89 nM T89988 CB9UO3 44447436 IC50 = 642 nM T89988 C49XWQ 44447446 IC50 = 229.09 nM T89988 CI8Q9M 44447766 IC50 = 3 nM T89988 C50JFH 44447775 IC50 = 4 nM T89988 CWY54R 44447782 IC50 = 6 nM T89988 C2UGM9 44447783 IC50 = 6 nM T89988 CSLU08 44447786 IC50 = 41 nM T89988 CRV6F7 44447789 IC50 = 45 nM T89988 CDI1F4 44447815 IC50 = 24 nM T89988 CMR4P3 44448776 IC50 = 50 nM T89988 CD3K4H 44448807 IC50 = 10 nM T89988 C12TPU 44448839 IC50 = 1 nM T89988 CB7F4C 44448879 IC50 = 1 nM T89988 CNPS37 44448915 IC50 = 2 nM T89988 C3UN9M 44448948 IC50 = 20 nM T89988 CUG0K5 44449030 IC50 = 20 nM T89988 CUV2A8 44449031 IC50 = 30 nM T89988 CV5G3U 44449054 IC50 = 2 nM T89988 C3NAM2 44449081 IC50 = 9 nM T89988 CIV30A 44449174 IC50 = 20 nM T89988 CU6M8T 44449175 IC50 = 80 nM T89988 CLB90E 44449204 IC50 = 2400 nM T89988 C6Q8HS 44449229 IC50 = 4800 nM T89988 CF5B8G 44453002 IC50 = 10000 nM T89988 CF0EB1 44453004 IC50 = 22000 nM T89988 C72NCT 44453133 IC50 > 10000 nM T89988 CEGW75 44453134 IC50 = 489 nM T89988 C9GNP8 44453171 IC50 = 473 nM T89988 C7PH5L 44453173 IC50 > 10000 nM T89988 CA0MZ6 44453203 IC50 > 5000 nM T89988 CALV41 44453204 IC50 > 5000 nM T89988 CSXO73 44453208 IC50 = 10000 nM T89988 C6G5AC 44453234 IC50 = 103 nM T89988 CESK25 44453268 IC50 = 305 nM T89988 C46MAN 44453298 IC50 = 5.5 nM T89988 C4ESA8 44453300 IC50 = 21 nM T89988 CH6C5F 44453325 IC50 = 53 nM T89988 CFH6C8 44453327 EC50 = 20 nM T89988 C0DM8U 44453329 IC50 = 121 nM T89988 C6M7IQ 44453330 IC50 = 21 nM T89988 CJV36D 44453365 IC50 = 5.3 nM T89988 CBNQ71 44453366 IC50 = 14 nM T89988 C2U5JW 44453368 IC50 = 6.1 nM T89988 C2JQ0A 44453369 IC50 = 2400 nM T89988 CI0PV7 44453370 IC50 = 2380 nM T89988 CV1E8J 44453372 IC50 = 59 nM T89988 CBCW46 44453373 IC50 = 35 nM T89988 CVC27Y 44453405 IC50 = 11 nM T89988 C1I9TO 44453407 IC50 = 20 nM T89988 CF8D2E 44453408 IC50 = 5.1 nM T89988 CE8X3Z 44453409 IC50 = 116 nM T89988 CBT74X 44453440 IC50 = 0.89 nM T89988 C9QKA4 44453441 IC50 = 116 nM T89988 CVL1R5 44453442 IC50 = 20 nM T89988 C06ICO 44453443 IC50 > 10000 nM T89988 CM9U2O 44453444 IC50 > 10000 nM T89988 C9Q1SV 44453471 IC50 = 43 nM T89988 CKX1I6 44453472 IC50 = 26 nM T89988 C3U2MW 44453473 IC50 = 643 nM T89988 CNT1L8 44453474 IC50 = 22 nM T89988 CPY9T6 44453475 IC50 > 10000 nM T89988 CY48QG 44453476 IC50 > 10000 nM T89988 CMBQ96 44453477 IC50 = 3100 nM T89988 C72HIV 44453505 IC50 > 5000 nM T89988 CEL4U0 44453507 IC50 = 74 nM T89988 CRZV62 44453533 IC50 = 730 nM T89988 CQ57XT 44453534 IC50 = 77 nM T89988 C2O5UN 44453535 IC50 = 300 nM T89988 CG0S3F 44453536 IC50 = 1360 nM T89988 C9X0RM 44453538 IC50 = 127 nM T89988 C8ZC4N 44453562 IC50 = 43 nM T89988 CBG8E7 44453563 IC50 = 2650 nM T89988 CMT4A6 44453565 IC50 = 630 nM T89988 CV85SI 44453587 IC50 > 10000 nM T89988 COK3C9 44453592 IC50 = 418 nM T89988 CWG31M 44453620 IC50 = 1550 nM T89988 C8ZA9E 44453621 IC50 > 10000 nM T89988 CY4ML1 44454793 IC50 = 115 nM T89988 CS2G0H 44454820 IC50 = 1.4 nM T89988 CT5N4E 44555481 IC50 > 50000 nM T89988 CQU5N6 44563038 IC50 = 1900 nM T89988 CR71SV 44563039 IC50 = 1300 nM T89988 CSQ4N3 44563071 IC50 = 960 nM T89988 CV2D1L 44563113 IC50 = 14 nM T89988 C5HIE4 44570713 IC50 = 112 nM T89988 C0OD7H 44570714 IC50 = 2 nM T89988 CQO26H 44570717 IC50 = 27 nM T89988 CF2N3O 44570718 IC50 = 7.7 nM T89988 C7ZYG6 44570779 IC50 = 135.7 nM T89988 C82AOH 44570780 IC50 = 227.5 nM T89988 CF56CE 44570781 IC50 = 23 nM T89988 CHB9E1 44571216 IC50 = 600 nM T89988 C2VC9W 44571218 IC50 = 4.8 nM T89988 CM4LZ8 44571257 IC50 = 19 nM T89988 CYCF52 44571258 IC50 = 61.5 nM T89988 C2OGV6 44573409 IC50 = 193.2 nM T89988 CZ4H9K 44573410 IC50 = 362 nM T89988 CGVT58 44573411 IC50 = 155.96 nM T89988 CYK18E 44573412 IC50 = 63.97 nM T89988 C09CJU 44573450 IC50 = 174.98 nM T89988 CKRY49 44573451 IC50 = 84.92 nM T89988 C6Z7DI 44573452 IC50 = 4.603 nM T89988 C3AG9N 44573485 IC50 = 4.6 nM T89988 C5OZX4 44573486 IC50 = 29.99 nM T89988 CR3XS9 44573487 IC50 = 35.97 nM T89988 C9FOB2 44573488 IC50 = 21.98 nM T89988 C9UH5E 44573535 IC50 = 630.96 nM T89988 CW7B8R 44573537 IC50 = 187 nM T89988 CO0FB9 44573538 IC50 = 187.07 nM T89988 CP9HC7 44573568 Ki = 50 nM T89988 C10UVI 44573569 IC50 = 418.79 nM T89988 C3RTY1 44573608 IC50 = 2.999 nM T89988 CWXH83 44573609 IC50 = 51 nM T89988 CBQ3N6 44573649 IC50 = 5.998 nM T89988 CCKN12 44573650 IC50 = 5.495 nM T89988 CYIP03 44573651 IC50 = 27.99 nM T89988 CQ2CP1 44573699 IC50 = 7 nM T89988 CBL9R6 44580424 IC50 = 1180 nM T89988 CD2V0I 44580590 IC50 = 4.3 nM T89988 C6MG8Q 44580591 IC50 = 6 nM T89988 CK78AN 44583280 IC50 = 24 nM T89988 CT78IF 44583281 IC50 = 6.5 nM T89988 CQI80O 44583282 IC50 = 16 nM T89988 C9KAN6 44583283 IC50 = 2.3 nM T89988 C8MIP6 44593554 IC50 = 1605 nM T89988 CTY83R 44593555 IC50 = 2 nM T89988 C9F8IU 44593561 IC50 = 3.3 nM T89988 C71ENV 44593562 IC50 = 238.78 nM T89988 CBR46V 44593563 IC50 = 0.3 nM T89988 CU7R2S 44593564 IC50 = 0.8 nM T89988 CSW0N7 44595711 IC50 = 11 nM T89988 C5IMW6 44612589 IC50 = 4500 nM T89988 C4D8RG 44612590 IC50 = 36 nM T89988 CU3C8Z 44612708 IC50 = 5779 nM T89988 CK3N1G 46206137 IC50 > 10000 nM T89988 CY2A9C 46240380 IC50 = 310 nM T89988 CIG71O 46240381 IC50 = 2700 nM T89988 CFY3L5 46240481 IC50 = 650 nM T89988 CPHB87 46240482 IC50 = 13 nM T89988 C8R1QX 46240484 IC50 = 60 nM T89988 CR0NX3 46240582 IC50 = 5300 nM T89988 CF9O5C 46240584 IC50 = 28 nM T89988 CV2X5E 46240585 IC50 = 70 nM T89988 CD1M3J 46240687 IC50 = 41 nM T89988 C63QWF 46240785 IC50 = 65 nM T89988 C3YU2T 46240895 IC50 = 36 nM T89988 CEH6U9 46241010 IC50 = 4 nM T89988 C43MLP 46241011 IC50 = 790 nM T89988 CJ7L3Z 46241120 IC50 = 100 nM T89988 C7PVU1 46241121 IC50 = 2820 nM T89988 CDZ3V6 46241509 IC50 = 56 nM T89988 CH8F5U 46241608 IC50 = 50 nM T89988 CD1H3B 46241609 IC50 = 250 nM T89988 CXJ7C5 46241610 IC50 = 17 nM T89988 C35CXM 46241611 IC50 = 71 nM T89988 C5Y8ZT 46241717 IC50 = 18 nM T89988 C8EX9T 46241718 IC50 = 43 nM T89988 CZK4H8 46241719 IC50 = 190 nM T89988 CK9H6B 46241720 IC50 = 170 nM T89988 CA05ZH 46241826 IC50 = 45 nM T89988 C3LD6V 46241827 IC50 = 220 nM T89988 CRJD47 46241829 IC50 = 190 nM T89988 C5TC2S 46830335 IC50 = 1.7 nM T89988 C1K7FL 46830336 IC50 = 3040 nM T89988 C5ZJM9 46842084 IC50 = 520 nM T89988 CPQ5E8 46842085 IC50 = 1730 nM T89988 C4Q6JH 46842086 IC50 = 750 nM T89988 CNX7H4 46842232 IC50 = 620 nM T89988 CU5W3P 46842233 IC50 = 3160 nM T89988 C5Y6MQ 46842235 IC50 = 660 nM T89988 CF8LO6 46842236 IC50 = 7520 nM T89988 CJDG46 46842381 IC50 = 1740 nM T89988 C2FE9H 46842382 IC50 = 6600 nM T89988 C1N4KX 46842383 IC50 = 580 nM T89988 CQN2H4 46865774 IC50 = 0.8 nM T89988 CPV2L4 46865775 IC50 = 0.5 nM T89988 CB8GE1 46884818 IC50 = 29 nM T89988 CHS4Q3 46884855 IC50 = 160 nM T89988 C4MQ0A 46884856 IC50 = 11 nM T89988 CCNT25 46884898 IC50 = 9 nM T89988 C3MSG2 46885027 IC50 = 9 nM T89988 CI5J4L 46885028 IC50 = 120 nM T89988 CA5W3K 46885029 IC50 = 170 nM T89988 C6QBR9 46885159 IC50 = 110 nM T89988 CMI8G7 46885160 IC50 = 1100 nM T89988 CB7XI0 46885213 IC50 = 2.6 nM T89988 CQ0M2Z 46885214 IC50 = 710 nM T89988 CB60AL 46885269 IC50 = 1860 nM T89988 C2VSQ4 46885270 IC50 > 10000 nM T89988 CLBQ50 46885271 IC50 > 10000 nM T89988 C1Z5OS 46886055 IC50 = 0.3 nM T89988 C7JO8A 46886056 IC50 = 51 nM T89988 CF83SA 46886057 IC50 = 4500 nM T89988 CA18BC 46886058 IC50 > 1000 nM T89988 CJ2U1P 46886059 IC50 = 284 nM T89988 C9QE0J 46886060 IC50 > 1000 nM T89988 CU9PR6 46886061 IC50 = 99 nM T89988 CNDL30 46886482 IC50 = 50 nM T89988 CTQ13P 46886507 IC50 = 311.5 nM T89988 C32NJX 46886508 IC50 = 278 nM T89988 CF8N0U 46886536 IC50 = 0.4 nM T89988 CZ59HO 46886537 IC50 = 151 nM T89988 C28IHA 46886538 IC50 = 3.5 nM T89988 C0UDN9 46886539 IC50 = 0.8 nM T89988 CK9E8N 46927116 IC50 = 36 nM T89988 C82HXR 46927117 IC50 = 7 nM T89988 CV28ZU 46944853 IC50 = 25 nM T89988 CT9P5G 46944854 IC50 = 32 nM T89988 CWH4K6 46944855 IC50 = 57 nM T89988 CC3O0S 46945254 IC50 = 35 nM T89988 C1UB8E 46945255 IC50 = 85 nM T89988 C4RZG5 46945857 IC50 = 44 nM T89988 CAK5J0 46946058 IC50 = 31 nM T89988 CY09UB 46946452 IC50 < 1000 nM T89988 CFH87K 46947816 IC50 = 13 nM T89988 CVEF51 49763568 IC50 = 5 nM T89988 C43LAE 49763569 IC50 = 390 nM T89988 CI6AR9 49763571 IC50 = 35 nM T89988 C78ICP 49763574 IC50 = 110 nM T89988 C65RMG 49763575 IC50 = 160 nM T89988 CQLN97 49763682 IC50 = 25 nM T89988 CY5ME3 49763685 IC50 = 80 nM T89988 C0ADU9 49763686 IC50 = 70 nM T89988 C1GVM0 49763804 IC50 = 61 nM T89988 C94ARN 49763931 IC50 = 21 nM T89988 C68SFM 49764196 IC50 = 22 nM T89988 CSW83Q 49764322 IC50 = 20 nM T89988 C1Z0UD 49764446 IC50 = 15 nM T89988 C5AD0E 49764447 IC50 = 21 nM T89988 C20WNR 49764700 IC50 = 210 nM T89988 CIZ86P 49764701 IC50 = 410 nM T89988 C95CPY 49798264 Ki = 251.19 nM T89988 C3SUN1 49798265 Ki = 31.62 nM T89988 CBG4T2 49798289 Ki = 125.89 nM T89988 C4HO3X 49798290 Ki > 3162.28 nM T89988 CK92RZ 49798291 Ki = 63.1 nM T89988 C70BOA 49798292 Ki = 39.81 nM T89988 C5LZJ7 49798323 Ki = 19.95 nM T89988 CX90YD 49798324 Ki > 3162.28 nM T89988 C8D3SA 49798325 Ki = 398.11 nM T89988 CMZT82 49798326 Ki = 630.96 nM T89988 CVD31B 49798327 Ki > 3162.28 nM T89988 CC42TS 49798347 Ki = 158.49 nM T89988 C4T3JR 49798348 Ki = 7.943 nM T89988 CQVG17 49798349 Ki = 3.162 nM T89988 C38JTB 49798350 Ki = 5.012 nM T89988 C94JQY 49798351 Ki = 398.11 nM T89988 C1WOS7 49798396 Ki = 794.33 nM T89988 CLD0Y3 49798397 Ki = 398.11 nM T89988 C3OMN2 49798398 Ki = 50.12 nM T89988 CG35HZ 49798399 Ki = 31.62 nM T89988 C3IDX4 49798434 Ki = 1.995 nM T89988 CQN90U 49798435 Ki = 1.585 nM T89988 CVG78D 49798436 Ki = 3.162 nM T89988 C62VRQ 49798437 Ki = 25.12 nM T89988 CR4FE3 49798438 Ki = 19.95 nM T89988 CY90CD 49798461 Ki = 10 nM T89988 CF8J6E 49798462 Ki = 12.59 nM T89988 C60QIU 49798463 Ki = 15.85 nM T89988 CD20QY 49798464 Ki = 199.53 nM T89988 CQP1H6 49798489 Ki = 50.12 nM T89988 CG42MY 49863167 IC50 = 2837.92 nM T89988 C9YB8V 49863168 IC50 = 9332.54 nM T89988 C41FAQ 49863199 IC50 = 1122.02 nM T89988 CTM2W6 49863200 IC50 = 1803.02 nM T89988 CQIV05 49863201 IC50 = 1224.62 nM T89988 C4SMG0 49863202 IC50 = 107.89 nM T89988 C6AP0W 49863225 IC50 = 42.95 nM T89988 C7JB8Z 50925394 IC50 = 0.95 nM T89988 C2T4IC 50991056 IC50 = 7.7 nM T89988 CI32TR 50992246 IC50 = 3 nM T89988 C8ICA4 51353692 IC50 > 10000 nM T89988 C4B0AF 51353693 IC50 > 10000 nM T89988 CX6B8U 52941377 IC50 = 2.9 nM T89988 CIBA52 52942863 IC50 = 120 nM T89988 C71MDG 52943756 IC50 = 7.4 nM T89988 CRKC87 52944966 IC50 = 17 nM T89988 CTF7Y6 52946110 IC50 > 1000 nM T89988 CRDI09 52947358 IC50 > 1000 nM T89988 CB4MN2 52947389 IC50 > 1000 nM T89988 CF9BQ7 52947417 IC50 = 649 nM T89988 CUFX45 52950180 IC50 = 47 nM T89988 CK0M6N 53317027 IC50 = 5 nM T89988 CT58US 53317028 IC50 = 3.2 nM T89988 C8BSM2 53317041 IC50 = 3.1 nM T89988 C8HO9F 53317526 IC50 = 221 nM T89988 CCN50W 53317527 IC50 = 232 nM T89988 C6FG7U 53318314 IC50 = 11.6 nM T89988 C5MFO3 53318315 IC50 = 13 nM T89988 C2PK1V 53318316 IC50 = 4.2 nM T89988 C0AS8E 53318853 IC50 = 2.5 nM T89988 C8K5QI 53318854 IC50 = 46.5 nM T89988 C1GH4U 53318855 IC50 = 116 nM T89988 C0VGT5 53319664 IC50 = 11.1 nM T89988 CZU3G0 53320171 IC50 = 22.7 nM T89988 CS2QA6 53320349 IC50 = 32 nM T89988 CI0R1F 53320350 IC50 = 17 nM T89988 CI2JU6 53320967 IC50 = 36.9 nM T89988 C1NAP2 53320968 IC50 = 130 nM T89988 CL0SO8 53320970 IC50 = 38.4 nM T89988 CNQ30U 53320973 IC50 = 4.3 nM T89988 C57FLU 53320974 IC50 = 75.9 nM T89988 C76HPL 53321427 IC50 = 45.5 nM T89988 C1HOS5 53321482 IC50 = 11.5 nM T89988 CW1TY6 53321483 IC50 = 10.6 nM T89988 C17BAO 53321484 IC50 = 27.6 nM T89988 CTHX71 53321503 IC50 = 18.5 nM T89988 CBJR38 53321615 IC50 = 39.5 nM T89988 CK2M9J 53321616 IC50 = 2.3 nM T89988 CFW3C6 53322299 IC50 = 14.6 nM T89988 CK2JD6 53322809 IC50 = 5.7 nM T89988 C35XLW 53322810 IC50 = 8.5 nM T89988 C8VM2O 53322811 IC50 = 9.3 nM T89988 C5BPW8 53322812 IC50 = 19.5 nM T89988 CYK8U9 53322813 IC50 = 294 nM T89988 C3JDS8 53322831 IC50 > 1000 nM T89988 CH6MZ9 53323653 IC50 = 3.5 nM T89988 C5J2DH 53323654 IC50 = 11.7 nM T89988 C3WY6T 53323664 IC50 = 15.2 nM T89988 CH3LK8 53324139 IC50 = 175 nM T89988 COYC36 53324140 IC50 = 46 nM T89988 C48XCJ 53324141 IC50 = 66 nM T89988 CO93PA 53324304 IC50 = 7 nM T89988 C09CEX 53324942 IC50 = 6.5 nM T89988 CHW4E1 53324943 IC50 = 12.8 nM T89988 CF93PO 53324944 IC50 = 17.5 nM T89988 C9YGA3 53325385 IC50 = 28 nM T89988 CM12CJ 53325460 IC50 = 3.2 nM T89988 CY15EU 53325639 IC50 = 6.2 nM T89988 CV4AO0 53326225 IC50 = 12.2 nM T89988 CU17IJ 53326226 IC50 = 14.7 nM T89988 C4N1PX 53326242 IC50 = 28 nM T89988 CHX40S 53326386 IC50 = 2.9 nM T89988 C5NS6A 53326645 IC50 = 17.3 nM T89988 CD1SK7 53326700 IC50 = 462 nM T89988 C8E0DF 53326701 IC50 = 15 nM T89988 C7PQ1Y 53326702 IC50 = 36 nM T89988 CRF7T6 53326703 IC50 = 34 nM T89988 CYH0F6 53326721 IC50 = 17 nM T89988 C2S5ZK 53326900 IC50 = 251 nM T89988 C6KP2D 53326901 IC50 = 13.9 nM T89988 CIT7E8 53389636 Ki = 3.467 nM T89988 CC8ME1 53389637 Ki = 1.9 nM T89988 CAH13N 53389641 Ki = 3.981 nM T89988 CM4U5G 53389660 Ki = 1.7 nM T89988 C13SIB 53389710 Ki = 2.291 nM T89988 CXW05M 53389845 Ki = 1.259 nM T89988 CS0Q8N 53389902 Ki = 0.4 nM T89988 C8GNX3 53389980 Ki = 16.6 nM T89988 C4AKQ1 54580188 IC50 = 18.3 nM T89988 CC72WM 54580189 IC50 = 68.6 nM T89988 C89MEB 54580190 IC50 = 15.5 nM T89988 CC3J5L 54581190 IC50 = 43.7 nM T89988 CG3HB9 54582215 IC50 = 40.1 nM T89988 C4KMX1 54582216 IC50 = 29.1 nM T89988 CD1AE2 54582217 IC50 = 20.9 nM T89988 CLX7U9 54583111 IC50 = 4.5 nM T89988 C3WZ9I 54583112 IC50 = 31.9 nM T89988 CYD20W 54583185 IC50 = 17.8 nM T89988 COQD25 54583186 IC50 = 9.2 nM T89988 CC19ZA 54583187 IC50 = 15.4 nM T89988 C9GFR1 54584109 IC50 = 500 nM T89988 C90AHI 54584164 IC50 = 28 nM T89988 CZ4S0B 54585107 IC50 = 18.3 nM T89988 C3TAR4 54585108 IC50 = 71.5 nM T89988 C8RTU2 54585109 IC50 = 19.7 nM T89988 CC6HY7 54586021 IC50 = 9.5 nM T89988 C7V0YA 54597147 Ki = 15 nM T89988 CGIP16 54754722 IC50 = 47 nM T89988 CX4LK5 54754723 IC50 = 86 nM T89988 C6LZ8B 54754724 IC50 = 32 nM T89988 CSA9I6 54754844 IC50 = 330 nM T89988 CEGJ53 54754845 IC50 = 510 nM T89988 C9NV8L 54754967 IC50 = 16 nM T89988 CI78YZ 54754968 IC50 = 2 nM T89988 CV3K8U 54754969 IC50 = 3 nM T89988 C6T8XS 54755079 IC50 = 12 nM T89988 CL2AU5 54755081 IC50 = 27 nM T89988 C2R6KO 54755083 IC50 = 63 nM T89988 C5LT0A 54755193 IC50 = 370 nM T89988 C3SD6W 54755560 IC50 = 7 nM T89988 C4GBT5 54755562 IC50 = 230 nM T89988 C0KZ4M 54755801 IC50 = 20 nM T89988 C2QP4W 54755919 IC50 = 20 nM T89988 CPWZ05 54756038 IC50 = 29 nM T89988 CJBW64 54756045 IC50 = 14 nM T89988 C0ZWL2 54756156 IC50 = 28 nM T89988 CFHI34 54768835 IC50 = 17 nM T89988 CLY35F 54768836 IC50 = 21 nM T89988 C9U4YQ 54768838 IC50 = 8 nM T89988 CO4FY1 54769305 IC50 = 15 nM T89988 CF39PC 54769752 IC50 = 19 nM T89988 CWN90Q 54771978 IC50 = 20 nM T89988 CUM4B5 54771980 IC50 = 5 nM T89988 CL7UD5 54772203 IC50 = 5 nM T89988 CH7K6J 54772204 IC50 = 7 nM T89988 C4E5YQ 54772205 IC50 = 7 nM T89988 C7Y8KR 54772206 IC50 = 7 nM T89988 C3UJ2D 56643545 IC50 = 4 nM T89988 C94RZF 56657929 IC50 = 19 nM T89988 COST81 56657930 IC50 = 4 nM T89988 C21NEQ 56659196 IC50 = 29 nM T89988 C7B9TW 56659197 IC50 = 33 nM T89988 CUM53N 56659295 IC50 = 20 nM T89988 C4IZL5 56661444 IC50 = 55 nM T89988 CQ25TB 56661451 IC50 = 7 nM T89988 CC3XP8 56661559 IC50 = 2600 nM T89988 C7K4TJ 56662695 IC50 = 7 nM T89988 C7SJH2 56664979 IC50 = 8 nM T89988 CC5S6K 56667036 IC50 = 45 nM T89988 C4X5DR 56668306 IC50 = 290 nM T89988 CF2N5W 56668309 IC50 = 82 nM T89988 C4SP2W 56668313 IC50 = 650 nM T89988 C31SKP 56668413 IC50 > 25000 nM T89988 CI5Y4E 56669631 IC50 = 200 nM T89988 CKV58T 56670477 IC50 > 25000 nM T89988 C34WPT 56671792 IC50 = 30 nM T89988 CXUJ14 56671793 IC50 = 11 nM T89988 C4UHW2 56671794 IC50 = 9 nM T89988 CG1JX9 56671795 IC50 = 11 nM T89988 CXIQ98 56671923 IC50 = 9 nM T89988 C19LWV 56671924 IC50 = 120 nM T89988 CE3Y0C 56671925 IC50 = 13 nM T89988 CET7K4 56672021 IC50 = 10000 nM T89988 CY26SL 56675205 IC50 = 6 nM T89988 C03LOT 56675300 IC50 = 530 nM T89988 CK9JX5 56675301 IC50 = 140 nM T89988 CU0H6Z 56675302 IC50 = 200 nM T89988 CR51UE 56676473 IC50 = 1400 nM T89988 C0KG7I 56676474 IC50 = 27 nM T89988 CBTG12 56677288 IC50 = 25 nM T89988 CU35WX 56677289 IC50 > 25000 nM T89988 C1E9CF 56677290 IC50 > 25000 nM T89988 CV23WU 56677291 IC50 > 25000 nM T89988 CCV03M 56677295 IC50 > 25000 nM T89988 CE3T1U 56677296 IC50 = 1200 nM T89988 CR8ZJ4 56678497 IC50 = 510 nM T89988 CD8IZ5 56678506 IC50 = 920 nM T89988 C7QW5F 56678507 IC50 = 14 nM T89988 C7MXE5 56678508 IC50 = 17 nM T89988 C2O4SY 56678640 IC50 = 2080 nM T89988 CKAU07 56680600 IC50 = 1000 nM T89988 C1BI5O 56681842 IC50 = 5400 nM T89988 CIW1T6 56683044 IC50 = 29 nM T89988 CKVB12 56683116 IC50 = 5 nM T89988 C0ZH9W 56683120 IC50 = 480 nM T89988 C9KMN5 56683121 IC50 = 37 nM T89988 CNS7H5 57335017 IC50 = 6.6 nM T89988 C6OX7Y 57343820 IC50 = 130 nM T89988 C3ME6N 57344218 IC50 = 190 nM T89988 CN0U5G 57344221 IC50 = 490 nM T89988 C6EGO0 57344296 IC50 = 36 nM T89988 C1GZ6S 57344297 IC50 = 270 nM T89988 C23CNI 57344298 IC50 = 64 nM T89988 CT92GZ 57344299 IC50 = 140 nM T89988 CBW8S6 57344303 IC50 = 16 nM T89988 C3ADF6 57344305 IC50 = 35 nM T89988 C5GV0P 57344307 IC50 = 83 nM T89988 C73ZNA 57344310 IC50 = 130 nM T89988 C9YZU2 57344314 IC50 = 900 nM T89988 C6MI0E 57344315 IC50 = 640 nM T89988 CVO80U 57344316 IC50 = 670 nM T89988 C4UC8E 57344317 IC50 = 980 nM T89988 CH7NM1 57344318 IC50 = 980 nM T89988 CI61XO 57391449 Ki = 40 nM T89988 CU39WF 57391450 Ki = 200 nM T89988 CW5GM2 57391487 IC50 = 950 nM T89988 CZOY39 57391591 IC50 = 6.6 nM T89988 CBEO41 57391765 IC50 = 7.3 nM T89988 CK9L1O 57391766 IC50 = 10.9 nM T89988 CN1Q4Y 57391767 IC50 = 2.7 nM T89988 CC53ND 57391768 IC50 = 7.8 nM T89988 CCZ85S 57391797 IC50 = 3700 nM T89988 CGR4B9 57392725 IC50 = 1878 nM T89988 CD97NH 57393218 Ki = 79 nM T89988 CF2WS8 57393219 Ki = 63 nM T89988 CRU9I7 57393220 Ki = 10 nM T89988 C3VI0X 57393248 IC50 > 25000 nM T89988 COE45G 57393249 IC50 = 740 nM T89988 C94QJG 57393347 IC50 = 12 nM T89988 CV4F2A 57393495 Ki = 63 nM T89988 C60XVA 57393496 Ki = 25 nM T89988 CW93MJ 57393497 Ki = 25 nM T89988 CHN9C0 57393530 IC50 = 59 nM T89988 CQW74A 57393531 IC50 = 310 nM T89988 CKJX42 57394938 Ki = 100 nM T89988 CA08MX 57394939 Ki = 631 nM T89988 CLFR28 57394966 IC50 = 25000 nM T89988 C4Y7BS 57394967 IC50 = 8600 nM T89988 CR37GS 57394968 IC50 = 9200 nM T89988 CY4JZ1 57394969 IC50 = 6000 nM T89988 C39SHX 57394970 IC50 = 15800 nM T89988 CC14HJ 57394971 IC50 > 25000 nM T89988 C7OF3Z 57395061 IC50 = 370 nM T89988 C3QCD9 57395216 IC50 = 9.3 nM T89988 C94MZO 57395217 IC50 = 3.2 nM T89988 CDIF34 57395218 IC50 = 2.6 nM T89988 C81ASJ 57395219 IC50 = 3 nM T89988 CD6F3G 57395221 Ki = 8 nM T89988 CKTL37 57396690 Ki = 794 nM T89988 CV9RJ7 57396722 IC50 = 5200 nM T89988 C7JOW2 57396723 IC50 = 2300 nM T89988 C5ZGD3 57396724 IC50 = 1300 nM T89988 CDY14H 57396725 IC50 = 1300 nM T89988 C6NPG0 57396726 IC50 = 11600 nM T89988 C0D3HL 57396832 IC50 = 130 nM T89988 CXB1F0 57396900 IC50 = 72 nM T89988 CH3CT2 57396901 IC50 = 27 nM T89988 CV4CN3 57396998 IC50 = 14 nM T89988 CO37CB 57396999 IC50 = 2.4 nM T89988 C5CYT8 57397001 Ki = 8 nM T89988 C7CHF8 57397013 IC50 = 4100 nM T89988 C9HF6A 57398458 Ki = 10 nM T89988 CK4E3W 57398492 IC50 > 25000 nM T89988 C3W1JY 57398493 IC50 = 9572 nM T89988 CO3UM0 57398494 IC50 = 1890 nM T89988 CQS9E4 57398590 IC50 = 340 nM T89988 CX8N3C 57398651 IC50 = 570 nM T89988 CYO6T8 57398750 IC50 = 4.9 nM T89988 CVF50W 57400125 Ki = 13 nM T89988 CH1KQ9 57400126 Ki = 13 nM T89988 CR09LY 57400127 Ki = 3 nM T89988 C6V8ET 57400128 Ki = 16 nM T89988 CNHU38 57400129 Ki = 2 nM T89988 C27JYV 57400160 IC50 = 50 nM T89988 CZ41PU 57400161 IC50 = 8100 nM T89988 CJ5X8T 57400162 IC50 > 25000 nM T89988 CV42YH 57400331 IC50 = 34 nM T89988 CWR51A 57400420 Ki = 4 nM T89988 C4O0ML 57400451 IC50 = 5.2 nM T89988 C2YVE5 57400452 IC50 = 12 nM T89988 C1N8YX 57401421 IC50 = 925 nM T89988 C67VKS 57401953 IC50 > 25000 nM T89988 C9SZ0F 57401954 IC50 = 38 nM T89988 CR6D1J 57402059 IC50 = 89 nM T89988 C2XM3P 57402124 IC50 = 180 nM T89988 CV54BI 57402219 IC50 = 1 nM T89988 CQ3JU8 57402220 IC50 > 1000 nM T89988 CE9TB4 57402254 IC50 = 2900 nM T89988 C5LG7S 57403699 IC50 = 2200 nM T89988 C8XIR4 57403700 IC50 = 1400 nM T89988 CG5X8H 57403701 IC50 > 25000 nM T89988 C5GI7L 57403755 IC50 > 25000 nM T89988 CRSG52 57403811 IC50 = 34 nM T89988 CJ2K4V 57403877 IC50 = 54 nM T89988 CM32RA 57656640 IC50 = 27 nM T89988 C0OJA5 57656641 IC50 = 17 nM T89988 CT8V9X 57656657 IC50 = 31 nM T89988 CH7BO0 57656701 IC50 = 5500 nM T89988 CMI4T3 57656713 IC50 = 64 nM T89988 CB30PQ 57656715 IC50 = 64 nM T89988 C51DOT 57656719 IC50 = 68 nM T89988 C2GHC7 57656729 IC50 = 2570 nM T89988 C6W3EJ 57656749 IC50 = 421 nM T89988 C1KAC6 57656808 IC50 = 797 nM T89988 CN7O1T 57656825 IC50 = 75 nM T89988 CHJ87A 57656833 IC50 = 3.5 nM T89988 CS6O1V 57656854 IC50 = 32 nM T89988 CPN5S4 57656869 IC50 = 262 nM T89988 CU8I2F 57656871 IC50 = 21 nM T89988 CD5W4E 57656887 IC50 = 202 nM T89988 C7NF4J 57656915 IC50 = 710 nM T89988 CQX1D5 57656921 IC50 = 58 nM T89988 C1QSF4 57656938 IC50 = 98 nM T89988 C5V0JI 57656942 IC50 = 220 nM T89988 C0YWT1 58509213 IC50 > 10000 nM T89988 CWFC53 59370257 IC50 = 0.65 nM T89988 CEB7T9 59370267 IC50 < 0.45 nM T89988 CN0C8R 60148505 IC50 = 6.5 nM T89988 CQR25M 66767933 IC50 < 0.45 nM T89988 CO62SG 66768099 IC50 < 0.45 nM T89988 CC81NU 66768640 IC50 = 4.9 nM T89988 C85HLV 67011331 IC50 = 3.4 nM T89988 C7CDA0 67220645 IC50 = 69 nM T89988 CC28AD 68003782 IC50 = 22 nM T89988 CXU2T6 68003962 IC50 = 15 nM T89988 C7ZA5Y 68003997 IC50 = 23 nM T89988 CQ4M8Y 68004002 IC50 = 40 nM T89988 CB7T0X 68004010 IC50 = 22 nM T89988 C9SZT4 68004011 IC50 = 19 nM T89988 C9BFS2 68004012 IC50 = 27 nM T89988 CX0B4G 68004016 IC50 = 38 nM T89988 C6U9NR 68004034 IC50 = 10 nM T89988 C8EM6J 68004094 IC50 = 72 nM T89988 CCO4A2 68004146 IC50 = 56 nM T89988 CFX59N 68070944 Ki = 24 nM T89988 C4D5IO 68616341 IC50 = 28 nM T89988 CCB1T5 68764898 IC50 = 0.24 nM T89988 C5O0JN 68764925 IC50 = 0.5 nM T89988 C70QJS 68767049 IC50 = 0.6 nM T89988 C8VU1C 68767078 IC50 = 2.7 nM T89988 C8XT7M 68767109 IC50 = 5.2 nM T89988 CP23JT 68767124 IC50 = 1.2 nM T89988 CKWJ72 68767577 IC50 = 0.2 nM T89988 C8U1DK 68767802 IC50 = 0.7 nM T89988 CS7T1U 68768752 IC50 = 2.2 nM T89988 CRM71Y 68768923 IC50 = 1.3 nM T89988 C6L3ZT 68769143 IC50 = 0.6 nM T89988 CHS3Z2 68769744 IC50 = 0.5 nM T89988 C2YRL3 68769802 IC50 = 3 nM T89988 C39SPK 68772423 IC50 = 0.9 nM T89988 C1UMP9 68867935 IC50 = 1.1 nM T89988 CWZU52 68988296 IC50 = 0.96 nM T89988 C5MP1I 69035439 IC50 = 1.2 nM T89988 CIU35O 69035677 IC50 = 1.9 nM T89988 C9UI0T 69212799 EC50 = 360 nM T89988 CPGC67 69285465 IC50 = 20 nM T89988 CM5XA1 69285531 IC50 = 13 nM T89988 C0QZ4U 69285563 IC50 = 33 nM T89988 C5T2GC 69285794 IC50 = 2.5 nM T89988 C8R4LZ 69286108 IC50 = 41 nM T89988 CNT95I 69286635 IC50 = 4.7 nM T89988 C1NY8Q 69315675 IC50 = 1700 nM T89988 C46QLW 69321774 IC50 = 440 nM T89988 CAU52S 70681271 IC50 = 158 nM T89988 C2K5HI 70681778 IC50 = 1055 nM T89988 CRZ9P2 70681779 IC50 > 10000 nM T89988 C8VE1I 70683350 IC50 = 3.8 nM T89988 CA1W4H 70683355 IC50 = 28000 nM T89988 CVUR18 70683619 IC50 = 860 nM T89988 C45LTY 70686028 IC50 > 10000 nM T89988 CSA38W 70687885 IC50 = 35 nM T89988 C4CI2T 70687886 IC50 = 84 nM T89988 CIS85H 70688149 IC50 = 26 nM T89988 C5M1GF 70689909 IC50 = 18 nM T89988 C9RDP5 70689914 IC50 = 11 nM T89988 C0QUO1 70689915 IC50 = 3.3 nM T89988 C7ESZ0 70691783 IC50 = 180 nM T89988 CTDY17 70691784 IC50 = 5 nM T89988 CNSJ34 70691785 IC50 = 10 nM T89988 C2GXN6 70692344 IC50 = 780 nM T89988 C3G7YH 70693849 IC50 = 10 nM T89988 CG7U4L 70696469 IC50 = 1458 nM T89988 CXS70G 70696470 IC50 = 449 nM T89988 C35YZQ 70697571 EC50 = 810 nM T89988 C5GM9Y 71190126 IC50 = 5 nM T89988 CG3DM1 71214709 Ki = 10 nM T89988 CG5V6I 71214710 Ki = 15.85 nM T89988 CA72CU 71214725 Ki = 39.81 nM T89988 CMSH09 71214976 Ki = 12.59 nM T89988 CRSA04 71226374 IC50 = 125 nM T89988 CSD6R9 71450657 Ki = 25.12 nM T89988 C8A0XW 71450658 Ki = 10 nM T89988 CW6C9V 71452241 IC50 = 33 nM T89988 C8YW2L 71452487 Ki = 100 nM T89988 C1TOE8 71452488 Ki = 50.12 nM T89988 C71FXH 71454246 Ki = 501.19 nM T89988 CD8I7C 71454247 Ki = 100 nM T89988 CSL01M 71454248 Ki = 12.59 nM T89988 C3EYK5 71456007 Ki = 1584.89 nM T89988 CHV16Z 71456008 Ki = 63.1 nM T89988 C6MHX5 71457815 Ki = 50.12 nM T89988 C3BXS9 71461438 Ki = 10 nM T89988 CRV73F 71461439 Ki = 100 nM T89988 C3P5HM 71461440 Ki = 31.62 nM T89988 C5E1FJ 71463165 Ki = 1258.93 nM T89988 C8VX0L 71463166 Ki = 251.19 nM T89988 CPU23H 71517239 IC50 = 4070 nM T89988 CLAF67 71517240 IC50 = 23 nM T89988 CYSI71 71517241 IC50 = 150 nM T89988 C8SR2Q 71517242 IC50 = 20 nM T89988 C4TGH7 71517401 IC50 = 45 nM T89988 CU28ZL 71517402 IC50 = 1258 nM T89988 C0BWE4 71517403 IC50 = 263 nM T89988 CU2TR7 71517573 IC50 = 59 nM T89988 C1XWC3 71517574 IC50 = 58 nM T89988 CZ5QD8 71517575 IC50 = 210 nM T89988 CGE96J 71517576 IC50 = 200 nM T89988 CFZ27L 71517577 IC50 = 8095 nM T89988 CK81FA 71517737 IC50 = 247 nM T89988 CVN31I 71518405 IC50 = 3300 nM T89988 CTL9E5 71518406 IC50 = 2329 nM T89988 C9V5RD 71518407 IC50 = 1529 nM T89988 CW39SU 71518408 IC50 = 699 nM T89988 CH5UM0 71518570 IC50 = 874 nM T89988 C6DIG9 71518571 IC50 = 3558 nM T89988 CZ0S5X 71518572 IC50 > 25000 nM T89988 CEJ1O6 71518573 IC50 > 25000 nM T89988 CQC14H 71518574 IC50 = 76 nM T89988 CXV79I 71518727 IC50 = 7927 nM T89988 CMKZ52 71518728 IC50 = 1070 nM T89988 CL05CZ 71518896 IC50 > 25000 nM T89988 C4UMA0 71518897 IC50 = 1100 nM T89988 C3Y2CP 71518898 IC50 = 200 nM T89988 CGO9T8 71519050 IC50 = 1500 nM T89988 CSU8J9 71519051 IC50 > 25000 nM T89988 C0E9LJ 71519052 IC50 = 5600 nM T89988 CK1GR7 71519053 IC50 = 4400 nM T89988 CGY45E 71519054 IC50 = 400 nM T89988 C29BZD 71519055 IC50 = 290 nM T89988 CR1IO9 71519224 IC50 = 34 nM T89988 CQ8F3O 71519225 IC50 = 1800 nM T89988 CE07SH 71519226 IC50 = 16 nM T89988 C2FE7Q 71519227 IC50 = 95 nM T89988 CP25YK 71519381 IC50 = 61 nM T89988 C3CT1R 71530223 IC50 = 22 nM T89988 C7XGD2 71552097 IC50 = 36 nM T89988 CQ31YB 71552260 IC50 = 39 nM T89988 CO3WL9 71552261 IC50 = 50 nM T89988 CU2R7W 71576618 Ki = 2.3 nM T89988 CI0GU8 71660496 IC50 > 48500 nM T89988 C5GE1T 71716742 IC50 = 88 nM T89988 CI8Q1K 71717723 Ki = 0.6 nM T89988 CP5NQ2 71718331 Ki = 1 nM T89988 CZ5C6V 71718930 Ki = 2 nM T89988 CC8JQ9 71719547 Ki = 1 nM T89988 CG30CF 71719764 IC50 = 130 nM T89988 CC80KL 71768688 IC50 = 16 nM T89988 CPX2W4 71768689 IC50 = 8.7 nM T89988 C4KUV6 71768721 IC50 = 62 nM T89988 CX39OE 71768722 IC50 = 2 nM T89988 CE5BJ7 71768725 IC50 = 16 nM T89988 C9NHU5 71768755 IC50 = 4 nM T89988 C65HBS 71768794 IC50 = 14 nM T89988 COE81F 71768798 IC50 = 59 nM T89988 C9ZKP0 71768830 IC50 = 29 nM T89988 CN9TQ3 71768831 IC50 = 330 nM T89988 CHQ15U 71768862 IC50 = 340 nM T89988 C8ERI3 71768864 IC50 = 27 nM T89988 C7ZY1J 71768865 IC50 = 1.5 nM T89988 C54JLD 71768897 IC50 = 370 nM T89988 CV53CZ 71768899 IC50 = 2130 nM T89988 CJY2C5 71768900 IC50 = 6.6 nM T89988 CKU6V5 71768931 IC50 = 35 nM T89988 C4EM1B 72945827 IC50 = 950 nM T89988 C1G5DP 72945830 IC50 = 69 nM T89988 C8RLE2 72946008 IC50 = 41 nM T89988 CDG6A2 72946010 IC50 = 99 nM T89988 C3N7RS 72946013 IC50 = 39 nM T89988 C37UZP 72946198 IC50 = 31 nM T89988 CF65HX 72946199 IC50 = 65 nM T89988 CI8Z0Q 72946200 IC50 = 82 nM T89988 C9FLS6 72946202 IC50 = 629 nM T89988 CA4L5S 72946204 IC50 = 126 nM T89988 CPA9G7 72946205 IC50 = 180 nM T89988 CF7WR3 72946381 IC50 = 28 nM T89988 CX82VR 72946384 IC50 = 1300 nM T89988 C7X2ZL 72946387 IC50 = 29 nM T89988 C16RLM 72946775 IC50 = 45 nM T89988 CP21YZ 72946982 IC50 = 118 nM T89988 CB51JH 72947191 IC50 = 87 nM T89988 CZR9S4 72947193 IC50 = 21 nM T89988 CMB52G 72947411 IC50 = 33 nM T89988 CN8U7J 72947413 IC50 = 395 nM T89988 CU9NB5 72947593 IC50 = 770 nM T89988 C7TIG1 72947595 IC50 = 27 nM T89988 CJQ04K 72948000 IC50 = 57 nM T89988 CO42FH 72948001 IC50 = 71 nM T89988 CFC70R 72948004 IC50 = 68 nM T89988 CXR6G5 73334813 Ki = 2.4 nM T89988 CT1RD0 73351183 EC50 = 630 nM T89988 CX9B4F 76167595 Ki = 2 nM T89988 CT2QF9 76314234 IC50 = 81 nM T89988 CSFB37 76314242 IC50 = 62 nM T89988 C2TLD8 76315270 IC50 = 10 nM T89988 CQT3F1 76321527 IC50 = 152 nM T89988 C8N9QM 76325121 IC50 = 1215 nM T89988 C1XL3H 76333441 IC50 = 39 nM T89988 C3Y0WL 76335990 IC50 = 300 nM T89988 CW1AZ2 86642531 IC50 = 0.13 nM T89988 C7TRY9 89844945 IC50 = 2.2 nM T89988 CE2Z4C 89845025 IC50 = 1.2 nM T89988 CTP94N 89845031 IC50 = 5 nM T89988 CN3DO5 89853102 IC50 = 1280 nM T89988 C9PSW7 90656015 IC50 = 5700 nM T89988 CTU8Z7 90656016 IC50 > 20000 nM T89988 C6N5DH 90656017 IC50 = 3170 nM T89988 CYTC65 90656018 IC50 > 20000 nM T89988 CZ1S2O 90656019 IC50 = 16100 nM T89988 C15QNG 90656020 IC50 = 2200 nM T89988 C3CAQ0 90656021 IC50 = 81 nM T89988 C6OI3C 90656022 IC50 = 180 nM T89988 C4FI1L 90656023 IC50 > 20000 nM T89988 CW4Z3B 90656024 IC50 > 20000 nM T89988 CK6QN4 90656025 IC50 = 30 nM T89988 CO73FL 90656026 IC50 = 190 nM T89988 COW7U5 90656027 IC50 = 0.25 nM T89988 C6ENV5 100951623 EC50 > 10000 nM T89988 CU29LP 118723021 Ki = 74 nM T89988 CZ1PV5 118723406 Ki = 270 nM T89988 CUGV43 118723408 Ki = 66 nM T89988 CK3S2X 118723411 Ki = 139 nM T89988 CP24GA 118723412 Ki = 90 nM T89988 CP10RK 118734571 Ki = 15 nM T89988 C2BWS4 118734572 Ki = 2.2 nM T89988 C75BLE 118734573 Ki = 31 nM T89988 CCP2L0 118734574 Ki = 4.6 nM T89988 C20SEZ 118734575 Ki = 15 nM T89988 CSOP75 118734576 Ki = 21 nM T89988 C8ZK9S 118734577 Ki = 4.9 nM T89988 CYOI62 118734578 Ki = 1.6 nM T89988 C94AOU 118734579 Ki = 4.4 nM T89988 CR8IY6 118734580 Ki = 13 nM T89988 C52KYS 118734581 Ki = 23 nM T89988 C5U1JI 118734582 Ki = 13 nM T89988 CDRN42 118734583 Ki = 7.9 nM T89988 C82WOS 118734584 Ki = 1.2 nM T89988 C50DNS 118734671 Ki = 49 nM T89988 CW7J0V 118734675 Ki = 55 nM T89988 CQ9N3Y 118734676 Ki = 11 nM T89988 CRJL05 118734678 Ki = 39 nM T89988 C52TGP 118734679 Ki = 75 nM T89988 C7RI8B 118734680 Ki = 10 nM T89988 CRF84D 118734681 Ki = 41 nM T89988 CGV9X0 118734682 Ki = 10 nM T89988 CAQ14V 118734683 Ki = 23 nM T89988 C47KNY 118734684 Ki = 12 nM T89988 CW08JS 118734685 Ki = 3.4 nM T89988 CIE93O 118734686 Ki = 2 nM T89988 C5K1DJ 118734687 Ki = 4.5 nM T89988 CNB69H 118734688 Ki = 13 nM T89988 CM9AJ8 118734689 Ki = 83 nM T89988 C1LNT2 118734690 Ki = 24 nM T89988 CG8FH2 118734691 Ki = 2 nM T89988 CT3MG4 118734692 Ki = 4.6 nM T89988 CRXS03 118734693 Ki = 199 nM T89988 CHPC27 118734694 Ki = 137 nM T89988 CA81LN 122178127 IC50 = 62 nM T89988 C2AWE9 122178128 IC50 = 1.8 nM T89988 CXN3E7 122181144 IC50 = 684 nM T89988 CQY5H1 122181145 IC50 = 7540 nM T89988 CJB1F7 122181146 IC50 = 1240 nM T89988 CM9PW3 122181147 IC50 = 180 nM T89988 C0V1MG 122181148 IC50 = 12000 nM T89988 C20HIU 122181149 IC50 = 318 nM T89988 CA0QB2 122181150 IC50 = 89 nM T89988 C1VM5E 122181151 IC50 = 462 nM T89988 CGRW01 122181152 IC50 = 163 nM T89988 C5KA8W 122181153 IC50 = 173 nM T89988 CYA7Z5 122181235 IC50 = 1600 nM T89988 CE5WF4 122181236 IC50 = 353 nM T89988 C8DC5N 122181237 IC50 = 6100 nM T89988 C0X6MH 122181238 IC50 = 17 nM T89988 CMOW05 127025086 IC50 = 1.2 nM T89988 CQD1C7 127025087 IC50 < 0.45 nM T89988 C2Y6EC 127025088 IC50 = 1.1 nM T89988 CGT84Q 127025089 IC50 = 9.2 nM T89988 CG32CV 127025091 IC50 = 41 nM T89988 CPU3B6 127025092 IC50 = 7.4 nM T89988 C5WC3V 127025093 IC50 = 1.7 nM T89988 CR5H4I 127025159 IC50 = 5406 nM T89988 CFL76Q 127025160 IC50 = 6605 nM T89988 CVJS82 127025444 IC50 = 9737 nM T89988 CZ80IQ 127025445 IC50 = 928 nM T89988 C7PY8T 127025446 IC50 = 284 nM T89988 CCWU81 127025447 IC50 = 254 nM T89988 C6BX2Y 127025448 IC50 = 1685 nM T89988 C1CE3P 127025460 IC50 = 150 nM T89988 C5AY2X 127025461 IC50 = 210 nM T89988 CWAU40 127025462 IC50 = 6151 nM T89988 C6XA7T 127025728 IC50 = 2637 nM T89988 CMXT79 127025729 IC50 = 3700 nM T89988 C57XLF 127025730 IC50 = 328 nM T89988 CHYK14 127026243 IC50 = 2.3 nM T89988 CL04JF 127027624 IC50 = 301 nM T89988 C8RK9W 127027625 IC50 = 744 nM T89988 CPUA26 127027626 IC50 = 3480 nM T89988 CL0DQ7 127027627 IC50 > 10000 nM T89988 C17CTI 127027628 IC50 = 114 nM T89988 CE45ZO 127027955 IC50 = 69 nM T89988 C1RSE3 127027956 IC50 = 249 nM T89988 C6SP7M 127028586 IC50 = 700 nM T89988 C71UIE 127028587 IC50 = 3418 nM T89988 C0ML7J 127028588 IC50 = 2967 nM T89988 C3YF7I 127028589 IC50 > 10000 nM T89988 CMJA67 127028590 IC50 = 1600 nM T89988 CU7DL4 127028591 IC50 = 8200 nM T89988 C7QWB2 127028592 IC50 = 438 nM T89988 CQ10RI 127029034 IC50 = 2.7 nM T89988 CPKQ90 127036603 IC50 = 550 nM T89988 CA4I9H 127036934 IC50 = 3700 nM T89988 CSD1X5 132572938 IC50 = 140 nM T89988 CK8XQ2 135981707 IC50 = 170 nM T89988 C9YAI3 136030597 IC50 > 10000 nM T89988 C2WT5B 137654404 IC50 = 3000 nM T89988 CGRA79 145953092 IC50 = 2502 nM T89988 C7ZFD4 145953762 IC50 = 638 nM T89988 CWVF94 145953765 IC50 = 3864 nM T89988 CQ2J5K 145954490 IC50 = 74 nM T89988 C0RE7W 145954949 IC50 = 336 nM T89988 C4BWN2 145955877 IC50 = 4936 nM T89988 CX96RN 145960485 IC50 = 720 nM T89988 C4R1XZ 145960924 IC50 = 7833 nM T89988 CW4N2T 145961260 IC50 = 1566 nM T89988 CB02GJ 145961667 IC50 = 19390 nM T89988 CKO9D2 145961759 IC50 = 1614 nM T89988 CD3IV4 145961961 IC50 = 1821 nM T89988 C32SJE 145961982 IC50 = 61 nM T89988 C4GL7Y 145962429 IC50 = 1261 nM T89988 CG3FT6 145962546 IC50 = 1731 nM T89988 C7Y8BD 145962575 IC50 = 390 nM T89988 C40AEX 145962604 IC50 = 5053 nM T89988 CNZ32U 145962608 IC50 = 550 nM T89988 CABC91 145962732 IC50 = 2466 nM T89988 CV8F3U 145963369 IC50 = 195 nM T89988 C72LVY 145963552 IC50 = 12330 nM T89988 C3UR2C 145963612 IC50 = 4450 nM T89988 CXR41S 145963669 IC50 = 2971 nM T89988 CFN4J8 145996522 Ki = 1.549 nM T89988 CXT09R 154572822 IC50 = 0.4 nM T89988 COP6C1 155491018 Ki = 0.3802 nM T89988 CVQ31N 155513284 Ki = 1.549 nM T89988 CW6CH0 155513605 Ki = 22.39 nM T89988 C7R1SZ 155513751 Ki = 316 nM T89988 CM7Y9H 155514261 IC50 = 8709.64 nM T89988 C70IOJ 155518928 Ki = 15.49 nM T89988 CMJU07 155520385 Ki = 4.074 nM T89988 CZ29FQ 155521447 Ki = 15 nM T89988 CN61LU 155522058 Ki = 51.29 nM T89988 CKX47L 155522874 Ki = 173.78 nM T89988 CBKQ30 155523645 Ki = 14.45 nM T89988 CW0R6Z 155526680 Ki = 213.8 nM T89988 CKR1O4 155527193 Ki = 20.89 nM T89988 C86OHR 155529593 IC50 = 1.9 nM T89988 CZ7TU0 155529754 Ki = 5.495 nM T89988 CCOP08 155530253 Ki = 154.88 nM T89988 CVS37C 155531379 IC50 = 1.4 nM T89988 C52QOY 155531561 Ki = 6.31 nM T89988 C0GAF2 155534565 Ki = 5.37 nM T89988 CF6DQ7 155535265 Ki = 158.49 nM T89988 CL0O2E 155535293 Ki = 3.467 nM T89988 CFDV10 155536512 Ki = 104.6 nM T89988 CE5SU4 155539148 Ki = 102.33 nM T89988 CK4I2Z 155540563 Ki = 288.4 nM T89988 CZ04TG 155540798 Ki = 2.188 nM T89988 CT9V0L 155541801 Ki = 2.951 nM T89988 CW71FQ 155543260 Ki = 3.467 nM T89988 C7FS8U 155545321 Ki = 12.88 nM T89988 C4J1ZL 155545804 Ki = 154.88 nM T89988 CRKZ36 155550777 Ki = 21.88 nM T89988 C03TXA 155551912 Ki = 2.089 nM T89988 CU32YB 155553131 Ki = 22.91 nM T89988 CYW9U3 155553573 Ki = 7.2 nM T89988 C3DB6L 155553917 Ki = 1.8 nM T89988 CT4NC3 155554106 Ki = 0.8318 nM T89988 C80LBZ 155554273 Ki = 0.6 nM T89988 C7X6VW 155559153 Ki = 66 nM T89988 C0TCG8 155560784 Ki = 2.455 nM T89988 C06NGD 155562719 Ki = 0.871 nM T89988 CF8JW6 155563012 Ki = 1.445 nM T89988 D0RM7J 44353447 IC50 = 17 nM T53904 D01SPD 69669724 IC50 = 480 nM T53904 D09NCT 53392492 IC50 = 54000 nM T53904 CMO39B 7493 Ki > 300000 nM T53904 CR85KY 10253 IC50 > 1000000 nM T53904 C5H7QS 9837038 IC50 = 91090 nM T53904 CUP73E 10103626 IC50 = 1000000 nM T53904 CM6Q3H 11788622 IC50 > 1000000 nM T53904 C4XC1Z 13548097 IC50 > 1000000 nM T53904 CYRZ62 15662041 IC50 = 24000 nM T53904 CCAM68 22959876 IC50 > 100000 nM T53904 C30EMN 24701909 IC50 = 18370 nM T53904 CZ8WG7 24831508 IC50 = 3.5 nM T53904 CUMF70 46899605 IC50 > 100000 nM T53904 C2DBN5 46899607 IC50 > 100000 nM T53904 C3G4QK 46899609 IC50 > 100000 nM T53904 CLK96Z 46899763 IC50 > 100000 nM T53904 CBOM64 46899765 IC50 > 100000 nM T53904 CA56RL 49831102 IC50 = 1.8 nM T53904 CU63QR 49847377 IC50 = 0.2 nM T53904 CZT4I8 49847378 IC50 = 0.3 nM T53904 CA72PE 49847379 IC50 = 1.1 nM T53904 CJ7H2B 49847753 IC50 = 1.4 nM T53904 C4V7EW 49848258 IC50 = 1.2 nM T53904 CP8TS6 49848895 IC50 = 0.3 nM T53904 C9COF5 49848896 IC50 = 0.3 nM T53904 CK0B1G 49848897 IC50 = 0.2 nM T53904 CP61VJ 49849002 IC50 = 0.3 nM T53904 C42SBF 49849005 IC50 = 1.4 nM T53904 CBM62Z 49849007 IC50 = 0.4 nM T53904 C05SEW 49849008 IC50 = 0.2 nM T53904 C78SAD 49849115 IC50 = 2.1 nM T53904 CF64IJ 49849120 IC50 = 0.2 nM T53904 CC9EB4 49849122 IC50 = 0.4 nM T53904 C2ORV5 49849123 IC50 = 6 nM T53904 CU7O4S 52942802 IC50 = 500000 nM T53904 C28RDF 54746913 IC50 = 3.6 nM T53904 C35JDV 54746961 IC50 = 3.6 nM T53904 CDL06K 54746964 IC50 = 2.4 nM T53904 C34DJP 57384236 IC50 = 0.8 nM T53904 CEOC15 57384237 IC50 = 2.1 nM T53904 CY50WC 57384238 IC50 = 2.3 nM T53904 C7S0ZR 57384239 IC50 = 1.8 nM T53904 C2XN1G 57384481 IC50 = 1.1 nM T53904 CR73IZ 57384482 IC50 = 0.7 nM T53904 CR2M5H 57384483 IC50 = 0.3 nM T53904 CQ72HI 57384749 IC50 = 3.7 nM T53904 C68KGE 57384750 IC50 = 1.6 nM T53904 CVK29R 57386523 IC50 = 1.7 nM T53904 C9S8MU 57386524 IC50 = 1.4 nM T53904 CMC8H6 57386782 IC50 = 1.1 nM T53904 CCT5D4 57386783 IC50 = 0.2 nM T53904 CC30XZ 57386784 IC50 = 8.2 nM T53904 C79BXP 57386785 IC50 = 0.9 nM T53904 CM6DV7 57387028 IC50 = 1.2 nM T53904 C0GS4F 57387282 IC50 = 0.3 nM T53904 C0TL9C 57387283 IC50 = 0.8 nM T53904 CRV2P5 57387539 IC50 = 0.2 nM T53904 CAU3G9 57387540 IC50 = 0.3 nM T53904 CL2AO8 57387541 IC50 = 0.3 nM T53904 C0XWL8 57387542 IC50 = 0.4 nM T53904 CC4DK0 57387775 IC50 = 1 nM T53904 C8DB9I 57387776 IC50 = 1 nM T53904 C73OLG 59186234 IC50 = 240 nM T53904 CCB65L 59603622 IC50 = 480 nM T53904 C4VU7J 70688210 IC50 = 5.5 nM T53904 CO7H3Q 71133989 IC50 = 2.1 nM T53904 C7K3JM 89812866 IC50 = 240 nM T53904 CUX19J 117632648 IC50 = 30000 nM T53904 CSEB74 117705981 IC50 = 570 nM T53904 CI5X2G 118978277 IC50 = 6.8 nM T53904 CH7WL3 118978299 IC50 = 11 nM T53904 CB3I9Z 118978325 IC50 = 6.3 nM T53904 CWH4I0 118978339 IC50 = 14 nM T53904 C6XD3H 118978341 IC50 = 3.3 nM T53904 CDBK07 118981498 IC50 = 2.2 nM T53904 CB23LS 118981525 IC50 = 12 nM T53904 C9F6RL 118981536 IC50 = 6.2 nM T53904 CF1E6T 118981546 IC50 = 11 nM T53904 C1ABC5 118981554 IC50 = 3.7 nM T53904 CR05OQ 118981555 IC50 = 5 nM T53904 CE9U5L 118981600 IC50 = 2.4 nM T53904 CO5XH7 118981638 IC50 = 4.9 nM T53904 CV84HB 118981731 IC50 = 3.1 nM T53904 CW89CV 118982285 IC50 = 3.8 nM T53904 C51RST 121245332 IC50 = 3.2 nM T53904 C2LI6C 121245745 IC50 = 5.9 nM T53904 C27WIY 121246694 IC50 = 27 nM T53904 C71YRT 121246805 IC50 = 2.3 nM T53904 CJU6X7 121246821 IC50 = 1.4 nM T53904 C1X3HT 121246837 IC50 = 4.9 nM T53904 C2UY6K 121246848 IC50 = 2.1 nM T53904 CRO04U 122540293 IC50 = 280 nM T53904 CQ5R9P 122540295 IC50 = 57 nM T53904 CB9K4N 122540308 IC50 = 34 nM T53904 C5ZIL1 122540317 IC50 = 67 nM T53904 C1KS9O 122540318 IC50 = 770 nM T53904 CPN71M 122540325 IC50 = 90 nM T53904 C5BFA8 122540341 IC50 = 1800 nM T53904 CPZ8I3 122540362 IC50 = 140 nM T53904 C6IEP4 122540388 IC50 = 50 nM T53904 CJ0RB3 122540392 IC50 = 39 nM T53904 CTG8N2 122540437 IC50 = 140 nM T53904 C6S2RC 122540446 IC50 = 13 nM T53904 CO34NP 122540461 IC50 = 1280 nM T53904 CZ0OW9 122540496 IC50 = 220 nM T53904 C6XL8K 122540512 IC50 = 3900 nM T53904 C81EIY 122540553 IC50 = 1370 nM T53904 C1ZMX3 122540617 IC50 = 10 nM T53904 C2EFG9 122540625 IC50 = 670 nM T53904 CK81UQ 122540630 IC50 = 8 nM T53904 C8K1DC 122540636 IC50 = 84 nM T53904 CTCL51 122540637 IC50 = 170 nM T53904 CD3VP5 122540661 IC50 = 6100 nM T53904 CI2ZX4 122540667 IC50 = 1870 nM T53904 CZ8M5Q 122540675 IC50 = 550 nM T53904 C3DOK6 122540683 IC50 = 74 nM T53904 CM1X0A 122540685 IC50 = 830 nM T53904 CLV75P 122540689 IC50 = 52 nM T53904 C38VFM 122540702 IC50 = 140 nM T53904 CAIU61 122540718 IC50 = 460 nM T53904 C1QXU7 122540722 IC50 = 25 nM T53904 C2LK0Y 122540724 IC50 = 34 nM T53904 CS61XJ 122540744 IC50 = 200 nM T53904 CYC48U 122540745 IC50 = 160 nM T53904 C1VOT7 122540750 IC50 = 460 nM T53904 CLT3K0 122540759 IC50 = 70 nM T53904 CG9T1H 134328388 IC50 = 270 nM T53904 CT57ZH 136069450 IC50 = 0.2 nM T53904 CFT9R3 136069453 IC50 = 0.5 nM T53904 CRPQ42 136069494 IC50 = 1.3 nM T53904 CK8Z3V 136069521 IC50 = 1.9 nM T53904 CPY1B2 136069522 IC50 = 17 nM T53904 CX0OM4 136069523 IC50 = 11 nM T53904 C6EU4D 136069524 IC50 = 38 nM T53904 CQA2Z1 136069531 IC50 = 4.5 nM T53904 CCH31A 136069532 IC50 = 0.4 nM T53904 CH8GV7 136069561 IC50 = 5.6 nM T53904 CQ1FS4 136069563 IC50 = 2 nM T53904 CQTB32 136205798 IC50 = 1.1 nM T53904 CV8QP3 136205832 IC50 = 0.2 nM T53904 CB93EM 136205833 IC50 = 0.5 nM T53904 C23FVD 137633446 IC50 > 100000 nM T53904 CPU1L2 137636406 IC50 = 5600 nM T53904 C8TN4G 137636671 IC50 = 55000 nM T53904 CG3F4E 137637795 IC50 > 100000 nM T53904 C1M6HB 137638932 IC50 = 2500 nM T53904 CFB79N 137641310 IC50 = 80000 nM T53904 C0DTF7 137641650 IC50 > 10000 nM T53904 C6PRQ9 137641829 IC50 > 10000 nM T53904 C34MZN 137642369 IC50 > 100000 nM T53904 CC7JI6 137646003 IC50 = 24000 nM T53904 C8NLW2 137648088 IC50 = 48000 nM T53904 CGX30Y 137648213 IC50 = 26000 nM T53904 CEWP67 137648313 IC50 > 10000 nM T53904 C78LJT 137649345 IC50 > 10000 nM T53904 CJ76HR 137649729 IC50 > 10000 nM T53904 C9AJ4B 137652165 IC50 > 10000 nM T53904 CU2IS6 137653429 IC50 = 9600 nM T53904 C25TUJ 137653793 IC50 > 10000 nM T53904 CD8HL9 137655479 IC50 > 10000 nM T53904 CWG40Z 137655745 IC50 > 10000 nM T53904 C9C3RJ 137657820 IC50 = 1300 nM T53904 C5DV0L 137658554 IC50 > 10000 nM T53904 C4XQH5 137659524 IC50 = 18000 nM T53904 CVB05O 137660951 IC50 = 28000 nM T53904 CD7LE9 137661677 IC50 = 61000 nM T53904 C2TB0E 137662021 IC50 = 26000 nM T53904 CG7R3L 155559901 IC50 = 3.2 nM T53904 D07IOY 10365 IC50 = 1500 nM T53904 D08IZY 3080614 IC50 = 842 nM T58449 D03ZBT 11626560 IC50 > 10000 nM T58449 D05SBO 46220502 IC50 = 300 nM T58449 D00UZR 5330286 IC50 > 10000 nM T58449 D05ADP 160355 IC50 = 480 nM T58449 D0CY1B 6420138 Ki > 10000 nM T58449 D0LF1U 5287969 IC50 = 875 nM T58449 D0S5RC 3025986 IC50 = 62 nM T58449 CB9F1O 447961 Ki = 70 nM T58449 C6A3LY 447962 Ki = 4012 nM T58449 CVX20F 9842276 IC50 = 1300 nM T58449 CVE1W8 10024433 Ki = 2804 nM T58449 C1KX3P 10248401 Ki > 10000 nM T58449 C9J3RM 10320107 Ki = 1080 nM T58449 CMY9D2 10340715 Ki > 10000 nM T58449 CC3L8Z 10430000 Ki > 10000 nM T58449 C69HPR 11257553 Ki = 2.3 nM T58449 CIWA03 11632150 Ki = 243 nM T58449 CEV5X2 11646645 Ki = 171 nM T58449 C2CVI7 11647020 Ki = 1395 nM T58449 C93KHF 11718021 Ki = 370 nM T58449 CJSV21 11744184 Ki > 10000 nM T58449 CCX39H 15979015 IC50 = 11000 nM T58449 CBV7T6 15979138 IC50 = 1000 nM T58449 CI5Q2D 15979261 IC50 = 410 nM T58449 C3ZC4Y 15979393 IC50 = 480 nM T58449 C6Z4CR 15979397 IC50 > 10000 nM T58449 C4D5UF 15979518 IC50 = 260 nM T58449 C1JMA7 15979519 IC50 > 2000 nM T58449 CARL15 15979630 IC50 > 3700 nM T58449 CXYU20 15979633 IC50 > 10000 nM T58449 CQD02P 15979747 IC50 > 10000 nM T58449 C8MGY5 15979751 IC50 = 210 nM T58449 CF9SK3 15979868 IC50 = 170 nM T58449 C7UEG5 15980106 IC50 = 160 nM T58449 CPJY86 15980107 IC50 = 705 nM T58449 CU87FW 15980108 IC50 > 10000 nM T58449 CQH37B 15980109 IC50 = 340 nM T58449 CB7JU8 15980233 IC50 > 10000 nM T58449 C7BS2R 16037674 IC50 > 10000 nM T58449 CB2H4D 16037675 IC50 = 530 nM T58449 C42DYS 16091079 IC50 > 20000 nM T58449 C5VPH9 16129448 IC50 = 2730 nM T58449 CQHK69 23646624 IC50 = 1500 nM T58449 C7YG1N 24759534 IC50 = 30 nM T58449 C4EG8R 24993189 IC50 > 10000 nM T58449 C5HZF2 44413509 IC50 = 20 nM T58449 C3D4FG 44413527 IC50 = 190 nM T58449 C3VRO9 44557921 IC50 > 10000 nM T58449 CGO1J5 46830766 Ki = 4240 nM T58449 CF7HK2 46830767 Ki = 2556 nM T58449 C2HJ1X 46830768 Ki = 2149 nM T58449 CKL1V8 49798556 IC50 > 20000 nM T58449 CCL3R5 49867929 IC50 = 21 nM T58449 C1DV2B 56932125 IC50 = 1760 nM T58449 C2VK6A 57404485 IC50 = 2100 nM T58449 CK6T1C 57404486 IC50 = 350 nM T58449 CQ80BX 57404487 IC50 = 317 nM T58449 CR1B9I 57867443 IC50 > 10000 nM T58449 C42IGJ 57867446 IC50 = 910 nM T58449 C18QUW 57867482 IC50 = 870 nM T58449 CIZ91X 57867490 IC50 = 960 nM T58449 C1VFJ8 57867505 IC50 = 940 nM T58449 C3Z5KS 57867516 IC50 > 10000 nM T58449 CFB7Q4 57867522 IC50 > 10000 nM T58449 CXJ63M 59603829 IC50 = 53 nM T58449 CQEU96 59603842 IC50 = 4.1 nM T58449 C37NKO 67129970 IC50 > 10000 nM T58449 CK80LJ 67130050 IC50 > 10000 nM T58449 C7GRV2 68755406 IC50 > 10000 nM T58449 CM8LY4 70681104 IC50 > 10000 nM T58449 CHC4P3 70685325 IC50 > 10000 nM T58449 C49QWD 70691636 IC50 = 26 nM T58449 CBE67N 71731769 IC50 < 5 nM T58449 CYG95S 72707651 IC50 = 1876 nM T58449 CNP0V5 72707724 IC50 = 1788 nM T58449 CU4A5Q 72707728 IC50 = 1645 nM T58449 CZAM98 72707790 IC50 = 1642 nM T58449 CP13FK 72707853 IC50 = 1423 nM T58449 C7VA5U 78161839 IC50 = 0.13 nM T58449 C2Y1RF 78162193 IC50 < 5 nM T58449 C4NM0V 78162195 IC50 < 5 nM T58449 CWR57U 78357763 IC50 = 27 nM T58449 C1HW4B 89735655 IC50 < 10 nM T58449 C8W9KV 91844733 IC50 = 40 nM T58449 CQCX41 118737057 IC50 > 10000 nM T58449 C4WGC7 119081415 IC50 = 194 nM T58449 C2BEH5 121443990 IC50 > 100 nM T58449 CP4Q7B 121444083 IC50 = 20 nM T58449 C9MIL3 122188249 IC50 = 841 nM T58449 C53AYQ 122188250 IC50 > 10000 nM T58449 CZO41H 122188251 IC50 > 10000 nM T58449 CLW25J 122188252 IC50 = 9244 nM T58449 C23PIE 122188253 IC50 > 10000 nM T58449 CE41KZ 122188254 IC50 > 10000 nM T58449 CHQT85 122188255 IC50 > 10000 nM T58449 CLAD59 122188256 IC50 > 10000 nM T58449 C3BXR2 122188258 IC50 > 10000 nM T58449 C67GYV 122188259 IC50 > 10000 nM T58449 CG8VX5 122188261 IC50 > 10000 nM T58449 C9ZKA1 122188262 IC50 > 10000 nM T58449 CQF9I2 122188263 IC50 > 10000 nM T58449 COGF57 122188264 IC50 > 10000 nM T58449 CPQ89G 122188266 IC50 = 3590 nM T58449 CVEB28 122188271 IC50 = 8750 nM T58449 C5E7WK 122188272 IC50 > 10000 nM T58449 CWIR28 122188273 IC50 > 10000 nM T58449 CB6I5A 122188274 IC50 > 10000 nM T58449 CA8VH1 122188275 IC50 = 1811 nM T58449 C2D5TF 122188281 IC50 > 10000 nM T58449 C93VST 122188282 IC50 = 1680 nM T58449 C4X7SD 122192466 IC50 > 10000 nM T58449 CM0A3E 124134260 IC50 < 100 nM T58449 COF75Z 126970673 IC50 = 300 nM T58449 C1SP3H 127030849 IC50 = 2780 nM T58449 CDJQ32 127051599 IC50 = 21 nM T58449 C1MTG5 134543905 IC50 = 20 nM T58449 C37ITY 135414445 IC50 = 6500 nM T58449 C5AG7L 135414460 IC50 = 56 nM T58449 CLXB05 135438541 IC50 = 300 nM T58449 CR48OH 135468068 IC50 = 39 nM T58449 CPE67T 135487516 IC50 = 11 nM T58449 CJ4V0A 135508121 IC50 = 310 nM T58449 C2JA3F 135520167 IC50 = 180 nM T58449 C25MKU 135559056 IC50 = 1300 nM T58449 CHW54V 135559057 IC50 = 4900 nM T58449 C4CJG9 135559058 IC50 > 100000 nM T58449 CCQ4J8 135559059 IC50 = 25 nM T58449 CDN21F 135559061 IC50 = 34 nM T58449 C8BJV6 135559062 IC50 = 18 nM T58449 CS4HA0 135559063 IC50 = 4000 nM T58449 C2BHG0 135559064 IC50 = 57 nM T58449 CMF9Y8 135559065 IC50 = 420 nM T58449 C61XZP 135559066 IC50 = 2300 nM T58449 CPC03V 135559067 IC50 = 480 nM T58449 C8G2TS 135559068 IC50 = 7000 nM T58449 CI1E8V 137634241 IC50 > 10000 nM T58449 CVU63L 139582016 IC50 = 3100 nM T58449 C8PH9S 139582017 IC50 = 17000 nM T58449 CR2GW6 145994117 IC50 = 3600 nM T58449 CYHW79 155530843 IC50 = 20 nM T58449 C1IHY8 155533514 IC50 > 200 nM T58449 C8OC5N 155537111 IC50 < 20 nM T58449 CETH36 155557337 IC50 < 20 nM T58449 CLXN40 155565350 IC50 = 193 nM T58449 D00ERW 44444843 Ki > 1525 nM T58449 D01MNK 25125014 IC50 = 250 nM T58449 D02QAZ 11612883 IC50 = 197 nM T58449 D03DZO 11715767 IC50 > 10000 nM T58449 D0LO5B 73602827 IC50 = 3.2 nM T58449 D0YZ7H 9797370 IC50 = 56700 nM T15139 CD74LR 292706 Ki = 27000 nM T15139 CGA5F2 346675 IC50 = 57500 nM T15139 CTHK18 895402 IC50 = 5600 nM T15139 C3M0VW 1838078 IC50 > 100000 nM T15139 C2GL0X 1869842 IC50 < 50000 nM T15139 CDT51Y 1951286 IC50 < 50000 nM T15139 C9N5XB 2026662 IC50 > 100000 nM T15139 CGX7T5 2120805 IC50 > 100000 nM T15139 CO9Y3Z 4355463 IC50 = 6800 nM T15139 CXS9F6 4566836 IC50 = 5400 nM T15139 CKZ7V6 4674993 IC50 = 7000 nM T15139 C9ID6V 4912070 IC50 > 100000 nM T15139 C1O3RJ 5010967 IC50 = 37200 nM T15139 CV8FZ1 6875399 IC50 = 35700 nM T15139 C1KF4O 8615611 IC50 > 57000 nM T15139 CFX96S 15544085 IC50 = 6600 nM T15139 CMV5X1 17011425 IC50 > 100000 nM T15139 CBXC05 24424330 IC50 = 8700 nM T15139 CF9J3R 49852772 IC50 = 37000 nM T15139 C9QSP2 49852889 IC50 = 8900 nM T15139 C4HU6B 49852897 IC50 = 11000 nM T15139 CYZC96 49852943 IC50 = 6400 nM T15139 C7AEH1 49853067 IC50 = 14000 nM T15139 C47SDM 49853091 IC50 = 10000 nM T15139 CES9G3 49853100 IC50 = 13000 nM T15139 C78HFB 49853142 IC50 = 37000 nM T15139 CU21EH 49853203 IC50 > 57000 nM T15139 C64EUF 49853209 IC50 = 6300 nM T15139 C2ZN7D 49853294 IC50 = 5300 nM T15139 C6ZCA3 49853368 EC50 = 17500 nM T15139 CYIC61 53257121 IC50 = 21000 nM T15139 CKA74G 101879233 IC50 = 68900 nM T15139 CMLW04 102205482 IC50 = 22800 nM T15139 C6W2ZN 118796328 EC50 = 2300 nM T15139 CMO57H 118947294 IC50 < 50000 nM T15139 C0X8KJ 118947349 IC50 > 100000 nM T15139 CBOS58 118947388 IC50 > 100000 nM T15139 CU53JP 118947412 IC50 < 50000 nM T15139 C1XZF7 118947462 IC50 > 100000 nM T15139 CB39WZ 118947481 IC50 > 100000 nM T15139 C8RCS4 118947495 IC50 > 100000 nM T15139 CN5J3Z 118947501 IC50 = 50000 nM T15139 CIZ72P 118947502 IC50 < 50000 nM T15139 CB4W1C 118947563 IC50 < 50000 nM T15139 C5MH7P 118947571 IC50 < 50000 nM T15139 C3PJB8 121485232 IC50 = 50000 nM T15139 C7BJ6G 121485242 IC50 = 10000 nM T15139 C91HSG 121485258 IC50 = 21000 nM T15139 CFIH36 121485269 IC50 = 8700 nM T15139 CEDA24 122418186 IC50 = 33000 nM T15139 C26VJM 130407999 IC50 = 30 nM T15139 C7P5EJ 130408291 IC50 = 10 nM T15139 CY65ND 130418263 IC50 = 153 nM T15139 CV1U2H 130429937 IC50 = 88100 nM T15139 CQ6AI9 130429939 IC50 = 160700 nM T15139 C6SFT7 130429940 IC50 = 9300 nM T15139 CR27LM 130429942 IC50 > 200000 nM T15139 CD5F7E 130429947 IC50 > 200000 nM T15139 C0MVF4 130429950 IC50 > 100000 nM T15139 CT48EP 130429983 IC50 > 200000 nM T15139 CHB9F5 130429986 IC50 > 100000 nM T15139 C18LPS 130429999 IC50 > 200000 nM T15139 C94VCX 130430007 IC50 > 200000 nM T15139 CNGD28 130430011 IC50 > 200000 nM T15139 C8LUX7 130430025 IC50 > 200000 nM T15139 CUE3P2 134429273 IC50 = 31000 nM T15139 CQAO64 134429274 IC50 = 8300 nM T15139 CW06KT 134429275 IC50 = 5800 nM T15139 CO2P5Y 134429276 IC50 = 9900 nM T15139 C5AD7I 134429279 IC50 = 12000 nM T15139 C5DS8E 134437716 IC50 = 19000 nM T15139 C8MWK9 134437740 IC50 = 5700 nM T15139 CW0DZ5 134437744 IC50 = 6300 nM T15139 C5NDX1 134437746 IC50 = 41000 nM T15139 C8T6YN 134437750 IC50 = 22000 nM T15139 CD8B6U 134437753 IC50 = 30000 nM T15139 CEL49B 134437755 IC50 = 20000 nM T15139 CPT52N 134437756 IC50 = 20000 nM T15139 C3OYN0 134437757 IC50 = 17000 nM T15139 C2OT5L 134437812 IC50 = 26000 nM T15139 CO8Q3N 134437824 IC50 = 15000 nM T15139 CH90ED 134437828 IC50 = 40000 nM T15139 C3ML0D 134437829 IC50 = 39000 nM T15139 CMS49R 134437832 IC50 = 38000 nM T15139 CXI18Q 134437838 IC50 = 9200 nM T15139 C3GPI7 134437841 IC50 = 11000 nM T15139 CMX8P1 134437848 IC50 = 11000 nM T15139 C8SW4G 134437869 IC50 = 6500 nM T15139 C8NKX2 134437870 IC50 = 11000 nM T15139 CCV31P 134437872 IC50 = 10000 nM T15139 CPNO39 134437877 IC50 = 7200 nM T15139 CVM23J 134437914 IC50 = 7700 nM T15139 CZQB64 134437925 IC50 = 17000 nM T15139 CY4AV9 135403154 IC50 = 34800 nM T15139 CTK6F0 136937731 IC50 > 100000 nM T15139 CBX7R0 137522167 IC50 = 1400 nM T15139 CR5O3C 137647070 IC50 > 100000 nM T15139 C3GKP5 137651355 IC50 > 100000 nM T15139 CS3QB9 137655343 IC50 > 100000 nM T15139 C21INE 137657956 IC50 > 100000 nM T15139 CG5HS1 138753630 Ki = 214 nM T15139 CVM80R 138756828 IC50 = 100 nM T15139 C8QC5T 138756829 IC50 = 400 nM T15139 CPR5Y3 138756830 IC50 = 300 nM T15139 CG3L7H 138756831 IC50 = 3 nM T15139 CV3D1R 138911337 IC50 = 2000 nM T15139 C21PYB 142427688 IC50 = 8 nM T15139 CZC62Y 142427749 IC50 = 4 nM T15139 CU4T6V 145960504 IC50 = 8000 nM T15139 CHX5N9 145960596 IC50 = 9700 nM T15139 CT9XH5 145960621 IC50 = 21000 nM T15139 CI40NB 145960758 IC50 = 4300 nM T15139 C7RW0X 145960898 IC50 = 23000 nM T15139 CU1IK7 145961091 IC50 = 50000 nM T15139 CNY09E 145961156 IC50 = 15000 nM T15139 C3P8LH 145961174 IC50 = 16000 nM T15139 CHQ56V 145961472 IC50 = 7300 nM T15139 C0T6SZ 145961708 IC50 = 59000 nM T15139 CP4LA9 145962107 IC50 = 24000 nM T15139 CAC5D9 145962456 IC50 = 14000 nM T15139 CY2KN7 145962789 IC50 = 8700 nM T15139 C3U9VD 145963193 IC50 = 12000 nM T15139 CS49BK 145963368 IC50 = 16000 nM T15139 CM64FH 145963685 IC50 = 7300 nM T15139 C96DLG 155510912 IC50 = 2500 nM T15139 C7VUG8 155512349 IC50 = 72 nM T15139 CSCH29 155513145 IC50 = 14 nM T15139 C32NXU 155515150 IC50 = 3300 nM T15139 CZ19YB 155516063 IC50 = 1580 nM T15139 CDK81A 155516285 IC50 = 15 nM T15139 CL2W0D 155516426 IC50 = 5200 nM T15139 CE2P4T 155516866 IC50 = 53800 nM T15139 CIAJ65 155516908 IC50 = 81 nM T15139 CWCT76 155517908 IC50 > 100000 nM T15139 CCN07T 155517974 IC50 = 287 nM T15139 CB2HW7 155518094 IC50 = 100 nM T15139 CZJ72G 155518421 IC50 = 6700 nM T15139 CK15XH 155518761 IC50 = 2368 nM T15139 CRH20E 155519110 IC50 > 100000 nM T15139 C24BQW 155522173 IC50 = 23200 nM T15139 C1NH8X 155523199 IC50 = 34 nM T15139 C73NSI 155525342 IC50 = 37 nM T15139 CY90TS 155525802 IC50 = 58 nM T15139 C2XIY9 155526005 IC50 = 39600 nM T15139 C7Q1EB 155526382 IC50 = 33000 nM T15139 C72UBT 155526686 IC50 = 25 nM T15139 CMGW68 155526835 IC50 = 22000 nM T15139 CM02HQ 155527973 IC50 = 1294 nM T15139 C0AUE1 155528104 IC50 = 2300 nM T15139 CB92UN 155529283 IC50 = 23400 nM T15139 CA58ZG 155531601 IC50 = 235 nM T15139 C17OHV 155532142 IC50 = 38100 nM T15139 CION96 155534368 IC50 = 30 nM T15139 CN12SJ 155535053 IC50 = 12100 nM T15139 CJN2M3 155536090 IC50 = 301 nM T15139 CB6D3O 155536637 IC50 > 100000 nM T15139 CT7L3S 155536748 IC50 = 1330 nM T15139 C6ND9J 155536777 IC50 = 5200 nM T15139 C4KTE5 155537075 IC50 = 51 nM T15139 C6LEK7 155537339 IC50 = 5700 nM T15139 CT5YL8 155537379 IC50 > 100000 nM T15139 CLB65J 155537992 IC50 > 100000 nM T15139 CTP4L0 155538389 IC50 = 900 nM T15139 C5GP6H 155538643 IC50 = 25 nM T15139 CS38OJ 155538775 IC50 = 1300 nM T15139 CKGW41 155541540 IC50 = 55400 nM T15139 CUT17I 155542117 IC50 = 4300 nM T15139 CT42PF 155542308 IC50 = 824 nM T15139 CXQ9T4 155542332 IC50 = 1400 nM T15139 C94XQG 155542973 IC50 = 28 nM T15139 C4D5ZQ 155544502 IC50 = 3100 nM T15139 C0OTJ1 155544677 IC50 = 209000 nM T15139 C1M4ZS 155545662 IC50 = 439 nM T15139 C86AEZ 155546222 IC50 > 100000 nM T15139 C3DON9 155546449 IC50 = 16200 nM T15139 CDM02P 155547534 IC50 = 42100 nM T15139 C2YUJ1 155550274 IC50 = 11700 nM T15139 CM8WK4 155550368 IC50 > 100000 nM T15139 C47GNZ 155552547 IC50 = 22000 nM T15139 C42UCY 155553773 IC50 = 235 nM T15139 CX16DK 155554240 IC50 = 70 nM T15139 C49EHO 155555646 IC50 = 12200 nM T15139 CNI86P 155556782 IC50 = 990 nM T15139 CWLB78 155557800 IC50 = 33700 nM T15139 CF03HW 155558291 IC50 = 341 nM T15139 CEIJ65 155558670 IC50 > 100000 nM T15139 C20MVN 155559066 IC50 = 1950 nM T15139 CMQP04 155559154 IC50 = 800 nM T15139 CD60PE 155559613 IC50 = 5830 nM T15139 CF4LH0 155562166 IC50 = 6000 nM T15139 C27QFZ 155562355 IC50 = 370 nM T15139 C3MN6X 155563952 IC50 = 21500 nM T15139 C5BP6R 155567916 IC50 = 100000 nM T15139 COJ5M8 155569162 IC50 = 1460 nM T15139 CU8K5P 155569553 IC50 = 28 nM T26368 D06ZII 969472 Ki > 15000 nM T26368 D07JVL 3016 Ki = 15 nM T26368 D0L9GG 2118 EC50 = 10 nM T26368 D0T1WN 5732 EC50 > 3000 nM T26368 D02XYB 3058746 IC50 = 4.6 nM T26368 D0CH7C 57336276 Ki = 4.7 nM T26368 D0HO2T 23581869 Ki = 230 nM T26368 D0Z9HW 23630026 Ki = 1680 nM T26368 C1W5EF 114888 Ki = 0.85 nM T26368 C7SZ9E 613843 IC50 > 10000 nM T26368 C12NWX 2729103 IC50 > 10000 nM T26368 CO61AF 2820320 IC50 > 10000 nM T26368 C59BWK 2820473 IC50 > 10000 nM T26368 CCX58U 9865233 Ki = 1.1 nM T26368 C7BA0Z 9908880 Ki = 2.3 nM T26368 CPC3U1 9971547 Ki = 6 nM T26368 CUSM85 10221761 Ki = 33.3 nM T26368 C15NXT 10926766 EC50 = 650 nM T26368 CK1S7J 10927005 EC50 = 375 nM T26368 CWK02D 10936672 EC50 = 94 nM T26368 C09PCZ 10971225 EC50 = 323 nM T26368 CJB1V2 11035207 EC50 = 291 nM T26368 CBV36I 11047145 EC50 = 231 nM T26368 CWO70Q 11673720 Ki = 2 nM T26368 CL4XD0 11783674 EC50 = 74 nM T26368 CTI32Y 15680235 EC50 = 1000 nM T26368 CZK75V 44364548 EC50 = 439 nM T26368 C0FN6W 44364725 EC50 = 112 nM T26368 CE8F3Y 44364734 EC50 = 90 nM T26368 COH5G6 44364735 EC50 = 111 nM T26368 C2VHW7 44364747 EC50 = 491 nM T26368 CZL2P0 44364907 EC50 = 38 nM T26368 CCX08E 44364918 EC50 = 346 nM T26368 C6J0GP 44561356 IC50 = 210 nM T26368 C9UW4V 44561357 IC50 = 550 nM T26368 CZR6A5 44561358 IC50 > 10000 nM T26368 C4IF7B 44561386 IC50 = 1000 nM T26368 C0PC5E 44561389 Ki = 83 nM T26368 CP5WT1 44561431 Ki = 500 nM T26368 CPJC74 44561432 Ki = 0.65 nM T26368 C0L1FI 44561433 Ki = 9.8 nM T26368 C4S7HF 44561434 Ki = 2610 nM T26368 CB4I1E 44561435 Ki = 166 nM T26368 C6J7DH 44561436 Ki > 300 nM T26368 CO2QA8 44561437 Ki = 182 nM T26368 CDN1A9 44561475 Ki = 369 nM T26368 CN24OF 46229639 Ki = 2364 nM T26368 C1BZN5 71584335 Ki = 24.9 nM T26368 CQ91VU 118278442 Ki = 7.9 nM T26368 CH0D4J 130439777 Ki = 55 nM T26368 C56XBU 130439778 Ki = 5000 nM T26368 C9N8LW 130439889 Ki = 79 nM T26368 C89LNZ 136118605 IC50 = 201 nM T26368 D06SOQ 6918451 Ki = 0.66 nM T26368 D09IHE 6918583 Ki = 1.4 nM T26368 D0E7PY 11624499 Ki = 4.6 nM T26368 D0M4CP 5081 Ki = 3.1 nM T26368 D0O9MG 5311203 Ki = 0.45 nM T25956 D02YNI 9936746 IC50 > 33000 nM T25956 D07SDQ 969516 IC50 = 6500 nM T25956 D0M2TS 71600087 IC50 = 63 nM T25956 D0PH9I 118693659 Ki < 10000 nM T25956 D0U2BH 65064 IC50 = 30000 nM T25956 CM2RK5 67254 IC50 = 118500 nM T25956 CK5QD7 73588 IC50 = 4850 nM T25956 CQ8A5W 91330 IC50 = 13700 nM T25956 CX16AI 122042 IC50 = 260 nM T25956 CHU6D4 343829 IC50 = 106000 nM T25956 CXCB27 393166 IC50 = 2430 nM T25956 CHR5Q8 395862 IC50 = 8280 nM T25956 CH1DM6 769739 IC50 = 6200 nM T25956 CO8HA9 832572 IC50 = 2600 nM T25956 COJ29X 890649 IC50 = 11000 nM T25956 CGZ7Y8 900269 IC50 = 14000 nM T25956 CM2Z5Q 1285941 Ki = 400 nM T25956 CS96HU 1367211 IC50 = 1800 nM T25956 CG1I7T 1550234 IC50 = 111000 nM T25956 CJWR09 1561807 IC50 = 81000 nM T25956 CS05BM 1600566 IC50 = 244100 nM T25956 C4EZ0H 1652812 IC50 = 660 nM T25956 C5DXU9 1797299 IC50 = 700 nM T25956 C6XQA3 1797300 IC50 = 700 nM T25956 CBIP78 2133789 IC50 = 1100 nM T25956 C8E9HY 2221149 IC50 = 1980 nM T25956 CBK1D6 2295854 IC50 = 2200 nM T25956 C4T8OV 2325816 IC50 = 8030 nM T25956 C1YZ8I 2327942 IC50 = 9350 nM T25956 CTVG84 2328663 IC50 = 8140 nM T25956 COTE61 2408437 IC50 = 24700 nM T25956 C1LNM0 2467794 IC50 = 12900 nM T25956 CZE13I 2816786 IC50 = 6740 nM T25956 C5F2BD 2854538 IC50 = 150000 nM T25956 CQUY78 2871948 Ki = 400 nM T25956 CAY86S 3312427 IC50 = 6200 nM T25956 C54MWY 3493274 IC50 = 1100 nM T25956 CG8F2A 3683950 IC50 = 15200 nM T25956 CMK3Q0 3801109 IC50 = 2800 nM T25956 CWJ93L 5124087 IC50 = 3700 nM T25956 C13OPQ 5352088 IC50 = 7000 nM T25956 C4FKS8 5467476 IC50 = 233000 nM T25956 CG1LV3 7333990 IC50 > 50000 nM T25956 CK4GM7 7574135 IC50 = 3000 nM T25956 CSX8V7 7897116 IC50 = 510 nM T25956 C2FM4R 9875131 IC50 = 5000 nM T25956 CH41UK 9992116 IC50 = 5350 nM T25956 C7NT2X 10311918 IC50 = 275000 nM T25956 CUD8X4 10355367 IC50 = 5710 nM T25956 C2QTW8 11052198 IC50 = 23000 nM T25956 C6EMN5 11114773 IC50 = 5000 nM T25956 CCTY51 11135781 Ki = 3900 nM T25956 C8OCA4 12005893 IC50 = 1800 nM T25956 CXP5S8 12006282 IC50 = 2000 nM T25956 C7U9KW 13099766 IC50 = 5740 nM T25956 C29QHR 13374635 IC50 = 1100 nM T25956 CP82EX 14117443 IC50 = 1900 nM T25956 C1ZIE7 16203604 IC50 = 168000 nM T25956 CW6TU0 16203606 IC50 = 5000 nM T25956 C1DM9I 18783165 IC50 = 95000 nM T25956 CWS8N7 22121498 IC50 = 1100 nM T25956 CI0FB7 24320099 IC50 = 1000 nM T25956 C46RLS 42609873 IC50 = 3000 nM T25956 C6Q7IJ 44564009 IC50 = 28000 nM T25956 CO3UF4 44564514 IC50 = 9900 nM T25956 CRK2E6 44564516 IC50 = 14400 nM T25956 C52BJH 44571034 IC50 = 3.2 nM T25956 C6BQ2N 44580829 Ki = 5100 nM T25956 CU46TX 45032907 IC50 = 7500 nM T25956 C87QKN 50899265 IC50 = 70 nM T25956 CG3PR6 52912222 IC50 = 31622.78 nM T25956 C4XCJ0 53257845 IC50 = 5920 nM T25956 CBOE48 56669892 IC50 = 5320 nM T25956 C6I7VX 60201924 IC50 < 5000 nM T25956 C1X7DC 60201925 IC50 < 5000 nM T25956 C6YD5U 60201926 IC50 = 5000 nM T25956 CLGW91 60201927 IC50 < 5000 nM T25956 CI3MA8 60201928 IC50 < 5000 nM T25956 C5OPX2 60201929 IC50 < 5000 nM T25956 CPR3T5 60201930 IC50 = 5000 nM T25956 C8EDT9 60202083 IC50 < 5000 nM T25956 CJTM92 60202084 IC50 < 5000 nM T25956 CCX28H 60202085 IC50 = 5000 nM T25956 CZ47SK 60202086 IC50 = 5000 nM T25956 C2Q0NP 60202087 IC50 < 5000 nM T25956 CD84NS 71481176 IC50 = 11 nM T25956 CBX37Z 72201043 IC50 = 58000 nM T25956 CX9CV2 76853637 IC50 = 57500 nM T25956 CQ1V6U 86302322 IC50 = 9190 nM T25956 CS3W6O 90667751 IC50 = 61900 nM T25956 CZBD29 90667752 IC50 = 151900 nM T25956 CF4W8Q 90667754 IC50 = 95300 nM T25956 CTA46H 91826273 Ki = 2000 nM T25956 CM9Y5S 102127780 IC50 = 3300 nM T25956 C8ZVB6 118734156 IC50 = 9800 nM T25956 CB58PX 118735300 IC50 = 2100 nM T25956 C6J0QZ 118735301 IC50 = 1600 nM T25956 CM29SP 118735302 IC50 = 5900 nM T25956 CIKU37 118735303 IC50 = 1500 nM T25956 C2CQ5J 118735304 IC50 = 11400 nM T25956 CPH4W9 118735305 IC50 = 8000 nM T25956 C96FHE 118735307 IC50 = 8500 nM T25956 CYWS40 118735308 IC50 = 5400 nM T25956 CA8P3R 118735309 IC50 = 31400 nM T25956 C0UR4G 118735310 IC50 = 4200 nM T25956 C6NI1C 118735317 IC50 = 26400 nM T25956 C3TG2V 118735320 IC50 = 1600 nM T25956 C0QY8M 118958122 IC50 = 60 nM T25956 CUWX94 119081692 IC50 = 270 nM T25956 CB83MK 121271792 IC50 = 51 nM T25956 CDH8M4 121373418 IC50 = 1.3 nM T25956 C47QXT 121376807 IC50 = 30 nM T25956 C7PRX6 124351359 IC50 = 750 nM T25956 CC1AX6 125920038 IC50 = 45000 nM T25956 C8C1ZL 126458860 IC50 = 3400 nM T25956 CD3AJ2 126797002 IC50 = 3700 nM T25956 CV4D8T 127030247 IC50 = 7000 nM T25956 CLB9N0 127033602 IC50 = 5000 nM T25956 CPIG89 127033885 IC50 = 22 nM T25956 CU2O8R 127045845 IC50 = 14100 nM T25956 CGDN94 132275066 IC50 = 1.2 nM T25956 CY46VZ 135423665 IC50 = 3100 nM T25956 C4KDT9 135457159 IC50 > 50000 nM T25956 CPY8E7 139341516 IC50 = 4000 nM T25956 C3HJI2 139341518 IC50 = 26900 nM T25956 CWK82L 139341520 IC50 > 33000 nM T25956 C3DGA7 139341522 IC50 = 17800 nM T25956 C4CHN3 139341523 IC50 = 34700 nM T25956 CRW7P5 139341524 IC50 = 5400 nM T25956 C98TAG 139341527 IC50 = 25100 nM T25956 CJ01EC 139341528 IC50 = 25100 nM T25956 C5F7OS 139341530 IC50 = 15600 nM T25956 COY2D4 139341532 IC50 = 57000 nM T25956 C6BV5E 139341541 IC50 = 16500 nM T25956 CWM81B 139341544 IC50 = 18600 nM T25956 CF1VL4 139341553 IC50 > 33000 nM T25956 CF8LU1 139341570 IC50 > 5000 nM T25956 C3SVA5 139341572 IC50 = 2200 nM T25956 CL9XU2 139341575 IC50 > 33000 nM T25956 C69JHS 139341584 IC50 > 33000 nM T25956 C7IN1U 139341589 IC50 > 100000 nM T25956 C0HT4J 139341591 IC50 > 100000 nM T25956 CF2D6W 139341726 IC50 > 100000 nM T25956 CI1H2T 139341727 IC50 > 100000 nM T25956 C9K8YX 139341747 IC50 > 100000 nM T25956 C4YMW6 139341818 IC50 > 100000 nM T25956 C8ZQ2U 141736359 IC50 = 1780 nM T25956 C5VNM4 141736367 IC50 = 49 nM T25956 C3YGJ5 145948689 IC50 = 200000 nM T25956 C96NCH 145950955 IC50 = 4450 nM T25956 C3ZV1O 145952497 IC50 = 5550 nM T25956 CB7R2C 145952522 IC50 = 8800 nM T25956 CTE74G 145954441 IC50 = 2510 nM T25956 C5WX1Y 145954899 IC50 = 52000 nM T25956 CRHG03 145955376 IC50 > 10000 nM T25956 CKO51W 145955422 IC50 > 10000 nM T25956 C3D8LO 145955588 IC50 = 60000 nM T25956 CN5YO3 145957310 IC50 = 510 nM T25956 C8JI5E 145957556 IC50 = 250000 nM T25956 C7C5WL 145958595 IC50 = 970 nM T25956 CM19OV 145959971 IC50 > 10000 nM T25956 C2OG9K 145964185 IC50 = 3900 nM T25956 C2I9YJ 145969602 IC50 = 3900 nM T25956 C15GYL 145973549 IC50 = 3900 nM T25956 CAD6O9 145975385 IC50 = 3900 nM T25956 CNHR01 145987968 IC50 > 50000 nM T25956 CBRE71 146047136 IC50 = 3857 nM T25956 CI1F6L 146204973 IC50 > 1000 nM T25956 CXG1V9 146204995 IC50 = 10 nM T25956 C2AJO8 146205056 IC50 = 2.6 nM T25956 CQM7N8 146205057 IC50 = 3 nM T25956 C9HWQ8 146205061 IC50 = 4 nM T25956 CH8E2N 146205066 IC50 = 1.9 nM T25956 CO4S3M 146205067 IC50 = 10 nM T25956 C1N5IH 146205070 IC50 = 7.5 nM T25956 CZN7D5 146205179 IC50 = 4.3 nM T25956 CZLO67 146205182 IC50 = 46 nM T25956 C5TXC2 146205184 IC50 = 3.7 nM T25956 CZU3B7 146205188 IC50 > 1000 nM T25956 CL4T3H 146205226 IC50 = 4.2 nM T25956 CUA52Y 146205228 IC50 = 2.4 nM T25956 CJ7Y0W 146205434 IC50 = 2.4 nM T25956 CY7GI4 146205498 IC50 = 30 nM T25956 CGYR94 146205502 IC50 = 14 nM T25956 CR3P4I 146205515 IC50 = 10 nM T25956 C8Z9OM 146205579 IC50 = 1.8 nM T25956 CQ1IX3 151484729 IC50 = 9610 nM T25956 CLZ34P 155512196 IC50 > 1000 nM T25956 CVJT64 155512236 IC50 = 290 nM T25956 C2WJ4O 155513273 IC50 > 10000 nM T25956 CYUW30 155514843 IC50 = 1600 nM T25956 CCI7T9 155515172 IC50 > 10000 nM T25956 C7E1TC 155516066 IC50 = 7310 nM T25956 CKM42V 155516765 IC50 > 10000 nM T25956 C2DI1Q 155516796 IC50 = 1130 nM T25956 CKR7F9 155518500 IC50 > 500 nM T25956 CG95RD 155519099 IC50 = 22 nM T25956 C2A1YU 155519665 IC50 = 2000 nM T25956 C5J8XK 155519829 IC50 = 470 nM T25956 CHD7V8 155520793 IC50 = 230 nM T25956 CMW49Z 155521226 IC50 = 860 nM T25956 C1MZC7 155522494 IC50 > 10000 nM T25956 CNL8O1 155522829 IC50 = 560 nM T25956 CE35PR 155523264 IC50 = 200 nM T25956 C3Y5XO 155523600 IC50 = 5000 nM T25956 C1SLG3 155524393 IC50 = 2400 nM T25956 CIA61E 155524527 IC50 = 5000 nM T25956 C63TIU 155524913 IC50 < 10000 nM T25956 CZ2FD5 155525448 IC50 = 6050 nM T25956 C87AZN 155525893 IC50 < 10000 nM T25956 C9OP3H 155527488 IC50 = 7130 nM T25956 C2T3OR 155528202 IC50 = 1800 nM T25956 C4XW9I 155528393 IC50 = 6000 nM T25956 CHR4K5 155528532 IC50 = 160 nM T25956 CKUM79 155528818 IC50 = 8600 nM T25956 C3LEV4 155529291 IC50 = 1800 nM T25956 CQEF61 155531348 IC50 > 10000 nM T25956 C8YNB3 155531682 IC50 < 10000 nM T25956 CHW29R 155532177 IC50 = 1950 nM T25956 C32MLY 155532996 IC50 > 10000 nM T25956 C1RPU0 155533512 IC50 > 2000 nM T25956 CK9S7N 155534073 IC50 > 10000 nM T25956 CBL5O0 155534637 IC50 > 10000 nM T25956 C9WB4Q 155534723 IC50 = 7400 nM T25956 C2RP4X 155535364 IC50 = 4400 nM T25956 C3W8XH 155536530 IC50 = 4 nM T25956 C95OQP 155536635 IC50 = 620 nM T25956 C1FEC3 155537172 IC50 = 580 nM T25956 CS3F4K 155537389 IC50 = 1.1 nM T25956 CFBE34 155538503 IC50 = 11 nM T25956 CX2Y9E 155538946 IC50 > 10000 nM T25956 CP4TW3 155539039 IC50 = 1700 nM T25956 C5KX7C 155539735 IC50 = 1530 nM T25956 CB5XE8 155539809 IC50 = 190 nM T25956 CZDW67 155540096 IC50 > 10000 nM T25956 C9KTW6 155540252 IC50 = 9800 nM T25956 CDR92H 155540348 IC50 = 5400 nM T25956 C7EOQ9 155540603 IC50 = 5000 nM T25956 C96MUR 155540976 IC50 = 3000 nM T25956 CIAT68 155542185 IC50 > 10000 nM T25956 CS3FY1 155543664 IC50 > 10000 nM T25956 CV0F2H 155544116 IC50 = 670 nM T25956 C9SUY7 155544858 IC50 = 1.3 nM T25956 COC7P0 155546490 IC50 = 2200 nM T25956 CTE76J 155547116 IC50 = 4600 nM T25956 CV56PN 155547836 IC50 = 4060 nM T25956 COHT62 155547999 IC50 = 8600 nM T25956 CX3UR0 155548318 IC50 = 2070 nM T25956 C71RPH 155548492 IC50 < 10000 nM T25956 C84GSF 155549456 IC50 < 10000 nM T25956 CP6AN5 155554496 IC50 > 10000 nM T25956 CUQ5F8 155556860 IC50 > 10000 nM T25956 CR0Y5U 155558481 IC50 = 24000 nM T25956 C8PUJ7 155558550 IC50 = 3730 nM T25956 CVL3T0 155559427 IC50 > 10000 nM T25956 CMD2A9 155559553 IC50 = 1400 nM T25956 C1TPW8 155559730 IC50 = 1800 nM T25956 CT3P5J 155559844 IC50 = 1170 nM T25956 CCY7V1 155559876 IC50 = 2800 nM T25956 CA9RW0 155560578 IC50 > 10000 nM T25956 C65CMJ 155561106 IC50 > 100 nM T25956 CQ70NE 155561894 IC50 = 73 nM T25956 CKR5A2 155563315 IC50 = 420 nM T25956 C8FD7C 155563587 IC50 = 1600 nM T25956 C2MNY1 155564022 IC50 > 10000 nM T25956 C1H9VW 155564054 IC50 > 10000 nM T25956 C2VR1B 155564237 IC50 > 10000 nM T25956 CT8S7I 155564925 IC50 = 4800 nM T25956 CK25GR 155565190 IC50 = 10000 nM T25956 C68CBM 155565352 IC50 = 12600 nM T25956 CM3SV1 155565651 IC50 = 7400 nM T25956 CY9GF7 155566211 IC50 = 12 nM T25956 CUK53M 155566805 IC50 > 10000 nM T25956 CP3B8C 155566822 IC50 = 7000 nM T25956 CZ5U4A 155568100 IC50 = 5800 nM T25956 CUDW40 155568215 IC50 = 1800 nM T25956 C4DE3Y 155568219 IC50 > 10000 nM T25956 D03XXT 72201027 IC50 = 230 nM T25956 D05RDP 992586 IC50 = 330 nM T25956 D07MTM 403 IC50 > 500000 nM T25956 D08XXD 17815 IC50 = 1400 nM T25956 D0E6JS 167551 IC50 = 8500 nM T25956 D0M6YZ 25226432 IC50 = 5000 nM T25956 D0P0IE 10205 IC50 = 2000 nM T25956 D0W3NA 87642 IC50 = 45940 nM T25956 D0YL8Z 1285940 IC50 = 9.8 nM T63414 D01BYB 5957 EC50 = 780000 nM T63414 D07QTG 66553218 IC50 = 5.012 nM T63414 D0CS2C 10161381 IC50 = 10 nM T63414 D0F4JK 11547499 IC50 = 1.3 nM T63414 D0H2UB 5361 EC50 = 92000 nM T63414 D0VI4N 90409366 IC50 = 3.467 nM T63414 D00PVH 16679492 IC50 = 39.81 nM T63414 D0FR8L 73442861 IC50 = 0.33 nM T63414 D0F8DL 176155 IC50 = 5000 nM T63414 CI15DO 265893 IC50 = 22.4 nM T63414 C1WDR8 331254 IC50 = 281.84 nM T63414 CX9F0T 331256 IC50 = 109.65 nM T63414 CCKT54 344276 IC50 = 414 nM T63414 CA3W5F 707096 IC50 = 522 nM T63414 CIWV85 746996 IC50 > 100000 nM T63414 CMUV80 766793 IC50 = 69800 nM T63414 CEBX03 779113 IC50 > 100000 nM T63414 CGJ9S2 921624 IC50 = 40800 nM T63414 C7BL5H 1478602 IC50 = 478 nM T63414 CN5T0V 1485975 IC50 = 125.89 nM T63414 CYV85L 2320735 IC50 > 10000 nM T63414 C3NPH7 2741121 IC50 = 501.19 nM T63414 CPD81K 2811018 IC50 = 320 nM T63414 CO8D1M 2812882 IC50 = 1400 nM T63414 C0S6BO 2831480 IC50 = 100 nM T63414 CR3FI4 2926477 IC50 = 4540 nM T63414 C6NAF0 2933256 IC50 = 7.943 nM T63414 C5J6IN 2941710 IC50 = 3981.07 nM T63414 C5HD9G 3079322 IC50 > 1000 nM T63414 C1RN5V 3454885 IC50 = 398.11 nM T63414 C47QZJ 3709284 IC50 = 398.11 nM T63414 CA5I3R 3872625 IC50 > 10000 nM T63414 CY68AQ 3932023 IC50 = 600 nM T63414 C81JUQ 4023622 IC50 = 3981.07 nM T63414 CM7W9S 4423333 IC50 = 125.89 nM T63414 C1V6ZX 4563797 IC50 = 501.19 nM T63414 C69OFV 4768671 IC50 = 4240 nM T63414 CPA28C 5052387 IC50 = 600 nM T63414 CJQ6M9 5151658 IC50 = 158.49 nM T63414 CN25AH 5176829 IC50 > 10000 nM T63414 CW1Q3Z 5229632 IC50 = 398.11 nM T63414 C01FHC 6466568 IC50 = 4960 nM T63414 C2WRS6 8923923 IC50 = 64.57 nM T63414 CL6DZ9 9045905 IC50 = 158.49 nM T63414 CT1K8I 9209741 IC50 = 1000 nM T63414 CSH1M6 9268807 IC50 = 79.43 nM T63414 CZDJ08 9270241 IC50 > 1000 nM T63414 CO1KY9 9821690 IC50 < 10000 nM T63414 CXE7T9 9821948 IC50 = 7.943 nM T63414 CU30FS 9878599 IC50 = 15848.93 nM T63414 CS05ET 9896790 IC50 = 1.3 nM T63414 CVL25E 9926842 IC50 = 10 nM T63414 CM74RK 9948588 IC50 = 158.49 nM T63414 CH05KP 9985155 IC50 = 50.12 nM T63414 C5VI1R 10086144 IC50 = 71.2 nM T63414 CST2B3 10115466 IC50 = 63.1 nM T63414 C05QVB 10117302 IC50 = 350 nM T63414 CYO93C 10126799 IC50 = 300 nM T63414 CM9OX5 10129577 IC50 = 132 nM T63414 C5JMC4 10139090 IC50 < 10000 nM T63414 CXYD23 10139173 IC50 < 10000 nM T63414 CT3SL2 10150143 IC50 = 4 nM T63414 COQU26 10153625 IC50 = 18.5 nM T63414 C2F5QT 10153639 IC50 = 97.7 nM T63414 CWHT56 10153662 IC50 = 100 nM T63414 CL30XQ 10153683 IC50 = 380 nM T63414 CVBZ07 10153700 IC50 = 12.3 nM T63414 CV71DN 10161380 IC50 = 0.23 nM T63414 CCA84W 10175779 IC50 = 70.8 nM T63414 C9RKJ2 10181729 IC50 < 10000 nM T63414 CMLT35 10190472 IC50 = 6 nM T63414 C0TJ1A 10197227 IC50 = 19.95 nM T63414 CKDG89 10202422 IC50 = 79.43 nM T63414 C0FK5C 10204578 IC50 = 63.1 nM T63414 CF7J5N 10212541 IC50 = 5.8 nM T63414 CZ29UQ 10219050 IC50 = 84.1 nM T63414 CDA5R8 10219058 IC50 = 15.8 nM T63414 C84RHX 10225191 IC50 < 10000 nM T63414 CBF8K0 10238746 IC50 = 15.85 nM T63414 CYJP45 10240451 IC50 = 101 nM T63414 C6ARI8 10240476 IC50 = 1122 nM T63414 C9IC5W 10276962 IC50 < 10000 nM T63414 C61FKR 10279659 IC50 = 500 nM T63414 C1GDY4 10290336 IC50 = 170 nM T63414 CXO1K8 10290342 IC50 = 79.43 nM T63414 CF6CX0 10290368 IC50 = 15.1 nM T63414 C5UX9N 10290391 IC50 = 600 nM T63414 C9DV4H 10290419 IC50 = 5.8 nM T63414 C0CY3U 10290496 IC50 = 176 nM T63414 C31FWT 10295970 IC50 < 10000 nM T63414 CSHM81 10297818 IC50 < 10000 nM T63414 CW28SB 10310632 IC50 = 10 nM T63414 C7Z0QM 10312629 IC50 = 28.8 nM T63414 C76XQR 10312667 IC50 = 13.5 nM T63414 C1C9ZI 10312693 IC50 = 12.59 nM T63414 CX56LQ 10312737 IC50 = 31.1 nM T63414 CF9JG2 10312739 IC50 = 33.9 nM T63414 CLN6Z9 10546931 IC50 = 560 nM T63414 COK26H 11007110 IC50 = 65.3 nM T63414 CPO5B9 11115244 IC50 < 1000 nM T63414 C2DJ7W 11167023 IC50 = 63.1 nM T63414 CCBW78 11179231 IC50 = 50.12 nM T63414 CJ3W8P 11187581 IC50 = 3 nM T63414 CRK5N7 11189340 IC50 = 63.1 nM T63414 CC21XM 11190463 IC50 = 50.12 nM T63414 C4V9WN 11199715 IC50 = 930 nM T63414 CK7I8C 11209712 IC50 = 630.96 nM T63414 C1Y5LT 11212938 IC50 = 100 nM T63414 CRS95A 11213305 IC50 = 100 nM T63414 CK61OS 11223687 IC50 = 31.62 nM T63414 CQM28B 11225321 IC50 = 100 nM T63414 COS8U3 11225680 IC50 = 31.62 nM T63414 CQ0C9T 11231942 IC50 = 316.23 nM T63414 CTWN36 11259677 IC50 = 79.43 nM T63414 CDOR07 11269479 IC50 = 100 nM T63414 CFPO95 11270845 IC50 = 10 nM T63414 C2XZ5B 11279679 IC50 = 10 nM T63414 CP25KE 11281239 IC50 = 63.1 nM T63414 CS6GY2 11294314 IC50 = 630.96 nM T63414 CA3I2Y 11327640 IC50 = 50.12 nM T63414 CIT65D 11350742 IC50 = 31.62 nM T63414 C8Z9LM 11351050 IC50 = 79.43 nM T63414 C4NPA1 11351142 IC50 = 39.81 nM T63414 C2XVW3 11351651 IC50 = 10 nM T63414 C6OE5H 11352109 IC50 = 50.12 nM T63414 C20GWS 11361743 IC50 = 79.43 nM T63414 CNE40H 11373994 IC50 = 63.1 nM T63414 CBI5L3 11374948 IC50 = 79.43 nM T63414 CI3RZ0 11386290 IC50 = 3.162 nM T63414 C8GJW2 11414871 IC50 = 125.89 nM T63414 CZF7H4 11418470 IC50 = 63.1 nM T63414 C2BE5J 11419335 IC50 <= 199.53 nM T63414 C07IEJ 11441307 IC50 = 25.12 nM T63414 C9S7LP 11442400 IC50 = 501.19 nM T63414 CRBG65 11453381 IC50 = 50.12 nM T63414 CBD6P3 11464418 IC50 = 19.95 nM T63414 CEXZ01 11465129 IC50 = 63.1 nM T63414 CQJ05C 11486676 IC50 = 63.1 nM T63414 C59BYU 11500704 IC50 = 31.62 nM T63414 CM2XS3 11503827 IC50 = 63.1 nM T63414 C92MUN 11507787 IC50 = 501.19 nM T63414 CWX01V 11508020 IC50 = 14.45 nM T63414 C2ND7T 11508207 IC50 = 3981.07 nM T63414 CAGV64 11509663 IC50 = 28.18 nM T63414 CBJ89G 11515022 IC50 = 39.81 nM T63414 CN9IS7 11516301 IC50 = 125.89 nM T63414 CR0MX4 11523472 IC50 = 23.99 nM T63414 C07CTD 11530196 IC50 = 12.59 nM T63414 CQG79J 11530593 IC50 = 25.12 nM T63414 CP3DM2 11530961 IC50 = 109.65 nM T63414 CZ40XE 11531460 IC50 = 63.1 nM T63414 CAW1T2 11537311 IC50 = 20.89 nM T63414 C1S2XY 11537418 IC50 = 199.53 nM T63414 CY52PW 11540045 IC50 = 100 nM T63414 C1RL5A 11543793 IC50 = 25118.86 nM T63414 C08CHM 11544727 IC50 = 18.2 nM T63414 C5A3FH 11546350 IC50 = 158.49 nM T63414 C9MZT6 11564932 IC50 = 25118.86 nM T63414 CIJ24Y 11566345 IC50 = 794.33 nM T63414 CTN61H 11573809 IC50 = 19.95 nM T63414 CXM10I 11574070 IC50 = 12.59 nM T63414 CNW65B 11602877 IC50 = 12589.25 nM T63414 C49UPR 11609203 IC50 = 15848.93 nM T63414 CC8NB2 11610500 IC50 = 12.59 nM T63414 C2QDJ4 11616778 IC50 = 63.1 nM T63414 C5JN4R 11625340 IC50 = 15 nM T63414 CV4I8J 11630893 IC50 = 100 nM T63414 C5T6EI 11639163 IC50 = 54.95 nM T63414 C57ZHK 11644745 IC50 = 7943.28 nM T63414 COVY38 11644924 IC50 = 15848.93 nM T63414 CX53OM 11652648 IC50 = 15.85 nM T63414 CIQ8C9 11652729 IC50 = 158.49 nM T63414 CJ0X3H 11652890 IC50 = 16.6 nM T63414 CC3ZM8 11653349 IC50 = 19.95 nM T63414 C94XDM 11658739 IC50 = 31622.78 nM T63414 CS3NX6 11681068 IC50 = 3981.07 nM T63414 CJQ19F 11687741 IC50 = 251.19 nM T63414 CXVQ78 11688382 IC50 = 630.96 nM T63414 CA1WS3 11690372 IC50 = 316.23 nM T63414 C7KP6B 11709854 IC50 = 50.12 nM T63414 C90UBJ 11709955 IC50 = 29.51 nM T63414 C45DFS 11744510 IC50 = 19 nM T63414 CC1US4 11749459 IC50 = 110 nM T63414 CN7CG3 11955514 IC50 = 199.53 nM T63414 CKX64A 11955519 IC50 = 190.55 nM T63414 C9YON1 11955520 IC50 = 141.25 nM T63414 CG81BJ 11955559 IC50 = 70.79 nM T63414 C8HW3J 11955560 IC50 = 52.48 nM T63414 C2MTY1 11955601 IC50 = 5.012 nM T63414 CGZ2U6 11955602 IC50 = 51.29 nM T63414 CCXO04 11955641 IC50 = 18.62 nM T63414 C8C1AH 11955642 IC50 = 1380.38 nM T63414 C8O6QT 11955678 IC50 = 57.54 nM T63414 CU5K7B 11955729 IC50 = 147.91 nM T63414 CX1KH4 11955771 IC50 = 407.38 nM T63414 CCPW09 11955827 IC50 = 173.78 nM T63414 CL96MS 11955828 IC50 = 11.75 nM T63414 CZU83X 11955880 IC50 = 131.83 nM T63414 CYC20M 11955881 IC50 = 70.79 nM T63414 C03GKP 11955920 IC50 = 33.88 nM T63414 CYR86X 11955922 IC50 = 34.67 nM T63414 C36WME 11955924 IC50 = 977.24 nM T63414 CPB15O 11955955 IC50 = 39.81 nM T63414 CL04FO 11955956 IC50 = 323.59 nM T63414 CSH71O 11955960 IC50 = 57.54 nM T63414 CXW68G 15486611 IC50 = 31 nM T63414 CX35SR 16678189 IC50 = 15.14 nM T63414 CZB32K 16678190 IC50 = 9.12 nM T63414 CHCM09 16678191 IC50 = 9.12 nM T63414 CVK63O 16678192 IC50 = 11.75 nM T63414 CF2UJ3 16678193 IC50 = 46.77 nM T63414 CE9Q6C 16678194 IC50 = 13.8 nM T63414 CK02CP 16678286 IC50 = 131.83 nM T63414 CD3S5H 16678288 IC50 = 190.55 nM T63414 CD96XF 16678386 IC50 = 190.55 nM T63414 CN14JM 16678387 IC50 = 77.62 nM T63414 COZ8V3 16678388 IC50 = 1047.13 nM T63414 CTF12U 16678389 IC50 = 13182.57 nM T63414 C69EPC 16678391 IC50 = 131.83 nM T63414 C2CNW4 16678483 IC50 = 48.98 nM T63414 CS6M5H 16678489 IC50 = 26.92 nM T63414 CJ2B6L 16678585 IC50 = 1288.25 nM T63414 CE9D7B 16678586 IC50 = 8912.51 nM T63414 CDK64U 16678694 IC50 = 58.88 nM T63414 CJ24DA 16678804 IC50 = 302 nM T63414 CVIU19 16678805 IC50 = 30.9 nM T63414 CUG98F 16678806 IC50 = 48.98 nM T63414 CY3AP8 16678807 IC50 = 19.95 nM T63414 CMKX09 16678903 IC50 = 57.54 nM T63414 C3HF2P 16678904 IC50 = 208.93 nM T63414 CZ39HD 16679400 IC50 = 15.85 nM T63414 CP42YQ 16679489 IC50 = 32.36 nM T63414 C48DST 16679490 IC50 = 67.61 nM T63414 CX20DE 16679491 IC50 = 10.96 nM T63414 C40AYD 16679493 IC50 = 354.81 nM T63414 C7QWN9 16679494 IC50 = 28.84 nM T63414 C09NSJ 16679590 IC50 = 30.9 nM T63414 CQ52JL 16679594 IC50 = 19.05 nM T63414 CIHK17 16679595 IC50 = 50.12 nM T63414 CZ6DV3 16679685 IC50 = 12.59 nM T63414 C9BE2D 16679686 IC50 = 28.18 nM T63414 C3IX1S 16748139 IC50 = 60 nM T63414 CK1C9G 16748140 IC50 > 1000 nM T63414 C9C6DJ 16748141 IC50 > 1000 nM T63414 C52NZH 16748261 IC50 > 1000 nM T63414 CX71LS 16748262 IC50 > 1000 nM T63414 CBAM38 16748263 IC50 > 1000 nM T63414 CHE60A 16748264 IC50 = 12.1 nM T63414 C0FR5J 16748265 IC50 > 1000 nM T63414 CR0E9D 16748266 IC50 > 1000 nM T63414 C1WU4K 16748384 IC50 > 1000 nM T63414 CWJT79 16748385 IC50 > 1000 nM T63414 C9Y7IB 16748386 IC50 > 1000 nM T63414 CTP6G1 16748387 IC50 > 1000 nM T63414 C5I0CX 16748388 IC50 > 1000 nM T63414 C5H8YP 16748389 IC50 > 1000 nM T63414 C10DVY 16748517 IC50 > 1000 nM T63414 CFM3I6 16748518 IC50 > 1000 nM T63414 CEMJ08 16748519 IC50 > 1000 nM T63414 CF3NI1 16748520 IC50 > 1000 nM T63414 CEX26A 16748521 IC50 = 130 nM T63414 CR4K2L 16748522 IC50 > 1000 nM T63414 CU1N4Z 16748628 IC50 > 1000 nM T63414 CID4T1 16748629 IC50 = 40.2 nM T63414 C64BCT 16748630 IC50 > 1000 nM T63414 C25LUG 16748631 IC50 > 1000 nM T63414 CJ9T3Q 16748632 IC50 > 1000 nM T63414 CGPI14 16748633 IC50 = 19.95 nM T63414 C05XNW 16748739 IC50 > 1000 nM T63414 CAKU80 16748740 IC50 = 800 nM T63414 C85QSE 16748741 IC50 > 1000 nM T63414 C4ZAP3 16748742 IC50 > 1000 nM T63414 CWK92R 16748743 IC50 = 35.1 nM T63414 C2Z9YL 16748744 IC50 = 900 nM T63414 CAG01I 16748850 IC50 = 39.81 nM T63414 C9N1AT 16748851 IC50 > 1000 nM T63414 C4Z1DH 16749266 IC50 > 1000 nM T63414 CX1F0R 16749371 IC50 > 1000 nM T63414 C6EM0D 16749372 IC50 = 90.2 nM T63414 CS69QB 16749373 IC50 > 1000 nM T63414 C7XE5Z 16749374 IC50 = 100 nM T63414 CHP82C 16749375 IC50 > 1000 nM T63414 CVH87I 16749376 IC50 > 1000 nM T63414 C0YM8U 18438679 IC50 = 238 nM T63414 C4WP3N 18438683 IC50 = 266 nM T63414 CQG7A5 18438690 IC50 = 95 nM T63414 CG0ZC7 18438692 IC50 = 280 nM T63414 C1Y2TM 18438700 IC50 = 490 nM T63414 C5OPF8 19796304 IC50 = 1 nM T63414 C2KI6R 20173059 IC50 = 2420 nM T63414 C3D9MI 20660005 IC50 = 63.1 nM T63414 C2YI9L 20660020 IC50 = 5.012 nM T63414 C3DT0V 20968164 IC50 = 316.23 nM T63414 CD8CM9 21093784 IC50 = 940 nM T63414 C9BJ7T 21093792 IC50 = 1300 nM T63414 CYA5O7 21093813 IC50 = 1100 nM T63414 C90NZQ 21093814 IC50 = 3600 nM T63414 C0BMP1 21093816 IC50 = 2800 nM T63414 C05FAL 21093905 IC50 = 794.33 nM T63414 COB7R6 22341299 IC50 = 50.12 nM T63414 CVF35Z 22644568 IC50 <= 31622.78 nM T63414 CP6F7H 22644657 IC50 <= 31622.78 nM T63414 CGU0Q2 22644665 IC50 <= 31622.78 nM T63414 C3GVJ2 23649368 IC50 = 132 nM T63414 CK76FP 23649427 Ki = 3.1 nM T63414 C49XAU 23654641 IC50 = 15.85 nM T63414 CC7H0G 23654661 IC50 = 630.96 nM T63414 C47PTE 23654663 IC50 = 251.19 nM T63414 CG39XH 23654666 IC50 = 7.943 nM T63414 C2PV0A 23654747 IC50 = 158.49 nM T63414 CSF46T 23654751 IC50 = 158.49 nM T63414 C1JEP4 23654752 IC50 = 39.81 nM T63414 C73PFO 23654815 IC50 = 2.512 nM T63414 CADC51 23654831 IC50 = 63.1 nM T63414 CKW05E 23654832 IC50 < 3162.28 nM T63414 C5NI0H 23654834 IC50 = 2.512 nM T63414 C5R2VB 24760653 IC50 = 1.995 nM T63414 C2QA6E 24760968 IC50 = 6.31 nM T63414 CMIJ42 24864649 IC50 = 11.48 nM T63414 CZ14WI 24864650 IC50 = 218.78 nM T63414 C6G7YS 24864651 IC50 = 33.88 nM T63414 CET91X 24865007 IC50 = 371.54 nM T63414 CXY74N 24865008 IC50 = 831.76 nM T63414 CRUS91 24865188 IC50 = 38.9 nM T63414 CZF70G 24883277 IC50 > 10000 nM T63414 CEH1K6 24894837 IC50 = 0.1995 nM T63414 C61OTM 24894840 IC50 = 0.05012 nM T63414 CV6B2Z 25011821 IC50 = 3.162 nM T63414 CFB7R4 25014313 IC50 = 0.01 nM T63414 CLA64S 25020193 IC50 = 15.85 nM T63414 C8Y2DG 25022679 IC50 > 10000 nM T63414 CC54IX 25022680 IC50 = 59 nM T63414 C4I6OJ 25032957 IC50 = 34 nM T63414 C68WHE 25061571 IC50 = 10 nM T63414 C39WZD 25061573 IC50 = 10 nM T63414 CZ8S3D 25106221 IC50 = 39.81 nM T63414 C1FER2 25106484 IC50 = 25.12 nM T63414 COEG07 25106658 IC50 = 316.23 nM T63414 C5RC1L 25106660 IC50 = 158.49 nM T63414 CM23AC 25106741 IC50 = 316.23 nM T63414 CPD29L 25106743 IC50 = 63.1 nM T63414 CFN59X 25106744 IC50 = 100 nM T63414 CQC4D9 25107017 IC50 = 50.12 nM T63414 CPJ30M 25107453 IC50 > 630.96 nM T63414 CLIZ02 25159047 IC50 = 28 nM T63414 CT78IL 25210349 IC50 = 31.62 nM T63414 C5F2OH 25809478 IC50 = 3981.07 nM T63414 C3LD7V 40075164 IC50 = 5950 nM T63414 COK46N 44139106 IC50 = 31.62 nM T63414 CJ4QG2 44139223 IC50 = 199.53 nM T63414 C6N8ZH 44139224 IC50 = 251.19 nM T63414 CEGZ59 44139225 IC50 = 251.19 nM T63414 CB0ZD7 44139226 IC50 = 316.23 nM T63414 CD3OL6 44139227 IC50 = 794.33 nM T63414 CZF1I8 44139348 IC50 = 3162.28 nM T63414 CDAY27 44139349 IC50 = 251.19 nM T63414 CA6Q9T 44139350 IC50 = 31622.78 nM T63414 CR19DY 44139351 IC50 = 5011.87 nM T63414 CMYX63 44139352 IC50 = 199.53 nM T63414 CJW89G 44139353 IC50 = 10 nM T63414 CRS4D7 44139469 IC50 = 1995.26 nM T63414 C97IUM 44139470 IC50 = 199.53 nM T63414 C9J4WA 44139598 IC50 = 100 nM T63414 CZ2Q7I 44139724 IC50 = 158.49 nM T63414 C47RUK 44139725 IC50 = 199.53 nM T63414 C9WD4T 44139726 IC50 = 251.19 nM T63414 CHS4Z6 44139727 IC50 = 316.23 nM T63414 C6WFB9 44139728 IC50 = 398.11 nM T63414 CK32IJ 44139877 IC50 = 1000 nM T63414 CJO78K 44139878 IC50 = 1584.89 nM T63414 CRLO92 44139879 IC50 = 794.33 nM T63414 CDM84Y 44139880 IC50 = 2511.89 nM T63414 C87ZUF 44139881 IC50 = 7943.28 nM T63414 C3H6PM 44139882 IC50 = 398.11 nM T63414 C9VJB2 44140001 IC50 = 630.96 nM T63414 CF7RH1 44140002 IC50 = 31.62 nM T63414 CE9WA1 44180167 IC50 = 310 nM T63414 CC14MU 44180168 IC50 = 250 nM T63414 CD51AN 44180169 IC50 = 180 nM T63414 C19ZDA 44241649 IC50 = 4310 nM T63414 CMH56F 44250460 IC50 = 19.95 nM T63414 CB91UW 44352797 IC50 < 10000 nM T63414 CD5MN7 44352798 IC50 = 630.96 nM T63414 C1RV2U 44352806 IC50 = 10000 nM T63414 CVZ85O 44352829 IC50 < 10000 nM T63414 C6FK0N 44352831 IC50 = 630.96 nM T63414 C7S4NI 44352852 IC50 = 6309.57 nM T63414 CW7O4M 44352866 IC50 < 10000 nM T63414 CGI63Q 44352867 IC50 < 10000 nM T63414 CIYE20 44352908 IC50 < 10000 nM T63414 CLR60K 44352910 IC50 < 10000 nM T63414 CNQ8Y9 44352911 IC50 < 10000 nM T63414 CN2RD8 44352912 IC50 < 10000 nM T63414 C3OY6E 44352913 IC50 < 10000 nM T63414 CF24SK 44352947 IC50 = 79.43 nM T63414 CYQ4A7 44352996 IC50 = 125.89 nM T63414 C3CUK0 44353025 IC50 = 158.49 nM T63414 C7D9EM 44353041 IC50 = 158.49 nM T63414 C9HGY8 44353139 IC50 = 199.53 nM T63414 CQ46IG 44353592 EC50 = 52000 nM T63414 CXM4D2 44374511 IC50 = 316 nM T63414 CAN0B9 44388794 IC50 = 63.1 nM T63414 CZ17CH 44388802 IC50 = 125.89 nM T63414 C57VAP 44388827 IC50 > 1000 nM T63414 CXUJ85 44388935 IC50 = 316.23 nM T63414 CH73BF 44388973 IC50 = 79.43 nM T63414 CRKP03 44388975 IC50 = 79.43 nM T63414 CPUT83 44389013 IC50 = 63.1 nM T63414 CMCQ81 44389040 IC50 > 3162.28 nM T63414 C5R3HZ 44391901 IC50 = 79.43 nM T63414 C50EJN 44412196 IC50 > 10000 nM T63414 CO3A0B 44440425 IC50 = 524.81 nM T63414 CT83UQ 44440428 IC50 = 602.56 nM T63414 COEL10 44440430 IC50 = 426.58 nM T63414 CIP1J7 44440432 IC50 = 1819.7 nM T63414 CV6IR5 44440433 IC50 = 6025.6 nM T63414 C1ZO2R 44440436 IC50 = 117.49 nM T63414 CV9W5I 44440439 IC50 = 144.54 nM T63414 C8K9MP 44440442 IC50 = 47.86 nM T63414 C3KF9Q 44440446 IC50 = 48.98 nM T63414 C26ZEO 44440449 IC50 = 912.01 nM T63414 C0YN6I 44440452 IC50 = 213.8 nM T63414 CCL5V1 44440456 IC50 = 331.13 nM T63414 COGQ18 44440459 IC50 = 138.04 nM T63414 CJ0N5Z 44446289 IC50 = 219 nM T63414 CYV62I 44446290 IC50 = 599 nM T63414 C70DYF 44446291 IC50 = 260 nM T63414 CB8SW5 44446292 IC50 = 256 nM T63414 CY5W3J 44446293 IC50 = 504 nM T63414 C9YWH1 44446294 IC50 = 1360 nM T63414 C4I1SC 44446295 IC50 = 539 nM T63414 CJ15XN 44446298 IC50 = 2010 nM T63414 CZXK03 44446299 IC50 = 724 nM T63414 C9Y0VR 44446300 IC50 = 319 nM T63414 CT9R6N 44446317 IC50 = 481 nM T63414 C4LCZ1 44446318 IC50 = 5880 nM T63414 CE0JT5 44446319 IC50 = 517 nM T63414 CDJM56 44446320 IC50 = 3540 nM T63414 C39KPW 44446321 IC50 = 780 nM T63414 C39MDY 44446322 IC50 = 725 nM T63414 CVS3W2 44446323 IC50 = 2460 nM T63414 CZ6J0T 44446324 IC50 = 1540 nM T63414 CP3R2U 44446325 IC50 = 861 nM T63414 C58XIQ 44446327 IC50 = 40 nM T63414 C9JP6I 44453720 IC50 = 67.61 nM T63414 C78FNH 44453771 IC50 = 45.71 nM T63414 CWZ92N 44453795 IC50 = 1621.81 nM T63414 CBA61W 44453817 IC50 = 288.4 nM T63414 CER54H 44453839 IC50 = 20.89 nM T63414 C46EXZ 44453840 IC50 = 154.88 nM T63414 CX5CV8 44453841 IC50 = 478.63 nM T63414 C6PAB1 44453843 IC50 = 47.86 nM T63414 CT3SA5 44453866 IC50 = 616.6 nM T63414 C14RXQ 44453867 IC50 = 3388.44 nM T63414 C7L6BX 44453869 IC50 = 102.33 nM T63414 C7O5BW 44453870 IC50 = 1862.09 nM T63414 CRM84K 44453893 IC50 = 363.08 nM T63414 CP76NZ 44453894 IC50 = 17.78 nM T63414 CSH25Q 44453895 IC50 = 45.71 nM T63414 CZC02W 44454976 IC50 = 140 nM T63414 CTH0Y1 44454978 IC50 = 51 nM T63414 C9DI8L 44454979 IC50 = 88 nM T63414 CZB07S 44455002 IC50 = 58 nM T63414 C4UJE8 44455036 IC50 = 190 nM T63414 C61QTH 44455104 IC50 = 220 nM T63414 CM0Q3T 44455110 IC50 = 430 nM T63414 C4GEW6 44455183 IC50 = 1300 nM T63414 CV9L8T 44455230 IC50 = 460 nM T63414 CG2BU3 44455253 IC50 = 70 nM T63414 CILG68 44455273 IC50 = 57 nM T63414 C2CW5X 44455277 IC50 = 94 nM T63414 CRQ15X 44455311 IC50 = 100 nM T63414 CSV9Z2 44455312 IC50 = 1500 nM T63414 C9BXO1 44455345 IC50 = 1000 nM T63414 CF3MU9 44455378 IC50 = 40 nM T63414 C8S4DG 44455380 IC50 = 60 nM T63414 C3Y2UZ 44455397 IC50 = 110 nM T63414 CXVM85 44455398 IC50 = 71 nM T63414 C7IKG2 44455425 IC50 = 46 nM T63414 CE9VI7 44455448 IC50 = 410 nM T63414 C2B3HJ 44455452 IC50 = 46 nM T63414 CPY02X 44455453 IC50 = 36 nM T63414 COWX27 44455454 IC50 = 40 nM T63414 CEUW63 44455455 IC50 = 310 nM T63414 CJOC69 44567813 IC50 = 25 nM T63414 CE2LB5 44567814 IC50 = 1030 nM T63414 C84VNX 44567815 IC50 = 540 nM T63414 CAH7Z4 44567845 IC50 > 10000 nM T63414 C5OVW0 44567848 IC50 = 780 nM T63414 CYF1R5 44567880 IC50 = 60 nM T63414 CB9SK6 44567881 IC50 = 112 nM T63414 C7FPK6 44567882 IC50 = 40 nM T63414 CQ2CU7 44567883 IC50 = 67 nM T63414 C10QEB 44567914 IC50 = 45 nM T63414 C0MIV1 44567915 IC50 = 130 nM T63414 CWY8Z4 44567916 IC50 = 250 nM T63414 CWP2D0 44567917 IC50 = 24900 nM T63414 CXYI51 44567972 IC50 = 480 nM T63414 C12TOE 44567973 IC50 = 1660 nM T63414 CZ0Q9L 44567974 IC50 = 1330 nM T63414 CJO97Q 44567975 IC50 = 60 nM T63414 CS2YF1 44568011 IC50 = 110 nM T63414 CPG8J6 44568014 IC50 = 93 nM T63414 CX9FB2 44571409 IC50 = 2660 nM T63414 C83OUL 44571411 IC50 = 4410 nM T63414 CR9N4X 44571929 IC50 = 440 nM T63414 C1RF3V 44571930 IC50 = 420 nM T63414 C29IPU 44571977 IC50 = 260 nM T63414 CJX40Z 44571979 IC50 = 400 nM T63414 C1LP0O 44571981 IC50 = 1120 nM T63414 CYX8R0 44572018 IC50 = 5020 nM T63414 C9QAH4 44572020 IC50 = 2560 nM T63414 CNK6G2 44572022 IC50 = 5400 nM T63414 CC5E4B 44572069 IC50 = 820 nM T63414 CZ87DW 44572070 IC50 = 420 nM T63414 C2NW7D 44572072 IC50 = 730 nM T63414 C87PRC 44572124 IC50 = 1530 nM T63414 CJM0C8 44572126 IC50 = 170 nM T63414 C8VO6R 44572127 IC50 = 1260 nM T63414 CGC93W 44572128 IC50 = 2600 nM T63414 CZ3MQ2 44572130 IC50 = 2810 nM T63414 C78EIN 44572132 IC50 = 3220 nM T63414 CAKV23 44576800 IC50 = 27.54 nM T63414 C3TK7V 44576833 IC50 < 1 nM T63414 CE12IZ 44576834 IC50 = 22.91 nM T63414 CRI8B3 44576835 IC50 = 275.42 nM T63414 C4C1FB 44576871 IC50 = 27.54 nM T63414 CX6EC5 45123697 IC50 = 50.12 nM T63414 CQJ49O 45267133 IC50 = 25.12 nM T63414 C9EM1X 45267162 IC50 = 15.85 nM T63414 CFE72S 45267185 IC50 = 501.19 nM T63414 CIF7D9 45267968 IC50 = 10 nM T63414 C48NUE 45269693 IC50 = 7.943 nM T63414 C92BPO 45269772 IC50 > 10000 nM T63414 CRYJ65 45270525 IC50 = 199.53 nM T63414 CG6A1U 45270543 IC50 = 0.3162 nM T63414 CJG3R6 45270588 IC50 = 19.95 nM T63414 C7GD3S 45271344 IC50 <= 10000 nM T63414 CC6UN5 45271415 IC50 > 10000 nM T63414 CA6DH8 45272316 IC50 > 10000 nM T63414 C2NOZ0 45273093 IC50 = 398.11 nM T63414 C8FBV6 45273094 IC50 <= 10000 nM T63414 C7C8SV 45273191 IC50 < 31622.78 nM T63414 C0RVP9 45486014 IC50 = 790 nM T63414 C1T6IN 45486047 IC50 = 13000 nM T63414 CZ0B3A 45486077 IC50 = 1450 nM T63414 CU3H1X 45486078 IC50 = 1280 nM T63414 CJ7R8B 45486080 IC50 = 1180 nM T63414 C3RF4L 45486083 IC50 = 740 nM T63414 CHW0Q6 45486085 IC50 = 850 nM T63414 C2LU4C 45486086 IC50 = 520 nM T63414 CI5G0S 45486088 IC50 = 1420 nM T63414 CG9OH1 45486091 IC50 = 1070 nM T63414 CBPD97 46175179 IC50 > 10000 nM T63414 C80DAS 46231312 IC50 > 10000 nM T63414 C6LJC9 46700791 IC50 = 251.19 nM T63414 C1I6PO 46830282 IC50 = 16 nM T63414 CM6L0H 46830291 IC50 = 27 nM T63414 C01TIE 46831210 IC50 = 33 nM T63414 CYJ24N 46831211 IC50 = 9 nM T63414 CLQ0S5 46831213 IC50 = 39 nM T63414 C2W8ID 46832336 IC50 = 23 nM T63414 CPE2Z1 46834939 IC50 = 104 nM T63414 CT2AE5 46834941 IC50 = 92 nM T63414 CHP14S 46834942 IC50 = 38 nM T63414 CA06XH 46886951 IC50 = 32 nM T63414 C7QL1Y 46886952 IC50 = 449 nM T63414 C5L3VP 46886953 IC50 = 17 nM T63414 CR2P7T 46886954 IC50 = 46 nM T63414 CU16JH 46886955 IC50 = 51 nM T63414 C46RHT 46887106 IC50 = 125.89 nM T63414 CTIN74 46887107 IC50 > 1000 nM T63414 C0UK6V 46887108 IC50 > 1000 nM T63414 CE13QO 46887141 IC50 > 1000 nM T63414 C7AID1 46887142 IC50 > 1000 nM T63414 CV1XW4 46887143 IC50 = 251.19 nM T63414 CDUO76 46887144 IC50 > 1000 nM T63414 CT6LC8 46887145 IC50 = 158.49 nM T63414 C0IZ2X 46887191 IC50 = 158.49 nM T63414 CFKC73 46887193 IC50 > 1000 nM T63414 CJB92T 46887194 IC50 > 1000 nM T63414 CLW5I3 46887195 IC50 > 1000 nM T63414 C3E4LZ 46887223 IC50 = 39.81 nM T63414 C9MO4K 46887224 IC50 = 10 nM T63414 CWC97Y 46887252 IC50 = 125.89 nM T63414 C9NFM0 46887253 IC50 = 199.53 nM T63414 CCZ9I6 46887477 IC50 = 40 nM T63414 CS0K7X 46887514 IC50 = 213 nM T63414 CLF08T 46887515 IC50 = 134 nM T63414 CCU0J8 46887516 IC50 = 232 nM T63414 C4LN5B 46887517 IC50 = 17 nM T63414 CD5F4G 46887518 IC50 = 32 nM T63414 C6TPL2 46887560 IC50 = 56 nM T63414 CM58OE 46887561 IC50 = 18 nM T63414 CBPU74 46887562 IC50 = 22 nM T63414 C1WBI0 46887563 IC50 = 8 nM T63414 CLV1W2 46918487 IC50 = 39.81 nM T63414 CY1OI8 49803437 IC50 = 932 nM T63414 CR1W5M 49863038 IC50 = 10 nM T63414 CLDK29 49863078 IC50 = 125.89 nM T63414 CH18IF 49863079 IC50 = 100 nM T63414 CGXC76 49863080 IC50 = 158.49 nM T63414 C5XZN3 49863081 IC50 > 1000 nM T63414 CW7Z8Q 49863082 IC50 = 12.59 nM T63414 C02NHY 49863083 IC50 = 398.11 nM T63414 CL45EU 49863107 IC50 = 158.49 nM T63414 CQN7K5 49863108 IC50 = 316.23 nM T63414 CE8FN5 49863109 IC50 = 63.1 nM T63414 CEB9H4 49864819 IC50 = 501.19 nM T63414 CPQ0C5 49864874 IC50 = 794.33 nM T63414 CY1NP4 49864875 IC50 = 100 nM T63414 CFWJ63 49864876 IC50 < 1000 nM T63414 CQ7K6V 49864877 IC50 = 100 nM T63414 C1VJ3X 49864911 IC50 = 31.62 nM T63414 CCN40K 49864912 IC50 = 158.49 nM T63414 CKBY67 49864913 IC50 = 398.11 nM T63414 CKTJ85 49864914 IC50 < 1000 nM T63414 CR0M7Y 49864915 IC50 = 25.12 nM T63414 CTV2R6 49864916 IC50 < 1000 nM T63414 C8Q0IP 49864946 IC50 < 1000 nM T63414 CNA3I9 49864947 IC50 = 79.43 nM T63414 C3VU2Y 49864948 IC50 = 630.96 nM T63414 CFT3V8 49864949 IC50 < 1000 nM T63414 CO1Y8A 49864950 IC50 = 630.96 nM T63414 C6Q5PX 49864951 IC50 = 100 nM T63414 C8Y0QK 49864952 IC50 = 630.96 nM T63414 CA1ZP4 49865005 IC50 < 1000 nM T63414 C9VB5R 49865006 IC50 = 12.59 nM T63414 CEQ42N 49865007 IC50 = 6.31 nM T63414 C9TX8W 49865008 IC50 = 1.585 nM T63414 CPO7N8 49865009 IC50 < 1000 nM T63414 CVLW35 49865010 IC50 = 100 nM T63414 CM3R5F 49865011 IC50 < 1000 nM T63414 CE93YS 49865054 IC50 = 158.49 nM T63414 C5UJL2 49865055 IC50 = 31.62 nM T63414 C0S2UE 50898450 IC50 = 10 nM T63414 C8P3FI 52543399 IC50 = 6410 nM T63414 CD52NL 52940698 IC50 = 3.981 nM T63414 CD4YE2 52941885 IC50 = 3.981 nM T63414 C7NV6R 52942125 IC50 = 31.62 nM T63414 C60DON 52943044 IC50 = 1.995 nM T63414 C3YWI6 52943045 IC50 = 10 nM T63414 CS46RU 52943071 IC50 = 5.012 nM T63414 CBRT15 52943107 IC50 = 79.43 nM T63414 CQ0B4W 52943108 IC50 = 25.12 nM T63414 CO9X7I 52943116 IC50 = 2.512 nM T63414 CYJ72M 52944502 IC50 = 0.631 nM T63414 CPG4J9 52944504 IC50 = 3.981 nM T63414 CM72WO 52946486 IC50 = 10 nM T63414 CC29MO 52946708 IC50 = 25.12 nM T63414 CWV76B 52947925 IC50 = 25.12 nM T63414 C78WQD 52947971 IC50 = 3.981 nM T63414 CDVR73 52949177 IC50 = 10 nM T63414 CM7B8F 53248666 IC50 = 14.79 nM T63414 C87LRM 53249126 IC50 = 11.48 nM T63414 C4KJN3 53357190 IC50 = 50 nM T63414 CFNV60 53357191 IC50 = 29 nM T63414 CV4NJ5 53357192 IC50 = 24 nM T63414 C3HO2R 53388310 IC50 = 3 nM T63414 C5BQU3 53388312 IC50 = 0.5 nM T63414 CG1L4T 54580621 IC50 = 64 nM T63414 CNI84W 54580632 IC50 = 41 nM T63414 C2OP1Q 54580633 IC50 = 132 nM T63414 CZJ87H 54580659 IC50 = 13.8 nM T63414 C3OZE5 54580660 IC50 = 21.88 nM T63414 C3RAB9 54580661 IC50 = 120.23 nM T63414 CE68YQ 54580681 IC50 = 74.13 nM T63414 CB7S6Y 54580682 IC50 = 54.95 nM T63414 CD9R1X 54580683 IC50 = 26.92 nM T63414 CWH45G 54581536 IC50 > 5000 nM T63414 CQW6Y4 54581643 IC50 = 25 nM T63414 CAF1W3 54581644 IC50 = 41 nM T63414 C9NYE7 54581645 IC50 = 64 nM T63414 CZB03V 54581673 IC50 = 16.6 nM T63414 C72LDF 54581674 IC50 = 27.54 nM T63414 CKVL16 54581675 IC50 = 82 nM T63414 CBT56Y 54581676 IC50 = 248 nM T63414 CJ82ZY 54581694 IC50 = 562.34 nM T63414 C90TNZ 54581695 IC50 = 1905.46 nM T63414 CUSK31 54581696 IC50 = 14.79 nM T63414 C4WJP0 54582634 IC50 = 141 nM T63414 C4OQ0E 54582635 IC50 = 470 nM T63414 C3M7BF 54582636 IC50 = 3207 nM T63414 C0MV6O 54582637 IC50 = 1236 nM T63414 CO6T7E 54582658 IC50 = 23.99 nM T63414 C5YMS4 54582659 IC50 = 43 nM T63414 C31HVQ 54582660 IC50 = 51 nM T63414 CEQK29 54582681 IC50 = 436.52 nM T63414 CO78WU 54582682 IC50 = 5623.41 nM T63414 CA35XM 54583586 IC50 = 121 nM T63414 C9E2DV 54583587 IC50 = 36 nM T63414 CL9HZ2 54583588 IC50 = 52 nM T63414 CZ36RH 54583589 IC50 = 439 nM T63414 CUIL26 54583619 IC50 = 40.74 nM T63414 CW6M0F 54583620 IC50 = 31.62 nM T63414 CC4ZP6 54583646 IC50 = 28.18 nM T63414 CB3N6C 54583647 IC50 = 38.9 nM T63414 C34SBA 54584488 IC50 = 185 nM T63414 CWV3S2 54584577 IC50 = 4065 nM T63414 C79HIA 54584578 IC50 = 117 nM T63414 CXC2J1 54584579 IC50 = 1471 nM T63414 CU19XD 54584620 IC50 = 74.13 nM T63414 CO5A6J 54584621 IC50 = 19.95 nM T63414 C2J6ED 54584622 IC50 = 70.79 nM T63414 CG7C0N 54584623 IC50 = 87.1 nM T63414 CC8JA2 54585434 IC50 = 42 nM T63414 CC5EH6 54585435 IC50 = 700 nM T63414 CW9AR7 54585517 IC50 = 158 nM T63414 CJ9R3L 54585518 IC50 = 114 nM T63414 C41NMK 54585519 IC50 = 143 nM T63414 CHA0L2 54585520 IC50 = 207 nM T63414 C5MCX8 54585545 IC50 = 39.81 nM T63414 CY3NR0 54585546 IC50 = 31.62 nM T63414 CAJ7W9 54585547 IC50 = 257.04 nM T63414 C7C4OB 54585548 IC50 = 42 nM T63414 CWO7F1 54585568 IC50 = 234.42 nM T63414 CB40QJ 54585569 IC50 = 15.85 nM T63414 CNRW68 54586397 IC50 = 200 nM T63414 C9MJH2 54586491 IC50 = 52 nM T63414 CS79DZ 54586492 IC50 = 111 nM T63414 C01NPQ 54586493 IC50 = 40 nM T63414 C85ZRN 54586494 IC50 = 114 nM T63414 C0E7LC 54586495 IC50 = 73 nM T63414 CXYL81 54586524 IC50 = 18.2 nM T63414 C1FYE9 54587413 IC50 > 5000 nM T63414 C0B5GH 54587523 IC50 = 35 nM T63414 CIL8Y6 54587524 IC50 = 43 nM T63414 C3VWR8 54587525 IC50 = 252 nM T63414 CNBI30 54587526 IC50 = 35 nM T63414 CSU91D 54587578 IC50 = 30.2 nM T63414 C7Y9QF 56589589 IC50 = 24 nM T63414 CW20CN 56658584 IC50 = 250 nM T63414 CA8W3B 56658585 IC50 = 1050 nM T63414 CXW93P 56658695 IC50 = 4800 nM T63414 CN2Y8B 56662034 IC50 = 6 nM T63414 C3X6SW 56662173 IC50 = 1600 nM T63414 CPO39Q 56662911 IC50 = 50.12 nM T63414 CV2IO3 56662912 IC50 = 158.49 nM T63414 CXF5Q2 56662950 IC50 = 199.53 nM T63414 C1HT4M 56665515 IC50 = 720 nM T63414 C0SN9Z 56665516 IC50 = 510 nM T63414 C3ZR5Q 56666388 IC50 = 50.12 nM T63414 CQE0H2 56666425 IC50 = 100 nM T63414 CNI50D 56666426 IC50 = 31.62 nM T63414 CJ6SG0 56666427 IC50 = 39.81 nM T63414 CS49UN 56668947 IC50 = 460 nM T63414 CT7SK3 56668948 IC50 = 240 nM T63414 C8JF5B 56669848 IC50 = 50.12 nM T63414 CZ0JP1 56672431 IC50 = 4600 nM T63414 C8WEG7 56675816 IC50 = 5200 nM T63414 CXW23S 56676617 IC50 = 100 nM T63414 C87VZL 56676618 IC50 = 50.12 nM T63414 CQV48D 56676619 IC50 = 50.12 nM T63414 C2SW4X 56679127 IC50 = 668 nM T63414 CJMO40 56679990 IC50 = 125.89 nM T63414 CQYN10 56679991 IC50 = 63.1 nM T63414 C2BQ9G 56683282 IC50 = 100 nM T63414 CEP6F0 56683327 IC50 = 63.1 nM T63414 C4LQK6 56683328 IC50 = 501.19 nM T63414 C9KI8H 57390667 IC50 = 50 nM T63414 CH6J9B 57392463 IC50 = 101 nM T63414 C5ZCB2 57392464 IC50 = 28 nM T63414 CQ5HO4 57392465 IC50 = 45 nM T63414 C9TLV4 57392466 IC50 = 1944 nM T63414 C8DE7B 57394171 IC50 = 388 nM T63414 CBAH26 57394172 IC50 = 276 nM T63414 CBMW74 57394173 IC50 = 700 nM T63414 C6WP2N 57394174 IC50 = 91 nM T63414 CF9NK7 57394175 IC50 = 52 nM T63414 CAJE41 57394176 IC50 = 39 nM T63414 CC4D5S 57394312 IC50 = 178 nM T63414 C0LX4E 57394313 IC50 = 85 nM T63414 C0NS6G 57395953 IC50 = 25 nM T63414 CT4X5P 57397748 IC50 = 110 nM T63414 C39CQX 57399409 IC50 = 108 nM T63414 CA57EW 57399410 IC50 = 104 nM T63414 C0WF7P 57399411 IC50 = 95 nM T63414 CE98JC 57399524 IC50 = 937 nM T63414 CD65TQ 57399525 IC50 = 870 nM T63414 C7S2RH 57399526 IC50 = 107 nM T63414 C4A9HB 57401171 IC50 = 55 nM T63414 CTN6K9 57401282 IC50 = 237 nM T63414 C4DUJ3 57401283 IC50 = 845 nM T63414 C0H2XN 57402932 IC50 = 137 nM T63414 CGH68E 57403034 IC50 = 269 nM T63414 CG1BC2 57403035 IC50 = 1036 nM T63414 C3POX4 57412481 IC50 = 900 nM T63414 CX50UV 57412482 IC50 = 1100 nM T63414 CT6Q4M 57412483 IC50 = 1400 nM T63414 CD6IN7 57412484 IC50 = 1500 nM T63414 CIXG79 57412485 IC50 = 620 nM T63414 C3F0YK 57412486 IC50 = 2500 nM T63414 CQF81U 57412565 IC50 = 1100 nM T63414 CNV98G 57412566 IC50 = 770 nM T63414 CC6BO8 57412567 IC50 = 1200 nM T63414 C84XCU 57412568 IC50 = 1900 nM T63414 C2WI7A 57412569 IC50 = 950 nM T63414 C56ICN 57412570 IC50 = 370 nM T63414 CL2ZY8 57412662 IC50 = 1100 nM T63414 C7ESN1 57412663 IC50 = 4200 nM T63414 CDQL71 57412664 IC50 = 320 nM T63414 CW1V0E 57412668 IC50 = 1200 nM T63414 CFS42I 57412745 IC50 = 380 nM T63414 C26MYQ 57412746 IC50 = 56 nM T63414 C81YML 57412747 IC50 = 42 nM T63414 CA1FY2 57412748 IC50 = 730 nM T63414 CJ7P2M 57412749 IC50 = 360 nM T63414 CV3H5P 57412750 IC50 = 340 nM T63414 CF1RD7 57412751 IC50 = 77 nM T63414 CY0CZ1 57412921 IC50 = 900 nM T63414 C67YRL 58227894 IC50 = 64 nM T63414 C0T1SR 58227950 IC50 = 82 nM T63414 CZEJ87 58228090 IC50 = 85 nM T63414 CT1EL4 58228091 IC50 = 151 nM T63414 CJ9EB3 58228418 IC50 = 78 nM T63414 CRSI26 58228496 IC50 = 120 nM T63414 CJ5Y4X 58228512 IC50 = 35 nM T63414 CS9LM2 59377426 IC50 = 23 nM T63414 CLPY52 59377517 IC50 = 20 nM T63414 C19YVT 59377518 IC50 = 8 nM T63414 C1JK7V 59377559 IC50 = 30 nM T63414 C4CD3N 59377565 IC50 = 27 nM T63414 CK23UQ 59377575 IC50 = 6 nM T63414 CQZ4H9 59377579 IC50 = 17 nM T63414 C24VHF 59377604 IC50 = 33 nM T63414 C0Z9CB 59377671 IC50 = 3800 nM T63414 C5T4CV 59377728 IC50 = 37 nM T63414 C3OY9U 59377733 IC50 = 40 nM T63414 C6GE1D 59377797 IC50 = 32 nM T63414 CHYU80 59377854 IC50 = 9 nM T63414 CDN3P6 59377867 IC50 = 12 nM T63414 CO4N7S 59377977 IC50 = 9 nM T63414 CM4EF3 59378034 IC50 = 9 nM T63414 C49IHZ 59760814 IC50 = 51 nM T63414 CO7PZ5 60168729 IC50 > 10000 nM T63414 C1IW8C 66598994 IC50 = 2.1 nM T63414 CTY7A5 66599177 IC50 = 7.9 nM T63414 C7W6RA 66599198 IC50 = 1.9 nM T63414 CFH6T5 66599261 IC50 < 10 nM T63414 CV6YT7 66599277 IC50 = 9.7 nM T63414 CB2U9J 67460623 Ki = 54.2 nM T63414 C0PK9J 70684134 IC50 = 13 nM T63414 C1XWD2 70690419 IC50 = 1400 nM T63414 CNW4E7 70690420 IC50 = 2800 nM T63414 CZ60JU 70692584 IC50 = 4.9 nM T63414 CL0JG7 70692585 IC50 = 210 nM T63414 C6IE1L 70794829 IC50 = 21 nM T63414 CH9Q0R 71450180 IC50 > 10000 nM T63414 CR64QG 71457337 IC50 > 10000 nM T63414 CR1L5W 71459185 IC50 = 1270 nM T63414 CSV43Z 71459189 IC50 > 10000 nM T63414 C0Y1JN 71462707 IC50 > 10000 nM T63414 CY9HC1 71464744 IC50 = 217 nM T63414 CIV3A7 71464745 IC50 = 666 nM T63414 CXH37V 71464746 IC50 = 220 nM T63414 CA1YJ5 71464747 IC50 = 133 nM T63414 CIU6C4 71464792 IC50 = 913 nM T63414 C31QEJ 71464793 IC50 = 72 nM T63414 CK5X2U 71464795 IC50 = 423 nM T63414 CJD57F 71464849 IC50 = 4880 nM T63414 CEO40G 71465164 IC50 = 3820 nM T63414 CU59BL 71465203 IC50 = 885 nM T63414 CP5CQ4 71465253 IC50 = 1820 nM T63414 CBI48D 71465254 IC50 = 1620 nM T63414 CIJ98Q 71465297 IC50 = 574 nM T63414 CATI79 71465298 IC50 = 789 nM T63414 CQV0T9 71465299 IC50 = 1010 nM T63414 CNUP45 71465300 IC50 = 5730 nM T63414 CH0FQ9 71465345 IC50 = 4990 nM T63414 CL03EH 71465347 IC50 = 11700 nM T63414 CAG4Z9 71465348 IC50 = 5650 nM T63414 C0AMR2 71465349 IC50 = 8770 nM T63414 CP5SD6 71465398 IC50 = 133 nM T63414 C3SWP9 71465399 IC50 = 7220 nM T63414 C6X3UJ 71465489 IC50 = 3760 nM T63414 CF2EL6 71466065 IC50 = 2140 nM T63414 CA65EM 71466067 IC50 = 1200 nM T63414 C4JH5Q 71466147 IC50 = 3430 nM T63414 CTZ90M 71466149 IC50 = 66 nM T63414 C6I0RB 71466213 IC50 = 107 nM T63414 CY5RP0 71466214 IC50 = 12 nM T63414 CQ5M0F 71466215 IC50 = 23 nM T63414 CNKP68 71466216 IC50 = 21 nM T63414 CLV2M3 71466284 IC50 = 131 nM T63414 C0VWJ2 71466285 IC50 = 25 nM T63414 C8C0KV 71466286 IC50 = 17 nM T63414 C60JFN 71466340 IC50 = 664 nM T63414 CUDK53 71466341 IC50 = 583 nM T63414 C4BOQ5 71466342 IC50 = 215 nM T63414 CBOT16 71466343 IC50 = 710 nM T63414 C5SAP9 71466396 IC50 = 30 nM T63414 C9YK3U 71466397 IC50 = 60 nM T63414 CIY5D8 71466398 IC50 = 169 nM T63414 CPV4S3 71466399 IC50 = 99 nM T63414 CNI81D 71466472 IC50 = 32 nM T63414 C5ELV2 71466473 IC50 = 166 nM T63414 C3YA7I 71466474 IC50 = 14 nM T63414 C80BPO 71466475 IC50 = 361 nM T63414 CJPR13 71625847 Ki = 12.59 nM T63414 C3U1YM 73669299 IC50 = 95200 nM T63414 C59FZS 76310220 IC50 = 3981.07 nM T63414 C4VIN2 76313910 IC50 = 3981.07 nM T63414 CB69EX 76324694 IC50 > 100000 nM T63414 C2BE9J 76853227 IC50 = 1.5 nM T63414 CS2N0Z 78153059 IC50 = 1.3 nM T63414 CQMB31 85470872 IC50 = 3.467 nM T63414 CA1CE3 86270720 IC50 = 4 nM T63414 C9TE7X 86271008 IC50 = 15 nM T63414 CMZV56 86271009 Ki = 40 nM T63414 CXN93A 86271108 IC50 = 2.188 nM T63414 C2KHM0 86271111 IC50 = 26 nM T63414 CN9MO7 86271494 IC50 = 4.8 nM T63414 CD6IJ1 86271658 IC50 = 4 nM T63414 CU4H0C 86271659 IC50 = 12 nM T63414 C5LD6M 86271660 IC50 = 89 nM T63414 C6ND4T 86271664 IC50 = 9 nM T63414 CWZ13M 86271758 IC50 = 14 nM T63414 C0D6MG 86271759 IC50 = 5 nM T63414 C3QR6J 86271850 IC50 = 10 nM T63414 CH3I6S 86271851 IC50 = 34 nM T63414 C2PE9L 86271853 IC50 = 78 nM T63414 C87QHD 86271941 IC50 = 9 nM T63414 CY01FH 86271942 IC50 = 30 nM T63414 CS74NP 86279014 IC50 = 6960 nM T63414 CQVL07 86279015 IC50 = 216 nM T63414 C6DX8V 86279088 IC50 = 3.4 nM T63414 C53GEN 86279089 IC50 = 72 nM T63414 C0ST4V 86279091 IC50 = 3.6 nM T63414 C58YOW 86279280 IC50 = 440 nM T63414 CW9KT6 86279350 IC50 = 1 nM T63414 C2NZE7 86279351 IC50 = 3.4 nM T63414 C4HLA3 86279411 IC50 = 4710 nM T63414 C38CMG 86279412 IC50 = 0.7 nM T63414 C5PLE7 86279413 IC50 = 0.2 nM T63414 C1EJ2H 86279414 IC50 = 0.5 nM T63414 CW7VE6 86279479 IC50 = 4.2 nM T63414 C7ETD9 86279481 IC50 = 0.5 nM T63414 C80FHL 86279482 IC50 = 0.6 nM T63414 CA35JQ 86279547 IC50 = 1.9 nM T63414 CR15JV 86279548 IC50 = 0.7 nM T63414 C5OM4Q 86279551 IC50 = 3.8 nM T63414 C8HK2T 86279746 IC50 = 4.3 nM T63414 CPJV10 86280878 IC50 = 19 nM T63414 C9ZS2N 86281547 IC50 = 28.1 nM T63414 C86FUO 86281680 IC50 = 4.5 nM T63414 CE68GI 86281948 IC50 = 240 nM T63414 CC3Z1H 86281949 IC50 = 8.5 nM T63414 CYK2T9 86282366 EC50 = 158 nM T63414 CA74MT 86282635 IC50 = 10 nM T63414 C3AS7V 86716303 IC50 = 0.79 nM T63414 CJ2NE0 88884677 IC50 = 9 nM T63414 CH8JM7 88954244 IC50 = 25 nM T63414 CO8M2K 90407576 Ki = 15.4 nM T63414 CA47VK 90408538 Ki = 22 nM T63414 CTC8B5 90408742 IC50 = 3538 nM T63414 CFG74P 90408756 IC50 = 7.3 nM T63414 CE4IT5 90408860 IC50 = 10 nM T63414 CZB5W4 90408922 IC50 = 880 nM T63414 C3E1CS 90409007 IC50 = 14 nM T63414 C1VA4O 90409557 IC50 = 1.9 nM T63414 C67XEH 90409637 IC50 = 114 nM T63414 CJ6E1S 90409668 IC50 = 28 nM T63414 CJPC93 90410264 IC50 = 1.7 nM T63414 C2FKB3 90410598 IC50 = 8 nM T63414 CB0RP3 90410604 IC50 = 8.318 nM T63414 CQ8ZW3 90410911 IC50 = 5.37 nM T63414 C2ZSD8 90444843 IC50 = 65 nM T63414 CR8KM2 90452359 IC50 = 77 nM T63414 CN9Y7U 90452374 IC50 = 12 nM T63414 C1EVN3 90455889 IC50 = 1.8 nM T63414 CAGK52 90456097 IC50 = 2 nM T63414 C5EC1H 90456171 IC50 = 19 nM T63414 C2JP5R 102004341 IC50 = 4.9 nM T63414 C4YI1F 108870288 IC50 = 3380 nM T63414 C1VF4Q 108870345 IC50 = 6750 nM T63414 CEFX57 117614925 IC50 = 14 nM T63414 CC5H9Y 117614990 IC50 = 11 nM T63414 C73LFS 118001660 IC50 = 809 nM T63414 CC37SU 118001939 IC50 = 810 nM T63414 CF57IP 118289475 IC50 = 18 nM T63414 C1YHC2 118566570 IC50 = 8.2 nM T63414 C9XV8C 118566572 IC50 = 36 nM T63414 C81DBJ 118566586 IC50 = 94 nM T63414 C0Z8PK 118566589 IC50 = 47 nM T63414 C16QEP 118566591 IC50 = 19 nM T63414 CGLB17 118566597 IC50 = 18 nM T63414 CWT5D6 118566606 IC50 = 140 nM T63414 C6VOL1 118566607 IC50 = 37 nM T63414 CCT20R 118566608 IC50 = 72 nM T63414 CSZ90X 118566610 IC50 = 89 nM T63414 C3H4AL 118566616 IC50 < 10 nM T63414 CY8P1K 118566647 IC50 = 27 nM T63414 C8XAS5 118566649 IC50 = 50 nM T63414 COZ29M 118566667 IC50 = 4.5 nM T63414 CM2YC8 118569729 IC50 = 230 nM T63414 CUI9F8 118569766 IC50 = 10 nM T63414 C2YU9O 118733180 IC50 = 14 nM T63414 CC74NF 118733181 IC50 = 12000 nM T63414 CQ5B1O 118733182 IC50 = 8960 nM T63414 C4T6YE 118733183 IC50 = 1970 nM T63414 CD26ZV 118733184 IC50 = 12200 nM T63414 CBI29Y 118733185 IC50 = 7720 nM T63414 CFCN02 118733187 IC50 = 355 nM T63414 CHWJ79 118733188 IC50 = 2290 nM T63414 C8F5WU 118733189 IC50 = 15 nM T63414 C9W3EM 118733190 IC50 = 27 nM T63414 CU5LV0 118733191 IC50 = 81 nM T63414 CPI50J 118733192 IC50 = 49 nM T63414 C03PZR 118733193 IC50 = 29 nM T63414 CVQU96 118733194 IC50 = 50 nM T63414 C69ZDL 118733195 IC50 = 542 nM T63414 CSQ21V 118733196 IC50 = 847 nM T63414 CXN07V 118733197 IC50 = 1670 nM T63414 C19UPL 118733198 IC50 = 3240 nM T63414 CAO73D 118949526 IC50 = 6.9 nM T63414 C79OSH 118949550 IC50 = 14 nM T63414 C7VL6I 118949555 IC50 = 1.4 nM T63414 C2KE6S 118949557 IC50 = 3.9 nM T63414 CN56FH 118949563 IC50 = 7.7 nM T63414 C8XWC1 118949568 IC50 = 15 nM T63414 CKL65X 118949576 IC50 = 23 nM T63414 CZQJ64 118949580 IC50 = 1670 nM T63414 CC3ZQ6 118949582 IC50 = 1560 nM T63414 CC03VS 118949592 IC50 = 12 nM T63414 C9LH2E 118950072 IC50 = 8.2 nM T63414 C7CPN2 118950092 IC50 = 8.7 nM T63414 C2BM9A 118950093 IC50 = 29 nM T63414 C4I2CJ 118950115 IC50 = 2.4 nM T63414 CWR8M4 118950147 IC50 = 7.7 nM T63414 CK74CV 118950157 IC50 = 8 nM T63414 CET0J1 118950171 IC50 = 8.5 nM T63414 CN71LF 118950176 IC50 = 3.2 nM T63414 CR3A8E 118950327 IC50 = 10 nM T63414 CE8G3M 118950384 IC50 = 55 nM T63414 C9UHO7 118950386 IC50 = 6.3 nM T63414 C6GJ2X 118950391 IC50 = 11 nM T63414 C1HJD2 118950410 IC50 = 10 nM T63414 C3GA0C 118950451 IC50 = 8.7 nM T63414 CI9MA2 118950452 IC50 = 12 nM T63414 CP0ZM7 118950460 IC50 = 7 nM T63414 CH5CU4 118950468 IC50 = 2.7 nM T63414 CD13JM 118950470 IC50 = 1370 nM T63414 CCX9B0 118950531 IC50 > 10000 nM T63414 CKG4N5 123779233 IC50 = 875 nM T63414 CPO7N5 124125214 IC50 = 10600 nM T63414 CJ5I8K 125478479 IC50 = 5.3 nM T63414 C68WFZ 127038803 IC50 = 252 nM T63414 CL0Y3F 127040183 IC50 > 10000 nM T63414 CM6QR9 127041723 IC50 = 1000 nM T63414 CD1N6H 127041895 IC50 > 10000 nM T63414 C1Z7PJ 127045201 IC50 = 1156.1 nM T63414 C34KHO 135603818 IC50 = 897 nM T63414 C3K1CM 135960707 IC50 = 6400 nM T63414 C3MR6C 136000710 IC50 = 1253.6 nM T63414 CN1VW6 137632041 IC50 = 18000 nM T63414 C5Q2HE 137632064 IC50 = 1557000 nM T63414 C6KC4F 137632084 IC50 = 389 nM T63414 CZ81QC 137633557 IC50 = 851 nM T63414 CC93IR 137635457 IC50 = 3020 nM T63414 CM6T5X 137635730 IC50 = 138 nM T63414 C0VRU5 137637027 IC50 = 100 nM T63414 CZH73L 137638115 IC50 = 132 nM T63414 CS2X8I 137638643 IC50 = 79 nM T63414 C5AIM2 137638655 IC50 = 186 nM T63414 CV5BE6 137640398 IC50 = 58 nM T63414 CPIG47 137640412 IC50 = 2 nM T63414 C9R8EP 137640871 IC50 = 214 nM T63414 CZ3VP0 137641909 IC50 = 51 nM T63414 CG3ZK6 137644370 IC50 = 933000 nM T63414 C6YO0L 137644636 IC50 = 40 nM T63414 CC3BS8 137646461 IC50 > 10000 nM T63414 CTKZ94 137646544 IC50 = 4034 nM T63414 C7BXL2 137646572 IC50 = 2399 nM T63414 C5GS2K 137646668 IC50 > 10000 nM T63414 CH3T7M 137649164 IC50 > 10000 nM T63414 C3PI9R 137650645 IC50 = 132000 nM T63414 CEJ6I1 137651790 IC50 > 10000 nM T63414 C4X0OY 137652052 IC50 = 366000 nM T63414 CJ2NS6 137652085 IC50 = 96000 nM T63414 C86LNH 137652744 IC50 = 58 nM T63414 CRB7N0 137652989 IC50 = 501 nM T63414 CM34CG 137655633 IC50 > 10000 nM T63414 CI0Q4V 137657140 IC50 > 10000 nM T63414 CKX62S 137658719 IC50 = 562 nM T63414 CNG5A9 137659120 IC50 = 417 nM T63414 CN6C9F 137660086 IC50 = 562 nM T63414 C8IEL0 137660769 IC50 = 4070 nM T63414 CVY90C 137661206 IC50 = 2455 nM T63414 C3JKD5 137661884 IC50 = 174 nM T63414 CRX48H 142737903 IC50 = 27 nM T63414 CGYE15 142737904 IC50 > 10000 nM T63414 CH9TP6 142737905 IC50 = 244 nM T63414 C6J8QD 142737906 IC50 = 702 nM T63414 C2K3ZM 142737910 IC50 = 32 nM T63414 C7PD9T 142737911 IC50 = 249 nM T63414 CW48KL 142737912 IC50 = 3520 nM T63414 C92ATU 142737914 IC50 = 202 nM T63414 CD8ZI3 142737915 IC50 = 312 nM T63414 CZD8J6 142737916 IC50 = 7 nM T63414 CEZ87J 142737917 IC50 = 210 nM T63414 C4TR6I 142737918 IC50 = 565 nM T63414 C5PS0V 142737919 IC50 = 1440 nM T63414 C3PT7Y 142737920 IC50 = 1.49 nM T63414 C43ZJQ 142737921 IC50 > 10000 nM T63414 CUC6I0 142737923 IC50 = 26 nM T63414 CU80EL 142737924 IC50 = 22 nM T63414 CH3X6D 142737925 IC50 > 10000 nM T63414 CPN42E 142737926 IC50 = 259 nM T63414 CST93I 142737929 IC50 = 269 nM T63414 C9SPQ7 142737930 IC50 = 37 nM T63414 CJG4Q0 142737931 IC50 = 400 nM T63414 CO23GR 142737932 IC50 = 0.49 nM T63414 CU78YD 142737933 IC50 = 430 nM T63414 CIC78M 142737934 IC50 = 155 nM T63414 CB42JQ 142737935 IC50 = 896 nM T63414 CGOA34 142737938 IC50 = 64 nM T63414 C35IFV 142737939 IC50 = 13 nM T63414 CY75NU 142737940 IC50 = 0.32 nM T63414 CEOY83 142737941 IC50 > 10000 nM T63414 C0I4TF 142737942 IC50 = 202 nM T63414 C0O4LP 142737943 IC50 = 143 nM T63414 C28KQI 142737944 IC50 = 58 nM T63414 C7B2HO 142737945 IC50 = 13 nM T63414 C3ZOV5 142737950 IC50 = 1.33 nM T63414 C37UNR 142737951 IC50 = 238 nM T63414 C9CLA6 142737953 IC50 = 4.28 nM T63414 C7ZQ4N 142737954 IC50 = 41 nM T63414 CI7P6A 142737955 IC50 = 0.11 nM T63414 CH52OW 142737956 IC50 = 1.76 nM T63414 CG23WO 142737957 IC50 = 152 nM T63414 CB52JH 142737959 IC50 = 187 nM T63414 C8R5LV 142737960 IC50 = 1570 nM T63414 CTK68D 142737961 IC50 = 22 nM T63414 C6WY0F 142737963 IC50 = 4.7 nM T63414 CF7Q9W 142737965 IC50 = 159 nM T63414 C2AE5F 145949409 IC50 = 10 nM T63414 CVUB13 145951660 IC50 = 62 nM T63414 C6MJF8 145951717 IC50 = 6 nM T63414 CT3YR8 145952273 IC50 = 54 nM T63414 CLV0D9 145953487 IC50 = 85 nM T63414 C0L3XO 145953515 IC50 = 723 nM T63414 C5F8OS 145953552 IC50 = 263 nM T63414 CW1ZS3 145953795 IC50 = 621 nM T63414 CYA15N 145954765 IC50 = 434 nM T63414 CI0BL7 145954866 IC50 = 8 nM T63414 C1H3YT 145956657 IC50 = 810 nM T63414 C8N4CA 145957051 IC50 = 120 nM T63414 CUK8L0 145957428 IC50 = 335 nM T63414 CBEA20 145958746 IC50 = 10 nM T63414 CYR3O9 145959117 IC50 = 12 nM T63414 CJ5XS2 145959607 IC50 = 18 nM T63414 CXPW20 145959674 IC50 = 108 nM T63414 CLS0X7 145960885 IC50 > 10000 nM T63414 CQK90X 145961422 IC50 = 7 nM T63414 C7M1NU 145962280 IC50 = 123 nM T63414 CD9P3E 145972418 IC50 = 861 nM T63414 CVO0B7 145972899 IC50 = 888 nM T63414 C5ZPH0 145974559 IC50 = 73 nM T63414 CQH5J2 155511022 Ki = 2.5 nM T63414 CPE58H 155514125 IC50 > 15000 nM T63414 CF6LV4 155514310 IC50 > 30000 nM T63414 C8F0TD 155517593 IC50 = 19 nM T63414 C5RO9U 155518243 IC50 = 103 nM T63414 CXV48Z 155520870 IC50 = 3.6 nM T63414 C1M6UJ 155522112 IC50 = 8.5 nM T63414 C1B9FT 155522567 IC50 = 7.4 nM T63414 CF7OT4 155523772 IC50 = 230 nM T63414 CM9CW2 155526224 IC50 > 100000 nM T63414 C1NOD4 155529242 IC50 > 100000 nM T63414 CX12AU 155529713 IC50 = 8530 nM T63414 C5BC9V 155529971 IC50 > 100000 nM T63414 CH0E9W 155530155 IC50 = 3.2 nM T63414 CP83MR 155530812 IC50 = 4.5 nM T63414 COU59G 155533299 IC50 = 22 nM T63414 C9DC1A 155534002 IC50 < 10 nM T63414 CL2YH0 155539805 IC50 = 3.9 nM T63414 COD7Q8 155543044 IC50 > 100000 nM T63414 CJVB92 155551147 Ki = 1.9 nM T63414 CZ9G8K 155559078 IC50 > 100000 nM T63414 C0PYX1 155562454 IC50 > 30000 nM T63414 C06HKI 155563184 IC50 = 3.4 nM T63414 CKOT58 155566246 IC50 = 44 nM T63414 CBS9Q8 10022445 IC50 = 6.31 nM T63414 CQB54V 11497646 IC50 = 25.12 nM T63414 C3D9RS 11526539 IC50 = 15.85 nM T63414 C9KV7B 11698695 IC50 = 79.43 nM T63414 CX24BZ 11741157 IC50 = 10 nM T63414 CR7HA4 135448190 IC50 = 100 nM T63414 CPXN13 135458217 IC50 = 63.1 nM T63414 C0G7OE 135965987 IC50 = 39.81 nM T63414 CBE09L 135966074 IC50 = 125.89 nM T63414 CT9RX6 136018716 IC50 = 398.11 nM T63414 CLU32R 19796273 IC50 = 15.85 nM T63414 CS3Q5J 23725174 IC50 = 79.43 nM T63414 C93RSL 24894834 IC50 = 1 nM T63414 CJBV47 24994779 IC50 = 398.11 nM T63414 CU8FD3 25013922 IC50 = 0.3981 nM T63414 C0WH3T 2818099 IC50 = 3981.07 nM T63414 CH96RX 45267182 IC50 = 199.53 nM T63414 CE2A7D 45267983 IC50 = 0.07943 nM T63414 CB1KJ0 45268902 IC50 = 31.62 nM T63414 C90SVN 45269779 IC50 = 316.23 nM T63414 C46KDJ 45270539 IC50 = 1.259 nM T63414 C89OVT 45271362 IC50 = 15.85 nM T63414 CYFG04 45271369 IC50 = 3.162 nM T63414 CDK3Y5 45271370 IC50 = 2.512 nM T63414 C23POI 45271376 IC50 = 79.43 nM T63414 COU15N 45273183 IC50 = 199.53 nM T63414 C2DL7Y 9865961 IC50 = 3.981 nM T63414 D00QLM 91557 EC50 > 100000 nM T63414 D02TNK 16121950 IC50 = 1800 nM T63414 D05DLI 16121949 IC50 = 700 nM T63414 D05QLT 11673921 IC50 = 123.03 nM T63414 D07QYU 4881 IC50 = 1180 nM T63414 D08DOG 25130235 IC50 > 100000 nM T63414 D0B1KT 15953802 IC50 > 10000 nM T63414 D0H2MA 6324599 IC50 = 536 nM T63414 D0M0XC 53325875 IC50 = 6.607 nM T63414 D0N6ES 5312126 IC50 = 12.59 nM T63414 D0Q1PO 53325874 IC50 = 9 nM T63414 D0U5ML 23232014 IC50 = 39.81 nM T53350 C1GR4N 9828276 IC50 = 10 nM T53350 C32JRZ 9843079 IC50 = 19000 nM T53350 CSM41Q 9849291 IC50 = 93 nM T53350 C94WDV 9858438 IC50 = 23 nM T53350 C4P5GL 9868381 IC50 = 60 nM T53350 CJ8DP1 9868672 IC50 = 290 nM T53350 CX9N3C 9870477 IC50 = 410 nM T53350 CU3TI0 9873209 IC50 = 73 nM T53350 C9KUZ3 9880993 IC50 = 31 nM T53350 CCO0V9 9885413 IC50 = 4500 nM T53350 CBD1T3 9887686 IC50 = 1000 nM T53350 CD79UJ 9890632 IC50 = 7 nM T53350 C5DW9S 9902427 IC50 = 28 nM T53350 C8NP7J 9915263 IC50 = 30 nM T53350 C1P5HF 9916545 Ki = 8 nM T53350 C5QFN3 9922714 IC50 = 122 nM T53350 CN4YK1 9923900 IC50 = 17 nM T53350 CG1A6B 9924640 IC50 = 9.3 nM T53350 CC5R1I 9925298 IC50 = 24 nM T53350 CPU59E 9928357 IC50 = 3000 nM T53350 C1OUM6 9936924 IC50 = 470 nM T53350 CMI06Q 9939403 Ki = 43 nM T53350 CWZC93 9947332 IC50 = 21 nM T53350 CZA4H5 9967696 IC50 = 21 nM T53350 CH4SM7 9968401 IC50 = 19 nM T53350 C8AQV3 9968741 IC50 = 2 nM T53350 CTC47X 9968907 IC50 = 92 nM T53350 C8K5VD 9969928 IC50 = 33 nM T53350 CC9KU8 9982365 IC50 = 9600 nM T53350 CM4AL0 10001331 IC50 = 160 nM T53350 C6MXW1 10054053 Ki = 7 nM T53350 CVTD42 10078499 Ki = 100 nM T53350 CYE7V4 10109052 IC50 = 23 nM T53350 CJG06C 10109498 IC50 = 10 nM T53350 CQ95BV 10109888 IC50 = 30 nM T53350 C9FGV3 10110893 IC50 = 98 nM T53350 CY6HZ7 10111132 IC50 = 26 nM T53350 CV9CN8 10111662 IC50 = 17 nM T53350 CQ0B1I 10112489 IC50 = 15 nM T53350 CHC04U 10112623 IC50 = 21 nM T53350 CJD98F 10117482 IC50 = 17 nM T53350 C6O2CN 10132603 IC50 = 6 nM T53350 CC4W1H 10132648 IC50 = 45 nM T53350 CZM7F4 10132758 IC50 = 36 nM T53350 CG1WB8 10133038 IC50 = 25 nM T53350 CH7A1G 10133089 IC50 = 23 nM T53350 CE0TP5 10134393 IC50 = 5 nM T53350 CI83LM 10136534 IC50 = 57 nM T53350 CXVW40 10155383 IC50 = 14 nM T53350 CXR42J 10155792 IC50 = 3 nM T53350 CIU30R 10156141 IC50 = 6 nM T53350 C23GXV 10159719 IC50 = 17 nM T53350 C0XWZ7 10160466 IC50 = 88 nM T53350 CF81HQ 10179230 IC50 = 17 nM T53350 CNK76U 10179252 IC50 = 38 nM T53350 C0F6JV 10180091 IC50 = 30 nM T53350 CEWF13 10180993 IC50 = 65 nM T53350 CW9DP6 10182462 IC50 = 26 nM T53350 CDS9A3 10184459 IC50 = 33 nM T53350 CJ64WB 10204279 IC50 = 26 nM T53350 CQI6D5 10205950 IC50 = 14 nM T53350 CYS9I2 10222243 IC50 = 25 nM T53350 CPSX26 10256361 Ki = 14 nM T53350 C1LR9B 10269446 IC50 = 29 nM T53350 CIRH04 10270164 IC50 = 6 nM T53350 CBE81L 10270207 IC50 = 17 nM T53350 C7HZ1M 10270281 IC50 = 32 nM T53350 C9P6RD 10271010 IC50 = 43 nM T53350 C3XD1E 10271240 IC50 = 21 nM T53350 C2MES9 10271604 Ki = 11 nM T53350 CSMH63 10272472 IC50 = 26 nM T53350 CWJ02G 10273315 IC50 = 37 nM T53350 CA6W7R 10279808 IC50 = 1.8 nM T53350 CU6QR7 10291655 IC50 = 324 nM T53350 CJTV12 10293283 IC50 = 8 nM T53350 C1JDV9 10294045 IC50 = 13 nM T53350 C5KW8A 10297713 IC50 = 107 nM T53350 CX6GU9 10462047 IC50 = 26 nM T53350 CE7G5A 10570770 IC50 = 18000 nM T53350 CB20LM 10594000 IC50 = 16000 nM T53350 C9OIB3 10686890 IC50 = 112000 nM T53350 CR3Q8Z 10691191 IC50 = 29000 nM T53350 C2DZT7 11399358 IC50 = 380 nM T53350 CAK3T6 11857267 IC50 = 300 nM T53350 C7GMV4 15923505 IC50 = 67 nM T53350 C81HZU 16748676 IC50 = 116 nM T53350 CM9A3U 16748677 IC50 = 154 nM T53350 CIA12S 16748678 IC50 = 32 nM T53350 CHJ8F5 16748680 IC50 = 3 nM T53350 CG7PV5 16748681 IC50 = 184 nM T53350 CT9B6F 16748784 IC50 = 6 nM T53350 CY9B0N 16748785 IC50 = 14 nM T53350 CU8WG1 16748786 IC50 = 74 nM T53350 CJ5RN8 16748788 IC50 = 46 nM T53350 C6F9LM 16748789 IC50 = 6 nM T53350 C0D4MW 16748790 IC50 = 59 nM T53350 CP05WD 16748896 IC50 = 18 nM T53350 CO2Q0D 16748897 IC50 = 13 nM T53350 C5VYB0 16748898 IC50 = 28 nM T53350 CXB10H 16748901 IC50 = 6 nM T53350 CYZ7R6 16749000 IC50 = 28 nM T53350 CJ1V6K 18325275 IC50 = 34000 nM T53350 C9FH2C 18337540 IC50 = 53 nM T53350 CR7JL9 18678862 IC50 = 1700 nM T53350 CG23VF 18678893 IC50 = 42000 nM T53350 C9EL0C 18678910 IC50 = 6700 nM T53350 CCX05P 18678912 IC50 = 900 nM T53350 C0XA5P 18678938 IC50 = 9100 nM T53350 CES6T4 23553780 IC50 = 8100 nM T53350 CL5C3M 23553781 IC50 = 81000 nM T53350 CA70EU 23553786 IC50 = 1000 nM T53350 CH4LV7 44273823 IC50 = 4.6 nM T53350 C5SW2F 44273953 IC50 = 37 nM T53350 CO4YF9 44273954 IC50 = 30 nM T53350 CLB7X0 44273997 IC50 = 200 nM T53350 C8NOD4 44273998 IC50 = 32 nM T53350 CE1NZ7 44273999 IC50 = 27 nM T53350 CT46MN 44274026 IC50 = 10 nM T53350 CN3WI7 44274027 IC50 = 860 nM T53350 C9ZL8U 44274028 IC50 = 9 nM T53350 C9FDN7 44274049 IC50 = 290 nM T53350 CH0OQ4 44274050 IC50 = 610 nM T53350 CY4MW8 44274066 IC50 = 670 nM T53350 CS6DI7 44274067 IC50 = 60 nM T53350 C72GYW 44274068 IC50 = 590 nM T53350 C2RI4D 44274069 IC50 = 32 nM T53350 C1WI6L 44274070 IC50 = 3.9 nM T53350 CTZ4I5 44274085 IC50 = 180 nM T53350 CY6W3R 44274086 IC50 = 592 nM T53350 CEG7R4 44274087 IC50 = 200 nM T53350 CE8H6I 44274103 IC50 = 170 nM T53350 C0IZ1H 44274105 IC50 = 120 nM T53350 CP3QO4 44274112 IC50 = 230 nM T53350 C1ASR6 44274113 IC50 = 230 nM T53350 CK20ZL 44274114 IC50 = 490 nM T53350 C43QAO 44274115 IC50 = 26 nM T53350 CUHA75 44274116 IC50 = 14 nM T53350 C9NWA5 44274119 IC50 = 210 nM T53350 CJE3L8 44274120 IC50 = 80 nM T53350 CAR8E4 44274121 IC50 = 110 nM T53350 CT6ZL8 44274122 IC50 = 180 nM T53350 C3TU4Y 44274123 IC50 = 260 nM T53350 CM49SA 44274124 IC50 = 120 nM T53350 CX9KL8 44274125 IC50 = 60 nM T53350 CJB2P6 44274138 IC50 = 440 nM T53350 CNOR83 44274139 IC50 = 190 nM T53350 C1UJ9L 44274140 IC50 = 24 nM T53350 C9I0LH 44274141 IC50 = 440 nM T53350 CR86EB 44274143 IC50 = 45 nM T53350 C3A0SC 44274144 IC50 = 40 nM T53350 CF1J9A 44274147 IC50 = 40 nM T53350 C38ALF 44274154 IC50 = 150 nM T53350 C72XAT 44274155 IC50 = 220 nM T53350 C9M4WO 44274156 IC50 = 390 nM T53350 CXO3T1 44274172 IC50 = 18 nM T53350 CK81FD 44274173 IC50 = 16 nM T53350 C96AKO 44274203 IC50 = 110 nM T53350 C21PRN 44274204 IC50 = 360 nM T53350 C27ZDC 44274205 IC50 = 100 nM T53350 CWTA79 44274218 IC50 = 70 nM T53350 CMCU38 44274219 IC50 = 220 nM T53350 CAM42I 44274231 IC50 = 36 nM T53350 C7PQW0 44274236 IC50 = 220 nM T53350 CZ2C1V 44274249 IC50 = 24 nM T53350 C59QHS 44274259 IC50 = 0.024 nM T53350 C4AC8N 44274266 IC50 = 93 nM T53350 C2KW9H 44274279 IC50 = 23 nM T53350 CSI8T7 44274281 IC50 = 52 nM T53350 CU5HD8 44274283 IC50 = 90 nM T53350 C4YK7D 44274293 IC50 = 380 nM T53350 C08XYH 44274294 IC50 = 350 nM T53350 CH1VP7 44274296 IC50 = 80 nM T53350 CBFJ67 44274297 IC50 = 50 nM T53350 CEFC32 44274298 IC50 = 76 nM T53350 CRKY46 44274304 IC50 = 50 nM T53350 C3AQ6Z 44274305 IC50 = 470 nM T53350 C8O2UH 44274306 IC50 = 380 nM T53350 CB57JP 44274308 IC50 = 6 nM T53350 CJ4MF1 44274321 IC50 = 23 nM T53350 C4OAW3 44274325 IC50 = 280 nM T53350 C79DWQ 44274335 IC50 = 490 nM T53350 C1K6BZ 44274336 IC50 = 470 nM T53350 CY9FG8 44274337 IC50 = 28 nM T53350 C3KE8M 44274338 IC50 = 250 nM T53350 C6TS1K 44274339 IC50 = 230 nM T53350 C31AUX 44274344 IC50 = 140 nM T53350 C4WTX2 44274345 IC50 = 130 nM T53350 C5Z1BX 44274346 IC50 = 120 nM T53350 C5HT9O 44298830 Ki = 530 nM T53350 C01FXR 44305976 IC50 = 170 nM T53350 C8TCI0 44305987 IC50 = 7800 nM T53350 C80BHF 44306001 IC50 = 6900 nM T53350 C47FRM 44306006 IC50 = 5500 nM T53350 CB83EW 44306022 IC50 = 5900 nM T53350 C1QEZ4 44306024 IC50 = 4000 nM T53350 CA65HW 44306031 IC50 = 160 nM T53350 CJP86D 44306032 IC50 = 110 nM T53350 C4Z3SB 44306046 IC50 = 5000 nM T53350 CI74SL 44306059 IC50 = 160 nM T53350 C2L3DS 44306061 IC50 = 140 nM T53350 CDAO08 44306089 IC50 = 1600 nM T53350 CQ54SA 44306104 IC50 = 45 nM T53350 C04ATH 44306105 IC50 = 38 nM T53350 CL81ID 44306111 IC50 = 4500 nM T53350 CJD9F3 44306112 IC50 = 1700 nM T53350 CAK90V 44306133 IC50 = 3400 nM T53350 CS5JA7 44306166 IC50 = 990 nM T53350 C8R5ED 44306169 IC50 = 61000 nM T53350 CYQA43 44306173 IC50 = 1600 nM T53350 CQ59PY 44306174 IC50 = 1400 nM T53350 CB5DP9 44306197 IC50 = 2300 nM T53350 CYH0S5 44306198 IC50 = 120 nM T53350 CD0EC6 44306207 IC50 = 23000 nM T53350 CFP38L 44306216 IC50 = 260 nM T53350 CUQ3M0 44306231 IC50 = 2300 nM T53350 CK1AZ5 44306250 IC50 = 58 nM T53350 C59LJH 44306251 IC50 = 50 nM T53350 CCJD47 44306255 IC50 = 910 nM T53350 CT4ER7 44306282 IC50 = 230 nM T53350 CN1X5U 44306301 Ki = 840 nM T53350 CAO79R 44306320 IC50 = 50 nM T53350 C4A1NU 44306323 IC50 = 97 nM T53350 CQ73OB 44306340 IC50 = 220 nM T53350 C9JU3H 44306342 Ki = 1010 nM T53350 COA2K7 44306344 IC50 = 45 nM T53350 CJOW08 44306353 IC50 = 290 nM T53350 CKOV20 44306362 IC50 = 7200 nM T53350 CAL78Z 44306370 Ki = 530 nM T53350 C9I1FG 44306381 IC50 = 92 nM T53350 CF3N8R 44306382 IC50 = 55 nM T53350 CYGB58 44306387 Ki = 28 nM T53350 C4ZVY9 44306397 IC50 = 78 nM T53350 CRJF47 44306406 Ki = 2500 nM T53350 C5OE6X 44306446 Ki = 1960 nM T53350 CO15BI 44306454 IC50 = 970 nM T53350 CEZ4L1 44306461 Ki = 86 nM T53350 C8KLP7 44306466 IC50 = 770 nM T53350 CW76MS 44306477 IC50 = 98 nM T53350 CTF39X 44306653 IC50 = 3600 nM T53350 CTF59Q 44306688 IC50 = 2100 nM T53350 COL7D9 44306723 IC50 = 1600 nM T53350 CFR9C0 44306781 Ki = 350 nM T53350 C7WG8A 44306791 Ki = 18 nM T53350 C9IJA0 44306792 Ki = 22 nM T53350 C5AJC4 44306813 Ki = 250 nM T53350 CDSF90 44306881 Ki = 960 nM T53350 CK4X2J 44306882 Ki = 410 nM T53350 C7BQ1I 44306927 Ki = 470 nM T53350 C1O2WB 44306928 Ki = 470 nM T53350 CP5XW3 44316117 Ki = 1200 nM T53350 C3FKY0 44316219 Ki = 480 nM T53350 C80EJB 44316220 Ki = 340 nM T53350 CCR96I 44316223 Ki > 40000 nM T53350 C3KO1L 44316224 Ki = 1300 nM T53350 C9JK5P 44316233 Ki = 33 nM T53350 C9OGB4 44316243 Ki = 120 nM T53350 CG0JD3 44316269 Ki = 110 nM T53350 C29VZC 44316280 Ki = 100 nM T53350 C3LDO9 44316287 Ki = 330 nM T53350 CP4DB2 44316304 Ki = 400 nM T53350 CF68JY 44316352 Ki > 40000 nM T53350 C5JU8G 44316384 Ki = 190 nM T53350 CLPI02 44316395 Ki > 40000 nM T53350 C7DR9J 44316410 Ki = 740 nM T53350 CT2WR0 44316411 Ki = 210 nM T53350 C1O6PM 44316416 Ki = 200 nM T53350 C68WVE 44316417 Ki > 1000 nM T53350 C9BW2T 44316431 Ki = 160 nM T53350 CLE51T 44316432 Ki = 620 nM T53350 CMJ5L3 44316433 Ki > 1000 nM T53350 C4TX3K 44316457 Ki = 1000 nM T53350 CP83EX 44316470 Ki = 63 nM T53350 C6Y7JO 44316471 Ki = 105 nM T53350 CD1HN0 44316491 Ki = 11 nM T53350 CAO35N 44316499 Ki = 98 nM T53350 CP46US 44316541 Ki = 40 nM T53350 CTM97P 44316585 Ki = 35 nM T53350 CJN80M 44316602 Ki = 1170 nM T53350 CO91HP 44316604 Ki = 300 nM T53350 CO6X2Z 44316605 Ki = 410 nM T53350 C20WNF 44316625 Ki = 1200 nM T53350 C0JK1Y 44316645 Ki = 280 nM T53350 CAQ56J 44316671 Ki = 15000 nM T53350 CKXI38 44316840 Ki = 90 nM T53350 C7CDN8 44316841 Ki = 260 nM T53350 CLOS38 44316842 Ki = 64 nM T53350 C9P7CY 44316843 Ki = 340 nM T53350 CJM90I 44316904 Ki = 660 nM T53350 CFX49E 44316925 Ki = 20 nM T53350 C2W9LI 44316927 Ki = 950 nM T53350 C7B9SL 44318117 IC50 = 90 nM T53350 C3SX8W 44318148 IC50 = 3400 nM T53350 CQ6TC7 44318149 IC50 = 750 nM T53350 CG2W9I 44318150 IC50 = 3000 nM T53350 C1ED4K 44318203 IC50 = 89 nM T53350 C0EH9V 44318204 IC50 = 50 nM T53350 C32ZDF 44318243 IC50 = 53 nM T53350 C24DQK 44318245 IC50 = 18000 nM T53350 C7XUE2 44318272 IC50 = 2500 nM T53350 C7G2RX 44318273 IC50 = 94 nM T53350 CBEZ01 44318274 IC50 = 130 nM T53350 CI7C8G 44318288 IC50 = 68000 nM T53350 C2F9XO 44318296 IC50 = 22000 nM T53350 CPJ16Z 44318297 IC50 > 800000 nM T53350 CWGZ92 44318298 IC50 = 200 nM T53350 CF1C9X 44318301 IC50 = 73 nM T53350 C30HZP 44318306 IC50 = 5100 nM T53350 CXK60H 44318313 IC50 = 19000 nM T53350 CA47VD 44318314 IC50 = 67000 nM T53350 C2NZ0E 44318318 IC50 = 19000 nM T53350 CO6W8R 44318319 IC50 = 15000 nM T53350 CG82RJ 44318322 IC50 = 190 nM T53350 CQI7M0 44318329 IC50 = 3600 nM T53350 CH1Q0L 44318330 IC50 = 2100 nM T53350 C03UAX 44318331 IC50 = 20000 nM T53350 C2MV3S 44318338 IC50 = 30 nM T53350 C3GRC5 44318342 IC50 = 5000 nM T53350 CZ5C6F 44318356 IC50 = 78 nM T53350 C80SHT 44318357 IC50 = 78 nM T53350 C2FKY8 44318358 IC50 = 67 nM T53350 CGL90Q 44318414 IC50 = 43 nM T53350 CQR2A6 44318427 IC50 = 32 nM T53350 C9N8LY 44318430 IC50 = 29 nM T53350 COJ62U 44318433 IC50 = 110 nM T53350 CIW74F 44318436 IC50 = 870 nM T53350 CE49MW 44318447 IC50 = 1900 nM T53350 CB7Z1P 44318448 IC50 = 500 nM T53350 C3KQ6A 44318456 IC50 = 2800 nM T53350 CRP2K0 44318459 IC50 = 1200 nM T53350 C8H9YV 44318467 IC50 = 730 nM T53350 C2GZ9S 44318550 IC50 = 90 nM T53350 CK24SZ 44318564 IC50 = 78 nM T53350 CWX35M 44318569 IC50 = 280000 nM T53350 C0T5IF 44318571 IC50 = 150 nM T53350 CXJ70N 44318604 IC50 = 200 nM T53350 CA5UZ3 44318618 IC50 = 250 nM T53350 CC28VP 44318623 IC50 = 220 nM T53350 CREH53 44318634 IC50 = 140 nM T53350 CAMI89 44318635 IC50 = 110 nM T53350 C9B7QK 44318638 IC50 = 210 nM T53350 C1X2YB 44318641 IC50 = 200 nM T53350 C9QD7J 44318698 IC50 = 44 nM T53350 CZY65J 44318699 IC50 = 43 nM T53350 CH7P8I 44318701 IC50 = 49 nM T53350 C4I6ME 44368970 IC50 = 8765 nM T53350 CIR84S 44369104 IC50 = 820 nM T53350 CC4PA1 44425137 IC50 = 75 nM T53350 C4DU9X 44425139 IC50 = 8 nM T53350 C9PE6F 44425140 IC50 = 27 nM T53350 CXAP75 44425141 IC50 = 20 nM T53350 CU5QV9 44425142 IC50 = 3 nM T53350 CW8RY1 44425150 IC50 = 6600 nM T53350 CKO5Q0 44462281 IC50 = 61 nM T53350 CP2SR3 44462304 IC50 = 65 nM T53350 C9QKB2 44462305 IC50 = 52 nM T53350 CDPC48 44462306 IC50 = 110 nM T53350 CAK94X 44563337 IC50 = 345000 nM T53350 C70UVG 44571513 IC50 = 40 nM T53350 CNLD24 44571552 IC50 > 2000 nM T53350 C8DN4W 44571586 IC50 = 73 nM T53350 C2K4VG 44571723 IC50 = 54 nM T53350 CX73PT 59033102 IC50 = 80 nM T53350 CJBV54 71450403 IC50 = 55000 nM T53350 C2OQC8 71450455 IC50 = 2200 nM T53350 CZB83P 71450456 IC50 = 400 nM T53350 C6FC0X 71450457 IC50 > 100000 nM T53350 CF2V0Z 71450458 IC50 = 28000 nM T53350 C7QK3J 71450459 IC50 = 10000 nM T53350 CGFB90 71452285 IC50 = 4700 nM T53350 CTL67I 71452286 IC50 = 42 nM T53350 CYQZ42 71452287 IC50 = 4900 nM T53350 C8J4HD 71452288 IC50 = 1700 nM T53350 CXPE73 71452290 IC50 = 40000 nM T53350 CF8YK2 71452291 IC50 = 1500000 nM T53350 CBO3M8 71452292 IC50 = 69000 nM T53350 C1KWB9 71454082 IC50 = 2300 nM T53350 CB8X0C 71454083 IC50 = 11000 nM T53350 C5J0NE 71454084 IC50 = 42000 nM T53350 CWZ7L2 71455769 IC50 = 166000 nM T53350 CQ63LJ 71455820 IC50 = 17000 nM T53350 C8YE3R 71455821 IC50 = 350 nM T53350 C7ZQB1 71455822 IC50 = 102000 nM T53350 CCDX81 71455823 IC50 = 23000 nM T53350 C10DWM 71457610 IC50 = 1000 nM T53350 CLP8O4 71457611 IC50 = 10000 nM T53350 CU69CF 71457612 IC50 = 2800 nM T53350 CUMY70 71459448 IC50 = 780 nM T53350 C5JDA8 71459505 IC50 = 73000 nM T53350 CJ15TM 71459506 IC50 = 18000 nM T53350 CFTB42 71459507 IC50 = 67000 nM T53350 C7SB0J 71459508 IC50 = 85000 nM T53350 CTBK47 71461245 IC50 = 13000 nM T53350 CGQM98 71461246 IC50 = 14000 nM T53350 CIZD69 71461247 IC50 = 9400 nM T53350 CFO6X9 71461248 IC50 = 167000 nM T53350 C6IB1K 71462974 IC50 = 7100 nM T53350 CX85QT 73346950 IC50 = 65000 nM T53350 C61RYQ 90662998 IC50 = 17000 nM T53350 CEZ3R0 91824149 IC50 < 1 nM T53350 CQ7KI2 118225750 Ki = 0.04 nM T53350 CUZ1D6 118225779 IC50 < 1 nM T53350 C4OD0K 118225789 IC50 = 32 nM T53350 CD8PA1 118225803 Ki = 0.0068 nM T53350 C6F8QV 118225829 IC50 < 1 nM T53350 C38RXZ 118225927 IC50 = 1 nM T53350 CI10PX 118225935 IC50 < 1 nM T53350 CN04JW 118225947 IC50 = 20 nM T53350 C4XUH1 118225963 IC50 = 1 nM T53350 C6E4SR 118226041 IC50 = 8 nM T53350 CLI7B8 118226146 IC50 = 25 nM T53350 C4FVJ1 135487604 IC50 = 10 nM T53350 CL9Y5Q 135678161 IC50 = 4000 nM T53350 C3AVY9 135712681 IC50 = 39 nM T53350 CJ9B6C 145963868 IC50 = 1250 nM T53350 C42AZM 145965977 IC50 > 10000 nM T53350 C8DF3N 145967770 IC50 = 160 nM T53350 CZ2XC4 145973252 IC50 = 6300 nM T53350 CZ4SB5 145976911 IC50 = 126 nM T53350 D02DQT 44274134 IC50 = 0.2 nM T53350 D0A4TC 446504 IC50 = 3000 nM T53350 D0NP8A 10370504 IC50 = 52000 nM T53350 D0P2TS 9818682 IC50 = 26 nM T49948 CNX79K 15303 IC50 = 2200 nM T49948 CFW1B7 736887 IC50 = 34000 nM T49948 CNSQ89 1241300 IC50 = 6900 nM T49948 CD2B0L 1714745 IC50 = 16000 nM T49948 CAFX17 2049595 IC50 = 79 nM T49948 C5VPU9 2735965 IC50 = 1800 nM T49948 CTVJ79 2737248 IC50 = 3400 nM T49948 CR3W9I 2769974 IC50 = 25000 nM T49948 CMP79R 2797430 IC50 = 4500 nM T49948 CY3N9K 2802558 IC50 = 280 nM T49948 C6R0PL 2811867 IC50 = 2700 nM T49948 C31SMO 2822041 IC50 = 200000 nM T49948 CDO08E 3691620 IC50 = 9000 nM T49948 CTX1Q3 4459133 IC50 = 5900 nM T49948 CXR6C0 5715203 IC50 = 530 nM T49948 C9A2SF 10658517 IC50 = 60000 nM T49948 C0KQ5I 16109339 IC50 = 82000 nM T49948 C2OT0I 16109340 IC50 = 37000 nM T49948 CKF72E 16109341 IC50 = 650 nM T49948 C13PVF 16109342 IC50 = 500000 nM T49948 C3FJH7 16109343 IC50 = 15000 nM T49948 CQ9ZK7 16109344 IC50 = 560000 nM T49948 CM4CJ3 44418971 IC50 = 6000 nM T86646 D04JEE 4946 IC50 = 4 nM T86646 D04VMT 5253 IC50 = 7200 nM T86646 D05DVP 5717 IC50 > 10000 nM T86646 D07MOX 439260 EC50 = 2600 nM T86646 D0I8FI 3779 EC50 = 30 nM T86646 D0O6IU 6041 EC50 = 6000 nM T86646 D0V4QS 135398745 Ki > 10000 nM T86646 D01VAB 2119 IC50 = 2.3 nM T86646 D08AWI 11430856 Ki > 2000 nM T86646 D0ZG9N 132337 Ki > 10000 nM T86646 CZUI83 2769 IC50 > 10000 nM T86646 CJQE97 5581 EC50 = 31 nM T86646 C4W1LV 58505 IC50 = 7000000 nM T86646 CVD0J9 66245 IC50 = 7200 nM T86646 CMWP80 121888 EC50 > 30000 nM T86646 CNWM94 489104 IC50 = 98 nM T86646 CSA6U7 489105 IC50 = 38000 nM T86646 CX6LW0 489106 IC50 = 4.3 nM T86646 C6WKB1 489107 IC50 = 25000 nM T86646 CIY21Q 547892 EC50 = 10 nM T86646 CI1O5D 9818958 IC50 = 2350000 nM T86646 CJ8LT7 9848518 IC50 > 10000 nM T86646 CT2C6K 9870702 IC50 > 10000 nM T86646 C6CZ3G 9906777 IC50 > 10000 nM T86646 CH5D3J 9928343 IC50 > 10000 nM T86646 C0FS3J 10142284 EC50 = 77 nM T86646 C6YW1R 12780318 EC50 = 20 nM T86646 C48KGC 12780320 EC50 = 30000 nM T86646 C8KVA9 14739875 IC50 = 150 nM T86646 C8D9YJ 14739876 IC50 = 43800 nM T86646 CHB84K 14739877 IC50 = 3900 nM T86646 C4QFC6 14739878 IC50 = 2900 nM T86646 CLV97P 14739879 IC50 = 192000 nM T86646 CJG6A4 14739880 IC50 = 12400 nM T86646 C2JIW3 14739881 IC50 = 61400 nM T86646 CBF70X 14739882 IC50 = 420 nM T86646 CL0ZW5 14739883 IC50 = 227000 nM T86646 CP5MC4 14739885 IC50 = 30900 nM T86646 CQBE07 14739886 IC50 = 12200 nM T86646 CB54QK 14739887 IC50 = 360000 nM T86646 CI1L9P 14739889 IC50 = 990 nM T86646 C21QMJ 14739890 IC50 = 2900 nM T86646 C25HZI 14739891 IC50 = 25800 nM T86646 CV8D7G 14739892 IC50 = 780 nM T86646 C4RO8H 14739896 IC50 = 15800 nM T86646 CIR0Q4 14739897 IC50 = 15700 nM T86646 CAQ69K 14739898 IC50 = 109000 nM T86646 C42CAQ 14739899 IC50 = 293000 nM T86646 C3XY0A 14739900 IC50 = 8400 nM T86646 C1R5FU 14739901 IC50 = 2300 nM T86646 CBQT63 14739905 IC50 = 40 nM T86646 C8NO3D 14739906 IC50 = 270 nM T86646 CD4JZ0 14739907 IC50 = 90 nM T86646 CE5LK3 14739908 IC50 = 3600 nM T86646 C6YCF8 14739909 IC50 = 3700 nM T86646 CE0PW2 16116807 EC50 > 30000 nM T86646 C8WLU1 19386048 EC50 > 30000 nM T86646 C1FRU8 44288600 IC50 > 10000 nM T86646 CJ2M7V 44329832 IC50 = 15700 nM T86646 C7YO1T 44329840 IC50 = 300 nM T86646 CNW2Y0 44336319 EC50 = 10 nM T86646 CC3D1O 45260430 EC50 > 30000 nM T86646 C0EQ5X 45264302 EC50 > 30000 nM T86646 CDI84E 71450922 IC50 > 10000 nM T86646 C5OU1T 135409492 Ki > 10000 nM T86646 C4PM9W 135515431 Ki > 10000 nM T86646 D03TPY 9885123 IC50 > 10000 nM T86646 D05KUM 135446209 Ki > 10000 nM T39321 D04XGT 31593 IC50 > 50000 nM T39321 D05EAM 4735 IC50 > 50000 nM T39321 D06IAR 60961 IC50 = 50000 nM T39321 D0NQ5I 65710 IC50 = 700000 nM T39321 CTS9E0 4624 IC50 = 8000 nM T39321 CV24FH 10228 IC50 = 208929.61 nM T39321 CKN4M5 14180 IC50 > 500000 nM T39321 C2J0PB 15048 IC50 = 8000000 nM T39321 CJ8NF1 24405 IC50 > 5000000 nM T39321 C1NQ8E 65188 IC50 = 194984.46 nM T39321 C7LF0S 68229 IC50 = 123026.88 nM T39321 CQG8F3 87216 IC50 = 3700000 nM T39321 CS4QG5 92208 Ki = 2800000 nM T39321 CQJ96I 125347 IC50 = 3100000 nM T39321 C3DS1E 446186 IC50 = 7000 nM T39321 C1CW3K 459890 IC50 = 8000 nM T39321 C6WY7U 463722 IC50 = 1800000 nM T39321 CU8B6Q 467916 IC50 = 300 nM T39321 CFU1T3 759292 IC50 = 144543.98 nM T39321 C9S2LO 4055843 IC50 = 38904.51 nM T39321 CS4KE7 5287846 IC50 = 54954.09 nM T39321 CHGO41 5363192 IC50 = 162181.01 nM T39321 CI2YH7 9924682 IC50 = 34003000 nM T39321 C9GWT6 9975183 IC50 = 600000 nM T39321 C9VF0R 9998966 IC50 > 10000000 nM T39321 CQ9RT8 10019035 IC50 > 4000000 nM T39321 CJ69UL 10029114 IC50 = 4000 nM T39321 CX6R0T 10045055 IC50 = 2400 nM T39321 C5L0IR 10049523 IC50 = 500000 nM T39321 C7G0JC 10066396 IC50 = 600 nM T39321 CHT5G7 10072244 IC50 = 200000 nM T39321 C0S3CH 10318843 IC50 = 700000 nM T39321 CR6AK3 10319600 IC50 = 400000 nM T39321 CP39MN 10334943 IC50 > 4000000 nM T39321 C76SQA 10337187 IC50 = 16982.44 nM T39321 C0LTR7 10339188 IC50 = 700000 nM T39321 CLN9P6 10341490 IC50 = 3000000 nM T39321 C8YDI5 10343681 IC50 = 6300000 nM T39321 CX1C3D 10348211 IC50 > 50000 nM T39321 C0KQT5 10360939 IC50 > 2000000 nM T39321 CWN87M 10368295 IC50 = 16000 nM T39321 CE7VQ8 10381084 IC50 > 4000000 nM T39321 CSTB14 10386525 IC50 = 200000 nM T39321 C07HWY 10393235 IC50 = 26000 nM T39321 C45RCF 10405158 IC50 = 10000 nM T39321 CRHU08 10408674 IC50 = 9000000 nM T39321 CR72DH 10428340 IC50 > 10000000 nM T39321 C0R1KB 10429225 IC50 = 3300 nM T39321 CCEL76 10431926 IC50 > 10000000 nM T39321 C2RPH3 10445321 IC50 = 1600000 nM T39321 C9NBJ1 10450657 IC50 > 4000000 nM T39321 CU25FM 10454854 IC50 = 500000 nM T39321 CKF0N9 10469836 IC50 > 2000000 nM T39321 CC3J4G 10476477 IC50 = 150000 nM T39321 C4HPM8 10528348 IC50 = 1200000 nM T39321 C4H0PY 10549805 IC50 = 600000 nM T39321 CVKI74 10620158 IC50 = 850000 nM T39321 CB4HC6 10668788 IC50 = 650000 nM T39321 CZ4QK0 10697288 IC50 = 25000 nM T39321 C87ACT 10740715 IC50 = 250000 nM T39321 C0KDO7 10792034 IC50 = 25000 nM T39321 CCSJ93 10834615 IC50 = 360000 nM T39321 C8C0TX 10835695 IC50 = 500000 nM T39321 CH6FQ5 10839640 IC50 = 5500 nM T39321 CXG08M 10940514 IC50 = 14000 nM T39321 C40FAS 10974017 IC50 = 40000 nM T39321 C4W2YD 11028195 IC50 = 7000 nM T39321 CKTO76 11028555 IC50 = 14000 nM T39321 CZF75Y 11114718 IC50 = 45000 nM T39321 C4BSO1 11124571 IC50 = 25000 nM T39321 C8T2GN 11512859 IC50 = 5000 nM T39321 C79IKG 11731457 IC50 = 12000 nM T39321 CRE0O4 11753045 IC50 = 6000 nM T39321 CH1O5K 11813682 IC50 = 12000 nM T39321 CHD9S0 11814031 IC50 = 7000 nM T39321 CN6S5T 11966381 IC50 = 8000 nM T39321 C2K4CN 15828698 IC50 = 590 nM T39321 CAF6E1 21829325 IC50 = 346736.85 nM T39321 CKQ84Y 24178170 IC50 > 10000 nM T39321 CSYD02 24863870 IC50 = 17782.79 nM T39321 C0GF7M 44306170 IC50 = 5000 nM T39321 C4NRA2 44306171 IC50 = 10000 nM T39321 CYZ5O4 44306177 IC50 = 30000 nM T39321 C7I8MA 44309784 IC50 = 85113.8 nM T39321 CAG5V7 44309804 IC50 = 5000 nM T39321 C3SI8V 44309810 IC50 = 52480.75 nM T39321 CHPX93 44309822 IC50 = 56234.13 nM T39321 C4D6ZN 44309832 IC50 = 30902.95 nM T39321 CH96VA 44309844 IC50 = 128824.96 nM T39321 CR9T2D 44309846 IC50 = 12000 nM T39321 CTK17A 44309997 IC50 = 74131.02 nM T39321 CMD14G 44310158 IC50 = 123026.88 nM T39321 CMS3I2 44310159 IC50 = 67608.3 nM T39321 CT7H5Q 44310180 IC50 = 64565.42 nM T39321 CYU58F 44310181 IC50 = 190546.07 nM T39321 CFB13G 46874050 IC50 = 240000 nM T39321 CB2UL5 46875344 IC50 = 250000 nM T39321 C90BVF 46875585 IC50 > 2000000 nM T39321 C3BPX0 46875590 IC50 = 750000 nM T39321 CS7HV0 46875985 Ki = 4000000 nM T39321 CP6K1F 46875998 Ki = 9000 nM T39321 CL1MK0 46876011 Ki = 1500000 nM T39321 C5OQ1D 46876042 Ki = 800000 nM T39321 C2QSA5 46876048 Ki = 3300000 nM T39321 C39XRD 46876082 IC50 = 8000000 nM T39321 C7Q3GH 46876205 IC50 = 340000 nM T39321 C5TMK8 46876222 IC50 > 5400000 nM T39321 CO25UZ 73356664 IC50 = 29000 nM T39321 C0Y8AZ 90662838 IC50 = 45000 nM T39321 CQT9A5 118719207 IC50 = 60 nM T39321 C0UO7C 118753751 IC50 = 100 nM T39321 CF1J8L 122185475 IC50 = 1340 nM T39321 CXHN49 122185488 IC50 = 1410 nM T39321 CUFZ63 122185495 IC50 = 2410 nM T39321 C5U1BH 135476505 IC50 = 56234.13 nM T39321 D02JEZ 5281426 IC50 = 616595 nM T39321 D03RFA 657378 IC50 > 5000000 nM T39321 D03ZMQ 323 IC50 = 691830.97 nM T39321 D05QOR 5280460 IC50 = 257039.58 nM T77400 D05GJW 20279 IC50 > 10000 nM T77400 D05MQK 110635 IC50 > 10000 nM T77400 D0C9SY 135400189 IC50 = 3100 nM T77400 D0D1HW 135409400 IC50 = 34000 nM T77400 D0E0SW 53708 IC50 = 520000 nM T77400 D0F8RA 2153 IC50 = 210000 nM T77400 D0F9GE 3108 IC50 = 3600 nM T77400 D0NJ3V 4680 IC50 = 2300 nM T77400 D0R5RR 119182 IC50 = 3120 nM T77400 D0Y9ZE 4197 IC50 = 200000 nM T77400 D0Z7ZM 135398744 IC50 > 10000 nM T77400 D01LCC 17754438 IC50 > 10000 nM T77400 D07GHV 60143346 IC50 = 1 nM T77400 D0T5PO 5092 IC50 > 16000 nM T77400 D0X0PP 59351313 IC50 > 30000 nM T77400 D01ITP 71295652 IC50 = 6 nM T77400 D05VBJ 71295299 IC50 = 69 nM T77400 D07EUB 46200734 IC50 = 2.99 nM T77400 D09BDD 56933838 IC50 = 14 nM T77400 D0WS3T 72706254 IC50 = 7900 nM T77400 D00SPK 23665864 IC50 = 15000 nM T77400 D00YPW 135399235 IC50 = 46800 nM T77400 D02EMR 151170 IC50 > 10000 nM T77400 D07FHZ 5087 IC50 = 390000 nM T77400 D08NXX 5487281 IC50 = 20000 nM T77400 D09SFV 3973 IC50 = 40000 nM T77400 D09UMA 55918 IC50 = 500000 nM T77400 D0BK6B 3021729 IC50 = 380000 nM T77400 CVQ0G5 1348 IC50 > 100000 nM T77400 C03NGJ 1713 IC50 > 100000 nM T77400 CO2Y3R 3698 IC50 = 580000 nM T77400 CH8J2B 4977 Ki = 600000 nM T77400 CCJ8F0 5353 IC50 = 200000 nM T77400 CGA17S 127779 Ki = 122000 nM T77400 CR8H1B 149028 IC50 = 68000 nM T77400 CK4VZ8 152034 IC50 = 17000 nM T77400 C0YK8A 155806 IC50 = 212000 nM T77400 COK69D 156890 IC50 = 57000 nM T77400 CH2P8A 158961 Ki = 700000 nM T77400 CVN23X 158962 Ki = 600000 nM T77400 C78DLE 205964 IC50 = 8700 nM T77400 CKH1C0 220780 Ki = 22400 nM T77400 C51LJV 223726 Ki = 6900 nM T77400 C7YV8R 656066 IC50 = 170 nM T77400 C8JLO0 2243267 IC50 = 4100 nM T77400 CWO8I2 3041753 IC50 = 108000 nM T77400 CK12OT 3814427 IC50 > 100000 nM T77400 C7BQ1N 5492386 IC50 > 100000 nM T77400 C0C9HP 6610310 IC50 > 100000 nM T77400 CB40PM 6918356 IC50 = 1300 nM T77400 CFJ62Y 9799389 IC50 > 10000 nM T77400 CZH08Y 9802738 IC50 > 20000 nM T77400 C2NK8E 9888568 IC50 = 984 nM T77400 CO87TV 9994528 IC50 > 100000 nM T77400 CB9EY5 9995187 IC50 > 100000 nM T77400 C39LZS 9999105 IC50 > 100000 nM T77400 C4ST7G 10017729 IC50 > 100000 nM T77400 C1FJ8H 10039594 IC50 > 10000 nM T77400 C2MGJ7 10117650 IC50 = 1700 nM T77400 CG8RW2 10142576 IC50 = 950 nM T77400 CB7XJ2 10216985 IC50 = 4850 nM T77400 CZ1Y8D 10232923 IC50 > 100000 nM T77400 CWG85T 10406931 IC50 = 9000 nM T77400 CF5O8D 10446136 IC50 = 33700 nM T77400 C6PXC2 10471556 IC50 > 100000 nM T77400 C4CN0V 10508072 IC50 > 100000 nM T77400 C7Z9YF 10579873 IC50 > 100000 nM T77400 C1O4KV 10626842 IC50 > 100000 nM T77400 CE65JO 10650764 IC50 > 100000 nM T77400 C9FR7P 10674875 IC50 > 100000 nM T77400 C4T8PS 10816641 IC50 > 100000 nM T77400 C41XSK 11065470 IC50 > 10000 nM T77400 C45VZC 11438405 IC50 = 40 nM T77400 C4ZYH9 11547485 IC50 > 10000 nM T77400 CUK49V 11988837 Ki = 24000 nM T77400 CFIO49 11988967 Ki = 37000 nM T77400 C2D0NG 11989101 Ki = 39000 nM T77400 C65ABT 11989102 Ki > 100000 nM T77400 C1B4XD 11992634 IC50 > 2000 nM T77400 CPX16N 11993169 IC50 > 2000 nM T77400 CE41YR 13059432 IC50 = 190000 nM T77400 C7SPV8 13233881 IC50 = 280000 nM T77400 C75JTV 13233882 IC50 = 260000 nM T77400 C9NR8P 13233885 IC50 = 71000 nM T77400 C4AK6E 13233889 IC50 = 380000 nM T77400 CZ50CU 13887375 IC50 = 190000 nM T77400 CL9KE4 13936986 IC50 = 70000 nM T77400 CB28RL 13936987 IC50 = 30000 nM T77400 CASB70 14099426 IC50 = 480000 nM T77400 CI3J7R 14099427 IC50 = 34000 nM T77400 CQ1LY8 14099432 IC50 = 39000 nM T77400 CUS17I 14099444 IC50 = 330000 nM T77400 CP5JU9 14099446 IC50 = 170000 nM T77400 C17HNR 14099449 IC50 = 110000 nM T77400 CH4S8D 14280990 IC50 = 30000 nM T77400 CD1Q4U 14280991 IC50 = 10000 nM T77400 C03ZNU 14280992 IC50 = 50000 nM T77400 CZ9WG1 14280994 IC50 = 30000 nM T77400 CL4AF3 14280995 IC50 = 10000 nM T77400 C1MK5R 14280996 IC50 = 100000 nM T77400 CCTP04 14280998 IC50 > 100000 nM T77400 CXH95F 14280999 IC50 = 100000 nM T77400 CZ6N0W 14281000 IC50 = 40000 nM T77400 CR1G8Y 14281001 IC50 = 100000 nM T77400 CJ6VF1 14281004 IC50 > 100000 nM T77400 C9MY5X 14281006 IC50 = 5500 nM T77400 CUFJ35 14281010 IC50 = 7000 nM T77400 CQ8TE3 14281011 IC50 > 100000 nM T77400 CSEC89 14281012 IC50 = 60000 nM T77400 CU0J8E 14281015 IC50 = 100000 nM T77400 CDP92K 14281016 IC50 = 6000 nM T77400 C6FCS9 14281018 IC50 = 8000 nM T77400 CUDO17 14281023 IC50 = 60000 nM T77400 CZ19AJ 14281024 IC50 = 10000 nM T77400 CY8PC6 14281025 IC50 = 5000 nM T77400 CBT8K9 14281026 IC50 = 5000 nM T77400 C3F7MZ 14281027 IC50 > 100000 nM T77400 CQ2YL0 14281033 IC50 = 50000 nM T77400 CCO0S1 15005567 IC50 > 100000 nM T77400 CW0UP4 15005571 IC50 = 7000 nM T77400 CE0DR4 15005574 IC50 = 7000 nM T77400 CAQ7J2 15005576 IC50 = 3000 nM T77400 C5Z8QA 15005579 IC50 > 100000 nM T77400 CJ72ZA 15005584 IC50 > 100000 nM T77400 CVA9B0 15005585 IC50 = 20000 nM T77400 C7QZO0 15005594 IC50 > 100000 nM T77400 CRA5G0 15005604 IC50 = 10000 nM T77400 C0X4QW 15065159 IC50 = 60000 nM T77400 CDS3L9 15065160 IC50 = 60000 nM T77400 CJAW97 15065161 IC50 > 100000 nM T77400 C1PZ8C 18734933 IC50 > 16000 nM T77400 C3LJ4B 19003750 IC50 = 58000 nM T77400 CJ95TM 20146320 IC50 = 170000 nM T77400 CW96SI 23624262 IC50 = 1000 nM T77400 C4S6VD 23654252 IC50 > 50000 nM T77400 C9WGI4 24802717 IC50 = 239 nM T77400 C20VHK 24871823 IC50 = 4560 nM T77400 C93DZI 25147798 IC50 > 50000 nM T77400 CPC08B 25179287 IC50 > 50000 nM T77400 COB03R 25179478 IC50 > 50000 nM T77400 CS7RC9 42629350 IC50 = 32 nM T77400 C7SGR9 42629353 IC50 = 75 nM T77400 C9CE2J 42629699 IC50 = 116 nM T77400 CP9TE3 42629700 IC50 = 21.9 nM T77400 CICF39 42629702 IC50 = 38 nM T77400 CMIX45 42629822 IC50 = 9.5 nM T77400 CM3X9S 42629827 IC50 = 11 nM T77400 CQN26J 42629945 IC50 = 47 nM T77400 CRX87A 42629953 IC50 = 14 nM T77400 C6O5FX 42630062 IC50 = 37 nM T77400 CR2VK6 42630063 IC50 = 135 nM T77400 C1A4UY 42630064 IC50 = 64 nM T77400 CWT8E7 42630065 IC50 = 237 nM T77400 CTS74L 42630069 IC50 = 153 nM T77400 C3P1XN 42630071 IC50 = 70.5 nM T77400 C2O1WH 42630072 IC50 = 70 nM T77400 CGU0S3 42630073 IC50 = 21.6 nM T77400 C71ZNR 42630180 IC50 = 62 nM T77400 C9UZW3 42630188 IC50 = 22 nM T77400 CX9ZT6 42630190 IC50 = 305 nM T77400 C4RHY0 42630191 IC50 = 108 nM T77400 CT6RS9 42630192 IC50 = 92 nM T77400 CYLS05 42630193 IC50 = 66 nM T77400 C7J0PY 42630314 IC50 = 621 nM T77400 CJC7B8 42630315 IC50 = 194 nM T77400 CYZL43 42630317 IC50 = 165 nM T77400 CH42OZ 42630318 IC50 = 83 nM T77400 C7X5AH 42630437 IC50 = 30 nM T77400 C8L7XT 42630438 IC50 = 300 nM T77400 C5IVS3 42630440 IC50 = 138 nM T77400 CGV5A0 42630796 IC50 = 35.6 nM T77400 CW8OB3 44243146 Ki > 10000 nM T77400 C7NHE8 44279839 IC50 = 130000 nM T77400 CK8Y4F 44286951 IC50 > 50000 nM T77400 COBW92 44301890 IC50 = 43000 nM T77400 C8A2JP 44311854 IC50 = 89000 nM T77400 C5SBO6 44311855 IC50 = 18000 nM T77400 CQ0S7E 44386000 IC50 > 50000 nM T77400 CHDN54 44386045 IC50 = 13000 nM T77400 CBT82J 44386129 IC50 > 50000 nM T77400 CV1F8W 44386133 IC50 = 27000 nM T77400 CP37LE 44386323 IC50 = 20000 nM T77400 C69DVN 44386324 IC50 > 50000 nM T77400 CWE39G 44386327 IC50 = 14000 nM T77400 CL7OS2 44386388 IC50 = 14000 nM T77400 C2RTX1 44386433 IC50 = 44000 nM T77400 CPQC46 44386434 IC50 > 25000 nM T77400 CD8VL7 44387049 IC50 = 19000 nM T77400 CC9HR5 44387117 IC50 = 66000 nM T77400 C8ZUQ5 44411688 IC50 = 431 nM T77400 CBL2J9 45263650 IC50 = 4600 nM T77400 C0D2MN 46186792 IC50 = 4 nM T77400 CR1K5E 46198523 IC50 = 9.3 nM T77400 C58BSW 46198541 IC50 = 101.6 nM T77400 C1BIJ2 46198546 IC50 = 142 nM T77400 CC42ER 46198694 IC50 = 39.4 nM T77400 C0WRO9 46198713 IC50 = 13.2 nM T77400 CON1M4 46199019 IC50 = 14 nM T77400 C5AND7 46199167 IC50 = 28.6 nM T77400 CKX1A6 46199301 IC50 = 3.31 nM T77400 CZU0H7 46199329 IC50 = 14.4 nM T77400 CD9LN1 46199458 IC50 = 5.31 nM T77400 CXG34R 46199487 IC50 = 15.8 nM T77400 CAL85J 46199794 IC50 = 974 nM T77400 CZF5C0 46199795 IC50 = 1950 nM T77400 CI9EA4 46199799 IC50 = 2055 nM T77400 C26RJV 46200090 IC50 = 172 nM T77400 C5WND9 46200233 IC50 = 196 nM T77400 CKIC45 46200238 IC50 = 775 nM T77400 CS46AE 46200399 IC50 = 589 nM T77400 C1S3BK 46200706 IC50 = 110 nM T77400 C4P5QJ 46200709 IC50 = 103 nM T77400 CV8Y6W 46200711 IC50 = 4.37 nM T77400 CK1N4X 46200728 IC50 = 15.1 nM T77400 CH9FU8 46200877 IC50 = 3390 nM T77400 CEZ3V4 46200878 IC50 = 35.9 nM T77400 C36XLQ 46209046 IC50 > 10000 nM T77400 C2Q4YT 46209162 IC50 > 10000 nM T77400 CJOE41 46209386 IC50 > 10000 nM T77400 C5IMB2 46239424 Ki > 10000 nM T77400 CKR9P7 46239425 Ki > 10000 nM T77400 CI1F5C 46239840 Ki >= 770 nM T77400 C26XVS 46240044 Ki >= 4793 nM T77400 CE4JU7 46842025 IC50 > 10000 nM T77400 CR8JC2 46842169 IC50 > 10000 nM T77400 C3P2IN 46933992 IC50 >= 57000 nM T77400 C3R9SZ 46957534 IC50 = 490 nM T77400 C3DH7C 49821302 IC50 = 81 nM T77400 C9Q6KE 49821304 IC50 = 36 nM T77400 CE8Y6Q 49821305 IC50 = 128 nM T77400 C3TVS5 49821396 IC50 = 71 nM T77400 CHA5Z0 49821469 IC50 = 325 nM T77400 C1AYP0 49821627 IC50 = 112 nM T77400 C85AXR 49821714 IC50 = 411 nM T77400 CZS03D 50902030 Ki > 4274 nM T77400 CH2Z1E 50902289 Ki > 7100 nM T77400 C4HJL2 50902291 Ki > 7950 nM T77400 C6A1IU 50902549 Ki > 2000 nM T77400 C3Y2AV 50903255 Ki > 2000 nM T77400 CGF65A 54670110 IC50 > 30000 nM T77400 C90ZLC 54670399 IC50 > 30000 nM T77400 COHX27 56648495 IC50 = 11.6 nM T77400 C4TGL7 56648496 IC50 = 27.5 nM T77400 C43WOF 56648497 IC50 = 19.5 nM T77400 CM3OI5 56648498 IC50 = 13.1 nM T77400 CM09EW 56648583 IC50 = 29.9 nM T77400 CIT68E 56648584 IC50 = 11.5 nM T77400 C9U0JW 56648585 IC50 = 7.4 nM T77400 C8O9PD 56648586 IC50 = 108 nM T77400 C52KXF 56648587 IC50 = 5.4 nM T77400 C9NC5E 56648588 IC50 = 276 nM T77400 CSZ6J1 56648589 IC50 = 299 nM T77400 CH6C3L 56648679 IC50 = 24.6 nM T77400 CCY79V 56648680 IC50 = 30 nM T77400 CL6Q1H 56648681 IC50 = 17 nM T77400 CR0C8I 56648683 IC50 = 24 nM T77400 C15YZK 56648684 IC50 = 40.6 nM T77400 C9Z8TP 56648763 IC50 = 18.4 nM T77400 C0HX6Z 56648767 IC50 = 40 nM T77400 C85VDI 56648768 IC50 = 89 nM T77400 CNE96P 56648857 IC50 = 23 nM T77400 CX86AQ 56648859 IC50 = 13.6 nM T77400 CLV5E3 56648860 IC50 = 14.7 nM T77400 C6QG0A 56648861 IC50 = 619 nM T77400 CL8QN3 56648862 IC50 = 501 nM T77400 C16DEO 56648951 IC50 = 42 nM T77400 CPC3T4 56654131 IC50 > 10000 nM T77400 C0YD3P 56928304 IC50 > 5000 nM T77400 C8RO6A 56929788 IC50 > 1000 nM T77400 C0ZF1L 57328385 IC50 = 2100 nM T77400 C4EGB7 57392860 IC50 = 27 nM T77400 CG3DF1 57392948 Ki > 10000 nM T77400 CE36TV 57394695 Ki > 10000 nM T77400 CPA3D1 57403394 Ki > 10000 nM T77400 C4XMB6 58547809 IC50 > 30000 nM T77400 CEB3G9 58547814 IC50 = 3030 nM T77400 C08QVG 58547833 IC50 = 11700 nM T77400 CFVG67 58547863 IC50 = 29700 nM T77400 CYZA38 58548077 IC50 = 12900 nM T77400 CWX3N7 59320301 IC50 > 10000 nM T77400 C7PB1U 59321218 IC50 = 2.06 nM T77400 CS32XI 59321284 IC50 = 346.5 nM T77400 C23WQA 59321310 IC50 = 944 nM T77400 CX45HS 59321315 IC50 = 80.6 nM T77400 CZ6C9L 59321318 IC50 = 864 nM T77400 C1OHZ0 59321339 IC50 = 722 nM T77400 C0EP5I 59341847 IC50 > 10000 nM T77400 CHQ28A 59341978 IC50 > 10000 nM T77400 CJ0YB8 59351288 IC50 > 10000 nM T77400 CCA1H6 59351376 IC50 > 10000 nM T77400 C1SX6A 60149170 IC50 = 0.3 nM T77400 C0AFM6 60150358 IC50 = 30.3 nM T77400 CE0Q1S 60152740 IC50 = 3 nM T77400 CJK53Q 60152741 IC50 = 4 nM T77400 CZ7OU4 60163253 IC50 = 8.2 nM T77400 C6C8RD 66802145 IC50 = 4900 nM T77400 C2D7LR 66967770 IC50 = 3465 nM T77400 C5BE3L 67021512 IC50 = 6100 nM T77400 CA53BN 68181843 IC50 = 2.01 nM T77400 CFV5P9 68181883 IC50 = 0.58 nM T77400 CY8J3O 68181896 IC50 = 0.53 nM T77400 C5OD4I 68181996 IC50 = 0.82 nM T77400 C8JN6C 68182075 IC50 = 1.08 nM T77400 CTJ46X 68594477 IC50 = 11.8 nM T77400 CV4X6K 68595169 IC50 = 23 nM T77400 C8E0XY 68596001 IC50 = 269 nM T77400 CJ80VI 68596013 IC50 = 1500 nM T77400 CL2H4T 68596452 IC50 = 894 nM T77400 C93IHS 68596628 IC50 = 2375.5 nM T77400 CDZ01B 68596639 IC50 = 1150 nM T77400 C1CD9S 68596902 IC50 = 50.4 nM T77400 C7PCW0 68597211 IC50 = 1998 nM T77400 CGJB21 68597401 IC50 = 3420 nM T77400 CHK4S0 68597804 IC50 = 1270 nM T77400 C10TGO 68598825 IC50 = 1220 nM T77400 CHX52Y 69561043 IC50 = 38 nM T77400 CCN10Q 70662473 IC50 > 1000 nM T77400 COI2P3 70679302 IC50 > 10000 nM T77400 CM3OP8 70686796 IC50 = 95.9 nM T77400 CHBT91 70686797 IC50 = 522 nM T77400 CC43LF 71074083 IC50 > 10000 nM T77400 C4P0XT 71092344 IC50 > 30000 nM T77400 C6DAG4 71092519 IC50 > 30000 nM T77400 C6VX8J 71093641 IC50 = 17.7 nM T77400 C87NJD 71114298 IC50 = 9 nM T77400 CLU1S6 71151948 IC50 = 5.9 nM T77400 CY9ZL0 71151966 IC50 = 280 nM T77400 C34XNL 71151981 IC50 = 9.7 nM T77400 C82AUP 71152059 IC50 = 2.2 nM T77400 C0C9JX 71152125 IC50 = 6.3 nM T77400 C5VUO9 71152240 IC50 = 2.8 nM T77400 CGTE48 71152251 IC50 = 30 nM T77400 CY3RW6 71152297 IC50 = 0.38 nM T77400 CN8W4I 71153086 IC50 = 6.2 nM T77400 CDZ4U5 71153104 IC50 = 21 nM T77400 C2TEH0 71153106 IC50 = 6.5 nM T77400 C1M0EN 71153110 IC50 = 4.4 nM T77400 C0M7ZG 71153186 IC50 = 29 nM T77400 CG9C3J 71153201 IC50 = 7.1 nM T77400 CT8W1G 71153209 IC50 = 10.4 nM T77400 CUW9X3 71153218 IC50 = 1.4 nM T77400 CD6C7M 71153238 IC50 = 0.28 nM T77400 C2NV4G 71153252 IC50 = 15 nM T77400 C74BDZ 71153260 IC50 = 263 nM T77400 CIM4L0 71153268 IC50 = 12.1 nM T77400 CCY3I0 71153278 IC50 = 1.7 nM T77400 CVW5J0 71153282 IC50 = 7.7 nM T77400 CH51WI 71153284 IC50 = 28 nM T77400 CYX69F 71153287 IC50 = 123 nM T77400 C3V5ZM 71153302 IC50 = 4.8 nM T77400 C40HNF 71153309 IC50 = 0.6 nM T77400 CM9DL8 71153318 IC50 = 8.9 nM T77400 C9NRH4 71153321 IC50 = 0.47 nM T77400 C0B4QF 71153327 IC50 = 39 nM T77400 CF7C0J 71153330 IC50 = 0.42 nM T77400 C3DT6Q 71153343 IC50 = 24 nM T77400 C2PE4N 71153351 IC50 = 6.3 nM T77400 C2HGI7 71153408 IC50 = 10 nM T77400 CU8MY9 71153417 IC50 = 30.5 nM T77400 CZTL75 71153427 IC50 = 6.1 nM T77400 C9GR3L 71153436 IC50 = 2.8 nM T77400 CP2SO9 71295337 IC50 = 15 nM T77400 C7LRS9 71305062 IC50 = 45 nM T77400 CR5NQ6 71450591 IC50 > 10000 nM T77400 CGD56M 71450592 IC50 > 10000 nM T77400 CZ1YN2 71452430 IC50 > 10000 nM T77400 CI1M8Q 71452431 IC50 > 10000 nM T77400 CKD9F3 71453591 IC50 = 16800 nM T77400 CX5D2O 71454197 IC50 > 10000 nM T77400 CJV1G2 71455939 IC50 > 10000 nM T77400 C8A4ME 71457746 IC50 > 10000 nM T77400 C3VKH8 71459650 IC50 > 10000 nM T77400 CT2D6E 71461384 IC50 > 10000 nM T77400 C5WS8U 71488840 IC50 = 2 nM T77400 CT4G2Y 71488842 IC50 = 3.4 nM T77400 C5D4IR 71488864 IC50 = 1.6 nM T77400 C4ES6V 71498916 IC50 = 5 nM T77400 CS61KO 71520599 IC50 = 19 nM T77400 C9MO5E 71520601 IC50 = 20 nM T77400 CIEW64 71520602 IC50 = 15 nM T77400 CT3IN6 71520691 IC50 = 7.3 nM T77400 C1D7QX 71520692 IC50 = 12 nM T77400 C71QXS 71520693 IC50 = 24 nM T77400 C4GNJ3 71598545 IC50 > 1000 nM T77400 CR9UP6 71624530 IC50 = 102 nM T77400 C2YCS7 71624531 IC50 = 54 nM T77400 C40NTG 71624532 IC50 = 23 nM T77400 C8RDG9 71624638 IC50 = 328 nM T77400 C7LFJ0 71624639 IC50 = 93 nM T77400 C03GMI 71624640 IC50 = 44 nM T77400 CZ4KC3 71624641 IC50 = 105 nM T77400 CUWS89 71624642 IC50 = 97 nM T77400 C5NU1X 71624751 IC50 = 505 nM T77400 CPBJ05 71624752 IC50 = 483 nM T77400 CFD0X9 71624753 IC50 = 586 nM T77400 CMQ7N9 71624754 IC50 = 156 nM T77400 C4FC1W 71624755 IC50 = 46 nM T77400 CO7X9M 71624869 IC50 = 14 nM T77400 C3OTL4 71624870 IC50 = 40 nM T77400 C4WN1T 71624871 IC50 = 70 nM T77400 C2UZC5 71624872 IC50 = 36 nM T77400 CZF6X3 71624873 IC50 = 18 nM T77400 CBX7F6 71624993 IC50 = 7 nM T77400 CJ1K6H 71624994 IC50 = 6.8 nM T77400 CG9ZJ8 71624995 IC50 = 1.3 nM T77400 CFL69D 71624996 IC50 = 3.4 nM T77400 CV69IU 71624997 IC50 = 9.3 nM T77400 C16JZP 71625120 IC50 = 1.2 nM T77400 C5CQM8 71625121 IC50 = 1.4 nM T77400 C7XL9G 71625122 IC50 = 1.8 nM T77400 C2N1FS 71625123 IC50 = 2.5 nM T77400 C61ULV 71625124 IC50 = 2.5 nM T77400 C7Z5GP 71625256 IC50 = 3 nM T77400 C9HG4F 71682930 IC50 = 1.72 nM T77400 C68SDB 71719394 IC50 = 6309.57 nM T77400 CZ0G2X 72165213 IC50 > 10000 nM T77400 C7XRY6 72190879 IC50 = 0.61 nM T77400 CM0PF5 72190880 IC50 = 1.6 nM T77400 CQ3GD7 72704434 Ki = 18000 nM T77400 CBM61I 73293715 IC50 > 10000 nM T77400 CHR7D0 73334611 IC50 = 1860 nM T77400 CS5XE8 73353458 IC50 = 840 nM T77400 C56RIA 73354963 IC50 = 259 nM T77400 C9ODB8 73387740 IC50 = 1320 nM T77400 C5X6GJ 73387742 IC50 = 12900 nM T77400 CT1E6V 73387743 IC50 = 3520 nM T77400 C7D1SJ 73387744 IC50 = 5390 nM T77400 CG89ET 73387745 IC50 = 923 nM T77400 C74TSX 73425972 IC50 = 3010 nM T77400 CWX3M6 73425973 IC50 = 4890 nM T77400 CEH2R6 73425974 IC50 = 1310 nM T77400 C9JE6M 75815419 IC50 = 47.6 nM T77400 CV35TH 89880131 IC50 = 80 nM T77400 C4EWJ2 89880132 IC50 = 500 nM T77400 CB9WX4 89880134 IC50 = 19 nM T77400 CKJ6N7 90005993 IC50 = 8.9 nM T77400 C9K4MZ 90006051 IC50 = 5.8 nM T77400 CF03DW 90168772 IC50 > 20000 nM T77400 CM6J9K 90168778 IC50 > 20000 nM T77400 CGJV10 90654177 IC50 = 4.9 nM T77400 C5H3ZQ 90654182 IC50 = 3.6 nM T77400 C1JPD6 91844700 IC50 = 5900 nM T77400 CYQV05 92471958 IC50 = 590 nM T77400 C2KVP3 117948953 IC50 = 2.8 nM T77400 CSCY01 117949009 IC50 = 66 nM T77400 CR87FK 117949032 IC50 = 62 nM T77400 C1XO7G 117949037 IC50 = 4100 nM T77400 C6WJN9 117949055 IC50 = 210 nM T77400 C9AW8C 117949072 IC50 = 24 nM T77400 C1COK8 117949123 IC50 = 250 nM T77400 COWG40 117949132 IC50 = 42 nM T77400 C0K7WT 117949138 IC50 = 8.7 nM T77400 CA74NJ 117949190 IC50 = 40 nM T77400 C74VEM 117949221 IC50 = 39000 nM T77400 C95TVN 117949229 IC50 = 33 nM T77400 C5H2ZV 117949248 IC50 = 910 nM T77400 CXEW03 117949270 IC50 = 72 nM T77400 CI3YX1 117949294 IC50 = 7.2 nM T77400 CHXA98 117949376 IC50 = 65 nM T77400 CZMJ97 117949378 IC50 = 29 nM T77400 CT3V0U 117949430 IC50 = 610 nM T77400 C8TE0J 117949497 IC50 = 3.5 nM T77400 C8LRE7 117949499 IC50 = 8100 nM T77400 CNE15J 117949533 IC50 = 77 nM T77400 C7FS2Y 118470919 IC50 = 10 nM T77400 CX0UN8 118470985 IC50 = 1 nM T77400 C4S5ZK 118471014 IC50 = 52 nM T77400 CB10HL 118471019 IC50 = 2 nM T77400 CNU8X4 118471029 IC50 = 2 nM T77400 C9F4PB 118471136 IC50 = 1 nM T77400 CQN46O 118471355 IC50 = 3 nM T77400 CS2QF5 118471479 IC50 = 47 nM T77400 C70LGE 118471483 IC50 = 0.8 nM T77400 CDA5Y3 118471525 IC50 = 80 nM T77400 CX0TQ7 118471706 IC50 = 3 nM T77400 CAM28L 118471717 IC50 = 14 nM T77400 CLU3C7 118471813 IC50 = 679 nM T77400 C8BN2I 118472547 IC50 = 7 nM T77400 CYQ74R 118479645 IC50 = 8 nM T77400 C04JTM 118479706 IC50 = 62 nM T77400 CL65RB 118479752 IC50 = 23 nM T77400 CVYK24 118556943 IC50 > 50000 nM T77400 CRA46I 118713812 IC50 = 404 nM T77400 C6RHL2 118736439 IC50 = 10 nM T77400 CZ1AM2 118736440 IC50 = 310 nM T77400 CXP31F 118736441 IC50 = 150 nM T77400 C8L7TA 118736442 IC50 = 5750 nM T77400 CP9T3B 118736443 IC50 = 2450 nM T77400 CVX94D 118736444 IC50 = 54 nM T77400 CM1X8H 118736445 IC50 = 190 nM T77400 CBW84D 118737979 IC50 = 6 nM T77400 CLR07H 118737980 IC50 = 95 nM T77400 C4CJR8 118737981 IC50 = 21 nM T77400 CLV60Q 118737982 IC50 = 3 nM T77400 CRJE23 122185011 IC50 = 5895 nM T77400 CS6M9C 122193679 IC50 > 100000 nM T77400 CY5S7B 126615633 IC50 = 52 nM T77400 CU52TA 126615644 IC50 = 987 nM T77400 CVX7U9 127029185 IC50 > 50000 nM T77400 C4UR7D 127038167 IC50 > 1000 nM T77400 C4H2TJ 127038168 IC50 = 395 nM T77400 CL9JT8 127038169 IC50 = 23.9 nM T77400 CN9BH4 127038170 IC50 = 2.06 nM T77400 CO2CI9 127038507 IC50 > 1000 nM T77400 CRF5C6 127038508 IC50 = 481 nM T77400 CJPX60 127038509 IC50 = 10.9 nM T77400 C7X2VQ 127038510 IC50 > 1000 nM T77400 C26EAG 127038511 IC50 = 65.7 nM T77400 CTM9E4 127038512 IC50 = 29.2 nM T77400 C6AQ2U 127038513 IC50 = 162 nM T77400 C6HZ8P 127038725 IC50 > 1000 nM T77400 CV1FM0 127038868 IC50 = 78.6 nM T77400 CADU23 127038869 IC50 = 3.49 nM T77400 C50MRW 127040517 IC50 = 46.8 nM T77400 CAG7Y1 127040518 IC50 > 1000 nM T77400 CLY63Q 127040519 IC50 = 98.6 nM T77400 C95LEY 127041240 IC50 > 100000 nM T77400 CW38DL 127042532 IC50 > 100000 nM T77400 CN5E6F 129010130 IC50 = 66.6 nM T77400 CRP5D9 131801460 Ki = 14.3 nM T77400 C16OKU 131801461 Ki = 237 nM T77400 CACJ46 132489333 IC50 = 362 nM T77400 C2P1IU 134129996 IC50 > 100000 nM T77400 CLE03O 134130328 IC50 > 100000 nM T77400 CSN6J0 134130563 IC50 > 100000 nM T77400 C0A1CZ 134131162 IC50 > 100000 nM T77400 CKYQ83 134587660 Ki = 642 nM T77400 CF24SY 134587670 Ki = 2340 nM T77400 CD9O8V 134587672 Ki = 4.3 nM T77400 CB8HO3 134587679 Ki = 19.6 nM T77400 CYDI92 134587729 Ki = 5.49 nM T77400 C4D5TR 134823954 IC50 = 7 nM T77400 C9IJK1 135566935 IC50 = 13000 nM T77400 C9Y7NH 136017768 IC50 = 1.59 nM T77400 C8UF7G 136087052 IC50 > 50000 nM T77400 C21FVA 136180322 IC50 = 560 nM T77400 CQW7T0 136197286 IC50 > 10000 nM T77400 C8TQ7A 136217455 IC50 > 50000 nM T77400 CMN10D 136239299 IC50 = 4.7 nM T77400 C1JUS2 137243509 IC50 > 100000 nM T77400 CPS12F 137286847 Ki = 195 nM T77400 C0KM1X 137288419 IC50 = 0.3 nM T77400 CC6TN9 137288423 IC50 = 0.6 nM T77400 CY3JA9 137348670 IC50 = 389.6 nM T77400 C50ZJS 137348671 IC50 = 7.1 nM T77400 C2N9VT 137348687 IC50 = 24 nM T77400 C64CQX 137631473 IC50 = 6100 nM T77400 C81LDE 137631646 IC50 = 3.1 nM T77400 C4OH1C 137631679 IC50 = 1200 nM T77400 C5ROI3 137631895 IC50 = 19.7 nM T77400 C2T4NC 137632277 IC50 = 16000 nM T77400 CC9T7R 137632951 IC50 = 19000 nM T77400 CU1R4L 137633190 IC50 > 100000 nM T77400 C8EV7L 137633354 IC50 = 1407 nM T77400 C6MB2D 137633899 IC50 = 21000 nM T77400 C9GJU6 137634998 IC50 = 206 nM T77400 CR31YE 137635321 IC50 = 85 nM T77400 CV6O7W 137635846 IC50 = 1.12 nM T77400 C4V0NA 137636043 IC50 = 15.6 nM T77400 CC9FP8 137636612 IC50 = 566.1 nM T77400 CME0R4 137636707 IC50 = 1000 nM T77400 C5NI2X 137636797 IC50 = 2107.4 nM T77400 C9XEK5 137637921 IC50 = 1520 nM T77400 CN7V2B 137638577 IC50 = 240.8 nM T77400 C2WA0G 137639069 IC50 = 27.7 nM T77400 CYXT20 137639195 IC50 = 792 nM T77400 CT3S0X 137640086 IC50 = 0.06 nM T77400 CKZ1V3 137640292 IC50 = 188.7 nM T77400 C13LPR 137640386 IC50 = 9.35 nM T77400 CAZJ94 137640735 IC50 = 0.92 nM T77400 CHJT03 137641277 IC50 = 146.4 nM T77400 CQ9TY5 137641733 IC50 = 70.1 nM T77400 C5E6TK 137642260 IC50 > 100000 nM T77400 C2F3KD 137642905 IC50 = 7000 nM T77400 C6VLU7 137642977 IC50 = 53 nM T77400 C9U8MJ 137643050 IC50 = 6500 nM T77400 CQP09A 137643189 IC50 = 480 nM T77400 C6ZIA0 137644259 IC50 = 5.94 nM T77400 CT95ED 137644401 IC50 = 7.8 nM T77400 CEW71T 137644414 IC50 = 2.4 nM T77400 C1L2AE 137644548 IC50 > 2000 nM T77400 CWUB18 137644904 IC50 = 5323.8 nM T77400 CY4K9V 137644985 IC50 = 297.8 nM T77400 CZ39VR 137645038 IC50 = 12 nM T77400 C4HC3F 137645688 IC50 = 1.3 nM T77400 CN7A5B 137645846 IC50 = 6.42 nM T77400 CF8PN0 137646373 IC50 = 1400 nM T77400 CH5T1N 137646636 IC50 = 24.4 nM T77400 C62WDH 137646854 IC50 > 100000 nM T77400 C27HUA 137647134 IC50 = 11 nM T77400 C9ILV2 137647474 IC50 = 49000 nM T77400 CIX4F6 137647559 IC50 = 5360 nM T77400 CYWR89 137647939 IC50 = 168 nM T77400 CHC24E 137648176 IC50 = 9.7 nM T77400 CYJ5Z4 137648284 IC50 = 3.54 nM T77400 CEI81F 137649219 IC50 = 10.9 nM T77400 C7YH2X 137649656 IC50 = 473 nM T77400 CU59SP 137649740 IC50 = 0.2 nM T77400 C4ZWI2 137649791 IC50 = 23000 nM T77400 C8YRB1 137649941 IC50 = 13.4 nM T77400 CQ21ZN 137650043 IC50 = 11.2 nM T77400 CR6M5K 137650215 IC50 = 9.26 nM T77400 CE4B5S 137651190 IC50 = 1012.7 nM T77400 CDYE95 137651309 IC50 > 100000 nM T77400 C18KXR 137651569 IC50 = 21 nM T77400 C6S2TD 137651868 IC50 = 3800 nM T77400 CIZX42 137651889 IC50 = 0.16 nM T77400 C6KX8Y 137651922 IC50 = 94.6 nM T77400 C05FML 137652023 IC50 > 100000 nM T77400 CDX5B4 137652246 IC50 = 140 nM T77400 CQ96UD 137652804 IC50 = 17.3 nM T77400 CI8OV2 137652839 IC50 = 2200 nM T77400 CIH38D 137652868 IC50 > 2000 nM T77400 CU8I3W 137653151 IC50 > 100000 nM T77400 CHLZ86 137653186 IC50 = 1.02 nM T77400 CS32XC 137653345 IC50 > 100000 nM T77400 CC5AK4 137654176 IC50 = 70000 nM T77400 CZV0W6 137654301 IC50 = 186 nM T77400 CSY3H9 137654828 IC50 = 3.59 nM T77400 CJT90A 137655626 IC50 = 423 nM T77400 CFW48A 137655833 IC50 = 0.23 nM T77400 C3EYO9 137656154 IC50 = 18.6 nM T77400 CM90RE 137656421 IC50 = 210 nM T77400 C0U1AS 137657330 IC50 = 69.2 nM T77400 CSX23V 137657865 IC50 = 28.6 nM T77400 CWC84D 137658255 IC50 = 52000 nM T77400 CM4CT5 137658915 IC50 = 199 nM T77400 CDE80H 137659658 IC50 = 3.19 nM T77400 C7FTC0 137660031 IC50 = 108.5 nM T77400 CY0V1N 137660078 IC50 = 7.8 nM T77400 C0GE7X 137660089 IC50 = 28000 nM T77400 CWAI46 137660568 IC50 = 3600 nM T77400 CTR5L7 137660971 IC50 = 28 nM T77400 C15IFJ 137662070 IC50 = 115 nM T77400 CJZD19 137662081 IC50 = 72 nM T77400 C6KYD7 137700754 IC50 > 10000 nM T77400 CM3UF7 137700779 IC50 > 20000 nM T77400 CPTE92 138319693 IC50 = 106 nM T77400 C2QLX3 138393292 IC50 > 50000 nM T77400 CSOF52 141737655 IC50 > 20000 nM T77400 C7SRA2 141737657 IC50 > 20000 nM T77400 CMIY07 141737666 IC50 > 20000 nM T77400 CC61SD 141737667 IC50 > 20000 nM T77400 C14CZJ 141737668 IC50 > 20000 nM T77400 CTNG49 141737674 IC50 > 20000 nM T77400 CJ38IC 141737676 IC50 > 20000 nM T77400 C1MC5Z 141737681 IC50 > 20000 nM T77400 CTUL23 141737690 IC50 > 20000 nM T77400 CMW20N 141737696 IC50 > 20000 nM T77400 CO1C4S 141737703 IC50 > 20000 nM T77400 CX9N1P 141737704 IC50 > 20000 nM T77400 C8HEG7 141737705 IC50 > 20000 nM T77400 CZTB36 145951354 IC50 = 6.9 nM T77400 C2AC1L 145963756 IC50 = 740 nM T77400 C2DKE6 145963778 IC50 > 10000 nM T77400 C8A3ES 145963852 IC50 > 10000 nM T77400 C6F8RD 145964089 Ki = 152 nM T77400 CN7EX8 145964626 Ki = 7810 nM T77400 CY69NH 145966741 IC50 = 620 nM T77400 C5RXC3 145967733 IC50 > 278000 nM T77400 CT89WH 145968235 IC50 = 670 nM T77400 CQ3RK6 145968854 IC50 = 233 nM T77400 CU2C0Y 145968972 IC50 = 18 nM T77400 C1U3IV 145969007 IC50 = 41 nM T77400 C7XA0G 145969034 IC50 = 66879 nM T77400 CH0ZK3 145969205 IC50 = 61 nM T77400 C8GDY6 145969532 IC50 = 1548 nM T77400 CH9I4O 145969561 IC50 = 2801 nM T77400 C2H9AP 145969697 IC50 = 422 nM T77400 CQ06JZ 145969912 IC50 = 6526 nM T77400 CP6QG9 145970031 IC50 = 5 nM T77400 CT3M9L 145971792 Ki = 11700 nM T77400 CHV59D 145971849 IC50 = 320 nM T77400 CH4D9S 145973243 IC50 = 1150 nM T77400 CCZ4U3 145974166 Ki = 97.2 nM T77400 CC7HN2 145974174 IC50 > 100000 nM T77400 C8P4GA 145974760 IC50 = 370 nM T77400 C6X3RQ 145975041 Ki = 15000 nM T77400 CWI73B 145976466 IC50 = 2.3 nM T77400 C9WR0G 145976954 Ki = 10100 nM T77400 C5N8AL 145977167 IC50 = 470 nM T77400 CUJZ04 145978143 IC50 > 10000 nM T77400 CK1BR0 145978345 IC50 > 100000 nM T77400 CVQ8I6 145978600 IC50 = 410 nM T77400 CKX3M5 145979083 IC50 = 1 nM T77400 C42ZAX 145979658 IC50 = 7.943 nM T77400 C93QTK 145979709 IC50 = 3.162 nM T77400 CA29ZL 145982452 IC50 = 3.981 nM T77400 CG7BR1 145987034 IC50 = 31 nM T77400 C5JXF1 145987164 IC50 = 1.995 nM T77400 CVMH95 145989382 IC50 = 3.162 nM T77400 CB5G0W 145990322 IC50 = 31.62 nM T77400 C0VQ7L 145990946 IC50 = 10 nM T77400 CZ6Y5L 145991256 IC50 = 5.012 nM T77400 CAM7X5 145991475 IC50 = 1.585 nM T77400 CHJ79V 145997874 IC50 > 10000 nM T77400 CM7TX2 148279038 IC50 > 100000 nM T77400 CM7N0S 155512334 IC50 = 1240 nM T77400 C9NVT8 155516688 IC50 = 3990 nM T77400 C5N0YD 155518781 IC50 = 11020 nM T77400 C7Z3CN 155520280 IC50 = 1940 nM T77400 CL8CU6 155521936 IC50 > 200000 nM T77400 CZPE14 155523280 IC50 = 5460 nM T77400 CWYF14 155523446 IC50 = 310 nM T77400 C1IJ5O 155526364 IC50 = 570 nM T77400 CC90XN 155526873 IC50 = 2630 nM T77400 CQ0AE6 155529518 IC50 = 40350 nM T77400 CT85RG 155530589 IC50 > 200000 nM T77400 CWKJ47 155532592 IC50 = 7270 nM T77400 CG0EC3 155536215 IC50 = 5940 nM T77400 CI4P1H 155537948 IC50 > 50000 nM T77400 C9J6VO 155540253 IC50 = 4280 nM T77400 CJ4GX7 155541617 IC50 = 3910 nM T77400 CMI8D9 155547380 IC50 = 4320 nM T77400 CSI4V9 155549683 IC50 = 5800 nM T77400 CX8DM0 155559762 IC50 = 16980 nM T77400 C9DMS4 155560624 IC50 > 50000 nM T77400 C2DA1W 155561694 IC50 = 72 nM T77400 C27FUB 155564688 IC50 = 3790 nM T77400 CQ2R0W 155568588 IC50 = 81 nM T77400 CWF2G3 71153391 IC50 = 1 nM T77400 D00YPO 14032753 IC50 = 46000 nM T77400 D05HFD 13936971 IC50 > 100000 nM T77400 D09GTN 13936969 IC50 > 100000 nM T77400 D09RKU 46239428 Ki > 10000 nM T77400 D0C2UJ 8974 IC50 > 10000 nM T77400 D0I6XA 149784 IC50 = 800 nM T77400 D0KD6S 44278378 IC50 = 17000 nM T77400 D0N6MR 10867033 IC50 = 80000 nM T77400 D0NI4Z 13936972 IC50 > 100000 nM T77400 D0R6MT 3758 IC50 = 4000 nM T77400 D0RC4F 72103 IC50 = 80000 nM T77400 D0T3UP 13724742 IC50 > 100000 nM T77400 D0V4WB 149790 IC50 = 635 nM T77400 D0V9MI 135564787 IC50 = 0.03 nM T77400 D0W3RR 10359339 IC50 = 6000 nM T07400 C9YJR2 9810788 IC50 < 500 nM T07400 CCO4K2 10188384 IC50 = 1750 nM T07400 C9WH7Y 24752728 Ki = 25 nM T07400 CL4VY2 71452357 IC50 = 1140 nM T07400 CLRZ53 71452359 IC50 = 5590 nM T07400 CE6QZ1 71452360 IC50 = 1240 nM T07400 CG1NU6 71452361 IC50 = 910 nM T07400 C6AYO7 71453726 IC50 = 16500 nM T07400 CFZ02E 71454135 IC50 = 1580 nM T07400 COE1Q3 71454136 IC50 = 1120 nM T07400 CCR73G 71455466 IC50 = 4600 nM T07400 C2D6WB 71455869 IC50 = 1210 nM T07400 C8M3TK 71455870 IC50 = 1910 nM T07400 CS8R7U 71455871 IC50 = 1720 nM T07400 CBP13J 71457675 IC50 = 1040 nM T07400 C27DBE 71457676 IC50 = 3180 nM T07400 CV9AI4 71459573 IC50 = 660 nM T07400 CI9U3N 71461319 IC50 = 1840 nM T07400 C4OH7I 71463041 IC50 = 2010 nM T07400 C6LQ4O 86304220 IC50 = 5400 nM T07400 CW1CK4 86304221 IC50 = 2500 nM T07400 CFMH38 86765239 IC50 = 1900 nM T07400 CVC9E4 86765240 IC50 = 1900 nM T07400 CGYJ35 90654926 IC50 = 18900 nM T07400 C31PFC 90654927 IC50 = 7800 nM T07400 CE0SJ3 90654928 IC50 = 5300 nM T07400 CUAO54 90664979 IC50 = 550 nM T07400 C4PN7Z 137635310 IC50 < 500 nM T40016 D04DJN 10635 IC50 = 540 nM T40016 D07BSQ 5994 Ki = 30.5 nM T40016 D0D1SG 5755 Ki = 1.14 nM T40016 D0D4HN 10607 IC50 = 14 nM T40016 D0EP0C 5833 Ki = 32.6 nM T40016 D0G3SH 31401 EC50 = 298700 nM T40016 D0G8BV 6450278 Ki = 252 nM T40016 D0IT2G 5743 EC50 = 0.1 nM T40016 D0Q4SD 443872 Ki = 3162.28 nM T40016 D0V9BD 2375 Ki > 100000 nM T40016 D0Y7IU 5281004 Ki = 1.3 nM T40016 D0Y7JU 9854489 IC50 = 0.03981 nM T40016 D0Z4EI 55245 IC50 = 0.008 nM T40016 D00JFE 56941241 IC50 = 990 nM T40016 D01SYU 10026128 IC50 = 10000 nM T40016 D03WNG 73051463 Ki = 7.2 nM T40016 D07MON 5311505 IC50 = 27 nM T40016 D07UIS 118092367 Ki = 12 nM T40016 D0HE7C 134415769 IC50 = 5.6 nM T40016 D0LI1C 44469321 IC50 > 30000 nM T40016 D0SZ1G 121248172 IC50 = 3.8 nM T40016 D0W8OJ 9854142 IC50 = 1.2 nM T40016 D0X1OW 86287635 IC50 = 9200 nM T40016 D0X9YP 67041274 IC50 = 0.056 nM T40016 D0TH6M 25204767 EC50 > 10000 nM T40016 D00PDG 44454750 Ki = 0.9 nM T40016 D02KAU 46871935 IC50 > 10000 nM T40016 D03KTE 16750192 Ki = 8300 nM T40016 D07EBU 135565424 IC50 > 10000 nM T40016 D09UFV 24825740 IC50 = 0.049 nM T40016 D0W5RL 9577221 IC50 = 120 nM T40016 C59UQE 6279 EC50 = 10 nM T40016 CD4XK3 156517 IC50 = 27000 nM T40016 CRL43B 192254 EC50 = 105300 nM T40016 CW90BT 441336 Ki = 0.7 nM T40016 C40YBS 444036 IC50 = 0.04 nM T40016 C2B0JA 674359 Ki = 1.3 nM T40016 C93EKR 674360 Ki = 26.2 nM T40016 CS6J4Z 1043068 IC50 > 100000 nM T40016 CJ02TD 3309795 IC50 > 10000 nM T40016 CKF71B 3463734 IC50 = 5700 nM T40016 CLBV35 3699263 IC50 = 480 nM T40016 C7X9AN 3728357 IC50 = 6900 nM T40016 CES83X 3775934 IC50 = 1600 nM T40016 C2EIT3 3789969 IC50 = 1300 nM T40016 C43BVE 3816305 IC50 = 735 nM T40016 CBIA94 3829166 IC50 > 10000 nM T40016 CMG30I 3832779 IC50 = 2600 nM T40016 CGH2L3 3854781 IC50 = 1800 nM T40016 CF2H8R 3865491 IC50 = 4600 nM T40016 CMK3N0 4110968 IC50 > 2000 nM T40016 C6JCL9 4163889 Ki = 33 nM T40016 C8V3MU 4193542 Ki = 24 nM T40016 CBFW65 4254945 Ki = 2.9 nM T40016 C9JP7D 4290639 Ki = 4500 nM T40016 CW23GV 4390931 Ki = 16 nM T40016 C5NDK3 4583408 IC50 > 10000 nM T40016 C0FRN6 4686093 IC50 = 4100 nM T40016 C9D6JM 4983635 IC50 > 10000 nM T40016 CBW8O6 5006871 IC50 = 2100 nM T40016 C7VQS6 5146911 IC50 > 10000 nM T40016 CDCK27 5185174 IC50 = 750 nM T40016 C16ZSG 6439929 Ki = 224 nM T40016 CG1U6P 7275458 IC50 = 55 nM T40016 CYI7T4 9802231 IC50 = 2.8 nM T40016 C7REX1 9805004 EC50 = 12.59 nM T40016 C82TUJ 9808265 IC50 = 19 nM T40016 CV87EA 9820084 IC50 = 40 nM T40016 C8A3WG 9820510 Ki > 10000 nM T40016 C06RXB 9821393 Ki = 2.1 nM T40016 C7HGB0 9822150 Ki = 236 nM T40016 CD9S5P 9825465 EC50 = 4 nM T40016 CT6OZ1 9825650 IC50 = 5.1 nM T40016 CW8LT0 9826255 IC50 = 18 nM T40016 CBS8M2 9839134 IC50 = 1756 nM T40016 C92CPK 9841404 Ki = 9200 nM T40016 CK7UC3 9841413 Ki > 10000 nM T40016 C7P6XH 9842832 Ki = 6500 nM T40016 CE9A6G 9845022 Ki = 210 nM T40016 C7RS9U 9846657 Ki = 3.3 nM T40016 CERF28 9861044 Ki = 8100 nM T40016 C3K4EU 9862027 Ki > 10000 nM T40016 CJN78I 9862597 IC50 = 35 nM T40016 C7XY1N 9863751 IC50 = 38 nM T40016 C01ZFV 9882789 IC50 = 35 nM T40016 CEM27C 9885473 Ki = 299 nM T40016 C8XSO2 9887578 Ki = 133 nM T40016 C6B9CZ 9888873 EC50 = 205 nM T40016 CZ5R9B 9890023 Ki = 11 nM T40016 CI4UK6 9890642 Ki = 2 nM T40016 CCM30W 9901180 Ki = 208 nM T40016 CJ7U3R 9904286 IC50 > 10000 nM T40016 C4KY8S 9904429 IC50 = 1316 nM T40016 C6SWK1 9904610 IC50 = 2581 nM T40016 CTI1J8 9905296 Ki = 8800 nM T40016 CE1TK2 9908041 Ki = 180 nM T40016 CG0B9U 9911589 IC50 = 3 nM T40016 CR4H6B 9919949 EC50 = 910 nM T40016 CMJG42 9921530 IC50 > 10000 nM T40016 C49UGC 9925244 Ki = 3.7 nM T40016 CUK3E9 9933829 IC50 = 26 nM T40016 C39EXP 9933936 IC50 = 430 nM T40016 CWX17A 9933946 IC50 = 707.95 nM T40016 C24FUO 9943699 IC50 = 1856 nM T40016 CXM67A 9946466 Ki = 106 nM T40016 C63MQU 9947042 Ki = 65 nM T40016 CCSX75 9949772 Ki = 1766 nM T40016 C6ZT3M 9950357 IC50 = 360 nM T40016 CKU64T 9952569 IC50 = 1 nM T40016 CW0ED9 9953456 IC50 = 146 nM T40016 CEM8L7 9969737 Ki = 2.1 nM T40016 C0Y1RE 9969849 Ki = 12.1 nM T40016 C95CAN 9978625 Ki = 0.146 nM T40016 CP2E8A 9979395 Ki = 2465 nM T40016 CP7F1R 9980041 IC50 = 7.6 nM T40016 C1QP8T 9993897 IC50 = 2500 nM T40016 COA3P9 9997031 IC50 > 2000 nM T40016 C47RUV 9998207 IC50 > 2000 nM T40016 C4V6RF 9998996 IC50 = 1.1 nM T40016 CU1ON0 9999068 Ki = 0.58 nM T40016 CL8V1C 9999671 IC50 = 565 nM T40016 CU4L7C 9999672 IC50 > 2000 nM T40016 C08OBS 10001663 IC50 > 2000 nM T40016 C0XDE9 10001914 IC50 = 194 nM T40016 CA5C6V 10002879 IC50 = 64 nM T40016 CW6P3G 10002931 IC50 = 6.3 nM T40016 C7FC9H 10004421 IC50 = 3.162 nM T40016 C3IE9K 10021634 IC50 = 355 nM T40016 CJ0O2X 10021826 IC50 > 2000 nM T40016 C52ADB 10023861 Ki = 4728 nM T40016 CN8BH3 10024007 IC50 = 5.8 nM T40016 CC4WY6 10024990 IC50 = 990 nM T40016 CSM0W3 10026120 IC50 = 690 nM T40016 C9RU8E 10027430 IC50 = 15.85 nM T40016 C9DH4U 10044332 IC50 = 0.6 nM T40016 C3ITG8 10044396 IC50 > 2000 nM T40016 C7WR0E 10044812 IC50 > 2000 nM T40016 CY6EH9 10046547 IC50 > 2000 nM T40016 C9I4JM 10046548 IC50 > 2000 nM T40016 CTL09O 10046928 EC50 = 2.7 nM T40016 CK50XF 10048063 IC50 > 2000 nM T40016 C3AXU8 10048339 EC50 = 10 nM T40016 C5E9SY 10064248 IC50 = 1.5 nM T40016 CC9Q5R 10067481 IC50 = 72.5 nM T40016 C0MG6I 10067556 IC50 > 2000 nM T40016 C2V9BW 10068183 IC50 = 710 nM T40016 CB5OZ0 10070722 IC50 = 400 nM T40016 CFY67M 10070808 Ki = 44 nM T40016 C7JQM6 10070842 IC50 = 800 nM T40016 CS9CO3 10071426 IC50 = 570 nM T40016 C9T4HR 10071810 IC50 = 77 nM T40016 C5MR6U 10071910 IC50 > 2000 nM T40016 CLO7H6 10072320 IC50 = 275 nM T40016 CUSC84 10090072 IC50 = 820 nM T40016 CQ3LD1 10091351 IC50 = 240 nM T40016 C2C7NE 10091387 IC50 > 2000 nM T40016 CRP4A3 10091735 IC50 > 2000 nM T40016 CT2Y1J 10092463 IC50 = 19 nM T40016 C16HAK 10094808 IC50 = 67 nM T40016 CC59OU 10110007 IC50 = 21 nM T40016 C3G2XJ 10110771 IC50 = 43 nM T40016 C5HM2D 10111302 IC50 = 62 nM T40016 CWR57A 10113229 Ki = 4.1 nM T40016 C62CGR 10125859 Ki = 14 nM T40016 CM4DK2 10125966 Ki = 2.7 nM T40016 CDBJ41 10126018 Ki = 9 nM T40016 CO97CW 10126196 Ki = 9.5 nM T40016 CR0DX5 10126475 IC50 = 855 nM T40016 CHS18G 10126476 IC50 = 945 nM T40016 CR0BP6 10126871 IC50 = 6.6 nM T40016 CV5PQ0 10126940 IC50 = 22 nM T40016 CVF40M 10127159 IC50 = 30 nM T40016 C3CRZ1 10127269 IC50 = 64 nM T40016 CPB60D 10127340 IC50 = 60 nM T40016 C1K8UF 10127593 IC50 = 7 nM T40016 C8VBQ0 10127709 IC50 = 9 nM T40016 CKMW98 10128037 EC50 = 45 nM T40016 C7CNX6 10128352 IC50 = 740 nM T40016 C8QRY9 10131608 IC50 = 382 nM T40016 CX6BP9 10134499 IC50 = 460 nM T40016 CWKL91 10136854 IC50 = 9 nM T40016 CS8I2Z 10138737 IC50 = 18 nM T40016 C1GI3D 10150743 IC50 = 55 nM T40016 CZKF71 10150825 IC50 = 10 nM T40016 CYR0U5 10150851 IC50 = 550 nM T40016 CVO1F7 10151165 IC50 = 24 nM T40016 C6EC1P 10151186 IC50 = 104 nM T40016 CQ14RM 10151357 IC50 = 45 nM T40016 C6U0FQ 10151473 IC50 = 61 nM T40016 CW4Y2K 10151995 IC50 = 120 nM T40016 CDV0H3 10152035 IC50 = 110 nM T40016 CR6N7C 10156793 Ki = 2.2 nM T40016 CP1M6Q 10157287 Ki = 487 nM T40016 C0MX7K 10157532 IC50 = 81 nM T40016 CKY6J8 10158491 IC50 = 41 nM T40016 CXO53S 10160645 IC50 = 28 nM T40016 C7DC1F 10162430 IC50 = 63 nM T40016 C4N8AV 10163106 IC50 = 13 nM T40016 C83WDN 10167930 IC50 = 2.1 nM T40016 CL0U4N 10172897 IC50 = 81 nM T40016 C56RYS 10173217 IC50 = 460 nM T40016 CG0VH8 10173354 IC50 = 66 nM T40016 CU6D8W 10173525 EC50 = 140 nM T40016 CP4Y6T 10173634 IC50 = 57 nM T40016 C14HMT 10173659 IC50 = 120 nM T40016 CE29WD 10174141 IC50 = 52 nM T40016 C5QDA4 10177869 IC50 = 180 nM T40016 C2P4IY 10177943 IC50 = 1430 nM T40016 CKGZ56 10178295 IC50 = 630 nM T40016 C8L7HJ 10179031 IC50 = 3 nM T40016 CNRZ84 10180123 IC50 = 10 nM T40016 CZ2L3V 10189211 IC50 = 19 nM T40016 CHK2V6 10193599 Ki = 5 nM T40016 C5SRU4 10193967 Ki = 62 nM T40016 C41YRZ 10194268 IC50 = 1125 nM T40016 CX4F7Z 10194607 IC50 = 275 nM T40016 CV0LE4 10194889 IC50 = 25.12 nM T40016 CJ1GX6 10195783 IC50 = 470 nM T40016 CRIH90 10210815 IC50 = 4.8 nM T40016 C8HDU9 10215137 EC50 = 15 nM T40016 C3O7WH 10215978 IC50 = 370 nM T40016 CX6FD1 10216117 Ki = 8.1 nM T40016 C1SG4N 10216152 IC50 = 1250 nM T40016 CD0YT7 10216465 IC50 = 46 nM T40016 C1FGX9 10216535 IC50 = 6 nM T40016 CW7QX2 10216536 IC50 = 38 nM T40016 CG9OH4 10216697 IC50 = 58 nM T40016 CXN4W1 10216788 IC50 = 580 nM T40016 CUGN98 10217411 IC50 = 77 nM T40016 C3XK0O 10217420 IC50 = 48 nM T40016 C54HJB 10221941 Ki = 9.9 nM T40016 CJ9BE0 10222329 IC50 = 7 nM T40016 CVAJ29 10223284 IC50 = 23 nM T40016 C84SRT 10223610 IC50 = 3 nM T40016 CEX46C 10224296 IC50 = 110 nM T40016 C0K1EX 10233467 IC50 = 2.2 nM T40016 CUYO17 10237223 IC50 = 610 nM T40016 C4KF2V 10237539 Ki = 511 nM T40016 CWYK62 10238100 IC50 = 15 nM T40016 C1R8GY 10238297 IC50 = 76 nM T40016 CNB1V3 10238624 EC50 = 420 nM T40016 CPGF94 10238831 IC50 = 191 nM T40016 C2AZH1 10238961 EC50 = 760 nM T40016 C56PQZ 10247253 IC50 = 116 nM T40016 CSA4R3 10252455 IC50 = 220 nM T40016 C7EGH2 10252527 IC50 = 10 nM T40016 C3C1OQ 10255490 IC50 = 3.09 nM T40016 C2N0XF 10269831 IC50 = 160 nM T40016 CR59SC 10271193 IC50 = 19 nM T40016 CPIS57 10271557 IC50 = 66 nM T40016 C4AS5M 10272127 IC50 = 216 nM T40016 CC4WT8 10272405 Ki = 13.9 nM T40016 C9UL4O 10272529 Ki = 12 nM T40016 C0D1BI 10274504 IC50 = 656 nM T40016 CKTL36 10275888 IC50 = 61 nM T40016 CQ6UW3 10283096 IC50 = 670 nM T40016 CZP75A 10286964 Ki = 8.1 nM T40016 CUQC81 10287415 IC50 > 1000 nM T40016 C5RC7X 10287444 IC50 = 30 nM T40016 CJT2G8 10287863 IC50 = 120 nM T40016 C1M6WY 10288006 IC50 = 17 nM T40016 CO6UP3 10288155 IC50 = 68 nM T40016 CNT3V9 10288528 IC50 > 2000 nM T40016 C6C2IK 10288565 IC50 = 81 nM T40016 C1I9JX 10288784 IC50 = 52 nM T40016 CNEO49 10289020 EC50 = 130 nM T40016 CMED59 10291237 IC50 = 117 nM T40016 CD03TA 10294824 IC50 = 289 nM T40016 C6TP2B 10295095 IC50 = 6 nM T40016 CZF4S5 10295116 IC50 = 9.2 nM T40016 C6JF1S 10296963 IC50 = 548 nM T40016 CUK42D 10297219 IC50 = 137 nM T40016 CLJU03 10298892 Ki = 2.4 nM T40016 C9UYG8 10309447 IC50 = 580 nM T40016 C8FM2D 10309755 IC50 = 340 nM T40016 C1OV7M 10309756 IC50 = 101 nM T40016 C9TI4A 10310063 IC50 = 56 nM T40016 CP9AE0 10310476 IC50 = 205 nM T40016 CV52EN 10310809 EC50 = 130 nM T40016 CR1L5N 10311251 EC50 = 120 nM T40016 C9FCQ5 10313926 IC50 = 194 nM T40016 C7RLW3 10314903 IC50 > 2000 nM T40016 CX7WS4 10316069 Ki = 154 nM T40016 CR9ON2 10316670 IC50 = 210 nM T40016 CP7CF8 10317646 EC50 = 21 nM T40016 CZFY94 10318044 IC50 = 804 nM T40016 CJB8R4 10319017 Ki = 331 nM T40016 CC4NU9 10319739 EC50 = 11.4 nM T40016 C7TQY8 10321412 IC50 > 2000 nM T40016 C0EJH9 10323216 IC50 = 4.677 nM T40016 C9L1FM 10325323 IC50 = 6.6 nM T40016 C6OI7M 10336208 IC50 > 2000 nM T40016 CEB82Z 10337245 Ki = 1777 nM T40016 C4QY5H 10337273 IC50 > 2000 nM T40016 C3PHW5 10339694 IC50 = 548 nM T40016 C8IAJ7 10339824 IC50 > 2000 nM T40016 CK20PF 10339825 IC50 > 2000 nM T40016 CQP1Y7 10340204 Ki = 152 nM T40016 C28SWP 10341012 IC50 > 2000 nM T40016 CQ01DG 10342379 IC50 = 980 nM T40016 CEW79S 10361500 IC50 > 2000 nM T40016 C3YU5D 10361560 IC50 = 12 nM T40016 CA20SQ 10362131 IC50 > 2000 nM T40016 CF2W3R 10362274 EC50 = 2.7 nM T40016 C2PSC1 10362449 IC50 > 2000 nM T40016 CMSA84 10362453 IC50 = 703 nM T40016 CEJ78I 10365592 IC50 = 45 nM T40016 C6QR5M 10366372 IC50 = 290 nM T40016 CDBZ06 10372181 IC50 = 86 nM T40016 C14AIB 10384345 IC50 = 34 nM T40016 C8KO5Z 10384804 IC50 = 65 nM T40016 C6RQK1 10386584 IC50 = 3.3 nM T40016 C59VXD 10386752 Ki = 0.8 nM T40016 C2MIC7 10388043 IC50 = 195 nM T40016 CBU68V 10406413 Ki = 0.95 nM T40016 C5SB4L 10407417 EC50 = 2.1 nM T40016 CEQW13 10407564 IC50 > 2000 nM T40016 CS5XF8 10408522 IC50 > 2000 nM T40016 CYZ5B6 10410448 EC50 = 5 nM T40016 C8ERB7 10411364 IC50 = 185 nM T40016 C4R6IF 10414489 IC50 = 25.12 nM T40016 CZ5CJ3 10423330 Ki = 5424 nM T40016 C3LF9D 10428026 IC50 > 2000 nM T40016 CFVP19 10428095 EC50 = 9.3 nM T40016 CJ6T4F 10428171 IC50 = 1015 nM T40016 CHR4W7 10429332 IC50 = 129 nM T40016 C03JBL 10429502 IC50 = 1.6 nM T40016 C37VXR 10432143 Ki = 3210 nM T40016 CAKV91 10434383 IC50 = 10 nM T40016 CFMI34 10440737 IC50 = 310 nM T40016 C1KE6C 10446402 IC50 = 2600 nM T40016 CI91JZ 10450619 IC50 = 1000 nM T40016 CK05HV 10450738 IC50 = 167 nM T40016 CT35HI 10452933 EC50 = 38 nM T40016 CS12VO 10453115 EC50 = 6 nM T40016 C0NT9D 10454007 IC50 = 5.3 nM T40016 CVQS04 10454813 IC50 = 6.7 nM T40016 CH49LB 10456872 EC50 = 24.2 nM T40016 C9LQ7R 10457600 IC50 = 5.012 nM T40016 C7R2OJ 10457897 IC50 = 5.012 nM T40016 C1H5RP 10458842 EC50 > 10 nM T40016 CYQ65Z 10472575 IC50 = 125 nM T40016 CK4NI1 10473865 IC50 = 280 nM T40016 COMX74 10474093 IC50 = 1.2 nM T40016 C85RBN 10474264 IC50 = 190 nM T40016 C1S9HE 10474749 IC50 = 395 nM T40016 CUL8O4 10475384 EC50 = 2.9 nM T40016 CN7KQ8 10475688 IC50 = 371 nM T40016 CGH31Z 10475742 EC50 = 1 nM T40016 C8O1QG 10476314 Ki = 913 nM T40016 CPX65M 10477088 IC50 = 64 nM T40016 CG3P0I 10478173 EC50 = 31.3 nM T40016 C5U3JY 10478638 IC50 = 5.1 nM T40016 CB3S1Q 10484201 IC50 = 2.1 nM T40016 CYE7C2 10496255 Ki = 3697 nM T40016 CT7IG5 10497270 Ki = 1657 nM T40016 CO35TR 10499308 Ki = 6386 nM T40016 C6FA1N 10501542 Ki = 2570 nM T40016 CA5OH2 10503046 Ki = 14 nM T40016 C5AP6C 10503520 Ki = 42 nM T40016 C5WP1Q 10517398 Ki = 8511 nM T40016 CR1OS9 10523126 Ki = 909 nM T40016 C5CDF0 10524606 Ki = 4109 nM T40016 CYS8J9 10546095 Ki > 10000 nM T40016 CB04AE 10593144 Ki = 2206 nM T40016 CBEC38 10596252 Ki = 60 nM T40016 C6G7JR 10596379 Ki = 193 nM T40016 CC8T7J 10598305 Ki = 59 nM T40016 CAD6L2 10618033 Ki = 1036 nM T40016 CMK8I6 10622122 Ki = 6.3 nM T40016 CO3V0S 10622594 Ki = 67 nM T40016 C57PFY 10643931 Ki = 864 nM T40016 C02ZMG 10643956 Ki = 58 nM T40016 CF08PC 10661117 Ki = 8215 nM T40016 CU9X3A 10665612 Ki = 1261 nM T40016 C69CNF 10667548 Ki = 680 nM T40016 CYNG45 10668755 Ki = 173 nM T40016 CS6YF0 10690456 Ki = 249 nM T40016 CYRQ10 10691647 Ki = 9.3 nM T40016 C6SP3O 10694256 Ki = 257 nM T40016 CVD2Y9 10717098 Ki = 100 nM T40016 CK2NM9 10717832 Ki = 250 nM T40016 CUG2Z9 10739308 Ki = 2199 nM T40016 CAT1X8 10741366 Ki = 34 nM T40016 C3H6CZ 10754393 Ki = 8356 nM T40016 CB3JD0 10763832 Ki = 39 nM T40016 C7HAB1 10782276 Ki = 4532 nM T40016 CNV27D 10783127 Ki = 2781 nM T40016 CNL1U7 10785305 Ki > 10000 nM T40016 C07BOR 10787258 Ki = 147 nM T40016 C10AMX 10805958 Ki = 2286 nM T40016 CBX48C 10807828 Ki = 2670 nM T40016 CN5WV4 10809583 Ki = 4417 nM T40016 C1CRQ5 10811045 Ki = 237 nM T40016 CL7JN6 10827013 Ki = 6812 nM T40016 CN1H5Z 10832792 Ki = 80 nM T40016 CA96PR 10860931 Ki = 7 nM T40016 C8KME1 10861665 Ki = 88 nM T40016 CHU9A4 10873317 IC50 = 77 nM T40016 CI5F0S 10881662 Ki = 33.8 nM T40016 CVG34R 10883247 Ki = 34 nM T40016 CK41RM 10892050 Ki > 10000 nM T40016 CNG7L9 10894018 Ki = 4.2 nM T40016 CP9FX4 10904951 Ki = 3200 nM T40016 C54IAT 10905085 Ki = 1800 nM T40016 C6EG2D 10906030 Ki = 5.32 nM T40016 CBD12K 10906044 IC50 = 320 nM T40016 C3BZD9 10916860 Ki = 6000 nM T40016 C1D8IK 10926892 Ki = 400 nM T40016 C2UG0A 10937849 Ki = 207 nM T40016 C2IJR9 10949091 Ki = 2100 nM T40016 CHU10G 10960295 Ki = 232 nM T40016 CT2BR8 10969959 Ki = 4.4 nM T40016 C0GX6P 10970905 Ki = 25 nM T40016 CV3QY8 10972344 Ki = 2.3 nM T40016 C07JFA 10993685 Ki = 386 nM T40016 CUC05J 11002535 Ki = 2.3 nM T40016 C8AY9Z 11003946 Ki = 51 nM T40016 C5U8ZE 11013870 Ki = 18 nM T40016 CMJ7F9 11013871 Ki = 2 nM T40016 C7E9XI 11015162 IC50 = 90 nM T40016 CRH3L8 11025398 IC50 = 250 nM T40016 CU02DM 11046701 Ki = 5.2 nM T40016 CF8UC7 11057125 Ki = 140 nM T40016 CUYB81 11057924 Ki = 6.6 nM T40016 CIH8K4 11066740 Ki = 5.96 nM T40016 CS7Q4F 11069511 Ki = 2.8 nM T40016 CI8GJ5 11079263 IC50 = 109 nM T40016 C09ZLY 11088436 Ki > 10000 nM T40016 C6T7CR 11089159 Ki = 9.3 nM T40016 C6HPL0 11089468 Ki = 1.9 nM T40016 C6LYG7 11090322 IC50 > 1000 nM T40016 CE2O8Y 11110616 Ki = 6.9 nM T40016 C69GXQ 11110815 Ki = 9 nM T40016 CDX2W3 11121575 Ki = 18 nM T40016 C1OJK3 11131414 Ki = 27.6 nM T40016 CBDG76 11132271 Ki > 5000 nM T40016 C6TJ8D 11132273 Ki = 3.8 nM T40016 CB03TK 11143041 EC50 = 99700 nM T40016 CXS6J7 11155441 Ki = 0.2 nM T40016 CJ7KZ9 11155655 Ki > 100000 nM T40016 CIX9T7 11177172 EC50 = 54.2 nM T40016 CP3D7X 11201812 IC50 = 10 nM T40016 CW0Z2J 11212626 IC50 = 4786.3 nM T40016 CL97OU 11212803 IC50 = 17 nM T40016 C4U0DF 11213029 EC50 = 0.2 nM T40016 CFH3Q8 11213179 Ki = 2.9 nM T40016 C81CJV 11214068 IC50 = 0.5 nM T40016 CLCM91 11224044 IC50 = 0.9 nM T40016 CF3AY1 11225369 IC50 = 3 nM T40016 CVR9L1 11226313 EC50 = 0.5 nM T40016 CRN4V2 11232136 IC50 > 3000 nM T40016 CW6P7A 11244720 EC50 = 3 nM T40016 C3DO9S 11248612 IC50 = 2.5 nM T40016 CYCR06 11256303 IC50 = 14 nM T40016 CXG0C2 11269006 IC50 = 1.5 nM T40016 C8XPZ4 11269445 IC50 = 57 nM T40016 C4HNB8 11269886 IC50 = 22 nM T40016 CSH2R3 11271731 EC50 = 4.5 nM T40016 CHXY45 11272042 EC50 = 0.4 nM T40016 CJLC62 11273833 IC50 = 330 nM T40016 CC0XI4 11279959 IC50 = 127 nM T40016 C4SC0W 11281576 EC50 = 2.2 nM T40016 C8YL6K 11282486 IC50 = 19 nM T40016 CUX0S2 11282904 Ki = 0.6 nM T40016 CIY9H5 11291999 IC50 = 6 nM T40016 C58MZD 11293264 IC50 = 0.4 nM T40016 C8UK5D 11302609 IC50 = 38 nM T40016 C24ILB 11302908 Ki = 2250 nM T40016 C0IQ9K 11304445 IC50 = 4 nM T40016 CLIB17 11304952 EC50 = 0.6 nM T40016 C0XUF2 11305564 IC50 = 1.9 nM T40016 C5C0MA 11316115 IC50 = 2.5 nM T40016 C0B2FT 11327284 IC50 = 5 nM T40016 CXC9G3 11327341 IC50 = 1400 nM T40016 C3OI8M 11330644 IC50 = 6.6 nM T40016 C1HZS7 11336351 IC50 = 73 nM T40016 CT9Y4O 11339440 IC50 > 3000 nM T40016 CGM2R9 11339795 IC50 = 562.34 nM T40016 CBPX74 11350176 IC50 = 26 nM T40016 CQ1NV4 11363810 Ki = 1.5 nM T40016 CUE7W0 11375176 EC50 = 1.5 nM T40016 C8FQ9B 11375180 IC50 = 2090 nM T40016 CP2DL0 11377050 IC50 = 500 nM T40016 C76VYN 11382721 IC50 = 230 nM T40016 CV4RO2 11384310 IC50 = 2 nM T40016 CXW40M 11384346 IC50 = 9 nM T40016 CU7IE0 11410199 IC50 = 5.4 nM T40016 CO20QH 11416730 IC50 = 120 nM T40016 C5KQY8 11417666 Ki = 225 nM T40016 C5WO0U 11429662 EC50 = 6.5 nM T40016 C8DXS2 11430241 EC50 = 0.7 nM T40016 CSGJ21 11430586 Ki = 1.9 nM T40016 C2D7HP 11442368 IC50 = 22 nM T40016 COQ7S4 11444087 Ki = 0.9 nM T40016 CV8XI7 11453933 EC50 = 0.6 nM T40016 C2BXU1 11454745 Ki = 4.3 nM T40016 C8Y5BF 11463839 EC50 = 19.5 nM T40016 CJEU23 11474124 IC50 = 77.3 nM T40016 CD2Q3F 11474917 IC50 = 3 nM T40016 CAT79U 11475733 EC50 = 1.9 nM T40016 CC75NQ 11477616 Ki = 0.6 nM T40016 CQ62KS 11485693 IC50 = 190 nM T40016 C9Q1NY 11494167 Ki = 1.3 nM T40016 CFLQ08 11495227 IC50 = 8.2 nM T40016 C03NYX 11495549 IC50 = 210 nM T40016 CJ1M8L 11495854 Ki = 17 nM T40016 CFB75K 11497883 Ki = 4.5 nM T40016 CK3RS0 11498018 Ki = 12 nM T40016 C0O7TM 11500993 Ki = 100 nM T40016 C3L4DF 11504875 EC50 = 75000 nM T40016 CR40IH 11516847 IC50 = 8 nM T40016 C4Q5XE 11517391 Ki = 6 nM T40016 CP4F8X 11517412 IC50 = 2.3 nM T40016 CB9D3A 11517558 IC50 = 11.22 nM T40016 CCL20N 11519406 Ki = 3 nM T40016 CS0M3B 11525591 Ki = 1.1 nM T40016 CE3I6O 11525793 IC50 = 12.59 nM T40016 C2PB6Z 11530605 Ki = 8 nM T40016 C1R6DC 11531942 IC50 = 37 nM T40016 C9SH1C 11532777 IC50 = 31.62 nM T40016 C0DS3E 11533163 Ki = 2.6 nM T40016 C7F0KV 11533276 IC50 = 19.95 nM T40016 CZ1HA3 11538472 IC50 = 16 nM T40016 CFC1Z4 11538799 IC50 = 26 nM T40016 C16YOG 11541310 Ki = 1.4 nM T40016 CNRP26 11545475 IC50 = 18 nM T40016 C8YBI3 11547009 Ki = 13 nM T40016 CP13VG 11547261 Ki = 41 nM T40016 CT45RM 11548068 IC50 = 1.202 nM T40016 CI90JB 11551816 IC50 = 10 nM T40016 C0J8UL 11551817 Ki = 4.4 nM T40016 C4FM3R 11553707 IC50 = 1.259 nM T40016 CBK60G 11559947 IC50 = 23 nM T40016 C1D9YS 11560003 IC50 = 15 nM T40016 C1XKY3 11561826 Ki = 18 nM T40016 C47ROU 11562491 Ki = 0.8 nM T40016 CB37YF 11566981 Ki = 1.8 nM T40016 C5UEY6 11567352 IC50 = 2.1 nM T40016 C8WJ2F 11567609 IC50 = 4.5 nM T40016 CXQ59S 11567630 IC50 = 99 nM T40016 C0PES1 11568433 IC50 = 1.95 nM T40016 CJ30TW 11568951 Ki = 2.5 nM T40016 C0QFC2 11569557 Ki = 12 nM T40016 CQ28XT 11569834 Ki = 0.6 nM T40016 C10AWO 11569892 IC50 = 794.33 nM T40016 C7AMJ5 11570728 Ki = 1.3 nM T40016 C1X7LS 11571692 EC50 = 50 nM T40016 CQ0U9D 11576238 IC50 = 25.12 nM T40016 CSQ32L 11577390 Ki = 1.4 nM T40016 CTA8J3 11583514 IC50 = 15.85 nM T40016 CQ43OD 11584668 Ki = 2.8 nM T40016 CEF7K8 11585049 EC50 = 173000 nM T40016 C0SCT6 11588584 IC50 = 31 nM T40016 C3MW1D 11589982 IC50 = 7.1 nM T40016 C03QYZ 11590471 IC50 = 15 nM T40016 CLN0C5 11591199 IC50 = 9.55 nM T40016 CZ4M8O 11591459 IC50 = 3.467 nM T40016 CEH7D2 11591552 Ki = 0.6 nM T40016 CV94WU 11591790 Ki = 26 nM T40016 CZO0L1 11595527 Ki = 5.8 nM T40016 CAO2P1 11596392 IC50 = 17 nM T40016 CJWP94 11596794 EC50 = 8.318 nM T40016 C53OBJ 11597965 Ki = 22 nM T40016 C54HCR 11598367 IC50 = 12.59 nM T40016 C3FJQ8 11602375 IC50 = 35000 nM T40016 C8RO4G 11611666 IC50 = 0.5012 nM T40016 C7PS2W 11612527 IC50 = 15.85 nM T40016 C7ME6V 11613022 IC50 = 9.55 nM T40016 CC0I2P 11613420 IC50 = 8.511 nM T40016 CSB97O 11617028 Ki = 0.3 nM T40016 CC49FR 11617298 Ki = 79 nM T40016 CR5DA0 11617684 Ki = 24 nM T40016 CI1D2W 11620916 Ki = 0.8 nM T40016 C1IEC7 11627493 IC50 = 11.48 nM T40016 CRF4E1 11631740 EC50 = 0.8 nM T40016 CW6R3T 11631784 Ki = 0.8 nM T40016 CRL3A7 11632925 IC50 = 25 nM T40016 CQB0E3 11633482 IC50 = 15 nM T40016 C9DNG1 11640164 IC50 = 4 nM T40016 CC4LE3 11640246 IC50 = 3.09 nM T40016 CB4E0S 11645780 Ki = 460 nM T40016 C3MHY7 11646048 IC50 = 5.3 nM T40016 C1RJ3I 11646689 IC50 = 9 nM T40016 CX3L5S 11647533 IC50 = 18 nM T40016 C2AD9C 11647851 Ki = 10 nM T40016 CU3K9V 11653520 Ki = 4.5 nM T40016 C4S5RG 11655053 IC50 = 34 nM T40016 C5L3GN 11656415 Ki = 1.6 nM T40016 CDOZ32 11661172 IC50 = 10 nM T40016 C1CEJ0 11663141 EC50 = 18.62 nM T40016 CEQR07 11663523 EC50 = 17.78 nM T40016 CH8F5J 11663592 IC50 = 5.012 nM T40016 C0LEZ3 11667800 IC50 = 14 nM T40016 C5XEN0 11668719 IC50 = 340 nM T40016 CCWJ64 11668984 IC50 = 48 nM T40016 CTE80K 11671653 Ki = 8.6 nM T40016 CM57PA 11682250 IC50 = 12 nM T40016 CZPK72 11682989 IC50 = 15 nM T40016 C1HA4U 11684596 IC50 = 125.89 nM T40016 C4QA6V 11685011 IC50 = 6.31 nM T40016 C8SY4D 11688929 Ki = 90 nM T40016 CCK83U 11690269 IC50 = 8 nM T40016 CH7I6J 11691206 IC50 = 12.59 nM T40016 CY07JH 11696378 IC50 = 51 nM T40016 CBU02W 11696959 IC50 = 4 nM T40016 C2S9IT 11697271 IC50 = 13 nM T40016 CGR32I 11697882 IC50 = 5 nM T40016 C42NIT 11697950 Ki = 340 nM T40016 C25NSM 11699191 IC50 = 8.128 nM T40016 C7VC2U 11699294 IC50 = 1380.38 nM T40016 C3OQH4 11703401 IC50 = 67 nM T40016 C75IBX 11704529 IC50 = 20 nM T40016 CGX54N 11704756 IC50 = 320 nM T40016 CI4JW3 11706478 Ki = 0.9 nM T40016 CO2N1W 11710364 IC50 = 9 nM T40016 C8OPA1 11710962 IC50 = 19 nM T40016 CW3N8H 11711766 IC50 = 280 nM T40016 C1TQX9 11712150 Ki = 15 nM T40016 C6AB0O 11712629 IC50 = 16.6 nM T40016 COEU05 11719039 IC50 = 60 nM T40016 CM3BG2 11724520 IC50 > 2000 nM T40016 C4OH1Y 11726899 Ki > 10000 nM T40016 C0VJ3I 11727825 Ki > 5000 nM T40016 CVA1S3 11728656 Ki = 5.42 nM T40016 CZ0B7H 11731863 Ki = 84 nM T40016 CYJ73N 11733546 IC50 = 40.9 nM T40016 CQO76Z 11741168 IC50 = 1400 nM T40016 CJC5A2 11741840 IC50 = 4.2 nM T40016 C87YNC 11741891 IC50 = 22 nM T40016 CH92VI 11743259 IC50 = 15 nM T40016 CV49MT 11747706 IC50 = 133 nM T40016 C5HLU8 11750204 IC50 = 1.4 nM T40016 C9UED8 11752131 EC50 = 0.2 nM T40016 CY1F4I 11752649 EC50 = 0.2 nM T40016 C3XF4G 11755231 IC50 = 7.943 nM T40016 CKD9R8 11757239 IC50 = 9.2 nM T40016 CEWP04 11771756 IC50 = 8.8 nM T40016 CQU0E7 11774868 IC50 = 14 nM T40016 COI0P1 11774981 IC50 = 510 nM T40016 CR70FP 11794088 Ki = 2379 nM T40016 CU7EJ1 11822858 Ki = 157 nM T40016 C5FRJ6 11825145 Ki = 18 nM T40016 C4U8KY 12085089 IC50 = 2 nM T40016 CEV10S 13278723 IC50 = 1.8 nM T40016 C7ICM3 15298636 IC50 = 18 nM T40016 C14LTD 15463551 IC50 = 10 nM T40016 CC15FW 16049465 IC50 = 2.3 nM T40016 CMZH47 16051364 IC50 > 10000 nM T40016 C3QOV0 16099227 IC50 = 10 nM T40016 CW6LO1 16099229 IC50 > 2000 nM T40016 C2R4PK 16099231 IC50 = 38 nM T40016 C9KM7X 16099232 IC50 = 120 nM T40016 C05CYN 16099234 IC50 = 950 nM T40016 CJQ8A1 16099236 IC50 = 6 nM T40016 CA72YW 16099237 IC50 = 780 nM T40016 CS07DB 16099238 IC50 = 4 nM T40016 C42ESN 16099240 IC50 = 5 nM T40016 CMZ91J 16099242 IC50 > 2000 nM T40016 CF69RC 16099243 IC50 > 2000 nM T40016 C60GEM 16099245 IC50 = 110 nM T40016 CE48CS 16099246 IC50 = 650 nM T40016 CTF2M7 16099247 IC50 = 4 nM T40016 CX9BK2 16099248 IC50 = 54 nM T40016 CN6PA9 16099249 IC50 = 28 nM T40016 C9Z6AK 16099250 IC50 = 10 nM T40016 C5Z8HR 16099251 IC50 = 11 nM T40016 CWK76M 16099252 IC50 = 3 nM T40016 CU1YV4 16099253 IC50 = 34 nM T40016 CN5VS8 16099254 IC50 = 125 nM T40016 CC24LB 16110489 EC50 > 10 nM T40016 C3BU9M 16216822 IC50 = 29 nM T40016 C1Q5SV 16220168 IC50 = 5600 nM T40016 CH6CN0 16658901 Ki = 8500 nM T40016 CU9LS2 16661702 EC50 = 7900 nM T40016 C9F2VT 16665286 IC50 = 3.9 nM T40016 C2H9EM 16665289 IC50 = 6.9 nM T40016 CT6Y5F 16665374 IC50 = 3.4 nM T40016 CI95KE 16665449 IC50 = 9.7 nM T40016 CYW0T9 16665451 IC50 = 12 nM T40016 CP8VM0 16665452 IC50 = 23 nM T40016 CPNJ02 16665453 IC50 = 5.7 nM T40016 C0OG7T 16665528 IC50 = 16 nM T40016 CMC9W0 16665533 IC50 = 12 nM T40016 CV3OM1 16665605 IC50 = 7.7 nM T40016 CCN5F6 16665606 IC50 = 795 nM T40016 CG5UM0 16665608 IC50 = 12 nM T40016 CLJ2U5 16666385 IC50 = 5.2 nM T40016 C1UY8J 16666386 IC50 = 1.47 nM T40016 CWR10T 16666470 IC50 = 5.4 nM T40016 CWEJ30 16666472 IC50 = 1.5 nM T40016 C0Y2OK 16721017 IC50 = 304 nM T40016 CE71BC 16722203 IC50 = 37.6 nM T40016 C92NRU 16727109 EC50 > 25000 nM T40016 CF6V2J 16730097 IC50 = 111 nM T40016 CWK35C 16730429 IC50 = 14000 nM T40016 C9BC0L 16732000 Ki > 10000 nM T40016 CLC2Z8 16739323 IC50 = 86.5 nM T40016 CAL7M5 16756781 IC50 = 34000 nM T40016 C3RPY2 17747503 IC50 = 6.3 nM T40016 CLNU15 17758014 EC50 = 0.2 nM T40016 C62WRI 17758132 EC50 = 0.2 nM T40016 C5GRB8 17758133 EC50 = 0.4 nM T40016 CSKX58 17758233 Ki = 1.2 nM T40016 C7CPW9 17758234 EC50 = 0.1 nM T40016 CI5KT6 17758236 EC50 = 0.5 nM T40016 CE8C5G 17758459 IC50 = 1 nM T40016 C32WCP 17758569 EC50 = 0.6 nM T40016 C05ARI 17758570 EC50 = 1.4 nM T40016 CX03YG 18188955 IC50 = 2 nM T40016 CQLU68 18189214 IC50 = 402 nM T40016 CH39OX 18504012 IC50 = 48 nM T40016 CYZ71G 18511908 IC50 = 370 nM T40016 C7ZIF9 18511910 IC50 = 2.9 nM T40016 CEFA90 18511931 IC50 = 34 nM T40016 CEDU50 18511945 IC50 = 96 nM T40016 C4EU2J 18511975 IC50 = 470 nM T40016 CL91CU 18511977 IC50 = 14 nM T40016 CQ4BF7 18511980 IC50 = 100 nM T40016 C9C8GH 18511994 IC50 = 48 nM T40016 CZO79P 18512002 IC50 = 58 nM T40016 C05YOA 18512008 IC50 = 56 nM T40016 C03SPA 18512022 IC50 = 47 nM T40016 CR5G8F 18512030 IC50 = 63 nM T40016 C7LFU4 18512032 IC50 = 320 nM T40016 CF6E2C 18512049 IC50 = 26 nM T40016 C1ZVD4 18512058 IC50 = 17 nM T40016 CGJ56E 18512087 IC50 = 36 nM T40016 C0C6BG 18512103 IC50 = 11 nM T40016 C49PLT 18512117 IC50 = 138 nM T40016 CX3B4O 18512130 IC50 = 3.9 nM T40016 C3C7ID 18512158 IC50 = 5.4 nM T40016 CJCF08 18512161 IC50 = 270 nM T40016 C7XC4K 18512162 IC50 = 1.4 nM T40016 C5YX7A 18512163 IC50 = 250 nM T40016 CR19ST 18512166 IC50 = 28 nM T40016 CB5C3I 18512168 IC50 = 11 nM T40016 CFI8E1 18512170 IC50 = 15 nM T40016 CM4B9R 18512171 IC50 = 220 nM T40016 CRP45C 18512178 IC50 = 1000 nM T40016 C64PAE 18512192 IC50 = 13 nM T40016 C14RFT 18512213 IC50 = 8.8 nM T40016 CTX2Z5 18512224 IC50 = 21 nM T40016 CL42KX 18512282 IC50 = 290 nM T40016 CX1FQ2 18512329 IC50 = 2.4 nM T40016 CEN14G 18512334 IC50 = 5.7 nM T40016 CD8JC6 18512366 IC50 = 120 nM T40016 CJG26V 18512380 IC50 = 1.5 nM T40016 CLX02Q 18512392 IC50 = 2.7 nM T40016 CXM9D1 18512399 IC50 = 60 nM T40016 CS9CI5 18551230 EC50 = 45 nM T40016 CBI64N 18551237 IC50 = 8 nM T40016 CLUA26 18551266 IC50 = 230 nM T40016 C5ZYJ0 20231824 Ki = 50 nM T40016 CEH7V5 20786216 IC50 = 6.31 nM T40016 CR73OM 21136439 IC50 = 892 nM T40016 CF0S6J 21210483 IC50 = 11700 nM T40016 C97WCO 21941658 EC50 = 10 nM T40016 CCI89R 21948853 IC50 = 1.995 nM T40016 CB2SF4 21948904 IC50 = 3.162 nM T40016 CP7S2I 21970730 IC50 = 289 nM T40016 C2ZP7V 22218142 IC50 > 10000 nM T40016 CWA9Q6 22284899 IC50 = 760 nM T40016 CY5Z4Q 22314851 IC50 = 13 nM T40016 C5N1HK 22314910 IC50 > 5000 nM T40016 C6R1WN 22314926 IC50 = 42 nM T40016 CDQ10L 22314947 IC50 = 150 nM T40016 C8XAR4 22314951 IC50 = 220 nM T40016 C84QJV 22314968 IC50 = 12 nM T40016 C4I7OB 22314982 IC50 = 23 nM T40016 CGWM75 22315021 IC50 = 320 nM T40016 C1GIZ6 22315043 IC50 = 20 nM T40016 C1QTK4 22398492 IC50 = 7 nM T40016 C6CSB4 22398502 IC50 = 160 nM T40016 CR8N1E 22398506 IC50 = 27 nM T40016 CM83TU 22398533 IC50 = 8 nM T40016 C34LHW 22398559 IC50 = 21 nM T40016 CJBW90 22398592 IC50 = 23 nM T40016 CEJ65O 22398627 IC50 = 8 nM T40016 CCYS56 22566499 IC50 = 303 nM T40016 CGE03P 22566506 IC50 = 260 nM T40016 CH29BV 22566507 IC50 = 116 nM T40016 C21YKI 22566509 IC50 = 404 nM T40016 CU8D7L 22566515 IC50 > 2000 nM T40016 CPQ9O5 22605977 IC50 = 2100 nM T40016 CCF52I 22605979 IC50 > 2000 nM T40016 CGY94Z 23433542 IC50 = 3200 nM T40016 CZ9L3J 23552303 IC50 = 87 nM T40016 CL0H7I 23595919 Ki = 303 nM T40016 C56STL 23595942 EC50 = 330.6 nM T40016 CP9SN1 23596227 Ki = 92.6 nM T40016 CNVC31 23596254 Ki = 82.5 nM T40016 C9O6RB 23596322 Ki = 4.1 nM T40016 CNLR52 23596329 Ki = 8.7 nM T40016 CMV6U7 23596330 Ki = 22.6 nM T40016 C4F7OG 23596337 Ki = 3.9 nM T40016 CJ0XR3 23625602 IC50 = 1.585 nM T40016 CF4UA3 23648072 IC50 = 1060 nM T40016 CSV4D3 23648197 EC50 = 19 nM T40016 CBI6J3 23648200 EC50 = 3 nM T40016 CT80JO 23648203 EC50 = 46 nM T40016 CD74QP 23648204 EC50 = 32 nM T40016 CHW3X2 23648205 EC50 = 3 nM T40016 C0VE5H 23648206 EC50 = 5 nM T40016 C7BLN0 23992759 Ki = 157.7 nM T40016 CWPH96 24180508 IC50 = 99 nM T40016 CS1KX2 24180659 Ki = 14 nM T40016 CZI4C6 24739672 Ki = 1860 nM T40016 CS23KY 24739834 Ki = 977 nM T40016 C1M9QG 24739836 Ki = 927 nM T40016 CG5SJ0 24739997 Ki = 1530 nM T40016 C7Z1HW 24740156 Ki = 780 nM T40016 CTE1N2 24748569 EC50 > 10000 nM T40016 CQ57SD 24748957 IC50 = 48.98 nM T40016 CWL9G2 24748958 IC50 = 8.128 nM T40016 C14ZOJ 24748959 EC50 = 41.69 nM T40016 CSP7E5 24748960 EC50 = 61.66 nM T40016 C8J3HZ 24748961 IC50 = 6.607 nM T40016 CXAJ63 24749047 IC50 = 7.244 nM T40016 CAS4V3 24749048 IC50 = 8.913 nM T40016 C6TAE7 24749049 IC50 = 1.585 nM T40016 C36ECZ 24749050 IC50 = 30.2 nM T40016 CMBK68 24749150 IC50 = 147.91 nM T40016 C7ZU9P 24749151 EC50 = 12.88 nM T40016 C4WYE7 24749678 Ki = 167 nM T40016 CY2JS4 24749684 Ki = 54.4 nM T40016 C2QHO3 24749808 Ki = 5.93 nM T40016 CR1G7M 24768971 EC50 = 3.981 nM T40016 CM8Y4V 24769095 IC50 = 0.7943 nM T40016 C5S6JN 24780149 IC50 = 6.31 nM T40016 CW5TJ7 24781731 IC50 = 15.85 nM T40016 CPVS80 24789142 EC50 = 4.1 nM T40016 C8OCU9 24789150 Ki = 1 nM T40016 CR48VC 24809711 EC50 = 7.943 nM T40016 CGC0D7 24816319 IC50 = 11 nM T40016 CNM45B 24850992 IC50 = 1510 nM T40016 C1JTW2 24851053 Ki = 0.257 nM T40016 CC53XL 24860583 Ki = 15 nM T40016 C5Y2TN 24873449 IC50 = 0.69 nM T40016 CGE0V4 24882669 IC50 = 10 nM T40016 C58RHY 24883011 IC50 = 2500 nM T40016 CW35CK 24883012 IC50 = 1800 nM T40016 C3SC0V 24883054 IC50 = 1700 nM T40016 C4SA6C 24883055 IC50 = 470 nM T40016 C5LZK2 24895096 IC50 = 34 nM T40016 CMH52V 24936311 Ki = 0.53 nM T40016 CA3O5Q 24936312 Ki = 10.2 nM T40016 COGP96 24936313 Ki = 5.14 nM T40016 C5WOB6 24936314 Ki = 0.72 nM T40016 CM8NR9 24936446 Ki = 1.74 nM T40016 CVY09S 24936449 Ki = 0.64 nM T40016 CD8JT0 24936598 Ki = 11 nM T40016 CT8L2W 24936727 Ki = 14 nM T40016 CFK6W8 24936729 Ki = 11 nM T40016 C1BR3F 24936732 Ki = 18 nM T40016 CBN24H 24936982 Ki = 1.7 nM T40016 C71KJS 24936984 Ki = 2.4 nM T40016 C65YPH 24937240 Ki = 5.7 nM T40016 C7YCB3 24937242 Ki = 12 nM T40016 C26TWN 24937362 Ki = 5 nM T40016 C26HUZ 24937363 EC50 = 10 nM T40016 CEV09L 24937493 Ki = 2.4 nM T40016 CZ91CN 24937934 IC50 = 0.3162 nM T40016 C4YTH3 24937935 IC50 = 0.1259 nM T40016 C9KFD4 24937936 IC50 = 0.07943 nM T40016 CXTL09 24945221 Ki = 2 nM T40016 CQFZ96 24945227 Ki = 3 nM T40016 CQ2FL3 24945386 Ki = 2 nM T40016 C5DW7P 24945389 Ki = 1 nM T40016 CTV40U 24945468 Ki = 4 nM T40016 CV03UT 24945548 Ki < 1 nM T40016 CYL54C 24945619 Ki < 1 nM T40016 C8L9PC 24945705 Ki = 10 nM T40016 C06PDG 24952192 Ki = 0.3 nM T40016 CG1CF9 24952193 Ki = 0.8 nM T40016 CZC7L8 24953162 IC50 = 0.91 nM T40016 C1CUZ4 24953163 IC50 = 13 nM T40016 CZB7M8 24953166 IC50 = 7.4 nM T40016 CU3A7E 24953513 IC50 = 37 nM T40016 CKML07 24954062 Ki = 1 nM T40016 C07FUV 24954066 Ki = 13 nM T40016 CP1G9U 24954421 Ki = 4 nM T40016 CNJS10 24954422 Ki = 169 nM T40016 CC4P9R 24954791 Ki = 2 nM T40016 CSD27Y 24954792 Ki = 4 nM T40016 CW7O3D 24954793 Ki = 4 nM T40016 CZ14BO 24954794 Ki = 2 nM T40016 C4W7BN 24954947 IC50 = 0.75 nM T40016 C6XC2R 24954951 IC50 = 1.4 nM T40016 CFK32R 24955041 Ki = 6 nM T40016 CL70XN 24955148 Ki = 2 nM T40016 CN9L1B 24955149 Ki = 1 nM T40016 CLJ87T 24955150 Ki = 8 nM T40016 CK96WS 24955151 Ki = 5 nM T40016 CVU18K 24955152 Ki = 5 nM T40016 CRBW74 24956466 Ki = 412 nM T40016 CYES17 24957737 Ki = 55 nM T40016 C85BHZ 24958028 IC50 = 12.59 nM T40016 C3VO7Q 24960588 EC50 = 39.81 nM T40016 C83YKB 24961057 Ki = 11 nM T40016 CQ3X6G 24961686 EC50 = 25.12 nM T40016 CZ89IP 24961687 EC50 = 6.31 nM T40016 CZG93W 24961689 EC50 = 251.19 nM T40016 CLY07O 24961690 EC50 = 50.12 nM T40016 C42YHP 24962051 IC50 = 316.23 nM T40016 C5W1IT 24962055 IC50 = 19.95 nM T40016 CN49EG 24962146 Ki = 151 nM T40016 CYEF46 24964075 Ki < 1 nM T40016 CVI3O1 24964440 Ki = 2 nM T40016 CS7WY4 24964443 Ki < 1 nM T40016 CIGM27 24983460 IC50 = 20 nM T40016 CP1VY8 24997743 IC50 = 98 nM T40016 CM2Z0U 25011854 IC50 = 0.66 nM T40016 CX7I2K 25012028 IC50 = 4.6 nM T40016 CR7GA9 25012190 IC50 = 0.05 nM T40016 CO9S6B 25013321 IC50 = 0.62 nM T40016 CHY0D7 25013322 IC50 = 0.13 nM T40016 C0J3CQ 25013326 IC50 = 0.25 nM T40016 CZE7X8 25013489 IC50 = 0.21 nM T40016 CAF85M 25013490 IC50 = 0.08 nM T40016 C0TPS5 25013653 IC50 = 2.9 nM T40016 CHN41A 25013654 IC50 = 0.03 nM T40016 CWU91M 25013811 EC50 = 1.3 nM T40016 CSH29L 25013812 IC50 = 0.04 nM T40016 C68SGK 25014203 IC50 = 3.1 nM T40016 C6SA2C 25014204 IC50 = 5.09 nM T40016 CKUA52 25014206 IC50 = 1.41 nM T40016 C0LO9C 25028373 EC50 = 50.12 nM T40016 C4H7UP 25048180 IC50 = 4100 nM T40016 C2G1JK 25053351 Ki > 30000 nM T40016 CAW8M0 25070694 IC50 > 3000 nM T40016 C3H0KR 25110774 Ki = 0.6 nM T40016 C4GLY1 25110785 Ki = 1.4 nM T40016 CCL91F 25110786 Ki = 0.8 nM T40016 C21XDY 25145083 Ki > 10000 nM T40016 CS6JQ1 25167502 Ki = 1.5 nM T40016 C0XPW9 25168896 IC50 = 210 nM T40016 CUL27D 25168900 IC50 = 95 nM T40016 CEV2D7 25205475 IC50 = 2 nM T40016 C9S0ZW 25205477 IC50 = 7 nM T40016 C49KHR 25206116 IC50 = 2 nM T40016 C87ZHT 25231296 IC50 = 0.9 nM T40016 CLY9W3 25235364 IC50 = 1.5 nM T40016 C3FW0Y 25257459 IC50 = 360 nM T40016 CVO06A 25257700 IC50 = 1100 nM T40016 CN03HI 25257925 IC50 = 17 nM T40016 CY6X2V 25258136 IC50 = 5.6 nM T40016 CS49WQ 25258137 IC50 = 3.5 nM T40016 CV4Y6N 25258138 IC50 = 6.2 nM T40016 C5NGC7 25258139 IC50 = 1.5 nM T40016 C1OJ6Z 25258140 IC50 > 1000 nM T40016 CWT31Y 25258141 IC50 > 1000 nM T40016 CJ68WY 25258142 IC50 = 21 nM T40016 CLX0P9 25258381 IC50 = 2.3 nM T40016 CM48WL 25258382 IC50 = 1500 nM T40016 CNLS64 25258386 IC50 = 2.5 nM T40016 CSG7P9 25258611 IC50 = 3 nM T40016 CN87ME 25258614 IC50 = 3.8 nM T40016 CX89HM 44138106 Ki = 1 nM T40016 C9LCJ5 44156980 IC50 = 4.8 nM T40016 CZAJ06 44193143 Ki = 6.2 nM T40016 CS36WU 44193144 Ki = 7.6 nM T40016 CXZ35T 44193145 Ki = 6.8 nM T40016 C2MOF7 44193146 Ki = 7.8 nM T40016 CWR6X1 44193147 Ki = 4.3 nM T40016 CF02JG 44193242 Ki = 14.3 nM T40016 C3JOW4 44193245 IC50 = 13 nM T40016 C9WB1Z 44193246 Ki = 16.1 nM T40016 CKDG10 44193342 Ki = 70 nM T40016 C4Q0SG 44193344 IC50 = 7.5 nM T40016 CK9ZL7 44193440 EC50 = 3.5 nM T40016 CYE8V6 44219884 IC50 = 8.3 nM T40016 C0R6PO 44220470 IC50 = 22 nM T40016 C0GW9R 44220471 IC50 = 16 nM T40016 C2ZV8C 44220675 IC50 = 20 nM T40016 CVF35J 44220676 IC50 = 8.5 nM T40016 CCR9E5 44220677 IC50 = 9.8 nM T40016 CU4Y0F 44222262 IC50 = 20 nM T40016 CR4O5D 44222437 IC50 = 16 nM T40016 CZHU72 44222438 IC50 = 12 nM T40016 CV6K2G 44222616 IC50 = 9.3 nM T40016 CXR5O7 44250279 IC50 = 62 nM T40016 C9QED8 44250280 IC50 = 17 nM T40016 CHGI03 44251606 IC50 = 13 nM T40016 C0OA6M 44264483 IC50 > 10000 nM T40016 COCE32 44264569 IC50 > 10000 nM T40016 CI0TN2 44264577 IC50 > 10000 nM T40016 CXOR54 44264579 IC50 > 10000 nM T40016 C01HSQ 44264588 IC50 > 10000 nM T40016 CP8OC7 44282950 Ki = 367 nM T40016 CT21MG 44292732 IC50 > 5000 nM T40016 CUS81V 44292816 IC50 = 310 nM T40016 CZ9MR4 44292832 IC50 = 40 nM T40016 C5QB1K 44292948 IC50 = 216.7 nM T40016 CBGI65 44293017 IC50 > 5000 nM T40016 CFR15U 44293099 IC50 = 310 nM T40016 CK8QL2 44293267 IC50 = 88 nM T40016 COF8L6 44293283 IC50 = 440 nM T40016 C9NO6K 44293320 IC50 = 15 nM T40016 C3LEM6 44293322 IC50 = 230 nM T40016 CMR51Y 44293351 IC50 = 23 nM T40016 C4C8ES 44293372 IC50 = 110 nM T40016 CJ6D4C 44294728 IC50 = 770 nM T40016 CJPD50 44294768 IC50 = 440 nM T40016 C6X2IH 44295653 Ki 10000 nM T40016 C1DBA2 44305237 IC50 = 324 nM T40016 CDB54J 44305270 IC50 = 177 nM T40016 C0XLN6 44305556 IC50 = 10 nM T40016 C17NWG 44305617 IC50 = 210 nM T40016 CHB82F 44305684 IC50 = 1929 nM T40016 C1UK4M 44305720 IC50 = 689 nM T40016 CTW67P 44305733 IC50 = 2170 nM T40016 CH4PU5 44305819 IC50 = 29 nM T40016 C7Y9TZ 44305822 IC50 = 31 nM T40016 CDXK57 44305874 IC50 = 3026 nM T40016 CP1MX9 44305909 IC50 = 1204 nM T40016 C6N1AR 44305929 IC50 = 1872 nM T40016 C9U6SZ 44306067 IC50 = 753 nM T40016 CE4S3K 44306078 IC50 = 812 nM T40016 C6OPD2 44306824 IC50 = 827 nM T40016 CLP97B 44310115 IC50 = 14000 nM T40016 C7F9NW 44310117 IC50 = 2700 nM T40016 CJ78FG 44310121 IC50 = 6600 nM T40016 CO7XP6 44310122 IC50 = 3800 nM T40016 CA73TS 44310248 IC50 = 25000 nM T40016 C2QV1X 44310288 IC50 = 220 nM T40016 CRT5J9 44310289 IC50 = 20 nM T40016 CD89XZ 44310345 IC50 = 1100 nM T40016 CKI2R0 44310353 IC50 = 1100 nM T40016 CQ17GY 44310359 IC50 = 2200 nM T40016 CKX52S 44310378 IC50 = 580 nM T40016 CD3X9U 44310397 IC50 = 850 nM T40016 CC2R3E 44310469 IC50 = 690 nM T40016 CMIG93 44310515 IC50 = 910 nM T40016 C7YKJ8 44310518 IC50 = 230 nM T40016 CV6AP0 44310535 IC50 = 42 nM T40016 C5A1XR 44310536 IC50 = 220 nM T40016 C7EWU8 44310595 IC50 = 130 nM T40016 CL42EC 44310626 IC50 = 110 nM T40016 CJH8Y1 44310641 IC50 = 570 nM T40016 CZ86HK 44310715 IC50 = 450 nM T40016 C4TU5G 44314208 IC50 = 16.7 nM T40016 CW21CA 44317747 Ki = 0.1 nM T40016 CT62WI 44341706 Ki = 394 nM T40016 CO10KF 44341745 Ki = 749 nM T40016 CP0AQ3 44341860 Ki = 130 nM T40016 CE62XL 44341871 Ki = 813 nM T40016 CIFK12 44341872 Ki = 158 nM T40016 C6KSD0 44341876 Ki = 51 nM T40016 CP6LV3 44341880 Ki = 533 nM T40016 C8RQS2 44342092 Ki = 260 nM T40016 CDGP02 44353994 IC50 = 188 nM T40016 C73CXK 44354006 Ki = 232 nM T40016 C0N3TD 44354884 IC50 = 900 nM T40016 CPQ2A6 44354885 Ki = 43 nM T40016 CM0G1V 44354886 IC50 = 780 nM T40016 CL6G3Q 44355066 IC50 = 35 nM T40016 C76OKZ 44370955 IC50 = 6.4 nM T40016 CZO25G 44371166 IC50 = 400 nM T40016 CILC83 44371259 IC50 = 1.4 nM T40016 CSAU31 44377064 IC50 > 10000 nM T40016 C7H9NC 44377081 IC50 > 10000 nM T40016 C60DYH 44377090 IC50 = 5800 nM T40016 CVH2R3 44377098 IC50 = 3000 nM T40016 CYLI63 44377110 IC50 > 10000 nM T40016 CQX39I 44377356 IC50 = 1400 nM T40016 C9FJW4 44377382 IC50 = 2100 nM T40016 C6SX0M 44393033 IC50 = 75 nM T40016 C7E9BC 44393047 IC50 = 460 nM T40016 CU4VI1 44393048 IC50 = 6.5 nM T40016 CM4DQ8 44393050 IC50 = 15 nM T40016 C2FJ0T 44393051 IC50 = 57 nM T40016 C8Y4RP 44393060 IC50 = 37 nM T40016 CK58MC 44393061 IC50 = 6.8 nM T40016 CTI0L9 44393062 IC50 = 23 nM T40016 CJ59US 44393181 IC50 = 71 nM T40016 CUK98X 44393182 IC50 = 170 nM T40016 C5NM4W 44393183 IC50 = 93 nM T40016 CFL1B2 44393188 IC50 > 1000 nM T40016 CMSV15 44393246 IC50 = 56 nM T40016 C12XBN 44393247 IC50 = 50 nM T40016 C89QJE 44394919 EC50 = 5.6 nM T40016 C5TY0K 44394965 IC50 = 165 nM T40016 C13SYV 44396250 Ki = 0.42 nM T40016 CB1P0S 44396251 Ki = 0.22 nM T40016 C0U5DZ 44396253 Ki = 0.16 nM T40016 CU3G0Y 44396254 Ki = 0.18 nM T40016 CHY1C3 44396271 Ki = 3 nM T40016 C29MBI 44396272 Ki = 2.1 nM T40016 C4TQ6N 44396282 Ki = 0.27 nM T40016 CH2Y3L 44396283 Ki = 0.27 nM T40016 CWZB52 44396284 Ki = 0.3 nM T40016 CD80LM 44396296 Ki = 0.4 nM T40016 C6SI5L 44396297 Ki = 0.39 nM T40016 CR4H1E 44396316 Ki = 0.42 nM T40016 C45LRH 44396317 Ki = 0.27 nM T40016 CPR85C 44396328 Ki = 0.22 nM T40016 CVF02B 44396329 Ki = 0.11 nM T40016 C5JG6H 44396330 Ki = 0.8 nM T40016 CA8V4G 44396331 Ki = 1.1 nM T40016 C57CPQ 44396332 Ki = 1.2 nM T40016 CGPV87 44396333 Ki = 6.5 nM T40016 CHG9O1 44396490 IC50 = 979 nM T40016 CPQL46 44396502 IC50 = 1812 nM T40016 CNH4C3 44396512 IC50 = 0.9 nM T40016 C1OYG3 44396526 IC50 = 870 nM T40016 CO25DV 44396547 IC50 = 1294 nM T40016 C7UP4O 44398565 IC50 = 5.012 nM T40016 CYCH34 44401707 IC50 = 9.1 nM T40016 CAG6T1 44401853 EC50 = 13 nM T40016 CA41SJ 44402030 IC50 = 10.2 nM T40016 C4PN2B 44402151 IC50 = 7.1 nM T40016 C61MGU 44402680 IC50 = 6.6 nM T40016 C9R8QP 44402681 IC50 = 8.5 nM T40016 CGL2T0 44402683 IC50 = 10 nM T40016 C63UET 44402699 IC50 = 8.4 nM T40016 C7VCZ5 44402711 IC50 = 7.1 nM T40016 CA5PI7 44402722 IC50 = 26 nM T40016 C2RLY1 44402736 IC50 = 2.2 nM T40016 CXI97U 44402746 IC50 = 8 nM T40016 C91WCI 44402753 IC50 = 5.6 nM T40016 CX4RZ6 44402754 IC50 = 5.5 nM T40016 C19KGF 44402755 IC50 = 18 nM T40016 CG4E3M 44402763 IC50 = 49 nM T40016 CRN9I4 44402766 IC50 = 10 nM T40016 C5Q6LX 44402767 IC50 = 3.1 nM T40016 CGRX27 44402769 IC50 = 24 nM T40016 C9R5SU 44402770 IC50 = 5.8 nM T40016 C7P6OT 44402796 IC50 = 10 nM T40016 C9XS4E 44402799 IC50 = 1.2 nM T40016 C1HE7G 44402805 IC50 = 2.1 nM T40016 CBUG70 44402817 IC50 = 2.7 nM T40016 CP1SY8 44402818 IC50 = 12 nM T40016 CBH76D 44402820 IC50 = 8.9 nM T40016 C7JU0O 44402832 IC50 = 21 nM T40016 CE5U1B 44402833 IC50 = 65 nM T40016 C36CWT 44402841 IC50 = 8.3 nM T40016 CW79UB 44402847 IC50 = 28 nM T40016 CP2IG4 44402961 IC50 > 2000 nM T40016 CXHF58 44403036 IC50 = 79 nM T40016 C25YCZ 44403037 IC50 > 2000 nM T40016 C6JNI4 44403038 EC50 = 2370 nM T40016 C45SOW 44403039 EC50 = 620 nM T40016 C1LUK3 44407314 IC50 = 2000 nM T40016 CA3B0O 44409475 Ki > 100 nM T40016 CYQZ19 44420005 IC50 = 481.5 nM T40016 CLA3J0 44420007 IC50 = 43 nM T40016 C1SFW5 44420010 IC50 = 0.7 nM T40016 C0C6FH 44420011 IC50 = 9 nM T40016 C0YG8R 44420014 IC50 = 0.4 nM T40016 CB1SU4 44420015 IC50 = 60.7 nM T40016 CHBG29 44420017 IC50 = 3.2 nM T40016 C5UIJ1 44420022 IC50 = 30.7 nM T40016 C91DUB 44420023 IC50 = 4.9 nM T40016 C2CJ6H 44420024 IC50 = 2.5 nM T40016 CAR8Y6 44420029 IC50 = 0.4 nM T40016 COD73E 44420033 IC50 = 1.5 nM T40016 CV38YP 44420040 IC50 = 0.7 nM T40016 CZFY86 44420051 IC50 = 1.5 nM T40016 C7I6RY 44420054 IC50 = 4.5 nM T40016 C5CW4E 44420057 IC50 = 0.1 nM T40016 CH1R7M 44420600 EC50 > 10 nM T40016 CF8N9J 44425531 IC50 = 204.3 nM T40016 CQ6R5N 44425537 IC50 = 33.4 nM T40016 CGY0M9 44425538 IC50 = 55.5 nM T40016 C6RGU2 44425539 IC50 = 166.9 nM T40016 CT7LE3 44425540 IC50 = 558 nM T40016 CT8Q9O 44425541 IC50 = 315 nM T40016 CE53FQ 44425542 IC50 > 3000 nM T40016 C0B6TU 44426753 Ki = 20 nM T40016 CO9JF7 44426754 Ki = 78 nM T40016 CV10KQ 44426759 Ki = 360 nM T40016 CF65BV 44426762 Ki = 470 nM T40016 CM01BZ 44426766 Ki = 19 nM T40016 C6EN4A 44426775 Ki = 154 nM T40016 CS5AL9 44426780 Ki = 227 nM T40016 CXZ4S3 44426781 Ki = 8.7 nM T40016 C8HO4K 44426782 Ki = 9.1 nM T40016 CXWC04 44426783 Ki = 31 nM T40016 C5OPU7 44426784 Ki = 14 nM T40016 CHT52I 44426787 Ki = 37 nM T40016 C35CJU 44426789 Ki = 45 nM T40016 C0FEN3 44426790 Ki = 7.1 nM T40016 CUK45W 44426792 Ki = 103 nM T40016 C19MJP 44426793 Ki = 4.9 nM T40016 CDN25Y 44426794 Ki = 46 nM T40016 C1ZDA4 44426795 Ki = 9.2 nM T40016 CFSH46 44426796 Ki = 6.5 nM T40016 CD0QH9 44426797 Ki = 47 nM T40016 C4FDY6 44427105 Ki = 4 nM T40016 C8OMK7 44427108 Ki = 1.8 nM T40016 C1M8YG 44427110 Ki = 0.9 nM T40016 CXO0S9 44427111 Ki = 0.6 nM T40016 C92VJT 44427112 Ki = 1.8 nM T40016 CY76PU 44427113 Ki = 4.8 nM T40016 C9AT0E 44427114 Ki = 2.7 nM T40016 CHMW84 44427115 Ki = 3 nM T40016 CM7TQ2 44427116 Ki = 31 nM T40016 C42FIO 44427117 Ki = 0.5 nM T40016 C79VAB 44427118 Ki = 1.1 nM T40016 CZM7N0 44430346 IC50 = 65.1 nM T40016 C2AJC1 44430347 IC50 = 64.8 nM T40016 C65HXP 44430353 IC50 = 62.7 nM T40016 C7O2JW 44430354 IC50 = 113.2 nM T40016 CK8QX3 44430355 IC50 = 51 nM T40016 CNB12D 44430370 IC50 = 56.6 nM T40016 CE36SB 44430377 IC50 = 48.9 nM T40016 CTS68I 44430382 IC50 = 36.3 nM T40016 C8BGC1 44430384 IC50 = 45.4 nM T40016 CI8JL5 44430385 IC50 = 43.5 nM T40016 CJ18XT 44430386 IC50 = 31.3 nM T40016 CG8KY9 44430387 IC50 = 22.1 nM T40016 CWR5Z1 44430388 IC50 = 80.3 nM T40016 CBST28 44430389 IC50 = 41.3 nM T40016 CUE9V4 44430390 IC50 = 65.8 nM T40016 C5CB2P 44430391 IC50 = 34.4 nM T40016 CV1DG2 44430392 IC50 = 175.3 nM T40016 C74CQT 44430393 IC50 = 341.6 nM T40016 CV6CM4 44430394 IC50 = 246.5 nM T40016 CEO60C 44430395 IC50 = 56 nM T40016 CVD9H1 44431137 IC50 > 10000 nM T40016 CD64XC 44431139 IC50 > 10000 nM T40016 C20KPU 44431142 IC50 = 1200 nM T40016 C12JEH 44431146 IC50 = 3600 nM T40016 CO4DF3 44431148 IC50 > 10000 nM T40016 C7ZDN6 44431150 IC50 = 1900 nM T40016 C3WSV5 44431167 IC50 = 1300 nM T40016 CXW14R 44431168 IC50 > 2000 nM T40016 CJR34C 44431169 IC50 > 2000 nM T40016 CP6L8E 44431172 IC50 > 2000 nM T40016 CIOW01 44431179 IC50 > 2000 nM T40016 CECG82 44431181 IC50 > 2000 nM T40016 C06NTR 44431183 IC50 > 2000 nM T40016 CQXD51 44431187 IC50 = 490 nM T40016 CLJC40 44431190 IC50 = 120 nM T40016 CL1XK9 44431202 IC50 = 79 nM T40016 C7VGK1 44433485 IC50 < 1000 nM T40016 C3E2QI 44433486 IC50 = 30.2 nM T40016 CK6P9M 44433489 IC50 = 7.586 nM T40016 CV4I9Z 44433491 IC50 = 5.888 nM T40016 C2R5SU 44433492 IC50 = 3.631 nM T40016 C4DFA6 44433500 IC50 = 4.677 nM T40016 C7IYB1 44433501 IC50 = 8.511 nM T40016 CR3OW8 44433502 IC50 = 3.715 nM T40016 C1Z0QH 44433503 EC50 = 1.202 nM T40016 C3SJ5V 44433504 Ki = 387 nM T40016 C2SCP7 44435606 IC50 > 1600 nM T40016 CH5E3L 44435611 IC50 > 1300 nM T40016 CDO62N 44435656 IC50 = 20 nM T40016 C9TP4C 44435662 IC50 = 19 nM T40016 C19TMW 44435663 IC50 = 27 nM T40016 C90WUC 44435667 IC50 = 21 nM T40016 CHFB89 44435668 IC50 = 11 nM T40016 C8IWK2 44435669 IC50 = 8 nM T40016 C8SG5B 44441950 Ki = 10 nM T40016 CWKU75 44441951 Ki = 10 nM T40016 C9EG5T 44441952 Ki = 3 nM T40016 CV0UD9 44441953 Ki = 9 nM T40016 C1OCJ7 44441954 IC50 = 10 nM T40016 CWH06J 44441955 Ki = 20 nM T40016 C9IS3X 44441956 Ki = 56.3 nM T40016 CJQ5G8 44441958 Ki > 3000 nM T40016 CU32PK 44441961 Ki = 59.8 nM T40016 CJ5E0V 44441962 Ki > 3000 nM T40016 C60DXZ 44442904 Ki > 10000 nM T40016 CIM40U 44442905 Ki > 10000 nM T40016 C8PIL1 44442906 Ki > 10000 nM T40016 CB3QN1 44442907 Ki > 10000 nM T40016 CY7UK6 44442908 Ki = 1200 nM T40016 CFX0E8 44442909 Ki > 5000 nM T40016 CV3S1P 44442910 Ki = 3700 nM T40016 C8KDU3 44442911 Ki > 10000 nM T40016 CW8CZ2 44442912 Ki = 1000 nM T40016 CTUE70 44442913 Ki = 4450 nM T40016 CA48OP 44442916 Ki = 3000 nM T40016 CXHK75 44442917 Ki = 1250 nM T40016 CL6ZK2 44442918 Ki = 800 nM T40016 C7YH5D 44442919 Ki = 196 nM T40016 CL7H0E 44442920 Ki = 216 nM T40016 CF7GX1 44442921 Ki = 1300 nM T40016 CMN07E 44442922 Ki > 10000 nM T40016 CJ3L7N 44442923 Ki = 163 nM T40016 CV4L6Z 44442924 Ki = 432 nM T40016 CT3B8Y 44442925 Ki = 193 nM T40016 CEQN26 44442926 Ki = 99 nM T40016 C7ZV0W 44442927 Ki = 4 nM T40016 C9E2QR 44442928 Ki > 10000 nM T40016 CO70RC 44442929 Ki = 55 nM T40016 C96ZLT 44442930 Ki = 1950 nM T40016 CE32IH 44442932 Ki = 2100 nM T40016 CG1VI4 44442933 Ki = 950 nM T40016 CFX2Z6 44442935 Ki = 137 nM T40016 C8JSW1 44442936 Ki = 750 nM T40016 CVQ5K4 44442937 Ki = 113 nM T40016 CIJ9N6 44442938 Ki = 64 nM T40016 CFM0Y1 44442939 IC50 = 3200 nM T40016 C31QCR 44442951 Ki = 76 nM T40016 CQGR94 44442953 Ki = 6 nM T40016 CNBU39 44442955 Ki = 4 nM T40016 C9LT3P 44442957 Ki = 5 nM T40016 C8PE5X 44442960 Ki = 9 nM T40016 C1GL4Z 44442962 Ki = 45 nM T40016 CK4YB1 44442964 Ki = 65 nM T40016 CHC51X 44442967 Ki = 99 nM T40016 CI37JQ 44442979 Ki = 15 nM T40016 C3RUQ9 44442980 Ki = 13 nM T40016 CZL8H0 44442982 Ki = 56 nM T40016 C8S1OM 44442983 Ki = 13 nM T40016 CQX76V 44442984 Ki = 2 nM T40016 COE4T0 44442986 Ki = 9 nM T40016 CY7M3O 44442988 Ki = 10 nM T40016 CMV0G6 44443285 IC50 = 210 nM T40016 CM2JI8 44443286 IC50 = 460 nM T40016 CAS57C 44443287 IC50 = 14000 nM T40016 CQY8H1 44443288 IC50 = 23 nM T40016 C4NQ1C 44443289 IC50 = 82 nM T40016 C0WMP8 44443290 IC50 = 540 nM T40016 CQ0N2S 44443291 IC50 > 10000 nM T40016 CW30DO 44443292 IC50 = 660 nM T40016 CH7B1G 44454500 Ki = 3.8 nM T40016 CDEP04 44454503 Ki = 1.4 nM T40016 CJY2X9 44454504 Ki = 1.2 nM T40016 C94YHC 44454533 Ki = 1 nM T40016 C1YSC6 44454535 Ki = 1.5 nM T40016 C3IW0D 44454537 Ki = 2.3 nM T40016 C9L5XM 44454539 Ki = 1.3 nM T40016 C48ZEN 44454540 Ki = 2.2 nM T40016 C2BQ0E 44454565 Ki = 1.7 nM T40016 CY78VG 44454566 Ki = 1.2 nM T40016 C2LJ6Q 44454567 Ki = 22 nM T40016 C30CHA 44454624 Ki = 2.1 nM T40016 CU7F5L 44454647 Ki = 2.4 nM T40016 CY7NS9 44454672 Ki = 0.8 nM T40016 CAT25W 44454673 Ki > 1000 nM T40016 CEFI01 44454699 Ki = 0.8 nM T40016 C41YOI 44454723 Ki = 0.5 nM T40016 C4ZVS8 44454724 Ki = 0.3 nM T40016 CEI8J6 44454725 Ki = 0.9 nM T40016 C0MG5R 44454751 Ki = 0.8 nM T40016 C49BKG 44454777 Ki = 0.8 nM T40016 C8KXU2 44454778 Ki = 0.5 nM T40016 C6S8ZH 44454802 Ki = 6.7 nM T40016 CC42DA 44454804 Ki = 1 nM T40016 CMB16K 44454805 Ki = 0.9 nM T40016 CE0Y5C 44454806 Ki = 1.6 nM T40016 CCU20Z 44454807 Ki = 8.6 nM T40016 CSV3G4 44454832 Ki = 1.6 nM T40016 CHX6B1 44454869 Ki = 1.1 nM T40016 CB5G1W 44454870 Ki = 3.4 nM T40016 CZ37QB 44454903 Ki = 1.5 nM T40016 CM6LE3 44454906 Ki = 3.7 nM T40016 CCB2O8 44454938 Ki = 9 nM T40016 CKXH14 44454942 Ki = 34 nM T40016 CYG7X4 44473146 IC50 = 0.062 nM T40016 CR5SI0 44476535 EC50 > 10000 nM T40016 C0B2ZT 44515373 IC50 = 0.032 nM T40016 C0MVJ3 44516035 IC50 = 0.051 nM T40016 CM29JD 44516036 IC50 = 1 nM T40016 CKHJ76 44517735 IC50 = 0.3162 nM T40016 CR19IH 44543858 IC50 = 180 nM T40016 C05HEP 44543860 IC50 = 45 nM T40016 C45ZHO 44543969 IC50 = 120 nM T40016 C27TZY 44543970 IC50 = 19 nM T40016 C25OXZ 44544094 IC50 = 370 nM T40016 C7JIF6 44544321 IC50 = 40 nM T40016 C1M4BL 44544711 IC50 = 2.4 nM T40016 CK1Z8P 44545482 IC50 = 43 nM T40016 CF6V4G 44563171 EC50 = 1.995 nM T40016 CSN41Q 44563745 EC50 = 2500 nM T40016 CP6F3O 44563746 EC50 = 33 nM T40016 C46TRW 44563747 EC50 = 1860 nM T40016 C80WGP 44565589 EC50 = 1067.3 nM T40016 CU40ER 44565590 EC50 = 1159.6 nM T40016 CJ39EH 44565614 EC50 = 678.1 nM T40016 C6WO3E 44565615 EC50 = 9.9 nM T40016 CQZ78D 44565616 EC50 = 12.3 nM T40016 CFZD18 44565646 Ki = 5.4 nM T40016 CK8MH3 44565647 Ki = 0.9 nM T40016 CEZ35O 44565648 Ki = 37.8 nM T40016 C6Q5DK 44569945 EC50 = 1.995 nM T40016 C8S3RZ 44570143 EC50 = 25.12 nM T40016 CD65UK 44570182 EC50 = 50.12 nM T40016 C14JOH 44570183 EC50 = 794.33 nM T40016 C06LMN 44570222 EC50 = 3.162 nM T40016 CK10JY 44570223 IC50 = 398.11 nM T40016 CBET53 44570224 EC50 = 251.19 nM T40016 C9TVI8 44570225 EC50 = 25.12 nM T40016 CVO8L1 44570275 EC50 = 50.12 nM T40016 C8BGL6 44585565 IC50 = 1300 nM T40016 C93AMI 44586093 IC50 = 36 nM T40016 CS81IL 44587000 IC50 = 3.6 nM T40016 CUNV59 44587001 IC50 = 2.8 nM T40016 CMN58Z 44587002 IC50 = 2.1 nM T40016 C9RX7K 44587056 IC50 = 21.5 nM T40016 C71CKD 44587057 IC50 = 17.4 nM T40016 C7LU9Z 44587058 IC50 = 2.4 nM T40016 CCJ6Z0 44587059 IC50 = 28.6 nM T40016 C68ZVD 44587197 IC50 = 0.5 nM T40016 CF93RA 44587198 IC50 = 55.1 nM T40016 CIHA86 44587199 IC50 = 352 nM T40016 C68JWV 44587218 IC50 = 12.3 nM T40016 C2USW6 44587219 IC50 = 5.7 nM T40016 CDBQ16 44587220 IC50 = 3.8 nM T40016 CUA45E 44587248 IC50 = 3.5 nM T40016 CC0V2T 44587249 IC50 = 5.8 nM T40016 COU07A 44587250 IC50 = 5.2 nM T40016 C91YAW 44587251 IC50 = 1.3 nM T40016 CJ3VI8 44593465 Ki = 1.3 nM T40016 C70MSI 44593549 EC50 = 158.49 nM T40016 CL8O7P 44769019 IC50 > 6309.57 nM T40016 C9PLK4 45263610 IC50 = 110 nM T40016 C78JKD 45265930 IC50 = 40 nM T40016 C1Z9XI 45267345 IC50 = 1400 nM T40016 CWKP29 45267349 IC50 = 150 nM T40016 CN8HI2 45267356 IC50 > 3000 nM T40016 CG6X9E 45267360 IC50 = 41 nM T40016 CJ10QV 45267605 IC50 = 0.7943 nM T40016 C3KD4Q 45267606 IC50 = 0.3981 nM T40016 CGN7S5 45267615 IC50 = 0.1995 nM T40016 CK04FJ 45267900 IC50 = 460 nM T40016 CPB29I 45268475 IC50 = 31.62 nM T40016 CV7JG9 45268476 IC50 = 25.12 nM T40016 CK0W2Z 45268480 IC50 = 7.943 nM T40016 CF0N2I 45268481 IC50 = 2.512 nM T40016 CF9B0L 45268482 IC50 = 5.012 nM T40016 CQ1F4T 45268485 IC50 = 0.3981 nM T40016 CX7ZG0 45268785 IC50 = 14 nM T40016 CD7T3W 45269091 IC50 = 68 nM T40016 C93BLG 45269348 IC50 = 0.2512 nM T40016 CJTC89 45269354 IC50 = 0.2512 nM T40016 CLSH89 45269632 IC50 = 23 nM T40016 CD61HS 45269633 IC50 = 5.7 nM T40016 CGIT19 45269634 IC50 = 550 nM T40016 C21HYG 45269951 IC50 = 7 nM T40016 CAP56V 45269952 IC50 = 110 nM T40016 CKG49L 45269958 IC50 = 21 nM T40016 C9FK5M 45270463 IC50 = 21 nM T40016 C8ICF3 45270464 IC50 = 480 nM T40016 CIR20D 45270774 IC50 = 20 nM T40016 C9D1IT 45270779 IC50 = 58 nM T40016 C6HZ3T 45271025 IC50 = 0.5012 nM T40016 CS6LO7 45271294 IC50 = 15 nM T40016 CS26QV 45271295 IC50 = 27 nM T40016 C1S8IW 45271296 IC50 = 26 nM T40016 C8GSB6 45271297 IC50 = 840 nM T40016 CJKN81 45271616 IC50 = 132 nM T40016 C08UBE 45272032 IC50 > 10000 nM T40016 C9MF3P 45272514 IC50 = 26 nM T40016 CBEC80 45273046 IC50 = 14 nM T40016 CT52NO 45273047 IC50 = 21 nM T40016 CZXN64 45273048 IC50 = 34 nM T40016 CUZ5C6 45273374 IC50 = 102 nM T40016 C4LK8X 45273665 IC50 = 3.162 nM T40016 CQ81DI 45273670 IC50 = 0.3162 nM T40016 CR8I9S 45486375 Ki = 2 nM T40016 CP35QW 45486376 Ki = 47 nM T40016 C4XDQ1 45486377 Ki = 11 nM T40016 CAT4C2 45486382 Ki = 7 nM T40016 CDA24N 45486383 Ki = 1 nM T40016 C9YM2G 45486384 Ki = 2 nM T40016 CX8HO5 45486385 Ki = 2.6 nM T40016 CJX89Y 45486393 EC50 = 2 nM T40016 C8K2DM 45486403 Ki = 2 nM T40016 CQT1C9 45486404 Ki = 5.2 nM T40016 C0RID5 45486424 Ki = 2.5 nM T40016 C0WQ4R 45486436 Ki = 21 nM T40016 COG73H 45486437 Ki = 2 nM T40016 C2NWO7 45486438 Ki = 2 nM T40016 CM8F4H 45486439 Ki = 9 nM T40016 CD7L1N 45486442 Ki = 8 nM T40016 CW20GE 45486443 Ki = 1 nM T40016 C5HL9V 45486450 Ki = 1.5 nM T40016 CW7J5K 45486451 Ki = 4 nM T40016 CJ6LH2 45486455 EC50 = 1.8 nM T40016 CL91NK 45486456 Ki = 2.5 nM T40016 C6OYN8 45486457 Ki = 1 nM T40016 C3KU7H 45486464 Ki = 3 nM T40016 C14DQK 45486465 Ki = 31 nM T40016 CR6P7Z 45486470 Ki = 3.9 nM T40016 CU3IY5 45486473 Ki = 2 nM T40016 CHRX37 45486474 Ki = 4.3 nM T40016 CY54HC 45486477 Ki = 2 nM T40016 CX8LZ0 45486478 Ki = 7.9 nM T40016 C7PMW0 45486484 Ki = 33 nM T40016 COD9R1 45486485 Ki = 2 nM T40016 CLT46H 45789439 Ki = 18 nM T40016 C1BYW8 46830503 IC50 = 3162.28 nM T40016 C04BWG 46830504 IC50 = 251.19 nM T40016 CY2ZJ0 46830505 IC50 = 3162.28 nM T40016 CC45TP 46830506 IC50 > 10000 nM T40016 CN7Q8A 46830507 IC50 = 398.11 nM T40016 C0QT3G 46830795 IC50 > 2511.89 nM T40016 C0JCX3 46830796 IC50 > 10000 nM T40016 CMS6R9 46830797 IC50 = 1258.93 nM T40016 CJIN74 46830798 IC50 = 3162.28 nM T40016 CRY31M 46830799 IC50 > 10000 nM T40016 CKA07I 46830800 IC50 = 501.19 nM T40016 C4XRF9 46830801 IC50 = 2511.89 nM T40016 C2NC3V 46831087 IC50 = 630.96 nM T40016 CXP6K3 46831397 IC50 = 794.33 nM T40016 C0QNC9 46831400 IC50 = 1258.93 nM T40016 CX6L7Q 46831696 IC50 = 19.95 nM T40016 CQ1IP3 46831697 IC50 = 1995.26 nM T40016 CL1KR4 46831698 IC50 = 31.62 nM T40016 C1DH9W 46831699 IC50 = 39.81 nM T40016 CASV14 46831700 IC50 = 1995.26 nM T40016 CTXY26 46831701 IC50 = 1584.89 nM T40016 CG0J5K 46831956 IC50 = 3162.28 nM T40016 CY3WK4 46831957 IC50 = 1995.26 nM T40016 CP19UN 46831958 IC50 = 15.85 nM T40016 CBJZ85 46831959 IC50 = 50.12 nM T40016 CE4VC8 46831960 IC50 = 251.19 nM T40016 CAR23U 46832233 IC50 = 125.89 nM T40016 CUAO43 46832234 EC50 = 316.23 nM T40016 CM40EP 46832235 IC50 = 15.85 nM T40016 CJ32XT 46832236 IC50 = 25.12 nM T40016 C81GUN 46832237 IC50 = 50.12 nM T40016 CT31AL 46832511 IC50 = 12.59 nM T40016 CR15XE 46832512 IC50 = 39.81 nM T40016 CW12GM 46832513 IC50 = 15.85 nM T40016 C0GTK8 46832514 EC50 = 199.53 nM T40016 C8HO0L 46832515 IC50 = 100 nM T40016 C2S6PL 46834818 IC50 > 10000 nM T40016 C9F5OB 46883794 IC50 = 63.1 nM T40016 C60NSG 46883795 IC50 = 63.1 nM T40016 CHNI89 46883838 IC50 = 158.49 nM T40016 C7KW8T 46883839 IC50 = 199.53 nM T40016 CM7EA1 46883840 IC50 = 199.53 nM T40016 C06JMN 46883842 IC50 = 251.19 nM T40016 CZSG25 46883893 IC50 = 251.19 nM T40016 CQD4K2 46883894 IC50 = 398.11 nM T40016 CMA7J9 46883895 IC50 = 398.11 nM T40016 CBY2M8 46883896 IC50 = 1000 nM T40016 CZDB52 46883897 IC50 > 6309.57 nM T40016 CZI1H6 46883898 IC50 > 6309.57 nM T40016 CV34LD 46883930 IC50 > 6309.57 nM T40016 CJ7TW5 46883931 IC50 > 6309.57 nM T40016 CTE7B2 46883932 IC50 > 6309.57 nM T40016 CAIF17 46883933 IC50 > 6309.57 nM T40016 CA9D4X 46883934 IC50 = 251.19 nM T40016 CXNT91 46883998 IC50 = 251.19 nM T40016 CCH3B0 46883999 IC50 = 251.19 nM T40016 CGSD50 46884000 IC50 = 316.23 nM T40016 C4VKF7 46884001 IC50 = 316.23 nM T40016 CHV9D6 46884030 IC50 = 501.19 nM T40016 CHW0T8 46884031 IC50 = 794.33 nM T40016 C68YXV 46884032 IC50 > 6309.57 nM T40016 CYB42R 46885327 Ki = 51 nM T40016 CA64WN 46885370 Ki = 6.9 nM T40016 C3S2EW 46885371 Ki = 18 nM T40016 CVD89I 46885372 Ki = 4.2 nM T40016 C1NX3S 46885418 Ki = 30 nM T40016 CXQ19B 46885419 Ki = 2465 nM T40016 C2X0TL 46885420 Ki = 3210 nM T40016 C3SB4Y 46885484 Ki = 4109 nM T40016 CNG65D 46888392 IC50 = 10000 nM T40016 C2WQ4M 46888393 IC50 = 2113 nM T40016 CTEY73 46888414 IC50 = 2089 nM T40016 C82NDU 46888415 IC50 = 178 nM T40016 CF97JD 46888416 IC50 = 52 nM T40016 CI4HJ9 46888439 IC50 = 72 nM T40016 CI6Q5G 46888440 IC50 = 99 nM T40016 CAE10V 46888443 IC50 = 30 nM T40016 C1N4WH 46888464 IC50 = 282 nM T40016 C5L7NY 46888465 IC50 = 54 nM T40016 CJK47T 46888466 IC50 = 35 nM T40016 C9QO6J 46888468 IC50 = 14 nM T40016 C6DB3K 46888487 EC50 = 93 nM T40016 C72MUY 46889765 IC50 > 5000 nM T40016 C6DVO1 46889848 IC50 > 10000 nM T40016 CZ90FC 46894119 IC50 > 25000 nM T40016 C3Q7RI 46913890 IC50 > 10000 nM T40016 CP91XE 46914741 IC50 > 10000 nM T40016 CTM2J5 46915203 IC50 > 10000 nM T40016 C75IFZ 46915353 IC50 > 10000 nM T40016 CX70GY 46915355 IC50 > 10000 nM T40016 C7NC4B 46917090 IC50 > 10000 nM T40016 C2LCJ7 46937290 IC50 = 3.3 nM T40016 CKQ8J3 46937431 IC50 = 8 nM T40016 CL7P3N 46938234 IC50 > 9497 nM T40016 CFJT93 46938236 IC50 = 6800 nM T40016 C8P7JH 46938914 IC50 = 860 nM T40016 CY95VK 46938915 IC50 = 690 nM T40016 CVX25Q 46938916 IC50 = 3 nM T40016 C2V5AT 46939019 IC50 = 12 nM T40016 C5R6GI 46939020 IC50 = 8 nM T40016 CF1BX0 46939115 IC50 = 27 nM T40016 C4P0EU 46939116 IC50 = 11 nM T40016 CD6B7X 46939395 IC50 = 1.4 nM T40016 C1KXF2 46939396 IC50 = 1700 nM T40016 CVRU79 46943298 Ki = 2.5 nM T40016 C4Z3NF 49652111 EC50 = 109500 nM T40016 CTG0U1 49652409 EC50 = 109000 nM T40016 CX0NO8 49782554 IC50 < 15848.93 nM T40016 CC7T8Q 49782555 EC50 < 15848.93 nM T40016 CD07EV 49782777 EC50 < 15848.93 nM T40016 C43UKW 49782778 IC50 < 9246.98 nM T40016 C2JTF0 49782779 EC50 < 15848.93 nM T40016 CS7KX9 49782780 EC50 < 15848.93 nM T40016 C36RYU 49782781 IC50 < 13489.63 nM T40016 C8OA0C 49782985 EC50 < 15848.93 nM T40016 C5Y6QU 49782986 IC50 = 3126.08 nM T40016 CB8V7R 49782987 EC50 < 15848.93 nM T40016 CU3S6H 49836028 Ki = 0.7 nM T40016 C96SLW 49851364 Ki = 1.2 nM T40016 C54IGW 49851365 Ki = 18.7 nM T40016 C0G1UO 49851366 Ki = 0.6 nM T40016 CN57XD 49851367 Ki = 20.7 nM T40016 CO5XW9 49851368 Ki = 4.6 nM T40016 CDN4K6 49851369 Ki = 0.4 nM T40016 C0K7OD 49851464 Ki = 0.9 nM T40016 C2JU6O 49851465 Ki = 7.3 nM T40016 CIO2F8 49851466 Ki = 1.1 nM T40016 C4YXN1 49851467 Ki = 0.7 nM T40016 C16OCR 49851468 Ki = 0.4 nM T40016 CI0MX2 49851469 Ki = 2.2 nM T40016 CA4UP7 49851577 Ki = 58.7 nM T40016 CFN03Q 49851580 Ki = 5.7 nM T40016 CUD91T 49862248 EC50 > 10000 nM T40016 CTKV39 49864176 IC50 > 10000 nM T40016 CHT86O 50925620 EC50 = 7300 nM T40016 CCM1T9 50938547 IC50 = 7.943 nM T40016 CZ8J1V 50942115 Ki = 1.7 nM T40016 C23OEF 50942312 EC50 = 12.59 nM T40016 CTHL29 50993207 EC50 = 5600 nM T40016 CH2M5E 50993208 EC50 = 50800 nM T40016 CC54NG 50993209 EC50 = 25300 nM T40016 CM2BI1 50993282 EC50 = 123500 nM T40016 C6DIX2 50993355 EC50 = 101000 nM T40016 CX1KO8 51346768 Ki = 523 nM T40016 C7N9TD 51346823 EC50 = 0.6 nM T40016 C0WDX3 51347001 Ki = 2.9 nM T40016 CF8DK7 51347002 Ki = 9.4 nM T40016 CTH45Q 52918523 IC50 = 0.17 nM T40016 CEC4I7 52941608 IC50 = 23 nM T40016 C6NR7I 52942081 EC50 > 10000 nM T40016 CDV90J 52942528 IC50 = 15.85 nM T40016 CZ1DS4 52943487 EC50 = 130000 nM T40016 C8Y9SU 52944898 IC50 > 1000 nM T40016 CTV7K1 53316621 EC50 = 5.012 nM T40016 CLC5U1 53316851 EC50 = 25.12 nM T40016 C82ATJ 53316852 EC50 = 25.12 nM T40016 C0YNS6 53317029 Ki = 2.3 nM T40016 C0KZW5 53317030 Ki = 2.4 nM T40016 CVNU71 53317031 Ki = 5 nM T40016 CY61KR 53317043 IC50 = 0.1995 nM T40016 C6EZS2 53317044 IC50 = 15.85 nM T40016 CO5GV1 53317045 IC50 = 5.012 nM T40016 CK5UT4 53317489 Ki = 157 nM T40016 CSY4T6 53317533 IC50 = 1.259 nM T40016 CB38MW 53317966 IC50 = 0.1259 nM T40016 C9Y0RM 53318166 EC50 = 10 nM T40016 CCT76B 53318167 EC50 = 12.59 nM T40016 CQ8K1O 53318317 Ki = 38.3 nM T40016 CO7Q4T 53318326 IC50 = 125.89 nM T40016 CQI41V 53318658 Ki = 436 nM T40016 CM0LU1 53318659 Ki = 10 nM T40016 CQBZ97 53318680 EC50 = 15 nM T40016 CAWQ20 53319309 IC50 = 12.59 nM T40016 CC8KA2 53319310 IC50 = 31.62 nM T40016 CPS1C0 53319665 EC50 = 5.7 nM T40016 CVIE23 53319666 Ki = 1.8 nM T40016 CUD48O 53320087 Ki = 6.39 nM T40016 C2CS5A 53320355 Ki = 2.2 nM T40016 C2DM5A 53320607 IC50 = 5.012 nM T40016 C4J1DL 53320608 IC50 = 63.1 nM T40016 C7Z0PN 53320971 IC50 = 3.8 nM T40016 C05MAE 53320972 Ki = 3.5 nM T40016 C58WMJ 53321241 Ki = 3 nM T40016 C5ITY0 53321440 IC50 = 6.31 nM T40016 C0US8P 53321674 IC50 = 7.943 nM T40016 CD2NZ1 53321685 IC50 = 5.7 nM T40016 CB67IZ 53321912 IC50 = 0.07943 nM T40016 CP9FI6 53321913 IC50 = 7.943 nM T40016 C7VWT1 53322135 EC50 = 31.62 nM T40016 C8ZB5U 53322300 EC50 = 0.9 nM T40016 CD2AW1 53322301 Ki = 11.7 nM T40016 CHQ5A9 53322303 Ki = 1.3 nM T40016 CO4ZQ2 53322313 IC50 = 0.2512 nM T40016 C97KUE 53322314 IC50 = 1.995 nM T40016 C63BYE 53322904 IC50 = 19.95 nM T40016 CDL2K7 53323256 IC50 = 3.981 nM T40016 CIQ28P 53323257 IC50 = 50.12 nM T40016 C4MJ9W 53323258 IC50 = 5.012 nM T40016 C4X3VU 53323259 IC50 = 1.995 nM T40016 CJD29K 53323475 EC50 = 3.981 nM T40016 CD0N1K 53323476 EC50 = 1000 nM T40016 CQ41DA 53323656 Ki = 9 nM T40016 C4I3OP 53323657 Ki = 0.9 nM T40016 CH8LW2 53323658 Ki = 106 nM T40016 CKRC57 53323670 IC50 = 0.3162 nM T40016 C9G2SP 53323671 IC50 = 5.012 nM T40016 CBM23P 53323672 IC50 = 50.12 nM T40016 C7K9RF 53323962 EC50 = 5.1 nM T40016 C4WC2R 53324599 IC50 = 7.943 nM T40016 C8EM1C 53324945 Ki = 3.1 nM T40016 CH2U4P 53324954 IC50 = 125.89 nM T40016 C16TGD 53325224 Ki = 416 nM T40016 CK2BN3 53325565 Ki = 10.4 nM T40016 CIU8H2 53325583 EC50 = 12.59 nM T40016 CLG69E 53325612 EC50 = 1.995 nM T40016 CYH3V0 53325642 Ki = 50.2 nM T40016 CP7Y9M 53326069 EC50 = 6.31 nM T40016 C7Q8CZ 53326228 EC50 = 0.4 nM T40016 CPFW50 53326229 EC50 = 0.2 nM T40016 C02REC 53326230 Ki = 19.6 nM T40016 C1Z0MJ 53326231 Ki = 8 nM T40016 C79XKL 53326232 Ki = 1 nM T40016 CXJ84N 53326233 Ki = 157 nM T40016 C68EWU 53326245 IC50 = 39.81 nM T40016 CTX3I2 53326246 IC50 = 3.162 nM T40016 CGX19M 53326247 IC50 = 794.33 nM T40016 C9HN7W 53326537 Ki = 132 nM T40016 CB71TJ 53326538 Ki = 12.2 nM T40016 C82DYI 53326614 Ki > 4290 nM T40016 C6K2OB 53328064 Ki = 0.66 nM T40016 CJCP75 53359074 Ki = 1.64 nM T40016 C9H5YE 53361128 EC50 > 10000 nM T40016 C9XT0F 53483966 EC50 = 2.97 nM T40016 CUR24K 53875787 IC50 = 340 nM T40016 C30XLO 54592009 IC50 = 597 nM T40016 CCJ42Y 56589543 IC50 = 3540 nM T40016 CW9OS3 56593697 Ki = 49.5 nM T40016 CU02PM 56593698 Ki = 1.2 nM T40016 CUX1B9 56593851 Ki = 3.8 nM T40016 CJ98FM 56593852 Ki = 4 nM T40016 CN0Q8R 56593853 Ki = 2.9 nM T40016 CEN7V4 56593854 Ki = 3.9 nM T40016 C1YGH6 56593980 Ki = 6 nM T40016 CV0JW2 56593981 Ki = 2.5 nM T40016 C8G0AR 56593982 Ki = 9.17 nM T40016 C47DRS 56593983 Ki = 5.48 nM T40016 C9W5DZ 56593984 Ki = 1.74 nM T40016 CV9OE8 56594117 Ki = 486 nM T40016 CA9ER8 56594118 Ki = 1.6 nM T40016 CXQ2R5 56594120 Ki = 1.3 nM T40016 C7ULR4 56594121 Ki = 1.68 nM T40016 C6ZR3U 56594268 Ki = 2.6 nM T40016 CKB34M 56594269 Ki = 2.7 nM T40016 C4P7JM 56594270 Ki = 1.96 nM T40016 CNOI17 56594271 Ki = 2.53 nM T40016 C42NTL 56594272 Ki = 3.08 nM T40016 CO0CR2 56594389 Ki = 8.6 nM T40016 CY0ZX3 56594392 Ki = 4.1 nM T40016 C7UVE6 56594518 Ki = 4.2 nM T40016 CH0M6A 56594523 Ki = 15.4 nM T40016 CR4U9K 56594613 IC50 = 4960 nM T40016 CV39IP 56595706 Ki = 7.1 nM T40016 CTSJ36 56595707 Ki = 10.5 nM T40016 C7KU1Y 56595708 Ki = 24 nM T40016 CEY96L 56595709 Ki = 2.5 nM T40016 CI1UN4 56661440 EC50 = 0.43 nM T40016 C1L0FO 56664884 EC50 = 0.38 nM T40016 CU5C3L 56668302 EC50 = 8.78 nM T40016 CI2E4M 56671781 EC50 = 0.71 nM T40016 CX5LM7 56671782 EC50 = 3.93 nM T40016 C4F7OS 56671783 EC50 = 7.35 nM T40016 CKHZ50 56675193 EC50 = 1.87 nM T40016 CUM21Y 56677234 Ki = 2.9 nM T40016 CBG79E 56681836 EC50 = 0.78 nM T40016 CR3P4L 56681837 EC50 = 1.75 nM T40016 CR4IK7 56681838 EC50 = 2.82 nM T40016 CF3G2M 56925477 IC50 = 3500 nM T40016 CZ7O8G 56925478 IC50 = 950 nM T40016 CW87RG 56925573 IC50 > 10000 nM T40016 C30DAL 56925669 IC50 = 5500 nM T40016 CQHA65 56925670 IC50 > 10000 nM T40016 CJP31U 56925671 IC50 > 10000 nM T40016 CI3S6F 56925790 IC50 > 10000 nM T40016 CTY1Q9 56925791 IC50 = 6900 nM T40016 CTG9I7 56926011 IC50 = 200 nM T40016 CL16UQ 56949326 IC50 < 10000 nM T40016 CX6Q9M 57390301 Ki = 1.6 nM T40016 CR3Y4C 57390331 IC50 = 1.4 nM T40016 C2PAW0 57390332 IC50 = 14.3 nM T40016 C26UES 57390369 EC50 = 22.4 nM T40016 C3Y9SF 57390753 IC50 = 61 nM T40016 C7R4HE 57390754 IC50 = 60 nM T40016 CM0SG2 57390990 IC50 = 87 nM T40016 CD1KG0 57391329 IC50 = 17.6 nM T40016 C1ETU3 57391330 IC50 = 23.5 nM T40016 C5Q0AF 57392164 IC50 = 2.1 nM T40016 C4SD8X 57392560 IC50 = 13 nM T40016 CU8AN3 57392780 IC50 = 88 nM T40016 CX12JM 57392781 IC50 = 3 nM T40016 C9OMW1 57392782 IC50 = 405 nM T40016 C6YQU8 57393091 IC50 = 17.2 nM T40016 C8BPN6 57393863 IC50 = 2.85 nM T40016 CS50GQ 57393864 IC50 = 9.7 nM T40016 C8S0HJ 57394288 IC50 = 23 nM T40016 C30JOV 57394501 IC50 = 7 nM T40016 C76QKN 57394818 IC50 = 70.2 nM T40016 CY6H7M 57394819 IC50 = 118 nM T40016 C8N0BF 57394833 IC50 = 722 nM T40016 CF8H1A 57394834 IC50 = 5.1 nM T40016 CDJ67U 57395566 Ki = 1 nM T40016 CW5V3Q 57395588 IC50 = 3.8 nM T40016 CM5UX2 57395589 IC50 = 2.2 nM T40016 CST3E8 57395590 IC50 = 2 nM T40016 C6J4SB 57395657 EC50 = 17.3 nM T40016 CINU04 57396254 IC50 = 8 nM T40016 C1O6JU 57396255 IC50 = 2 nM T40016 CSUH91 57396585 IC50 = 41.3 nM T40016 CSRF70 57396586 IC50 = 305 nM T40016 C4BV3D 57396601 IC50 = 5.8 nM T40016 CG9A3H 57396602 IC50 = 4.4 nM T40016 CU4M9T 57396603 IC50 = 1.69 nM T40016 CA49PX 57398362 IC50 = 57.2 nM T40016 CS2MU7 57398378 IC50 = 46.5 nM T40016 CELN93 57398379 IC50 = 37.9 nM T40016 C24YLG 57399054 Ki = 2.4 nM T40016 C0CNX7 57399075 IC50 = 15.9 nM T40016 C54BJR 57399499 IC50 = 142 nM T40016 CVOB64 57399718 IC50 = 6 nM T40016 CT7X2V 57400021 IC50 = 68.7 nM T40016 C4B8RP 57400033 IC50 = 69.3 nM T40016 C0FA2Q 57400034 IC50 = 6 nM T40016 CACH70 57400817 EC50 = 535 nM T40016 CM29BO 57400818 IC50 = 1.9 nM T40016 CY7IE5 57400819 IC50 = 18 nM T40016 CG9KZ2 57400871 EC50 = 14.1 nM T40016 CF83VM 57401459 Ki = 1.94 nM T40016 CJ4LR2 57401460 Ki = 15.7 nM T40016 C7W3YD 57401479 IC50 = 39 nM T40016 C4GIL8 57401833 IC50 = 11.4 nM T40016 C84EUP 57402578 EC50 = 50 nM T40016 CQB6W2 57402579 IC50 = 3.7 nM T40016 C6RX7O 57403004 IC50 = 45 nM T40016 C6IPK0 57403199 Ki = 0.67 nM T40016 CR6L7E 57403222 IC50 = 49 nM T40016 CG2J6D 57403536 IC50 = 7.3 nM T40016 C81TNW 57403537 IC50 = 13.5 nM T40016 C86WRQ 57403538 IC50 = 43.8 nM T40016 CDP21S 57403554 IC50 = 36 nM T40016 C7NX0F 57432086 IC50 = 13.4 nM T40016 CLP69J 57432087 IC50 = 17 nM T40016 CPU6W7 57473898 IC50 = 35 nM T40016 CEJ25K 57473899 IC50 = 10 nM T40016 CUJ08D 57474008 IC50 = 10 nM T40016 C2U1GQ 57524309 IC50 = 125 nM T40016 C3NHX4 57651527 IC50 = 97 nM T40016 CR2J4D 57651532 IC50 = 1600 nM T40016 CW1XC2 57651533 IC50 = 23 nM T40016 C0MTP4 57651538 IC50 = 75 nM T40016 CJ1B4P 57651564 IC50 = 18 nM T40016 CBY05F 57651578 IC50 = 80 nM T40016 C7P3UH 57651588 IC50 = 240 nM T40016 C2QG9T 57651604 IC50 = 42 nM T40016 CJD46O 57651617 IC50 = 410 nM T40016 CSV5U6 57651649 IC50 = 160 nM T40016 CD74EG 57651658 IC50 = 220 nM T40016 COUM81 57666295 Ki = 2.6 nM T40016 CO02KN 57666296 Ki = 4.1 nM T40016 C9Y5ZN 57666298 Ki = 4.6 nM T40016 CQF1I7 57666299 Ki = 1.7 nM T40016 CKS5N7 57666309 Ki = 4.4 nM T40016 C3WG0L 57666312 Ki = 0.5 nM T40016 CB4Y7X 57666322 Ki = 2.4 nM T40016 CS5W9Q 57666329 IC50 = 2.3 nM T40016 CK1PB7 57666331 Ki = 15 nM T40016 C2WL8X 57666350 IC50 = 0.4 nM T40016 CR0F3Y 57666355 IC50 = 0.1 nM T40016 CBDI87 57666363 Ki = 3.1 nM T40016 CBMZ45 57666378 Ki = 2.7 nM T40016 C43GDR 57666397 IC50 = 1.1 nM T40016 CNX5C4 57666415 Ki = 1.9 nM T40016 CZX0O6 57690890 IC50 = 6.9 nM T40016 CN6Q0O 57690891 IC50 = 28 nM T40016 CTM6K5 57690900 IC50 = 7.2 nM T40016 CV0WT1 57690902 IC50 = 3.8 nM T40016 CHDO84 57690904 IC50 = 8.8 nM T40016 C6PKR9 57690906 IC50 = 2 nM T40016 CD5T6X 57690907 IC50 = 4.1 nM T40016 CH45LN 57736637 Ki > 100 nM T40016 C1KZT3 57906156 IC50 > 10000 nM T40016 C3IN9F 57983276 IC50 > 10000 nM T40016 CJ6Y1B 58026134 IC50 = 27 nM T40016 CV1RX3 58026153 IC50 = 28 nM T40016 C19XQV 58026164 IC50 = 2 nM T40016 CR7H3O 58026170 IC50 = 140 nM T40016 C7XL3D 58026176 IC50 = 19 nM T40016 C8S3EQ 58064714 IC50 = 2770 nM T40016 CL42XF 58064726 IC50 = 4800 nM T40016 CPL9A6 58064729 IC50 > 10000 nM T40016 CA0SH5 58064735 IC50 > 10000 nM T40016 C47AUR 58392644 Ki = 0.76 nM T40016 CLU6V4 58392650 Ki = 0.57 nM T40016 CV6G4D 58392653 EC50 = 248 nM T40016 C9CQS0 58392665 Ki = 0.66 nM T40016 CTMC05 58392676 Ki = 0.39 nM T40016 CXF39M 58392685 Ki = 4.8 nM T40016 C9FK1W 58392705 EC50 = 63.9 nM T40016 CSE2H6 58392714 Ki = 0.52 nM T40016 C7FXH3 58392721 Ki = 1.1 nM T40016 C9IAL0 58392730 Ki = 0.71 nM T40016 CBY7Q3 58392757 Ki = 0.57 nM T40016 CWX3L0 58392759 EC50 = 1.3 nM T40016 CJDN90 58392790 Ki = 0.62 nM T40016 CC5L9W 58392802 Ki = 9.8 nM T40016 CO59DQ 58392803 EC50 = 45 nM T40016 CD9V7K 58392806 EC50 = 54.9 nM T40016 C0AZ1T 58392807 Ki = 0.66 nM T40016 CE5S4N 58392813 EC50 = 15.2 nM T40016 C1U8YQ 58392816 Ki = 0.66 nM T40016 CJH51L 58392825 Ki = 1.9 nM T40016 C4C2FT 58599563 IC50 = 7 nM T40016 CWAD17 58731166 Ki <= 500 nM T40016 CI7XQ5 58731245 Ki <= 500 nM T40016 CI6XF5 58742295 IC50 = 0.6 nM T40016 CVGS24 58742335 IC50 = 100 nM T40016 CNW46Q 58742348 IC50 = 211 nM T40016 CUAY18 58742377 IC50 = 22 nM T40016 C4I8UG 58742381 IC50 = 38 nM T40016 CRYK21 58742385 IC50 = 0.79 nM T40016 C0JL7A 58973277 IC50 = 1.15 nM T40016 CV8B1K 59233333 Ki = 69 nM T40016 CN3YR2 59233334 Ki = 35 nM T40016 CY38HG 59233337 Ki = 35 nM T40016 CUX4E7 59233347 Ki = 46 nM T40016 CO63VJ 59233364 Ki = 53 nM T40016 CW3Z2B 59251049 EC50 = 977 nM T40016 C3VD2R 59251055 Ki = 1.51 nM T40016 C14FAP 59251075 Ki = 2 nM T40016 CTZ10A 59251088 Ki = 1.9 nM T40016 C2A9JO 59251119 Ki = 0.81 nM T40016 CHM67D 59251186 Ki = 1.15 nM T40016 C14OUW 59252742 Ki = 7.2 nM T40016 CN4J2B 59252759 Ki = 21 nM T40016 CL91EP 59252761 Ki = 8.1 nM T40016 CZW0C6 59252766 Ki = 36 nM T40016 COH4C0 59252776 Ki = 47 nM T40016 CE9PF6 59252796 Ki = 21 nM T40016 C0WL5E 59252800 Ki = 9.8 nM T40016 CR24NL 59252804 Ki = 19 nM T40016 CR3D9I 59252811 Ki = 46 nM T40016 CV49FS 59252819 Ki = 8.8 nM T40016 C1IOL3 59252821 Ki = 7.5 nM T40016 C5F8SX 59252827 Ki = 1.9 nM T40016 CVT75O 59252830 Ki = 29 nM T40016 C4EV6L 59252842 Ki = 84 nM T40016 CWUE23 59252846 Ki = 7 nM T40016 CA3W0U 59252850 Ki = 1.1 nM T40016 C9F3JN 59252853 Ki = 14 nM T40016 C5B9WH 59252854 Ki = 12 nM T40016 C4K3RM 59252869 Ki = 10 nM T40016 CTM0O8 59252882 Ki = 13 nM T40016 C1VDO0 59266722 IC50 = 1.1 nM T40016 CN6CO4 59272917 IC50 = 0.21 nM T40016 C10MEG 59272918 IC50 = 0.92 nM T40016 CM2L1N 59272923 IC50 = 0.19 nM T40016 CIDC27 59339621 IC50 = 0.04 nM T40016 CQF0V6 59339664 IC50 = 0.02 nM T40016 CF0CQ2 59339738 IC50 = 0.09 nM T40016 CORQ09 59339810 IC50 = 0.029 nM T40016 CC3QG0 59419621 Ki = 18 nM T40016 C4NHO7 59419641 Ki = 5 nM T40016 CYZI85 59556974 IC50 > 10000 nM T40016 C5DU8H 59612841 Ki < 1 nM T40016 CMR3W0 59769897 Ki > 100 nM T40016 C5C3AO 59770003 Ki = 0.226 nM T40016 C9CF2N 59770543 Ki > 100 nM T40016 CI8JB6 59786564 IC50 = 44 nM T40016 C1OE0C 59786572 IC50 = 2.8 nM T40016 COM20D 59786577 IC50 = 100 nM T40016 CH3QT2 59786587 IC50 = 6.6 nM T40016 C2TNO8 60026286 IC50 = 560 nM T40016 CZE5J8 60026377 IC50 = 8 nM T40016 CJ34GW 60026481 IC50 = 59 nM T40016 CJ7E6C 60026483 IC50 = 2 nM T40016 C0LDS2 60026592 IC50 = 11 nM T40016 C31PTC 60026641 IC50 = 9 nM T40016 C67NSE 60026675 IC50 = 13 nM T40016 C6GP5R 60026731 IC50 = 5 nM T40016 C5M8HV 60026772 IC50 = 5 nM T40016 CI36XS 60026787 IC50 = 2 nM T40016 C3JD8M 60026802 IC50 = 14 nM T40016 CE9MI4 60026817 IC50 = 5 nM T40016 C3UQ8M 60026849 IC50 = 7 nM T40016 C04EKW 60026878 IC50 = 18 nM T40016 CM3Y0X 60026895 IC50 = 22 nM T40016 CH5CQ7 60202645 Ki = 4 nM T40016 CIX6M8 66549685 Ki = 19 nM T40016 C5TKZ8 66549686 Ki = 7 nM T40016 C7T5RU 66549878 Ki = 5 nM T40016 C9YN2F 66549879 Ki = 11 nM T40016 C3WQ9J 66549880 Ki = 11 nM T40016 C7DF3G 66549881 Ki = 8 nM T40016 C64VNT 66549882 Ki = 3 nM T40016 C4WER8 66549883 Ki = 557 nM T40016 C69DEI 66550094 Ki = 22 nM T40016 COY2Q0 66550095 Ki = 400 nM T40016 C3THV1 66550096 Ki = 24 nM T40016 C4KM3Y 66550097 Ki = 18 nM T40016 CNDC81 66550098 Ki = 49 nM T40016 CR8X7I 66550099 Ki > 50 nM T40016 CE3QS0 66550320 Ki = 139 nM T40016 C5RMY8 66550321 Ki = 188 nM T40016 CB0VD7 66550322 Ki = 21 nM T40016 CT90BP 66550324 Ki = 8 nM T40016 CSU9T5 66550325 Ki = 28 nM T40016 CJKH71 66550524 Ki = 9 nM T40016 CZ47TU 66550726 Ki = 19 nM T40016 CIN7W5 66550727 Ki = 9 nM T40016 CH7JS8 66550729 Ki = 16 nM T40016 C1CXY9 66996546 IC50 > 10000 nM T40016 CH39DP 67053383 IC50 = 70 nM T40016 C3LF8O 67053425 IC50 = 100 nM T40016 CU5C7T 68327007 Ki > 50 nM T40016 C4UC3D 68833523 IC50 = 0.3 nM T40016 C35MCV 69075970 IC50 = 1800 nM T40016 CNQ8T5 69571559 IC50 = 10 nM T40016 CP7ME8 70681366 IC50 = 5.57 nM T40016 C28NIR 70681401 IC50 = 101 nM T40016 CO2V3L 70681433 IC50 = 29.2 nM T40016 CQ0Z1H 70682700 IC50 = 1642 nM T40016 CEK7F6 70683461 IC50 = 0.63 nM T40016 C5YF1S 70683462 IC50 = 1.5 nM T40016 C0Y7VR 70683502 IC50 = 400 nM T40016 CK8H0A 70683527 IC50 = 0.32 nM T40016 C1V8BT 70683528 IC50 = 0.6 nM T40016 CLCX98 70684785 IC50 = 235 nM T40016 CARO49 70685018 Ki = 0.17 nM T40016 CJIF98 70685568 IC50 = 6.6 nM T40016 CV6S0D 70685569 IC50 = 3.12 nM T40016 C9A4VY 70685580 IC50 = 3.43 nM T40016 CK3U2R 70685600 IC50 = 2.1 nM T40016 C0A5RP 70685628 IC50 = 0.5 nM T40016 CT08DF 70685651 IC50 = 22.1 nM T40016 CJ31YF 70687711 IC50 = 4.4 nM T40016 CZLJ82 70687712 IC50 = 7.3 nM T40016 CCR59B 70687725 IC50 = 7.5 nM T40016 C65IRX 70687751 IC50 = 107 nM T40016 C2DIO4 70687776 IC50 = 1.8 nM T40016 C3K1FC 70687805 IC50 = 4.3 nM T40016 CSZA04 70687806 IC50 = 6.6 nM T40016 C8BEI2 70687807 IC50 = 14.9 nM T40016 C0AEY1 70689007 IC50 > 10000 nM T40016 C6QW5H 70689008 IC50 = 46 nM T40016 C2HP8J 70689009 IC50 = 801 nM T40016 C52VZQ 70689010 IC50 = 1278 nM T40016 C1GCA5 70689011 IC50 = 1601 nM T40016 CD29ZL 70689757 IC50 = 14.8 nM T40016 CA2Z5T 70689778 IC50 = 44.7 nM T40016 CKJ64D 70689802 IC50 = 86.4 nM T40016 C4JUQ2 70689803 IC50 = 88.7 nM T40016 CZ8XA6 70689821 IC50 = 18.3 nM T40016 C2X4VH 70689840 IC50 = 4.7 nM T40016 CH74ZQ 70689841 IC50 = 127 nM T40016 CWR1T7 70691113 IC50 = 1910 nM T40016 CE41BJ 70691114 IC50 = 722 nM T40016 CWK43T 70691115 IC50 = 96 nM T40016 CM1WP7 70691918 IC50 = 28.8 nM T40016 CA2U1S 70691919 IC50 = 3.7 nM T40016 C4NC7P 70691920 IC50 = 2.8 nM T40016 CSRB01 70691940 IC50 = 179 nM T40016 CT45PM 70691941 IC50 = 2.9 nM T40016 C8MHT9 70691942 IC50 = 30.5 nM T40016 CD19KG 70691967 IC50 = 1.99 nM T40016 CPH9W3 70691968 IC50 = 1.6 nM T40016 CT7KY2 70691995 IC50 = 26.7 nM T40016 C7PKB1 70691996 IC50 = 27.2 nM T40016 C32MBT 70693235 IC50 = 820 nM T40016 CXI23M 70693236 IC50 = 4.6 nM T40016 CX0IR5 70693237 IC50 = 1256 nM T40016 CE02OB 70693238 IC50 = 298 nM T40016 CLE0R8 70693239 IC50 = 111 nM T40016 CXA43E 70693965 IC50 = 4.7 nM T40016 CYO30E 70693966 IC50 = 0.89 nM T40016 CE60JR 70693992 IC50 = 1.06 nM T40016 CF4D9M 70694011 IC50 = 1.89 nM T40016 C6ZK1Y 70695317 IC50 = 1423 nM T40016 C9SPT1 70696092 IC50 = 12.4 nM T40016 CI4EG2 70696161 IC50 = 8.9 nM T40016 CE7P8B 70696162 IC50 = 61.3 nM T40016 CBJ0D6 70697330 IC50 > 9000 nM T40016 CGLJ86 70697331 IC50 = 1200 nM T40016 C9QTP1 70697332 IC50 = 4.5 nM T40016 C5QPC0 70697572 Ki = 0.21 nM T40016 CUH71V 71239417 IC50 > 1000 nM T40016 C95CVQ 71245268 Ki = 0.67 nM T40016 C9GC3P 71245282 Ki = 0.52 nM T40016 CM90EO 71245304 Ki = 0.52 nM T40016 CV1QJ5 71245432 Ki = 0.71 nM T40016 C1W0KS 71245462 Ki = 0.57 nM T40016 CP0C6L 71245590 Ki = 0.52 nM T40016 C0NWE2 71451108 Ki = 155 nM T40016 C94FCP 71452686 IC50 = 2300 nM T40016 C8OT4U 71452929 Ki < 1 nM T40016 C0BFS4 71452930 Ki = 58 nM T40016 CLRN15 71452931 Ki > 400 nM T40016 CF7G5Q 71454032 Ki = 98 nM T40016 C35HYI 71456433 Ki = 2 nM T40016 CLM4X2 71456434 Ki = 3 nM T40016 CF08ME 71457470 Ki = 669 nM T40016 C15EYZ 71457556 Ki > 1500 nM T40016 CJR7C5 71460130 Ki = 15 nM T40016 C39VNO 71460131 Ki = 1 nM T40016 CUZQ62 71460135 Ki > 400 nM T40016 CEO5G4 71461616 IC50 = 2800 nM T40016 CHEM26 71461848 Ki = 40 nM T40016 C1MHC0 71467246 IC50 = 6900 nM T40016 C4B0IC 71467248 IC50 = 5800 nM T40016 CVB70W 71508604 EC50 = 2090 nM T40016 CGS13D 71508641 EC50 = 1440 nM T40016 CG6ZR3 71508642 EC50 > 10000 nM T40016 C82UIW 71508688 EC50 = 90 nM T40016 CQCD26 71508715 EC50 = 1500 nM T40016 C13ALQ 71508716 EC50 > 10000 nM T40016 CT52JE 71508749 EC50 > 10000 nM T40016 CV0F5Y 71508789 EC50 = 2810 nM T40016 COI72X 71508790 EC50 = 550 nM T40016 C9XHS2 71508832 EC50 = 690 nM T40016 C92GOZ 71508833 EC50 = 350 nM T40016 CYW34A 71519686 IC50 = 3400 nM T40016 CGK4S8 71543393 Ki > 6020 nM T40016 C83YJF 71544946 IC50 > 5000 nM T40016 CT9Y5D 71549558 IC50 = 3800 nM T40016 C8ZX0F 71549573 IC50 = 11000 nM T40016 CZ8Y7O 71549829 IC50 = 4900 nM T40016 CPFL57 71549843 EC50 > 20000 nM T40016 CY8SP0 71549969 IC50 = 17000 nM T40016 CX6JR5 71550242 IC50 = 3100 nM T40016 C6WIA2 71550244 IC50 = 3000 nM T40016 CSHT69 71550657 IC50 > 5000 nM T40016 C1JP3D 71712294 Ki = 0.7 nM T40016 C0B6GE 71716762 EC50 > 10000 nM T40016 CRDK79 71717362 EC50 = 6200 nM T40016 C5NU0T 71721539 IC50 = 32500 nM T40016 CP5KM8 72163477 IC50 > 10000 nM T40016 CA6O4K 72163478 IC50 > 10000 nM T40016 C27XWS 72163479 IC50 = 4700 nM T40016 C6M9CN 72163480 IC50 = 3800 nM T40016 CL8AH4 72163481 IC50 > 10000 nM T40016 CB2SD9 72163621 IC50 = 2000 nM T40016 CU6NA8 72163622 IC50 = 2100 nM T40016 CTEV75 72163623 IC50 = 1600 nM T40016 CER73F 72163624 IC50 = 2200 nM T40016 CC8VM7 72163625 IC50 > 10000 nM T40016 CS69AC 72163626 IC50 = 9100 nM T40016 CAJ0H5 72163627 IC50 = 4900 nM T40016 C1D3EU 72163754 IC50 = 5000 nM T40016 C1G3ES 72163755 IC50 = 1100 nM T40016 C92WND 72188913 Ki = 13 nM T40016 CP8AC2 72188914 EC50 = 2.4 nM T40016 CA6FO5 72188915 Ki = 6.7 nM T40016 C0IZU8 72188916 EC50 = 0.5 nM T40016 C8UT9I 72188920 Ki = 15 nM T40016 CMKD06 72188921 Ki = 85 nM T40016 C85XAF 72189208 Ki = 7.9 nM T40016 C8ETZ0 72189209 Ki = 4 nM T40016 C1ERA6 72192163 Ki = 0.16 nM T40016 C8IUW4 72192289 Ki = 2.7 nM T40016 CG7D0N 72192290 Ki = 0.9 nM T40016 C34FBN 72544603 IC50 = 2195 nM T40016 CJ62YO 72547740 Ki = 0.12 nM T40016 C4K8DR 72547975 Ki = 0.22 nM T40016 CPA19X 72548209 Ki = 0.83 nM T40016 CN48HM 72548212 Ki = 0.23 nM T40016 C7IA0J 72548214 Ki = 0.14 nM T40016 CJ34IN 72548216 Ki = 0.14 nM T40016 CBF76T 72548443 Ki = 0.16 nM T40016 CELT72 72548445 Ki = 0.17 nM T40016 C8F9MA 72548670 Ki = 0.41 nM T40016 CY9HV3 72548678 Ki = 0.21 nM T40016 CO1PV2 72548922 Ki = 0.13 nM T40016 CV4G5E 72548925 Ki = 0.21 nM T40016 CX7CM5 72549154 Ki = 0.14 nM T40016 CZBE28 72549155 Ki = 0.25 nM T40016 C8JTK6 72549156 Ki = 0.19 nM T40016 CG06BL 72549381 Ki = 28 nM T40016 C1XGF0 72549624 Ki = 0.22 nM T40016 CSC10N 72549625 Ki = 0.73 nM T40016 CN3W7R 72549852 Ki = 10 nM T40016 COFJ20 72549853 Ki = 69 nM T40016 CT0RY5 72550282 Ki = 0.1 nM T40016 CJ48YS 72550284 Ki = 0.21 nM T40016 C6S3FW 72550951 Ki = 0.14 nM T40016 C1C6SR 72551176 Ki = 0.14 nM T40016 CLA3Y9 72710581 Ki = 0.268 nM T40016 CXB45U 72724690 IC50 = 2 nM T40016 CI2K6C 72725442 IC50 = 83 nM T40016 C0W2UD 72725443 IC50 = 23 nM T40016 CQ5D1B 72725444 IC50 = 230 nM T40016 C2PJV7 72725445 IC50 = 110 nM T40016 CQ4Z2C 72725446 IC50 = 10 nM T40016 C47IMQ 72725447 IC50 = 160 nM T40016 CJSK52 72725491 IC50 = 11 nM T40016 CS6J4T 72725492 IC50 = 48 nM T40016 C41FYD 72725493 IC50 = 10 nM T40016 CUG96L 72725494 IC50 = 10 nM T40016 CFHJ16 72725495 IC50 = 78 nM T40016 CW7IY3 72725496 IC50 = 62 nM T40016 CSV1I7 72725497 IC50 = 15 nM T40016 COV09R 72725548 IC50 = 25 nM T40016 CTE01I 72725549 IC50 = 250 nM T40016 C09ZFS 72725550 IC50 = 89 nM T40016 C2Z7QT 72725551 IC50 = 3 nM T40016 C0K2CP 72725552 IC50 = 120 nM T40016 C37MEN 72725553 IC50 = 27 nM T40016 CYSM01 72725554 IC50 = 23 nM T40016 C3POU0 72736045 EC50 = 0.1 nM T40016 CFQK42 73051162 Ki = 0.14 nM T40016 CL3MJ4 73051163 Ki = 0.08 nM T40016 C45NKJ 73051309 Ki = 0.2 nM T40016 CZ2AM8 73051786 Ki = 0.23 nM T40016 CN7CI1 73346216 Ki = 1.42 nM T40016 CPQY04 73346217 Ki = 2.4 nM T40016 CYU73F 73346218 Ki = 285 nM T40016 CW93GP 73346219 Ki = 196 nM T40016 C3A9QB 73346225 Ki = 11 nM T40016 CCJ4V5 73349253 EC50 = 0.66 nM T40016 C0MTX8 73350834 Ki = 2.3 nM T40016 CW0Q8A 73350835 Ki = 3.6 nM T40016 C9LSH7 73350845 Ki = 17 nM T40016 C5YC4W 73352322 Ki = 0.93 nM T40016 CI16HS 73353799 Ki = 17 nM T40016 C2X6KY 73355320 Ki = 0.87 nM T40016 C02PXY 73356866 Ki = 1.3 nM T40016 COU49R 76314656 IC50 = 5 nM T40016 C95NBT 76314657 IC50 = 21 nM T40016 CD7TQ2 76314998 IC50 = 260 nM T40016 CZ08OF 76317198 IC50 = 120 nM T40016 CR5B2V 76317199 IC50 = 15 nM T40016 C5YFZ6 76318225 IC50 = 11 nM T40016 CS25MH 76318649 IC50 = 62 nM T40016 CG3HM7 76321650 Ki > 100 nM T40016 C0RK5D 76321918 IC50 = 13 nM T40016 C7GI5W 76328818 Ki > 100 nM T40016 C3IC5B 76329113 IC50 = 840 nM T40016 C1RB6X 76329114 IC50 = 9 nM T40016 C8NUF6 76329495 IC50 = 270 nM T40016 CP8M1Z 76332766 IC50 = 5 nM T40016 CKDI18 76332767 IC50 = 8 nM T40016 CW35KY 76336757 IC50 = 17 nM T40016 CK21EY 77461202 IC50 = 2 nM T40016 CIU65X 86280440 Ki = 1.22 nM T40016 CZLU45 86710000 Ki = 0.48 nM T40016 CJ6Q7K 86710002 Ki = 4.6 nM T40016 CT50AL 87539277 IC50 = 39.81 nM T40016 CAVY94 87591264 IC50 = 2.1 nM T40016 CY05IC 87733533 IC50 = 3.981 nM T40016 CBH60W 89400603 Ki = 0.52 nM T40016 C9EH7I 89500376 Ki = 2390 nM T40016 C0EQS7 89501406 Ki > 3120 nM T40016 C8JG7O 89510193 Ki = 462 nM T40016 C0VB9S 89953995 Ki = 12 nM T40016 CK29LG 89954151 Ki = 7.6 nM T40016 CFKJ67 89954179 Ki = 0.88 nM T40016 CP68TD 89954189 Ki = 3.1 nM T40016 C6HPE2 89954292 Ki = 31 nM T40016 CPHU03 89954366 Ki = 1.3 nM T40016 C2MPT3 89954418 Ki = 0.64 nM T40016 C0PU6X 89954457 Ki = 0.29 nM T40016 CM38BS 89954484 Ki = 9.7 nM T40016 CQ5WA1 89954525 Ki = 0.15 nM T40016 CU45GK 89954608 Ki = 0.32 nM T40016 CIX49O 89954622 Ki = 11 nM T40016 CXW1Q6 89954759 Ki = 0.59 nM T40016 C90OKR 89954788 Ki = 0.19 nM T40016 CKMB42 89954841 Ki = 0.29 nM T40016 CDH31J 89954858 Ki = 6.6 nM T40016 C9A4ZX 89955032 Ki = 0.42 nM T40016 C4HDM0 89955037 Ki = 0.33 nM T40016 CM5V8H 89955158 Ki = 0.32 nM T40016 CK5D1A 90395281 IC50 > 20000 nM T40016 CQ06RH 90654508 IC50 = 1300 nM T40016 C6VZ7X 90656360 IC50 > 10000 nM T40016 CNCB43 90656361 IC50 > 10000 nM T40016 C4BA8W 90656430 IC50 = 32000 nM T40016 C0Q5MF 90656551 IC50 = 10000 nM T40016 CQM94C 90656552 IC50 = 10000 nM T40016 CA95DL 90656553 IC50 > 10000 nM T40016 C7G4UN 90656554 IC50 > 10000 nM T40016 CXK9Q8 90656555 IC50 > 10000 nM T40016 CJ1X6I 90656556 IC50 = 32 nM T40016 CC0E1Z 90656557 IC50 = 85 nM T40016 CHI35V 90662883 EC50 = 21.1 nM T40016 CA9PL8 91663316 IC50 = 22300 nM T40016 CE4Z3U 102313488 IC50 = 10000 nM T40016 CF67IH 117917065 EC50 = 3.2 nM T40016 CFG2T8 117917077 Ki = 69.4 nM T40016 CDZ31K 117917098 Ki = 1.5 nM T40016 CW27MY 118063735 EC50 > 10000 nM T40016 C6BQ8K 118092322 Ki = 60 nM T40016 C43QTL 118092331 Ki = 120 nM T40016 CZ7DT3 118092342 Ki = 24 nM T40016 CL47CF 118092345 Ki = 44 nM T40016 CGD29J 118092358 Ki = 68 nM T40016 CSK83H 118092376 Ki = 34 nM T40016 CD7RS9 118599615 Ki = 31.62 nM T40016 C70AOV 118599714 Ki = 630.96 nM T40016 C8XLO9 118599727 Ki = 2511.89 nM T40016 CW7G4T 118599742 Ki = 125.89 nM T40016 C9L5EW 118599756 Ki = 5011.87 nM T40016 CVIW94 118599769 Ki = 316.23 nM T40016 CFS28Y 118599779 Ki = 3162.28 nM T40016 CREN83 118707969 Ki = 2.5 nM T40016 CC2I1P 118707970 Ki = 12.9 nM T40016 C7XD9E 118707971 Ki = 8.5 nM T40016 CF60IG 118707972 Ki = 8.7 nM T40016 CZB1G7 118707973 Ki = 110.5 nM T40016 C3XOR9 118707974 Ki = 6.9 nM T40016 CDA17Q 118707975 Ki = 5.7 nM T40016 CTKA86 118707976 Ki = 8.7 nM T40016 CVW2B3 118707977 Ki = 7.4 nM T40016 CLS7C1 118707978 EC50 = 1.2 nM T40016 C9LV0M 118707979 Ki = 1.6 nM T40016 CV4DC0 118707980 Ki = 0.7 nM T40016 COJB29 118707981 Ki = 1.9 nM T40016 C3TLR1 118707982 EC50 = 0.6 nM T40016 CMW3N5 118707983 Ki = 2 nM T40016 C72VHF 118707984 Ki = 7.3 nM T40016 C06ZWX 118707985 Ki = 4 nM T40016 C6Y5JG 118723171 IC50 = 300 nM T40016 CE3I9T 118723172 IC50 = 24 nM T40016 C13AIC 118723173 IC50 = 21 nM T40016 C21SWI 118723174 IC50 = 56 nM T40016 CKR24J 118723175 IC50 = 60 nM T40016 C28YZF 118723176 IC50 = 170 nM T40016 C6AGI7 118723177 IC50 > 2000 nM T40016 C4QO8E 118723178 IC50 = 260 nM T40016 C31RJM 118735258 IC50 = 5.2 nM T40016 C1IC6W 118735259 IC50 = 47 nM T40016 C70CMF 118735260 IC50 = 20.1 nM T40016 C6FDB4 118735261 IC50 = 35.4 nM T40016 C20TNQ 118735262 IC50 = 650 nM T40016 CKWU27 118735263 IC50 = 79 nM T40016 CVZ95N 118735264 IC50 = 28 nM T40016 CLE9O2 121248060 IC50 = 1.7 nM T40016 CPVF94 121248184 EC50 = 5.6 nM T40016 C61QKR 121248207 EC50 = 2.7 nM T40016 CG13LX 122178361 IC50 = 2900 nM T40016 C9LIR4 122179356 Ki = 16 nM T40016 CUI57B 122179357 IC50 < 30 nM T40016 C9U1QL 122179358 Ki = 146 nM T40016 CTQZ35 122179359 Ki = 106 nM T40016 CR98CI 122179360 Ki = 28 nM T40016 C24FBP 122179361 Ki > 384 nM T40016 CGF74Y 122179362 Ki > 384 nM T40016 C10YVG 122179363 Ki > 384 nM T40016 C0OR2H 122186738 Ki = 654 nM T40016 CU0Y8B 122186739 Ki = 39.8 nM T40016 CWF0Q4 122186740 Ki = 115 nM T40016 CBE6Q8 122186741 Ki = 2.67 nM T40016 CX13DR 122186742 Ki = 0.543 nM T40016 CJ74HX 122186743 Ki = 53.7 nM T40016 C05VWL 122186744 Ki = 1.32 nM T40016 CNX5H4 122186745 Ki = 5.45 nM T40016 C4E5JI 122186746 Ki = 1410 nM T40016 CQ6BG8 122186747 Ki = 5.04 nM T40016 CH8O2M 122186748 Ki = 3.06 nM T40016 C4LRN1 122186749 Ki = 94.6 nM T40016 CN9C2T 122192181 IC50 > 31622.78 nM T40016 CCK36V 127029882 IC50 > 5000 nM T40016 CFY1P0 127029884 IC50 = 651 nM T40016 CLDC46 127031152 IC50 > 37000 nM T40016 C60SMC 127031153 IC50 > 12000 nM T40016 CWG34O 127036544 Ki = 0.47 nM T40016 CY0WZ9 129295280 IC50 = 5.6 nM T40016 C65RIZ 129295282 IC50 = 33.6 nM T40016 CM62UE 129295287 IC50 = 14.6 nM T40016 CR23ZG 129295311 IC50 = 47.2 nM T40016 C2LVO7 129295370 IC50 = 57.9 nM T40016 CTI04S 129295372 IC50 = 52.1 nM T40016 C4G2ID 129304679 IC50 = 16.1 nM T40016 CGK48C 129304682 IC50 = 43 nM T40016 CEVZ49 129304683 IC50 = 16.6 nM T40016 CM4LD6 129304687 IC50 = 19.5 nM T40016 C6XAZ5 129304688 IC50 = 17.5 nM T40016 C85QXL 129304691 IC50 = 205 nM T40016 CR3YV9 129304702 IC50 = 16.7 nM T40016 CS2UB8 129304733 IC50 = 28 nM T40016 COU93J 129304741 IC50 = 43 nM T40016 C7K2IE 129304748 IC50 = 9.6 nM T40016 C2GJ8T 129304757 IC50 = 13.3 nM T40016 C7MRB5 129304758 IC50 = 7.5 nM T40016 CN0UA7 129304771 IC50 = 48 nM T40016 CBSJ31 129304830 IC50 = 12.4 nM T40016 C1H0UX 129304861 IC50 = 16 nM T40016 C9ELW1 132275097 IC50 = 2.4 nM T40016 C12UNI 132502971 IC50 = 1430 nM T40016 CK3P0W 132502972 IC50 = 3150 nM T40016 CFT2A4 134132246 EC50 = 47 nM T40016 CP7U8D 134133225 IC50 = 0.62 nM T40016 CNE2Y4 134134891 IC50 = 0.9 nM T40016 COYD80 134135818 IC50 = 1.4 nM T40016 C79OUF 134136440 EC50 = 149 nM T40016 CH9KN0 134136493 EC50 = 1861 nM T40016 C4UX7Z 134137342 EC50 = 0.11 nM T40016 C9TG2N 134137487 IC50 = 0.1585 nM T40016 CED46P 134138613 IC50 = 0.07 nM T40016 C8HY9A 134141623 IC50 = 37 nM T40016 CRJ12I 134141987 IC50 = 558 nM T40016 CNS5V7 134144852 EC50 = 280 nM T40016 CS4P3B 134145141 IC50 = 91 nM T40016 CK10EC 134145786 IC50 = 2400 nM T40016 C0XRT2 134146077 IC50 = 0.09 nM T40016 CVS65Y 134148910 EC50 = 265 nM T40016 CTPU54 134149674 EC50 = 100 nM T40016 C46HMP 134149836 IC50 = 455 nM T40016 CM0TA5 134149846 IC50 = 8.83 nM T40016 CD3E2J 134149965 EC50 = 0.04 nM T40016 CX9T1H 134150995 IC50 = 0.4 nM T40016 C87YMA 134156029 IC50 = 1870 nM T40016 CY7ZM4 134157373 EC50 = 240 nM T40016 CNBM96 134157739 IC50 = 84 nM T40016 CD58OH 134157814 EC50 = 0.05 nM T40016 C30HIQ 134415607 IC50 = 12.2 nM T40016 C3Y2NT 134415609 IC50 = 52.2 nM T40016 CQ53DW 134415610 IC50 = 116 nM T40016 CO32XF 134415624 IC50 = 10.3 nM T40016 CRP1C4 134415742 IC50 = 12.7 nM T40016 C1U9HD 134415745 IC50 = 13.9 nM T40016 CB09XQ 134415864 IC50 = 20.6 nM T40016 CU6Y5D 134415868 IC50 = 35.8 nM T40016 C1GY2T 135156251 EC50 > 10000 nM T40016 CY8U6E 135459005 IC50 > 100000 nM T40016 CBA2F6 135513268 IC50 > 50000 nM T40016 CTF0J3 135567449 Ki = 50.12 nM T40016 CN24YZ 135567451 Ki = 251.19 nM T40016 CPF3B4 135567452 Ki = 7.943 nM T40016 C34JMK 135571931 IC50 > 100000 nM T40016 C5MXO2 136000568 Ki = 0.6 nM T40016 CD07ZO 136000655 Ki = 7 nM T40016 CM6OX5 136000656 Ki = 0.8 nM T40016 CZ2D6U 136059148 Ki = 2.2 nM T40016 C6HOU3 136059149 Ki = 2 nM T40016 CE1G9O 136059150 Ki = 3.8 nM T40016 C7LSN6 136088946 EC50 = 0.6 nM T40016 C1F4BY 136088947 Ki = 0.7 nM T40016 CRJ9V5 136088948 IC50 = 3.5 nM T40016 C1M3WU 136088949 Ki = 1.5 nM T40016 CR4X3Q 136088950 Ki = 5.8 nM T40016 CI4RW5 136088951 Ki = 31 nM T40016 C4OX9M 136088952 Ki = 0.4 nM T40016 C2JV0P 136088953 Ki = 2700 nM T40016 C98CLF 136098616 Ki = 5.7 nM T40016 CEP7N9 136254190 IC50 = 3 nM T40016 C1B2KD 137631905 IC50 = 0.156 nM T40016 C38MWL 137632612 IC50 > 1000 nM T40016 CC10WR 137632878 IC50 > 30000 nM T40016 CE48UI 137633773 IC50 > 30000 nM T40016 COI80Z 137634236 IC50 = 12.59 nM T40016 CQ6J5I 137637753 IC50 > 30000 nM T40016 C5B4PZ 137637922 IC50 > 30000 nM T40016 CAHT60 137638938 IC50 > 30000 nM T40016 CPD87Y 137639726 IC50 = 19.95 nM T40016 CGCA32 137639839 IC50 > 30000 nM T40016 CEGX68 137640275 IC50 = 0.12 nM T40016 C8TBZ4 137641110 IC50 = 24.3 nM T40016 CZRS94 137641411 IC50 > 30000 nM T40016 CXQ8P3 137641761 IC50 > 30000 nM T40016 C6E0AL 137642668 IC50 = 5770 nM T40016 C0T3HQ 137643401 IC50 > 30000 nM T40016 C46QZA 137647155 IC50 = 7870 nM T40016 C0K4BJ 137648403 IC50 = 464 nM T40016 C30ZJF 137648477 IC50 = 6.31 nM T40016 CJE8B2 137648715 IC50 > 30000 nM T40016 C4SJD8 137650072 IC50 = 7480 nM T40016 CAS7B9 137651118 IC50 = 3590 nM T40016 CRYF53 137651691 IC50 = 1970 nM T40016 CW9Y6S 137651919 IC50 = 12.7 nM T40016 CWZ06G 137652587 IC50 = 5420 nM T40016 CO92KL 137654415 IC50 = 15.85 nM T40016 C5MXU1 137655191 IC50 = 0.066 nM T40016 C1CM0L 137656584 IC50 > 30000 nM T40016 C75CDY 137658459 IC50 = 2040 nM T40016 CP46JS 137658546 IC50 > 30000 nM T40016 COT7M8 137659850 IC50 > 30000 nM T40016 C7JKI9 137660091 IC50 > 1000 nM T40016 CZ49NM 137660168 IC50 = 2020 nM T40016 CQWG60 137661608 IC50 = 0.15 nM T40016 CZWT36 137661763 IC50 > 30000 nM T40016 C54OHS 137661940 IC50 = 2110 nM T40016 C7EKA2 138911324 IC50 = 8.5 nM T40016 C96ONI 141538600 IC50 = 58.3 nM T40016 CR6Y2I 141538601 IC50 = 28.5 nM T40016 CR5Y9P 145949269 IC50 = 1.93 nM T40016 CW3Y0H 145949340 IC50 > 20000 nM T40016 CP5U7Q 145949975 EC50 = 57 nM T40016 COKU96 145950643 IC50 = 32 nM T40016 CPK5U1 145951022 IC50 > 20000 nM T40016 CKT24R 145951943 IC50 > 20000 nM T40016 CD49VI 145953389 IC50 = 18.1 nM T40016 CU19EN 145958055 IC50 = 11.2 nM T40016 C5U3JV 145958117 IC50 = 8.5 nM T40016 CORP09 145958365 EC50 = 17.4 nM T40016 CR6T8S 145959457 IC50 = 64 nM T40016 CU84AB 145963803 IC50 < 3.2 nM T40016 C9AH5J 145964455 IC50 < 4 nM T40016 C72QDJ 145964714 IC50 = 9.3 nM T40016 CSJ60M 145964914 EC50 = 3.5 nM T40016 C2QB3L 145964915 IC50 < 4.1 nM T40016 CX94YN 145965573 IC50 < 0.34 nM T40016 CF0PO7 145965716 IC50 = 57 nM T40016 CS8G3K 145965784 EC50 = 29 nM T40016 C9Y6RT 145965869 IC50 = 7.1 nM T40016 CE9PD6 145966463 IC50 = 160 nM T40016 CW61TA 145966634 IC50 = 1.6 nM T40016 C14OAC 145966706 IC50 = 2 nM T40016 CVT2B5 145971542 IC50 = 7.2 nM T40016 C1V7EP 145972549 EC50 = 13 nM T40016 C34ENO 145972998 IC50 < 1.6 nM T40016 C71PDT 145973741 IC50 = 21 nM T40016 C8DFZ5 145973994 IC50 = 6.1 nM T40016 C0V1TU 145974260 EC50 = 3.5 nM T40016 CM9QN8 145974940 IC50 = 42 nM T40016 CJFS50 145975057 IC50 = 4.7 nM T40016 C19HXS 145975460 IC50 = 11 nM T40016 C2GUH7 145975580 EC50 = 23 nM T40016 CH87UD 145976543 IC50 = 120 nM T40016 C7CUS0 145976724 IC50 < 0.42 nM T40016 CBOW92 145977353 IC50 = 39 nM T40016 C32VLX 145977741 IC50 = 449 nM T40016 C1PMA8 145977753 EC50 = 87 nM T40016 CJY2W5 145978475 IC50 < 6.8 nM T40016 C5T7IK 147930449 Ki = 316.23 nM T40016 C30SYM 155459658 IC50 = 62 nM T40016 CGB78J 155459666 IC50 = 73.7 nM T40016 C0MF5X 155512827 IC50 = 9.5 nM T40016 C28RHM 155514304 Ki = 1995.26 nM T40016 CE2YJ9 155514399 Ki = 79.43 nM T40016 CQF09V 155516050 Ki = 630.96 nM T40016 CELU49 155517819 Ki > 15848.93 nM T40016 C2E4XV 155518137 Ki = 12589.25 nM T40016 C4QAB0 155518139 Ki > 15848.93 nM T40016 C6VIG2 155518655 IC50 = 1012 nM T40016 CCO0Z4 155519877 Ki = 199.53 nM T40016 CC5JZ4 155520100 IC50 > 1000 nM T40016 COF3R4 155520306 IC50 = 0.41 nM T40016 C8BD6Y 155522508 Ki = 398.11 nM T40016 C71VIK 155525344 Ki = 1258.93 nM T40016 C1WAQ6 155527406 Ki = 1258.93 nM T40016 C5T2QN 155528866 Ki = 158.49 nM T40016 CQM89D 155529443 Ki = 1.585 nM T40016 CR0N3F 155529454 Ki = 125.89 nM T40016 CB0XS4 155529625 Ki > 15848.93 nM T40016 C5Y4FK 155531943 IC50 = 6 nM T40016 C3HFZ6 155534085 Ki > 15848.93 nM T40016 CF52DM 155535034 Ki = 1.259 nM T40016 CXR2W1 155536089 IC50 = 4016 nM T40016 C3FON4 155537084 Ki > 12589.25 nM T40016 CJH5I3 155538097 IC50 = 135 nM T40016 COP7X8 155539171 IC50 > 10000 nM T40016 C78ISM 155540009 IC50 = 202 nM T40016 C28KPU 155540268 IC50 = 20 nM T40016 C84LKI 155540713 IC50 = 130 nM T40016 CIAW80 155544156 IC50 = 1051 nM T40016 C76OVS 155544396 Ki > 12589.25 nM T40016 C25HEV 155545046 IC50 > 1000 nM T40016 CR6UY8 155545121 IC50 = 1644 nM T40016 C1XGF5 155546726 IC50 = 17.6 nM T40016 CC36TR 155546752 IC50 = 89 nM T40016 CJ9T5D 155548288 IC50 = 10 nM T40016 C6H2ML 155552723 Ki = 316.23 nM T40016 CW8BH4 155554673 Ki = 1258.93 nM T40016 C9WV3L 155556878 Ki = 1000 nM T40016 CR5ZI2 155557239 Ki = 1258.93 nM T40016 CPY83L 155558503 Ki > 15848.93 nM T40016 C0FEP8 155559859 IC50 > 1000 nM T40016 CQ7HG2 155561626 Ki = 2.512 nM T40016 CBM45A 155563942 IC50 > 1000 nM T40016 CD4K6Z 155564467 Ki = 19.95 nM T40016 CS25QB 155564604 IC50 = 111 nM T40016 C7YK6N 155565026 IC50 = 870 nM T40016 CPX2J5 155566857 Ki > 15848.93 nM T40016 C79WFJ 155567245 Ki > 15848.93 nM T40016 CME1B7 155567676 Ki = 6309.57 nM T40016 CWQI82 136130172 Ki = 370 nM T40016 D00DNY 3213 IC50 = 90000 nM T40016 D00ZGW 46883841 IC50 = 199.53 nM T40016 D01ETZ 261000 Ki = 9.65 nM T40016 D01NVD 46830196 IC50 = 100 nM T40016 D02UID 16734800 IC50 = 1000 nM T40016 D05XVM 18189209 IC50 = 1937 nM T40016 D05ZUX 44207909 Ki >= 1000 nM T40016 D07KWO 9823099 IC50 = 2.4 nM T40016 D08KQM 24816375 Ki = 2.4 nM T40016 D09FQL 16756780 IC50 = 900 nM T40016 D09OKK 9951771 Ki = 564 nM T40016 D0D6GI 46888441 EC50 = 93 nM T40016 D0EG5G 46888467 EC50 = 19 nM T40016 D0F1SS 44605900 IC50 > 1000 nM T40016 D0GR5L 9906282 Ki = 1.4 nM T40016 D0J7XZ 9819614 Ki = 0.17 nM T40016 D0L5IC 9820558 Ki = 0.1 nM T40016 D0M0RS 11560224 Ki > 1000 nM T40016 D0N8UD 46888391 IC50 = 86 nM T40016 D0O5ZG 44305900 IC50 = 1914 nM T40016 D0PR2T 16756782 IC50 = 13000 nM T40016 D0S9KH 63052 IC50 = 600 nM T40016 D0T2RY 9948320 Ki >= 1000 nM T40016 D0T4SL 72512 IC50 = 90000 nM T40016 D0V4RZ 25113722 IC50 = 7200 nM T40016 D0XS0R 44433505 Ki = 1758 nM T99834 C9SYZ3 3708153 EC50 = 22300 nM T99834 C8PDE1 14686324 EC50 = 42500 nM T99834 C45BQH 132585194 EC50 = 4800 nM T42048 D02YNI 9936746 Ki = 4 nM T42048 D05ICT 132010322 Ki = 4.9 nM T42048 D07OFM 46943432 Ki = 30.3 nM T42048 D0M2TS 71600087 Ki = 12.2 nM T42048 D0PH9I 118693659 Ki = 63.1 nM T42048 D0ZW4W 46907787 Ki = 6.6 nM T42048 D09SFV 3973 IC50 = 13700 nM T42048 C92EYR 1503595 IC50 = 30000 nM T42048 CIG94A 13953713 IC50 = 12589.25 nM T42048 C3VRO9 44557921 IC50 > 10000 nM T42048 C98BLM 49871817 IC50 = 19.1 nM T42048 CG3PR6 52912222 IC50 = 0.631 nM T42048 CBXV52 52932793 IC50 = 316.23 nM T42048 CJE59U 52932930 IC50 = 1258.93 nM T42048 CSZ2T6 52932933 IC50 = 3162.28 nM T42048 CN87IR 52933159 IC50 = 1258.93 nM T42048 CG6OL4 52933160 IC50 = 794.33 nM T42048 CP8Y9K 52933161 IC50 = 1000 nM T42048 CK8Z4P 52933165 IC50 = 3162.28 nM T42048 CKC17F 52933403 IC50 = 1000 nM T42048 CD08ZX 52933405 IC50 = 1000 nM T42048 C1T7VQ 52933407 IC50 = 1258.93 nM T42048 CO8VX9 52933655 IC50 = 1584.89 nM T42048 C6G7BE 52933893 IC50 = 1000 nM T42048 C7VN1E 52934039 IC50 = 501.19 nM T42048 CUZE18 52934122 IC50 = 1000 nM T42048 CN16FE 52934128 IC50 = 1995.26 nM T42048 CTS13B 52934275 IC50 = 630.96 nM T42048 CNOH36 52935183 IC50 = 199.53 nM T42048 CLRH53 52935478 IC50 = 794.33 nM T42048 CJIB35 53054190 IC50 = 4700 nM T42048 C6V8YR 53054191 IC50 = 13000 nM T42048 C09HTR 53054200 IC50 = 1000 nM T42048 CUS8F7 53054236 IC50 = 4800 nM T42048 CX5QN4 53054237 IC50 = 14000 nM T42048 CD2TY9 53054238 IC50 = 6500 nM T42048 C47GAW 53054240 IC50 = 5400 nM T42048 CVH2G1 53054241 IC50 = 2200 nM T42048 CF9E2V 53054248 IC50 = 1900 nM T42048 CRWK92 53054249 IC50 = 5900 nM T42048 CSXI51 53054250 IC50 = 1800 nM T42048 CM12EL 53054251 IC50 = 1900 nM T42048 CY5L3J 53054252 IC50 = 4000 nM T42048 CWV76Y 53054258 IC50 = 700 nM T42048 CIU8P7 53054259 IC50 = 500 nM T42048 CVX3R0 53054274 IC50 = 3000 nM T42048 CB05OM 53054276 IC50 = 1100 nM T42048 CLR97U 53054289 IC50 = 1000 nM T42048 CJ6E2Q 53054291 IC50 = 3300 nM T42048 C1WSZ4 53054297 IC50 = 1500 nM T42048 C7A2XC 53054319 IC50 = 2000 nM T42048 C0J1EO 53054320 IC50 = 3800 nM T42048 CK68UF 53054321 IC50 = 800 nM T42048 CJY5S2 53054322 IC50 = 3200 nM T42048 C1YW5L 53054324 IC50 = 2100 nM T42048 C8Q6WG 53054325 IC50 = 1000 nM T42048 C9V5LX 53318989 IC50 = 220 nM T42048 C1KWY4 54759170 IC50 = 2500 nM T42048 C7HK2C 56924692 IC50 = 1100 nM T42048 CX6SD9 56950289 IC50 = 3000 nM T42048 CZ6NE0 56950420 IC50 = 1400 nM T42048 CJ5BE9 56950421 IC50 = 2200 nM T42048 CL96VQ 56950422 IC50 = 1300 nM T42048 CCLD98 56950423 IC50 = 8600 nM T42048 CZD7G2 56950424 IC50 = 4200 nM T42048 CPQ0B7 56950425 IC50 = 8600 nM T42048 CL90DK 56950426 IC50 = 700 nM T42048 CF9IJ1 56950561 IC50 = 700 nM T42048 CH24QC 56950562 IC50 = 8200 nM T42048 CU62NO 56950563 IC50 = 11000 nM T42048 CRD86M 56950564 IC50 = 11000 nM T42048 CNQ2L5 56950565 IC50 = 21000 nM T42048 CB3A1Z 56950566 IC50 = 8400 nM T42048 C5ADP4 56950567 IC50 = 13000 nM T42048 CFW0D1 57339435 IC50 = 501.19 nM T42048 CF8B4E 60498769 IC50 = 62000 nM T42048 CPY59D 67195867 IC50 = 25118.86 nM T42048 CN3KZ8 68161075 IC50 = 316.23 nM T42048 C49IOA 68161669 IC50 = 398.11 nM T42048 CJ7N3M 68184870 IC50 = 1000 nM T42048 CT4Z2A 68184871 IC50 = 398.11 nM T42048 CEX74I 68186034 IC50 = 5011.87 nM T42048 C25INY 68204735 IC50 = 630.96 nM T42048 CMC7V5 70664240 IC50 = 630.96 nM T42048 C1I6OH 70681167 IC50 = 3162.28 nM T42048 C7GJW9 70681170 IC50 = 316.23 nM T42048 C8H4JX 70681173 IC50 = 501.19 nM T42048 C6NYK2 70681174 IC50 = 398.11 nM T42048 C8KBJ0 70683271 IC50 = 501.19 nM T42048 CXD3F9 70691699 IC50 = 251.19 nM T42048 CL8Y9N 71450297 IC50 = 630.96 nM T42048 C6CQT5 71462842 IC50 = 1584.89 nM T42048 CIPN50 71760902 Ki = 35 nM T42048 C2AFW1 72702849 IC50 = 501.19 nM T42048 C3R1IL 72703043 IC50 = 100000 nM T42048 CK9O6W 72705811 IC50 = 6309.57 nM T42048 C5TB9S 77843982 Ki = 110 nM T42048 CS6XE0 77846025 Ki = 3.2 nM T42048 COZ8S1 78319129 Ki = 290 nM T42048 C4IF8T 78425807 Ki = 10 nM T42048 CFE7R3 86270928 Ki = 10 nM T42048 C53QEW 86669224 IC50 = 6309.57 nM T42048 CEDL57 89657555 IC50 = 7 nM T42048 CZJ8W9 90387575 Ki = 4.2 nM T42048 C1W3XP 112499930 IC50 = 1800 nM T42048 C6A1RW 118120978 IC50 = 1710 nM T42048 CHB87O 118120979 IC50 = 1320 nM T42048 CPN74M 118719856 IC50 = 501.19 nM T42048 CE8DL3 118719857 IC50 = 794.33 nM T42048 COEU47 118719858 IC50 = 1258.93 nM T42048 CX05SW 118719859 IC50 = 630.96 nM T42048 CRCG07 118719860 IC50 = 501.19 nM T42048 C03XDG 118719861 IC50 = 630.96 nM T42048 C3ML2F 118719862 IC50 = 398.11 nM T42048 CZ67WF 118719863 IC50 = 25118.86 nM T42048 C0HR9Y 118719864 IC50 = 501.19 nM T42048 C7F4EP 118719865 IC50 = 316.23 nM T42048 CA40QV 118719866 IC50 = 501.19 nM T42048 CZ8QI6 118719867 IC50 = 1000 nM T42048 C8NRI9 118719868 IC50 = 794.33 nM T42048 C3Y2WT 118719869 IC50 = 794.33 nM T42048 C52HPM 118719870 IC50 = 501.19 nM T42048 CUT97H 118719871 IC50 = 501.19 nM T42048 CBE68N 118719872 IC50 = 1258.93 nM T42048 C29WRE 118719873 IC50 = 501.19 nM T42048 C8J0TY 118719874 IC50 = 1000 nM T42048 CZR10C 118719875 IC50 = 2511.89 nM T42048 C35AWU 118719876 IC50 = 1584.89 nM T42048 C3QJ5L 122181550 IC50 > 50118.72 nM T42048 CO25IW 122191031 IC50 >= 10000 nM T42048 C4WGV6 122191040 IC50 = 10000 nM T42048 CDY43J 122191048 IC50 >= 10000 nM T42048 C4GYP3 126521168 IC50 = 25 nM T42048 CL2PG5 126521180 IC50 = 18 nM T42048 CQV90I 126521354 IC50 = 16 nM T42048 C1DOG4 126521586 IC50 = 10 nM T42048 CRY0S6 126563516 IC50 = 14 nM T42048 CN0D6M 126563562 IC50 = 13 nM T42048 CKB36S 126563576 IC50 = 11 nM T42048 CX79NH 126563597 IC50 = 39 nM T42048 C2K5XG 126563611 IC50 = 23 nM T42048 CZ06NR 126563612 IC50 = 44 nM T42048 CM5P2Z 126563615 IC50 = 36 nM T42048 C15ILF 126564427 IC50 = 10 nM T42048 CHO12Y 126564469 IC50 > 10000 nM T42048 CB2AS4 126564470 IC50 = 9 nM T42048 CBW08I 126564471 IC50 = 19 nM T42048 CD78GB 126564481 IC50 = 21 nM T42048 CNP2L7 126564832 IC50 = 14 nM T42048 C58PNK 126564833 IC50 = 21 nM T42048 CHPV09 126564847 IC50 = 12 nM T42048 CJZW04 126564858 IC50 = 13 nM T42048 CH14FC 127032939 IC50 = 4800 nM T42048 CS4NG8 127033568 IC50 = 31700 nM T42048 C9L1OG 130345579 Ki = 2.5 nM T42048 CRNY32 135397673 Ki = 0.18 nM T42048 CV4X7R 135566898 Ki = 1640 nM T42048 CU2F1G 135566900 Ki = 220 nM T42048 C5F3LV 135567026 IC50 > 100000 nM T42048 CW94QO 136226511 Ki = 240 nM T42048 CO71RI 137285009 IC50 = 2241 nM T42048 CS9MR6 137285011 IC50 = 2193 nM T42048 CFXE14 137321203 IC50 = 31.62 nM T42048 CXN4U1 137321204 IC50 = 1258.93 nM T42048 C4VNB8 137369426 IC50 = 52 nM T42048 CU5N8O 137701509 IC50 = 11200 nM T42048 CQ6XB7 139030526 IC50 = 31622.78 nM T42048 C1G9LA 139035062 Ki = 5.3 nM T42048 CG6X3A 142535938 IC50 = 42 nM T42048 CD6U7X 145925666 IC50 = 246.3 nM T42048 C1HLK5 145951928 IC50 = 21 nM T42048 CV83ED 145972103 Ki = 17 nM T42048 CK20BY 145988169 Ki = 42.4 nM T42048 C9FIY4 153534005 IC50 > 20000 nM T42048 CFD6H1 155352361 IC50 = 51000 nM T42048 CFK2B1 155352401 IC50 = 200000 nM T42048 C76QMK 155513141 Ki = 8.2 nM T42048 C27LFN 155514936 IC50 = 770 nM T42048 C6OP0S 155535292 Ki = 11.1 nM T42048 C0HI7N 155536879 IC50 = 456 nM T42048 CUX25H 155547195 Ki = 13.9 nM T42048 CZA5N1 155561689 IC50 > 20500 nM T42048 C7ICA9 155564455 IC50 = 78 nM T42048 D00XRH 91820725 IC50 = 19952.62 nM T42048 D03LIP 13953710 IC50 = 28.4 nM T42048 D09HBR 135566899 Ki = 100 nM T42048 D09VHS 3971 IC50 = 11500 nM T42048 D0F5TZ 91827383 IC50 = 7943.28 nM T42048 D0N5BI 91668541 IC50 > 50118.72 nM T42048 D0WU1S 52912189 Ki = 7.2 nM T09572 D0A3CL 49801838 IC50 = 27 nM T09572 D0TV4N 9865843 Ki = 5.5 nM T09572 D0U0YR 11520239 IC50 = 3 nM T09572 D00RUE 60169095 IC50 = 20 nM T09572 D03KWP 71660914 IC50 = 48 nM T09572 D0C5RD 71719525 IC50 = 50 nM T09572 D0HH1O 71731806 IC50 = 17 nM T09572 D0MT7T 71816518 IC50 = 6.8 nM T09572 D0Q1NA 71660917 IC50 = 77 nM T09572 D0V8FC 60169096 IC50 = 30 nM T09572 C97FYX 702501 IC50 = 43000 nM T09572 C12OHT 1252415 Ki = 11300 nM T09572 CQ6BS4 2276336 Ki = 8100 nM T09572 CUM8T0 2729098 IC50 = 109 nM T09572 CRA9T2 2729502 Ki = 347 nM T09572 CVE13J 2881764 Ki = 11900 nM T09572 CSM9V8 3410248 IC50 = 114 nM T09572 CX6CF2 3611477 IC50 = 82 nM T09572 C2EN7Y 4219492 IC50 = 59 nM T09572 CB9WS0 4653788 IC50 > 2000 nM T09572 C5I9SA 4826270 Ki = 7800 nM T09572 C39UDN 5312114 IC50 = 3500 nM T09572 CBJD49 5817261 IC50 = 56 nM T09572 CRV52B 6621104 IC50 = 30 nM T09572 CP5X6Z 9799244 EC50 = 96 nM T09572 C5GL6S 9799726 Ki = 29 nM T09572 CA4Z7C 9801165 Ki < 1 nM T09572 C8XGV3 9804849 IC50 = 16 nM T09572 CYIT28 9806086 IC50 = 50 nM T09572 C1NQC6 9807658 IC50 = 4.9 nM T09572 C2MIW9 9821717 IC50 = 2 nM T09572 C5RIY7 9824428 IC50 = 250 nM T09572 C1J9MV 9824856 IC50 = 6 nM T09572 CG3X9R 9828622 IC50 = 300 nM T09572 CJZ9L7 9829942 IC50 = 5 nM T09572 CX2PO5 9844702 IC50 = 17 nM T09572 C0Q8UT 9848699 Ki = 24 nM T09572 C2PU9N 9851676 Ki = 11 nM T09572 CAKP95 9866552 IC50 = 10 nM T09572 CSTG23 9866745 IC50 = 2 nM T09572 C74RZP 9887476 IC50 = 2.7 nM T09572 C34NSZ 9887864 IC50 = 7 nM T09572 C6EK5P 9888078 IC50 > 100 nM T09572 C9BRE3 9895005 Ki = 6.4 nM T09572 CY1P7H 9895868 IC50 = 140 nM T09572 CTZ48N 9910346 IC50 = 1.9 nM T09572 C5YM8X 9915039 Ki = 0.17 nM T09572 CIP6V7 9932896 IC50 = 0.54 nM T09572 C4L1GA 9934033 IC50 = 3.4 nM T09572 CDY39E 9934161 IC50 = 9 nM T09572 CSWJ86 9954518 Ki = 19.95 nM T09572 CTUO16 9955811 IC50 = 1300 nM T09572 CT7AP4 9978378 IC50 = 11 nM T09572 C5FB3N 9978428 IC50 = 5 nM T09572 CMY73F 9978490 IC50 = 7 nM T09572 C9XH3V 9978508 IC50 = 5.5 nM T09572 CF41ZD 9980157 IC50 = 16 nM T09572 C7TPF5 9983233 IC50 = 2 nM T09572 CVL8X0 9984325 Ki = 45 nM T09572 C9Y6GX 9985634 Ki = 9.772 nM T09572 CS6Q2J 9985881 Ki = 34 nM T09572 CV2D9B 9986014 Ki = 14 nM T09572 C4T2XD 9986044 Ki = 10 nM T09572 CP8WR3 9999058 IC50 = 62 nM T09572 CG14IV 10000146 IC50 = 0.9 nM T09572 CQL12P 10004545 Ki = 0.6 nM T09572 C6OI1A 10005009 IC50 = 1.9 nM T09572 C6Q0IN 10007632 Ki = 823 nM T09572 CXL43G 10008279 Ki = 16 nM T09572 CZ45JK 10024145 IC50 = 6 nM T09572 C4U8JG 10024171 IC50 = 5.9 nM T09572 C3O2EL 10024175 IC50 = 15 nM T09572 C8M2YA 10025637 IC50 = 10 nM T09572 C3NPS8 10025899 IC50 = 12 nM T09572 CS14OM 10027853 IC50 = 1.5 nM T09572 CP9JI2 10029161 Ki = 59 nM T09572 C9XTE6 10029835 Ki = 35 nM T09572 CRJ41C 10029836 Ki = 63 nM T09572 C4XK0H 10031575 Ki = 7 nM T09572 C0UQ4M 10036257 IC50 > 2000 nM T09572 CD4KM9 10041636 IC50 = 120 nM T09572 C02OIU 10047339 IC50 = 28 nM T09572 CA2ZW7 10050565 IC50 = 4.1 nM T09572 C4IS6W 10053890 Ki = 25 nM T09572 CGHX74 10053937 Ki = 10.96 nM T09572 CFA8Y5 10054046 Ki = 2600 nM T09572 C5T6CZ 10059666 IC50 > 2000 nM T09572 C0Y9JS 10067783 IC50 = 0.9 nM T09572 C8PH7Y 10070016 IC50 = 11 nM T09572 CM5S6R 10070680 IC50 = 21 nM T09572 C2Z4FO 10073563 IC50 = 790 nM T09572 CCN5S8 10073934 IC50 = 2.9 nM T09572 CRQL64 10075375 IC50 = 4 nM T09572 C3T7HL 10077022 Ki = 1800 nM T09572 CWD1K0 10077403 Ki = 6.8 nM T09572 C1UCY7 10098577 Ki = 38 nM T09572 CR3MJ4 10099409 Ki = 24 nM T09572 C3FME5 10100662 Ki = 16 nM T09572 C2D6TX 10113523 Ki = 1.2 nM T09572 CNCP64 10114686 IC50 = 0.88 nM T09572 CQ3U9H 10115919 Ki = 2.6 nM T09572 C8MJ1U 10117415 Ki = 1.4 nM T09572 CXJ79U 10118862 Ki = 0.31 nM T09572 CT5GK7 10118863 Ki = 0.45 nM T09572 CX4IA7 10126754 EC50 = 380 nM T09572 C7IFU2 10127348 EC50 = 96 nM T09572 CG7Z9I 10128764 Ki = 1428 nM T09572 COS3D1 10128900 Ki = 2.2 nM T09572 CEO59I 10129026 Ki = 281 nM T09572 CW5O4B 10129036 Ki = 52 nM T09572 C3FS7G 10129058 Ki = 18 nM T09572 CJ05QL 10129135 Ki = 76 nM T09572 C1XK6M 10139496 Ki = 15.85 nM T09572 CTND76 10139873 Ki = 100 nM T09572 CDN19U 10140070 Ki = 6 nM T09572 C8MTR3 10140707 Ki = 4.3 nM T09572 CCSW12 10141528 Ki = 5.5 nM T09572 CP9Q6O 10142124 Ki = 2.6 nM T09572 CFL14Q 10142464 Ki = 37 nM T09572 CX9EI2 10143421 Ki = 19 nM T09572 CZ95DQ 10143980 Ki = 15 nM T09572 CPR42N 10149893 IC50 = 8300 nM T09572 CZT7L9 10150552 EC50 = 110 nM T09572 C2L3HU 10150954 EC50 = 210 nM T09572 CD9V8P 10150955 IC50 = 3 nM T09572 C2X9YI 10152629 Ki = 99 nM T09572 C9VP5L 10152726 Ki = 523 nM T09572 CVGB64 10152879 Ki = 4 nM T09572 C9TQ1J 10159452 IC50 = 2.7 nM T09572 CLW3P2 10159789 Ki = 7.4 nM T09572 C2V1TA 10159797 Ki = 19.95 nM T09572 CRW17C 10160079 Ki = 398.11 nM T09572 CBV5S9 10161039 Ki = 1.5 nM T09572 C8ALH2 10164110 Ki = 2.6 nM T09572 CJ5HL7 10165163 Ki = 2.1 nM T09572 CX36LA 10165503 Ki = 2.5 nM T09572 CZQ69G 10165656 Ki = 27 nM T09572 CFQM97 10166038 Ki < 100 nM T09572 C9EJT4 10166088 Ki = 131 nM T09572 C6ZPK7 10173726 IC50 = 4.5 nM T09572 CC2F7Z 10173787 IC50 = 18 nM T09572 CM9KF2 10174522 Ki = 241 nM T09572 CO2XG1 10174940 Ki = 1.6 nM T09572 CH25WF 10174984 Ki = 2 nM T09572 CX48ZP 10184368 Ki = 4.7 nM T09572 CF8Q2N 10185187 Ki = 50 nM T09572 C47RGT 10186370 Ki = 35 nM T09572 CUO81F 10186375 Ki = 5.4 nM T09572 CQP58G 10186594 Ki = 0.98 nM T09572 C80YEW 10188732 Ki = 82 nM T09572 CM0RA3 10195637 Ki = 4.1 nM T09572 CGJ7D9 10195667 Ki = 18 nM T09572 C9OB3S 10196098 Ki = 3 nM T09572 C2K1LR 10196214 Ki = 178 nM T09572 CBX4C2 10196316 Ki = 21 nM T09572 CD9N3H 10196460 Ki = 3 nM T09572 CYT8S5 10196576 Ki = 9 nM T09572 C5EGZ8 10196608 Ki = 16 nM T09572 C0OB2A 10196742 Ki = 49 nM T09572 CV9H1P 10202381 IC50 = 1000 nM T09572 C6M4SO 10203421 Ki = 3.3 nM T09572 C1V9WG 10204047 Ki = 1.1 nM T09572 CUL57F 10204151 Ki = 0.84 nM T09572 C48NGR 10206922 Ki = 5.6 nM T09572 C63SDN 10209344 Ki = 0.63 nM T09572 CMY61O 10210351 Ki = 20 nM T09572 CDK26C 10217978 Ki = 7.1 nM T09572 CIC0H8 10218194 Ki = 77 nM T09572 CH7BP9 10218547 Ki = 2162 nM T09572 CX7KR8 10218604 Ki = 23 nM T09572 CB4VT6 10224210 Ki = 2.2 nM T09572 CA1YM8 10225681 IC50 = 1.995 nM T09572 C7YUF6 10226765 Ki = 0.98 nM T09572 CP25NG 10229815 Ki = 46 nM T09572 CKMB46 10230235 Ki = 26 nM T09572 C78KEN 10230490 Ki = 0.41 nM T09572 CEO3C0 10230947 Ki = 10 nM T09572 CNHR93 10231050 IC50 = 160 nM T09572 CX5S8V 10231341 Ki = 1.2 nM T09572 CT50QF 10238912 Ki = 13 nM T09572 C2AV9K 10239389 Ki = 215 nM T09572 CWTM13 10239448 Ki = 180 nM T09572 CY3B9V 10239505 Ki = 6 nM T09572 C9ZR5W 10239639 Ki = 690 nM T09572 C8GUX5 10239907 Ki = 9 nM T09572 C8R7NE 10239929 Ki = 1667 nM T09572 C2JY5L 10239930 Ki = 786 nM T09572 C4M9EA 10248906 IC50 = 30 nM T09572 CY3C6Z 10250850 IC50 = 24 nM T09572 CC94UL 10255474 IC50 = 850 nM T09572 CC7K0Q 10256914 Ki = 29 nM T09572 CRI6L0 10257135 Ki = 12 nM T09572 C9U7QP 10257298 Ki = 23 nM T09572 C46ALH 10258364 IC50 = 0.71 nM T09572 CK7W0O 10273126 Ki = 2.4 nM T09572 CM8Q4V 10274635 IC50 = 7 nM T09572 CZ7TK1 10277136 Ki = 79.43 nM T09572 C4HN5M 10277257 Ki = 398.11 nM T09572 CNY7O0 10280331 Ki = 61 nM T09572 C7GFV9 10281308 Ki = 7.2 nM T09572 CQAM65 10289494 Ki = 3 nM T09572 CD32KO 10289615 Ki = 2.5 nM T09572 C8GUV6 10295411 Ki = 63.1 nM T09572 C97VMZ 10297428 Ki = 9.2 nM T09572 CS6AF7 10298251 Ki = 1.4 nM T09572 C7JB9Z 10301472 Ki = 1.6 nM T09572 CP4MX9 10303281 Ki = 12 nM T09572 C3ZJY6 10303307 IC50 = 79 nM T09572 CA5PV1 10304239 Ki = 40 nM T09572 C16TVN 10310161 IC50 = 12 nM T09572 C2IG7F 10310316 IC50 = 2.8 nM T09572 C5NVX2 10310772 Ki = 3 nM T09572 CUZ0N7 10310778 IC50 > 4000 nM T09572 C8X2OD 10311260 Ki = 1174 nM T09572 CS5YX7 10311798 Ki = 141 nM T09572 C51CRS 10312052 Ki = 13 nM T09572 CHR1A3 10312086 Ki = 3247 nM T09572 CCRI74 10312244 Ki = 16 nM T09572 CMC1G5 10319824 IC50 = 2410 nM T09572 CQ9RL7 10325994 Ki = 36 nM T09572 CVO3N7 10344176 IC50 = 6.4 nM T09572 C3YB4P 10345121 IC50 = 1.9 nM T09572 CSB63G 10345845 IC50 = 0.46 nM T09572 CIW12H 10347752 Ki = 15 nM T09572 CHE8C4 10347753 Ki = 138 nM T09572 C3LZ7G 10347754 Ki = 13 nM T09572 CC3GW1 10348080 Ki = 15 nM T09572 C3WC2E 10348147 Ki = 54 nM T09572 C3KOI9 10348749 Ki = 24 nM T09572 C9FI8M 10360874 IC50 = 0.4 nM T09572 CQG45X 10361342 IC50 = 30 nM T09572 CMD9J2 10385550 IC50 > 100000 nM T09572 C3C2LS 10386162 IC50 = 20 nM T09572 CP4S9C 10386529 IC50 = 77 nM T09572 CAI68E 10388351 IC50 = 5 nM T09572 CF17HN 10388352 IC50 = 20 nM T09572 CL83KQ 10388797 IC50 = 16 nM T09572 C36BOF 10389430 IC50 = 63 nM T09572 CESG32 10389978 IC50 = 6.1 nM T09572 C7W4TF 10391177 IC50 = 2.7 nM T09572 C39PRE 10392311 Ki = 22 nM T09572 C5EXD4 10408758 IC50 = 149 nM T09572 CS6MA7 10413283 IC50 = 1 nM T09572 CWU0O3 10415704 Ki = 9.3 nM T09572 CYD95P 10433825 IC50 = 6 nM T09572 C6T7WB 10434776 IC50 = 50 nM T09572 CFV7D4 10436090 IC50 = 8.1 nM T09572 C2LYJ4 10436663 Ki = 26 nM T09572 CV9KC4 10436862 Ki = 138 nM T09572 C5SX2J 10443228 IC50 > 2000 nM T09572 C07KPU 10456755 IC50 = 88 nM T09572 CY17SB 10459635 IC50 = 0.71 nM T09572 CGQ62I 10460913 Ki > 1000 nM T09572 CO42XC 10461033 Ki = 16 nM T09572 CN85WI 10480652 IC50 = 3450 nM T09572 COLB47 10481477 IC50 = 1 nM T09572 C8GV3E 10483604 Ki = 119 nM T09572 CHI65E 10483729 Ki = 5100 nM T09572 CSP9I7 10483799 Ki > 1000 nM T09572 CV5GD3 10483882 Ki > 1000 nM T09572 C8SK7B 11156521 Ki = 7.3 nM T09572 CUD3I6 11156790 Ki = 14 nM T09572 C7SZD0 11165058 IC50 = 90 nM T09572 C52FBG 11166395 IC50 = 10 nM T09572 CLY23H 11168108 Ki = 16.3 nM T09572 C19UHW 11168186 Ki = 1.8 nM T09572 C6Y7LA 11168831 Ki = 1.9 nM T09572 CJ30VR 11168918 Ki = 6.7 nM T09572 C0N1BS 11169159 Ki = 21.3 nM T09572 CCA26O 11178792 IC50 = 71 nM T09572 CRW5M2 11190261 IC50 = 146 nM T09572 C9W0VG 11191034 Ki = 1.7 nM T09572 C7YZ1U 11191656 Ki = 6.8 nM T09572 CPS26T 11201645 IC50 = 0.9 nM T09572 C50SKJ 11201867 IC50 = 67 nM T09572 C24JXQ 11204090 IC50 = 83 nM T09572 C8AS3V 11211551 IC50 = 178 nM T09572 C7E9AN 11222404 IC50 = 3.3 nM T09572 CX47OL 11236807 Ki = 4.7 nM T09572 CC62PB 11238080 Ki = 2.7 nM T09572 CSPC85 11238695 Ki = 20 nM T09572 C64KCU 11238718 Ki = 1145 nM T09572 CW07ZE 11246373 IC50 = 369 nM T09572 CAS5P8 11247985 Ki = 19 nM T09572 CZ98EU 11259253 IC50 = 5 nM T09572 CIM40L 11259560 IC50 > 10000 nM T09572 CKBJ08 11260997 Ki = 8.2 nM T09572 C2U7OP 11270012 Ki = 7.4 nM T09572 CB8ZS6 11270984 IC50 = 558 nM T09572 C7JP8R 11272081 Ki = 8.4 nM T09572 CFZP19 11282448 IC50 = 287 nM T09572 CJ3Q4Y 11282697 Ki = 233 nM T09572 CCWK17 11284878 IC50 = 140 nM T09572 C49PQG 11292322 IC50 = 35 nM T09572 CCG2J7 11295707 Ki = 12.5 nM T09572 C4JK1H 11296279 IC50 = 320 nM T09572 CU4L6M 11304816 IC50 = 58 nM T09572 CP98MD 11306487 Ki = 98 nM T09572 CN38VE 11307645 Ki = 1.5 nM T09572 CK9E2Y 11317465 Ki = 20 nM T09572 CK4P6A 11317824 Ki = 20.7 nM T09572 CO7CX6 11318577 Ki = 391 nM T09572 CCU9P8 11318709 Ki = 39 nM T09572 CWT28O 11328029 IC50 = 6 nM T09572 C7R2ZE 11329623 Ki = 5.6 nM T09572 C47VRG 11329860 Ki = 6.2 nM T09572 CR1BG6 11330800 Ki = 3000 nM T09572 CZ6FG9 11340348 Ki = 3.1 nM T09572 C5R2GO 11340894 Ki = 139 nM T09572 CR1K5W 11342160 IC50 = 250 nM T09572 CVGM47 11351174 IC50 = 78 nM T09572 CHJ73G 11353174 Ki = 2.2 nM T09572 C36OES 11374857 IC50 = 160 nM T09572 C43HJQ 11376081 Ki = 4 nM T09572 CQ58NT 11376122 Ki = 27 nM T09572 CU3V1H 11387603 Ki = 197 nM T09572 C3XR6W 11408441 IC50 = 5 nM T09572 C7MVN8 11409615 Ki = 70.8 nM T09572 CBL42Y 11410080 Ki = 327.6 nM T09572 CI8X2J 11410430 Ki = 25.7 nM T09572 CI80HK 11410594 Ki = 405 nM T09572 CF6XZ1 11419337 IC50 = 12 nM T09572 C2RXD8 11419338 IC50 = 46 nM T09572 C0EHV3 11419666 IC50 = 24.5 nM T09572 CI3RU9 11419776 IC50 = 15 nM T09572 C26DPU 11420203 Ki = 7.1 nM T09572 C28YHB 11420543 Ki = 11 nM T09572 C69OFJ 11420621 Ki = 5.8 nM T09572 CB51KQ 11433168 Ki = 26 nM T09572 CXY0L4 11442761 IC50 = 4 nM T09572 CTAI65 11452967 Ki = 6 nM T09572 CJP2I6 11453830 IC50 = 1985 nM T09572 C09HMW 11454965 Ki = 4.9 nM T09572 C50BVO 11455871 Ki = 4.9 nM T09572 CKU5J7 11464405 IC50 = 4 nM T09572 C5JFE2 11467626 Ki = 14.2 nM T09572 CN54JD 11476556 IC50 = 772000 nM T09572 CI6CY2 11489130 Ki = 8.9 nM T09572 C1I3TF 11489588 Ki = 13.7 nM T09572 CMQ86R 11495432 IC50 = 5 nM T09572 C6L8DU 11495754 IC50 = 2.1 nM T09572 C9YME5 11496313 IC50 = 1.6 nM T09572 CZG39V 11496739 IC50 = 2.3 nM T09572 CQF0N9 11496824 Ki = 92 nM T09572 CE0FW1 11497179 Ki = 15 nM T09572 CSG7A1 11497180 Ki = 87 nM T09572 CZIE58 11502008 IC50 = 5.8 nM T09572 COC9S1 11504274 IC50 = 6 nM T09572 CEGY35 11504793 Ki = 180 nM T09572 CRVH23 11504906 Ki = 2.8 nM T09572 C10FVQ 11505089 IC50 = 13 nM T09572 CCP2Z0 11510399 IC50 = 4 nM T09572 CB59MV 11510669 IC50 = 145 nM T09572 C72BCW 11510887 IC50 = 266 nM T09572 CTKH79 11511219 IC50 = 25 nM T09572 CW6C2K 11511638 Ki = 2190 nM T09572 CXH3M7 11511671 Ki = 9.6 nM T09572 C9DE5V 11511776 IC50 = 15 nM T09572 C2B6YR 11512135 IC50 = 5.9 nM T09572 CVW89A 11512221 Ki = 6.6 nM T09572 CEPN59 11516903 IC50 = 45 nM T09572 C7O3YC 11517116 IC50 > 1000 nM T09572 CKH3R6 11518999 Ki = 3.3 nM T09572 CI1H6G 11519341 Ki > 3000 nM T09572 CW4V9C 11519451 Ki = 1.8 nM T09572 CZN1S8 11519652 Ki = 3000 nM T09572 CB86YA 11525369 IC50 = 57 nM T09572 C1TLH5 11526309 IC50 = 78 nM T09572 CGU14V 11526592 Ki = 30 nM T09572 CMCE20 11526824 IC50 = 93 nM T09572 CL04IY 11527169 Ki = 44 nM T09572 CQ7LC4 11531010 IC50 = 8 nM T09572 C24VTF 11531660 IC50 = 41 nM T09572 C4W2IN 11533195 IC50 = 35 nM T09572 C8W1XB 11533835 Ki = 8 nM T09572 CQ08DH 11539632 IC50 = 85 nM T09572 C5NA7O 11541231 Ki = 1615 nM T09572 C3E9MH 11545677 IC50 = 9 nM T09572 CP8I4R 11546687 IC50 = 734 nM T09572 CI15ZK 11547011 Ki = 3.3 nM T09572 CE34IS 11547939 IC50 = 9.7 nM T09572 CX6IL5 11548234 IC50 = 1.5 nM T09572 C69YGT 11548597 Ki = 3.5 nM T09572 C0KYZ7 11553316 IC50 = 163 nM T09572 CW4QS9 11553648 IC50 = 150 nM T09572 C0I6EV 11553871 IC50 = 1.585 nM T09572 CZD24Q 11554412 IC50 = 3 nM T09572 CPM70L 11554989 IC50 = 48 nM T09572 C64NID 11555572 IC50 = 37 nM T09572 CNWU65 11556070 IC50 = 2 nM T09572 C5WKO2 11559625 IC50 = 18 nM T09572 C7J9IY 11560917 IC50 = 6 nM T09572 CXR53E 11561126 IC50 = 0.5 nM T09572 C0XQ1U 11561155 IC50 = 120 nM T09572 CS5M0K 11562056 Ki = 52 nM T09572 CF8E0C 11562129 IC50 = 100 nM T09572 CDP1L5 11562138 IC50 = 2 nM T09572 CX3HC8 11563017 IC50 = 11 nM T09572 CY0N7L 11563153 IC50 = 340 nM T09572 C59SVL 11563383 IC50 = 21 nM T09572 CMFZ35 11568741 IC50 = 339 nM T09572 C2BIP8 11568782 IC50 = 29 nM T09572 C0J3VR 11569300 IC50 = 32 nM T09572 CAEY52 11569327 Ki = 2 nM T09572 CAC92H 11569340 IC50 = 302 nM T09572 CN0S1H 11570031 IC50 = 31 nM T09572 CJ9RX4 11570040 Ki = 3.5 nM T09572 C8FXD6 11577410 Ki = 2.3 nM T09572 CN87ZF 11577588 IC50 = 22 nM T09572 C2YIV1 11577708 Ki = 727 nM T09572 CXKA03 11581666 IC50 = 3628 nM T09572 CM0H2R 11583049 IC50 = 2 nM T09572 CZ6C8H 11583193 IC50 = 1 nM T09572 CPA3J7 11583744 IC50 = 2.7 nM T09572 CNT0J4 11583747 IC50 = 2 nM T09572 CP07QN 11583835 IC50 = 20 nM T09572 C70NAD 11583925 IC50 = 330 nM T09572 CS6OE5 11584710 Ki = 2.5 nM T09572 COE14C 11589812 IC50 = 38 nM T09572 CNB39X 11591169 IC50 = 50 nM T09572 C5SOE3 11591542 IC50 = 380 nM T09572 CLW26H 11591644 IC50 = 8 nM T09572 CD6Y3F 11592099 IC50 = 2 nM T09572 C3E9YV 11592199 IC50 = 88 nM T09572 CLEA14 11592317 Ki = 129 nM T09572 CMAF85 11596311 IC50 = 6.6 nM T09572 CAU85E 11597758 IC50 = 313 nM T09572 C9OU8J 11598355 IC50 = 2 nM T09572 CE0N5F 11599186 IC50 = 16 nM T09572 C0H3WV 11599681 IC50 = 5360 nM T09572 CKI9D5 11599973 IC50 = 6 nM T09572 CS1EL0 11603897 IC50 = 7 nM T09572 CRAO19 11604236 IC50 = 297 nM T09572 CCL5H9 11605260 IC50 = 1050 nM T09572 C97GBU 11605775 IC50 = 49 nM T09572 CEF85Q 11605821 Ki = 11 nM T09572 CC5R1Q 11610423 Ki = 2.3 nM T09572 CP4VN0 11611530 IC50 = 60 nM T09572 C9I5GN 11612098 IC50 = 19 nM T09572 CYB0H4 11612847 Ki = 190 nM T09572 CM03ZX 11613073 IC50 = 1.7 nM T09572 CDA48G 11613696 Ki = 3.7 nM T09572 CP9T8V 11613829 Ki = 9.3 nM T09572 CG1RP5 11619850 IC50 = 3 nM T09572 CDT2Y7 11620005 IC50 = 540 nM T09572 CIO53A 11627085 IC50 = 44 nM T09572 C2NC0H 11627122 IC50 = 9 nM T09572 CHS10O 11627316 Ki = 13 nM T09572 CGEX14 11627530 IC50 = 1.3 nM T09572 C3CI5V 11627700 Ki = 6 nM T09572 CVA6R9 11628136 Ki = 41 nM T09572 CEK0Z8 11628328 IC50 = 25 nM T09572 C6CXP5 11628547 Ki = 221 nM T09572 CA90RE 11632484 IC50 = 20 nM T09572 C7H9VD 11632909 IC50 = 461 nM T09572 CCN9E6 11633862 IC50 = 90 nM T09572 CE70ZA 11634061 IC50 = 42 nM T09572 CX36IC 11634230 IC50 = 98 nM T09572 CP46KM 11634329 Ki = 13 nM T09572 CBW24J 11634823 IC50 = 38 nM T09572 C75FNR 11634886 IC50 = 26 nM T09572 CDE1G8 11635187 IC50 = 25 nM T09572 C8Y9AL 11635230 IC50 = 99 nM T09572 C8LU4M 11635274 Ki = 4.8 nM T09572 CUN3R9 11635332 IC50 = 74 nM T09572 C0PQ9D 11635674 Ki = 1.8 nM T09572 C5U4HW 11635715 Ki = 67 nM T09572 CY3IN5 11640515 IC50 = 24 nM T09572 C8SBV2 11641333 Ki = 605 nM T09572 CH79OL 11641948 IC50 = 15 nM T09572 CUG36W 11642443 Ki = 37 nM T09572 CLFC12 11642491 Ki = 96 nM T09572 CKM2Z4 11646818 IC50 = 10 nM T09572 CJQK24 11647458 IC50 = 10 nM T09572 C5A4YW 11648240 IC50 = 13 nM T09572 CTLK95 11648753 Ki = 8.9 nM T09572 CK2SO9 11648912 IC50 = 0.1 nM T09572 C1XZ5S 11648976 Ki = 161 nM T09572 C0WAT8 11649549 IC50 = 3 nM T09572 CE57QF 11653882 IC50 = 20 nM T09572 C8I7UT 11654412 IC50 = 5.6 nM T09572 CM0J9D 11654904 IC50 > 1000 nM T09572 CRF2O3 11655701 Ki = 18 nM T09572 CFHR60 11655790 IC50 > 1000 nM T09572 CP09GF 11655872 IC50 = 29 nM T09572 CTW7H9 11656044 IC50 = 151 nM T09572 CI3YO9 11656489 IC50 = 29 nM T09572 C35CMI 11656728 Ki = 1300 nM T09572 CT0YF3 11656805 Ki = 160 nM T09572 C2TDF5 11656916 Ki = 71.4 nM T09572 C6Q7TC 11657090 Ki = 22 nM T09572 CJ8OS7 11662564 IC50 = 158 nM T09572 C1F9VA 11662657 IC50 = 4 nM T09572 CESA67 11662906 IC50 = 22 nM T09572 CZ0KM9 11663109 IC50 > 1000 nM T09572 C91WGJ 11664086 Ki = 32 nM T09572 CW0C5S 11664134 Ki = 3000 nM T09572 C5NI1G 11670645 Ki = 648 nM T09572 CMXQ27 11671178 Ki = 2.9 nM T09572 CX3WF2 11676200 IC50 = 710 nM T09572 CXB59V 11676220 IC50 = 1.4 nM T09572 C0R5KF 11677277 IC50 = 2 nM T09572 CW1MI7 11677806 IC50 = 109 nM T09572 CW0N1P 11678040 Ki = 4.4 nM T09572 C4KG5D 11678370 IC50 = 140 nM T09572 C8UVK4 11678666 Ki = 394 nM T09572 CD7C4O 11683259 IC50 = 5.4 nM T09572 CEHG64 11683903 IC50 = 16 nM T09572 CG76YZ 11684745 IC50 = 45 nM T09572 C8S2RG 11691468 Ki = 16.98 nM T09572 CR0JZ3 11691995 IC50 = 54 nM T09572 C8CWF4 11692133 Ki = 7 nM T09572 CKX65Z 11692293 IC50 = 519 nM T09572 C3HOB4 11692382 Ki = 167 nM T09572 CJ6C2T 11692643 Ki = 29 nM T09572 C6QKV2 11698276 Ki = 380 nM T09572 C17ZOJ 11698592 Ki = 3.6 nM T09572 CW5Z4U 11698729 Ki = 340 nM T09572 C3D1IX 11698964 Ki = 33 nM T09572 CMZ94P 11699265 Ki = 15 nM T09572 CYR87W 11705240 IC50 = 19 nM T09572 CR6BE5 11705485 IC50 = 29 nM T09572 CG2LE3 11706442 IC50 = 39 nM T09572 CE1FU8 11706443 IC50 = 41 nM T09572 C16BRA 11706744 Ki = 4 nM T09572 CKZJ72 11710969 IC50 > 1000 nM T09572 CIZQ65 11711452 IC50 = 7 nM T09572 CL3H6E 11712583 IC50 = 39 nM T09572 C8V9XO 11712898 IC50 = 29 nM T09572 C1MV6S 11713027 IC50 = 1.4 nM T09572 CWQ67V 11713742 IC50 = 23 nM T09572 C74DRE 11719291 IC50 = 7 nM T09572 C87WCU 11719447 Ki = 1 nM T09572 CIR3H9 11719877 Ki = 8.2 nM T09572 CO29BN 11719912 IC50 = 39 nM T09572 CQV4D8 11720881 Ki = 61 nM T09572 C3CSB2 11740891 IC50 = 26 nM T09572 CG70PF 11743571 IC50 = 2 nM T09572 C7IR0M 11752320 IC50 = 5.2 nM T09572 CFB78R 11752339 Ki = 7.9 nM T09572 C6T9RV 11752579 Ki = 7.1 nM T09572 CIB4J8 11752750 Ki = 3 nM T09572 C0REU4 11756387 Ki = 38 nM T09572 C8KZ7Y 11758076 Ki = 11 nM T09572 C15NMU 11758499 Ki = 9.7 nM T09572 CDT5W6 11775399 IC50 = 1.4 nM T09572 C7JD4S 11775505 IC50 = 71 nM T09572 CMT60I 11778029 IC50 = 310 nM T09572 CX20YM 11785261 Ki = 9.2 nM T09572 CJZ1S6 11785262 Ki = 8.8 nM T09572 C3URN6 11785761 Ki = 11.4 nM T09572 CCA5X9 11786179 Ki = 374 nM T09572 CF5X6S 11786476 Ki = 166 nM T09572 CQ3UA0 11837128 IC50 = 191 nM T09572 C8MT6W 11973798 IC50 = 427 nM T09572 CA54WB 11973799 IC50 = 13 nM T09572 C09SBY 11973800 IC50 = 966 nM T09572 C4G3JS 11973801 IC50 = 53 nM T09572 CJ51DI 11973802 IC50 = 1690 nM T09572 CW4V0D 11973803 IC50 > 2000 nM T09572 C0X9SH 11973913 IC50 > 2000 nM T09572 CY6F0Q 11973915 IC50 > 2000 nM T09572 CYA98F 11973916 IC50 = 1140 nM T09572 CTQ2M5 11974030 IC50 = 178 nM T09572 C9OQ1D 11974034 IC50 = 351 nM T09572 C1NEZ7 11974035 IC50 = 187 nM T09572 CRP64S 11974126 IC50 = 132 nM T09572 CYF81E 11974128 IC50 > 2000 nM T09572 C68TIS 11974129 IC50 = 1480 nM T09572 CU3J7M 11974130 IC50 = 59 nM T09572 CN38YH 11974131 IC50 = 137 nM T09572 C05LEI 11974132 IC50 = 393 nM T09572 C72WDJ 11974227 IC50 = 99 nM T09572 C1BXQ6 11974228 IC50 = 418 nM T09572 C5W7EA 11974229 IC50 = 601 nM T09572 C3C2EN 11974230 IC50 = 171 nM T09572 CAN81B 11974231 IC50 = 31 nM T09572 C2QW4A 11974233 IC50 = 2150 nM T09572 CHJ84N 11974345 IC50 = 159 nM T09572 CNCP71 11974346 IC50 = 39 nM T09572 C7W6UZ 11975326 IC50 = 192 nM T09572 CJ82RK 11975327 IC50 = 24 nM T09572 C8KJU9 11975436 IC50 = 75 nM T09572 C3EU8T 11975438 IC50 = 60 nM T09572 CJ0M5S 11975440 IC50 > 700 nM T09572 CGHS90 11993892 IC50 = 2 nM T09572 CC67HK 11993893 IC50 = 0.89 nM T09572 CY2R0H 11993894 IC50 = 1.3 nM T09572 CTR36W 11993895 IC50 = 6.1 nM T09572 CH46NZ 11993896 IC50 = 6.2 nM T09572 CY93VJ 11993897 IC50 = 37 nM T09572 CKJ40R 11994017 IC50 = 3.2 nM T09572 C2X1FE 11994018 IC50 = 6918 nM T09572 COYJ12 11994019 IC50 = 3.4 nM T09572 C2XV4Y 11994136 IC50 = 8.5 nM T09572 CZO24Q 11994137 IC50 = 25 nM T09572 CU4ZI8 11994138 IC50 = 24 nM T09572 CE0D8U 11994273 IC50 > 10000 nM T09572 C87MRI 11994275 IC50 = 31.6 nM T09572 CUT45B 11994276 IC50 > 10000 nM T09572 CO9RD2 11994277 IC50 = 5 nM T09572 CB47ZX 11994412 IC50 = 0.87 nM T09572 C2TXD4 11994413 IC50 = 1.1 nM T09572 C1FLA4 11994414 IC50 = 3.1 nM T09572 CP3ID2 11994659 IC50 = 1.3 nM T09572 CX49YR 11994660 IC50 = 2.5 nM T09572 C8WS7J 11994661 IC50 = 5.7 nM T09572 CID9L3 11994662 IC50 = 29 nM T09572 CNOW76 11994780 IC50 = 1.4 nM T09572 CKS43A 11994784 IC50 = 1.1 nM T09572 C75HYU 11994786 IC50 = 1.1 nM T09572 CXJ16Z 11994909 IC50 > 10000 nM T09572 C79ATS 11994910 IC50 = 1412 nM T09572 C9SDQ6 11994911 IC50 = 2.7 nM T09572 CGJD13 11994912 IC50 = 0.75 nM T09572 CH52LD 11994913 IC50 = 1.3 nM T09572 CDI85R 11995024 IC50 = 0.91 nM T09572 CB8E2J 11995025 IC50 = 2 nM T09572 C1F3KB 11995026 IC50 = 38 nM T09572 CL8U5H 11995028 IC50 = 9.5 nM T09572 CUTI13 11995136 IC50 = 794 nM T09572 C6X5QK 11995137 IC50 = 3980 nM T09572 C7CQ0R 11995138 IC50 = 40 nM T09572 C65FGL 11995139 IC50 = 478 nM T09572 CO3S6Y 11995140 IC50 = 36 nM T09572 CUG9Q0 11995141 IC50 = 200 nM T09572 CA0TX2 11995240 IC50 = 63 nM T09572 CM12WP 11995241 IC50 = 87 nM T09572 C7VYA1 11995242 IC50 = 1 nM T09572 C6AT2K 11995243 IC50 = 5.6 nM T09572 C48VEJ 11995244 IC50 = 1.5 nM T09572 C5RE4A 11995245 IC50 = 3.1 nM T09572 C56OSH 11995342 IC50 = 3.1 nM T09572 CV28MQ 11995343 IC50 = 19 nM T09572 C19YGN 11995344 IC50 = 3.8 nM T09572 C9L5UO 11995345 IC50 = 3.5 nM T09572 CR8C7Y 11995346 IC50 = 4168 nM T09572 CDV83P 11995347 IC50 = 2.3 nM T09572 COUR13 11995441 IC50 = 5.3 nM T09572 CZ23MA 11995442 IC50 = 3.5 nM T09572 C91ZIU 11995443 IC50 = 7.7 nM T09572 CKF0H1 11995444 IC50 = 3.2 nM T09572 CG9Z2R 11995445 IC50 = 7 nM T09572 C0QSD9 11995552 IC50 = 4.9 nM T09572 CY07CV 11995644 IC50 = 1258 nM T09572 CZQ39K 11995645 IC50 = 501 nM T09572 CE2OQ3 11995646 IC50 = 31 nM T09572 C41NIS 11995647 IC50 = 501 nM T09572 CSJ72B 11995648 IC50 = 0.74 nM T09572 CM6P0A 12002494 IC50 > 5000 nM T09572 CZ0UY2 12020149 Ki = 20 nM T09572 C9L6BY 12020151 IC50 = 100 nM T09572 CR64CY 12020152 Ki = 51 nM T09572 C42JBR 12020156 IC50 = 270 nM T09572 C61WZV 12020161 Ki = 108 nM T09572 CLP70H 12020164 Ki = 191 nM T09572 CN3FB9 12020168 Ki = 795 nM T09572 CICW40 12020169 Ki = 266 nM T09572 CY6BQ4 15133403 EC50 = 140 nM T09572 C7WB4Y 15981934 Ki > 5000 nM T09572 CL50KS 15983730 Ki = 220 nM T09572 CD39IP 15983731 Ki > 5000 nM T09572 CM1I3Z 15983732 Ki > 5000 nM T09572 C4QLI2 15983733 Ki = 341 nM T09572 CGUZ74 15983734 Ki > 5000 nM T09572 C8PFB1 15983862 Ki = 357 nM T09572 C9A0LX 15983863 Ki > 5000 nM T09572 C76FSJ 15983864 Ki = 707 nM T09572 CDT5B7 15983865 Ki = 2060 nM T09572 C43HRS 15983866 Ki > 5000 nM T09572 CXW37K 15987265 IC50 = 5 nM T09572 CQ2H5X 15987638 IC50 = 2630 nM T09572 C8FV4Y 16006976 Ki = 6 nM T09572 CL2PB7 16006977 Ki = 7 nM T09572 CKJ76E 16006978 IC50 = 2.2 nM T09572 CB0JD2 16037921 Ki = 1 nM T09572 CX9W7Q 16043220 Ki = 21 nM T09572 CFM31I 16043291 Ki = 0.6 nM T09572 CB6LK8 16046114 Ki = 19.95 nM T09572 CR78OW 16046124 Ki = 3.981 nM T09572 CD65KI 16046157 Ki = 51 nM T09572 CA5YN3 16049789 IC50 = 0.3 nM T09572 C3LK2C 16072132 Ki = 3 nM T09572 CRU35S 16106513 Ki = 77 nM T09572 CJ4M0E 16110074 Ki = 31.62 nM T09572 CU37CY 16116777 Ki = 39.81 nM T09572 CJLX24 16192241 IC50 = 11000 nM T09572 C72BAI 16659061 Ki = 78 nM T09572 C23NUI 16659197 Ki = 140 nM T09572 COC0B8 16659239 Ki = 16000 nM T09572 CYS2H0 16659240 IC50 = 20 nM T09572 CFXU61 16718619 IC50 = 13 nM T09572 C7K5AW 16721015 IC50 = 1 nM T09572 CV5F3P 16739263 IC50 = 29 nM T09572 CO1W7Z 16739310 Ki = 8 nM T09572 CTB2D8 16739324 Ki = 10 nM T09572 CGCY91 16742745 IC50 = 154 nM T09572 C2IJ3D 16742746 IC50 = 7 nM T09572 C4URY2 16742747 IC50 = 20 nM T09572 C8V1KM 16745235 IC50 = 3 nM T09572 CDK04H 16745305 Ki = 43 nM T09572 C96RYO 17173466 IC50 = 23000 nM T09572 COL97Q 17484866 IC50 = 6500 nM T09572 C7HA3N 17545006 IC50 = 23000 nM T09572 C5SO0V 17848895 IC50 = 190 nM T09572 CSTQ69 17989325 Ki = 398.11 nM T09572 CJ7Z4X 17989329 Ki = 19.95 nM T09572 CWC4K6 17989356 Ki = 125.89 nM T09572 CL2QF0 17989369 Ki = 15.85 nM T09572 CYV93L 17989373 Ki = 50.12 nM T09572 C5P3IU 17989383 Ki = 316.23 nM T09572 CKX23J 17989406 Ki = 31.62 nM T09572 C5X4FZ 17989409 Ki = 25 nM T09572 C6SZ0G 17989439 Ki = 82 nM T09572 CVSB32 18361509 IC50 > 1000 nM T09572 CI46GT 18435902 IC50 = 1.8 nM T09572 C2DFS4 18435980 IC50 = 6.6 nM T09572 C03YQS 18435984 IC50 = 35 nM T09572 CQ86SW 18435986 IC50 = 48 nM T09572 C0IPE3 18435988 IC50 = 23 nM T09572 CFYX59 18436038 IC50 = 2 nM T09572 C37CPM 18436043 IC50 = 1600 nM T09572 CCS6E4 18436055 IC50 = 0.74 nM T09572 C7MUE8 18436066 IC50 = 0.36 nM T09572 C9HN3G 18436075 IC50 = 9.2 nM T09572 CA9UL8 18436082 IC50 = 1.4 nM T09572 CDQS35 18436083 IC50 = 1.4 nM T09572 C1WJ0Z 18436085 IC50 = 10 nM T09572 C3CYE7 18436094 IC50 = 0.92 nM T09572 C56SPK 18436095 IC50 = 110 nM T09572 C5Z8FL 18436109 IC50 = 170 nM T09572 CF7Q1R 18436112 IC50 = 3.7 nM T09572 CS24AR 18436114 IC50 = 0.53 nM T09572 C34WKZ 18436115 IC50 = 2.2 nM T09572 C0H7OP 18436117 IC50 = 1 nM T09572 CXL27Y 18436118 IC50 = 100 nM T09572 C0ST8U 18436119 IC50 = 3.2 nM T09572 C7X1SY 18436120 IC50 = 4.1 nM T09572 C9F2DA 18436123 IC50 = 25 nM T09572 C32IMY 18436125 IC50 = 26 nM T09572 CW6HU8 18436126 IC50 = 18 nM T09572 CCN82B 18436129 IC50 = 73 nM T09572 CAP6L1 18672590 Ki = 31.62 nM T09572 CBR6Q7 20608969 Ki = 61 nM T09572 COF9E8 20608974 Ki = 19 nM T09572 CWSB30 20608975 Ki = 13 nM T09572 C7PL9M 20608976 Ki = 42 nM T09572 CG9R3I 20608977 Ki = 40 nM T09572 C9U6JQ 20608981 Ki = 8 nM T09572 CC1RB9 20608989 Ki = 190 nM T09572 C2H1YF 20608991 Ki = 25 nM T09572 C8Q0XO 20608992 Ki = 45 nM T09572 C8CUT0 20608996 Ki = 249 nM T09572 CVGY56 20609011 Ki = 63 nM T09572 C7N6XY 20609018 Ki = 30 nM T09572 C78UWI 20609028 Ki = 128 nM T09572 C2PF3N 20779393 Ki = 11 nM T09572 C3QGN7 20779413 Ki = 11 nM T09572 C1R4BJ 20779426 Ki = 300 nM T09572 C84VKA 20779429 Ki = 39 nM T09572 C9NK0T 20779441 Ki = 155 nM T09572 CW81IR 20779442 Ki = 281 nM T09572 CSV2M0 20817761 IC50 = 4 nM T09572 C85YPN 20817762 IC50 = 24 nM T09572 CO29QJ 20817763 IC50 = 16 nM T09572 C7X4ND 20817800 IC50 = 44 nM T09572 CS4AU1 20817821 IC50 = 5 nM T09572 CZC89U 20817846 IC50 = 88 nM T09572 CHB01Q 20817864 IC50 = 97 nM T09572 CGP04L 20877140 Ki = 20900 nM T09572 C9OMT8 21062990 IC50 = 65 nM T09572 CD90IG 21062991 IC50 = 140 nM T09572 CTCV19 21062998 IC50 = 7.4 nM T09572 CXC0F1 21062999 IC50 = 11 nM T09572 C01EQU 21063019 IC50 > 10000 nM T09572 C89XCE 21063022 IC50 > 1000 nM T09572 CJRD60 21101400 Ki = 39.81 nM T09572 CSU46X 21101402 Ki = 25.12 nM T09572 CXA8V1 21101416 Ki = 1000 nM T09572 CHZ4L6 21108056 IC50 = 11 nM T09572 CVS4D7 21108099 IC50 = 100 nM T09572 CD3O2Y 21108114 IC50 = 34 nM T09572 CYU8L1 21108117 IC50 = 20 nM T09572 C8R7XC 21108118 IC50 = 30 nM T09572 C48PMV 21939767 IC50 = 91 nM T09572 CIS5W2 21939881 IC50 = 230 nM T09572 CZ1GI7 21939887 IC50 = 350 nM T09572 CLD4C5 21939898 IC50 = 1.6 nM T09572 CC98QY 21939900 IC50 = 10000 nM T09572 CFS7G5 21939902 IC50 = 2.8 nM T09572 CDKT72 21939915 IC50 = 8.4 nM T09572 C4R6QP 21939935 IC50 = 380 nM T09572 CG63ZA 21939937 IC50 = 1.4 nM T09572 CI9R2D 21939940 IC50 = 380 nM T09572 CD8GZ7 21939950 IC50 = 2.2 nM T09572 CU7Z2B 21940008 IC50 = 17 nM T09572 C12GZE 21940052 IC50 = 190 nM T09572 CBQV01 21940083 IC50 = 1.9 nM T09572 C1MD6T 22018856 IC50 = 2 nM T09572 CK0GB9 22018896 IC50 = 12 nM T09572 CBO1J2 22018914 IC50 = 5 nM T09572 C0FJO5 22018919 IC50 = 10 nM T09572 CZUW58 22018932 IC50 = 5 nM T09572 C92HPN 22018944 IC50 = 1 nM T09572 C5SG9E 22018945 IC50 = 2 nM T09572 C2FYN1 22018957 IC50 = 0.5 nM T09572 CSQ1H0 22018964 IC50 = 1 nM T09572 CCQ6M7 22018997 IC50 = 6 nM T09572 CTQG86 22018999 IC50 = 2 nM T09572 C10MAZ 22251624 IC50 = 1.8 nM T09572 CY2PZ8 22254547 IC50 > 10000 nM T09572 C0G7FB 22254553 IC50 > 2000 nM T09572 CV64TI 22254570 IC50 = 808 nM T09572 COW3D8 22254571 IC50 = 137 nM T09572 CAL1Q8 22254581 IC50 = 60 nM T09572 CTH7J3 22254632 IC50 = 115 nM T09572 C16HAP 22348022 IC50 = 1.1 nM T09572 CCU37W 22348066 IC50 = 15 nM T09572 C82XIL 22348140 IC50 = 0.8 nM T09572 CY0WA7 22348155 IC50 = 1.2 nM T09572 C5PS4N 22348219 IC50 = 34 nM T09572 C6KJ0C 22348261 IC50 = 3 nM T09572 CJ67AV 22421739 IC50 = 6600 nM T09572 CITM21 22421741 IC50 = 727000 nM T09572 CO8AL0 22421743 IC50 = 251 nM T09572 CY39TI 22421749 IC50 = 230 nM T09572 C6TDY7 22421750 IC50 = 24800 nM T09572 C5UX4T 22422406 IC50 = 250 nM T09572 CTH09W 22427041 IC50 = 327 nM T09572 CLA5H0 23022394 IC50 = 32 nM T09572 CJ86XR 23022422 IC50 = 1.8 nM T09572 C26ESM 23022499 IC50 = 13 nM T09572 CT13GQ 23022509 IC50 = 4.3 nM T09572 C46HAR 23022536 IC50 = 1.7 nM T09572 CJS4U2 23022589 IC50 = 100 nM T09572 C81XUE 23027035 IC50 = 13 nM T09572 C5LCB2 23027181 IC50 = 58 nM T09572 CR5H1I 23027211 IC50 = 4.8 nM T09572 CC2L1B 23027245 IC50 = 16 nM T09572 CQ45SO 23027402 IC50 = 6.5 nM T09572 CG9M4Y 23027411 IC50 = 10 nM T09572 CC6R2O 23027527 IC50 = 6 nM T09572 CB4TK6 23027679 IC50 = 2.5 nM T09572 CLBE26 23027806 IC50 = 2.3 nM T09572 CW86DG 23027830 IC50 = 25 nM T09572 C9S3NP 23120512 IC50 = 4.4 nM T09572 C4Z9DB 23120540 IC50 = 1000 nM T09572 CJC1Y9 23120543 IC50 > 1000 nM T09572 C40PSL 23120550 IC50 = 2.5 nM T09572 CEH84I 23120564 IC50 = 4.8 nM T09572 C01LMH 23120572 IC50 = 2 nM T09572 C14ABC 23120575 IC50 = 6.8 nM T09572 C5RY1K 23120576 IC50 = 5.6 nM T09572 CV5ES9 23120580 IC50 = 17 nM T09572 CF67MJ 23120582 IC50 = 11 nM T09572 CYM4Q8 23120586 IC50 = 4 nM T09572 CK8Y2C 23532172 IC50 = 580 nM T09572 C1JOZ3 23532179 IC50 = 100 nM T09572 CJ6O3B 23532180 IC50 = 50 nM T09572 C45MIS 23532181 IC50 = 20 nM T09572 C3P9AQ 23567276 Ki = 240 nM T09572 CYQ35D 23567283 Ki = 130 nM T09572 CVO89E 23567290 Ki = 280 nM T09572 C9CRK8 23567310 Ki = 1641 nM T09572 C8OK2Q 23567355 Ki = 122 nM T09572 CK71DM 23567391 Ki = 205 nM T09572 CV5LK9 23567394 Ki = 1080 nM T09572 C7GP0L 23567408 Ki = 300 nM T09572 C0Q8AU 23567432 Ki = 1223 nM T09572 CL9B6S 23567477 Ki = 135 nM T09572 CX7QH0 23567513 Ki = 100 nM T09572 C2DIJ7 23573799 Ki = 21 nM T09572 CKXV10 23593464 IC50 = 3.4 nM T09572 C6L9NA 23593468 IC50 = 19 nM T09572 CNSZ98 23593471 IC50 = 1300 nM T09572 CO1D9V 23593472 IC50 = 220 nM T09572 C7R5TE 23593474 IC50 = 18 nM T09572 CQ80SP 23626228 Ki = 107 nM T09572 CX7B9D 23657037 IC50 = 29 nM T09572 CGI6M2 23658492 IC50 = 45.71 nM T09572 C4C3HR 24780883 IC50 = 4.4 nM T09572 CH15KN 24808474 IC50 = 3 nM T09572 C59IBZ 24857597 Ki = 9.7 nM T09572 CB4LY1 24857598 Ki = 2.6 nM T09572 C56KFT 24952055 EC50 = 60 nM T09572 C8TB2K 24952056 EC50 = 40 nM T09572 C2L9DI 24952417 EC50 = 20 nM T09572 C2GAX4 24952418 IC50 = 13 nM T09572 CX5QB0 24952419 EC50 = 20 nM T09572 C40XUR 24952765 IC50 = 3 nM T09572 CX83WL 24963343 Ki = 6 nM T09572 CD1AO6 25017033 Ki = 5.2 nM T09572 C1HK0Y 25017297 Ki = 38 nM T09572 CE7UZ8 25017298 Ki = 14 nM T09572 C9Y2LZ 25017299 Ki = 48 nM T09572 CIL04A 25017300 Ki = 28 nM T09572 CIL0E6 25017571 Ki = 4.2 nM T09572 C8FE1I 25017572 Ki = 6.1 nM T09572 C9X5AB 25018073 Ki = 59 nM T09572 C7ZR3G 25018075 Ki = 1679 nM T09572 CHQ86P 25054013 Ki = 3.1 nM T09572 C7EQ5T 25054288 Ki = 4.7 nM T09572 CCEY27 25054289 Ki = 11.2 nM T09572 C0PIZ8 25054550 Ki = 17.3 nM T09572 C20JHU 25054551 Ki = 33 nM T09572 CG8C7J 25054804 Ki = 12 nM T09572 C2FP5D 25056872 Ki = 24.3 nM T09572 C6Z3CE 25057124 Ki = 22.6 nM T09572 C0TYE6 25057388 Ki = 4.7 nM T09572 CE12CD 25057645 Ki = 43.4 nM T09572 C1K9VQ 25057911 Ki = 9.4 nM T09572 CH4PI7 25057913 Ki = 30.4 nM T09572 C8L6JE 25058425 IC50 = 1 nM T09572 C9WI7E 25110804 Ki = 3 nM T09572 CWVK74 25113835 IC50 = 3 nM T09572 CZH60W 25113838 IC50 = 8 nM T09572 CN8XF7 25114064 IC50 = 42 nM T09572 C9XL7R 25114065 IC50 = 56 nM T09572 CU10OY 25114067 IC50 = 4 nM T09572 CCQE40 25114068 IC50 = 16 nM T09572 CAW76X 25114286 IC50 = 1 nM T09572 CPD2X6 25114287 IC50 = 4 nM T09572 CCN5Y9 25114722 IC50 = 5 nM T09572 CCF8W5 25114723 IC50 = 19 nM T09572 CN5F7X 25114724 IC50 = 213 nM T09572 CS85TU 25114948 IC50 = 300 nM T09572 C38NAY 25115173 IC50 = 32 nM T09572 CPU90J 25115618 IC50 = 2 nM T09572 C9PQR0 25115619 IC50 = 10000 nM T09572 CT61UB 25115621 IC50 = 29 nM T09572 C1U6ES 25115852 IC50 = 74 nM T09572 CQLV30 25115854 IC50 = 10 nM T09572 CQ2U9N 25115855 IC50 = 5 nM T09572 C9V8QS 25115856 IC50 = 24 nM T09572 C57IBX 25116079 IC50 = 5 nM T09572 C0WG3P 25116082 IC50 = 3 nM T09572 CV6H9C 25116306 IC50 = 747 nM T09572 CMO7K5 25116307 IC50 = 7 nM T09572 C6X3MP 25116308 IC50 = 9 nM T09572 C9FOR4 25116309 IC50 = 60 nM T09572 CV71WE 25205149 Ki = 15 nM T09572 CSY73Q 25205150 Ki = 275 nM T09572 CI60SN 25205152 Ki = 13 nM T09572 C76DEF 25205153 Ki = 24 nM T09572 CS1MG9 25205316 Ki = 25 nM T09572 CK0AS8 25205317 Ki = 11 nM T09572 C8CY6O 25205318 Ki = 5 nM T09572 CY1M9Q 25205319 Ki = 3.4 nM T09572 CP6KO3 25205320 Ki = 23 nM T09572 C86NIQ 25205321 Ki = 26 nM T09572 C8YBX7 25205493 Ki = 539 nM T09572 C0ZBD5 25205827 Ki = 19 nM T09572 CWBS82 25205829 Ki = 5.8 nM T09572 C3DF9J 25206134 Ki = 272 nM T09572 CJ94XT 25206298 Ki = 99 nM T09572 C82KIH 25206454 Ki = 2.8 nM T09572 CP7EJ2 25206612 Ki = 3.9 nM T09572 C7XQG1 25206616 Ki = 16 nM T09572 CNQ57R 25207583 Ki > 1000 nM T09572 CRCF01 30979231 IC50 = 20000 nM T09572 C8ECM1 44143489 IC50 = 375 nM T09572 C2HY7L 44143490 IC50 = 365 nM T09572 CZ08GX 44143491 IC50 > 750 nM T09572 CU54OE 44143492 IC50 = 12 nM T09572 CIN95X 44143493 IC50 = 19 nM T09572 CRJ9P8 44143494 IC50 = 24 nM T09572 CYI1M0 44143495 IC50 = 4 nM T09572 CZ81KR 44143496 IC50 = 6.7 nM T09572 CSO6G3 44143497 IC50 = 27 nM T09572 C3J2EK 44143498 IC50 = 30 nM T09572 CN7G3T 44143499 IC50 = 23 nM T09572 C12KQP 44143500 IC50 = 135 nM T09572 CKN78A 44143501 IC50 = 428 nM T09572 C2U0LK 44143502 IC50 = 41 nM T09572 CS5K8F 44143503 IC50 = 3.1 nM T09572 C21VSY 44143504 IC50 = 8.8 nM T09572 C3BUH1 44143505 IC50 = 900 nM T09572 CMY45F 44188279 Ki = 0.18 nM T09572 CT48EW 44193451 IC50 = 41 nM T09572 CV5Y8E 44193624 IC50 = 28 nM T09572 CLXI76 44193625 IC50 = 22 nM T09572 CEWK48 44193792 Ki = 4.2 nM T09572 CUT6B9 44194383 Ki = 15 nM T09572 CW29OF 44194482 Ki = 168 nM T09572 C3WE8T 44194579 Ki = 7 nM T09572 CJQ9T7 44194749 Ki = 3.6 nM T09572 C5L6WO 44194849 Ki = 4.5 nM T09572 CXM7T5 44194850 Ki = 2.7 nM T09572 C1HJE6 44194853 Ki = 6.7 nM T09572 CG65PL 44194954 Ki = 4.2 nM T09572 C76ONX 44219756 IC50 = 0.09 nM T09572 C7QS6G 44250210 IC50 = 17 nM T09572 C64ASH 44250211 IC50 = 65 nM T09572 CPG1J4 44388058 Ki = 18500 nM T09572 C7P4WR 44388077 Ki = 22500 nM T09572 C4G8DW 44388096 IC50 = 6800 nM T09572 C9RT3L 44388141 Ki = 11000 nM T09572 CR0H7L 44388201 Ki = 84 nM T09572 CL93KW 44388215 Ki = 2.2 nM T09572 C8N3YM 44388219 Ki = 13 nM T09572 C4S8VZ 44388227 Ki = 5.2 nM T09572 CFJB61 44388263 Ki = 140 nM T09572 C2CT4S 44388265 Ki = 250 nM T09572 CFQ06P 44388271 Ki = 164 nM T09572 CRIH18 44388273 Ki > 10000 nM T09572 C0E8ON 44388277 Ki = 110 nM T09572 C3GEC4 44388280 Ki > 10000 nM T09572 CEQ6Y2 44388289 Ki = 13 nM T09572 C3HEM4 44388293 Ki = 12 nM T09572 CV70XA 44388294 Ki = 14 nM T09572 CSB35R 44388303 Ki = 16 nM T09572 CR1UM2 44388308 Ki > 10000 nM T09572 CT9V3N 44388309 Ki = 4300 nM T09572 CNA6Q3 44388311 Ki = 43 nM T09572 C3OUS8 44388314 Ki = 52 nM T09572 CI3O4R 44388345 Ki > 10000 nM T09572 CQWD51 44388355 Ki = 2400 nM T09572 CU6NJ1 44388365 Ki = 34 nM T09572 C4IF0M 44388368 Ki > 10000 nM T09572 CMV89X 44388380 Ki > 10000 nM T09572 C0I5RS 44388395 Ki > 10000 nM T09572 C8W2XV 44388409 Ki = 3.1 nM T09572 CNL7F3 44388417 Ki = 5.9 nM T09572 C52KHP 44388425 Ki = 31 nM T09572 CZH08E 44388427 Ki = 130 nM T09572 CI72GN 44388428 Ki = 5.5 nM T09572 CR51FP 44388442 Ki = 8.6 nM T09572 C51CXM 44388451 Ki = 3000 nM T09572 CT0F4Y 44388559 IC50 = 299 nM T09572 CLJ51W 44389354 Ki = 48 nM T09572 CY4H3V 44389375 Ki = 64 nM T09572 C9K6JZ 44389378 Ki = 67 nM T09572 C2FA9Y 44389379 Ki = 5.3 nM T09572 CDX17Y 44389390 Ki = 96 nM T09572 CTZ7M3 44389391 Ki = 7.3 nM T09572 CDW69Y 44389392 Ki = 20 nM T09572 CE8PA6 44389403 Ki = 18 nM T09572 C6UQ3V 44389404 Ki = 14 nM T09572 CKB9H8 44389405 Ki = 82 nM T09572 C92DLV 44389406 Ki = 31 nM T09572 C07KJE 44389422 Ki = 75 nM T09572 C0COV7 44389440 Ki = 83 nM T09572 CU2PK6 44389461 Ki = 1019 nM T09572 C7ME0A 44389484 Ki = 142 nM T09572 CVZ1J6 44389490 Ki = 22 nM T09572 C6ORK9 44389509 Ki = 57 nM T09572 CT58NE 44389521 Ki = 1043 nM T09572 C51XMO 44389526 Ki = 64 nM T09572 CH1SO4 44389533 Ki = 1096 nM T09572 CX2BO7 44389546 Ki = 456 nM T09572 CA6P7D 44389590 Ki = 98 nM T09572 CTMI35 44389604 Ki = 460 nM T09572 CE25YT 44390369 IC50 = 5800 nM T09572 CFH3C2 44390385 IC50 = 960 nM T09572 C6LJC2 44390456 IC50 = 5600 nM T09572 CHGY52 44390499 IC50 = 1500 nM T09572 CK7G4S 44390706 IC50 = 5.9 nM T09572 C69OXU 44390707 IC50 = 170 nM T09572 CS16BQ 44390710 IC50 = 15 nM T09572 C9GTA2 44390713 IC50 = 9.5 nM T09572 C0B5MU 44390715 IC50 = 5 nM T09572 CBA36Y 44390726 IC50 = 2 nM T09572 C9GTB7 44390730 IC50 = 10 nM T09572 CPQ63J 44390733 IC50 = 35 nM T09572 CHO04I 44390742 IC50 = 9.4 nM T09572 CHL23R 44390748 IC50 = 1200 nM T09572 CZN1R2 44390750 IC50 = 4.5 nM T09572 C3TEB2 44390752 IC50 = 320 nM T09572 C85MAY 44390768 IC50 = 6.8 nM T09572 C5BA0Y 44390778 IC50 = 4.6 nM T09572 CN3U4V 44390787 IC50 = 38 nM T09572 CT8D4X 44393379 IC50 = 124 nM T09572 CVS4K0 44394569 IC50 = 290 nM T09572 C9GI5M 44394572 IC50 = 80 nM T09572 CAN86X 44394573 IC50 = 50 nM T09572 CSK4Z8 44394587 IC50 = 660 nM T09572 C9RD7J 44394591 IC50 = 10 nM T09572 C8HU9L 44394592 IC50 = 90 nM T09572 C79UNY 44394596 IC50 = 730 nM T09572 C63GOP 44394602 IC50 > 2000 nM T09572 CQ1M6N 44394604 IC50 = 2170 nM T09572 C24HUY 44394605 IC50 = 360 nM T09572 C9GY1S 44394606 IC50 = 30 nM T09572 C6SGC9 44394607 IC50 = 530 nM T09572 CSF04I 44394609 IC50 = 1 nM T09572 CA1H6D 44394611 IC50 = 5 nM T09572 C9Q1WO 44394628 IC50 > 2000 nM T09572 C67EUA 44394638 IC50 = 520 nM T09572 CC6HG0 44394639 IC50 = 70 nM T09572 CPK8S4 44394643 IC50 > 2000 nM T09572 CLRE30 44394644 IC50 = 340 nM T09572 C0XFU6 44394650 IC50 = 1 nM T09572 CJ78KQ 44394676 IC50 = 10 nM T09572 CY3ZO1 44394683 IC50 = 10 nM T09572 CHL3U0 44394684 IC50 = 580 nM T09572 CZ0B4R 44394697 IC50 > 10000 nM T09572 CFXI09 44394698 IC50 = 7 nM T09572 CW8RI7 44394705 IC50 = 38.6 nM T09572 CV7M6B 44394715 IC50 > 2000 nM T09572 CQ8IE0 44394725 IC50 = 7 nM T09572 CNHG32 44394726 IC50 = 2 nM T09572 CGFO71 44394763 IC50 = 10 nM T09572 CICX23 44394764 IC50 = 140 nM T09572 C57FPS 44394769 IC50 = 1.2 nM T09572 C19TJC 44394770 IC50 = 2.7 nM T09572 CJTQ96 44394774 IC50 = 306 nM T09572 C4HGJ3 44394780 IC50 > 10000 nM T09572 C1M2VQ 44394791 IC50 > 2000 nM T09572 C25PUB 44394792 IC50 = 6 nM T09572 C1NH3W 44394793 IC50 > 2000 nM T09572 CT9R3J 44394798 IC50 = 2.2 nM T09572 CLPC86 44394799 IC50 = 20.5 nM T09572 C0AQ9Y 44394800 IC50 = 1 nM T09572 C0P3SE 44394807 IC50 = 210 nM T09572 CBH9C8 44394824 IC50 = 5 nM T09572 CZN6A8 44394825 IC50 = 149 nM T09572 C6X8ZK 44394826 IC50 = 41 nM T09572 CP39MA 44394854 IC50 = 1640 nM T09572 CQ6CE2 44394855 IC50 = 240 nM T09572 C1SGN4 44394856 IC50 = 5 nM T09572 C0L8SO 44394858 IC50 > 2000 nM T09572 C35PHE 44394859 IC50 = 50 nM T09572 C6FVP1 44394860 IC50 = 30 nM T09572 CX1ZS5 44394861 IC50 = 13000 nM T09572 CHC4X1 44394863 IC50 > 2000 nM T09572 CM8P9R 44394864 IC50 = 25.6 nM T09572 CMKO91 44394866 IC50 = 10 nM T09572 C4BXR3 44394877 IC50 > 2000 nM T09572 CMR24H 44394881 IC50 > 2000 nM T09572 CYS57R 44394882 IC50 > 2000 nM T09572 CBUM52 44394883 IC50 = 80 nM T09572 COQ63G 44394890 IC50 = 100 nM T09572 CX5F2L 44394891 IC50 = 2 nM T09572 C3OVG9 44394906 IC50 > 2000 nM T09572 CTE35F 44394907 IC50 = 5.3 nM T09572 CG34PA 44394908 IC50 = 540 nM T09572 C1RD0C 44394909 IC50 = 110 nM T09572 C9I6AV 44394910 IC50 = 4700 nM T09572 C0KLA9 44394921 IC50 = 640 nM T09572 CI7RP8 44394922 IC50 = 30 nM T09572 CQ2Z0P 44394925 IC50 = 3200 nM T09572 C8G5RJ 44394926 IC50 = 960 nM T09572 C8O1VN 44394931 IC50 = 7900 nM T09572 C69ZSF 44394939 IC50 = 370 nM T09572 C90YMX 44394943 IC50 > 10000 nM T09572 CW3NK2 44394944 IC50 = 5900 nM T09572 CAOI08 44394946 IC50 = 130 nM T09572 C30MBJ 44394948 IC50 = 200 nM T09572 CTE91Q 44394958 IC50 = 1970 nM T09572 C2KM0Q 44394959 IC50 = 20 nM T09572 CB8NG3 44394961 IC50 = 640 nM T09572 C9R8NZ 44394966 IC50 = 11000 nM T09572 C49NZX 44394972 IC50 = 2500 nM T09572 CBN80V 44394973 IC50 = 2450 nM T09572 C0R9QC 44394977 IC50 > 100000 nM T09572 C8JO6R 44394978 IC50 > 100000 nM T09572 CE7HN6 44394983 IC50 = 1480 nM T09572 C1SQA9 44394986 IC50 = 250 nM T09572 C5I0CR 44394987 IC50 = 18000 nM T09572 CO5X7L 44394997 IC50 = 3500 nM T09572 CNW8A9 44394998 IC50 = 710 nM T09572 C7NM0Q 44394999 IC50 = 1920 nM T09572 C3MB6U 44395000 IC50 > 100000 nM T09572 C1JR7F 44395001 IC50 = 5800 nM T09572 C8Z5WY 44395007 IC50 = 1900 nM T09572 CY45BV 44395008 IC50 > 100000 nM T09572 CZ6G8X 44395012 IC50 = 15800 nM T09572 CKXF13 44395013 IC50 > 100000 nM T09572 CSUM01 44395019 IC50 = 140 nM T09572 CEC3Z2 44395021 IC50 = 3900 nM T09572 CGY19E 44395022 IC50 = 4800 nM T09572 CUQ04R 44395076 IC50 = 5820 nM T09572 CC48AI 44395082 IC50 = 8800 nM T09572 C67MQP 44396196 IC50 = 8200 nM T09572 CDH9A0 44396800 Ki = 3 nM T09572 C1Q3KE 44396807 Ki = 2 nM T09572 CK24UL 44396904 Ki = 310 nM T09572 C06GEV 44396952 IC50 = 90 nM T09572 C34UGT 44396975 Ki = 63 nM T09572 C3QE2M 44396985 Ki = 61 nM T09572 CJO81G 44397008 IC50 = 50 nM T09572 C5LY2S 44397009 IC50 = 110 nM T09572 CG9L7A 44397018 Ki = 3 nM T09572 CCO72P 44397026 IC50 = 50 nM T09572 C4V9XD 44397031 Ki = 10 nM T09572 C1YAO3 44397033 IC50 = 4300 nM T09572 CR7I9Z 44397048 IC50 = 230 nM T09572 C6DTI3 44397052 IC50 > 2000 nM T09572 CXP1H2 44397086 Ki = 3 nM T09572 CZXN03 44397087 Ki = 7 nM T09572 CQZ9M6 44397095 Ki = 3 nM T09572 C5NR9X 44397099 IC50 = 5190 nM T09572 CSY42I 44397103 Ki = 6000 nM T09572 C0DE8P 44397114 Ki = 1 nM T09572 C8VPO7 44397120 IC50 = 510 nM T09572 CJ3HW9 44397126 Ki = 190 nM T09572 C1O0AT 44397127 IC50 = 50 nM T09572 CVD8J2 44397128 IC50 = 60 nM T09572 CN26GO 44397145 Ki = 1800 nM T09572 C2I9VT 44397163 Ki = 37 nM T09572 CD15XJ 44397167 Ki = 19 nM T09572 C41YAD 44397168 Ki = 3300 nM T09572 CT3IG2 44397174 IC50 > 10000 nM T09572 C0IOB2 44397175 IC50 = 300 nM T09572 CM83JY 44397194 IC50 = 20 nM T09572 CO8EI5 44397200 Ki = 320 nM T09572 CFY3U9 44397202 IC50 = 10 nM T09572 CR6YG0 44397203 Ki > 10000 nM T09572 C1MQ3T 44397215 IC50 = 320 nM T09572 CQ73UR 44397221 IC50 = 90 nM T09572 CL8IY3 44397227 Ki = 900 nM T09572 C4CQT2 44397243 Ki = 3400 nM T09572 C58DRB 44397245 Ki = 4 nM T09572 CZ30KL 44397254 Ki = 3 nM T09572 C92RCK 44397262 IC50 = 30 nM T09572 CB2ZN8 44397263 IC50 > 2000 nM T09572 C5IXH8 44397273 Ki = 5 nM T09572 CSI3G7 44397278 IC50 = 490 nM T09572 CX3ED1 44397288 Ki = 2 nM T09572 C6DZQ0 44397293 Ki = 4 nM T09572 CFP9Y1 44397302 Ki = 14 nM T09572 CZK80P 44397303 IC50 = 1040 nM T09572 CZKY29 44397309 Ki = 12 nM T09572 C7R3EV 44397310 IC50 = 110 nM T09572 C9IZO5 44397312 Ki = 2400 nM T09572 CLC7N8 44397323 Ki = 150 nM T09572 CP6I4E 44397329 IC50 = 1950 nM T09572 CB5ZQ7 44397330 IC50 > 2000 nM T09572 C9X3JV 44397350 Ki = 16 nM T09572 CV72OU 44397425 IC50 = 90 nM T09572 C82FLB 44397454 IC50 = 2990 nM T09572 CMJ67E 44397476 IC50 = 3 nM T09572 C9AM8F 44397477 IC50 > 2000 nM T09572 CSRG09 44397479 Ki = 2 nM T09572 CI2VP7 44397480 IC50 = 320 nM T09572 C6LJB5 44397497 Ki = 5 nM T09572 CS07BY 44397560 IC50 = 120 nM T09572 CR2DJ8 44397605 IC50 = 1610 nM T09572 C5B2YW 44397606 IC50 = 280 nM T09572 CPB7Q4 44397630 Ki = 2 nM T09572 CS4IW6 44397636 IC50 = 330 nM T09572 C0QM4W 44397716 IC50 = 1560 nM T09572 C4HR6C 44399507 Ki = 7.1 nM T09572 CH39TA 44399610 Ki = 2.7 nM T09572 CL06NB 44401276 IC50 > 10000 nM T09572 CDS4Y1 44401368 IC50 = 6700 nM T09572 C93HAW 44401395 IC50 = 2700 nM T09572 C4RN8A 44401449 IC50 = 83 nM T09572 C49USD 44401460 IC50 > 10000 nM T09572 CHGX51 44401508 IC50 = 2900 nM T09572 CIKD90 44401552 IC50 = 2900 nM T09572 C8VQ3B 44401591 IC50 = 1900 nM T09572 CT46VH 44401616 IC50 = 810 nM T09572 CIXE76 44401626 IC50 = 140 nM T09572 CER15G 44401671 IC50 = 6000 nM T09572 CR1D2K 44402861 Ki > 100000 nM T09572 CW4Z1L 44403445 IC50 = 370 nM T09572 C4UDG8 44403454 IC50 = 370 nM T09572 CT6IX9 44403467 IC50 = 6 nM T09572 CBN6J3 44403468 IC50 = 20 nM T09572 CRWC57 44403471 IC50 = 110 nM T09572 CT0U6C 44403472 IC50 = 80 nM T09572 C5Q0OF 44403473 IC50 = 2010 nM T09572 CJ1U2V 44403474 IC50 = 30 nM T09572 C3Y2ST 44403477 IC50 = 9 nM T09572 CHZI37 44403478 IC50 = 680 nM T09572 C1JRE0 44403479 IC50 = 70 nM T09572 CF6QJ8 44403480 IC50 = 30 nM T09572 C1FOP8 44403483 IC50 = 560 nM T09572 CT2GD3 44403484 IC50 = 260 nM T09572 C1P5JF 44403486 IC50 = 1980 nM T09572 CF7Z6C 44403487 IC50 = 20 nM T09572 CE27XC 44403490 IC50 = 160 nM T09572 CI4S5Z 44403491 IC50 = 220 nM T09572 C5I7ZO 44403492 IC50 = 160 nM T09572 CUZH85 44403493 IC50 = 20 nM T09572 CWCJ58 44403498 IC50 = 90 nM T09572 C6OWP7 44403499 IC50 = 50 nM T09572 CE9W5D 44403500 IC50 = 410 nM T09572 CSP0T1 44403501 IC50 = 60 nM T09572 CXH8U1 44403505 IC50 = 40 nM T09572 CLK27J 44403506 IC50 = 30 nM T09572 C5D1NZ 44403507 IC50 = 20 nM T09572 CWP5R7 44403511 IC50 = 9 nM T09572 C39ZVY 44403513 IC50 = 9 nM T09572 CHS0Y9 44403516 IC50 = 70 nM T09572 C1V6BP 44403517 IC50 = 4 nM T09572 CEJF46 44403518 IC50 = 6 nM T09572 C5UG0H 44403522 IC50 = 20 nM T09572 C8I1JU 44403523 IC50 = 10 nM T09572 C41YLX 44403524 IC50 = 60 nM T09572 CNW95X 44403527 IC50 = 90 nM T09572 CFS35E 44403528 IC50 = 50 nM T09572 CB02DH 44403533 IC50 = 390 nM T09572 C65YJN 44403535 IC50 = 190 nM T09572 C4U3FN 44403538 IC50 = 70 nM T09572 C19IBE 44403539 IC50 = 140 nM T09572 C2OMY6 44403547 IC50 = 410 nM T09572 C0TO1J 44403548 IC50 = 10 nM T09572 CQ08CG 44403733 IC50 = 1800 nM T09572 CZE89R 44403747 IC50 = 95 nM T09572 CR7BQ9 44403748 IC50 = 438 nM T09572 CQ4W5H 44403749 IC50 = 442 nM T09572 C81ISR 44403750 IC50 = 224 nM T09572 CLGA83 44403765 IC50 = 6.1 nM T09572 CBA93S 44403849 IC50 > 10000 nM T09572 CD3FE4 44405399 Ki = 287 nM T09572 CQDZ37 44405408 IC50 = 50 nM T09572 C2DAJ8 44405409 IC50 = 330 nM T09572 CA75TW 44405412 IC50 = 5200 nM T09572 C8A2RI 44405415 IC50 = 30 nM T09572 CW5KU8 44405417 Ki = 159 nM T09572 CVP74K 44405418 Ki = 48 nM T09572 C0N4IL 44405421 Ki = 48 nM T09572 C5F2LI 44405430 IC50 = 4500 nM T09572 C5T9CU 44405431 IC50 = 1380 nM T09572 C79OPX 44405435 Ki = 23 nM T09572 CDJF17 44405436 Ki = 70 nM T09572 CT42XM 44405437 Ki = 151 nM T09572 CF57KL 44405439 Ki = 18 nM T09572 C37XOM 44405444 Ki = 76 nM T09572 C74WZI 44405458 IC50 > 2000 nM T09572 C5V3EU 44405459 IC50 = 200 nM T09572 CW80JL 44405461 Ki = 16 nM T09572 CBS4P2 44405463 IC50 = 50 nM T09572 C5KLO6 44405464 IC50 = 5 nM T09572 CJRW91 44405468 IC50 = 40 nM T09572 C29JXR 44405477 IC50 = 850 nM T09572 C27IXA 44405481 IC50 = 1060 nM T09572 CB78MN 44405482 IC50 = 70 nM T09572 C9V7MC 44405486 IC50 = 520 nM T09572 CX64ET 44405487 IC50 = 220 nM T09572 C16CPT 44405488 IC50 = 280 nM T09572 CN4KP9 44405501 Ki = 31 nM T09572 C1T3AR 44405517 IC50 = 440 nM T09572 CTW14K 44405518 IC50 = 1820 nM T09572 CC38GX 44405519 IC50 = 70 nM T09572 CJ2OV1 44405557 IC50 = 930 nM T09572 CH7XF0 44405560 IC50 = 20 nM T09572 C1GA2K 44405570 IC50 = 50 nM T09572 CN2W1H 44405612 IC50 = 20 nM T09572 CB79VL 44405618 IC50 = 20 nM T09572 CTI27L 44405619 IC50 = 560 nM T09572 CU08QO 44405645 IC50 = 40 nM T09572 C3H4OS 44405646 IC50 = 20 nM T09572 CD4H0S 44405651 IC50 = 9 nM T09572 C7DY8R 44407478 IC50 > 10000 nM T09572 C7TXS3 44407479 IC50 = 2540 nM T09572 CY70WO 44407629 IC50 = 2 nM T09572 C29UTK 44407667 IC50 = 17 nM T09572 CBL19U 44407710 IC50 = 3.7 nM T09572 CBU72F 44407711 IC50 = 83 nM T09572 C0BY6Z 44407836 IC50 = 4.7 nM T09572 CP5D3Y 44407860 IC50 = 91 nM T09572 C3JLT1 44407870 IC50 = 14 nM T09572 C8TP0Q 44407875 IC50 = 3.7 nM T09572 C8FTO7 44407934 IC50 = 2100 nM T09572 C7MEY5 44407944 IC50 = 33 nM T09572 CRS49X 44407950 IC50 = 2760 nM T09572 CB0LM3 44407951 IC50 = 125 nM T09572 CUEI62 44407956 IC50 = 44 nM T09572 CU34HG 44407965 IC50 > 10000 nM T09572 CV9R8K 44407966 IC50 = 105 nM T09572 CYOP29 44407967 IC50 = 474 nM T09572 CK13PD 44407989 IC50 = 6970 nM T09572 CF3X7M 44407990 IC50 > 10000 nM T09572 CR8B7D 44407991 IC50 = 5.7 nM T09572 CWUS42 44407997 IC50 = 9460 nM T09572 C70DWK 44408013 IC50 = 23 nM T09572 CG9HB0 44408014 IC50 = 3280 nM T09572 CA72TP 44408020 IC50 = 568 nM T09572 C6IT1B 44408027 IC50 = 15 nM T09572 CVS92Y 44408028 IC50 = 7.1 nM T09572 CP8A0C 44408081 IC50 = 210 nM T09572 CG5JN8 44408093 IC50 = 162 nM T09572 CT9Q7Z 44408099 IC50 = 271 nM T09572 CU4JK5 44408108 IC50 = 5.3 nM T09572 COGK24 44408109 IC50 = 2.4 nM T09572 CBJY53 44408117 IC50 = 18 nM T09572 CUS7R1 44409479 Ki = 15 nM T09572 C1DTI6 44409527 Ki = 15.1 nM T09572 CKEP27 44409689 Ki = 974 nM T09572 CYP37K 44410821 IC50 = 5 nM T09572 CJI8T3 44410823 IC50 = 62 nM T09572 C01JXU 44410838 IC50 = 72 nM T09572 C1LYC9 44410849 IC50 = 0.9 nM T09572 CGF17I 44410876 IC50 = 12 nM T09572 CF0O7N 44410878 IC50 = 34 nM T09572 CL1XV7 44410904 IC50 = 53 nM T09572 C4P5TW 44410944 IC50 = 12 nM T09572 CFSD50 44412624 Ki = 51 nM T09572 C1CPT2 44412682 Ki = 46 nM T09572 CG6J5R 44412683 Ki = 92 nM T09572 CQ7P1N 44412686 Ki = 48 nM T09572 CVJF97 44412837 Ki = 26 nM T09572 CRPQ04 44412852 Ki = 1.2 nM T09572 CV1ZX4 44412960 Ki = 193 nM T09572 C43CDI 44413138 Ki = 132 nM T09572 C2SOJ1 44413259 Ki = 95 nM T09572 C8OT1W 44413271 Ki = 77 nM T09572 C1AJ8V 44413283 Ki = 3.9 nM T09572 CHG2A7 44413297 Ki = 10.3 nM T09572 C6V5YR 44413299 Ki = 31 nM T09572 C7PC5N 44413309 Ki = 26 nM T09572 C4YMR8 44413312 Ki = 31 nM T09572 CXC97Y 44413326 IC50 = 130 nM T09572 C0IBW4 44413345 Ki = 464 nM T09572 C9U8FY 44413382 Ki = 7.2 nM T09572 CDG5Q2 44413398 Ki = 99 nM T09572 C64UZT 44413428 Ki = 174 nM T09572 CK8C1H 44413470 Ki = 15.5 nM T09572 C34LQB 44413471 Ki = 45 nM T09572 CG7KI9 44413472 Ki = 20 nM T09572 CGY94E 44413473 Ki = 10.1 nM T09572 C7X5HF 44413474 Ki = 10.3 nM T09572 CCKU08 44413475 Ki = 15 nM T09572 CS5WN4 44413480 Ki = 64 nM T09572 CB5GI6 44414309 Ki = 3 nM T09572 C3IB1L 44414310 Ki = 8.8 nM T09572 C79XQN 44414318 Ki = 4.4 nM T09572 CJ1V0F 44414319 Ki = 13 nM T09572 C9MV4A 44414327 Ki = 10 nM T09572 CZI1Y9 44414342 Ki = 24 nM T09572 CS5VO0 44414356 Ki = 24 nM T09572 C2XK7V 44414357 Ki = 14 nM T09572 C5M6ZU 44414368 Ki = 120 nM T09572 CIJ8D5 44414375 Ki = 4.8 nM T09572 C52EQN 44414391 Ki = 7.2 nM T09572 CMV9H6 44414392 Ki = 13 nM T09572 C2N7PZ 44414399 Ki = 3.1 nM T09572 CE36JR 44414432 Ki = 4.1 nM T09572 C2BXH0 44414444 Ki = 25 nM T09572 C1X5TM 44414451 Ki = 2 nM T09572 CXQK29 44414455 Ki = 18 nM T09572 C3CA5G 44414461 Ki = 57 nM T09572 CU8VR5 44414464 Ki = 15.1 nM T09572 C2D9BH 44414465 Ki = 115 nM T09572 CEL21T 44414466 Ki = 28 nM T09572 CKB82R 44414475 Ki = 2.1 nM T09572 CB5F4W 44414481 Ki = 29 nM T09572 CY1VH7 44414483 Ki = 28 nM T09572 C96BYD 44414497 Ki = 1.6 nM T09572 C3DP8X 44414499 Ki = 19 nM T09572 CHG0S9 44414506 Ki = 56 nM T09572 CH7P4X 44414518 Ki = 10 nM T09572 CG7J0K 44414520 Ki = 1.4 nM T09572 CTE9S2 44414522 Ki = 138 nM T09572 CX2F6A 44414528 Ki = 8.6 nM T09572 CJ0FN4 44414540 Ki = 7.1 nM T09572 CL0H1X 44414542 Ki = 78 nM T09572 CR1CS5 44414552 Ki = 43 nM T09572 CBJF79 44414570 Ki = 16 nM T09572 C7E6RX 44414571 Ki = 4.7 nM T09572 C2I9CV 44414576 Ki = 5.4 nM T09572 CSEN81 44414589 Ki = 5.4 nM T09572 C97FHL 44414600 Ki = 2.6 nM T09572 C10IPW 44414601 Ki = 46 nM T09572 CS1B0T 44414606 Ki = 15 nM T09572 CG6R9J 44414622 Ki = 2.7 nM T09572 C6E7RW 44414649 Ki = 8.5 nM T09572 C9KHE1 44414650 Ki = 17 nM T09572 C40PGW 44414651 Ki = 139 nM T09572 CWIM26 44414654 Ki = 6.8 nM T09572 CGI4F7 44415364 Ki = 10.47 nM T09572 CPJ4V5 44415378 Ki = 18.62 nM T09572 CWJE81 44415381 Ki = 630 nM T09572 CC25QM 44415385 Ki = 4786.3 nM T09572 CMV57G 44415389 Ki = 13 nM T09572 CN1M4Z 44415396 Ki = 398.11 nM T09572 CRHQ87 44415401 Ki = 39.81 nM T09572 C29JXK 44415402 Ki = 23.99 nM T09572 C1T2DR 44415407 Ki = 630.96 nM T09572 C83UJR 44415409 Ki = 51 nM T09572 CRUT01 44415410 Ki = 53 nM T09572 C75SYA 44415413 Ki = 16 nM T09572 CR34JS 44415414 Ki = 41.69 nM T09572 CH91UG 44415419 Ki = 1000 nM T09572 C9WRN5 44415425 Ki = 33.88 nM T09572 C7VT5P 44415426 Ki = 53.7 nM T09572 CV9S7J 44415427 Ki = 51 nM T09572 CFZ90J 44415431 Ki = 43.65 nM T09572 C09SEJ 44415439 Ki = 38 nM T09572 C0TZ3O 44415440 Ki = 28.84 nM T09572 CPM3R9 44415446 Ki = 28 nM T09572 C7NH2F 44415451 Ki = 8 nM T09572 C5IV2C 44415459 Ki = 33 nM T09572 CL1KM8 44415460 Ki = 25.7 nM T09572 CGHJ29 44415461 Ki = 14 nM T09572 COW3P7 44415462 Ki = 26.92 nM T09572 COLW46 44415463 Ki = 47.86 nM T09572 C5Z9UM 44415465 Ki > 10000 nM T09572 CU2LQ5 44415466 Ki = 3981.07 nM T09572 CX76TL 44415467 Ki = 73 nM T09572 CTS2L6 44415483 Ki = 16.6 nM T09572 CI05LE 44415491 Ki = 22 nM T09572 CQKB40 44415501 Ki = 109.65 nM T09572 CO8X2W 44415512 Ki = 180 nM T09572 CN9GY5 44415516 Ki = 48.98 nM T09572 C0OG4J 44415524 Ki = 14 nM T09572 C86OHN 44415525 Ki = 20.89 nM T09572 CL17YI 44415526 Ki = 19.95 nM T09572 CY6C2D 44415533 Ki = 18.62 nM T09572 C6HSF3 44416140 Ki = 41 nM T09572 CZG1L2 44416172 Ki = 77 nM T09572 CZ38VN 44416173 Ki = 87 nM T09572 CT79MH 44416174 Ki = 799 nM T09572 C9FT7Y 44416178 Ki = 46 nM T09572 CV8JU0 44416212 IC50 = 25.12 nM T09572 CN78HS 44416223 Ki = 95 nM T09572 CKD7I4 44416224 Ki = 191 nM T09572 CKP27D 44416225 Ki = 77 nM T09572 C58WVT 44416231 IC50 = 5.012 nM T09572 CE93MV 44416232 IC50 = 199.53 nM T09572 CAO4W7 44416255 IC50 = 1584.89 nM T09572 C5B3IQ 44416261 Ki = 24 nM T09572 CBC5O3 44416272 IC50 = 25.12 nM T09572 CITW25 44416275 Ki = 927 nM T09572 C2AO6C 44416287 Ki = 718 nM T09572 C9F2PM 44416296 IC50 = 19.95 nM T09572 C0LQ3D 44416297 IC50 = 1258.93 nM T09572 CVXO51 44416302 IC50 = 5.012 nM T09572 CD9J7M 44416303 IC50 = 3162.28 nM T09572 CGC7V2 44416310 Ki = 108 nM T09572 C8IPQ2 44416311 Ki = 73 nM T09572 CUN0J8 44416314 IC50 = 1.259 nM T09572 CKJ1N7 44416315 IC50 = 6.31 nM T09572 CFI41O 44416316 IC50 = 1.585 nM T09572 CN4O2X 44416322 Ki = 43 nM T09572 CHL8D7 44416336 IC50 = 1 nM T09572 CB7H1J 44416337 IC50 = 2.512 nM T09572 CV13DW 44416344 Ki > 1000 nM T09572 C8XCL1 44416346 Ki = 455 nM T09572 C5SI3O 44416348 IC50 = 12.59 nM T09572 CRJ97I 44416350 IC50 = 100 nM T09572 CPUD71 44416357 Ki = 115 nM T09572 CLXG42 44416362 IC50 = 3981.07 nM T09572 CF19EV 44416363 IC50 = 125.89 nM T09572 CU64KI 44416364 Ki = 35 nM T09572 CX59PC 44416376 IC50 = 6.31 nM T09572 CA98PR 44416377 IC50 = 3.162 nM T09572 CQV5J1 44416381 Ki = 168 nM T09572 C4BJR5 44416388 Ki = 25.12 nM T09572 CB7P8K 44416389 Ki = 158.49 nM T09572 CP7H2Q 44416390 Ki = 5.012 nM T09572 CF0BM8 44416391 Ki = 414 nM T09572 CRO95N 44416402 Ki = 398.11 nM T09572 CFUA54 44416405 Ki = 4.9 nM T09572 CAE2D0 44416428 Ki = 251.19 nM T09572 C8P2XM 44416451 Ki < 6309.57 nM T09572 C32IYJ 44416472 Ki = 251.19 nM T09572 C2F3EY 44416474 Ki = 102 nM T09572 C70GBX 44416475 Ki = 1408 nM T09572 CNL35D 44416479 Ki = 31.62 nM T09572 CVF1B8 44416480 Ki = 251.19 nM T09572 C4AOQ9 44416495 Ki = 79.43 nM T09572 C4SP0A 44416498 Ki = 39.81 nM T09572 C42WEU 44416502 Ki = 50.12 nM T09572 C7IB2N 44416503 Ki = 50.12 nM T09572 CVA3M1 44416504 Ki < 10000 nM T09572 C15TAE 44416521 Ki = 39.81 nM T09572 CO0QD7 44416522 Ki = 2511.89 nM T09572 CEH6A9 44416536 Ki < 10000 nM T09572 C4L8UP 44416539 Ki = 39.81 nM T09572 C79YPB 44416540 Ki < 10000 nM T09572 CPE1L9 44416553 Ki = 50.12 nM T09572 C3UIT1 44416554 Ki = 79.43 nM T09572 CF0E9H 44416559 Ki = 125.89 nM T09572 C1VT2K 44416561 Ki = 63.1 nM T09572 CBP2N5 44416579 Ki = 199.53 nM T09572 C75GYI 44416580 Ki = 501.19 nM T09572 CJ4D5N 44416584 Ki = 79.43 nM T09572 C9CD8Z 44416585 Ki = 158.49 nM T09572 C6H0BL 44416586 Ki = 25.12 nM T09572 C9VS6Z 44416587 Ki = 1153 nM T09572 C87FGN 44416606 Ki = 50.12 nM T09572 CAF18G 44416607 Ki = 60 nM T09572 CC1Y0W 44416623 Ki = 5011.87 nM T09572 CZ7W0E 44416624 Ki < 10000 nM T09572 C4RS6H 44416627 Ki = 310 nM T09572 CF3HG1 44416628 Ki = 3544 nM T09572 C8A5HU 44416629 Ki = 31 nM T09572 CT4DU9 44416650 Ki = 20119 nM T09572 C7JV9E 44416651 Ki = 0.631 nM T09572 CFZ0H1 44416664 Ki = 63.1 nM T09572 CN3UQ7 44416670 Ki = 1.995 nM T09572 C8ZI4H 44416671 Ki = 0.9 nM T09572 CGB3S0 44416689 Ki = 803 nM T09572 C6BD0R 44416711 Ki = 199.53 nM T09572 CE5MY9 44416713 Ki = 195 nM T09572 CSRK76 44416714 Ki = 19.95 nM T09572 C1YV3D 44416735 Ki = 79.43 nM T09572 CV7BA5 44416736 Ki < 10000 nM T09572 C0V4BK 44416737 Ki = 142 nM T09572 C95RCN 44416738 Ki = 310 nM T09572 CX0R4H 44416751 IC50 = 100 nM T09572 CJ08ZR 44416753 Ki = 25 nM T09572 C3O7GK 44416757 Ki = 3.981 nM T09572 CA28XT 44416777 IC50 = 5.012 nM T09572 C16WUL 44416781 Ki = 3600 nM T09572 CY6T2S 44416782 Ki = 18 nM T09572 C0SX4T 44416786 Ki = 12.59 nM T09572 CK1UJ6 44416797 Ki = 1000 nM T09572 CD2U4N 44416798 Ki = 316.23 nM T09572 C9R1UT 44416800 Ki = 1.585 nM T09572 CMHX86 44416801 Ki = 5 nM T09572 CGMX09 44416814 IC50 = 6.31 nM T09572 CL53YH 44416815 IC50 = 6.31 nM T09572 CAT0B7 44416816 Ki = 2511.89 nM T09572 C4OX7Y 44416817 Ki = 1995.26 nM T09572 CSRH79 44416828 IC50 = 25.12 nM T09572 C0VJ9B 44416833 Ki = 133 nM T09572 C94QFT 44416837 IC50 = 1.995 nM T09572 CAZW24 44416838 IC50 = 5.012 nM T09572 CD9Q0Y 44416839 Ki = 136 nM T09572 C81JPB 44416840 Ki = 110 nM T09572 CRMS24 44416841 Ki = 794.33 nM T09572 C0WCI8 44416845 IC50 = 6.31 nM T09572 C7SIK0 44416851 IC50 = 31.62 nM T09572 CP64OW 44416857 IC50 = 1.585 nM T09572 C1UMD2 44416858 IC50 = 31.62 nM T09572 C4W8ST 44416859 Ki = 1.9 nM T09572 CG46MT 44416862 Ki = 6 nM T09572 CKNF68 44416871 IC50 = 19.95 nM T09572 CI35XF 44416872 IC50 = 5.012 nM T09572 CP4YB0 44416875 IC50 = 3.981 nM T09572 CT62LG 44416877 Ki = 2.4 nM T09572 C8ELH9 44416880 Ki = 500 nM T09572 C76SRF 44416881 Ki = 2 nM T09572 CWS2B9 44416890 IC50 = 3.162 nM T09572 CDNH81 44416895 Ki = 3.7 nM T09572 C2FX5H 44416898 Ki = 10 nM T09572 CPNY68 44416910 Ki = 197 nM T09572 CLP16U 44416911 Ki = 1.585 nM T09572 C0X5HE 44416916 Ki = 63.1 nM T09572 C0OMX6 44416923 IC50 > 1000 nM T09572 CE0SK3 44416928 Ki = 126 nM T09572 CB9RO3 44416929 Ki = 91 nM T09572 CZ8CS2 44416935 IC50 = 5.012 nM T09572 C5G7KA 44416946 IC50 > 1000 nM T09572 CC9KR4 44416947 IC50 > 1000 nM T09572 C74ATQ 44416949 IC50 = 25.12 nM T09572 C87RVU 44416955 IC50 = 5.012 nM T09572 C5MI0P 44416956 IC50 = 12.59 nM T09572 C5C7QR 44416964 IC50 > 1000 nM T09572 CILD84 44416966 Ki = 773 nM T09572 C5MY6P 44416968 Ki = 79.43 nM T09572 C7BI9T 44416969 Ki = 10 nM T09572 CIEB89 44416970 Ki = 10 nM T09572 C9WRP8 44416975 IC50 = 2511.89 nM T09572 CW2I3N 44416976 IC50 = 10 nM T09572 C9QU0R 44416989 Ki = 7.943 nM T09572 C8BQ3P 44416990 Ki = 31.62 nM T09572 CTC30S 44416995 IC50 = 12.59 nM T09572 C5C1PE 44417017 IC50 = 170 nM T09572 C0DV8X 44417021 IC50 = 2.512 nM T09572 CGNK93 44417022 IC50 = 7.943 nM T09572 C05LZR 44417024 Ki = 2.512 nM T09572 CZ5SQ3 44417025 Ki = 5 nM T09572 CFPC71 44417043 IC50 = 15.85 nM T09572 CZ4Q5J 44417044 IC50 = 3.162 nM T09572 C2LW3E 44417061 Ki = 84 nM T09572 CE8KJ6 44417066 IC50 = 5.012 nM T09572 C0NI5V 44417067 IC50 = 15.85 nM T09572 C0A2FS 44417069 Ki = 15.85 nM T09572 CK92GD 44417083 IC50 = 7.943 nM T09572 CCX9R4 44417140 IC50 = 31.62 nM T09572 CXLI76 44417145 IC50 = 6.31 nM T09572 CQP8L9 44417146 IC50 = 5.012 nM T09572 C7WY1L 44417150 IC50 = 10 nM T09572 C0YZ7M 44417151 IC50 = 6.31 nM T09572 CT3KX7 44417481 IC50 > 2000 nM T09572 C0V7EJ 44417821 EC50 = 370 nM T09572 CA61IW 44417822 IC50 = 10000 nM T09572 C0Y8UH 44417823 EC50 = 120 nM T09572 CYAD92 44417824 IC50 = 4000 nM T09572 CG0E3N 44417825 IC50 = 1700 nM T09572 CPX53N 44417827 IC50 = 1100 nM T09572 CU72ZV 44417828 Ki = 27 nM T09572 C46RHE 44417829 Ki = 56 nM T09572 C8AQU5 44417830 Ki = 1000 nM T09572 CR0G9W 44417831 Ki = 286 nM T09572 CYNX47 44417832 IC50 = 0.7 nM T09572 CC0P6Y 44417833 Ki = 133 nM T09572 CLHV60 44417834 Ki > 100000 nM T09572 CDT9M1 44417835 Ki = 8.6 nM T09572 C3F4ZC 44417836 Ki = 86 nM T09572 CAO59Y 44417837 Ki = 170 nM T09572 C0NPX2 44417838 EC50 = 500 nM T09572 C8QB4F 44417839 Ki = 36 nM T09572 C1OL9Y 44417840 Ki = 40 nM T09572 CPF38S 44417841 Ki = 18 nM T09572 C7D4FK 44417842 Ki = 9 nM T09572 C8XC5O 44417843 IC50 = 2.3 nM T09572 CC26DZ 44417844 EC50 = 71 nM T09572 CNQ02C 44417845 EC50 = 40 nM T09572 C1EHB3 44417846 IC50 = 1.4 nM T09572 C3QP7X 44417847 EC50 = 3600 nM T09572 C9TN8Y 44417848 EC50 = 740 nM T09572 CO51ID 44417849 Ki = 232 nM T09572 C96QJO 44417850 Ki = 7 nM T09572 CNX80R 44417851 Ki > 100000 nM T09572 CAI3K8 44417852 Ki = 484 nM T09572 CA7T1X 44417853 Ki = 67 nM T09572 CT7WS4 44417854 Ki = 65 nM T09572 C1MEX3 44417855 Ki = 13 nM T09572 CZO51X 44417856 EC50 = 990 nM T09572 C1JQ5P 44417857 EC50 = 310 nM T09572 CG05EA 44417858 IC50 = 190 nM T09572 CP8AF3 44417859 Ki = 32 nM T09572 CP72QS 44417860 Ki = 62 nM T09572 C1W4VB 44417861 Ki = 12 nM T09572 C05HMG 44417862 Ki = 17 nM T09572 CB10YP 44417863 Ki = 28.2 nM T09572 CB62CN 44417864 IC50 = 95 nM T09572 CQNF68 44417865 Ki = 125 nM T09572 CU7XD8 44417866 IC50 = 1100 nM T09572 C57FVT 44417867 IC50 = 130 nM T09572 CV4EF6 44417868 Ki = 441 nM T09572 CL8X5U 44417869 Ki = 25 nM T09572 C0ODM7 44417870 Ki = 625 nM T09572 C3FO0H 44417871 Ki = 23 nM T09572 CT8FJ0 44417872 Ki = 8070 nM T09572 CI60HL 44417873 EC50 = 910 nM T09572 CC61GR 44417874 IC50 = 9 nM T09572 C6A2YW 44417875 EC50 = 118 nM T09572 CCD0P3 44417876 Ki = 142 nM T09572 CGWI26 44417877 EC50 = 520 nM T09572 CT27KD 44417878 Ki = 505 nM T09572 CA34LP 44417879 Ki = 2.5 nM T09572 C42RJO 44417880 Ki = 205 nM T09572 CU9JD6 44417881 Ki = 136 nM T09572 CN25SX 44417882 Ki > 100000 nM T09572 C21ZCB 44417883 IC50 = 1797 nM T09572 C6HJ3K 44417885 Ki = 169 nM T09572 CRT85J 44417886 EC50 = 2800 nM T09572 CG1WM8 44417887 Ki = 3.3 nM T09572 C89TAB 44417888 IC50 = 20 nM T09572 CK76AM 44417889 Ki = 32 nM T09572 CPE50S 44417890 IC50 = 76 nM T09572 CQS6G2 44417891 Ki = 93 nM T09572 CO0U5H 44417892 IC50 = 300 nM T09572 CAK9U7 44417893 Ki = 52000 nM T09572 C26CUN 44417894 IC50 = 13 nM T09572 C35KLS 44417895 Ki = 146 nM T09572 CL5XO4 44417897 IC50 = 11 nM T09572 CKI1W2 44417898 IC50 = 750 nM T09572 CM9QI8 44417899 IC50 = 21 nM T09572 C6UAH2 44417900 Ki = 2480 nM T09572 CWO51Q 44417901 Ki = 145 nM T09572 CI16UJ 44417902 IC50 = 1267 nM T09572 C0US4Z 44417903 IC50 = 18 nM T09572 C8GK5Q 44417904 Ki = 24 nM T09572 CHC7G9 44417905 Ki = 11 nM T09572 C9BDI1 44417906 IC50 = 95 nM T09572 CC3S6F 44417907 IC50 = 3700 nM T09572 C3GW2E 44417908 Ki = 94000 nM T09572 CKQ92G 44417909 Ki = 22 nM T09572 CN2G7U 44417910 IC50 = 43 nM T09572 C46KMH 44417911 IC50 = 4 nM T09572 C2XJW5 44417912 Ki = 5294 nM T09572 CPDW02 44417913 Ki = 184 nM T09572 CY46AB 44417914 Ki = 270000 nM T09572 C9HN5T 44417915 IC50 = 800 nM T09572 C5HA7X 44417916 Ki = 18 nM T09572 CM2UC6 44417917 IC50 = 25 nM T09572 CD62PS 44417918 Ki = 100000 nM T09572 CW1D3V 44417919 Ki = 11 nM T09572 CCU69N 44417920 Ki = 62000 nM T09572 CFR6H4 44417921 IC50 = 12 nM T09572 C3CM4J 44417922 Ki = 12 nM T09572 CH0T1F 44417923 Ki = 15000 nM T09572 C4WU0N 44417924 Ki = 30000 nM T09572 CTUV23 44417925 IC50 = 10 nM T09572 CE96RJ 44417926 Ki = 20 nM T09572 C27PHW 44417927 Ki = 47 nM T09572 CEZH78 44417928 Ki = 103 nM T09572 CT0B1U 44417929 Ki = 8700 nM T09572 CB8IZ1 44417930 IC50 = 3 nM T09572 CPO9R1 44417931 IC50 = 622 nM T09572 C7F4LM 44417933 Ki = 2482 nM T09572 CS9AZ3 44417934 Ki = 82 nM T09572 CH08OA 44417936 IC50 = 2010 nM T09572 C7W8KZ 44417937 IC50 = 166 nM T09572 CH3QM1 44417938 IC50 = 47 nM T09572 CP1U0Z 44417939 IC50 = 19 nM T09572 C3B4LO 44417940 IC50 = 180 nM T09572 C7IJZ9 44417941 IC50 = 25 nM T09572 CP5K2A 44417942 IC50 = 2700 nM T09572 CM6H8T 44417943 IC50 = 45 nM T09572 CHSE12 44417944 EC50 = 110 nM T09572 C89EBO 44417945 IC50 = 3 nM T09572 C42OAE 44417946 IC50 = 763 nM T09572 CQ7M6F 44417947 EC50 = 250 nM T09572 C70AVF 44417948 EC50 = 68 nM T09572 CZK6C5 44417949 IC50 = 4 nM T09572 C3WT1V 44417950 Ki = 15 nM T09572 CM76IN 44417952 IC50 = 96 nM T09572 C6F9MN 44417953 Ki = 23 nM T09572 C3P1JG 44417954 Ki = 727 nM T09572 CLOU53 44417955 IC50 = 961 nM T09572 C2OH0S 44417956 IC50 = 5 nM T09572 COA19M 44417957 IC50 = 5 nM T09572 CDF0V4 44417959 EC50 = 90 nM T09572 C3SVB8 44417960 Ki = 3465 nM T09572 C6HTW2 44417961 IC50 = 112 nM T09572 CF7QS3 44417962 EC50 = 160 nM T09572 C6TJL5 44417963 Ki = 497 nM T09572 C5GDU7 44417965 Ki = 4 nM T09572 CFU91G 44417966 IC50 = 0.3 nM T09572 C7JFN6 44417967 Ki = 148 nM T09572 C93GJO 44417968 IC50 = 313 nM T09572 CH6F8D 44417969 Ki = 228 nM T09572 CM2YT3 44417970 IC50 = 1814 nM T09572 C9RKO4 44417971 IC50 = 512 nM T09572 CNVM62 44417972 IC50 = 952 nM T09572 CF91YW 44417973 IC50 = 13 nM T09572 C3C5PN 44417974 IC50 = 212 nM T09572 CE3Q5V 44417975 IC50 = 210 nM T09572 CDT71X 44417976 IC50 = 88 nM T09572 CH2RQ7 44417977 IC50 = 243 nM T09572 C2JM1K 44417979 IC50 = 18.5 nM T09572 C6K9JW 44417981 IC50 = 904 nM T09572 C6D2EQ 44417982 IC50 = 240 nM T09572 CFU0Y7 44417983 IC50 = 1034 nM T09572 CJZ82I 44417984 Ki = 570 nM T09572 CM2EL7 44417985 Ki = 890 nM T09572 CY2I0A 44417986 IC50 = 311 nM T09572 CTYW15 44417987 Ki = 625 nM T09572 C07FSQ 44417988 IC50 = 443 nM T09572 CG63SF 44417989 Ki = 260 nM T09572 CLS47Q 44417991 IC50 = 172 nM T09572 CM4VL9 44417992 EC50 = 300 nM T09572 C7CP8I 44417993 Ki = 118 nM T09572 C8OZD0 44417994 IC50 = 122 nM T09572 CNR9E4 44417995 IC50 = 26 nM T09572 C2GZ9T 44417996 IC50 = 1100 nM T09572 CE0FS4 44417998 EC50 = 150 nM T09572 CQ3LS1 44417999 EC50 = 340 nM T09572 CWR70L 44418000 Ki = 99 nM T09572 CRP5I2 44418002 IC50 = 4 nM T09572 CP7YV8 44418003 EC50 = 904 nM T09572 C6Q7ZM 44418004 Ki = 129 nM T09572 CF4E1N 44418005 IC50 = 78 nM T09572 C8BH6G 44418006 IC50 = 1008 nM T09572 CFUG30 44418008 IC50 = 490 nM T09572 C8DIV9 44418009 IC50 = 36 nM T09572 CRO92C 44418010 IC50 = 40 nM T09572 CE51ZC 44424061 Ki = 16 nM T09572 CU78DE 44424062 Ki = 10 nM T09572 C5OXM1 44424063 Ki = 12 nM T09572 CR6TA2 44424064 Ki = 19 nM T09572 CEIA14 44424065 Ki = 194 nM T09572 CA2D9R 44424066 Ki = 4 nM T09572 CO26JC 44424067 IC50 = 38 nM T09572 CINY58 44424068 Ki = 374 nM T09572 C41UFQ 44424069 Ki = 19 nM T09572 C5THN9 44424070 IC50 = 3 nM T09572 C0G2QJ 44424071 Ki = 25 nM T09572 CLAW52 44424072 Ki = 2000 nM T09572 CUL09D 44424073 Ki = 1200 nM T09572 C7O9PT 44424166 Ki = 132 nM T09572 C8MJ5Y 44424167 Ki = 1884 nM T09572 C7GS8T 44424168 Ki = 20 nM T09572 COD05N 44424169 Ki = 373 nM T09572 C6Y3NT 44424170 Ki = 54 nM T09572 C1V5YS 44424171 Ki = 15 nM T09572 COU9D8 44424172 Ki = 20 nM T09572 CSU96B 44424173 Ki = 48 nM T09572 CZ48SF 44424174 Ki = 134 nM T09572 CA2TK3 44424175 Ki = 539 nM T09572 C4DSJ0 44424176 Ki = 2213 nM T09572 CR2GP1 44424177 Ki = 16 nM T09572 CWJ41D 44424178 Ki = 23 nM T09572 C9IC7X 44424179 Ki = 15 nM T09572 C51PEO 44424180 Ki = 7 nM T09572 CA76NC 44424181 Ki = 15 nM T09572 CP4H0T 44424182 Ki = 15 nM T09572 CKE61I 44424183 Ki = 22 nM T09572 CW8NM4 44424184 Ki = 53 nM T09572 CZ6LD4 44424185 Ki = 15 nM T09572 CSA9H2 44424186 Ki = 11 nM T09572 C9AP8V 44424187 Ki = 5 nM T09572 C7R3WV 44424188 Ki = 2.7 nM T09572 CQ6Z7X 44424189 Ki = 5.7 nM T09572 CP2W3Y 44424190 Ki = 2.1 nM T09572 CEHP70 44424191 Ki = 6 nM T09572 CBAW19 44424192 Ki = 7.6 nM T09572 CV48KH 44424193 Ki = 4.5 nM T09572 CO7A5C 44424194 Ki = 2.8 nM T09572 C7L0KT 44424195 Ki = 10.4 nM T09572 C36ROD 44424196 Ki = 2 nM T09572 CH1Z3R 44424197 Ki = 60 nM T09572 C3PMT9 44424198 Ki = 34 nM T09572 CK5ZM9 44424199 Ki = 27 nM T09572 CM5UV2 44424200 Ki = 92 nM T09572 COHK30 44424201 Ki = 92 nM T09572 CJ1S6F 44424202 Ki = 7.8 nM T09572 CPI5B7 44424203 Ki = 142 nM T09572 C59RHN 44424204 Ki = 34 nM T09572 CC7PE6 44424205 Ki = 48 nM T09572 CC45EG 44424206 Ki = 4.1 nM T09572 CNDW09 44424207 Ki = 29 nM T09572 CVKE34 44424208 Ki = 8.7 nM T09572 C5EMG3 44424209 Ki = 9.4 nM T09572 CAG2L4 44424210 Ki = 5.2 nM T09572 C04VIZ 44424211 Ki = 12 nM T09572 C51ZVB 44424212 Ki = 1.6 nM T09572 C08JMU 44424213 Ki = 1.6 nM T09572 CDB0G8 44424214 Ki = 10 nM T09572 CX21FM 44424215 Ki = 1.9 nM T09572 C8B2SV 44424216 Ki = 4.4 nM T09572 CCVG85 44424217 Ki = 11 nM T09572 CGA81M 44424218 Ki = 1.2 nM T09572 C25WLJ 44424224 Ki = 8.7 nM T09572 C5SM3Y 44424225 Ki = 181 nM T09572 C4FET2 44424228 Ki = 312 nM T09572 CBQ6F5 44424229 Ki = 7.2 nM T09572 CC4J1W 44424231 Ki = 5.4 nM T09572 CJ15CH 44424232 Ki = 21 nM T09572 C28AFI 44424233 Ki = 26 nM T09572 CC1KS2 44424234 Ki = 9.7 nM T09572 C4TDJ7 44424235 Ki = 80 nM T09572 C3PLC4 44424236 Ki = 211 nM T09572 CP90FZ 44424237 Ki = 295 nM T09572 CH2R7W 44424238 Ki = 559 nM T09572 C8BT1N 44424244 Ki = 2.3 nM T09572 CVJ2L5 44424246 Ki = 18 nM T09572 C9P1QG 44424247 Ki = 31 nM T09572 CR9L4I 44424249 Ki = 21 nM T09572 C45NIL 44424250 Ki = 54 nM T09572 CNB09T 44424252 Ki = 46 nM T09572 C2IMP0 44424253 Ki = 13 nM T09572 CW9ZC2 44424254 Ki = 9.9 nM T09572 C6OW2Z 44424255 Ki = 15 nM T09572 C4GSN5 44424256 Ki = 2.4 nM T09572 CO86IG 44424258 Ki = 3.3 nM T09572 C5F8PY 44424259 Ki = 8.9 nM T09572 C7BW3R 44424260 Ki = 146.89 nM T09572 C13AXK 44424261 Ki = 30 nM T09572 C7V2AY 44424262 Ki = 1969 nM T09572 CH17YP 44424263 Ki = 116.95 nM T09572 CW53QE 44424265 Ki = 51 nM T09572 C47BAF 44424266 Ki = 316 nM T09572 C32PLE 44424267 Ki = 85 nM T09572 C63AUS 44424268 Ki = 31 nM T09572 C1D8YR 44424269 Ki = 4.2 nM T09572 CJ25WE 44424270 Ki = 57 nM T09572 C89EXO 44425789 Ki = 50 nM T09572 C89LGK 44425790 Ki = 2100 nM T09572 CG3MY4 44425792 Ki = 1100 nM T09572 C1N0EW 44425793 Ki = 200 nM T09572 CN2I8O 44425794 Ki = 340 nM T09572 C7LMS4 44425795 Ki = 115 nM T09572 CH02JZ 44425796 Ki = 150 nM T09572 COX87N 44425797 Ki = 400 nM T09572 C89PUR 44425798 Ki = 25 nM T09572 CUP51V 44425799 Ki = 340 nM T09572 C3N2GM 44425800 Ki = 300 nM T09572 C2AE6C 44425801 Ki = 1500 nM T09572 CH04WE 44425802 Ki = 89 nM T09572 C9D4LQ 44425803 Ki = 44 nM T09572 C3REX2 44425804 Ki = 330 nM T09572 C4L5ZP 44425805 Ki = 640 nM T09572 CK7T3L 44425806 Ki = 315 nM T09572 CT1N9U 44425807 Ki = 20 nM T09572 C52ZIS 44425809 Ki = 13 nM T09572 CU7YW1 44425810 Ki = 10 nM T09572 C0WVT1 44425811 Ki = 8 nM T09572 C46FWV 44425812 Ki = 230 nM T09572 CYR4W7 44425814 Ki = 9300 nM T09572 CP1ZY6 44425815 Ki > 10000 nM T09572 CE3A2G 44425817 Ki = 20 nM T09572 CCV7H3 44425818 Ki = 210 nM T09572 C6JY8V 44425820 Ki = 620 nM T09572 CNV50P 44425821 Ki = 150 nM T09572 CA4KO2 44425822 Ki = 8000 nM T09572 C3KP5U 44425823 Ki = 2900 nM T09572 CX7TS1 44425824 Ki = 92 nM T09572 C7IF1X 44425825 Ki = 19 nM T09572 CWZ4G7 44425826 Ki = 280 nM T09572 CE2R3N 44425827 Ki = 180 nM T09572 CADK60 44425828 Ki = 100 nM T09572 CNFI93 44425830 Ki = 84 nM T09572 CY5HW2 44425832 Ki = 12 nM T09572 CKJ03V 44425834 IC50 = 5 nM T09572 CYJ20S 44425835 Ki = 6 nM T09572 C1IVD0 44425837 Ki = 45 nM T09572 CXPO87 44425839 Ki = 6 nM T09572 CBMT90 44430452 Ki = 17 nM T09572 CODL74 44430453 Ki = 6 nM T09572 CAE2N5 44430455 Ki = 5 nM T09572 CMKP65 44430458 Ki = 1 nM T09572 C8OQV2 44430459 Ki = 4 nM T09572 CNW86X 44430460 Ki = 2 nM T09572 C62BSV 44430463 Ki = 3 nM T09572 CB97TH 44430465 Ki = 50 nM T09572 CW01JX 44430468 Ki = 4 nM T09572 CU6I1H 44430471 Ki = 4 nM T09572 CJ9C8U 44430475 Ki = 3 nM T09572 C12TLF 44430476 Ki = 7 nM T09572 CQ59YW 44430477 Ki = 7 nM T09572 CH38CM 44430478 Ki = 17 nM T09572 CT37LP 44430479 Ki = 80 nM T09572 CZ8WO4 44430480 Ki = 69 nM T09572 C1UMX3 44430481 Ki = 154 nM T09572 CP6U2S 44430482 Ki = 15 nM T09572 C5YQ3O 44430483 Ki = 5 nM T09572 C2OT9F 44430484 Ki = 49 nM T09572 C7TEZ2 44430485 Ki = 17 nM T09572 C8J0LH 44430486 Ki = 39 nM T09572 CX1D3I 44430487 Ki = 21 nM T09572 C5K1DQ 44430488 Ki = 46 nM T09572 CRT5O9 44430489 Ki = 26 nM T09572 CAG1M5 44430490 Ki = 143 nM T09572 CX03CA 44430493 Ki = 14 nM T09572 CTM7G1 44430494 Ki = 8 nM T09572 CTK8S7 44430495 Ki = 70 nM T09572 CIG9Y6 44430496 Ki = 19 nM T09572 CR5EU8 44430498 Ki = 18 nM T09572 CX81ZL 44430499 Ki = 28 nM T09572 CKOL19 44430500 Ki = 14 nM T09572 C09UFN 44430501 Ki = 45 nM T09572 CJ81UG 44434143 Ki = 22 nM T09572 C15TRQ 44434144 Ki = 431 nM T09572 C16UDV 44434145 Ki = 99 nM T09572 CC03AH 44434146 Ki = 45 nM T09572 C5H1MB 44434148 Ki = 17 nM T09572 CYNE36 44434149 Ki = 19 nM T09572 CVFM10 44434151 Ki = 13.1 nM T09572 CA98YS 44434152 Ki = 73 nM T09572 CN80KD 44434153 Ki = 117 nM T09572 CM6LD3 44434154 Ki = 6.1 nM T09572 CY45FT 44434155 Ki = 171 nM T09572 CZ18JV 44434156 Ki = 4 nM T09572 C7LD6V 44437494 Ki = 543.25 nM T09572 C1I2BU 44437495 Ki = 1445.44 nM T09572 CS9UQ1 44437496 Ki = 425 nM T09572 C4SV8L 44437497 Ki = 186 nM T09572 CO8DT9 44437498 Ki = 2640 nM T09572 C9R8WN 44437499 Ki = 5860 nM T09572 C3ZDU4 44437500 Ki > 1000 nM T09572 CP36JI 44437501 Ki = 6025.6 nM T09572 CCMV89 44437514 Ki = 6380 nM T09572 CO20QU 44437515 Ki > 1000 nM T09572 CRD6O8 44437516 Ki = 312.61 nM T09572 CW09ML 44437517 Ki = 273 nM T09572 CE5OX7 44437518 Ki > 1000 nM T09572 CXH06Q 44437519 Ki = 509 nM T09572 CYK2O7 44437520 Ki = 257.04 nM T09572 CAV9L2 44437522 Ki = 421 nM T09572 C4HZX3 44437523 Ki = 595 nM T09572 CXBE83 44437524 Ki = 214.78 nM T09572 C4X0AD 44437525 Ki = 254 nM T09572 CPLN85 44437526 Ki = 947 nM T09572 CTKX20 44437528 Ki = 213.8 nM T09572 CE08HO 44437541 Ki = 169.82 nM T09572 C7VBE4 44437542 Ki = 1200 nM T09572 CV6S2Q 44437544 Ki = 1080 nM T09572 CYC56F 44437547 Ki = 388 nM T09572 CPDS73 44437553 Ki = 96.6 nM T09572 CZ9L4F 44437555 Ki = 204 nM T09572 C1AU2N 44437557 Ki = 251 nM T09572 C61UVK 44437558 Ki = 144 nM T09572 C0IQ8W 44437609 Ki = 149 nM T09572 CBG34A 44437612 Ki = 143 nM T09572 CC1L2V 44437614 Ki = 165.96 nM T09572 CJQ1X5 44437620 Ki = 769 nM T09572 CS3GI1 44437622 Ki = 173 nM T09572 CEB9V8 44438737 IC50 > 2000 nM T09572 CJ79PE 44438739 IC50 = 1520 nM T09572 C9T7JL 44438740 IC50 = 773 nM T09572 CB9S3W 44438741 IC50 = 165 nM T09572 CL20OD 44438742 IC50 = 64 nM T09572 C71UWM 44438745 IC50 = 4010 nM T09572 CBJ5R9 44438747 IC50 = 31 nM T09572 C5VFD8 44438748 IC50 = 15 nM T09572 CW8GU6 44438753 IC50 = 86 nM T09572 CS9D3H 44438755 IC50 = 26 nM T09572 C65EMO 44440586 Ki = 260 nM T09572 C6FGD1 44440587 Ki = 101 nM T09572 C8ZA4N 44440588 Ki = 1090 nM T09572 CZ1L5J 44440593 Ki = 1000 nM T09572 C9IBX4 44440599 Ki = 176 nM T09572 C0NBF9 44442050 IC50 = 3590 nM T09572 CUC4A6 44442051 IC50 > 33000 nM T09572 C7EH8P 44442053 IC50 = 3 nM T09572 C8EAD0 44442054 IC50 = 411 nM T09572 C03OKE 44442056 IC50 = 5010 nM T09572 C9BKO7 44442058 IC50 = 106 nM T09572 CZVQ72 44442059 IC50 = 119 nM T09572 CBTV83 44442060 IC50 = 2990 nM T09572 CW41ZF 44442061 IC50 = 2300 nM T09572 C23MNK 44442062 IC50 = 2130 nM T09572 C1PEQ4 44442063 IC50 = 68 nM T09572 CANQ03 44442064 IC50 = 7 nM T09572 CC6S0I 44442065 IC50 = 25 nM T09572 CXJ52D 44442066 IC50 = 571 nM T09572 CD5G2R 44442067 IC50 = 847 nM T09572 CE0Y1I 44442068 IC50 = 2520 nM T09572 CO3V4T 44442069 IC50 = 4800 nM T09572 C4CRF6 44442070 IC50 = 9920 nM T09572 CE52RC 44442071 IC50 = 97 nM T09572 C2A0OM 44442090 IC50 = 8 nM T09572 CX5J6I 44442093 IC50 = 231 nM T09572 C10KDT 44442095 IC50 = 0.1 nM T09572 CR3KI9 44442097 IC50 = 54 nM T09572 CE4LG3 44442098 IC50 = 1390 nM T09572 CLU51Z 44442100 IC50 = 5100 nM T09572 C06WTB 44442118 IC50 = 22 nM T09572 CPW23O 44442119 IC50 = 89 nM T09572 CT3N0B 44442120 IC50 = 13 nM T09572 C8VEW9 44442121 IC50 = 28 nM T09572 C2Y1XP 44442124 IC50 = 61 nM T09572 CK57FP 44442130 IC50 = 58 nM T09572 CGLN40 44442134 IC50 = 16 nM T09572 C13TNE 44442135 IC50 = 50 nM T09572 C2FAQ7 44442139 IC50 = 9 nM T09572 CBN4Q3 44442144 IC50 = 35 nM T09572 CSQN12 44442148 IC50 = 80 nM T09572 C0SMR6 44442151 IC50 = 33 nM T09572 CBV07Y 44442153 IC50 = 20 nM T09572 C4Z8HF 44442156 IC50 = 39 nM T09572 CV3ZI1 44454966 Ki = 25 nM T09572 CU8EX2 44455336 Ki = 0.5 nM T09572 COU5A6 44455367 Ki = 47 nM T09572 C7B1KA 44455368 Ki = 10 nM T09572 CQKH50 44455414 Ki = 5 nM T09572 CK4O6B 44455417 Ki = 20 nM T09572 C0I6SN 44455443 Ki = 31 nM T09572 CRN57M 44455444 Ki = 5.2 nM T09572 CQ0WM7 44469273 IC50 = 2.6 nM T09572 CNW41S 44539369 Ki = 2920 nM T09572 CJE2Q6 44555375 IC50 = 1.2 nM T09572 C4LJ6X 44557554 IC50 = 19 nM T09572 C2X1BC 44562403 IC50 = 804 nM T09572 CK2GC9 44562404 IC50 = 104 nM T09572 C21KTW 44562405 IC50 = 903 nM T09572 COQ7L5 44562415 IC50 = 82 nM T09572 CX39BW 44562416 IC50 = 2340 nM T09572 CZVN14 44562441 IC50 > 33000 nM T09572 C7C5GX 44562442 IC50 = 43 nM T09572 C6X1CW 44562443 IC50 = 9650 nM T09572 CC57QH 44562461 IC50 = 1500 nM T09572 CZT5U2 44562462 IC50 = 927 nM T09572 CTV75H 44562479 IC50 = 347 nM T09572 CHN81A 44562480 IC50 = 2140 nM T09572 CCY92R 44562481 IC50 = 636 nM T09572 C4WAK1 44562499 IC50 = 3050 nM T09572 CH40TM 44562500 IC50 = 29 nM T09572 C1NG5P 44562501 IC50 = 111 nM T09572 C4IK2N 44562521 IC50 = 2260 nM T09572 CP80OG 44562522 IC50 = 104 nM T09572 CE5M8W 44562523 IC50 = 1250 nM T09572 CK6PR8 44562524 IC50 = 169 nM T09572 C9QW4M 44562542 IC50 = 313 nM T09572 CYDB09 44562543 IC50 = 303 nM T09572 C6USZ1 44562544 IC50 = 269 nM T09572 CEJ3G1 44562545 IC50 = 122 nM T09572 C59XKS 44562562 IC50 = 113 nM T09572 CAPH48 44562563 IC50 = 58 nM T09572 C9XD5G 44562564 IC50 = 67 nM T09572 CJB05V 44562565 IC50 = 66 nM T09572 C1SUW5 44562600 IC50 = 71 nM T09572 C81IMZ 44573820 IC50 = 9.6 nM T09572 CEF6J8 44573821 IC50 = 2.1 nM T09572 CT2FW6 44573822 IC50 = 2.1 nM T09572 C4I5UB 44573823 IC50 = 19 nM T09572 CXWQ34 44573931 IC50 = 1.7 nM T09572 C6U0EY 44573932 IC50 = 9.9 nM T09572 C04SIR 44573964 IC50 = 125 nM T09572 CAT49R 44574008 IC50 = 0.15 nM T09572 C0VQ8Y 44574357 IC50 = 54 nM T09572 CQZ1Y2 44574358 IC50 = 42 nM T09572 C0SOD6 44574359 IC50 = 42 nM T09572 C95TVW 44592169 Ki = 3.16 nM T09572 COR08L 44592214 Ki = 3.3 nM T09572 CO0RY5 44592215 Ki = 3 nM T09572 CO6X8L 44592256 IC50 = 83.18 nM T09572 CO6ES5 44592257 IC50 = 104.71 nM T09572 CD06ZV 45178545 IC50 = 18000 nM T09572 C3BWP6 45266975 Ki = 1413 nM T09572 CJVC17 45266979 Ki = 30 nM T09572 CP1UX8 45267015 Ki = 3473 nM T09572 C1N5ZL 45267385 IC50 = 55 nM T09572 C4AZD3 45267386 IC50 = 444 nM T09572 C8LPF5 45267399 IC50 = 597 nM T09572 C8PR5X 45267430 IC50 = 21 nM T09572 C17EPN 45267561 IC50 = 83 nM T09572 CA4ZJ2 45267565 IC50 = 260 nM T09572 CNZ95W 45267576 IC50 = 100 nM T09572 CVPT19 45267577 IC50 = 5.4 nM T09572 C7SJ4A 45267654 IC50 = 300 nM T09572 CM23AU 45267709 IC50 = 196 nM T09572 CGB32I 45267714 IC50 = 21 nM T09572 CO3Y0N 45267724 IC50 = 120 nM T09572 CI7KZ2 45267735 IC50 = 17 nM T09572 CC5OP0 45267739 IC50 = 27 nM T09572 CXJ8H3 45267746 IC50 = 152 nM T09572 CCS2E7 45267809 Ki = 17380 nM T09572 CV4W6Y 45267812 Ki = 1951 nM T09572 CZ8G9K 45267814 Ki = 4560 nM T09572 C37UGL 45267827 Ki = 149 nM T09572 CH4V7J 45267849 IC50 = 11765 nM T09572 CP85WO 45268247 IC50 = 71 nM T09572 CW5C8M 45268457 IC50 = 320 nM T09572 C4G1SL 45268465 IC50 = 48 nM T09572 C84UTO 45268470 IC50 = 4 nM T09572 COZ7J8 45268527 IC50 = 130 nM T09572 C7VZR5 45268637 IC50 = 112 nM T09572 CV1IR5 45268644 IC50 = 412 nM T09572 CXSQ09 45268694 Ki = 2334 nM T09572 CJFQ65 45268721 Ki = 5642 nM T09572 CGL25F 45268725 Ki = 3567 nM T09572 CPH10U 45269335 IC50 = 102 nM T09572 C63KED 45269336 IC50 = 44 nM T09572 CHR31D 45269555 Ki = 5114 nM T09572 CA3MZ6 45269996 IC50 = 417 nM T09572 C5DIS2 45270014 IC50 = 5 nM T09572 CF0DL4 45270139 IC50 = 35 nM T09572 CC14UH 45270147 IC50 = 330 nM T09572 C2UNR9 45270157 IC50 = 160 nM T09572 CPG7D6 45270273 IC50 = 617 nM T09572 C0J6BO 45270297 IC50 = 138 nM T09572 C23PMF 45270302 IC50 = 125 nM T09572 C9WNG1 45270303 IC50 = 46 nM T09572 C4SXQ3 45270319 IC50 = 66 nM T09572 C26DVR 45270386 Ki = 2056 nM T09572 C7LW6A 45270392 Ki = 5 nM T09572 CL71EJ 45270393 Ki = 312 nM T09572 CKLX79 45270416 IC50 = 1800 nM T09572 C3A0NB 45270802 IC50 = 4 nM T09572 C35TNH 45270803 IC50 = 150 nM T09572 C3GLV8 45270841 IC50 = 28 nM T09572 CD5OS6 45270850 IC50 = 67 nM T09572 C42GYR 45271095 IC50 = 13 nM T09572 C1F5RT 45271103 IC50 = 236 nM T09572 CCN0F4 45271111 IC50 = 40 nM T09572 CS9M8B 45271114 IC50 = 36 nM T09572 CY70FL 45271134 IC50 = 10 nM T09572 C5YL6K 45271219 Ki = 105 nM T09572 C97WCQ 45271221 Ki = 1078 nM T09572 CR3S4Z 45271246 Ki = 13890 nM T09572 CO04UR 45271549 IC50 = 145 nM T09572 C13PCQ 45271633 IC50 = 8 nM T09572 C3OA8C 45271642 IC50 = 30 nM T09572 CP7CX1 45271647 IC50 = 142 nM T09572 CH1PS3 45271663 IC50 = 173 nM T09572 CM4ZX1 45271673 IC50 = 17 nM T09572 CJN52K 45271829 IC50 = 26 nM T09572 CF9L1B 45271839 IC50 = 4.8 nM T09572 CIWH57 45271907 IC50 = 7.1 nM T09572 C12DAS 45271908 IC50 = 11 nM T09572 C36SRE 45271994 IC50 = 81.8 nM T09572 C73LNM 45272006 IC50 = 111 nM T09572 CMYT82 45272014 IC50 = 23 nM T09572 C60DPZ 45272024 IC50 = 82 nM T09572 C2MKZ1 45272040 IC50 = 308 nM T09572 CWD50J 45272111 Ki = 15606 nM T09572 C7O1UV 45272117 Ki = 4678 nM T09572 C5CEH0 45272120 Ki = 133 nM T09572 C6FCW0 45272539 IC50 = 66 nM T09572 CKI1W9 45272701 IC50 = 8.2 nM T09572 CJ52PS 45272816 IC50 = 49 nM T09572 CD6FR7 45272837 IC50 = 57 nM T09572 C3GUS5 45272853 IC50 = 38 nM T09572 C2YI4R 45272942 Ki = 2584 nM T09572 CY65HN 45272944 Ki = 36588 nM T09572 C3F7SQ 45272984 Ki = 4135 nM T09572 C7QZG5 45272985 Ki = 9332 nM T09572 CYD3P4 45273335 IC50 = 0.87 nM T09572 C9JQT2 45273392 IC50 = 815 nM T09572 CPTE06 45273401 IC50 = 40 nM T09572 CG4YS2 45273406 IC50 = 144 nM T09572 CZ7R6G 45273623 IC50 = 30 nM T09572 C2K6RW 45273638 IC50 = 140 nM T09572 C2AB8E 45273642 IC50 = 122 nM T09572 CSGK15 45273659 IC50 = 61 nM T09572 CKM6P4 45273703 IC50 = 4.6 nM T09572 CLFN69 45273777 IC50 = 28 nM T09572 CP7OZ1 45273778 IC50 = 90 nM T09572 COD72W 45273783 IC50 = 63 nM T09572 CCJR41 45273790 IC50 = 63 nM T09572 C3TZ8X 45273801 IC50 = 19 nM T09572 CX9T5I 45273802 IC50 = 11 nM T09572 CX9LC1 45273887 IC50 = 3057 nM T09572 C2GKC7 45278576 Ki = 124 nM T09572 C81XVO 45278577 Ki = 17 nM T09572 CVD12N 45278578 Ki = 13 nM T09572 CY9SZ3 45278579 Ki = 0.7 nM T09572 CPT17U 45278657 Ki = 76 nM T09572 CQ4J0K 45278977 Ki = 26 nM T09572 C79CHB 45279061 Ki = 3.4 nM T09572 C35VWA 45279062 Ki = 6.5 nM T09572 CH3YM7 45279064 Ki = 6.5 nM T09572 C9GZ5B 45279148 Ki = 2.4 nM T09572 C6DU8B 45279233 Ki = 9 nM T09572 CT30ZQ 45279319 Ki = 28 nM T09572 CJ20EF 45279321 Ki = 15 nM T09572 CE7WZ3 45279402 Ki = 2.3 nM T09572 C8XY6M 45279488 Ki = 21 nM T09572 C0Y2PW 45279489 Ki = 3.5 nM T09572 C7DXG1 45279490 Ki = 0.5 nM T09572 CER6A7 45279491 Ki = 86 nM T09572 C2K8NV 45279493 Ki = 4.4 nM T09572 CX01LN 45279583 Ki = 4.8 nM T09572 CR0N4Z 45279585 Ki = 0.4 nM T09572 C7XI9W 45279680 Ki = 12 nM T09572 C84XIH 45279772 Ki = 15 nM T09572 CZF27R 45279773 Ki = 5.3 nM T09572 C58PTY 45279868 Ki = 3.1 nM T09572 CJO30G 45279869 Ki = 0.8 nM T09572 CL0D6F 45279871 Ki = 13 nM T09572 CYUP42 45279872 Ki = 9.1 nM T09572 CWM86N 45484974 IC50 = 46 nM T09572 CN1OK5 45484984 IC50 = 210 nM T09572 CGLF37 45484995 IC50 = 120 nM T09572 C4X8LF 45485002 IC50 = 26 nM T09572 CQL2O6 45485003 IC50 = 81 nM T09572 C3NFA0 45485004 IC50 = 200 nM T09572 CIX49Y 45485018 IC50 = 230 nM T09572 CHWT32 45485028 IC50 = 7.6 nM T09572 CI97CR 45485029 IC50 = 100 nM T09572 CBZ02X 45485038 IC50 = 64 nM T09572 C7GQ2P 45485043 IC50 = 600 nM T09572 CGOS24 45485061 IC50 = 8 nM T09572 CLX9C8 45485062 IC50 = 2.9 nM T09572 C9JG7Q 45485063 IC50 = 4 nM T09572 C53PKX 45485077 IC50 = 9.6 nM T09572 CREA46 45487283 IC50 = 3.5 nM T09572 C04UFC 45487284 IC50 = 4.4 nM T09572 C7PF5S 45487309 IC50 = 3.5 nM T09572 CTCP93 45487326 IC50 > 1000 nM T09572 CXS6B7 45487330 IC50 = 29 nM T09572 C8ZP0F 45487331 IC50 = 5.4 nM T09572 CF8J3Q 45487356 IC50 = 11 nM T09572 C6KSR1 45487366 IC50 = 30 nM T09572 CSI8X4 45487371 IC50 > 1000 nM T09572 C6FVJ7 45487372 IC50 = 5 nM T09572 C1SEH5 45487375 IC50 > 1000 nM T09572 C1AM2G 45487382 IC50 = 5.9 nM T09572 CC1SO0 45487383 IC50 = 3.3 nM T09572 C3QU2C 45487384 IC50 = 7 nM T09572 COF5G1 45487385 IC50 = 11 nM T09572 C7LQ4D 45487390 IC50 = 5.2 nM T09572 CAB4D7 45487391 IC50 = 4.9 nM T09572 CK9I3H 45487392 IC50 = 34 nM T09572 CMX27T 45487640 IC50 = 2.6 nM T09572 C5NO1K 45487641 IC50 = 45 nM T09572 CR10DI 45487647 IC50 = 1.4 nM T09572 CS17WK 45487652 IC50 = 3.5 nM T09572 CAQ2D8 45487653 IC50 = 6.8 nM T09572 C3A7QW 45487657 IC50 = 4.6 nM T09572 CB9K2G 45487660 IC50 = 1.3 nM T09572 CJ8R3S 45487668 IC50 = 0.22 nM T09572 CN1V0Y 45487671 IC50 = 0.12 nM T09572 CWH0O7 45487673 IC50 = 6.3 nM T09572 CCZR81 45487674 IC50 = 0.35 nM T09572 CTB2P0 46188603 IC50 = 241 nM T09572 C3UN9A 46188959 IC50 = 1173 nM T09572 CS6P3L 46878210 Ki = 338 nM T09572 C07TYF 46899578 IC50 = 1750 nM T09572 C4D0HN 46899579 IC50 = 450 nM T09572 CYSC07 46899581 IC50 = 540 nM T09572 CI05ZH 46899582 IC50 = 1160 nM T09572 C7JP6X 46902024 IC50 = 120 nM T09572 CS46RV 46902025 IC50 = 1660 nM T09572 C08OLW 46902026 IC50 = 920 nM T09572 CHU2O6 46933537 IC50 = 2 nM T09572 C9YZ5I 46933538 IC50 = 0.6 nM T09572 C8A0LD 49801837 IC50 = 23 nM T09572 CG3VX4 49865653 IC50 = 45 nM T09572 CMHY97 49865654 IC50 = 21 nM T09572 C9I0SK 49865678 IC50 = 68 nM T09572 CE09ML 49865679 IC50 = 71 nM T09572 CH5WD6 49865680 IC50 = 35 nM T09572 C9OKI3 49865708 IC50 = 269 nM T09572 CT98KS 49865738 IC50 = 600 nM T09572 CGXO13 49865739 IC50 = 35 nM T09572 C0V2OU 49865789 IC50 = 140 nM T09572 CZ9H6T 49865790 IC50 = 261 nM T09572 CC6B0N 49865868 IC50 = 110 nM T09572 C7Z5TE 49865869 IC50 = 528 nM T09572 C7OF6U 49865870 IC50 = 1620 nM T09572 CI52NU 49865871 IC50 = 87 nM T09572 C5TN3P 49865927 IC50 = 10 nM T09572 CBJ87H 49865928 IC50 = 15 nM T09572 CPHK47 49865929 IC50 = 112 nM T09572 CROD23 49865975 IC50 = 646 nM T09572 C15SMZ 49865976 IC50 = 88 nM T09572 C3G6MD 49865977 IC50 = 336 nM T09572 CBW0I6 49866034 IC50 = 1450 nM T09572 CIP9U4 49866035 IC50 = 13 nM T09572 CS8OU5 49866036 IC50 = 37 nM T09572 C3HI5E 49866086 IC50 = 678 nM T09572 C4PR5M 49866087 IC50 = 566 nM T09572 CEA02K 49866088 IC50 = 9 nM T09572 CK6AX0 49866089 IC50 = 106 nM T09572 C1N4YP 50908737 Ki = 4.9 nM T09572 C3SJ6Y 50908738 Ki = 2.6 nM T09572 C92GDH 50908739 Ki = 2.4 nM T09572 CIRP71 52917998 IC50 = 7 nM T09572 CT0B1S 52917999 IC50 = 12 nM T09572 CFX76G 52918016 IC50 = 12 nM T09572 C47RHB 52918017 IC50 = 27 nM T09572 C9SE1W 52940981 Ki = 33.96 nM T09572 CV8Q3Y 52941054 Ki = 20 nM T09572 C4NUM9 52941152 Ki = 14 nM T09572 CH4X0U 52941195 Ki = 14 nM T09572 CW6CG4 52941272 Ki = 20.99 nM T09572 CFI49B 52941492 Ki = 16 nM T09572 C1HS4J 52941518 Ki = 8.71 nM T09572 CUV8I6 52941526 Ki = 37.7 nM T09572 C9NX0A 52941539 Ki = 7.6 nM T09572 CZM85N 52941615 Ki = 11 nM T09572 CMN74I 52941621 Ki = 8.4 nM T09572 C1YLX8 52941699 Ki = 5.2 nM T09572 C34WMT 52942456 Ki = 3.8 nM T09572 CAH6F7 52942539 Ki = 4.977 nM T09572 CQ20HZ 52942540 Ki = 15 nM T09572 CJOB30 52942547 Ki = 5.2 nM T09572 CIN1J9 52942550 Ki = 62 nM T09572 C79HTE 52942685 Ki = 2.799 nM T09572 CXK65J 52942795 Ki = 11 nM T09572 CT8UE5 52942796 Ki = 5.6 nM T09572 C13YUX 52942885 Ki = 1.901 nM T09572 CXYD26 52943353 Ki = 21.98 nM T09572 C6BZO9 52943420 Ki = 5.395 nM T09572 C2GR9I 52943485 Ki = 28.97 nM T09572 CWX75K 52943587 Ki = 8.892 nM T09572 C0SML4 52943689 Ki = 47.97 nM T09572 CFTH05 52943690 Ki = 59.98 nM T09572 CD3H8P 52943712 Ki = 295.12 nM T09572 CX2RY7 52943873 Ki = 1.6 nM T09572 C8R4JF 52943912 Ki = 23.01 nM T09572 CE0MV7 52943913 Ki = 15 nM T09572 C3GQC4 52943978 Ki = 15 nM T09572 CE84SY 52944068 Ki = 708 nM T09572 C2U4VH 52944540 Ki = 181.13 nM T09572 C0U8RC 52944577 Ki = 47.97 nM T09572 C6L3EG 52944805 Ki = 6300 nM T09572 CV9B7X 52944859 Ki = 17.99 nM T09572 CPV63Q 52944920 Ki = 46.03 nM T09572 C0C2TV 52944948 Ki = 92.04 nM T09572 CEB4J0 52944997 Ki = 7.8 nM T09572 C5DCJ2 52945048 Ki = 2.099 nM T09572 CV6T4N 52945087 Ki = 1.6 nM T09572 C6HNI1 52945088 Ki = 30.97 nM T09572 CT8X7J 52945129 Ki = 10.99 nM T09572 C1MHT3 52945130 Ki = 1.199 nM T09572 CK7JS2 52945154 Ki = 15 nM T09572 CC1NT2 52945806 Ki = 7.762 nM T09572 CG8Z4H 52945863 Ki = 4.102 nM T09572 CXZI97 52946021 Ki = 133.97 nM T09572 C83GRH 52946062 Ki = 26 nM T09572 C9J6PV 52946082 Ki = 20 nM T09572 CTS78H 52946137 Ki = 33.96 nM T09572 CTF7I1 52946184 Ki = 2.698 nM T09572 C6X9RM 52946259 Ki = 5.998 nM T09572 C6HBD0 52947025 Ki = 3500 nM T09572 CK1FT4 52947054 Ki = 7.194 nM T09572 CU86TE 52947140 Ki = 132.13 nM T09572 CL6TY3 52947141 Ki = 20.99 nM T09572 C6CBM4 52947251 Ki = 14 nM T09572 CN6EW2 52947267 Ki = 53.95 nM T09572 CSJ0U6 52947270 Ki = 17 nM T09572 CW6MI3 52947297 Ki = 128 nM T09572 C8PLT3 52947314 Ki = 373.25 nM T09572 CD1P9I 52947331 Ki = 15 nM T09572 C5W8CU 52947407 Ki = 13 nM T09572 CBG8U3 52947408 Ki = 8.71 nM T09572 CXHO23 52947539 Ki = 4.498 nM T09572 C1EY0A 52947542 Ki = 4.395 nM T09572 CTS9E4 52947550 Ki > 5000 nM T09572 CAHV60 52947558 Ki = 7.6 nM T09572 CZ19DQ 52947578 Ki = 1200 nM T09572 C4UN6O 52947610 Ki = 6.998 nM T09572 CCIG41 52947616 Ki = 12.6 nM T09572 C7KTG3 52948254 Ki = 6600 nM T09572 C5M3KF 52948459 Ki > 1000 nM T09572 CRK14T 52948531 Ki = 53.95 nM T09572 CP2EZ8 52948553 Ki = 30.97 nM T09572 C03ORG 52948635 Ki = 5.702 nM T09572 CZ51UD 52948636 Ki = 3.304 nM T09572 CU6QX1 52948758 Ki = 10.4 nM T09572 C76WHV 52948835 Ki = 25 nM T09572 C7SAC6 52948857 Ki = 1.2 nM T09572 CERH05 52948916 Ki = 2.399 nM T09572 C62QLU 52948951 Ki = 9.397 nM T09572 C4EOB2 52949472 Ki = 15 nM T09572 CNG60D 52949479 Ki = 311.89 nM T09572 C25FGA 52949693 Ki = 79.98 nM T09572 C61XZN 52949768 Ki = 9.705 nM T09572 CD26UA 52949812 Ki = 26.98 nM T09572 C3N6DP 52949912 Ki = 11.99 nM T09572 CS02MO 52949941 Ki = 7.2 nM T09572 C0M7FO 52949955 Ki = 7.603 nM T09572 C94WRG 52949956 Ki = 84.92 nM T09572 CQYM81 52950112 Ki = 10.99 nM T09572 CHNX58 53317305 IC50 = 30 nM T09572 CDH87Y 53317306 IC50 = 5.9 nM T09572 CK3MZ0 53317307 IC50 = 7.7 nM T09572 CG6CM0 53317308 IC50 > 1000 nM T09572 CV9W1B 53317524 IC50 = 650 nM T09572 C13SNK 53318592 IC50 = 18 nM T09572 CGWD27 53318593 IC50 = 6.7 nM T09572 C54SRN 53318594 IC50 = 6.8 nM T09572 C74CVF 53318595 IC50 = 16 nM T09572 CK1ZI3 53318801 IC50 = 24 nM T09572 C1VDP8 53319915 IC50 > 1000 nM T09572 CWLQ84 53320117 IC50 = 23 nM T09572 CJ7RL2 53321222 IC50 = 640 nM T09572 CML70D 53321223 IC50 = 3.8 nM T09572 C4BW7G 53322554 IC50 = 12 nM T09572 C98PDX 53322555 IC50 = 4.2 nM T09572 C0HC8D 53324076 IC50 = 7 nM T09572 CHRK49 53324269 IC50 = 180 nM T09572 C6IDZ5 53325163 IC50 = 150 nM T09572 CS3L5G 53325164 IC50 = 22 nM T09572 COD2Y6 53325165 IC50 = 51 nM T09572 CX1RG6 53325166 IC50 > 1000 nM T09572 C9ZF4V 53326457 IC50 = 18 nM T09572 C1UZ8E 54579971 IC50 = 4600 nM T09572 CTA9K1 54579972 IC50 = 3120 nM T09572 C1GXF9 54579973 IC50 = 14 nM T09572 CLW26Q 54580457 IC50 = 70 nM T09572 C8W4CO 54580458 IC50 = 530 nM T09572 CTN5U4 54580459 IC50 = 1130 nM T09572 CQ8E0H 54580923 IC50 = 3180 nM T09572 CQ6V1E 54581466 IC50 = 310 nM T09572 CA2Y3W 54581468 IC50 = 100 nM T09572 C1PWI9 54581469 IC50 > 10000 nM T09572 C8NE4S 54581980 IC50 = 2600 nM T09572 CBK79N 54581986 IC50 > 10000 nM T09572 CUN59X 54582014 IC50 = 840 nM T09572 C5S1ZK 54582015 IC50 = 350 nM T09572 CL02CG 54582016 IC50 > 10000 nM T09572 CGA01C 54582476 IC50 = 360 nM T09572 C2CAO0 54582957 IC50 = 31 nM T09572 CZ3DW2 54582958 IC50 = 170 nM T09572 CM56TD 54582959 IC50 > 10000 nM T09572 CS3P4K 54582960 IC50 = 1600 nM T09572 CD0WT4 54582961 IC50 = 91 nM T09572 C72AXY 54583209 IC50 = 5380 nM T09572 C2DEZ6 54583449 IC50 > 10000 nM T09572 C1R7PQ 54583912 IC50 = 2300 nM T09572 CP0WN1 54583922 IC50 > 10000 nM T09572 CN6E9W 54583953 IC50 = 250 nM T09572 C6UED1 54583954 IC50 = 41 nM T09572 C68OSI 54584181 IC50 = 30 nM T09572 CRZY72 54584417 IC50 > 10000 nM T09572 C3VO1U 54584857 IC50 = 4800 nM T09572 CR3ON1 54584904 IC50 = 2050 nM T09572 C3C8QF 54584905 IC50 = 640 nM T09572 C0V6NH 54584906 IC50 = 2200 nM T09572 CKM78Q 54584907 IC50 > 10000 nM T09572 C7UY2T 54584908 IC50 = 150 nM T09572 CJ03KM 54585374 IC50 = 670 nM T09572 C0TC3L 54585375 IC50 = 410 nM T09572 C7PI2T 54585376 IC50 = 3800 nM T09572 CVE5B9 54585377 IC50 = 170 nM T09572 CIU2O3 54585378 IC50 = 170 nM T09572 C8JUO0 54585827 IC50 = 3200 nM T09572 C0C2BE 54585833 IC50 = 1520 nM T09572 C10GJU 54585861 IC50 = 940 nM T09572 CPX76L 54585862 IC50 = 1520 nM T09572 CW31VH 54585863 IC50 = 24 nM T09572 C2M9RO 54585864 IC50 = 30 nM T09572 CD71UB 54586089 IC50 = 50 nM T09572 CU1F9B 54586090 IC50 > 6000 nM T09572 C5K7CF 54586330 IC50 = 160 nM T09572 CM86YJ 54586331 IC50 = 1020 nM T09572 CA68VP 54586332 IC50 > 10000 nM T09572 CH15VT 54586333 IC50 > 10000 nM T09572 CLUV37 54586334 IC50 > 10000 nM T09572 CSY9Q5 54586798 IC50 > 10000 nM T09572 C3HE2I 54586826 IC50 = 2620 nM T09572 C27KZJ 54586827 IC50 > 10000 nM T09572 CI5G2O 54587365 IC50 > 10000 nM T09572 CAL94R 54587366 IC50 > 10000 nM T09572 CX74PC 54587367 IC50 > 10000 nM T09572 CI4ON9 54587368 IC50 = 140 nM T09572 C7Y3PM 56589628 IC50 = 5.6 nM T09572 CCG6D9 56597407 IC50 = 34 nM T09572 CAC5B2 56597542 IC50 = 27 nM T09572 CTK41N 56597689 IC50 = 21 nM T09572 CN54TH 56597851 IC50 = 23 nM T09572 CZNV53 56597988 IC50 = 22 nM T09572 CI6B8D 56597990 IC50 = 93 nM T09572 CSU5C1 56597991 IC50 = 25 nM T09572 CJ4V0G 56598130 IC50 = 29 nM T09572 CK6VF3 56598528 IC50 = 19 nM T09572 C5F8IX 56666754 IC50 = 9.9 nM T09572 CKQ47D 56666755 IC50 = 4.6 nM T09572 CT0JY2 56666756 IC50 = 33 nM T09572 CQO6F8 56673711 IC50 > 10000 nM T09572 C8MAJ6 56673713 IC50 = 5.5 nM T09572 C7BDU4 56673714 IC50 = 140 nM T09572 CES2I1 56680348 IC50 = 6.8 nM T09572 CYE9C0 56683679 IC50 = 50 nM T09572 C3OM0R 57390252 IC50 = 61 nM T09572 CVM2Z0 57390738 IC50 = 40 nM T09572 C4AVT1 57390739 IC50 = 91 nM T09572 CB6R2C 57391027 IC50 = 86 nM T09572 C3I2XE 57391028 IC50 = 11 nM T09572 C56RAV 57391029 IC50 > 1000 nM T09572 CCTK32 57391030 IC50 = 480 nM T09572 CZ4FY6 57391045 IC50 = 46 nM T09572 C0P1NW 57391572 IC50 = 200 nM T09572 CWL86O 57391573 IC50 = 3300 nM T09572 CBY5V0 57391574 IC50 = 180 nM T09572 CP8Y0U 57391575 IC50 > 20000 nM T09572 CVA0I2 57392546 IC50 = 14 nM T09572 CM7NG4 57392547 IC50 = 5 nM T09572 C8SEO1 57392548 IC50 = 380 nM T09572 CT06UE 57392549 IC50 = 12 nM T09572 CHOU93 57392823 IC50 = 22 nM T09572 C4VSR8 57392824 IC50 = 4.7 nM T09572 C0GK5W 57392835 IC50 = 19 nM T09572 CBX75K 57393331 IC50 = 200 nM T09572 CKW2R8 57393332 IC50 = 0.9 nM T09572 CVP38Z 57394271 IC50 = 20 nM T09572 CW8T3G 57394272 IC50 = 20 nM T09572 C2EWB0 57394273 IC50 = 423 nM T09572 CRB28X 57394274 IC50 = 7 nM T09572 C4O0AK 57394275 IC50 = 50 nM T09572 CI7J8D 57394546 IC50 > 1000 nM T09572 CX0AM8 57394547 IC50 > 1000 nM T09572 CA3YG5 57395049 IC50 = 700 nM T09572 C19CVL 57395050 IC50 = 40 nM T09572 CC64OF 57396018 IC50 = 20 nM T09572 CX6EZ4 57396019 IC50 = 30 nM T09572 C39VRQ 57396020 IC50 = 50 nM T09572 C74WKY 57396021 IC50 = 34 nM T09572 C8IU0W 57396022 IC50 = 27 nM T09572 CV26IT 57396293 IC50 = 1200 nM T09572 CWY6C2 57396294 IC50 = 4.5 nM T09572 C5SV9H 57396295 IC50 > 1000 nM T09572 C5W2PA 57396309 IC50 > 1000 nM T09572 CWJ94D 57396310 IC50 = 77 nM T09572 C4VP7L 57397816 IC50 = 120 nM T09572 CFXQ13 57397817 IC50 = 14 nM T09572 CNG7U5 57397818 IC50 = 141 nM T09572 C4ULN0 57397819 IC50 = 6 nM T09572 CP9SC0 57397820 IC50 = 27 nM T09572 CW0DC8 57398087 IC50 = 20 nM T09572 C80BEV 57398088 IC50 = 2.8 nM T09572 CM17JZ 57398089 IC50 > 1000 nM T09572 C4HM7E 57398090 IC50 > 1000 nM T09572 CRVU80 57398576 IC50 = 1000 nM T09572 CY6X5S 57399486 IC50 = 15 nM T09572 CRX4D5 57399487 IC50 = 179 nM T09572 C6DY7F 57399740 IC50 = 3.9 nM T09572 C3LYG6 57399741 IC50 = 12 nM T09572 CO2I5T 57399742 IC50 = 62 nM T09572 C0QHE2 57400241 IC50 = 400 nM T09572 C8A1RB 57400242 IC50 > 20000 nM T09572 CJ58YB 57401248 IC50 = 170 nM T09572 C2PC7Q 57401249 IC50 = 20 nM T09572 C2EHU3 57401250 IC50 = 30 nM T09572 C8OAM4 57401251 IC50 = 96 nM T09572 CB0M3A 57401252 IC50 = 30 nM T09572 CEM23S 57401507 IC50 = 19 nM T09572 CF71QU 57401508 IC50 = 70 nM T09572 CF97AB 57401509 IC50 = 6.7 nM T09572 CFY5N4 57401510 IC50 = 8.1 nM T09572 CMVO87 57401511 IC50 > 1000 nM T09572 C8MR2T 57401531 IC50 = 280 nM T09572 C34RTG 57402044 IC50 = 100 nM T09572 CLDV18 57402045 IC50 = 1000 nM T09572 C1ZPE7 57402226 IC50 = 136 nM T09572 CQI16H 57402500 IC50 = 450 nM T09572 CJFE03 57402992 IC50 = 20 nM T09572 CA6O0N 57402993 IC50 = 26 nM T09572 CHIW16 57403264 IC50 = 900 nM T09572 CV8HP7 57403265 IC50 > 1000 nM T09572 CFW3Y9 57403266 IC50 > 1000 nM T09572 CI5D1U 57403267 IC50 > 1000 nM T09572 C9MZU0 57403281 IC50 > 1000 nM T09572 C6WPC8 57403783 IC50 = 180 nM T09572 C7XW5S 57403784 IC50 = 3 nM T09572 CGO38J 57403785 IC50 = 50 nM T09572 C1L8YD 57404359 IC50 = 140 nM T09572 C8SX7A 57404360 IC50 = 110 nM T09572 C0Q1OZ 57404374 IC50 = 440 nM T09572 CXL13R 57521366 IC50 = 5.3 nM T09572 CV9ZT0 57522468 IC50 = 1.9 nM T09572 CRM9Q6 57522701 IC50 = 7.8 nM T09572 C7MT4F 57522703 IC50 = 2 nM T09572 CXUY90 57522704 IC50 = 4.4 nM T09572 C4EUO7 57522816 IC50 = 2.5 nM T09572 C6ZEW3 57522945 IC50 = 3.4 nM T09572 C2J8QB 57522946 IC50 = 2.4 nM T09572 CA2Y5C 57522947 IC50 = 2 nM T09572 CY2GW3 57522948 IC50 = 12 nM T09572 CF9X1V 57522949 IC50 = 5.5 nM T09572 CTPD32 57522950 IC50 = 3.8 nM T09572 C2WD7Q 57523086 IC50 = 1.5 nM T09572 CR7KU6 57845728 IC50 = 10 nM T09572 CPZ0W6 57890345 IC50 = 1 nM T09572 CDU52G 57890370 IC50 = 3 nM T09572 CXBS52 58423512 Ki = 13 nM T09572 C1YJH4 58646147 IC50 = 3.4 nM T09572 C6F4PY 59135471 IC50 = 50 nM T09572 CW8E6V 59135474 EC50 = 30 nM T09572 CO6TL1 59135478 EC50 = 30 nM T09572 CMNY97 59135479 IC50 = 63 nM T09572 C7WM1C 59135482 IC50 = 5.9 nM T09572 C7H4EZ 59135485 IC50 = 560 nM T09572 C2TD0S 59135486 IC50 = 230 nM T09572 CU4Z5R 59135490 IC50 = 340 nM T09572 CG1QE0 59135492 EC50 = 53 nM T09572 CDX98T 59691557 IC50 = 38 nM T09572 CUAY97 59691584 IC50 = 634 nM T09572 CDB34N 59691661 IC50 = 899 nM T09572 CV8U3A 59691704 IC50 = 94 nM T09572 C1MVB2 59835725 IC50 = 8 nM T09572 CZ6EF7 59835728 IC50 = 5 nM T09572 CMG1L8 59835758 IC50 = 8 nM T09572 C4Y8OJ 59835766 IC50 = 35 nM T09572 CG7JS4 59835780 IC50 = 4 nM T09572 C6I5DJ 59835799 IC50 = 12 nM T09572 C65CNM 59835853 IC50 = 10 nM T09572 CY30SJ 59835871 IC50 = 10 nM T09572 CK52CM 59835874 IC50 = 17 nM T09572 C42PAO 59835879 IC50 = 4 nM T09572 C4K2AL 59835909 IC50 = 78 nM T09572 C7SFO5 60130264 IC50 = 1 nM T09572 CA41LH 60130278 IC50 = 2 nM T09572 CIX06K 60130301 IC50 = 10 nM T09572 CIU8R5 60130302 IC50 = 29 nM T09572 C8HYR7 60130337 IC50 = 6 nM T09572 C70YHU 60130349 IC50 = 68 nM T09572 CGF54X 60150483 IC50 = 16 nM T09572 C1XTB5 60168816 IC50 = 70 nM T09572 CK0BH9 60168817 IC50 = 410 nM T09572 CA84NS 60168818 IC50 = 80 nM T09572 C0SJI9 60168913 IC50 = 120 nM T09572 C65BWQ 60168914 IC50 = 720 nM T09572 CE4I2W 60168915 IC50 = 160 nM T09572 C2S9DZ 60168916 IC50 = 1910 nM T09572 CJE24S 60169097 IC50 = 40 nM T09572 CNC6K8 60169098 IC50 = 60 nM T09572 C4BEU6 60169181 IC50 = 100 nM T09572 CD04TV 60169182 IC50 = 60 nM T09572 C7ZS9G 60169184 IC50 = 50 nM T09572 CU3X8A 60169185 IC50 = 80 nM T09572 CM8N0C 60169263 IC50 = 50 nM T09572 CO23GN 66877080 IC50 = 470 nM T09572 CX5H4B 69603769 IC50 = 220 nM T09572 C5AMB2 70681113 IC50 = 7 nM T09572 C59GPT 70681114 IC50 = 160 nM T09572 CO9Z6H 70681115 IC50 = 215 nM T09572 C8BP2U 70681116 IC50 = 158 nM T09572 CV0B8H 70681117 IC50 = 350 nM T09572 C4E1OI 70681197 IC50 = 171 nM T09572 CDH5M3 70681198 IC50 = 142 nM T09572 C14POJ 70681213 IC50 = 15 nM T09572 CV0X2S 70681214 IC50 = 20 nM T09572 C71GOK 70681215 IC50 = 66 nM T09572 CUWS85 70681216 IC50 = 21 nM T09572 CEP43U 70681217 IC50 = 19 nM T09572 C5MZT4 70681299 Ki = 210.86 nM T09572 C7HO6W 70683237 IC50 = 270 nM T09572 CYS92Z 70683241 IC50 = 59 nM T09572 C7FGW6 70683286 IC50 = 116 nM T09572 CL8FX4 70683287 IC50 = 30 nM T09572 CPJN73 70683299 IC50 = 81 nM T09572 CY7LX9 70683300 IC50 = 94 nM T09572 C3NR1Z 70683781 IC50 = 40 nM T09572 CXL0Y8 70685336 IC50 = 96 nM T09572 C53CDS 70685337 IC50 = 9 nM T09572 C08BEC 70685338 IC50 = 15 nM T09572 CDEZ93 70685346 IC50 = 258 nM T09572 CV0WI4 70685347 IC50 = 150 nM T09572 CCXF74 70685395 IC50 = 340 nM T09572 C2WS0G 70685396 IC50 = 86 nM T09572 CHZ6Y4 70685397 IC50 = 270 nM T09572 CYR86Q 70685398 IC50 = 26 nM T09572 CLUJ28 70685407 IC50 = 16 nM T09572 CH9EK3 70685408 IC50 = 69 nM T09572 CZO15N 70685409 IC50 = 4 nM T09572 C3HM0V 70685410 IC50 = 18 nM T09572 CXPR84 70687361 IC50 = 4000 nM T09572 CCRF61 70687470 IC50 = 146 nM T09572 CC3YQ9 70687471 IC50 = 180 nM T09572 CL79FG 70687472 IC50 > 10000 nM T09572 CALE31 70687473 IC50 = 18 nM T09572 C0YZF1 70687477 IC50 = 4 nM T09572 CEZ95O 70687478 IC50 = 237 nM T09572 C3P8VA 70687479 IC50 = 100 nM T09572 CEF40L 70687536 IC50 = 208 nM T09572 CPHD56 70687537 IC50 = 196 nM T09572 C59DKB 70687538 IC50 = 32 nM T09572 COY81J 70687549 IC50 = 31 nM T09572 CT8A1Y 70687550 IC50 = 26 nM T09572 C5UI4H 70687551 IC50 = 31 nM T09572 CE8FW5 70687552 IC50 = 26 nM T09572 CE6M1I 70688018 IC50 = 10 nM T09572 CGX8O4 70689518 IC50 > 10000 nM T09572 CT6NC1 70689519 IC50 = 91 nM T09572 C7GY1R 70689520 IC50 = 116 nM T09572 C7HY1M 70689525 IC50 = 27 nM T09572 C8K6GH 70689526 IC50 = 156 nM T09572 C1O6EB 70689527 IC50 = 59 nM T09572 CVYC02 70689594 IC50 = 40 nM T09572 C5JZ0U 70689595 IC50 = 54 nM T09572 C39VHU 70689596 IC50 = 91 nM T09572 C6RD9J 70689612 IC50 = 11 nM T09572 CQA6H0 70691333 IC50 = 22 nM T09572 C4GOS0 70691526 IC50 > 3000 nM T09572 CHX2V3 70691648 IC50 = 690 nM T09572 CJ8C3H 70691649 IC50 = 115 nM T09572 CC1G3W 70691650 IC50 = 33 nM T09572 CJ7VK5 70691651 IC50 = 45 nM T09572 C6HPK5 70691652 IC50 = 15 nM T09572 CYJS32 70691653 IC50 = 7 nM T09572 C7NI4U 70691655 IC50 > 10000 nM T09572 C2BEO6 70691656 IC50 = 67 nM T09572 CJQA94 70691720 IC50 = 107 nM T09572 C27ECJ 70691721 IC50 = 62 nM T09572 C9N0ZJ 70691722 IC50 = 24 nM T09572 CB71AI 70691723 IC50 = 230 nM T09572 CDI17T 70691724 IC50 = 4125 nM T09572 CM1W5S 70691725 IC50 = 35 nM T09572 CD3N0U 70691736 IC50 = 10 nM T09572 C31VLM 70691737 IC50 = 225 nM T09572 CK03LJ 70691738 IC50 = 14 nM T09572 C8CL4G 70691739 IC50 = 56 nM T09572 C4PH6G 70693620 IC50 = 3800 nM T09572 C2EGO8 70693732 IC50 = 30 nM T09572 C9Y0GP 70693733 IC50 = 3 nM T09572 C50FLK 70693734 IC50 = 10 nM T09572 C94PEU 70693737 IC50 = 33 nM T09572 C7R6XS 70693792 IC50 = 73 nM T09572 C0MN5C 70693793 IC50 = 83 nM T09572 CKTG14 70693794 IC50 = 575 nM T09572 C7OWB6 70693795 IC50 = 1800 nM T09572 CS79JT 70693796 IC50 = 57 nM T09572 CYE09Q 70693807 IC50 = 13 nM T09572 CHT37L 70693808 IC50 = 27 nM T09572 CY48LR 70693809 IC50 = 45 nM T09572 CO4G8Z 70693810 IC50 = 31 nM T09572 CA9NO7 70695565 Ki = 21 nM T09572 CYP9F5 70695851 IC50 = 246 nM T09572 C0CZ8Y 70695852 IC50 = 7300 nM T09572 C0OYQ4 70695853 IC50 = 163 nM T09572 C20EKP 70695854 IC50 = 213 nM T09572 CZ92AV 70695855 IC50 = 23 nM T09572 CJ61GF 70695859 IC50 = 208 nM T09572 C5SK0T 70695860 IC50 = 636 nM T09572 C6RM8L 70695913 IC50 = 670 nM T09572 CM6JE8 70695914 IC50 = 201 nM T09572 CY17NO 70695915 IC50 = 220 nM T09572 C7CF9D 70695916 IC50 = 182 nM T09572 C35IPG 70695917 IC50 = 255 nM T09572 CIW1D8 70695918 IC50 = 23 nM T09572 C8UD2I 70695929 IC50 = 170 nM T09572 CG0D4A 70695930 IC50 = 112 nM T09572 CW71LQ 70696356 IC50 = 0.76 nM T09572 C87MGT 71226277 IC50 = 20 nM T09572 C4J8MI 71226400 IC50 = 20 nM T09572 C1WP5Y 71226964 IC50 = 16 nM T09572 C1B9KV 71227161 IC50 = 45 nM T09572 CI8E6U 71227163 IC50 = 20 nM T09572 C26UYS 71450863 Ki = 3.9 nM T09572 CAEM97 71450908 Ki = 1188 nM T09572 CFEI76 71660915 IC50 = 40 nM T09572 C9I3GO 71714121 Ki = 14 nM T09572 CB2S3Z 71716477 IC50 = 4130 nM T09572 CF18UN 71716478 IC50 = 1040 nM T09572 CB0O6P 71716479 IC50 = 510 nM T09572 C5P6AH 71716480 IC50 = 5650 nM T09572 C0WF7K 71717084 IC50 = 3100 nM T09572 C2TNF8 71717085 IC50 = 10000 nM T09572 C0IL4X 71717086 IC50 = 2780 nM T09572 CNWZ92 71717700 IC50 = 340 nM T09572 CCLZ30 71717701 IC50 = 10000 nM T09572 CSZU90 71718317 IC50 = 210 nM T09572 C4JFS2 71718318 IC50 = 130 nM T09572 CIK12B 71718319 IC50 = 440 nM T09572 CKQ23I 71718910 IC50 = 180 nM T09572 CZOR72 71718911 IC50 = 7110 nM T09572 CMP54N 71719522 IC50 = 320 nM T09572 CVE7I3 71719523 IC50 = 190 nM T09572 CE0IQ4 71719524 IC50 = 2000 nM T09572 CJ9SP8 71719526 IC50 = 90 nM T09572 CK21FD 71720118 IC50 = 300 nM T09572 C2IJ4F 71720119 IC50 = 540 nM T09572 C3OM4R 71720120 IC50 = 80 nM T09572 C7D6VL 71720121 IC50 = 2010 nM T09572 CR1CA7 71730269 IC50 = 8.7 nM T09572 CF14LT 71730661 IC50 = 24 nM T09572 C7LX2Q 71730663 IC50 = 16 nM T09572 C9SN7I 71731948 IC50 = 33 nM T09572 CS5PA1 71732078 IC50 = 17 nM T09572 C8VJ7O 73356649 IC50 = 230 nM T09572 C1Q2HP 76324350 Ki <= 1500 nM T09572 C6BEM8 86582974 IC50 = 35 nM T09572 C1LJW9 89689924 IC50 = 12 nM T09572 C7S8ON 89690124 IC50 = 72 nM T09572 CHP67R 89690222 IC50 > 1000 nM T09572 CX01FB 89690237 IC50 = 92 nM T09572 CD3RU2 89690239 IC50 = 410 nM T09572 CP4Z8K 89690292 IC50 = 240 nM T09572 C9KT2U 89690293 IC50 > 1000 nM T09572 CK6AR1 89690294 IC50 > 1000 nM T09572 CRQ1S5 89690318 IC50 = 42 nM T09572 C7Y3BZ 89690333 IC50 > 1000 nM T09572 C24NIJ 89690365 IC50 = 37 nM T09572 C4W0KZ 89690368 IC50 = 380 nM T09572 C6TG1E 89690379 IC50 = 47 nM T09572 CJ42SW 89690396 IC50 = 24 nM T09572 C8IZG5 89690573 IC50 = 120 nM T09572 CG9X7P 89690574 IC50 = 7.7 nM T09572 CSQ84D 89690600 IC50 = 78 nM T09572 CLPT46 89690607 IC50 = 25 nM T09572 CJ6V7S 89690622 IC50 = 95 nM T09572 CN8VQ4 89690864 IC50 = 35 nM T09572 C8KT3J 89690957 IC50 = 34 nM T09572 CLI0S8 89690968 IC50 > 1000 nM T09572 CG1LS2 89690973 IC50 = 160 nM T09572 CQ0YA2 89691019 IC50 = 76 nM T09572 CE04BI 89691032 IC50 = 45 nM T09572 C0AYJ8 89691044 IC50 = 17 nM T09572 CU1X2I 89691057 IC50 = 85 nM T09572 C20YIN 89691065 IC50 = 41 nM T09572 C0XB6N 89691096 IC50 = 16 nM T09572 CE9C1Y 89691111 IC50 > 1000 nM T09572 CQB43P 89691143 IC50 = 100 nM T09572 CENL63 89691144 IC50 = 73 nM T09572 CP3I8Z 89691162 IC50 = 28 nM T09572 CZ5M8J 89691193 IC50 = 240 nM T09572 CUF15D 89691216 IC50 = 600 nM T09572 CZV10H 89691247 IC50 = 37 nM T09572 C9OV4S 89691264 IC50 > 1000 nM T09572 CZSL41 89691284 IC50 = 90 nM T09572 C9J6WL 89691349 IC50 > 1000 nM T09572 CHAI64 89691416 IC50 = 44 nM T09572 CX90VG 89691439 IC50 = 26 nM T09572 C2ZY0O 89691440 IC50 = 150 nM T09572 CP93JH 89691535 IC50 = 34 nM T09572 C50ODP 89702205 IC50 > 1000 nM T09572 CXR3A4 89702226 IC50 = 24 nM T09572 C4B8VD 89702233 IC50 = 17 nM T09572 CD94UH 89702341 IC50 > 1000 nM T09572 C0GS9K 89702355 IC50 = 180 nM T09572 C70YGQ 89702382 IC50 > 1000 nM T09572 CQE21B 89702566 IC50 = 14 nM T09572 C7BNF2 89798657 IC50 = 10 nM T09572 CYW7P8 89798658 IC50 = 13 nM T09572 C6BID5 90469437 IC50 = 38 nM T09572 C2IN9R 90666094 IC50 = 15 nM T09572 C9R7TC 90666095 IC50 = 3 nM T09572 C0KWI9 90666096 IC50 = 0.9 nM T09572 CXM6Q2 90666097 IC50 = 8 nM T09572 CMU2J7 90666098 IC50 = 34 nM T09572 CS71ZE 90666251 IC50 = 1004 nM T09572 CKV42Z 90666252 IC50 = 172 nM T09572 CIA63Z 90666253 IC50 = 817 nM T09572 C8YHD2 90666254 IC50 = 271 nM T09572 C90CGQ 90666255 IC50 = 138 nM T09572 CC07QH 90666256 IC50 = 47 nM T09572 CMO4T3 90666257 IC50 = 259 nM T09572 CWM0V6 90666258 IC50 = 3250 nM T09572 CT53ER 90666259 IC50 = 184 nM T09572 C6H5CY 90666260 IC50 = 46 nM T09572 CI2AQ3 90666261 IC50 = 651 nM T09572 CR0NA6 90666262 IC50 = 11 nM T09572 C8B5IV 90666263 IC50 = 27 nM T09572 CX6ZO5 90666264 IC50 = 15 nM T09572 C7J1IK 90666265 IC50 = 14 nM T09572 CCX69F 90666266 IC50 = 12 nM T09572 C45NLU 90666267 IC50 = 96 nM T09572 CR9HQ7 91759552 IC50 = 70 nM T09572 CS5A8P 91759588 IC50 = 57 nM T09572 C8XFV3 101007561 IC50 = 5128.61 nM T09572 CJMR89 117798671 IC50 = 90 nM T09572 CO2L5Z 117798675 IC50 = 140 nM T09572 C48XKW 117798680 IC50 = 230 nM T09572 CYU6B5 117798688 IC50 = 210 nM T09572 CN84IO 117798692 IC50 = 170 nM T09572 C54ISX 117798744 IC50 = 31 nM T09572 CM3F4S 117798780 IC50 = 130 nM T09572 CI2K4J 117816748 IC50 = 74 nM T09572 CL1Z6U 117816753 IC50 = 110 nM T09572 C1A3HV 117816804 IC50 = 43 nM T09572 CIET51 121386280 IC50 > 1000 nM T09572 C09BDS 122184557 IC50 = 2 nM T09572 CK35BS 122184558 IC50 = 8 nM T09572 CED1I6 122184559 IC50 = 470 nM T09572 C6JG4U 122184560 IC50 = 8 nM T09572 CTJO50 122184561 IC50 = 3 nM T09572 CZ1MA3 122184562 IC50 = 11 nM T09572 CH37IW 122184563 IC50 = 5 nM T09572 C5JTD9 122184564 IC50 = 36 nM T09572 CF2YG3 122184565 IC50 = 15 nM T09572 CRPW64 122184566 IC50 = 33 nM T09572 CACV74 122184567 IC50 = 700 nM T09572 CMR65S 122184568 IC50 = 420 nM T09572 CNC14U 122184569 IC50 = 360 nM T09572 CFC4P3 122184570 IC50 = 247 nM T09572 CJR48E 122184670 IC50 = 17 nM T09572 C7YA0Q 122184671 IC50 = 4 nM T09572 C6RP0N 122184672 IC50 = 21 nM T09572 CLP36J 122184673 IC50 = 151 nM T09572 CQT2K8 122184674 IC50 = 2530 nM T09572 CSIL49 122184687 IC50 = 251 nM T09572 CN0CB1 122184690 IC50 > 3000 nM T09572 C5Y0KX 122184691 IC50 = 95 nM T09572 C18ZKO 122184692 IC50 = 20 nM T09572 C0XJK1 122184693 IC50 = 6 nM T09572 C97APV 122184694 IC50 = 10 nM T09572 CLK94O 122184695 IC50 = 3 nM T09572 CWSF63 122184696 IC50 = 24 nM T09572 CW8L5K 122184697 IC50 = 9 nM T09572 CI4SF6 122184698 IC50 = 15 nM T09572 CDHE98 122184699 IC50 = 4 nM T09572 CIU9W5 122184700 IC50 = 92 nM T09572 CU2PG6 122184701 IC50 = 13 nM T09572 CKG74I 122184702 IC50 = 13 nM T09572 CZ0I1K 122184703 IC50 = 186 nM T09572 C65COE 122184704 IC50 = 15 nM T09572 CHS9N7 122184705 IC50 = 22 nM T09572 CWM9Q7 122184706 IC50 = 10 nM T09572 CZ2VB1 122184832 IC50 = 7 nM T09572 CJ0V1K 122184885 IC50 = 25 nM T09572 C2CHR3 123471111 IC50 = 34 nM T09572 CY6WF8 127025096 IC50 = 210 nM T09572 CELT51 127025110 IC50 = 270 nM T09572 C5IK3Q 127025395 IC50 = 94 nM T09572 CG28ML 127028868 IC50 = 69 nM T09572 CYP9E6 127028869 IC50 = 99 nM T09572 CS9YL7 127029623 IC50 = 3.8 nM T09572 CJO31V 127029624 IC50 = 3 nM T09572 C5P9RC 127029625 IC50 > 1000 nM T09572 C34PRW 127029630 IC50 > 1000 nM T09572 CK18EL 127029631 IC50 > 1000 nM T09572 C7S2DW 127029632 IC50 = 990 nM T09572 CFN3Y4 127029759 IC50 = 150 nM T09572 CZDO76 127030069 IC50 = 22 nM T09572 C8WD7N 127030070 IC50 = 23 nM T09572 C9GHX6 127030071 IC50 = 39 nM T09572 C0OKZ3 127030367 IC50 = 30 nM T09572 CEP0T2 127030368 IC50 = 35 nM T09572 CF4V0J 127031338 IC50 = 11 nM T09572 CZ6A2D 127031339 IC50 = 43 nM T09572 CZ6P7H 127031354 IC50 = 40 nM T09572 C5BTJ9 127031355 IC50 = 50 nM T09572 CB7XP0 127031356 IC50 = 39 nM T09572 C4F3QY 127031621 IC50 = 28 nM T09572 CB7Y6D 127031622 IC50 = 15 nM T09572 CUO4V9 127031623 IC50 = 44 nM T09572 CFG8U2 127031907 IC50 = 1000 nM T09572 CI9ZB4 127031908 IC50 = 61 nM T09572 C3NE8G 127031909 IC50 = 150 nM T09572 CYZH79 127032787 IC50 = 1200 nM T09572 C7AK5Z 127033095 IC50 = 75 nM T09572 C3UKI0 127033096 IC50 = 200 nM T09572 C9MD2C 127033672 IC50 = 140 nM T09572 C1YR3E 127033673 IC50 = 220 nM T09572 C5ITG3 127033945 IC50 = 70 nM T09572 C05XCQ 137635978 IC50 = 3235.94 nM T09572 C5PV0E 137640352 Ki = 15 nM T09572 CK5HG6 137644041 EC50 = 1042 nM T09572 CXH16S 137655884 IC50 = 1862.09 nM T09572 CME6U8 137657882 IC50 = 4265.8 nM T09572 CFC7Z0 155516078 IC50 = 17380 nM T09572 CX1A0M 155516949 IC50 = 6.8 nM T09572 C4TY3K 155520135 IC50 = 890 nM T09572 CLJU26 155522708 IC50 = 5100 nM T09572 CG4YE1 155524512 IC50 = 4300 nM T09572 CQ9PM4 155527803 IC50 = 129 nM T09572 C4AJ7V 155528494 IC50 = 105 nM T09572 C9RUQ4 155531314 IC50 = 4.9 nM T09572 CJ2S8K 155538229 IC50 = 40 nM T09572 CRC90P 155541584 IC50 > 3000 nM T09572 C0E4VQ 155562407 IC50 = 228 nM T09572 C6CTA5 155569743 IC50 = 1300 nM T09572 D00AWM 9826520 IC50 = 0.5012 nM T09572 D00MSU 22254580 IC50 = 492 nM T09572 D01NOZ 16665072 IC50 = 28 nM T09572 D01OYC 10262766 IC50 = 5310 nM T09572 D01OZL 10466405 IC50 = 36 nM T09572 D01PFN 22254575 IC50 = 432 nM T09572 D02FQG 54579974 IC50 = 25 nM T09572 D02QXF 11776033 IC50 = 860 nM T09572 D03BIQ 11189610 IC50 = 100 nM T09572 D03CDM 10399674 IC50 = 1070 nM T09572 D03FJK 10083869 IC50 = 20 nM T09572 D03FNQ 11281523 IC50 = 9 nM T09572 D03SEC 10443307 IC50 = 789 nM T09572 D04OOK 3787955 Ki = 7500 nM T09572 D05HFC 10466406 IC50 = 199 nM T09572 D05MEW 14514271 Ki = 302 nM T09572 D05QTT 11691555 Ki = 8.5 nM T09572 D05TVU 22254551 IC50 = 90 nM T09572 D05UZY 11539096 IC50 = 3 nM T09572 D05ZUX 44207909 EC50 = 128.82 nM T09572 D06KLQ 44403742 IC50 = 16 nM T09572 D07EPU 11155432 IC50 = 164 nM T09572 D07HQP 10353806 IC50 = 580 nM T09572 D07IUE 22254582 IC50 = 53 nM T09572 D07WFH 3575822 Ki = 7500 nM T09572 D07XEA 10332650 IC50 = 137 nM T09572 D08OQO 10198125 IC50 = 437 nM T09572 D08SOE 11994411 IC50 = 0.39 nM T09572 D09RGM 3747253 Ki = 1700 nM T09572 D0AT3U 44418001 IC50 = 1000 nM T09572 D0AT5N 56835134 IC50 = 1 nM T09572 D0AU6T 10377914 IC50 = 132 nM T09572 D0C5RQ 10300618 Ki = 19.95 nM T09572 D0C7ED 57523087 IC50 = 1.5 nM T09572 D0C9DP 11153928 IC50 = 9 nM T09572 D0D2PL 22266820 IC50 = 1590 nM T09572 D0ES2Y 22254604 IC50 = 32 nM T09572 D0F3VX 10466478 IC50 = 606 nM T09572 D0G6DS 10421932 IC50 = 818 nM T09572 D0I7FK 10038053 IC50 = 640 nM T09572 D0J7MM 11440762 IC50 = 390 nM T09572 D0K0KR 9895867 IC50 = 160 nM T09572 D0K5JA 10399494 IC50 = 361 nM T09572 D0K5QJ 11188955 IC50 = 70 nM T09572 D0K5XL 11440885 IC50 = 1930 nM T09572 D0L4WB 10244148 IC50 = 349 nM T09572 D0LJ4Q 10420382 IC50 = 1100 nM T09572 D0M3HZ 9927967 IC50 = 15 nM T09572 D0N6OL 11452268 IC50 = 58 nM T09572 D0P4CQ 10377822 IC50 = 191 nM T09572 D0P5QW 57521365 IC50 = 1.1 nM T09572 D0S7IJ 10083101 IC50 = 823 nM T09572 D0U1OX 10421933 IC50 = 201 nM T09572 D0V2IR 10353807 IC50 = 326 nM T09572 D0V9KF 22254540 IC50 = 722 nM T09572 D0W7ZM 10443853 IC50 = 614 nM T95558 D0EY0A 42636350 IC50 = 80 nM T95558 D02NRD 9865421 IC50 > 10000 nM T95558 D0M0NT 46926360 IC50 > 30000 nM T95558 D0U5NY 10435589 IC50 > 10000 nM T95558 CL21WZ 3168855 IC50 > 20000 nM T95558 C9A4YR 11892264 IC50 = 600 nM T95558 CKRN07 25118654 IC50 > 100000 nM T95558 CH3L6V 25192656 IC50 = 28000 nM T95558 C7URI3 25235407 IC50 > 10000 nM T95558 CM2G4X 42797508 IC50 > 50000 nM T95558 CAX57D 46850597 IC50 > 30000 nM T95558 CCY12P 46946735 IC50 > 50000 nM T95558 CW6EA0 52917768 IC50 = 1300 nM T95558 CBHT83 56840376 IC50 > 50000 nM T95558 CV8W4T 56933229 IC50 > 10000 nM T95558 C0QMK7 58064355 IC50 > 10000 nM T95558 C03EFU 59440893 IC50 > 30000 nM T95558 CW2LD6 70686525 IC50 > 20000 nM T95558 CY08FK 71571356 IC50 > 10000 nM T95558 C49QLP 71602372 IC50 > 10000 nM T95558 CR13XU 71602433 IC50 > 10000 nM T95558 C38SOR 71602434 IC50 > 10000 nM T95558 C3ZR8K 71603028 IC50 > 10000 nM T95558 CP97OC 71603093 IC50 > 10000 nM T95558 CAHY94 71603095 IC50 > 10000 nM T95558 C3IHF5 71603097 IC50 > 10000 nM T95558 CQ1K6W 71603210 IC50 > 10000 nM T95558 C9D1QC 71603211 IC50 > 10000 nM T95558 C8JKL2 71603212 IC50 > 10000 nM T95558 CJTR16 71766152 IC50 = 20 nM T95558 CVNX92 71766153 IC50 = 34 nM T95558 CGSV54 71766156 IC50 = 1.3 nM T95558 C5JV1P 71812623 IC50 > 20000 nM T95558 C9NE1Y 89853814 IC50 = 31 nM T95558 C47OKQ 89854212 IC50 = 17 nM T95558 C9FCS1 90644592 IC50 = 10000 nM T95558 CEC50G 91884614 IC50 > 30000 nM T95558 C4J9DB 118916617 IC50 = 120 nM T95558 C8EF1P 118916631 IC50 = 180 nM T95558 C2RBF7 118918048 IC50 = 2 nM T95558 CSBO65 122179027 IC50 > 30000 nM T95558 C75SHP 122188924 IC50 > 100000 nM T95558 C8HN7U 122189249 IC50 > 40000 nM T95558 CNV03S 122189255 IC50 > 100000 nM T95558 C48MIR 127034747 IC50 > 12000 nM T95558 C8UX4Q 127034759 IC50 = 540 nM T95558 CTM46H 127034938 IC50 = 500 nM T95558 C8VYP5 127034939 IC50 = 2200 nM T95558 C4OB5T 127035411 IC50 = 3 nM T95558 CUQ1Z6 127035947 IC50 = 140 nM T95558 CRI96L 127035948 IC50 = 1600 nM T95558 CTN0J4 127035949 IC50 = 300 nM T95558 CZV70W 127035950 IC50 = 60 nM T95558 CJ5OX8 127035951 IC50 = 3460 nM T95558 C1M5NI 127035952 IC50 = 4 nM T95558 CGET82 134586817 IC50 = 579 nM T95558 C6B5US 137628648 IC50 > 10000 nM T95558 C42PLT 145962320 IC50 > 50000 nM T95558 CLP89H 145963384 IC50 > 50000 nM T95558 C4MQU9 145980134 IC50 = 37 nM T95558 CQR0O2 155524798 IC50 = 17 nM T20302 D0ZD2M 16720766 IC50 > 1000 nM T20302 CP81AT 11655576 IC50 = 100000 nM T20302 C0YCU9 59671423 IC50 > 10000 nM T72702 D01FFA 72301 IC50 = 22.78 nM T72702 D0Y3KG 3121 IC50 = 1500000 nM T72702 D07SDQ 969516 IC50 = 13.16 nM T72702 D0I7IB 5222465 IC50 = 1000000 nM T72702 D0M8FD 4261 IC50 = 6000 nM T72702 C1WK2E 5417 IC50 = 14.98 nM T72702 CGO94B 34458 IC50 = 8.35 nM T72702 CQD56Z 73299 IC50 = 0.221 nM T72702 CEC2H3 73309 IC50 = 0.054 nM T72702 CHV19R 127026 IC50 = 6.46 nM T72702 C1ND9W 161665 IC50 = 152.43 nM T72702 C5Y6QK 261619 IC50 = 12.17 nM T72702 CHB7D2 453215 IC50 = 187.26 nM T72702 CS5PK2 640180 IC50 = 0.053 nM T72702 C2K4YZ 715840 IC50 = 13.37 nM T72702 CG1I7T 1550234 IC50 > 200 nM T72702 C4L7CX 1550330 IC50 = 0.26 nM T72702 CPU3R4 1550699 IC50 > 200 nM T72702 CC40IA 1909086 IC50 = 0.94 nM T72702 C5LGJ1 5282362 IC50 = 0.12 nM T72702 CM3T9J 5377817 IC50 = 15.39 nM T72702 C85WLD 5927890 IC50 = 141.98 nM T72702 CUYD15 9986341 IC50 = 0.095 nM T72702 CH5ZD8 10079039 IC50 = 9.581 nM T72702 CFJR86 11600024 IC50 = 36 nM T72702 C2VEB7 11753144 IC50 = 4.678 nM T72702 C56NRA 11957383 IC50 = 20 nM T72702 CF4W7L 12269810 IC50 = 968.9 nM T72702 CR0EG4 12302577 IC50 = 1.294 nM T72702 CCLH20 12313091 IC50 = 36.41 nM T72702 C4QK6B 13518132 IC50 = 15.95 nM T72702 C5U0AR 14189384 IC50 = 0.035 nM T72702 C6ZUG1 15061351 IC50 = 63.06 nM T72702 C5B1CH 15604798 Ki = 33 nM T72702 C6VZ1N 15942655 Ki = 800 nM T72702 CC5VF9 16007120 Ki = 2.6 nM T72702 CC7Y0D 16066741 IC50 = 590 nM T72702 CVB82P 17809181 IC50 = 89 nM T72702 C52BRP 21120798 IC50 = 0.28 nM T72702 CM87QX 21633122 IC50 = 10.61 nM T72702 CYE8Z0 23646853 Ki = 335 nM T72702 CF7JA3 23646854 Ki = 270 nM T72702 CRI3Y5 23646855 Ki = 350 nM T72702 CHUX39 23646856 Ki = 61.5 nM T72702 C6IT8J 23646857 Ki = 57 nM T72702 CFT69V 23646858 Ki = 130 nM T72702 C93HOM 23646859 Ki = 110 nM T72702 CTZ1K0 23646860 Ki = 100 nM T72702 CV3B5R 23646861 Ki = 330 nM T72702 CI2Q6A 23646862 Ki = 830 nM T72702 C2WK6E 23646863 Ki = 57 nM T72702 CVCZ14 23646864 Ki = 47 nM T72702 C2N6OU 23646865 Ki = 100 nM T72702 C6WGE2 23646866 Ki = 88 nM T72702 C54VSD 23646867 Ki = 28 nM T72702 C3GAY7 23646868 Ki = 60 nM T72702 CCD14G 23646869 Ki = 190 nM T72702 CXOF04 23646870 Ki = 58 nM T72702 C3W5LA 23646871 Ki = 160 nM T72702 CW5CX0 23646872 Ki = 130 nM T72702 CG91AX 23646873 Ki = 2700 nM T72702 CE75AW 23646874 Ki = 155 nM T72702 C4MO5W 23646875 Ki = 17000 nM T72702 CB8VS0 23646876 Ki = 130000 nM T72702 CU1L5O 23646877 Ki = 2000 nM T72702 C1COD6 23646878 Ki = 9500 nM T72702 CM5F3L 23646879 Ki = 220 nM T72702 CD01TF 23646880 Ki = 610 nM T72702 C58PMJ 23646881 Ki = 850 nM T72702 CXHL61 23646883 Ki = 72 nM T72702 C40ESI 44407593 IC50 = 120 nM T72702 CG3F5V 44407595 IC50 = 130 nM T72702 CJT68D 44407597 IC50 = 27 nM T72702 CH5L1B 44407599 IC50 = 31 nM T72702 C6M0JA 44407601 IC50 = 92 nM T72702 CLX0M1 44407607 IC50 = 210 nM T72702 CM8V2B 44407609 IC50 = 570 nM T72702 C4O0GT 44407611 IC50 = 180 nM T72702 CFZ12R 44407613 IC50 = 590 nM T72702 CMIF29 44407615 IC50 = 110 nM T72702 CX79CA 44407617 IC50 = 600 nM T72702 CCQ4O8 44407688 IC50 = 1600 nM T72702 C26PJY 44407814 IC50 = 47 nM T72702 C3GW8V 44407816 IC50 = 17 nM T72702 C7UCD4 44407818 IC50 = 150 nM T72702 C4S6FL 44407820 IC50 = 180 nM T72702 C51QCV 44407822 IC50 = 16 nM T72702 C5VW4Y 44407825 IC50 = 43 nM T72702 C2E0JC 44407841 IC50 = 48 nM T72702 C7QK8H 44407843 IC50 = 16 nM T72702 C36OIS 44407846 IC50 = 63 nM T72702 C3KTD2 44407848 IC50 = 170 nM T72702 CVSE54 44407974 IC50 = 240 nM T72702 C9N1SL 44407977 IC50 = 130 nM T72702 CW9L7N 44407979 IC50 = 2400 nM T72702 CUPX36 44407981 IC50 = 190 nM T72702 C71TKS 44407986 IC50 = 73 nM T72702 CGBR83 44407988 IC50 = 290 nM T72702 CZ69GQ 44408053 IC50 = 97 nM T72702 CJ3P4D 44408067 IC50 = 67 nM T72702 CG6H0U 44415561 Ki = 220 nM T72702 C3LCV6 44415581 Ki = 81 nM T72702 COY95B 44415713 Ki = 15 nM T72702 CSM18R 44415714 Ki = 20 nM T72702 CE3NH9 44415737 Ki = 1.3 nM T72702 CQ25XV 44421779 IC50 = 1300 nM T72702 CAP6F0 44421800 IC50 = 19000 nM T72702 CV1FC6 44421801 IC50 = 19000 nM T72702 CYE0W3 44421802 IC50 = 2200 nM T72702 CP1O3U 44421803 IC50 = 860 nM T72702 CNPU85 44421804 IC50 = 91000 nM T72702 CS3TC8 44421807 IC50 = 191000 nM T72702 C71ECV 44421808 IC50 = 8500 nM T72702 CF3AQ6 44421810 IC50 = 2400 nM T72702 CRX5K3 44421813 IC50 = 4200 nM T72702 C8OMB1 44421816 IC50 = 4200 nM T72702 C7VY0B 44421822 IC50 = 3200 nM T72702 CVJ85S 44421826 IC50 = 690 nM T72702 C4DYF3 44421831 IC50 = 300 nM T72702 CWVX31 44421837 IC50 = 150 nM T72702 CD58ZY 44421845 IC50 = 180 nM T72702 CQX8V2 44421851 IC50 = 300 nM T72702 CLV9Z6 46905970 IC50 = 380 nM T72702 CSX46R 57580978 IC50 = 376.52 nM T72702 C0B7OW 71508815 IC50 = 12.61 nM T72702 CA2LK1 71508816 IC50 = 118.8 nM T72702 C5GYN6 71508817 IC50 = 1501.43 nM T72702 CQDU73 71508864 IC50 = 555.37 nM T72702 CDB2C5 71508865 IC50 = 3.75 nM T72702 CQ2N0J 71508866 IC50 = 201.93 nM T72702 C2K3CV 71524613 IC50 = 6.75 nM T72702 C50YDS 71716758 IC50 = 38.59 nM T72702 CGU06V 71717958 IC50 = 8.79 nM T72702 CQY27U 71719784 IC50 = 16.8 nM T72702 CPK1H2 135450157 Ki = 2 nM T72702 CBU2E4 135469660 Ki = 44 nM T72702 CSW47P 135528873 Ki = 13 nM T72702 CQ3YN8 135530560 Ki = 4 nM T72702 C9Q7BK 135543038 Ki = 35 nM T72702 C9Q1TW 135543055 Ki = 43 nM T72702 C43KYW 135547926 Ki = 14 nM T72702 C89IBC 135547960 Ki = 13 nM T72702 CE2B7G 136094792 Ki = 12 nM T72702 CAW5Q0 136094793 Ki = 12 nM T72702 C2MZX6 137632271 IC50 = 0.028 nM T72702 C9HUM3 137634350 IC50 = 0.801 nM T72702 C61AWC 137635791 IC50 = 0.64 nM T72702 C3I4UR 137639091 IC50 = 0.078 nM T72702 CKNA04 137652993 IC50 = 0.221 nM T72702 D02KKU 12313704 IC50 = 0.221 nM T72702 D0IO0I 6474893 IC50 > 200 nM T72702 D0J6RQ 6437306 IC50 = 2.58 nM T72702 D0L7OM 6917970 IC50 = 104.58 nM T72702 D0PG8M 5467477 IC50 = 0.96 nM T72702 D0SJ2Q 10494 IC50 = 4.975 nM T72702 D0W1PV 6918328 IC50 = 200 nM T40103 D0J6AU 10152654 IC50 > 10 nM T40103 D0HM5J 118253852 IC50 > 20000 nM T40103 D04ZIJ 5478883 IC50 > 100000 nM T40103 CMW5A9 4430623 Ki = 251000 nM T40103 CESY50 5288259 IC50 > 500 nM T40103 C0XQP7 6917747 IC50 > 100000 nM T40103 CN26IL 9547980 Ki > 30000 nM T40103 COBW38 9821383 IC50 > 100000 nM T40103 CLB5G0 10025017 IC50 > 500 nM T40103 C2N9CS 10062713 IC50 = 18 nM T40103 CSO96K 10127748 IC50 > 5000 nM T40103 CKZ15P 10129236 IC50 > 5000 nM T40103 C5NEX6 10174161 IC50 > 5000 nM T40103 C1YR4T 10174359 IC50 > 2000 nM T40103 CY7DQ2 10288811 IC50 > 2000 nM T40103 CF5NB6 10668225 Ki = 160000 nM T40103 C5GD2S 10746284 Ki = 137000 nM T40103 CT9D8H 10765270 Ki = 210000 nM T40103 CG7D0X 10770036 Ki = 93000 nM T40103 CN0F8E 11199915 IC50 > 100000 nM T40103 CFI8L5 11502586 IC50 > 13000 nM T40103 C98EQF 11545899 IC50 = 230 nM T40103 CU57OC 11705307 IC50 > 100000 nM T40103 C8D7BS 11771234 Ki = 3700 nM T40103 CP4H9E 12737307 Ki = 89000 nM T40103 C31MCN 13186896 IC50 > 100000 nM T40103 C6XPN4 16664855 IC50 = 2653 nM T40103 CFY7O6 22988664 Ki = 354000 nM T40103 CZ8DI1 23643986 Ki = 137 nM T40103 CZPF48 23648277 IC50 > 50000 nM T40103 CN0VA7 24822701 IC50 > 50000 nM T40103 CQU38W 24900755 IC50 > 30000 nM T40103 C2S8VB 24901099 IC50 = 6591 nM T40103 CIN28B 24901100 IC50 > 10000 nM T40103 CD2EH0 24901101 IC50 > 10000 nM T40103 CS7B3F 24901102 IC50 > 100000 nM T40103 CGI0U2 25023791 Ki > 10000 nM T40103 C73KLE 25209862 IC50 > 30000 nM T40103 C25ELB 44143088 IC50 = 125.89 nM T40103 C9QDC0 44143091 IC50 = 645.65 nM T40103 C8Y9NQ 44219712 IC50 > 100000 nM T40103 C5VBI8 44368657 Ki = 260000 nM T40103 CP7KW2 44391459 IC50 = 580 nM T40103 C9W3HN 44391474 IC50 = 40 nM T40103 CV71WQ 44391475 IC50 = 8300 nM T40103 CTRP74 44394287 IC50 = 5000 nM T40103 CP7X6J 44394353 IC50 > 5000 nM T40103 C79NFU 44394458 IC50 > 12000 nM T40103 CD73QR 44398649 Ki = 0.46 nM T40103 CHQF16 44398651 Ki = 1.4 nM T40103 C4ALQ9 44398659 Ki > 13000 nM T40103 CD18YP 44402055 IC50 > 2000 nM T40103 CU8TB9 44402056 IC50 > 5000 nM T40103 CD4TP7 44402158 IC50 > 13000 nM T40103 CO6BG2 44402160 IC50 > 13000 nM T40103 C0AJC4 44402175 IC50 > 13000 nM T40103 CX9O2Q 44402263 IC50 > 13000 nM T40103 C89MOT 44402291 IC50 > 13000 nM T40103 C4ZMP9 44408016 IC50 > 13000 nM T40103 C25RIN 44408049 IC50 = 190 nM T40103 CS6X7V 44426055 IC50 > 100000 nM T40103 C8IB2W 44426056 IC50 > 100000 nM T40103 C8Z4WO 44459967 IC50 = 14454.4 nM T40103 C86ORE 44459987 IC50 = 16218.1 nM T40103 CLH74F 44565900 IC50 = 91760 nM T40103 CMIP10 44565901 IC50 > 100000 nM T40103 C70BXJ 44565925 IC50 = 66520 nM T40103 CS6YO0 44566187 IC50 = 145 nM T40103 CSF17Z 44566188 IC50 > 100000 nM T40103 CJP3U5 44566195 IC50 > 100000 nM T40103 CUFJ57 44566196 IC50 = 32570 nM T40103 CI7P2B 49797571 IC50 > 50000 nM T40103 CI59MV 49797572 IC50 > 50000 nM T40103 C96CKU 49797573 IC50 > 50000 nM T40103 CZM3L7 71520324 Ki = 129000 nM T40103 C63ROI 71717313 Ki = 221000 nM T40103 CGFK60 101201806 IC50 = 29000 nM T40103 C8E4WS 102323332 IC50 = 9800 nM T40103 C8X6JG 145970039 Ki = 329000 nM T40103 C51ZEH 145970706 Ki = 462000 nM T40103 CM53FT 145986712 Ki = 7000 nM T40103 CN6U8D 145988823 Ki = 108000 nM T40103 C5MWT1 145990477 Ki = 1300 nM T40103 CHD79T 44408017 IC50 > 13000 nM T40103 CO0N3S 44408050 IC50 > 13000 nM T40103 D05WZF 10129151 IC50 > 5000 nM T40103 D08KCA 72429 Ki = 9200 nM T40103 D09FGQ 123985 IC50 = 190 nM T40103 D0G2QG 44343301 IC50 = 40 nM T40103 D0L9VP 5287864 Ki = 1400 nM T40103 D0T7QF 10420833 IC50 > 13000 nM T40103 D0VE0F 10062714 IC50 > 13000 nM T40103 D0Y5IQ 44255320 IC50 = 10000 nM T34296 D00MDP 466151 Ki = 0.038 nM T34296 D04AIT 5280445 IC50 = 10050 nM T34296 D0K8KX 5280343 IC50 = 8460 nM T34296 D0S0LZ 54671203 IC50 = 40000 nM T34296 D05VZE 119031 IC50 = 2 nM T34296 D0A4RF 657061 IC50 = 0.6 nM T34296 D0HG5M 11452716 IC50 = 8 nM T34296 D0MW3H 9824350 Ki = 0.53 nM T34296 D0G1LL 74221072 IC50 = 47000 nM T34296 D0N6ZA 74221131 IC50 > 100000 nM T34296 D0UM5R 74221070 IC50 = 4800 nM T34296 D00UCC 9827497 IC50 = 3.3 nM T34296 D01DVX 9847838 IC50 = 461 nM T34296 D03BOZ 3342298 IC50 = 0.01 nM T34296 D0N8NK 11641563 IC50 = 4.7 nM T34296 D0P8YC 5362422 IC50 = 5 nM T34296 D0Q1CD 6918336 Ki = 1470 nM T34296 D0T9HG 132519 IC50 = 5.2 nM T34296 CNA81R 1836 Ki = 65 nM T34296 CZ45IU 4219 IC50 = 6.4 nM T34296 CFY8Q2 4230 IC50 = 1.3 nM T34296 C7ROG5 177347 IC50 = 1570 nM T34296 CV60YH 445010 IC50 = 3 nM T34296 C4D7TS 448002 IC50 = 3 nM T34296 CZDY56 645394 IC50 = 9900 nM T34296 CU6X2H 647218 IC50 = 15300 nM T34296 CY58CV 651056 IC50 = 4700 nM T34296 C4UMB1 651101 IC50 = 9400 nM T34296 C78NPG 651441 IC50 = 2500 nM T34296 CA70CP 664499 IC50 = 4000 nM T34296 CS4O7K 685005 IC50 = 31000 nM T34296 CP1Q6R 703233 IC50 = 67000 nM T34296 C2OCU9 779459 IC50 > 1000000 nM T34296 CEBX21 1016400 IC50 = 7700 nM T34296 CXNA13 1201165 IC50 = 4700 nM T34296 CH82ZT 1201321 IC50 = 1590 nM T34296 CAM10Y 1204907 IC50 = 640 nM T34296 C9IFC6 1348435 IC50 = 22000 nM T34296 C7K3JR 1358229 IC50 = 5890 nM T34296 C6UZ1A 1383990 IC50 = 6970 nM T34296 CVA63S 1506964 IC50 = 900 nM T34296 C4X0MZ 1870548 IC50 = 12600 nM T34296 CZ9TI3 2053915 IC50 = 39810.72 nM T34296 CN9C8D 2140735 IC50 = 120000 nM T34296 CJ3EF9 2221136 IC50 = 3600 nM T34296 CN6E3U 2366268 IC50 = 1900 nM T34296 CSL5X7 2369069 IC50 = 8100 nM T34296 CJ1LK6 2568387 IC50 = 25118.86 nM T34296 C0I9ZT 2571427 IC50 = 8400 nM T34296 C65UHI 2966106 IC50 = 6800 nM T34296 COH0C4 2994402 IC50 > 100000 nM T34296 C5Z9PF 2999799 IC50 = 13300 nM T34296 CO1HF6 3109990 IC50 = 24700 nM T34296 CP09YC 3109994 IC50 = 10900 nM T34296 CM72OK 3236108 IC50 = 12000 nM T34296 C5QT9A 3240046 IC50 = 3500 nM T34296 C6C3QR 3243814 IC50 = 23300 nM T34296 C0PB5H 3380837 IC50 = 177000 nM T34296 CME24U 3649035 IC50 = 24000 nM T34296 CT8PU3 3671894 IC50 > 67000 nM T34296 C3EI6T 4085085 IC50 = 14000 nM T34296 CBN96T 4358655 IC50 = 10000 nM T34296 CP8D7Y 4478236 IC50 = 75.86 nM T34296 CQ4VL5 5287415 IC50 = 0.7 nM T34296 CW5SE3 5288615 IC50 = 2.4 nM T34296 CJ3QI1 5288814 IC50 = 2330 nM T34296 C1R5CO 5289109 IC50 = 72 nM T34296 CA5D1J 5289110 IC50 = 8 nM T34296 CKM71T 5289111 IC50 = 6600 nM T34296 C7BPU5 5310930 IC50 > 40000 nM T34296 CVLS16 5319161 IC50 = 7620 nM T34296 C1CM3J 6005649 IC50 = 55270 nM T34296 C9S1VI 6006930 IC50 = 3990 nM T34296 C5OMB7 6102708 IC50 = 8 nM T34296 C0M3LR 6323382 IC50 = 3 nM T34296 CJG2B7 6476333 IC50 = 11090 nM T34296 CL5DH0 6479915 IC50 = 29030 nM T34296 CI86PQ 6539651 IC50 = 1.7 nM T34296 CQEF36 6539670 IC50 = 2 nM T34296 CP7BG0 6852146 IC50 = 1.3 nM T34296 CN5L2B 6852147 IC50 = 2.6 nM T34296 CP2XK7 6882342 IC50 = 140000 nM T34296 C0FQW9 7063077 Ki = 175 nM T34296 C9UPD8 9794928 IC50 = 1480 nM T34296 CA0ZH1 9798114 IC50 = 86 nM T34296 C7NP9Z 9798247 IC50 = 3 nM T34296 C78EKW 9798637 IC50 = 8 nM T34296 C80WFI 9800763 IC50 = 4.4 nM T34296 C76RCQ 9801569 IC50 = 155 nM T34296 C68HMJ 9801786 IC50 = 3019.95 nM T34296 CM9GH8 9802180 IC50 = 1 nM T34296 CIXD67 9802768 IC50 < 1 nM T34296 C83FVW 9803207 IC50 = 1 nM T34296 C3QS5H 9803407 IC50 = 47 nM T34296 CUSD58 9803469 IC50 = 89 nM T34296 C4QCG9 9803771 IC50 = 5 nM T34296 C23VTC 9804342 IC50 = 3 nM T34296 C49HNU 9805016 IC50 = 1 nM T34296 CXSU10 9805304 IC50 = 83 nM T34296 CO4D0U 9805473 IC50 = 1 nM T34296 C1HP7E 9805710 IC50 = 67 nM T34296 CT8X1F 9806970 IC50 = 321 nM T34296 CTK6J8 9808181 IC50 = 2300 nM T34296 C67XKV 9808391 IC50 = 3 nM T34296 CS07BM 9808594 IC50 = 3 nM T34296 C9RQM7 9808674 IC50 = 0.35 nM T34296 C5CE8A 9809470 IC50 = 4.5 nM T34296 C32ODL 9818295 IC50 = 182 nM T34296 C0R2KN 9818588 IC50 > 10000 nM T34296 CC9VY4 9819420 IC50 = 33 nM T34296 C1VT4J 9819974 IC50 = 26 nM T34296 CQG86S 9820708 IC50 = 2 nM T34296 CN4AP6 9821427 IC50 = 3.49 nM T34296 C6KJ9W 9822461 IC50 = 5.3 nM T34296 C6IX7G 9822926 IC50 = 0.15 nM T34296 CVN5Z3 9823395 IC50 = 30 nM T34296 CUZ25T 9825237 IC50 = 9 nM T34296 C3AEF4 9825692 IC50 = 5 nM T34296 CDJB86 9825720 IC50 = 0.016 nM T34296 CXL65P 9825920 Ki > 5000 nM T34296 CL0G8K 9825927 IC50 = 100 nM T34296 CVSJ72 9826275 IC50 = 1 nM T34296 C7W3TG 9826481 IC50 = 289 nM T34296 CPW60S 9827023 IC50 = 34.6 nM T34296 CXTY18 9827218 IC50 = 290 nM T34296 C24CZI 9827635 IC50 = 7 nM T34296 C2TU0C 9827807 IC50 = 2 nM T34296 CC1NG5 9829581 IC50 = 20 nM T34296 C8WH1Q 9840355 IC50 = 14 nM T34296 CU7FM2 9840390 IC50 = 44 nM T34296 CEAZ87 9840395 IC50 = 84 nM T34296 C9PW7L 9841168 Ki = 206 nM T34296 C5XL7R 9841323 IC50 = 0.2 nM T34296 CRP01H 9841401 Ki = 130 nM T34296 CA7DJ9 9842114 IC50 = 2.4 nM T34296 CQ5L0D 9842167 IC50 = 500 nM T34296 CH63ZI 9842332 IC50 = 12 nM T34296 CC1TB5 9842343 IC50 = 148 nM T34296 C6YT5W 9843479 IC50 = 41.5 nM T34296 C9N5PA 9843679 IC50 = 0.77 nM T34296 C49UOA 9844245 IC50 = 6.5 nM T34296 CK76RW 9845271 IC50 = 29 nM T34296 CD31XZ 9845513 IC50 = 365 nM T34296 CEB90C 9846418 IC50 = 1 nM T34296 C4D2MY 9846507 IC50 = 2 nM T34296 C0KP9H 9847092 IC50 = 2 nM T34296 CE9AL3 9847113 IC50 < 0.1 nM T34296 C6SV1X 9847843 IC50 = 1 nM T34296 CG14CO 9848625 IC50 = 358 nM T34296 C92EJW 9849379 IC50 = 5 nM T34296 CX3EW2 9849576 IC50 = 155 nM T34296 CHVL24 9849957 IC50 = 3 nM T34296 C4IEK0 9850035 IC50 = 0.2 nM T34296 C9P1BH 9851086 IC50 = 1 nM T34296 C5DGI9 9851911 IC50 = 4.5 nM T34296 CC70WV 9858468 IC50 = 107 nM T34296 CECR39 9860227 IC50 = 3450 nM T34296 CR37HQ 9861014 IC50 = 751 nM T34296 C5TUJ7 9862317 IC50 = 7 nM T34296 CS5JT6 9864502 IC50 = 4 nM T34296 CGUF07 9865358 IC50 = 5.7 nM T34296 CU51IV 9865936 IC50 = 2 nM T34296 CI8Z0R 9866250 IC50 = 0.75 nM T34296 CP4Y7O 9867411 IC50 = 6 nM T34296 C0YN1X 9867935 IC50 = 33 nM T34296 CK3F1T 9868079 IC50 = 28 nM T34296 C2L9SU 9868329 IC50 = 2 nM T34296 CJS23I 9868333 Ki > 5025 nM T34296 C5O0GC 9868490 IC50 = 97 nM T34296 CRI23M 9868515 IC50 = 52 nM T34296 C4K2GH 9868577 IC50 = 2 nM T34296 C4ZR7O 9868713 IC50 = 77 nM T34296 C24JSB 9868858 IC50 = 33 nM T34296 C5IJH2 9869068 IC50 = 15 nM T34296 CT76IN 9869441 IC50 = 2 nM T34296 CA6G0W 9869598 IC50 = 2 nM T34296 CZO6K4 9869819 IC50 = 0.4 nM T34296 C5ELS6 9869902 IC50 = 2 nM T34296 CMEA71 9869947 IC50 = 1.1 nM T34296 CA48SX 9870269 IC50 = 1.9 nM T34296 C25-SEP 9870933 IC50 = 701 nM T34296 C5QFG1 9871290 IC50 = 2 nM T34296 CSM16R 9871355 IC50 = 302 nM T34296 CHU9I8 9871883 IC50 = 0.1 nM T34296 CU9L3X 9879183 IC50 > 10000 nM T34296 CG41SV 9879575 IC50 > 10000 nM T34296 C0TCJ2 9880675 Ki = 904 nM T34296 C0NA6S 9880842 IC50 = 100 nM T34296 C0QY4U 9883809 IC50 = 946 nM T34296 C9XSN0 9883962 IC50 = 4760 nM T34296 C2OHV3 9885051 IC50 = 34 nM T34296 CKFD90 9885716 IC50 = 38 nM T34296 CG35XZ 9885916 IC50 = 1000 nM T34296 CZBK85 9886177 IC50 = 78 nM T34296 CHT08B 9886916 IC50 = 0.65 nM T34296 C2M4EC 9887473 Ki > 5025 nM T34296 C1STP9 9887771 IC50 = 1.2 nM T34296 CFG4Q2 9887831 IC50 = 9 nM T34296 C3ZG6O 9887870 IC50 = 8 nM T34296 CC87LP 9888280 IC50 = 2 nM T34296 CD76WB 9888485 IC50 = 2 nM T34296 CVP45O 9888530 IC50 = 231 nM T34296 CJS0E5 9888649 IC50 = 8 nM T34296 CB2YG7 9889128 IC50 = 2 nM T34296 CD1U5P 9889190 IC50 = 20.89 nM T34296 C4AVN6 9889449 IC50 = 200 nM T34296 CZD2E3 9889870 IC50 = 4 nM T34296 C26SZX 9890226 IC50 = 0.6 nM T34296 CWN19T 9890526 IC50 = 12.2 nM T34296 CD79UJ 9890632 IC50 > 100000 nM T34296 CNX78A 9890733 IC50 = 1 nM T34296 CMD0S2 9891009 IC50 = 47 nM T34296 C20LGF 9891255 IC50 = 31 nM T34296 C9YD2O 9891259 IC50 = 16 nM T34296 CU65HY 9891358 IC50 = 1.2 nM T34296 C3QSE6 9891814 IC50 = 5 nM T34296 CPT4C6 9892042 IC50 = 427 nM T34296 CR50BS 9892336 IC50 = 27 nM T34296 C1KV7J 9892518 IC50 = 26 nM T34296 CH69LT 9892815 IC50 < 0.1 nM T34296 CZU7Y4 9892876 IC50 = 129 nM T34296 CX82KN 9893236 IC50 = 1.4 nM T34296 C2G5AQ 9894201 IC50 = 908 nM T34296 CSIB97 9896504 IC50 = 23 nM T34296 C6Q4JF 9903007 IC50 = 22 nM T34296 C2R5CX 9905493 IC50 = 1.8 nM T34296 CD78ZQ 9907286 IC50 = 0.9 nM T34296 CYHN04 9908006 IC50 = 7 nM T34296 CKWF30 9908681 IC50 = 22 nM T34296 CQ8Y9T 9909624 IC50 = 0.37 nM T34296 CJ3K1I 9910075 IC50 = 2137.96 nM T34296 C4E6LR 9910544 IC50 = 150 nM T34296 C6NUE9 9910550 IC50 = 3 nM T34296 CP4LS8 9910727 IC50 = 498 nM T34296 C2GMQ0 9912235 IC50 = 119 nM T34296 C62VZI 9912382 IC50 = 12 nM T34296 C8VJ9Z 9913053 IC50 = 1 nM T34296 CI5A3G 9913301 IC50 = 3 nM T34296 C3AZP0 9913479 IC50 = 1.4 nM T34296 CX1Q5C 9913489 IC50 = 1 nM T34296 C7ZY1L 9914029 IC50 = 248 nM T34296 CU9B3E 9914147 IC50 = 20 nM T34296 CX3C2G 9914326 IC50 = 72 nM T34296 CM39FU 9915194 IC50 = 2377 nM T34296 CA3FW0 9918908 IC50 = 0.008 nM T34296 CM7UO8 9924798 IC50 = 24 nM T34296 CBPD13 9926779 IC50 = 37 nM T34296 CSA12Z 9927353 IC50 = 57 nM T34296 C26ZPC 9929976 IC50 = 2 nM T34296 C1KX3E 9930058 IC50 = 2 nM T34296 CLJ61Q 9931505 IC50 = 2 nM T34296 C67PBX 9932128 IC50 = 11 nM T34296 CJI5A7 9932167 IC50 = 2 nM T34296 CY79AT 9932263 IC50 = 1.2 nM T34296 C03GVA 9932290 Ki = 210 nM T34296 C3VO2E 9932958 IC50 = 12 nM T34296 CT2KM9 9933083 IC50 = 100 nM T34296 CDXR37 9933197 IC50 = 0.4 nM T34296 C2EUL8 9933259 IC50 = 34 nM T34296 CX17KQ 9933408 IC50 = 104.71 nM T34296 C57WSD 9934240 IC50 = 42 nM T34296 CGJZ78 9934997 IC50 = 29 nM T34296 C65ION 9935032 IC50 = 0.2 nM T34296 C1HRU9 9936228 IC50 = 3.8 nM T34296 CDRC76 9936405 IC50 = 317 nM T34296 CH9G5D 9936469 IC50 = 9.5 nM T34296 C7GJF8 9936712 IC50 = 5 nM T34296 CG38KL 9936728 Ki = 2.3 nM T34296 CE59TP 9936926 IC50 = 758.58 nM T34296 C12ZGS 9945200 IC50 = 396 nM T34296 C0MLZ6 9945553 IC50 = 2000 nM T34296 CA30JY 9946988 IC50 = 520 nM T34296 C6TH4I 9947270 IC50 = 708 nM T34296 C16HTN 9948666 Ki = 17 nM T34296 C52IUJ 9949603 IC50 = 2000 nM T34296 CWO48K 9952436 IC50 = 1.5 nM T34296 C8C3DL 9953278 IC50 = 580 nM T34296 C9OY4Z 9953817 IC50 = 9 nM T34296 CABI45 9954117 IC50 = 11 nM T34296 C8RXN6 9954304 IC50 = 869 nM T34296 C6GA8D 9954513 IC50 = 11 nM T34296 CH9YL3 9954604 IC50 = 3 nM T34296 C37VXK 9954605 IC50 = 2 nM T34296 CK9HX0 9955125 IC50 = 0.4 nM T34296 CMV37W 9955127 IC50 = 49 nM T34296 CWE6N8 9955640 IC50 = 3 nM T34296 C3ZLA1 9956465 IC50 = 40 nM T34296 C3Q2UJ 9956686 IC50 = 0.25 nM T34296 C56GFP 9956833 IC50 = 3 nM T34296 CQ80MP 9957107 IC50 = 7 nM T34296 C5I0VJ 9957500 IC50 = 233 nM T34296 CN76XI 9957653 IC50 = 1 nM T34296 CPJR82 9957875 IC50 = 3 nM T34296 CYJ35F 9958085 IC50 = 0.12 nM T34296 CWE4D3 9958604 IC50 = 6 nM T34296 CNHT34 9959421 IC50 = 0.4 nM T34296 CN8TK0 9959428 IC50 = 1691 nM T34296 C9DRB7 9966028 IC50 = 185 nM T34296 CYK75X 9967932 IC50 > 10000 nM T34296 C0HL2X 9976697 IC50 = 0.9 nM T34296 C09LSY 9979489 Ki > 5025 nM T34296 CUA65C 9982414 IC50 = 0.95 nM T34296 CO09PN 9983251 IC50 = 0.9 nM T34296 CJGR30 9983604 IC50 = 0.7 nM T34296 C3KX1B 9998685 Ki = 3 nM T34296 C8W5UK 9999879 IC50 = 527 nM T34296 C59WEK 10001843 IC50 < 0.1 nM T34296 CR7T3J 10009978 Ki = 50 nM T34296 CJ6H8O 10019658 IC50 = 1 nM T34296 C71YGT 10025307 Ki = 4.169 nM T34296 C5PKZ1 10029419 IC50 = 0.09 nM T34296 CM52RO 10030422 IC50 = 14 nM T34296 CJR59P 10031295 Ki > 5025 nM T34296 C7J9ZF 10039403 IC50 = 64 nM T34296 CNA3G4 10042214 IC50 = 12 nM T34296 C07DLO 10046817 IC50 = 290 nM T34296 CHF92V 10047100 Ki = 2.692 nM T34296 CLXN48 10047373 IC50 = 1 nM T34296 C1N9UX 10050222 IC50 = 154 nM T34296 CLZ87W 10051236 Ki = 753 nM T34296 C21ULC 10052150 IC50 = 0.16 nM T34296 CSHD67 10054852 IC50 = 0.4 nM T34296 CJK0R1 10074190 IC50 = 1 nM T34296 CPS4R9 10076090 IC50 = 0.8 nM T34296 CPKC43 10093147 IC50 = 4 nM T34296 C5W4ZA 10094362 IC50 = 40 nM T34296 C2XV5J 10098250 IC50 = 1 nM T34296 C3V2HW 10099112 IC50 = 12 nM T34296 CXV2Y3 10109170 Ki = 1055 nM T34296 C0G7IY 10114318 Ki = 470 nM T34296 C9T2AW 10116042 IC50 = 10 nM T34296 CVK61T 10116047 IC50 = 11 nM T34296 C78JHL 10116107 Ki = 570 nM T34296 CP5L0W 10117663 Ki = 3869 nM T34296 C7OPQ8 10118047 IC50 = 0.4 nM T34296 CU3ZM2 10118633 IC50 > 1000 nM T34296 C2F8KW 10119294 IC50 = 1 nM T34296 CPA4R9 10119730 IC50 = 7 nM T34296 C7A8MI 10120093 IC50 = 0.2 nM T34296 C0Q9DW 10120586 IC50 = 20 nM T34296 C0KHW5 10120930 IC50 = 50 nM T34296 CP65KL 10125869 Ki = 55 nM T34296 CPTG57 10126378 IC50 = 122 nM T34296 CY2N3D 10127629 Ki > 5020 nM T34296 C1N4MJ 10127670 Ki > 5020 nM T34296 CIL09Z 10127889 Ki > 5020 nM T34296 CYU19P 10127901 Ki = 3530 nM T34296 C07KFI 10128313 Ki > 5020 nM T34296 CB3I6K 10128659 Ki > 5020 nM T34296 C6ZK3A 10128916 Ki > 5020 nM T34296 CS54CQ 10133565 IC50 > 10000 nM T34296 C0SVY1 10134897 IC50 = 4019 nM T34296 C9EWX5 10135125 IC50 = 13 nM T34296 C7KR3Y 10136680 Ki = 320 nM T34296 CNU93J 10136924 Ki = 650 nM T34296 C1CDF2 10136925 Ki = 300 nM T34296 CJ9EX4 10138303 Ki = 3810 nM T34296 C6UXD7 10138936 IC50 = 85 nM T34296 CU6Y9T 10140438 Ki > 5025 nM T34296 CE75BY 10140776 Ki = 1206 nM T34296 CIH36M 10141214 IC50 = 0.2 nM T34296 C5DA1U 10141270 IC50 = 4 nM T34296 C5H1ZM 10141426 IC50 = 1 nM T34296 C6MSI0 10141443 IC50 = 7300 nM T34296 CLXF15 10141613 Ki > 5000 nM T34296 C7VF1K 10141614 Ki = 2613 nM T34296 CWB5O4 10142326 Ki > 5000 nM T34296 CPXB21 10143028 Ki > 5025 nM T34296 C23WZR 10143587 Ki > 5000 nM T34296 CAM6U7 10143672 IC50 = 6 nM T34296 C82SMW 10144091 IC50 = 3 nM T34296 CD3U8E 10150649 Ki = 7 nM T34296 CJMV83 10152887 IC50 = 3.3 nM T34296 CZW98O 10156375 Ki = 55 nM T34296 CPY87U 10158366 IC50 > 10000 nM T34296 CYO8D2 10159633 Ki > 5025 nM T34296 CHUA34 10160545 IC50 = 2.4 nM T34296 CQ41YI 10161391 Ki > 5025 nM T34296 CCU9S1 10162155 IC50 = 1 nM T34296 C7SXD4 10162245 Ki = 3266 nM T34296 CO6PS3 10162900 Ki = 130 nM T34296 CR5H6E 10163627 Ki > 5025 nM T34296 CZO5V4 10164317 IC50 = 0.4 nM T34296 CCM0Y8 10165180 Ki = 603 nM T34296 CE10MK 10165419 IC50 = 7 nM T34296 CP02FJ 10165420 IC50 = 7 nM T34296 C0K7HT 10165868 IC50 = 1 nM T34296 C9X8YZ 10172500 IC50 = 130 nM T34296 CB3Q9L 10172753 IC50 = 61.2 nM T34296 CA81UR 10173271 IC50 = 10000 nM T34296 C6IW4O 10173876 Ki > 5020 nM T34296 CV7ES2 10174780 IC50 = 1.7 nM T34296 C8NAM9 10174791 IC50 = 1 nM T34296 CN6I1L 10174798 IC50 = 0.54 nM T34296 CZL72O 10175020 IC50 = 0.45 nM T34296 C4QY3V 10175210 Ki = 5020 nM T34296 C84ZQD 10175219 Ki = 1310 nM T34296 C5JM1A 10179045 IC50 > 10000 nM T34296 CD4AO0 10180362 IC50 = 2200 nM T34296 CCX3T6 10183064 Ki > 15000 nM T34296 CS6X2R 10183408 IC50 = 2 nM T34296 C6OE9H 10183692 IC50 > 10000 nM T34296 CDM94B 10183693 Ki > 5000 nM T34296 C2GV5Q 10183755 IC50 = 65 nM T34296 CH04IS 10184457 IC50 = 2 nM T34296 C3E9NF 10184537 Ki > 5000 nM T34296 CTDP62 10184579 Ki > 5000 nM T34296 CXQ8N0 10185100 Ki = 3136 nM T34296 C2OM9G 10186288 IC50 = 16 nM T34296 CK0P3F 10186536 Ki > 5025 nM T34296 CV7YI1 10186544 Ki > 5000 nM T34296 CA9FG4 10187181 IC50 = 4 nM T34296 CY9W6L 10194183 IC50 = 13.5 nM T34296 C51RPY 10195069 Ki > 5020 nM T34296 CY36NO 10196425 Ki > 5020 nM T34296 C63JGO 10196445 IC50 = 0.68 nM T34296 C0U9KC 10199401 IC50 = 32 nM T34296 C5CUM9 10202769 Ki > 5025 nM T34296 CX8BS3 10203685 Ki > 5025 nM T34296 C4FSU0 10203714 IC50 = 0.88 nM T34296 CE1LI3 10204303 Ki = 120 nM T34296 C32RAQ 10204620 Ki > 5000 nM T34296 C7AU0H 10205886 IC50 = 26 nM T34296 CQFP69 10206106 Ki = 370 nM T34296 CS1CA5 10207780 Ki = 653 nM T34296 C4K1MJ 10208262 Ki > 5025 nM T34296 CV4DG9 10209314 IC50 = 2 nM T34296 CD76KE 10209382 Ki > 5025 nM T34296 CT62UX 10215925 IC50 = 57 nM T34296 CVQA31 10216178 IC50 = 18 nM T34296 CXRT17 10218227 IC50 = 0.73 nM T34296 C7Y2US 10218353 Ki = 3720 nM T34296 C1C7AH 10223757 Ki > 5025 nM T34296 C92BVJ 10223963 IC50 = 21 nM T34296 CV5X8A 10224181 IC50 = 0.67 nM T34296 CGKU70 10224396 Ki = 250 nM T34296 C7K1OR 10224602 IC50 = 2000 nM T34296 CLH71C 10225319 Ki > 5025 nM T34296 C2X1KF 10226116 Ki = 753 nM T34296 C9CSG3 10226996 IC50 = 8.2 nM T34296 CJ46HR 10227522 IC50 = 2 nM T34296 CUE63Q 10227853 Ki > 5000 nM T34296 C19DFP 10227854 Ki > 5000 nM T34296 CSDG58 10228529 IC50 = 255 nM T34296 C7T0WH 10229644 IC50 = 1.8 nM T34296 CD2HP3 10230012 Ki > 5000 nM T34296 CLJ3Y9 10230286 IC50 = 1 nM T34296 CCRM18 10231253 IC50 = 1.1 nM T34296 CCTY95 10237492 Ki = 5020 nM T34296 CRF32B 10237550 Ki = 10 nM T34296 CNO8Z1 10237571 IC50 = 1.54 nM T34296 CF5PO0 10237938 IC50 = 3000 nM T34296 CWR7E2 10237960 IC50 = 6.5 nM T34296 CBG59O 10238145 IC50 = 13.9 nM T34296 C91DMB 10239619 IC50 = 0.36 nM T34296 CG70QJ 10239685 IC50 = 0.93 nM T34296 CCQ9V5 10239716 Ki > 5020 nM T34296 C8LQP4 10253358 IC50 = 0.65 nM T34296 C2V4MP 10253549 IC50 = 1.9 nM T34296 CQF3V9 10253673 IC50 = 34.67 nM T34296 CJKD83 10268288 IC50 > 10000 nM T34296 CMNA19 10270268 IC50 > 10000 nM T34296 C2MES9 10271604 Ki = 91000 nM T34296 CBJE75 10272162 IC50 = 11.7 nM T34296 CGP97S 10274748 Ki = 180 nM T34296 CU67RC 10275101 IC50 = 2.7 nM T34296 CES6A5 10276821 Ki = 804 nM T34296 C0GU6B 10277568 IC50 = 2 nM T34296 CY6K1G 10277706 Ki = 3266 nM T34296 C9OAE1 10277812 IC50 = 3 nM T34296 C2UAM8 10278729 IC50 = 1 nM T34296 C5Z2IG 10278742 IC50 = 0.8 nM T34296 C6KR5M 10278934 IC50 = 9 nM T34296 C3IG0K 10280852 IC50 < 0.1 nM T34296 C7TWG0 10289551 Ki > 5020 nM T34296 CJ63ER 10289607 Ki > 5020 nM T34296 CR48SA 10289842 Ki > 5210 nM T34296 CP0I5Y 10291146 IC50 > 10000 nM T34296 CLP72J 10293348 IC50 > 10000 nM T34296 CS69YG 10293394 IC50 = 9000 nM T34296 CB82ZF 10294766 IC50 = 90 nM T34296 CDU36Y 10296475 Ki = 1330 nM T34296 C48IRP 10296785 Ki = 140 nM T34296 CQ1Z0G 10298111 IC50 = 900 nM T34296 CN14MI 10298369 Ki > 5025 nM T34296 C25EKM 10299665 Ki = 753 nM T34296 C1BR6A 10300063 Ki > 5025 nM T34296 C80VEU 10300077 Ki > 5025 nM T34296 CFAU84 10301584 Ki > 5025 nM T34296 CP5AU1 10302088 Ki > 5025 nM T34296 C35LHB 10309800 IC50 = 244 nM T34296 CE1C7H 10310082 IC50 = 0.15 nM T34296 CE1KM9 10311498 Ki = 3950 nM T34296 C4MC8P 10311673 IC50 = 2 nM T34296 CP3D5K 10311698 IC50 = 0.57 nM T34296 COBH25 10311898 IC50 = 0.88 nM T34296 C4R9ZK 10311997 Ki = 95 nM T34296 CE6MB0 10312141 Ki = 356 nM T34296 CDO9J3 10318516 Ki = 110 nM T34296 CIDW49 10319098 Ki > 5025 nM T34296 CG23FV 10320328 IC50 = 0.6 nM T34296 CJ6XM1 10321516 IC50 = 1 nM T34296 CJWH74 10321975 Ki > 5025 nM T34296 CY08WJ 10322755 Ki > 5000 nM T34296 C3QDH0 10340642 Ki = 1.9 nM T34296 CL8YC0 10346590 IC50 = 0.05 nM T34296 C94ANQ 10347529 IC50 = 0.8 nM T34296 C4K9MO 10355923 Ki = 2200 nM T34296 CWIM61 10364088 IC50 = 10 nM T34296 CL4B2U 10364155 IC50 = 16900 nM T34296 CI0T8K 10366352 Ki > 5025 nM T34296 CBTO07 10370226 Ki > 5025 nM T34296 CP9WG5 10389610 IC50 = 1.8 nM T34296 CY2G0R 10391428 Ki > 5025 nM T34296 C8O1XU 10392082 IC50 = 0.1 nM T34296 C8Y7EZ 10393391 IC50 = 28 nM T34296 CFKA79 10395015 Ki = 653 nM T34296 C1SJ4K 10435554 IC50 = 20 nM T34296 C7XE1L 10437629 IC50 = 4000 nM T34296 C5WV1N 10439082 Ki = 442 nM T34296 C54UDR 10453826 IC50 = 400 nM T34296 C8M9FE 10462640 Ki = 15700 nM T34296 CX38EB 10467565 IC50 = 460 nM T34296 CNQZ36 10483139 Ki = 0.66 nM T34296 C9XC8Y 10493383 IC50 = 79 nM T34296 C6KD0A 10498747 IC50 = 1 nM T34296 CZ2UY0 10502046 IC50 = 2.3 nM T34296 C36OMW 10502172 IC50 = 1 nM T34296 C5V8HJ 10502382 IC50 = 0.8 nM T34296 CJZ5T8 10502487 IC50 > 10000 nM T34296 CSN17G 10502708 IC50 = 0.9 nM T34296 CBNM82 10503128 IC50 < 0.4 nM T34296 C9LJR5 10503737 IC50 = 137 nM T34296 C5Y4IA 10504081 IC50 = 478 nM T34296 C2C7TE 10504472 IC50 < 0.5 nM T34296 CH6S8Y 10505729 IC50 > 10000 nM T34296 C6D7JF 10506147 IC50 = 36 nM T34296 C7S0DB 10506158 IC50 = 24 nM T34296 CBT12Q 10522080 IC50 = 0.7 nM T34296 CC2F5Y 10522311 IC50 = 1 nM T34296 CZ36JW 10523383 IC50 = 580 nM T34296 CQEH42 10524134 IC50 < 0.5 nM T34296 CYU87N 10524260 IC50 < 0.4 nM T34296 COT07L 10525329 IC50 = 8 nM T34296 C61GSD 10525562 IC50 = 2.5 nM T34296 C14XUW 10526101 IC50 = 3 nM T34296 CJK6G1 10526509 IC50 < 0.1 nM T34296 CWLD37 10526788 IC50 = 1 nM T34296 CHS9Q5 10527785 IC50 = 0.8 nM T34296 CJ0D7G 10528505 IC50 = 1.3 nM T34296 CYGU41 10529315 IC50 = 2137.96 nM T34296 CO2R0P 10544323 IC50 = 21 nM T34296 C4PK0U 10549114 IC50 = 1 nM T34296 C4TA1K 10549256 IC50 < 0.4 nM T34296 CHCI01 10549577 IC50 = 0.4 nM T34296 C2HJ1U 10549764 IC50 = 1 nM T34296 CRHP20 10550304 IC50 = 1.5 nM T34296 C7WQ5Z 10550399 IC50 = 2 nM T34296 CNQ75F 10551139 IC50 = 21 nM T34296 CCH0K3 10551483 IC50 = 2.1 nM T34296 CC2FM6 10551489 IC50 > 1600 nM T34296 C5UD0A 10551910 IC50 = 21 nM T34296 CI8XG0 10554869 IC50 = 7 nM T34296 CT7O9M 10569678 IC50 = 11 nM T34296 C8RWE4 10569743 IC50 = 105 nM T34296 CE14GM 10570702 IC50 = 6 nM T34296 CS9Y3Q 10573446 IC50 = 0.5 nM T34296 C61IUN 10574937 IC50 = 3.3 nM T34296 C1KH7E 10578728 IC50 = 154 nM T34296 CIUO27 10593253 IC50 = 1 nM T34296 CUTS47 10594564 IC50 = 37 nM T34296 CN4Y6H 10594565 IC50 = 53 nM T34296 CYNC76 10596158 IC50 = 10 nM T34296 C0R8ND 10599533 IC50 < 0.4 nM T34296 CQCW86 10599579 IC50 < 0.4 nM T34296 CW18QK 10599594 IC50 = 0.4 nM T34296 CR1JI4 10600645 IC50 = 0.9 nM T34296 C6RH4O 10601640 IC50 = 4.5 nM T34296 CG32FM 10613145 IC50 = 18 nM T34296 CZD9B3 10617580 IC50 = 1.9 nM T34296 CL02BO 10618584 IC50 = 16 nM T34296 C0JGS3 10621776 IC50 = 3 nM T34296 CL5QN9 10622296 IC50 = 1.9 nM T34296 CL62YC 10622822 IC50 = 9.2 nM T34296 CZJB31 10622970 IC50 = 2.9 nM T34296 CL67UQ 10623250 IC50 = 478.63 nM T34296 CGB29T 10625771 IC50 = 0.5 nM T34296 C98KGO 10625860 IC50 = 3.2 nM T34296 C8UY9P 10639050 IC50 > 30000 nM T34296 C7KGM3 10642071 IC50 = 0.7 nM T34296 CWRY91 10642128 IC50 = 3.6 nM T34296 CI2QB9 10642965 IC50 < 1 nM T34296 C2O1XM 10647817 IC50 = 2.8 nM T34296 C5RWF4 10648802 IC50 = 2 nM T34296 C6S1KA 10649216 IC50 > 10000 nM T34296 C27QHB 10663143 IC50 = 1.7 nM T34296 C97KZU 10665624 IC50 = 43 nM T34296 CF0E6H 10668745 IC50 = 23 nM T34296 CAI72H 10670246 IC50 = 0.7 nM T34296 CY6QC1 10670819 IC50 = 4.1 nM T34296 CPG5O2 10671155 IC50 = 2.4 nM T34296 C17LYV 10672346 IC50 = 48.98 nM T34296 CMU74I 10672857 IC50 = 269.15 nM T34296 CXTP56 10688727 IC50 < 0.5 nM T34296 C0OJ9C 10689683 IC50 = 5 nM T34296 CSA80H 10692194 IC50 = 1 nM T34296 CS5CL7 10692307 IC50 = 0.5 nM T34296 CR5KF8 10692994 IC50 = 710 nM T34296 CDI12G 10693559 IC50 = 1.3 nM T34296 CB70DA 10693592 IC50 = 0.9 nM T34296 CVML68 10693881 IC50 = 1 nM T34296 CZGC63 10695865 IC50 = 102.33 nM T34296 CW6CF7 10696226 IC50 = 1 nM T34296 C6MWX8 10696713 IC50 = 26.92 nM T34296 C1YFC3 10696977 IC50 = 223.87 nM T34296 C4BME8 10697140 IC50 = 254 nM T34296 CG38ZD 10714323 IC50 = 27 nM T34296 C4IWF2 10714988 IC50 = 1 nM T34296 CO9KV7 10715115 IC50 = 0.3 nM T34296 CE1D6G 10716217 IC50 = 0.2 nM T34296 C0ZX6T 10717308 IC50 = 5 nM T34296 C7OSW8 10718200 IC50 < 0.4 nM T34296 C35MRE 10719092 IC50 = 0.4 nM T34296 CVW81M 10719595 IC50 = 114.82 nM T34296 C4J1WN 10721454 IC50 = 2 nM T34296 CI4SQ2 10732349 IC50 = 500 nM T34296 C51DZG 10737732 IC50 = 48 nM T34296 C1LS5U 10738104 IC50 = 1 nM T34296 CL74TG 10738165 IC50 < 0.4 nM T34296 C76ANK 10739335 IC50 = 1 nM T34296 C0T2VK 10740460 IC50 = 1.698 nM T34296 CKJD45 10741133 IC50 = 650 nM T34296 CL64BU 10741592 IC50 < 0.4 nM T34296 C4MQ8L 10742072 IC50 < 0.4 nM T34296 CKX5R3 10742142 IC50 = 21.88 nM T34296 CHW23E 10742387 IC50 = 2.7 nM T34296 CCH94Q 10743507 IC50 = 1.3 nM T34296 C9ILP3 10745718 IC50 = 13 nM T34296 CE09PI 10757715 IC50 = 5 nM T34296 C0BAE9 10763583 IC50 = 2037 nM T34296 C68THN 10763851 IC50 < 0.2 nM T34296 CAG53Y 10764489 IC50 = 5.6 nM T34296 C0ZJB9 10764600 IC50 = 57 nM T34296 CJE76M 10764871 IC50 = 0.7 nM T34296 CQ0KM4 10765140 IC50 < 0.4 nM T34296 C3P2TS 10766036 IC50 = 144.54 nM T34296 CN6P1J 10766950 IC50 = 17 nM T34296 CWR5Z3 10767105 IC50 = 58.88 nM T34296 CR4I1E 10767157 IC50 = 125.89 nM T34296 C7Q2EM 10767236 IC50 = 2 nM T34296 CQ7J4I 10769007 IC50 = 344 nM T34296 C2FA7J 10787997 IC50 = 1 nM T34296 C16XQR 10788211 IC50 = 0.4 nM T34296 C0DFB9 10788617 IC50 < 0.2 nM T34296 CNAE08 10788733 IC50 = 7 nM T34296 CXQD12 10789326 IC50 = 1659.59 nM T34296 CKV2O8 10789493 IC50 = 0.7 nM T34296 C45UGJ 10789671 IC50 < 0.4 nM T34296 C9NZ4W 10789711 IC50 = 1 nM T34296 CHWG02 10790787 IC50 = 88 nM T34296 CWCD73 10805054 IC50 = 4 nM T34296 C1WZ4S 10805349 IC50 = 1 nM T34296 CN8I3Z 10808172 IC50 = 11 nM T34296 CT1AI4 10810573 IC50 = 2 nM T34296 CV3ZA5 10812444 IC50 = 54 nM T34296 CZB7L2 10812929 IC50 < 1 nM T34296 C4TF0K 10813874 IC50 = 0.1 nM T34296 CCIL63 10813879 IC50 < 0.4 nM T34296 CIUN51 10814028 IC50 = 144.54 nM T34296 CS7BY4 10816934 IC50 = 4 nM T34296 CX2E1C 10829071 IC50 = 0.5 nM T34296 C3AI5Z 10831752 IC50 = 150 nM T34296 CLK9P7 10832592 IC50 = 18.4 nM T34296 CF50HD 10832925 IC50 = 26 nM T34296 C5OG4U 10833497 IC50 = 102 nM T34296 CH90ZB 10834348 IC50 = 4.3 nM T34296 C48PYQ 10836923 IC50 = 1.4 nM T34296 CH8OV4 10837276 IC50 = 2.5 nM T34296 CF40VH 10837557 IC50 = 0.8 nM T34296 CY4J9A 10838149 IC50 = 0.9 nM T34296 CA76MU 10840059 IC50 = 2754.23 nM T34296 CN5MJ6 10853865 IC50 = 3390 nM T34296 C3UCL2 10854279 IC50 = 9 nM T34296 CBQ70P 10874312 IC50 = 16.2 nM T34296 CXY47P 10875332 IC50 = 2.8 nM T34296 C3AY8O 10885569 IC50 = 31 nM T34296 CAU0I3 10885834 IC50 = 2.399 nM T34296 CG1I4Y 10886343 IC50 = 2 nM T34296 CF5L1R 10886549 IC50 = 4 nM T34296 CPJ0I8 10896934 IC50 = 808 nM T34296 CU7YE0 10896986 IC50 = 0.5 nM T34296 CX93MR 10907320 IC50 = 27 nM T34296 CAH70N 10914350 IC50 = 37 nM T34296 CF9NT3 10914471 IC50 = 141 nM T34296 CGI2T1 10928606 IC50 = 275 nM T34296 CXHA75 10928874 IC50 = 5.37 nM T34296 C40PRC 10929100 IC50 = 19 nM T34296 CXY4L6 10929354 IC50 = 417 nM T34296 CDSQ41 10929404 IC50 = 391 nM T34296 C4JC9O 10930047 IC50 = 3.02 nM T34296 CLIR35 10938505 IC50 = 2 nM T34296 CWO29J 10940364 IC50 = 80 nM T34296 C9YOU4 10951375 IC50 = 14 nM T34296 CJI1G0 10951750 IC50 = 0.8 nM T34296 C3K1BL 10959017 IC50 = 11 nM T34296 C5ZV9Q 10962137 IC50 = 11 nM T34296 CR9J5B 10983887 IC50 = 5.1 nM T34296 CSI5G1 10992109 IC50 = 6 nM T34296 CCX0L6 10994350 IC50 = 5.1 nM T34296 C9C8SA 11001101 IC50 = 64 nM T34296 C4PNK3 11006191 IC50 = 407 nM T34296 CS4FL3 11012667 IC50 = 12 nM T34296 C5JE9G 11014504 IC50 = 14 nM T34296 C9WPH7 11016072 Ki > 15000 nM T34296 CBE68H 11016073 Ki > 15000 nM T34296 CG2DK0 11016448 IC50 = 1 nM T34296 CF30UR 11016519 IC50 = 5.3 nM T34296 CODQ51 11016616 IC50 = 0.3981 nM T34296 C6IHF5 11026991 IC50 > 100 nM T34296 C23KPN 11050468 IC50 = 4.5 nM T34296 C9RU4I 11059620 IC50 = 29.5 nM T34296 C1N5PT 11070986 IC50 = 13.8 nM T34296 C18EIZ 11071831 IC50 = 1 nM T34296 CM9EP0 11077031 IC50 = 188 nM T34296 C5MUD2 11078779 IC50 = 85 nM T34296 CG0A4C 11081333 IC50 = 32 nM T34296 C05MUK 11081992 IC50 = 3.2 nM T34296 CS29GX 11091928 IC50 = 15 nM T34296 C16WBE 11092175 IC50 = 12 nM T34296 CE8V9B 11092295 IC50 = 11.8 nM T34296 CR8ZA7 11092551 IC50 = 195 nM T34296 CX69YN 11093502 IC50 = 1.6 nM T34296 C6CLV8 11101735 IC50 = 319 nM T34296 CR4V2D 11101785 Ki = 620 nM T34296 C8CK3E 11102531 IC50 = 66 nM T34296 CEAI92 11112993 IC50 = 1 nM T34296 CY1SR9 11113744 IC50 = 140 nM T34296 CB2I5K 11123701 IC50 = 55 nM T34296 C8YVE5 11123989 IC50 = 13 nM T34296 CNBG53 11124956 IC50 = 2.3 nM T34296 C2YBQ7 11134935 IC50 = 6.9 nM T34296 C8DMW5 11135133 IC50 = 1.8 nM T34296 CD3N8B 11135304 IC50 = 23 nM T34296 CPO02F 11142863 IC50 = 1.4 nM T34296 C3V4ZX 11143285 IC50 = 12 nM T34296 C9H1CW 11156691 IC50 = 2.3 nM T34296 CMKT17 11168614 IC50 = 8 nM T34296 C63CLD 11169065 IC50 = 220 nM T34296 CVI3F8 11188429 IC50 = 3687 nM T34296 CPA84O 11192618 IC50 = 32 nM T34296 CO5VN2 11201367 IC50 > 10000 nM T34296 CET3R7 11201814 IC50 = 284 nM T34296 C43ONW 11202395 Ki = 4314 nM T34296 CO87YZ 11215538 IC50 = 19 nM T34296 CIZW31 11226189 IC50 = 4.3 nM T34296 C72UCB 11233687 IC50 = 68 nM T34296 CS15WB 11236105 IC50 = 38 nM T34296 CJZ3P6 11257884 Ki = 0.54 nM T34296 CD1FT8 11258906 IC50 = 7 nM T34296 CJM90S 11259332 IC50 = 6.72 nM T34296 C2OJ8Q 11272747 IC50 = 9.5 nM T34296 CC62RY 11279665 IC50 = 38 nM T34296 CJX60I 11284255 IC50 = 6.5 nM T34296 C6LJM4 11284404 IC50 = 3 nM T34296 CP17ID 11284983 IC50 = 2.3 nM T34296 C1IW7N 11292680 IC50 = 4.1 nM T34296 C8C5AV 11294179 Ki > 10000 nM T34296 CLH50U 11318841 IC50 = 7.1 nM T34296 C1SN8I 11319030 IC50 = 3.2 nM T34296 C91LBZ 11319396 IC50 = 58 nM T34296 C48JVH 11327633 IC50 = 2200 nM T34296 C9FW7I 11330706 IC50 = 15 nM T34296 C0XR3B 11330861 IC50 = 11 nM T34296 C49CDU 11335940 IC50 = 970 nM T34296 CQH57S 11342435 IC50 = 1.8 nM T34296 CZ8B0D 11349945 Ki < 5 nM T34296 CYAK73 11353754 IC50 = 3 nM T34296 CTQK48 11373358 Ki > 5025 nM T34296 C5KU3Z 11376005 IC50 = 6.1 nM T34296 CL8QO7 11382562 IC50 = 900 nM T34296 CNZ0T5 11386918 IC50 = 5 nM T34296 CEM0A7 11387990 IC50 = 25 nM T34296 C9KVB7 11394505 IC50 = 32 nM T34296 C9ABX8 11397130 Ki > 5025 nM T34296 CF78WB 11398934 IC50 = 7.8 nM T34296 C2EUO5 11417011 IC50 > 10000 nM T34296 C30PFC 11421763 IC50 = 6.4 nM T34296 CK95HW 11429232 Ki = 1.2 nM T34296 C01FLQ 11441438 Ki < 5 nM T34296 C5NAJ3 11449819 IC50 = 72 nM T34296 COS67B 11456566 IC50 = 2.1 nM T34296 C96DRO 11466734 IC50 = 3.7 nM T34296 C7QF0G 11467517 IC50 = 13 nM T34296 C1KP2Q 11473879 Ki > 5025 nM T34296 C5QEZ8 11483818 IC50 = 18 nM T34296 CX9IY2 11496709 IC50 = 95.6 nM T34296 C3RJ8Z 11496896 IC50 = 4 nM T34296 C6HU4N 11503290 IC50 = 28 nM T34296 CJ46KN 11508259 Ki = 3.6 nM T34296 CWS35C 11510523 IC50 = 13600 nM T34296 C5VUM2 11517085 Ki = 510 nM T34296 CQ9E6J 11519157 IC50 = 2.6 nM T34296 C5MO0U 11526826 IC50 = 15 nM T34296 C9Y6LH 11533683 IC50 = 4440 nM T34296 C5V8UA 11540282 IC50 = 184 nM T34296 C1NZB9 11548265 IC50 = 1.1 nM T34296 CC4GZ0 11554178 IC50 = 2.69 nM T34296 CE3HA6 11556698 Ki = 4000 nM T34296 CNZV95 11561070 IC50 = 16.4 nM T34296 CCW1B8 11569185 IC50 = 5.4 nM T34296 CW5A4S 11569716 IC50 = 2.2 nM T34296 CL9K7T 11583525 IC50 = 8.5 nM T34296 CTQ87G 11599024 IC50 = 4560 nM T34296 CVGC49 11603611 Ki = 2 nM T34296 C7L1NB 11604052 IC50 = 184 nM T34296 C8IWM1 11605689 IC50 = 1.2 nM T34296 C0VCJ8 11613810 IC50 = 6.3 nM T34296 CC2YD9 11618883 IC50 = 4.24 nM T34296 C9EOY7 11619541 IC50 = 11 nM T34296 CCBS59 11634234 IC50 = 157 nM T34296 CNY92D 11640694 Ki = 7000 nM T34296 C1U3EX 11656290 IC50 = 9.8 nM T34296 C3LZP9 11662242 IC50 = 120 nM T34296 CPIN09 11668791 IC50 = 19.3 nM T34296 CRF7V9 11691964 IC50 = 1.1 nM T34296 C3U6ZR 11697504 Ki = 20000 nM T34296 C1NGT6 11698000 IC50 = 18 nM T34296 C4BGI2 11698938 IC50 = 1336 nM T34296 C2BJ3X 11716217 Ki = 12860 nM T34296 CCD93H 11730086 Ki = 180 nM T34296 C7CED0 11733417 IC50 = 791 nM T34296 CI0KL2 11733573 IC50 = 11 nM T34296 C27SBC 11734162 IC50 = 1 nM T34296 C6HV8Z 11752434 IC50 = 3 nM T34296 CG8U3H 11753351 IC50 = 25 nM T34296 CO8QT0 11753905 Ki = 490 nM T34296 CJ4G5D 11754907 IC50 = 18.1 nM T34296 CE6OS0 11755521 IC50 = 1.288 nM T34296 CL4NF5 11756420 IC50 = 0.11 nM T34296 CUC9R5 11758082 IC50 = 0.7 nM T34296 C2KU3D 11760296 IC50 = 6 nM T34296 CKM6P2 11795228 IC50 = 4.2 nM T34296 CCSD72 11795621 IC50 = 2.1 nM T34296 C46KHU 11796490 IC50 = 1.3 nM T34296 C47OIA 11797154 IC50 = 0.8 nM T34296 CCD4W2 11797992 IC50 = 1.1 nM T34296 CHQR96 11798386 IC50 = 0.2 nM T34296 C2YD4N 11809525 IC50 = 39 nM T34296 C1NRV6 11811437 IC50 = 9 nM T34296 CQ9HE2 11811551 IC50 = 264 nM T34296 CLW3F1 11812791 IC50 = 55.3 nM T34296 CH3SV6 11813493 IC50 = 296 nM T34296 C7BK5P 11825105 IC50 = 0.4 nM T34296 CKEM29 11827006 IC50 = 162 nM T34296 C4XR5G 11963536 IC50 = 2277 nM T34296 C02BWA 11967143 Ki > 2000 nM T34296 CB80OT 12000718 IC50 = 0.03 nM T34296 C43PJZ 12000720 IC50 = 1.3 nM T34296 CUQM03 12074753 IC50 = 1100 nM T34296 CKND02 12074756 IC50 = 1100 nM T34296 C4I1TJ 12074757 IC50 = 3700 nM T34296 CJ8W2C 12074758 IC50 = 800 nM T34296 C0K8ZX 12404978 IC50 > 500000 nM T34296 CB1F2E 12971983 IC50 = 825 nM T34296 CJY6X7 12971984 IC50 = 281 nM T34296 CZYE40 12971985 IC50 = 331 nM T34296 C8TH1O 14177156 IC50 > 500000 nM T34296 CKN3R1 15430588 IC50 = 291 nM T34296 C63MFQ 15435266 IC50 = 7 nM T34296 CZ0NL1 15484680 IC50 = 16 nM T34296 C70TDZ 15503645 IC50 = 136 nM T34296 C16TEM 15516782 IC50 = 18 nM T34296 CV1HA9 15516783 IC50 = 2 nM T34296 CEKN36 15520981 IC50 = 0.35 nM T34296 CXUG10 15546245 IC50 = 50 nM T34296 CU7CM3 15551877 IC50 = 56 nM T34296 C2WHJ4 15859211 IC50 = 555 nM T34296 C5FA3L 15871222 IC50 = 12 nM T34296 C6R1LD 15985818 IC50 = 96 nM T34296 C6HM9P 16069178 IC50 = 0.034 nM T34296 CS46XU 16126723 IC50 = 1.6 nM T34296 CC1K9A 16651091 IC50 > 398107.17 nM T34296 CT40DY 16651117 IC50 = 31622.78 nM T34296 C91EXN 16655061 IC50 = 259 nM T34296 CY7DO3 16718635 IC50 = 0.062 nM T34296 CBIH04 16719299 IC50 = 0.024 nM T34296 CP82IZ 16719300 IC50 = 0.054 nM T34296 CQS0F5 16719301 IC50 = 0.036 nM T34296 C97REC 16719303 IC50 = 0.14 nM T34296 C75XDI 16730519 IC50 > 5000 nM T34296 C2W1VA 16739287 Ki = 1200 nM T34296 C3S2TQ 17754305 IC50 = 2920 nM T34296 C6O3KA 17781194 IC50 = 0.53 nM T34296 CIR7S8 17866387 IC50 = 3 nM T34296 CL1H9W 17866459 IC50 = 20 nM T34296 C9RNH3 17866675 IC50 = 12 nM T34296 CCGR13 17897285 IC50 = 3 nM T34296 C2ZAX1 18002715 Ki > 5000 nM T34296 C12UGK 18002722 Ki = 503 nM T34296 C0IYW8 18002726 Ki > 5000 nM T34296 C8N1DM 18002729 Ki = 754 nM T34296 CCG96A 18002736 Ki = 955 nM T34296 C5MLG1 18002745 Ki > 5000 nM T34296 CXT4H2 18002752 Ki > 5000 nM T34296 C26WHK 18002758 Ki = 1708 nM T34296 CV90XS 18002764 Ki > 5000 nM T34296 C8KPM7 18002765 Ki > 5000 nM T34296 CMJ0K3 18002771 Ki > 5000 nM T34296 C2CO9Z 18002775 Ki > 5000 nM T34296 CK8FS7 18173159 IC50 = 101 nM T34296 CX10BM 18173179 IC50 = 65 nM T34296 CQO70Y 18173222 IC50 = 485 nM T34296 C6AW0H 18365436 IC50 = 17 nM T34296 C1QIU4 18368941 IC50 = 15000 nM T34296 C0VJG4 18368975 IC50 = 15000 nM T34296 CI53DY 18379040 Ki > 5025 nM T34296 CB1U5T 18379077 Ki > 5025 nM T34296 CSX97G 18379115 Ki > 5025 nM T34296 CJHL25 18379123 Ki > 5025 nM T34296 CR0B8G 18379149 Ki > 5025 nM T34296 CS4V5K 18379187 Ki > 5025 nM T34296 CCTY94 18379210 Ki > 5025 nM T34296 CA6K5S 18379235 Ki > 5025 nM T34296 CCSK49 18379254 Ki > 5025 nM T34296 CP4T7S 18379435 Ki > 5025 nM T34296 C9Y5GX 18379443 Ki > 5025 nM T34296 CS2H6J 18396836 IC50 = 250 nM T34296 C1WUJ0 18512732 IC50 < 1000 nM T34296 CA0JF9 18512733 IC50 = 15000 nM T34296 C8EIC6 18512737 IC50 = 5900 nM T34296 C50AEZ 18616892 IC50 = 1.7 nM T34296 CRI35F 19366819 IC50 = 1500 nM T34296 CC4KN8 19366830 IC50 = 1 nM T34296 CS70KY 19366867 IC50 = 0.4 nM T34296 CE73XW 19366873 IC50 = 700 nM T34296 CK8MP3 20620240 Ki = 0.13 nM T34296 CPC4G6 20620273 Ki = 2 nM T34296 C26UJT 20620561 IC50 = 0.9 nM T34296 C2E3CY 20620614 IC50 = 0.2 nM T34296 CVEX54 20620688 IC50 = 0.9 nM T34296 CV1SD8 20620714 IC50 = 0.2 nM T34296 C3GAC4 20620715 IC50 = 3.3 nM T34296 C7QV8K 20620757 IC50 = 1.6 nM T34296 CVO73Y 20620827 IC50 = 8.2 nM T34296 CQ14NY 20620831 IC50 = 8 nM T34296 C5RQ8A 20620860 IC50 = 1.7 nM T34296 CPK09X 20651316 IC50 = 1 nM T34296 C30EAU 20651317 IC50 = 305 nM T34296 C48TWB 20728102 IC50 > 5000 nM T34296 C18RXS 20735191 IC50 < 0.1 nM T34296 C4I1OM 20735209 IC50 = 9 nM T34296 CF1CK9 20735364 IC50 = 1 nM T34296 C09JTR 21130554 IC50 = 0.4 nM T34296 CW1JS2 21130555 IC50 = 24000 nM T34296 C6VP1T 21130556 IC50 = 0.3 nM T34296 C15UGO 21130558 IC50 = 24 nM T34296 C9H3IG 21130559 IC50 = 1.6 nM T34296 C8Q2OD 21130561 IC50 = 2.4 nM T34296 C25FAD 21130562 IC50 = 0.6 nM T34296 C3FAU5 21130572 IC50 = 600 nM T34296 C19AEV 21130574 IC50 = 400 nM T34296 CW2Q5A 21130590 IC50 = 160 nM T34296 C9HMC0 21130591 IC50 = 161 nM T34296 CM92DX 21304705 IC50 = 9 nM T34296 CJ0Y9V 21304706 IC50 = 7 nM T34296 C5X1YM 21304708 IC50 = 11 nM T34296 C0Z3LD 21304710 IC50 = 1 nM T34296 C8F5AH 21310747 IC50 = 26 nM T34296 CG18HB 21310751 IC50 = 19 nM T34296 CEW0M3 21310753 IC50 = 11 nM T34296 CC2L1Z 21310756 IC50 = 959 nM T34296 C0T2QX 21310757 IC50 = 24 nM T34296 CWM7F2 21310775 IC50 = 138 nM T34296 CNEW70 21310777 IC50 = 50 nM T34296 CY12PI 21310778 IC50 = 42 nM T34296 CV10FJ 21310779 IC50 = 134.9 nM T34296 CPT4E5 21310780 IC50 = 982 nM T34296 CJ2U7K 21310781 IC50 = 728 nM T34296 C5SG2L 21310789 IC50 = 84 nM T34296 C3TI6Y 21310790 IC50 = 1 nM T34296 C87BMF 21310824 IC50 = 14 nM T34296 C26IPQ 21310829 IC50 = 11 nM T34296 CIB1X5 21310851 IC50 = 43 nM T34296 C6OZL3 21310926 IC50 = 113 nM T34296 C72BVA 21310934 IC50 = 717 nM T34296 CUJ6A1 21310984 IC50 = 137 nM T34296 C96REO 21584504 IC50 = 15 nM T34296 C8N6DH 21931010 IC50 = 0.53 nM T34296 CA6E9I 21931045 IC50 = 7.5 nM T34296 CN16ZT 21931049 IC50 = 0.63 nM T34296 C8IBZ2 21931061 IC50 = 0.4 nM T34296 CVS02H 21931065 IC50 = 1.6 nM T34296 CM9XW7 21931067 IC50 = 0.35 nM T34296 C27BZI 21931069 IC50 = 7.8 nM T34296 CO46GR 21931088 IC50 = 3.4 nM T34296 CS2KZ5 21931099 IC50 = 2.4 nM T34296 C7PQU4 21931103 IC50 = 6.1 nM T34296 CLQ58R 21931105 IC50 = 0.34 nM T34296 CWCN52 21931106 IC50 = 1 nM T34296 CX6QD0 21931115 IC50 = 12 nM T34296 COJ2R8 21931118 IC50 = 0.84 nM T34296 C94BWM 21931138 IC50 = 0.46 nM T34296 CIC4S9 22004232 IC50 = 7 nM T34296 C5FWN2 22248619 IC50 = 77 nM T34296 CH6U1G 22338710 IC50 = 75 nM T34296 CO91AD 22341241 Ki > 5025 nM T34296 CJW3E0 22482219 IC50 = 194 nM T34296 CE5DH1 22484408 IC50 = 1.8 nM T34296 CZT05X 22484417 Ki = 1.6 nM T34296 CZT64B 22484431 Ki = 1.5 nM T34296 C1O7RC 22485248 IC50 = 70 nM T34296 CAM10T 22485252 IC50 = 0.8 nM T34296 CBJS34 22485260 IC50 < 0.1 nM T34296 C9MU7N 22485263 IC50 = 6 nM T34296 CEGJ03 22485276 IC50 = 2.9 nM T34296 C7VB8G 22485289 IC50 = 0.3 nM T34296 CNB02I 22485291 IC50 = 0.1 nM T34296 CAY3N6 22485292 IC50 = 2.7 nM T34296 C94OCJ 22485302 IC50 = 0.25 nM T34296 C3YL5X 22485311 IC50 = 0.25 nM T34296 C80RSQ 22485314 IC50 = 0.2 nM T34296 CWA03L 22485327 IC50 = 0.3 nM T34296 C6JRW5 22485340 IC50 = 0.1 nM T34296 C5JZF1 22485344 IC50 = 0.8 nM T34296 CI7MY5 22485346 IC50 = 0.25 nM T34296 CI1YL7 22485347 IC50 = 0.2 nM T34296 C25OBD 22485356 IC50 = 0.45 nM T34296 C7I0EW 22485367 IC50 = 0.3 nM T34296 CL64TJ 22485368 IC50 = 0.6 nM T34296 CT4GF9 22485381 IC50 = 27.7 nM T34296 C27NDB 22485386 IC50 = 1.2 nM T34296 CTJ9I3 22485392 IC50 = 0.5 nM T34296 C3MG9P 22485396 IC50 = 1.9 nM T34296 CZY10U 22485408 IC50 = 5.5 nM T34296 C89AGT 22485413 IC50 = 0.6 nM T34296 C03NLM 22485417 IC50 = 0.1 nM T34296 C8GHU9 22485432 IC50 = 0.5 nM T34296 CIN18B 22598309 IC50 = 15.1 nM T34296 C2X3VB 22598316 IC50 = 1.57 nM T34296 C9BT5F 22626996 IC50 = 114 nM T34296 C7ITG0 22644780 IC50 = 20.89 nM T34296 CIQ76F 22644837 IC50 = 5 nM T34296 CYJ48I 22644895 IC50 = 36 nM T34296 CQB36V 22644965 IC50 = 4 nM T34296 CVM1O6 22644970 IC50 = 7 nM T34296 C0K1GE 22645081 IC50 = 20 nM T34296 C2Q4XK 22707806 IC50 = 0.2 nM T34296 CD4Z6P 22707833 IC50 = 20 nM T34296 CMYK90 22707860 IC50 < 0.1 nM T34296 CDQ12R 22712799 IC50 = 100000 nM T34296 CX40LP 22712801 IC50 = 75000 nM T34296 CVF9M4 22922043 IC50 = 42520 nM T34296 CIYA45 22985930 IC50 = 0.1 nM T34296 CF75MS 23017979 IC50 = 25000 nM T34296 CQJ3S4 23018008 IC50 = 7000 nM T34296 C9IW3E 23433373 IC50 = 6700 nM T34296 C4VG8C 23506747 IC50 = 433 nM T34296 CK97AT 23506779 IC50 = 68 nM T34296 CP94QR 23506783 IC50 = 11 nM T34296 CX32YK 23513795 IC50 = 10 nM T34296 C6IZ1S 23513821 IC50 = 69 nM T34296 CPNM93 23513825 IC50 = 59 nM T34296 CML90Q 23513831 IC50 = 54 nM T34296 C87RTM 23513845 IC50 = 327 nM T34296 CNSU58 23513850 IC50 = 135 nM T34296 C4R2AJ 23625454 IC50 = 3199 nM T34296 CD3U8A 23627203 Ki = 1700 nM T34296 CL24JR 23655078 IC50 = 470 nM T34296 COIZ43 23655713 IC50 = 9140 nM T34296 CURM98 23655714 IC50 > 100000 nM T34296 CO90JC 23655717 IC50 > 100000 nM T34296 C56NMQ 23655910 IC50 = 34000 nM T34296 C9QZX5 23655911 IC50 = 3260 nM T34296 CA8W3K 23656106 IC50 = 384 nM T34296 CU4R7T 23656291 IC50 = 11 nM T34296 CVZ2M1 23656293 IC50 = 10 nM T34296 CL5C1I 23656295 IC50 = 59 nM T34296 CZP12E 23656450 IC50 = 24 nM T34296 CA2PY5 23657418 IC50 = 10 nM T34296 CN9TY1 23657419 IC50 = 1340 nM T34296 C9FHZ1 23657421 IC50 = 50 nM T34296 CY9LF1 23657422 IC50 = 0.9 nM T34296 C28SPW 23657691 IC50 = 14000 nM T34296 CVJ1T7 23657695 IC50 = 41000 nM T34296 CAL05Q 23657697 IC50 = 30000 nM T34296 C3TWS6 24178109 Ki = 2.7 nM T34296 C35QME 24742028 IC50 = 0.8 nM T34296 CXEP14 24754176 IC50 > 100000 nM T34296 CSQ9E4 24754248 IC50 > 22000 nM T34296 CX16GL 24754251 IC50 > 100000 nM T34296 COY8K0 24754252 IC50 > 100000 nM T34296 CG3J2L 24768528 IC50 = 860 nM T34296 CQCJ17 24768595 IC50 = 0.2 nM T34296 CUS47E 24795059 IC50 = 65 nM T34296 CDRP74 24801536 IC50 = 1.61 nM T34296 CI61SG 24801701 IC50 = 31.1 nM T34296 C18FRG 24807817 IC50 = 55000 nM T34296 CW3X0F 24852010 IC50 = 6.8 nM T34296 C6YPS8 24852048 IC50 = 2.5 nM T34296 C4LXM8 24860420 IC50 = 1600 nM T34296 CK0CI6 24860421 IC50 = 1038 nM T34296 CZI59C 24860423 IC50 = 2075 nM T34296 CE29HI 24860424 IC50 = 6882 nM T34296 CT10JE 24860425 IC50 = 772 nM T34296 CRC98J 24860426 IC50 = 584 nM T34296 C8MKR0 24860427 IC50 = 2476 nM T34296 C3S6DX 24860428 IC50 = 30 nM T34296 C2LNE4 24860429 IC50 = 2912 nM T34296 CF4D0X 24860430 IC50 = 12000 nM T34296 C4FI5C 24901479 IC50 = 62 nM T34296 C6F0ZP 24901485 IC50 = 2.6 nM T34296 C4SP3O 24936157 IC50 = 0.19 nM T34296 CBUA83 24936183 IC50 = 7.3 nM T34296 C0EA5F 24936382 IC50 = 0.062 nM T34296 CB94KU 24958549 IC50 > 100000 nM T34296 CU3W7Y 24960377 IC50 > 200000 nM T34296 CNCA57 25004194 Ki = 4.677 nM T34296 CAQ9Z1 25022681 Ki > 5025 nM T34296 CA86UE 25049752 Ki = 2.2 nM T34296 C82NLV 25049754 Ki = 46 nM T34296 C6QFV4 25049756 Ki = 42 nM T34296 C4HVF2 25064051 IC50 = 93 nM T34296 C64BZH 25064052 IC50 = 1.22 nM T34296 CZ2TG0 25064053 IC50 = 1135 nM T34296 C3S8OA 25064054 IC50 = 277 nM T34296 CA64KF 25064283 IC50 = 456 nM T34296 C94MXR 25064485 IC50 = 200 nM T34296 CD9T2O 25064489 IC50 = 809 nM T34296 C3BC9Z 25064704 IC50 = 1286 nM T34296 C23TDS 25064904 IC50 = 632 nM T34296 C54MLN 25064905 IC50 = 56 nM T34296 C7T2UO 25064906 IC50 = 334 nM T34296 C16AIC 25064907 IC50 = 1353 nM T34296 CL9N8I 25064908 IC50 = 147 nM T34296 CJP30U 25065108 IC50 = 235 nM T34296 CMZV31 25065109 IC50 = 217 nM T34296 C03NHX 25065111 IC50 = 23 nM T34296 CE72DR 25065318 IC50 = 500 nM T34296 CEK1Y2 25065514 IC50 = 109 nM T34296 C3F5LH 25065515 IC50 = 500 nM T34296 CB0Z5P 25065946 IC50 = 1100 nM T34296 CJWD41 25066149 IC50 = 25000 nM T34296 CI4A7E 25066153 IC50 = 6000 nM T34296 CN9UM1 25066154 IC50 > 25000 nM T34296 CEU95V 25066364 IC50 > 25000 nM T34296 C0FJK5 25066365 IC50 > 25000 nM T34296 CZY4L8 25066366 IC50 > 25000 nM T34296 C2ZS5J 25066563 IC50 = 65 nM T34296 C6CMU0 25066564 IC50 = 180 nM T34296 CZO08G 25066566 IC50 = 100 nM T34296 C58KNZ 25066763 IC50 = 10 nM T34296 CVR52U 25066764 IC50 = 120 nM T34296 C8IBO5 25066765 IC50 = 10 nM T34296 CP85RV 25067176 IC50 = 59 nM T34296 CXP6V8 25067178 IC50 = 1.1 nM T34296 CD2KA4 25102047 IC50 = 4.6 nM T34296 CRW96X 25102048 IC50 = 2.2 nM T34296 CQ3O9P 25102050 IC50 = 0.68 nM T34296 CSHA26 25102051 IC50 = 1.4 nM T34296 C7ADO2 25102197 IC50 = 0.25 nM T34296 CX6D9J 25138245 Ki = 700 nM T34296 C7A6JQ 25138250 Ki = 2000 nM T34296 CR35QP 25144971 IC50 < 25 nM T34296 C0Y5BC 25145683 IC50 < 25 nM T34296 CB7V8Y 25147773 IC50 = 0.12 nM T34296 CEP9Q2 25180867 IC50 = 0.33 nM T34296 C7EH0J 25181615 Ki = 0.3 nM T34296 C6EWF1 25183622 Ki = 1.5 nM T34296 CAH7T2 25183623 Ki = 4.2 nM T34296 CXG2S6 25183625 Ki = 5.8 nM T34296 CHR2P1 25183768 Ki = 4.4 nM T34296 C8IM5D 25263230 IC50 = 120 nM T34296 C7PTR2 25263231 IC50 = 34000 nM T34296 C9MR1P 25263232 IC50 = 670 nM T34296 CW9MK2 25263233 IC50 = 600 nM T34296 CX9L6V 25263234 IC50 = 25446 nM T34296 CJE4M1 25263235 IC50 > 25000 nM T34296 CJ1H5A 25263236 IC50 = 100 nM T34296 C2CGD1 25263237 IC50 = 10 nM T34296 C57UXR 25263238 IC50 = 220 nM T34296 CO4K7N 25263239 IC50 = 2.1 nM T34296 C3TGE2 25263240 IC50 = 3.3 nM T34296 C06WRU 25263241 IC50 = 505 nM T34296 C95AVW 25263242 IC50 = 97 nM T34296 CXT42G 25263243 IC50 = 361 nM T34296 C50DHY 25263244 IC50 = 2500 nM T34296 C6R7SI 25263245 IC50 = 25000 nM T34296 C0H3RD 42627769 IC50 = 1810 nM T34296 CPO1Z3 44123600 Ki = 0.19 nM T34296 CWS64Q 44143474 IC50 = 8624 nM T34296 C7HV5Q 44143475 IC50 = 1900 nM T34296 C06IJY 44143476 IC50 = 440 nM T34296 CVM82U 44143477 IC50 = 415 nM T34296 C5XEB8 44143478 IC50 = 204 nM T34296 CJQF59 44143479 IC50 = 105 nM T34296 C0ZW7S 44143480 IC50 = 349 nM T34296 C7K0YS 44143481 IC50 = 1110 nM T34296 CWU1K0 44143482 IC50 = 835 nM T34296 CA29EQ 44143483 IC50 = 57 nM T34296 CA5P3E 44143484 IC50 = 1451 nM T34296 C7ER1N 44143485 IC50 = 266 nM T34296 C8YNO3 44143486 IC50 = 80 nM T34296 CLJG93 44143487 IC50 = 393 nM T34296 CJB54F 44143488 IC50 = 926 nM T34296 C9LF6X 44143582 IC50 = 0.3 nM T34296 CIH43B 44143583 IC50 = 11 nM T34296 CRO9K7 44143584 IC50 = 0.75 nM T34296 CNT3R8 44143585 IC50 = 6.8 nM T34296 C9TXG7 44143586 IC50 = 1058 nM T34296 CYW27E 44143587 IC50 = 575 nM T34296 C7XOT1 44143588 IC50 = 90 nM T34296 CQ2RN8 44143589 IC50 = 18 nM T34296 CF40SE 44143590 IC50 = 50 nM T34296 CIDW75 44143591 IC50 = 1325 nM T34296 CS7M0P 44143592 IC50 = 145 nM T34296 CKL4T2 44143593 IC50 = 9 nM T34296 CA25DI 44143594 IC50 = 0.7 nM T34296 CW95HZ 44143595 IC50 = 48 nM T34296 CCH26N 44143596 IC50 = 0.5 nM T34296 C6LM5N 44143597 IC50 = 61.5 nM T34296 C9QME0 44143598 IC50 = 9000 nM T34296 CI8Y0R 44143599 IC50 = 197 nM T34296 CE7X2W 44143600 IC50 = 1.3 nM T34296 CYJ0Z4 44143601 IC50 = 12.1 nM T34296 CP1UO5 44143602 IC50 = 300 nM T34296 CP8L7N 44143603 IC50 = 0.6 nM T34296 C6MSK3 44143604 IC50 = 1800 nM T34296 CRL6C0 44143605 IC50 = 0.8 nM T34296 C09OTR 44143606 IC50 = 390 nM T34296 CTM85Q 44143607 IC50 = 25 nM T34296 CV8BO6 44143608 IC50 = 1.3 nM T34296 C8HR2I 44143609 IC50 = 3.9 nM T34296 C90ISP 44143610 IC50 = 3.5 nM T34296 C2J5IT 44143611 IC50 = 2 nM T34296 CO9N4R 44143612 IC50 = 1 nM T34296 C85DBI 44143613 IC50 = 0.8 nM T34296 CQZ2W1 44143614 IC50 = 105 nM T34296 CAP7M2 44143615 IC50 = 60 nM T34296 C3DX9H 44143616 IC50 = 0.9 nM T34296 CIY4K3 44143617 IC50 = 0.6 nM T34296 CRQ0T5 44143618 IC50 = 0.5 nM T34296 COP5G1 44143619 IC50 = 0.4 nM T34296 CM45NB 44143620 IC50 = 110 nM T34296 C20COZ 44143621 IC50 = 1.6 nM T34296 CZC0U7 44143622 IC50 = 13.5 nM T34296 CR4ZF1 44143623 IC50 = 2.8 nM T34296 CZU83Q 44143624 IC50 = 16 nM T34296 CS26DC 44143625 IC50 = 8 nM T34296 C8B3VE 44143626 IC50 = 3.6 nM T34296 CG78RF 44143627 IC50 = 0.9 nM T34296 C8VQS4 44143628 IC50 = 1.7 nM T34296 CKV3C6 44143629 IC50 = 1.4 nM T34296 CK21NW 44143630 IC50 = 1.2 nM T34296 C4ELQ8 44143631 IC50 = 0.7 nM T34296 C9S8YH 44143632 IC50 = 0.7 nM T34296 CCZP24 44143633 IC50 = 230 nM T34296 C3VBX4 44143634 IC50 = 4 nM T34296 CU02HY 44143635 IC50 = 280 nM T34296 C16VZT 44143636 IC50 = 6.9 nM T34296 CSQ0V9 44143637 IC50 = 123 nM T34296 C27UYE 44143638 IC50 = 7.6 nM T34296 C5K2OM 44143639 IC50 = 188 nM T34296 CI7H6E 44143640 IC50 = 49 nM T34296 CH1IR0 44144307 IC50 = 43550 nM T34296 CEC98Q 44182306 IC50 = 430 nM T34296 C6CPZ7 44182307 IC50 = 620 nM T34296 CT80ED 44219901 Ki = 8.2 nM T34296 C94JVY 44219902 IC50 = 41 nM T34296 C7J6GH 44219903 IC50 = 63 nM T34296 C9J7WL 44219904 IC50 = 260 nM T34296 CRQ71E 44219905 IC50 = 600 nM T34296 C4Z0ID 44219906 IC50 = 91 nM T34296 CRNA25 44220092 IC50 = 25 nM T34296 C9T5ZF 44220093 IC50 = 1.4 nM T34296 CV38TE 44222825 IC50 = 15 nM T34296 CJI73R 44222826 IC50 = 7.2 nM T34296 CGQ30N 44222827 Ki = 5.8 nM T34296 CCI64J 44224245 IC50 = 106 nM T34296 C4P2GX 44236892 IC50 = 63 nM T34296 C9RD3F 44236893 IC50 = 57 nM T34296 CTMW04 44236894 IC50 = 31 nM T34296 C7U2CY 44236895 IC50 = 180 nM T34296 C84HYM 44236896 IC50 = 88 nM T34296 C1KY4B 44236897 IC50 = 17 nM T34296 C4PO8V 44236898 IC50 = 245 nM T34296 C8IJ2C 44236899 IC50 = 1550 nM T34296 CG52XV 44236900 IC50 = 6000 nM T34296 C72XPC 44236901 IC50 = 460 nM T34296 C4TDM2 44236902 IC50 = 480 nM T34296 CJW1A3 44236903 IC50 = 290 nM T34296 C9DNJ0 44236904 IC50 > 50000 nM T34296 CW1AF0 44236905 IC50 = 220 nM T34296 CDM1X4 44236906 IC50 = 32 nM T34296 C81SZN 44236907 IC50 = 6 nM T34296 CQ1YS7 44236908 IC50 = 40 nM T34296 C0B2LG 44236909 IC50 = 6 nM T34296 CDI34Y 44236910 IC50 = 25 nM T34296 C6MQO3 44236911 IC50 = 2 nM T34296 C0OY8X 44236912 IC50 = 4 nM T34296 CLRT69 44247751 IC50 = 4.1 nM T34296 CX4VZ8 44248449 IC50 = 40 nM T34296 C3JP6F 44248450 IC50 = 225 nM T34296 CD94XA 44248451 IC50 > 1000 nM T34296 C90ZLT 44248570 IC50 = 187 nM T34296 CF8G2N 44248571 IC50 = 269 nM T34296 CSY0M2 44248572 IC50 = 140 nM T34296 CHM1D7 44248573 IC50 = 1093 nM T34296 CM3Y8J 44248697 IC50 > 1000 nM T34296 CCXS75 44248811 IC50 = 370 nM T34296 CUSR91 44248815 IC50 = 215 nM T34296 COU3Y8 44266817 IC50 = 81.28 nM T34296 CUA5E0 44266818 IC50 = 33 nM T34296 CG23BI 44266830 IC50 = 14.13 nM T34296 CTX92S 44272249 IC50 = 416 nM T34296 CG92WS 44272353 IC50 = 252 nM T34296 CO2Z6K 44272475 IC50 = 5 nM T34296 C63KSL 44272540 IC50 = 47 nM T34296 C20JLP 44272837 IC50 = 123 nM T34296 C4YM6S 44272911 IC50 = 214 nM T34296 C6ON3U 44273235 IC50 = 1590 nM T34296 CSJ50I 44275605 IC50 = 1600 nM T34296 C8CB4A 44275752 IC50 = 14 nM T34296 CVI56W 44275768 IC50 = 300 nM T34296 CV3IQ8 44275769 IC50 = 180 nM T34296 C1O4TU 44275790 IC50 = 2000 nM T34296 CV2WC5 44275791 IC50 = 1600 nM T34296 CUD36E 44275806 IC50 = 110 nM T34296 CPXV83 44275825 IC50 = 1100 nM T34296 CZK8S5 44275954 IC50 = 30 nM T34296 CIK26Z 44276134 IC50 > 3000 nM T34296 C6S3GN 44283598 IC50 = 5 nM T34296 CXE73H 44283613 IC50 = 3 nM T34296 CP3L2U 44283938 IC50 = 170 nM T34296 CET62P 44287169 IC50 > 30000 nM T34296 CJG20R 44287181 IC50 = 6100 nM T34296 CHNI65 44287384 IC50 >> 30000 nM T34296 CB72PO 44287385 IC50 = 27000 nM T34296 C5CT4M 44287386 IC50 = 5100 nM T34296 CS4Z7D 44287398 IC50 = 12000 nM T34296 CF1QK7 44287413 IC50 > 30000 nM T34296 CJ7VW3 44291166 IC50 = 12 nM T34296 C51TQK 44291531 IC50 = 3.8 nM T34296 CF21CS 44291532 IC50 = 3 nM T34296 CU75TB 44291559 IC50 = 96 nM T34296 C06JAO 44291626 IC50 = 20 nM T34296 C2Y0PK 44302023 IC50 = 21 nM T34296 C5S3UO 44302024 IC50 = 11 nM T34296 C8ERW6 44302042 IC50 = 11 nM T34296 CFQ68V 44302071 IC50 = 37 nM T34296 CWB83G 44302076 IC50 = 7 nM T34296 CY1J9U 44302096 IC50 = 17 nM T34296 C5TF4K 44302162 IC50 = 13 nM T34296 CW94ZQ 44302164 IC50 = 200 nM T34296 C5X1WY 44302183 IC50 = 21 nM T34296 C7G3BN 44302200 IC50 = 36 nM T34296 CZP20C 44302339 IC50 = 22 nM T34296 CO73BW 44302357 IC50 = 13 nM T34296 CPC25G 44302409 IC50 = 54 nM T34296 C4NDA2 44302416 IC50 = 26 nM T34296 C24ZWF 44302429 IC50 = 29 nM T34296 C5H6OV 44302627 IC50 = 43 nM T34296 C6QR7C 44302634 IC50 = 67 nM T34296 CG8KJ0 44302661 IC50 = 8 nM T34296 CX1M3Q 44302666 IC50 = 16 nM T34296 CBQ7P3 44302751 IC50 = 21 nM T34296 C36CQP 44302952 IC50 = 32 nM T34296 C4SJF3 44309329 IC50 = 1 nM T34296 C7ED1H 44309330 IC50 = 2 nM T34296 C1E3KF 44309437 IC50 = 4 nM T34296 CH3SU2 44309482 IC50 = 1752 nM T34296 C6N5SL 44309531 IC50 = 18 nM T34296 CO7TS8 44309532 IC50 = 38 nM T34296 CQ7Z0W 44309533 IC50 = 163 nM T34296 CJ0L4P 44309550 IC50 = 3 nM T34296 C6J3WN 44309662 IC50 = 3 nM T34296 CY96UH 44309686 IC50 = 6 nM T34296 C49MHR 44309863 IC50 = 661 nM T34296 CMW0U4 44309879 IC50 = 39 nM T34296 CK6BT0 44309901 IC50 = 142 nM T34296 C5WZR7 44309939 IC50 = 44 nM T34296 C2BLO9 44314811 IC50 = 13 nM T34296 CSY5R3 44314812 IC50 = 17 nM T34296 C0BJ7X 44314813 IC50 = 54 nM T34296 C1V9FZ 44315040 IC50 = 19 nM T34296 C02YGK 44315041 IC50 > 300 nM T34296 C64MTA 44315075 IC50 = 7.7 nM T34296 C85WJB 44315076 IC50 = 9.4 nM T34296 CXLD02 44315105 IC50 = 43 nM T34296 CIJ8H3 44315114 IC50 = 37 nM T34296 C5G7OS 44315115 IC50 = 24 nM T34296 CBP7S0 44315139 IC50 = 44 nM T34296 C4GR1C 44315140 IC50 = 58 nM T34296 CWS3E8 44315141 IC50 = 18 nM T34296 CPAT25 44315142 IC50 = 7.7 nM T34296 C9YK1H 44315143 IC50 = 30 nM T34296 CH48TD 44315155 IC50 = 210 nM T34296 C3VB1J 44315156 IC50 = 31 nM T34296 C79QEK 44315157 IC50 = 11 nM T34296 C62FXJ 44315244 IC50 = 8.3 nM T34296 CB0VI3 44315245 IC50 = 4.3 nM T34296 C4BWR2 44315286 IC50 = 70 nM T34296 CH4YI9 44315311 IC50 = 13 nM T34296 COVF49 44315312 IC50 = 10 nM T34296 C50IQE 44315333 IC50 = 7 nM T34296 C1LC5H 44315334 IC50 = 29 nM T34296 CKAL69 44315860 IC50 = 2 nM T34296 C0HR5Q 44316157 IC50 = 3.981 nM T34296 C5RJ6F 44316310 IC50 = 6 nM T34296 CSA5P7 44316333 IC50 = 1 nM T34296 CS5V0J 44316334 IC50 = 531 nM T34296 CS7D5E 44317086 IC50 = 5 nM T34296 CH70XB 44317451 IC50 = 233 nM T34296 C89IQW 44318090 IC50 = 3 nM T34296 C15WQO 44323336 IC50 = 2.2 nM T34296 C9UOW2 44323407 IC50 = 65 nM T34296 C4C1WD 44323426 IC50 = 4.6 nM T34296 C85JGD 44323430 IC50 = 45.71 nM T34296 CKP12T 44323431 IC50 = 10.4 nM T34296 C4R8OD 44323432 IC50 = 17 nM T34296 COQ6U7 44323456 IC50 = 5.1 nM T34296 CL07GT 44323526 IC50 = 26 nM T34296 CZRF63 44323527 IC50 = 16 nM T34296 CT9M4F 44323539 IC50 = 10.96 nM T34296 CQG24X 44323540 IC50 = 6.2 nM T34296 CND4Y1 44323633 IC50 = 89.13 nM T34296 CBN51C 44324159 IC50 = 87.1 nM T34296 CT01XC 44324546 IC50 = 400 nM T34296 CK5F4S 44324646 IC50 = 400 nM T34296 C6BJ7X 44324656 IC50 = 800 nM T34296 CE6VR2 44324878 IC50 = 400 nM T34296 CYLN13 44324879 IC50 = 2900 nM T34296 CBI48M 44324889 IC50 = 300 nM T34296 CEQ43S 44324934 IC50 = 4000 nM T34296 CRM0C1 44325233 IC50 = 2000 nM T34296 CN0GX1 44325234 IC50 = 200 nM T34296 C5STC3 44325248 IC50 = 300 nM T34296 C2ZH0F 44327181 IC50 = 195 nM T34296 C8V3AO 44327386 IC50 = 41 nM T34296 C0UC5H 44327407 IC50 = 18 nM T34296 C6TPB1 44327409 IC50 = 8 nM T34296 C8ZI0P 44327432 IC50 = 146 nM T34296 CVJ9Q6 44327443 IC50 = 28 nM T34296 C4R9WM 44327681 IC50 = 27 nM T34296 CR40TV 44327695 IC50 = 207 nM T34296 C6IM7G 44327755 IC50 = 28 nM T34296 CHU2P7 44328876 IC50 = 2 nM T34296 C0KA4S 44328937 IC50 = 3 nM T34296 CLT8B6 44328971 IC50 = 4 nM T34296 C7J0ZI 44329016 IC50 = 2 nM T34296 CW24VN 44329040 IC50 = 2 nM T34296 C9J0VO 44329253 IC50 = 2 nM T34296 C90CHA 44329405 IC50 = 600 nM T34296 CB0G1H 44329644 IC50 = 2000 nM T34296 CK9HO7 44329673 IC50 = 100 nM T34296 C07GRS 44329693 IC50 = 19.95 nM T34296 CBH16R 44329694 IC50 = 39.81 nM T34296 CG3E7A 44329712 IC50 = 8 nM T34296 C9SN6I 44329713 IC50 = 199.53 nM T34296 CZ2FW6 44329725 IC50 = 100 nM T34296 CDKI48 44329741 IC50 = 39.81 nM T34296 CK3M2H 44329742 IC50 = 200 nM T34296 C39RDS 44329886 IC50 = 7.943 nM T34296 C3YAF6 44329898 IC50 = 7000 nM T34296 C63RHP 44329909 IC50 = 20 nM T34296 CVQA75 44329910 IC50 = 79.43 nM T34296 C84SLI 44329926 IC50 = 10 nM T34296 CJS6B1 44329927 IC50 = 40 nM T34296 C9R1ZE 44330132 IC50 = 25000 nM T34296 CLU8I7 44330135 IC50 = 3300 nM T34296 C1IE0S 44330147 IC50 = 40000 nM T34296 CPG7N2 44330149 IC50 = 3300 nM T34296 CYP6S4 44330152 IC50 = 5000 nM T34296 CMGA28 44330163 IC50 = 22000 nM T34296 CD0L6S 44331932 IC50 = 3 nM T34296 CHIG68 44331976 IC50 = 6 nM T34296 CF4JN0 44331983 IC50 = 3 nM T34296 CG2AH4 44331984 IC50 = 4 nM T34296 CPB96A 44332003 IC50 = 6 nM T34296 C6RE3I 44332107 IC50 = 0.7 nM T34296 C3L1HQ 44332161 IC50 = 6 nM T34296 CG2Q8W 44332306 IC50 = 84 nM T34296 CY0MQ9 44332313 IC50 = 7 nM T34296 CFP3X8 44334949 IC50 = 96 nM T34296 CV5RF0 44334963 IC50 = 519 nM T34296 C4AOZ7 44334981 IC50 = 218 nM T34296 CXW59C 44334982 IC50 = 22.3 nM T34296 CCH1W8 44334983 IC50 = 3.7 nM T34296 CQ0UI1 44335017 IC50 = 44.2 nM T34296 CX58SB 44335240 IC50 = 5.5 nM T34296 CA96JG 44335285 IC50 = 17 nM T34296 C0Y2CZ 44339375 IC50 = 17 nM T34296 CP12TJ 44339394 IC50 = 4 nM T34296 COR15M 44339402 IC50 = 11 nM T34296 CU5NI2 44339444 IC50 = 6 nM T34296 CISO73 44339448 IC50 = 8 nM T34296 C4QKI6 44339451 IC50 = 7 nM T34296 CEUP59 44339452 IC50 = 4 nM T34296 CU7DZ9 44339462 IC50 = 98 nM T34296 CLT8C6 44339543 IC50 = 3 nM T34296 C6M4UR 44339544 IC50 = 127 nM T34296 C5PQ1B 44339569 IC50 = 7 nM T34296 CA65PF 44339570 IC50 = 20 nM T34296 C4W8LS 44339571 IC50 = 19 nM T34296 COUE24 44339575 IC50 = 40 nM T34296 CMA2L3 44339647 IC50 = 4 nM T34296 CE3MT4 44341611 Ki = 4700 nM T34296 CJTZ45 44341652 Ki = 200000 nM T34296 CE0PL2 44341937 IC50 = 2 nM T34296 C2S1GO 44341947 IC50 = 1.5 nM T34296 C5FG4N 44341974 IC50 = 4.6 nM T34296 CN4UP5 44341977 IC50 = 14 nM T34296 C2S7PL 44341987 IC50 = 0.97 nM T34296 C6EY7C 44342019 IC50 = 24 nM T34296 CK4WL8 44342020 IC50 = 19 nM T34296 C8WH0C 44342056 IC50 = 0.93 nM T34296 CT68XS 44342103 IC50 = 13 nM T34296 CWYV36 44342115 IC50 = 9.7 nM T34296 CER9M5 44342120 IC50 = 0.93 nM T34296 C0KO4U 44342125 IC50 = 0.87 nM T34296 CA1X5L 44342131 IC50 = 49 nM T34296 CIS5M3 44342135 IC50 = 4.6 nM T34296 C80EKJ 44342143 IC50 = 5 nM T34296 C29IPJ 44342160 IC50 = 1.3 nM T34296 CVNF08 44342224 IC50 = 1.5 nM T34296 C5PAS4 44342236 IC50 = 210 nM T34296 CMI0T2 44342251 IC50 = 1.7 nM T34296 CAN54Y 44342308 IC50 = 25 nM T34296 CR9G4Y 44342410 IC50 = 0.56 nM T34296 CD3Y9N 44342428 IC50 = 0.65 nM T34296 CTQ6P4 44344631 IC50 = 2300 nM T34296 CCF94Z 44349787 IC50 = 3.1 nM T34296 C1L2GF 44350073 IC50 = 133 nM T34296 CQ5RN6 44350101 IC50 = 682 nM T34296 CE2X3Q 44350116 IC50 > 100 nM T34296 CQ60YD 44360219 IC50 = 2.1 nM T34296 CT4C6P 44360260 IC50 = 4 nM T34296 CY5I3O 44360286 IC50 = 7.5 nM T34296 C40OCB 44360287 IC50 = 1.4 nM T34296 C90CYD 44367175 IC50 = 3 nM T34296 C2DV0R 44367276 IC50 = 0.4 nM T34296 C5BAW2 44367284 IC50 < 0.4 nM T34296 C2YG5E 44367285 IC50 = 8 nM T34296 CUDF82 44367309 IC50 = 2 nM T34296 CI0ZD9 44371783 IC50 = 176 nM T34296 C4VR5M 44371799 IC50 = 338 nM T34296 C4FHG7 44371800 IC50 = 131 nM T34296 CZ5I8B 44386229 IC50 = 475 nM T34296 C0S7EU 44389231 IC50 = 2500 nM T34296 CN8F1Q 44389253 IC50 > 1200 nM T34296 CB71LT 44389285 IC50 = 270 nM T34296 CZ6PU7 44389401 Ki = 0.33 nM T34296 C40BHI 44389462 Ki = 54 nM T34296 CO7P6Y 44389492 Ki = 5.8 nM T34296 CS1N5F 44389516 Ki = 25 nM T34296 CX25WY 44389537 Ki = 934 nM T34296 CB1RD0 44389551 Ki = 1100 nM T34296 CO4W0Y 44389552 Ki = 0.95 nM T34296 C3YPG6 44390245 IC50 = 8 nM T34296 COG80H 44390258 IC50 = 307 nM T34296 C0U3XR 44390274 IC50 = 363 nM T34296 CAC3F2 44390281 IC50 = 225 nM T34296 CRE9G2 44390289 IC50 = 11 nM T34296 CN41JE 44390299 IC50 = 19.95 nM T34296 C5VBL2 44390300 IC50 = 8.913 nM T34296 C4YUK7 44390304 IC50 = 88 nM T34296 C47EZV 44390314 IC50 = 446 nM T34296 CF65OK 44390317 IC50 = 30.9 nM T34296 CV45JT 44390322 IC50 = 180 nM T34296 C3GU1Q 44390323 IC50 = 52 nM T34296 CAZ2B4 44390326 IC50 = 1063 nM T34296 C2Y7MR 44390338 IC50 = 395 nM T34296 CA47CR 44390351 IC50 = 128 nM T34296 CYW89M 44390352 IC50 = 140 nM T34296 CPK9Z6 44390355 IC50 = 311 nM T34296 CEJH75 44390356 IC50 = 17 nM T34296 CWYM93 44390391 IC50 = 142 nM T34296 C3EZ0W 44391336 IC50 = 19 nM T34296 C1E5JC 44391341 IC50 = 0.54 nM T34296 CT5Y1X 44391344 IC50 = 19 nM T34296 CP0QS3 44391345 IC50 = 4.1 nM T34296 CR0Y3D 44391350 IC50 = 3.1 nM T34296 CMTB94 44391351 IC50 = 3.1 nM T34296 CC7QW9 44391352 IC50 = 1 nM T34296 C0FC5U 44391354 IC50 = 0.61 nM T34296 CMS1Z6 44391356 IC50 = 1.4 nM T34296 CA3NH7 44391357 IC50 = 6 nM T34296 CTK65L 44391360 IC50 = 8 nM T34296 C0S4YB 44391365 IC50 = 53 nM T34296 CN4GJ0 44391366 IC50 = 56 nM T34296 CKL09S 44391376 IC50 = 150 nM T34296 CVTB31 44391377 IC50 > 300 nM T34296 C2R8AW 44391389 IC50 = 390 nM T34296 C3BPI8 44391397 IC50 = 2.1 nM T34296 CW90KP 44391398 IC50 = 1.4 nM T34296 C1N8KB 44391410 IC50 = 18 nM T34296 CB0HI5 44391419 IC50 = 0.87 nM T34296 C5XSH0 44391424 IC50 = 140 nM T34296 CFH41S 44391425 IC50 = 0.95 nM T34296 C49DCW 44391434 IC50 = 9.2 nM T34296 CZ89IE 44391435 IC50 = 5.9 nM T34296 CP0AU9 44391440 IC50 = 3.8 nM T34296 C9BMR7 44391444 IC50 = 0.87 nM T34296 CR4U6B 44391445 IC50 = 3.1 nM T34296 CH59GY 44391449 IC50 = 5 nM T34296 CU7N6G 44391450 IC50 = 3.6 nM T34296 CD5TX3 44391460 IC50 = 190 nM T34296 CCK39J 44391461 IC50 = 3.1 nM T34296 C3V1PB 44391476 IC50 = 1.7 nM T34296 C37DHM 44391486 IC50 = 28 nM T34296 CMGB67 44393214 IC50 = 20 nM T34296 CA1S5T 44393217 IC50 = 21 nM T34296 CSC6N1 44393218 IC50 = 53 nM T34296 CBO9E6 44393239 IC50 = 33 nM T34296 CQNR83 44393261 IC50 = 47 nM T34296 CT1LM8 44393266 IC50 = 17 nM T34296 C0SGF6 44393279 IC50 = 17 nM T34296 CYFC07 44393295 IC50 = 67 nM T34296 C24INM 44393328 IC50 = 32 nM T34296 C15IZJ 44393358 IC50 = 12 nM T34296 C3HP5Q 44393383 IC50 = 19 nM T34296 CS06PD 44393394 IC50 = 42 nM T34296 CFA83O 44393414 IC50 = 97 nM T34296 CCO3S9 44393444 Ki = 1758 nM T34296 CNO4P6 44393516 Ki = 377 nM T34296 C5OIK4 44393520 Ki > 5000 nM T34296 CDG2K7 44393747 IC50 = 1 nM T34296 CWUV21 44393760 IC50 = 140 nM T34296 CQ6WZ5 44393836 IC50 = 5 nM T34296 CR58XA 44393837 IC50 = 1.3 nM T34296 CIH8T9 44393838 IC50 = 28 nM T34296 CK95WI 44393841 IC50 = 46 nM T34296 CAC72Q 44393867 IC50 = 38 nM T34296 CFR4G2 44393892 IC50 = 0.43 nM T34296 CMBJ97 44393897 IC50 = 0.39 nM T34296 CF3M5K 44393910 IC50 = 13 nM T34296 C4YJI9 44393913 IC50 = 300 nM T34296 C0E8BQ 44393936 IC50 = 17 nM T34296 CGU63Q 44393964 IC50 > 300 nM T34296 C8P0IG 44393980 IC50 = 15 nM T34296 CP24NE 44394027 IC50 = 9.8 nM T34296 CHP81Z 44394038 IC50 = 1.1 nM T34296 CKB7S1 44394067 IC50 > 300 nM T34296 CZB81D 44395506 IC50 = 1 nM T34296 CKV57D 44399071 IC50 = 2.8 nM T34296 C0NSO4 44399233 IC50 = 2.1 nM T34296 CRL5D0 44399252 IC50 = 14 nM T34296 CHL9S2 44399294 Ki > 5020 nM T34296 CD49UI 44399312 Ki = 4020 nM T34296 C7IDB0 44399341 IC50 = 3.5 nM T34296 C2UDW8 44399397 IC50 = 7.8 nM T34296 CA0DV5 44399432 IC50 = 1.2 nM T34296 C95RKA 44399451 IC50 = 188 nM T34296 CIA8T3 44399555 Ki > 5020 nM T34296 CV2CQ0 44399635 IC50 = 6.5 nM T34296 CJWB10 44399637 IC50 = 19 nM T34296 CW83LM 44399638 IC50 = 0.5 nM T34296 C7XCI6 44399665 IC50 = 53 nM T34296 CW9MD1 44399704 IC50 = 36 nM T34296 C2JMC1 44399712 IC50 = 4.3 nM T34296 CD8Q2Y 44399731 IC50 = 8 nM T34296 CC16YQ 44399733 IC50 = 1.4 nM T34296 C9KGL0 44404474 IC50 = 0.61 nM T34296 C92KDG 44404475 IC50 = 0.4 nM T34296 C07CGB 44404477 IC50 = 9.5 nM T34296 C7VH3G 44404484 IC50 = 5.9 nM T34296 CC29XL 44404490 IC50 = 55 nM T34296 CCN16G 44404500 IC50 = 17 nM T34296 C69GZU 44404501 IC50 = 3.4 nM T34296 CY6WL5 44404502 IC50 = 1.9 nM T34296 CWGQ46 44404503 IC50 = 4.9 nM T34296 CLXM58 44404504 IC50 = 3.8 nM T34296 C1F9HO 44404506 IC50 = 67 nM T34296 CLU41O 44404507 IC50 = 27 nM T34296 C30DKN 44404553 IC50 = 0.1 nM T34296 C7Z0OH 44404761 IC50 = 83 nM T34296 CIC60V 44406452 IC50 = 4.4 nM T34296 C1F0DR 44406571 IC50 = 20 nM T34296 CT7CD3 44409041 IC50 = 14 nM T34296 CJ2Q8Z 44409042 IC50 = 86 nM T34296 CY3KF2 44409047 IC50 = 17 nM T34296 CT01JW 44409066 IC50 = 4 nM T34296 CJNE37 44409163 IC50 = 2 nM T34296 CVA69I 44409164 IC50 = 4 nM T34296 C9I0JW 44409184 IC50 = 27 nM T34296 C1JSU2 44409197 IC50 = 7 nM T34296 CW4BM3 44409214 IC50 = 8 nM T34296 CVRL76 44409215 IC50 = 2 nM T34296 C9F7HR 44409221 IC50 = 9 nM T34296 CJ70LK 44409222 IC50 = 7 nM T34296 C5J1PS 44409261 IC50 = 1 nM T34296 C06EZF 44409365 IC50 = 7 nM T34296 CV5AW8 44409366 IC50 = 29 nM T34296 C9PS4Q 44409369 IC50 = 24 nM T34296 C1S4GD 44409389 IC50 = 14 nM T34296 C69CGM 44409390 IC50 = 23 nM T34296 C1SKI7 44409405 IC50 = 48 nM T34296 C84ZSL 44411052 Ki = 3 nM T34296 CUE29K 44411053 Ki = 19 nM T34296 C6IKL1 44411602 IC50 = 1.4 nM T34296 CEB0S4 44411823 IC50 = 0.8 nM T34296 CVM7Y3 44413975 IC50 = 24 nM T34296 C4X0GA 44413977 IC50 = 14 nM T34296 CH01EO 44413978 IC50 = 13 nM T34296 CBT0P2 44413982 IC50 = 21 nM T34296 CIJ39D 44413983 IC50 = 39 nM T34296 C9BA0V 44413987 IC50 = 79 nM T34296 CHN85S 44414002 IC50 = 74 nM T34296 C2OJ4B 44414029 IC50 = 177 nM T34296 CF02QK 44419926 IC50 = 1.1 nM T34296 CR1Y6A 44419932 IC50 = 0.85 nM T34296 CVAC97 44419939 IC50 = 3.4 nM T34296 CONP58 44419944 IC50 = 3.9 nM T34296 CYA7G4 44419949 IC50 = 0.4 nM T34296 CNA02B 44419955 IC50 = 6.1 nM T34296 C0Y8RP 44419959 IC50 = 2.6 nM T34296 C0LI1C 44419992 IC50 = 0.84 nM T34296 C5UB4S 44419996 IC50 = 8 nM T34296 CZ5KM8 44421257 IC50 > 10000 nM T34296 CT5PC9 44422672 IC50 = 3.3 nM T34296 CS9D5U 44422720 IC50 = 1.1 nM T34296 CNWM05 44422723 IC50 = 4.2 nM T34296 C58LAY 44422724 IC50 = 13 nM T34296 CDQU41 44422736 IC50 = 63 nM T34296 CVUB56 44422737 IC50 = 24 nM T34296 CB8G2W 44422743 IC50 = 15 nM T34296 CFX42T 44422744 IC50 = 820 nM T34296 C9EL7F 44422749 IC50 = 480 nM T34296 CK5H7O 44429877 IC50 = 4000 nM T34296 CQL1X9 44429878 IC50 = 238 nM T34296 C1CYV2 44429879 IC50 = 295 nM T34296 C7AXP9 44429880 IC50 = 136 nM T34296 CXOS97 44429881 IC50 = 72 nM T34296 C2MQ0I 44429882 IC50 = 43 nM T34296 CQ5PT8 44429883 IC50 = 130 nM T34296 CQRO36 44429884 IC50 = 1159 nM T34296 CM27YB 44429885 IC50 = 155 nM T34296 C9JH0T 44429886 IC50 = 24.4 nM T34296 CD2B3T 44429887 IC50 = 205 nM T34296 C6V1CO 44429888 IC50 = 2040 nM T34296 CBC6W4 44429889 IC50 = 56 nM T34296 C7A0LF 44429890 IC50 = 166 nM T34296 CS0M3L 44429891 IC50 = 385 nM T34296 CX93QY 44429892 IC50 = 147 nM T34296 C8QKS0 44429894 IC50 = 23 nM T34296 CBS47K 44429896 IC50 = 38 nM T34296 CI7TG1 44429897 IC50 = 229 nM T34296 CLJ48T 44429898 IC50 = 195 nM T34296 C3F9CK 44429899 IC50 = 144 nM T34296 C8PVF7 44429900 IC50 = 117 nM T34296 C6U0TK 44429901 IC50 = 104 nM T34296 CBK9M5 44429902 IC50 = 190 nM T34296 C72YFT 44429903 IC50 = 354 nM T34296 CMO9Q3 44429905 IC50 = 449 nM T34296 C8BHL5 44431844 IC50 > 5000 nM T34296 CR1DN9 44431845 IC50 > 5000 nM T34296 CHFB16 44431846 IC50 > 5000 nM T34296 C0C3ZT 44431847 IC50 > 5000 nM T34296 CS49GV 44431848 IC50 > 5000 nM T34296 C4AVK5 44431849 IC50 > 5000 nM T34296 C5DH4Q 44431850 IC50 > 5000 nM T34296 CLHE45 44431851 IC50 > 5000 nM T34296 CYG29L 44431852 IC50 > 5000 nM T34296 C4OF5L 44431853 IC50 > 5000 nM T34296 CWU7G8 44434565 IC50 = 122 nM T34296 C70MGQ 44440455 Ki > 5025 nM T34296 CDY53F 44440460 Ki > 5025 nM T34296 CTB9P6 44440461 Ki = 392 nM T34296 C63RLK 44440462 Ki > 5025 nM T34296 C23JBO 44440463 Ki > 5025 nM T34296 CT9P3Y 44440464 Ki > 5025 nM T34296 CX32AM 44440465 Ki > 5025 nM T34296 C6FOC7 44440466 Ki > 5025 nM T34296 CMPX37 44440467 Ki > 5025 nM T34296 CV4F6Z 44440468 Ki > 5025 nM T34296 C6K8VB 44440469 Ki > 5025 nM T34296 C4Y0UM 44440470 Ki > 5025 nM T34296 CHU49A 44440471 Ki > 5025 nM T34296 C8OI4L 44440472 Ki > 5025 nM T34296 CV58YW 44441018 Ki > 5025 nM T34296 CV85PN 44441019 Ki > 5025 nM T34296 C5O2WK 44441020 Ki > 5025 nM T34296 CU67WS 44441021 Ki > 5025 nM T34296 CXZ53B 44441022 Ki = 2462 nM T34296 C8S7UT 44441023 Ki > 5025 nM T34296 CT4PZ9 44441024 Ki > 5025 nM T34296 CU9GE6 44441025 Ki > 5025 nM T34296 CB2IT4 44441026 Ki > 5025 nM T34296 CN4X2F 44441027 Ki = 3136 nM T34296 CPF45Y 44441028 Ki > 5025 nM T34296 CAM23N 44441029 Ki > 5025 nM T34296 C23BPG 44441030 Ki > 5025 nM T34296 C5YMT6 44441031 Ki > 5025 nM T34296 C9A6GJ 44441032 Ki > 5025 nM T34296 CYSU19 44441033 Ki > 5025 nM T34296 CB9P0C 44442303 IC50 = 1200 nM T34296 C7HO0Y 44442304 IC50 = 1100 nM T34296 CAR3S2 44442305 IC50 = 1170 nM T34296 CZK0A9 44442306 IC50 = 2860 nM T34296 C71MCV 44442307 IC50 = 1200 nM T34296 CN70HO 44442308 IC50 = 1110 nM T34296 CVE5P0 44442309 IC50 = 840 nM T34296 CGS18B 44442311 IC50 = 1010 nM T34296 CIZL27 44442312 IC50 = 1370 nM T34296 CCFV76 44442313 IC50 = 1190 nM T34296 CZ2PE6 44442315 IC50 = 950 nM T34296 C2N8BW 44442316 IC50 = 1740 nM T34296 CGR6E7 44442318 IC50 > 16666 nM T34296 C97ZHM 44442319 IC50 > 16666 nM T34296 C3DIB8 44442320 IC50 > 16666 nM T34296 C9IQD0 44444485 IC50 = 8.9 nM T34296 C64FGU 44444487 IC50 = 2.9 nM T34296 CR4O1V 44444516 IC50 = 138 nM T34296 CGZ20Y 44444519 IC50 = 7.33 nM T34296 CV4MK5 44444526 IC50 = 12 nM T34296 CI20ZD 44444531 IC50 = 0.6 nM T34296 C91QFR 44444569 IC50 = 0.49 nM T34296 CG3P8M 44444573 IC50 = 0.11 nM T34296 CO46QB 44444576 IC50 = 0.96 nM T34296 C9L4DH 44444578 IC50 = 0.1 nM T34296 CBC28D 44444580 IC50 = 0.4 nM T34296 CV0CI2 44444582 IC50 = 0.08 nM T34296 CL4BX1 44445917 IC50 = 15.85 nM T34296 CKW5G7 44445918 IC50 = 1 nM T34296 CE0O2Z 44445919 IC50 = 20.89 nM T34296 CSKN69 44455242 IC50 = 4 nM T34296 C3J1SV 44455676 IC50 = 11 nM T34296 C38VBL 44455836 IC50 = 13.4 nM T34296 CG0Z7I 44478924 IC50 = 2700 nM T34296 CFO27Y 44478926 IC50 = 84 nM T34296 CBZJ29 44478927 IC50 = 25 nM T34296 CRJ24K 44479197 IC50 = 12 nM T34296 CGOH82 44479198 IC50 = 940 nM T34296 CLV56M 44479199 IC50 = 78 nM T34296 CY92OQ 44479458 IC50 = 20000 nM T34296 CH1QG9 44479459 IC50 = 260 nM T34296 CB1NT7 44479460 IC50 = 62 nM T34296 C0JQ9L 44479699 IC50 = 74 nM T34296 C0DN1Q 44479700 IC50 = 55000 nM T34296 CTG24W 44479702 IC50 = 1800 nM T34296 CGZ49M 44479703 IC50 = 190 nM T34296 CAK94X 44563337 IC50 = 213 nM T34296 CY1A8V 44564505 IC50 = 3 nM T34296 C47XUD 44571675 IC50 > 200000 nM T34296 CQ7W5I 44580110 Ki > 5000 nM T34296 CWD32S 44580184 IC50 = 2277 nM T34296 CH8QS0 44596287 IC50 = 0.6 nM T34296 CW5A2D 44608129 IC50 = 8 nM T34296 CT7KX5 44608938 IC50 = 33 nM T34296 CJRP30 44608939 IC50 = 26 nM T34296 COI5K3 44608942 IC50 = 28 nM T34296 CS4C5T 44609098 IC50 = 2 nM T34296 CMLV87 44609099 IC50 = 28 nM T34296 C3T9SV 44609100 IC50 = 2.9 nM T34296 C0KR6J 44626353 IC50 = 1130 nM T34296 C25QLI 44626354 IC50 = 3760 nM T34296 CA1YC9 44626604 Ki = 19 nM T34296 CK6S5H 44626708 Ki = 1200 nM T34296 C0EJ1F 44626709 Ki = 30 nM T34296 CZR23J 44626710 Ki > 10000 nM T34296 CQB06H 44626711 Ki = 24 nM T34296 C19LWR 44634267 IC50 = 0.58 nM T34296 CZP79X 45268488 IC50 = 6.1 nM T34296 CK50JB 45268522 IC50 = 35 nM T34296 C2B0GI 45268787 Ki = 1.5 nM T34296 CVG5I2 45269378 IC50 = 11 nM T34296 CQC5Y4 45269386 IC50 = 14 nM T34296 CACH13 45269631 IC50 = 9.4 nM T34296 C2HI5Q 45269910 IC50 = 13800 nM T34296 C84JSF 45269911 IC50 = 60000 nM T34296 CTOH60 45270200 IC50 = 7.1 nM T34296 C2H5IY 45271017 IC50 = 7.4 nM T34296 C0YT8W 45271893 IC50 = 4.8 nM T34296 CVNO86 45271894 IC50 = 2.3 nM T34296 C7OQB3 45271912 IC50 = 13 nM T34296 C3SWC7 45272759 IC50 = 40 nM T34296 C36HRP 45377138 IC50 = 14 nM T34296 C6B7ZY 45377564 IC50 = 90 nM T34296 C5HAR6 45377565 IC50 = 150 nM T34296 CZYH47 45377567 IC50 = 56000 nM T34296 CKR0Q8 45377703 IC50 = 120 nM T34296 CMPE63 45482676 IC50 = 7900 nM T34296 CGH1U8 45482997 IC50 = 50200 nM T34296 C8AUI5 45482999 IC50 > 98000 nM T34296 C9W7IP 45483016 IC50 = 26100 nM T34296 CPB42K 45483022 IC50 = 33500 nM T34296 CBG76X 45483023 IC50 = 41900 nM T34296 CDW4C8 45483036 IC50 > 98000 nM T34296 CSX5I9 46175170 IC50 = 3.4 nM T34296 C56WVI 46184724 Ki = 3600 nM T34296 C8A3ER 46207232 IC50 = 2 nM T34296 CNF8R2 46207262 IC50 = 28 nM T34296 CT85VJ 46207292 IC50 = 2 nM T34296 CFW09H 46207358 IC50 = 6 nM T34296 C2W1KN 46225418 Ki = 65.3 nM T34296 CEVP65 46225419 Ki = 75.9 nM T34296 CA9QD6 46225437 Ki = 43.4 nM T34296 C25OWI 46225438 Ki = 36.7 nM T34296 CVL2I0 46225439 Ki = 2.1 nM T34296 CHKW61 46225440 Ki = 227 nM T34296 CTU9S1 46225452 Ki = 18.1 nM T34296 C9L8TO 46225453 Ki = 16.5 nM T34296 CJO87P 46225454 Ki = 22.3 nM T34296 C9KM3H 46225455 Ki = 5.3 nM T34296 CF12SQ 46225473 Ki = 28.6 nM T34296 CD6M3V 46225474 Ki = 3.6 nM T34296 C45RIP 46225475 Ki = 4.4 nM T34296 CW0G8P 46225476 Ki = 0.18 nM T34296 CGK72P 46225491 Ki = 2.5 nM T34296 CW42CR 46225492 Ki = 31.3 nM T34296 CJS16C 46225493 Ki = 4.2 nM T34296 C9WDJ6 46225506 Ki = 22.1 nM T34296 CV0G1O 46225507 Ki = 6.7 nM T34296 CG3SX7 46225508 Ki = 1.5 nM T34296 CP8NT9 46225509 Ki = 0.16 nM T34296 C7S1QD 46225519 Ki = 1.5 nM T34296 CWY81P 46225520 Ki = 7.5 nM T34296 C0ZIX3 46225521 Ki = 1.4 nM T34296 C6LY8C 46225536 Ki = 0.26 nM T34296 CZO14V 46225537 Ki = 0.62 nM T34296 C7HNV9 46225538 Ki = 0.22 nM T34296 CL2U4Z 46829322 Ki = 1 nM T34296 CH0Z1E 46844314 Ki > 40000 nM T34296 C7IXV6 46849757 IC50 > 10000 nM T34296 C20BTY 46856241 Ki = 3300 nM T34296 C5L8GF 46871738 IC50 = 0.6 nM T34296 CR1KF7 46871739 IC50 = 1 nM T34296 C8Q6YR 46871740 IC50 = 0.42 nM T34296 C58YSM 46871741 IC50 = 4 nM T34296 CR96AK 46890762 IC50 = 90 nM T34296 C5G9FX 46890763 IC50 = 6.7 nM T34296 COP78K 46890764 IC50 = 18 nM T34296 C60QSB 46890765 IC50 = 6 nM T34296 CQ5P9V 46890766 IC50 = 6.7 nM T34296 CB90YN 46890767 IC50 = 12.2 nM T34296 CUA7L6 46890821 IC50 = 10.7 nM T34296 C9BNQ7 46890822 IC50 = 6.4 nM T34296 CTF20Y 46890823 IC50 = 30 nM T34296 CR3QW7 46891107 IC50 = 2.7 nM T34296 C5MK3A 46891108 IC50 = 7.7 nM T34296 CQ5E1H 46891109 IC50 = 9 nM T34296 C0NW9D 46891110 IC50 = 130 nM T34296 C91LGI 46891170 IC50 = 8 nM T34296 CGI5B4 46891171 IC50 = 20 nM T34296 CZPM12 46891172 IC50 = 0.63 nM T34296 C2V6MW 46891173 IC50 = 1.9 nM T34296 CZWT45 46891207 IC50 = 28.6 nM T34296 CFE58Q 46891208 IC50 = 3.3 nM T34296 C8S7QX 46891209 IC50 = 2.4 nM T34296 C5Y0MN 46891255 IC50 = 17.5 nM T34296 CJ16SE 46891256 IC50 = 0.7 nM T34296 C7Y9TE 46891257 IC50 = 42.5 nM T34296 C7DT6W 46891258 IC50 = 32.7 nM T34296 CLF7Y4 46891311 IC50 = 28.8 nM T34296 C2IN7Y 46891312 IC50 = 35 nM T34296 CNXU57 46891313 IC50 = 11.3 nM T34296 CJB5D0 46891314 IC50 = 33.7 nM T34296 CVK0E5 46891356 IC50 = 11.4 nM T34296 C89RPO 46891357 IC50 = 7 nM T34296 CVB6K4 46891358 IC50 = 11 nM T34296 C67WEK 46891359 IC50 = 11.4 nM T34296 CPQ37V 46891414 IC50 = 70 nM T34296 C5LTI6 46891459 IC50 = 35 nM T34296 C92FBL 46891460 IC50 = 24.5 nM T34296 C1A0OE 46891522 IC50 = 9 nM T34296 C2I6FV 46891523 IC50 = 6.2 nM T34296 CAZ9Q5 46891524 IC50 = 4.4 nM T34296 CG02KB 46891525 IC50 = 50 nM T34296 C7ZG8J 46891526 IC50 = 18.1 nM T34296 CRQ13J 46891580 IC50 = 50 nM T34296 CERM39 46891581 IC50 = 28 nM T34296 CN8WF9 46891582 IC50 = 45 nM T34296 C86RLM 46891583 IC50 = 25.1 nM T34296 CM7S5T 46891584 IC50 = 40 nM T34296 CRY18A 46891617 IC50 = 26.8 nM T34296 C0S9WB 46919610 Ki = 3500 nM T34296 C6U1ZJ 46934733 IC50 = 24 nM T34296 CX89ON 46935023 IC50 = 11 nM T34296 CJ5U9I 46935024 IC50 = 8 nM T34296 CE3H7I 46938726 IC50 = 0.2 nM T34296 C9T0HR 46938727 IC50 = 0.6 nM T34296 C0YR7M 46938728 IC50 < 0.1 nM T34296 C2S7PK 46942365 Ki = 1.7 nM T34296 C2TE8J 47162079 IC50 = 39000 nM T34296 CE35HQ 49865150 IC50 = 100 nM T34296 C6YF2O 49865151 IC50 = 3300 nM T34296 CW5Q1C 49865207 IC50 = 110 nM T34296 C1FT8V 49865208 IC50 = 140 nM T34296 C0MC4H 49865209 IC50 = 75 nM T34296 CG17QX 49865271 IC50 = 180 nM T34296 CAR87K 49865272 IC50 = 330 nM T34296 CD8NS5 49865273 IC50 = 310 nM T34296 CJ5R6M 49865325 IC50 = 72 nM T34296 C6K2OQ 49865326 IC50 = 140 nM T34296 C8JM0Q 49865327 IC50 = 8 nM T34296 C0FJ1B 49865379 IC50 = 42 nM T34296 CD45PA 49865380 IC50 = 31 nM T34296 CF4VU8 49865381 IC50 = 10 nM T34296 CY1LX7 49865382 IC50 = 4 nM T34296 C16SGP 49865429 IC50 = 9 nM T34296 C6LI1B 49865430 IC50 = 100 nM T34296 C4GOT9 49865431 IC50 = 29 nM T34296 CFS08O 49865432 IC50 = 27 nM T34296 C6QYN3 49865473 IC50 = 3 nM T34296 C8QH3B 49865474 IC50 = 7 nM T34296 CE0M1T 49865521 IC50 = 25 nM T34296 CX67WT 49865522 IC50 = 9 nM T34296 CFRI63 49865523 IC50 = 36 nM T34296 CJR6H7 49865573 IC50 = 5 nM T34296 C7XW1Q 50907084 Ki = 1.7 nM T34296 C8RL5Q 50907292 Ki = 18 nM T34296 CUD7O0 50941549 IC50 > 10000 nM T34296 CX8N4D 50990920 IC50 = 430 nM T34296 CXF4V3 50990921 IC50 > 8100 nM T34296 CU2SX3 51355576 Ki = 7730 nM T34296 CLA96C 53232689 Ki = 0.6 nM T34296 C3BGW0 53233015 Ki > 40000 nM T34296 CZ06OY 53233469 IC50 = 0.66 nM T34296 CMQZ70 53242178 IC50 > 31000 nM T34296 CC9HK5 53245646 IC50 = 79.43 nM T34296 CRI92N 53311230 IC50 = 100 nM T34296 CB09MA 53318910 IC50 = 7.6 nM T34296 C47DIU 53318911 IC50 = 530 nM T34296 CC6DR2 53318912 IC50 = 23000 nM T34296 CWH47R 53319228 Ki = 2.9 nM T34296 C7V1NC 53320225 IC50 = 2300 nM T34296 CVH2B7 53320226 IC50 > 16000 nM T34296 CO8QK2 53320227 IC50 = 350 nM T34296 CNS3F2 53321542 IC50 = 16000 nM T34296 C1N2BX 53322876 IC50 = 2300 nM T34296 CSYW40 53322877 IC50 = 27000 nM T34296 CGUC59 53322878 IC50 = 4600 nM T34296 C3QHA6 53322879 IC50 > 4500 nM T34296 C1VNZ9 53324198 IC50 = 180 nM T34296 C0H7FQ 53324260 IC50 = 6700 nM T34296 CZD9L1 53324788 IC50 = 3800 nM T34296 CU7YG9 53325497 IC50 = 260 nM T34296 C4G1HK 53325498 IC50 = 17000 nM T34296 CO5L1I 53325499 IC50 = 14000 nM T34296 CZA03W 53326760 IC50 = 370 nM T34296 CM53CG 53326761 IC50 = 6100 nM T34296 CWR6T4 53326860 IC50 = 570 nM T34296 C6Y2EV 53374826 IC50 > 100000 nM T34296 CQ04KO 53389286 IC50 = 3 nM T34296 C1IFJ8 53957122 IC50 = 97000 nM T34296 CBL30Y 54181369 IC50 > 10000 nM T34296 CSUW40 54352406 IC50 = 18 nM T34296 C3M8GZ 54580051 IC50 = 46000 nM T34296 CL0WM9 54580052 IC50 > 10000 nM T34296 CK26XF 54580053 IC50 > 10000 nM T34296 CS1LM9 54580054 IC50 = 154 nM T34296 C3LF0P 54580544 Ki = 3.7 nM T34296 CA8U9V 54580837 IC50 = 8 nM T34296 C8PE1G 54581030 IC50 = 570 nM T34296 CVO09J 54581546 Ki = 0.66 nM T34296 CWB2Q6 54581896 IC50 = 1.2 nM T34296 CVK72M 54582073 IC50 = 940 nM T34296 CBK18O 54582074 IC50 > 10000 nM T34296 CP2F1B 54582075 IC50 > 10000 nM T34296 CZNU23 54582076 IC50 > 10000 nM T34296 C0U5HZ 54582077 IC50 > 4100 nM T34296 CSTG96 54582078 IC50 = 1400 nM T34296 C8SG9Y 54582079 IC50 > 10000 nM T34296 CZI6S3 54582080 IC50 = 5900 nM T34296 CD09BZ 54582543 IC50 = 0.7 nM T34296 CH6Q2Z 54583016 IC50 > 10000 nM T34296 C3V9LQ 54583017 IC50 = 260 nM T34296 CT80KQ 54583018 IC50 > 600 nM T34296 CPT4L5 54583019 IC50 = 8400 nM T34296 CK52YD 54583511 Ki = 1.7 nM T34296 CF0SK8 54583712 IC50 = 0.3 nM T34296 CBEV27 54584024 IC50 = 1700 nM T34296 CM87DP 54584025 IC50 = 1100 nM T34296 C28GKQ 54585927 IC50 > 10000 nM T34296 CAZ76E 54586892 IC50 = 4600 nM T34296 CM0OQ3 54586893 IC50 > 10000 nM T34296 CK1NS7 54586894 IC50 > 10000 nM T34296 CMC4Y1 54586895 IC50 > 10000 nM T34296 C2MKX5 54586896 IC50 = 2000 nM T34296 CU91QP 54586897 IC50 > 10000 nM T34296 CI08RQ 54586898 IC50 = 780 nM T34296 C6PRI4 54586899 IC50 > 10000 nM T34296 CG37UX 54587429 Ki = 1.2 nM T34296 CL9SC3 54587769 Ki = 14100 nM T34296 CGH0S7 54589400 IC50 > 100000 nM T34296 C9P5ES 54752445 IC50 = 0.7 nM T34296 C0HKC9 54752446 IC50 = 0.4 nM T34296 CIV16T 56659712 IC50 = 25118.86 nM T34296 C06AWP 56659713 IC50 > 398107.17 nM T34296 CTM86X 56659714 IC50 = 251.19 nM T34296 CFZ48A 56659715 IC50 = 501.19 nM T34296 CC94RE 56663176 IC50 = 3162.28 nM T34296 C5EA4B 56666624 IC50 = 50118.72 nM T34296 CCSY94 56666625 IC50 > 398107.17 nM T34296 C40WKH 56670032 IC50 = 19952.62 nM T34296 C5GOU2 56670033 IC50 = 5011.87 nM T34296 C9MW0X 56670034 IC50 = 125.89 nM T34296 C5FE3V 56673547 IC50 > 398107.17 nM T34296 C4TSJ8 56673548 IC50 = 25118.86 nM T34296 CFLI43 56673549 IC50 > 100000 nM T34296 CADI17 56673550 IC50 > 398107.17 nM T34296 CG0N3B 56673551 IC50 = 398.11 nM T34296 CF98LT 56676871 IC50 = 50118.72 nM T34296 C4EHL2 56676872 IC50 = 316.23 nM T34296 CP98QO 56680187 IC50 = 25118.86 nM T34296 CG8D6A 56680188 IC50 = 63.1 nM T34296 CA8R2T 56680189 IC50 = 2511.89 nM T34296 C62FZC 56835063 IC50 = 1980 nM T34296 CKJ9S1 56835167 IC50 = 9.5 nM T34296 C21CLZ 56835168 IC50 = 52 nM T34296 C0L2TS 56835169 IC50 = 300 nM T34296 CKEV19 56850269 IC50 > 500000 nM T34296 C13DBR 56850270 IC50 > 500000 nM T34296 C05CTJ 56850271 IC50 = 15000 nM T34296 CX8QD5 56850272 IC50 = 82000 nM T34296 C1I9RE 56850407 IC50 = 9600 nM T34296 CVJ90W 56850408 IC50 = 2500 nM T34296 CPI5G0 56850409 IC50 = 2400 nM T34296 CFR3E5 56850410 IC50 > 26000 nM T34296 CRE5O1 56850411 IC50 = 250 nM T34296 CK47BT 56928417 IC50 = 3.5 nM T34296 C8TH2F 56945850 IC50 = 48 nM T34296 CD72TG 56945851 IC50 = 16 nM T34296 C8J4SC 56945854 IC50 = 87 nM T34296 C1AIZ6 56945963 IC50 = 9 nM T34296 CXQC91 56945964 IC50 = 51 nM T34296 CM4H9D 56945965 IC50 = 94 nM T34296 CUT4S2 56946063 IC50 = 605 nM T34296 C2CQR8 56946064 IC50 = 7 nM T34296 C2H8PG 56946065 IC50 = 23 nM T34296 CW2P6A 56946167 IC50 = 21 nM T34296 CT8S3G 56946168 IC50 = 40 nM T34296 C8YID1 56970123 IC50 > 300000 nM T34296 CI5A2O 56970124 IC50 = 5200 nM T34296 CTW18D 56970125 IC50 = 3200 nM T34296 CIK96H 56970340 IC50 = 2600 nM T34296 C1SBD6 56970341 IC50 = 4900 nM T34296 CHA5Q6 56970342 IC50 = 4900 nM T34296 C7A5GT 56970550 IC50 = 5500 nM T34296 C10BMZ 57127110 IC50 > 10000 nM T34296 CQU16V 57339411 Ki = 49 nM T34296 C6LM3B 57339412 Ki = 14 nM T34296 CNVG85 57339413 Ki = 12 nM T34296 C0IU4S 57390230 IC50 = 9.6 nM T34296 CCN3K2 57390233 IC50 = 4300 nM T34296 CJ49DO 57390234 IC50 = 24700 nM T34296 CU34JA 57390237 IC50 = 4000 nM T34296 C9SD5O 57390259 IC50 = 1.4 nM T34296 CI0X9S 57391136 IC50 = 0.6 nM T34296 CD9J1C 57391201 IC50 = 79.43 nM T34296 C6ZAX3 57391202 IC50 = 316.23 nM T34296 C1POE0 57391203 IC50 = 100 nM T34296 CN2H9K 57391204 IC50 = 39.81 nM T34296 CR8MW2 57391205 IC50 = 10 nM T34296 CA25DM 57391224 IC50 = 7 nM T34296 C6P9XK 57391225 IC50 = 18 nM T34296 CJC7M9 57392022 IC50 = 1.1 nM T34296 CAL94F 57392025 IC50 = 2.6 nM T34296 CA6L5W 57392045 IC50 = 2 nM T34296 CH1I4N 57392901 IC50 = 13 nM T34296 C7CV1B 57392902 IC50 = 361 nM T34296 C25FAK 57392903 IC50 = 1.8 nM T34296 C4CK0Q 57392968 IC50 = 79.43 nM T34296 CNQ9B2 57392969 IC50 = 199.53 nM T34296 CU3SG5 57392970 IC50 = 5011.87 nM T34296 C4NYE5 57392971 IC50 = 2511.89 nM T34296 CTYP14 57392972 IC50 = 50.12 nM T34296 C5VB0U 57392973 IC50 = 25.12 nM T34296 CMQL31 57392974 IC50 = 100 nM T34296 C39OHF 57392975 IC50 = 79.43 nM T34296 CX89EL 57392993 IC50 = 32 nM T34296 CB64TD 57393744 IC50 = 5.6 nM T34296 C3CA9G 57393746 IC50 = 0.1 nM T34296 CP5BX6 57394607 IC50 = 3 nM T34296 CA09RY 57394649 IC50 = 10 nM T34296 CDCW73 57394678 IC50 = 220000 nM T34296 CH6BA3 57394709 IC50 = 31.62 nM T34296 CD1CO2 57394710 IC50 = 2511.89 nM T34296 CNOH63 57394711 IC50 = 74 nM T34296 C1CYK9 57394729 IC50 = 15 nM T34296 C9JC3H 57394730 IC50 = 2.2 nM T34296 C80FML 57394731 IC50 = 3.2 nM T34296 CYFJ06 57394732 IC50 = 242 nM T34296 C27AQN 57395458 IC50 = 1.4 nM T34296 C10PRG 57395459 IC50 = 0.7 nM T34296 C42XNM 57395460 IC50 = 4.6 nM T34296 C17DMO 57395461 IC50 = 0.1 nM T34296 CZX7S9 57395466 IC50 = 2.7 nM T34296 CQ4JU6 57395492 IC50 = 12 nM T34296 COXA03 57396390 IC50 = 7 nM T34296 CO17CH 57396398 IC50 = 12 nM T34296 CDES09 57396473 IC50 = 19.95 nM T34296 CONH52 57396474 IC50 = 50.12 nM T34296 CV51ME 57396475 IC50 = 100 nM T34296 C7QD2T 57396476 IC50 = 398.11 nM T34296 CJB27Z 57396489 IC50 = 12 nM T34296 C34RZI 57396490 IC50 = 1 nM T34296 CBY21D 57397314 IC50 = 1.4 nM T34296 CD6Q9F 57398187 IC50 = 180 nM T34296 CSX81J 57398194 IC50 = 165 nM T34296 CBH82N 57398195 IC50 = 0.3 nM T34296 C2INW7 57398264 IC50 > 10000 nM T34296 C0YHM7 57398273 IC50 = 1.3 nM T34296 C5R1PU 57398274 IC50 = 34 nM T34296 CR59KW 57398991 IC50 = 450 nM T34296 C0ZL1D 57399843 IC50 = 100 nM T34296 CI6WB3 57399844 IC50 = 3892 nM T34296 C5SVE2 57399911 IC50 = 316.23 nM T34296 CZ4GX2 57399912 IC50 = 31.62 nM T34296 C4J5LE 57399913 IC50 = 63.1 nM T34296 CH1J9Q 57399914 IC50 = 63.1 nM T34296 CGTF67 57399915 IC50 = 630.96 nM T34296 CI6AZ8 57399916 IC50 = 1584.89 nM T34296 CAKW95 57399917 IC50 > 10000 nM T34296 CD50CO 57399918 IC50 = 50.12 nM T34296 C82HGR 57399936 IC50 = 480 nM T34296 CAX15U 57399937 IC50 = 603 nM T34296 C5U9NO 57400708 IC50 = 1 nM T34296 CBZ36R 57401604 IC50 = 0.05 nM T34296 CM9D3A 57401688 IC50 = 251.19 nM T34296 CF02UP 57401689 IC50 = 12.59 nM T34296 CVO56U 57401690 IC50 = 63.1 nM T34296 CN27EP 57401691 IC50 = 39.81 nM T34296 CJLZ14 57401692 IC50 = 25.12 nM T34296 C2AI8P 57401693 IC50 = 100 nM T34296 CLNT30 57401717 IC50 = 24 nM T34296 CKL68A 57401718 IC50 = 3.6 nM T34296 COP3C5 57402482 IC50 = 7.1 nM T34296 C6HZ1P 57402483 IC50 = 5.2 nM T34296 CGMQ47 57402485 IC50 = 2.2 nM T34296 C37JZN 57402486 IC50 = 1600 nM T34296 CT26AL 57403355 IC50 = 176 nM T34296 C6OQH8 57403420 IC50 = 10 nM T34296 C2Z6EC 57403421 IC50 = 100 nM T34296 CA5Z2V 57403422 IC50 = 50.12 nM T34296 C9O5HA 57403423 IC50 = 1000 nM T34296 CK68EY 57403424 IC50 = 79.43 nM T34296 CQN8L6 57403445 IC50 = 2.2 nM T34296 C2L1SE 57403446 IC50 = 1.3 nM T34296 C2MH8O 57523473 IC50 = 0.09 nM T34296 C57CEM 57523505 IC50 = 1 nM T34296 CS8W4L 57523538 IC50 = 10 nM T34296 CIT7B9 57523539 IC50 = 6 nM T34296 C56QXU 57523540 IC50 = 4 nM T34296 CX8IU3 57523541 IC50 = 18 nM T34296 CE8CL9 57523575 IC50 = 5 nM T34296 CWUP89 57523576 IC50 = 0.006 nM T34296 CT2QS3 57523577 IC50 = 0.02 nM T34296 CK6M0Y 57523578 IC50 = 0.04 nM T34296 C0HVU7 57523611 IC50 = 1 nM T34296 C5Q0ND 57523641 IC50 = 6 nM T34296 CWH7V8 57561293 IC50 = 684 nM T34296 C1PHI6 57708731 IC50 = 0.078 nM T34296 C1MW3I 57708751 IC50 = 0.027 nM T34296 CE27US 57708758 IC50 = 0.026 nM T34296 C2PF5O 57708776 IC50 = 0.043 nM T34296 CF2Z7W 57708783 IC50 = 0.033 nM T34296 C76ABG 57708790 IC50 = 0.1 nM T34296 C9KV2W 57708792 IC50 = 1.5 nM T34296 CE36GP 57708799 IC50 = 0.29 nM T34296 CK6H4D 57708802 IC50 = 0.44 nM T34296 CX5B1P 57708811 IC50 = 0.093 nM T34296 CA3E8P 57708824 IC50 = 0.091 nM T34296 CQ1E7H 57708842 IC50 = 0.059 nM T34296 C23QGY 57708843 IC50 = 4.9 nM T34296 C4NCK5 57708858 IC50 = 0.29 nM T34296 C2J5CW 57708880 IC50 = 2.6 nM T34296 CSO4R8 57708881 IC50 = 0.057 nM T34296 CS25LJ 57708883 IC50 = 0.074 nM T34296 C1K6AP 57708886 IC50 = 0.064 nM T34296 CY1N3J 57792153 IC50 = 1230 nM T34296 CCKD80 58307579 Ki = 28 nM T34296 C1EJ4S 59379730 Ki = 0.59 nM T34296 CK93UZ 59788426 IC50 = 1.3 nM T34296 C8ITK7 59794408 IC50 = 59.1 nM T34296 CSO3W8 59794423 IC50 = 28.9 nM T34296 C6JE9N 59794437 IC50 = 11.5 nM T34296 C7ECU2 59794447 IC50 = 21 nM T34296 C52ESR 66559934 IC50 > 50000 nM T34296 C57ARI 66560021 IC50 > 25000 nM T34296 CU58DB 66560022 IC50 > 25000 nM T34296 C16RDM 66560389 IC50 = 7900 nM T34296 C8RZG9 66560479 IC50 = 7900 nM T34296 C5AQG2 68724898 Ki = 16.6 nM T34296 CC2UE5 68726681 Ki = 0.2 nM T34296 CJU60O 68793626 Ki = 6.3 nM T34296 CMG96N 68794188 Ki = 32.9 nM T34296 C9AL6F 68794211 Ki = 47.2 nM T34296 C7A5PI 68795150 Ki = 21.2 nM T34296 C4IPW3 68795152 Ki = 3.8 nM T34296 CNS46M 68795882 Ki = 29.3 nM T34296 CHL56C 68799256 Ki = 1.4 nM T34296 CT2K3G 70265758 Ki = 2.7 nM T34296 CHRO48 70266605 Ki = 11.7 nM T34296 C34LYX 70266607 Ki = 7.7 nM T34296 COD03W 70267879 Ki = 0.25 nM T34296 CG38ZM 70267887 Ki = 4.5 nM T34296 C3CEL7 70267989 Ki = 23.8 nM T34296 CJHN06 70268164 Ki = 38.5 nM T34296 C50CAL 70268171 Ki = 2.1 nM T34296 CWP71E 70269104 Ki = 16.5 nM T34296 CVWI31 70269555 Ki = 1.2 nM T34296 CGD3B2 70269997 Ki = 5.8 nM T34296 C0GKT8 70685026 IC50 = 3.9 nM T34296 C8B6WD 70688393 IC50 = 18520 nM T34296 CGR3J2 70688394 IC50 = 13170 nM T34296 CFM0Q5 70690777 IC50 = 0.5 nM T34296 CY4E9Z 70692916 IC50 > 100000 nM T34296 C0HE2P 70694634 IC50 = 24490 nM T34296 CI8X5B 71449151 IC50 = 4 nM T34296 CMW3O0 71451330 Ki > 200000 nM T34296 CDZ3P2 71453147 Ki = 28 nM T34296 CKW2Q5 71453375 IC50 = 25000 nM T34296 CX3I5C 71458120 IC50 = 17 nM T34296 C3L7SD 71533484 IC50 = 70 nM T34296 CZH5S9 71533485 IC50 = 134 nM T34296 CGM72Q 71540498 IC50 = 11 nM T34296 CXA1I5 71540599 IC50 = 164 nM T34296 C7CV9E 71540600 IC50 = 23 nM T34296 CA4BP6 71540601 IC50 = 648 nM T34296 CMZ3T2 71540715 IC50 = 155 nM T34296 CXY83G 71540716 IC50 = 44 nM T34296 C1ZH2G 71540717 IC50 = 106 nM T34296 CT4UD5 71540831 IC50 = 104 nM T34296 CP7SX8 71540832 IC50 = 225 nM T34296 C9IW7R 71540833 IC50 = 23 nM T34296 CH5J4A 71602247 IC50 = 22 nM T34296 CH53IU 71602248 IC50 = 386 nM T34296 C97EWQ 71602249 IC50 = 220 nM T34296 CNX9B1 71652215 IC50 = 1.5 nM T34296 C7RZN9 71652216 IC50 = 19 nM T34296 C0NTU7 71652382 IC50 = 0.65 nM T34296 CA5XS1 71652383 IC50 = 62 nM T34296 CYS46I 71652677 IC50 = 4500 nM T34296 CX67VE 71654516 IC50 = 5400 nM T34296 C7DMX5 71680709 Ki = 50 nM T34296 CFPM82 71680710 Ki = 27 nM T34296 C9ZOM7 71680866 Ki = 2 nM T34296 CQ68LT 71680868 Ki > 200000 nM T34296 CV3X1T 71682766 Ki = 200 nM T34296 C5EAO8 71682767 Ki = 160 nM T34296 C80EYX 71682913 Ki = 3400 nM T34296 CIBD03 71682914 Ki = 230 nM T34296 C41BYG 71682915 Ki = 15 nM T34296 C93XEI 71682916 Ki = 10 nM T34296 CQ29PJ 71682917 Ki = 100000 nM T34296 CFWN65 71683062 Ki = 28000 nM T34296 C3L4XU 71718301 IC50 = 12.2 nM T34296 C3E2VT 71814508 IC50 = 1.4 nM T34296 CR2L4T 71814509 IC50 = 1.4 nM T34296 CF21LN 71814684 IC50 = 0.69 nM T34296 C4YM2D 71814685 IC50 = 1.8 nM T34296 CZW1P6 71814686 IC50 = 2.7 nM T34296 C5SI6C 71814687 IC50 = 3.6 nM T34296 CDXZ25 71814688 IC50 = 0.88 nM T34296 CIZ7K1 71814857 IC50 = 1.9 nM T34296 C4W9TJ 71814858 IC50 = 2.9 nM T34296 CJH9K3 71814859 IC50 = 4.7 nM T34296 CCMN52 71814860 IC50 = 5.3 nM T34296 CZ9BC5 71814861 IC50 = 1.6 nM T34296 CU28BE 71815035 IC50 = 0.82 nM T34296 C7HN2J 71815036 IC50 = 3.3 nM T34296 CKV2U5 71817094 Ki = 19 nM T34296 CHDS52 71817095 Ki = 10 nM T34296 C5LZH0 71817097 Ki = 1 nM T34296 C50SID 71817098 Ki = 35 nM T34296 CN83DB 71817100 Ki = 6 nM T34296 CDX2F9 72984326 IC50 = 2.17 nM T34296 CUKG79 73292708 IC50 = 9 nM T34296 C5D3CJ 73292709 IC50 = 1 nM T34296 CL69NM 73292710 IC50 = 1 nM T34296 CQ4RO1 73292711 IC50 = 0.05 nM T34296 C7CT2E 73292869 IC50 = 6 nM T34296 CA0LS6 73292870 IC50 = 0.04 nM T34296 CJU3V6 73292871 IC50 = 0.09 nM T34296 C3PGF2 73292872 IC50 = 1 nM T34296 C0O8VM 73292873 IC50 = 0.3 nM T34296 CBR9I5 73293034 IC50 = 0.1 nM T34296 C9FD2C 73293035 IC50 = 3 nM T34296 C7LP5J 73293036 IC50 = 0.07 nM T34296 C9PQG1 73293037 IC50 = 7 nM T34296 C4PF1H 73293038 IC50 = 0.07 nM T34296 CE39WF 73293196 IC50 = 0.1 nM T34296 CU96XE 73293197 IC50 = 1 nM T34296 CGC51Z 73293198 IC50 = 0.7 nM T34296 CC83FW 73293199 IC50 = 0.6 nM T34296 CS6T8M 73293200 IC50 = 0.3 nM T34296 CW5IQ0 73345859 Ki = 3 nM T34296 CS9AY8 73346035 IC50 = 544.6 nM T34296 CSB01W 73346036 IC50 = 47.3 nM T34296 CCV78D 73346037 IC50 = 14 nM T34296 CUDF74 73347568 IC50 = 31.5 nM T34296 CQ7KG2 73347569 IC50 = 8445 nM T34296 C2B4HW 73349096 IC50 = 1080 nM T34296 CK0TR7 73349097 IC50 = 3.8 nM T34296 C57LGA 73349098 IC50 = 5.1 nM T34296 C25SOB 73349251 IC50 = 0.04 nM T34296 CW01EA 73349535 IC50 > 100000 nM T34296 CFV9Q5 73352169 IC50 = 7329 nM T34296 CA2X8C 73352170 IC50 = 17.7 nM T34296 CXT5V1 73352171 IC50 = 1051 nM T34296 C7Z9MF 73352172 IC50 = 1617 nM T34296 C43WKX 73353429 Ki = 1 nM T34296 CK42DO 73353430 Ki = 5 nM T34296 CNW2C8 73353628 IC50 = 71.2 nM T34296 CYV0L6 73353629 IC50 = 13.8 nM T34296 CG6R7T 73353630 IC50 = 6980 nM T34296 C6H5TU 73354941 Ki = 10 nM T34296 C1HLC9 73355128 IC50 = 2.8 nM T34296 CX8HV9 73355129 IC50 = 178 nM T34296 C06BPT 73355130 IC50 = 18.2 nM T34296 C0K9RX 73355131 IC50 = 53.8 nM T34296 CEHB08 73356503 Ki = 323 nM T34296 C4SXT6 73356696 IC50 = 8.3 nM T34296 CA5T7P 73603957 IC50 = 4200 nM T34296 C8VN1R 74221194 IC50 = 1100 nM T34296 CUB7V9 76329513 IC50 = 0.5 nM T34296 C21FEO 76331549 IC50 = 43 nM T34296 CX39OW 76331563 IC50 = 216 nM T34296 C9CY5K 76335167 IC50 = 127 nM T34296 CKD41G 81689861 IC50 = 1000 nM T34296 CUE7G4 86287514 IC50 = 7000 nM T34296 CGQ8F3 86287515 IC50 = 930 nM T34296 CJ37XE 86287516 IC50 = 2500 nM T34296 COV8I9 86291010 IC50 = 1114 nM T34296 CO2FL5 90137145 IC50 = 320 nM T34296 CRT54C 101910871 IC50 = 30000 nM T34296 C1W5NH 118718816 IC50 = 150 nM T34296 C5ZS4E 118722686 IC50 = 720 nM T34296 CIZB24 118722687 IC50 = 3100 nM T34296 C5C0ZX 118722688 IC50 = 4700 nM T34296 CNF86U 121493953 Ki = 0.008 nM T34296 CJFS09 122190237 IC50 = 1800 nM T34296 CF9C4N 127025165 IC50 = 5.37 nM T34296 CH59PY 127025166 IC50 = 93.8 nM T34296 COGJ69 127025217 Ki = 119 nM T34296 CF45SG 127025218 Ki = 110 nM T34296 CD36QJ 127025222 Ki = 4 nM T34296 CO1DJ9 127027301 IC50 = 2.41 nM T34296 CPG8E6 127027350 Ki = 33.6 nM T34296 CXS26T 127027351 Ki = 14.1 nM T34296 CM7B5S 127029507 IC50 = 1030 nM T34296 C6HA8I 127029508 IC50 > 100000 nM T34296 CPM3N2 127029509 IC50 = 73.1 nM T34296 C3B9EY 127029510 IC50 > 100000 nM T34296 CKNI84 127050262 IC50 = 6 nM T34296 CYA92R 130282633 IC50 = 1300 nM T34296 CO3QE2 130282636 IC50 = 1200 nM T34296 CTN42D 132941363 IC50 = 18000 nM T34296 C83FAY 134130294 Ki = 57.5 nM T34296 C9J7UE 134152374 IC50 = 11 nM T34296 CN9D7G 134155756 IC50 = 0.12 nM T34296 C7K4PA 135412054 IC50 = 920 nM T34296 C31VAN 135412231 Ki = 800 nM T34296 C2VKE8 135414653 IC50 = 16500 nM T34296 CHV2U1 135438561 IC50 = 0.0039 nM T34296 CN30DX 135438809 IC50 = 1600 nM T34296 C4FVJ1 135487604 IC50 = 49600 nM T34296 C8R4FB 135546884 Ki = 1526 nM T34296 C6GR3K 135567051 IC50 = 0.2 nM T34296 C1MOD4 135567320 IC50 = 3.4 nM T34296 CZ0NP3 135924162 IC50 = 36 nM T34296 C2R1MP 135982287 IC50 = 1.7 nM T34296 CFX24R 135982332 IC50 = 16 nM T34296 CWP01Y 135982353 IC50 = 9.4 nM T34296 CR2A9D 135982354 IC50 = 29 nM T34296 CQP35S 135982356 IC50 = 65 nM T34296 CAJ75N 135995993 IC50 = 0.03 nM T34296 CASN17 135995994 IC50 = 0.15 nM T34296 C8EWM3 135995995 IC50 = 0.04 nM T34296 CAO12W 135995996 IC50 = 34 nM T34296 C5BO6Y 135995997 IC50 = 0.99 nM T34296 C6VP7Q 135995998 IC50 = 0.16 nM T34296 CG96KF 135995999 IC50 = 2.9 nM T34296 C5QMP6 135996000 IC50 = 9.7 nM T34296 CYOZ82 135996001 IC50 = 4.3 nM T34296 CI8E5D 135996002 IC50 = 1.6 nM T34296 C5PA8K 135996003 IC50 = 0.52 nM T34296 CATJ83 135996004 IC50 = 0.69 nM T34296 CNJ8H9 135996005 IC50 = 0.31 nM T34296 CW6YS4 135996006 IC50 = 0.53 nM T34296 C1Z8HS 135996007 IC50 = 2.2 nM T34296 C4CB9Z 135996008 IC50 = 8.6 nM T34296 CZWJ74 135996009 IC50 = 25 nM T34296 C1P9QA 135996010 IC50 = 5 nM T34296 C3ZNT0 135996011 IC50 > 10000 nM T34296 CH3J7W 135996012 IC50 = 2200 nM T34296 C7FA3X 135996013 IC50 = 6.3 nM T34296 C2EZ0T 135996014 IC50 = 9.8 nM T34296 CM48OV 135996015 IC50 = 23 nM T34296 CS3Y8H 135996016 IC50 = 1.8 nM T34296 CZ3R8J 135996017 IC50 = 110 nM T34296 CVZC21 135996018 IC50 = 27 nM T34296 C29AGZ 136036767 IC50 >= 100000 nM T34296 CMXL16 136036768 IC50 = 25000 nM T34296 C8WP2X 136036769 IC50 = 55880 nM T34296 CO19FB 136036770 IC50 = 89430 nM T34296 CQS0B6 136036777 IC50 = 55880 nM T34296 CU5IK0 136036779 IC50 = 64000 nM T34296 C49YHB 136036783 IC50 >= 100000 nM T34296 CU54MP 136036786 IC50 = 158 nM T34296 C12UID 136036787 IC50 = 32000 nM T34296 CR9Q6H 136054467 IC50 = 1.6 nM T34296 CYH23I 136054468 IC50 = 0.59 nM T34296 CZ8DW1 136054472 IC50 = 0.38 nM T34296 C9H0DL 136054473 IC50 = 1.7 nM T34296 CX7MI0 136054475 IC50 = 0.3 nM T34296 CA5JR6 136054481 IC50 = 0.24 nM T34296 CO2VU9 136054484 IC50 = 0.36 nM T34296 CV47JN 136054485 IC50 = 0.11 nM T34296 CZ48WO 136054487 IC50 = 0.071 nM T34296 CR9CY5 136054490 IC50 = 0.26 nM T34296 C8FGT0 136054495 IC50 = 0.23 nM T34296 CGH39U 136054498 IC50 = 0.19 nM T34296 C2TO7Y 136054508 IC50 = 1.5 nM T34296 CG70BZ 136054516 IC50 = 0.051 nM T34296 CSM57W 136054520 IC50 = 0.052 nM T34296 CXNG40 136118011 Ki > 5025 nM T34296 C1IOH9 136118012 Ki = 4314 nM T34296 CIEW62 136380958 IC50 = 0.17 nM T34296 CHOA14 136814721 IC50 = 26910 nM T34296 CFJ3I6 136814723 IC50 >= 100000 nM T34296 C9HS7J 137287436 IC50 = 0.0032 nM T34296 C4N8VM 137348731 IC50 = 356 nM T34296 CLE8B1 137348732 IC50 = 9.4 nM T34296 C7FQ6W 137348733 IC50 = 2.2 nM T34296 CAZ87R 137631621 IC50 = 35 nM T34296 CQ3GZ0 137632187 Ki = 36 nM T34296 C0I6RH 137632487 IC50 = 1.9 nM T34296 C4KQR9 137635016 Ki = 1.6 nM T34296 C0R5ZT 137635841 IC50 = 32 nM T34296 CU5G8I 137636679 IC50 = 86 nM T34296 C4UMY5 137636781 IC50 = 159 nM T34296 C1RID9 137636861 IC50 = 175 nM T34296 CNM8J4 137638970 IC50 = 5.495 nM T34296 C7Y0FB 137642170 IC50 = 111 nM T34296 CR8H9Z 137644167 IC50 = 4.4 nM T34296 CDOQ29 137644394 IC50 = 36.31 nM T34296 C0Y5JA 137644464 IC50 = 1.6 nM T34296 CB8M6U 137646865 Ki = 1.7 nM T34296 C04KVQ 137647395 IC50 = 14 nM T34296 CK4LE6 137647628 IC50 = 17.9 nM T34296 CHI2E1 137648744 IC50 = 11.75 nM T34296 CXV6J5 137648746 Ki = 0.47 nM T34296 C1U2QR 137651063 IC50 = 25 nM T34296 C9CIY6 137651719 IC50 = 0.3 nM T34296 CZ51XB 137651858 Ki = 24.5 nM T34296 CS80YI 137652598 IC50 = 340 nM T34296 C5Y8RP 137654086 IC50 = 258 nM T34296 CKH37T 137657100 Ki = 190 nM T34296 CZB75K 137657128 IC50 = 16.9 nM T34296 CRD46H 137658344 IC50 = 58 nM T34296 C3ER5O 137658673 IC50 = 128 nM T34296 CEQ8I9 137659945 IC50 = 89 nM T34296 CC3I9B 137660260 Ki = 9.2 nM T34296 CHO70T 137660954 IC50 = 149 nM T34296 C4H0EM 137661370 IC50 = 257 nM T34296 CZ8H6N 137661550 IC50 = 16000 nM T34296 C1IF6L 137661809 IC50 = 20.89 nM T34296 C1Q2BP 145949247 IC50 > 5000 nM T34296 C6TD4M 145949288 IC50 = 2600 nM T34296 CN9RD6 145949408 IC50 = 1200 nM T34296 C5FWA2 145949488 IC50 = 2.5 nM T34296 CZS1N7 145949693 IC50 = 1.9 nM T34296 CYG32L 145950058 IC50 > 5000 nM T34296 CU53BP 145950331 IC50 = 2.5 nM T34296 CY8C4A 145950332 IC50 = 7.8 nM T34296 CAJ25P 145951291 IC50 = 38 nM T34296 C3EF7N 145952515 IC50 = 5.5 nM T34296 CW1GS2 145952760 IC50 = 18.7 nM T34296 CFN1R7 145952843 IC50 = 7.3 nM T34296 CM6T2O 145953417 IC50 = 1300 nM T34296 C6FYK8 145953609 IC50 > 5000 nM T34296 CV80WQ 145954107 IC50 = 9.4 nM T34296 C16VNH 145954604 IC50 = 12.9 nM T34296 CQF50V 145954863 IC50 = 2.4 nM T34296 C8QW9G 145955776 IC50 = 13 nM T34296 CH0ZO5 145955778 IC50 = 14.4 nM T34296 CFDZ62 145955866 IC50 = 2000 nM T34296 CVZ5U7 145955868 IC50 = 6.9 nM T34296 C8TPR1 145956198 IC50 = 43.2 nM T34296 CR8U7Y 145956318 IC50 = 4.4 nM T34296 C4S8LU 145956764 IC50 = 153 nM T34296 CUS0Y9 145957234 IC50 = 9.1 nM T34296 CUO69Q 145957392 IC50 = 88 nM T34296 CX94UK 145957493 IC50 = 289 nM T34296 C6MHN7 145957508 IC50 = 20 nM T34296 C5K7PV 145958060 IC50 = 1.6 nM T34296 CBE02W 145958354 IC50 = 5.1 nM T34296 CQL4O0 145959327 IC50 = 8.5 nM T34296 CUAT97 145960347 IC50 = 18 nM T34296 CZ76WA 145962290 IC50 > 5000 nM T34296 C27MTZ 145962695 IC50 = 148 nM T34296 CRY63E 145963538 IC50 = 6.4 nM T34296 CVCL61 145963739 IC50 = 8.4 nM T34296 C72NJI 145968012 IC50 = 403 nM T34296 CRK13Q 145969600 IC50 = 51 nM T34296 C1FPG2 145972660 IC50 = 6.4 nM T34296 CN73DF 145972870 IC50 = 69 nM T34296 C3F0AD 145973196 IC50 > 2000 nM T34296 CJF73O 145973630 IC50 = 7.1 nM T34296 CX7M9L 145976456 IC50 = 697 nM T34296 CPD1B0 145977213 IC50 = 7.1 nM T34296 C9Z5DX 145978402 IC50 = 274 nM T34296 CZ25LW 155512044 IC50 = 23000 nM T34296 CV10AF 155512426 IC50 = 11 nM T34296 CFHU79 155514943 IC50 = 57 nM T34296 CF64GH 155518335 Ki = 562 nM T34296 CL16UE 155520835 IC50 = 5000 nM T34296 C59YHT 155522902 IC50 = 636 nM T34296 CC5FA9 155529859 IC50 = 4320 nM T34296 CQUA53 155531128 IC50 = 939 nM T34296 C7TP3R 155531151 IC50 > 10000 nM T34296 CJN8X5 155542058 Ki = 1.6 nM T34296 CWEG57 155545190 IC50 = 0.7 nM T34296 C1FP0M 155548067 IC50 = 39 nM T34296 C9AOK6 155550135 IC50 > 10000 nM T34296 C3BA9L 155561798 IC50 = 0.07 nM T34296 CP9YX2 155567218 IC50 = 3400 nM T34296 C8D5VK 155567855 IC50 = 2300 nM T34296 C5U9LI 155569346 IC50 = 280 nM T34296 CLT4Y6 10138589 Ki = 260 nM T34296 C5U3AO 57394286 IC50 = 645 nM T34296 D00KSS 18411961 IC50 = 50 nM T34296 D01OCR 19366856 IC50 = 4 nM T34296 D01UNE 44580457 Ki = 15.7 nM T34296 D02ECA 448942 IC50 = 270 nM T34296 D02EFQ 10549609 IC50 = 16 nM T34296 D02PKO 44294636 IC50 = 500 nM T34296 D03AMR 9849669 Ki = 10 nM T34296 D03FEI 15516781 IC50 = 45 nM T34296 D03SNK 644601 IC50 = 280 nM T34296 D04GOO 10111838 IC50 = 1350 nM T34296 D04UBY 45483018 IC50 = 52000 nM T34296 D04VPH 45376872 IC50 = 4 nM T34296 D05PZV 796420 IC50 = 1700 nM T34296 D05THD 44478925 IC50 = 1400 nM T34296 D07DRT 46175162 Ki = 1.7 nM T34296 D07GEL 10344307 Ki = 0.45 nM T34296 D07MJD 44479701 IC50 = 260 nM T34296 D08ELY 9838786 IC50 = 22 nM T34296 D09GLA 4368 IC50 = 7.943 nM T34296 D09XUQ 19366844 IC50 = 6 nM T34296 D09ZOA 25049753 Ki = 2 nM T34296 D0A0FY 44479457 IC50 = 28000 nM T34296 D0A4TC 446504 Ki = 1.27 nM T34296 D0B3UN 44580458 Ki = 49 nM T34296 D0C1EQ 20348772 IC50 = 95200 nM T34296 D0D7UA 10267279 IC50 = 0.5 nM T34296 D0F4UT 21496278 IC50 = 95900 nM T34296 D0G3YZ 11391583 IC50 = 12000 nM T34296 D0H2PA 9886977 Ki = 0.5 nM T34296 D0H6CK 10160968 Ki > 5025 nM T34296 D0I0WP 649391 IC50 = 13300 nM T34296 D0K0YX 44626352 IC50 = 2450 nM T34296 D0K3RC 44294677 IC50 = 1 nM T34296 D0L6ND 10089677 IC50 = 0.47 ug.mL-1 T34296 D0LB0N 45483008 IC50 > 98000 nM T34296 D0LL8I 9830392 IC50 = 17 nM T34296 D0LM2K 45483015 IC50 = 11300 nM T34296 D0N0FX 19366816 IC50 = 22 nM T34296 D0N6CD 10565532 IC50 = 100 nM T34296 D0NP8A 10370504 IC50 = 73 nM T34296 D0Q4TA 10044321 Ki = 20 nM T34296 D0R5MR 15052873 IC50 = 400 nM T34296 D0S9OL 10155934 IC50 = 2700 nM T34296 D0T1FR 44457233 IC50 > 100000 nM T34296 D0TL3N 45482998 IC50 > 98000 nM T34296 D0V9GS 651854 IC50 = 1300 nM T34296 D0W2UK 6914621 Ki = 1417 nM T34296 D0XE4B 15516780 IC50 = 32 nM T34296 D0XK7G 10445302 Ki = 8 nM T34296 D0Y5IQ 44255320 IC50 = 5000 nM T34296 D0Z7EF 2777 IC50 = 10000 nM T78709 D01AZG 5073 Ki = 21 nM T78709 D01FFA 72301 Ki > 5000 nM T78709 D01ZII 2726 Ki = 673 nM T78709 D03SKR 2803 Ki = 3235.94 nM T78709 D03WEX 9966051 Ki = 9.5 nM T78709 D04JCN 47811 Ki = 1.8 nM T78709 D04JEE 4946 IC50 = 3981.07 nM T78709 D05MBZ 129211 Ki = 0.79 nM T78709 D05XGO 11154555 Ki = 2.6 nM T78709 D05ZIK 4205 Ki > 18 nM T78709 D06FPQ 77992 Ki = 62 nM T78709 D06OSM 91273 Ki = 5.8 nM T78709 D06YFA 31101 Ki = 24 nM T78709 D09IOI 2170 Ki = 221 nM T78709 D0B3UJ 115237 EC50 > 10000 nM T78709 D0CQ0Z 33630 Ki = 356 nM T78709 D0D1AL 3559 IC50 = 1500 nM T78709 D0F2PO 4828 Ki = 22.4 nM T78709 D0G8NN 119570 Ki = 6514 nM T78709 D0H3HM 60795 Ki = 1.7 nM T78709 D0H6QU 6005 Ki = 296 nM T78709 D0H7KF 5002 Ki = 79.43 nM T78709 D0K0KH 656665 Ki = 5.3 nM T78709 D0K0MW 30668 Ki = 125.89 nM T78709 D0K0VO 5639 Ki = 213 nM T78709 D0K8KX 5280343 EC50 > 100000 nM T78709 D0NG7O 60857 Ki = 78.6 nM T78709 D0P0OU 11978813 Ki = 0.12 nM T78709 D0R1JV 60854 Ki = 1.585 nM T78709 D0R6RO 4184 IC50 = 398.11 nM T78709 D0R9EQ 5095 Ki = 1706 nM T78709 D0S9CB 6918248 EC50 = 630.96 nM T78709 D0S9MU 5078 Ki = 140 nM T78709 D0T3KI 4440 Ki = 45 nM T78709 D0T6QX 5736 Ki = 330 nM T78709 D0U2OO 2477 Ki = 3.1 nM T78709 D0UA0I 28693 Ki = 2.3 nM T78709 D0V4QS 135398745 Ki = 610 nM T78709 D0W5HK 216239 Ki = 1181 nM T78709 D0WV3U 4893 Ki > 10 nM T78709 D0X6BV 6918314 EC50 = 0.12 nM T78709 D0X7KB 28864 Ki = 0.4 nM T78709 D0Z1RV 135398737 Ki = 6.38 nM T78709 D0Z6UC 5358 Ki = 230 nM T78709 D01GEB 219050 IC50 = 0.8 nM T78709 D07YVK 9818479 Ki = 73 nM T78709 D09GHO 5311258 Ki = 22 nM T78709 D09IRN 21071390 Ki = 3936 nM T78709 D0F8HS 11741361 EC50 = 389.05 nM T78709 D0HZ2E 5311271 Ki > 10000 nM T78709 D0L3JI 188942 Ki = 180 nM T78709 D0LI1C 44469321 IC50 > 10000 nM T78709 D0N1HW 5311200 Ki = 6620.9 nM T78709 D0P2QO 132787 Ki = 0.7943 nM T78709 D0R9HI 11256720 Ki = 2370 nM T78709 D0T8KA 11151899 Ki = 6.5 nM T78709 D0W5EH 6918388 IC50 < 6 nM T78709 D0X2XF 177336 Ki < 10000 nM T78709 D0Y2GJ 44182694 Ki = 5.05 nM T78709 D0R1PZ 10248159 EC50 = 10 nM T78709 D00OWF 5280953 Ki > 10000 nM T78709 D00KZF 2419 Ki = 0.3715 nM T78709 D01DAW 208951 Ki = 9.3 nM T78709 D01RAE 133079 Ki > 1600 nM T78709 D01VAB 2119 Ki = 21.6 nM T78709 D01WJZ 60820 Ki = 1.7 nM T78709 D02FNU 56971 Ki = 6 nM T78709 D02JMI 9888211 Ki = 2.512 nM T78709 D02VUX 11697676 Ki = 3.7 nM T78709 D02VZP 57347 EC50 = 6.607 nM T78709 D03ITI 183092 Ki = 92 nM T78709 D03QMR 5685 Ki = 2.089 nM T78709 D03TNA 5025739 Ki > 10000 nM T78709 D03ZZH 9887537 Ki = 0.7943 nM T78709 D06DZI 107780 Ki = 70 nM T78709 D07BCO 5684 Ki = 0.1585 nM T78709 D08AWI 11430856 Ki = 5.1 nM T78709 D09WHM 208917 Ki = 1.5 nM T78709 D0B7SP 11292933 Ki = 0.3981 nM T78709 D0EE6L 3038495 Ki = 81 nM T78709 D0G1RT 132059 IC50 = 3.162 nM T78709 D0G5ZL 132792 Ki = 1.9 nM T78709 D0K9JP 9928332 Ki = 2 nM T78709 D0L9SN 4431 Ki = 0.6 nM T78709 D0M7LV 5761 Ki = 1.1 nM T78709 D0O9EM 208928 Ki = 175 nM T78709 D0OS6O 60149 Ki = 33 nM T78709 D0P9FT 148842 Ki = 5.9 nM T78709 D0Q2JS 10436045 Ki = 100 nM T78709 D0R5GS 55191 Ki = 13 nM T78709 D0T1SF 9909448 Ki = 1092 nM T78709 D0Y0RW 66004 IC50 = 5.012 nM T78709 D0YP7L 6604889 Ki < 5 nM T78709 D0Z7AW 9820261 Ki = 180 nM T78709 C5JG6U 2689 IC50 = 46.77 nM T78709 CZUI83 2769 Ki = 794.33 nM T78709 C0H8GR 3191 IC50 = 47 nM T78709 C0OCW6 6240 Ki = 673 nM T78709 C3H5DF 7172 Ki = 63000 nM T78709 C5H9CN 9287 Ki = 3162.28 nM T78709 COD41I 17371 Ki = 256 nM T78709 CVD75F 20810 Ki = 1.3 nM T78709 C9E6DA 21171 Ki > 5000 nM T78709 CFGH18 27620 Ki = 12 nM T78709 C6WDL7 49756 Ki = 200 nM T78709 CPW9B5 65752 Ki > 100000 nM T78709 C06GWQ 72340 EC50 > 100000 nM T78709 CJV28G 90285 IC50 = 2.4 nM T78709 C10XRB 99652 Ki = 32000 nM T78709 CN9GK1 104911 Ki = 0.31 nM T78709 CI24CD 120540 Ki = 43.2 nM T78709 CBS9J2 124433 Ki = 3.58 nM T78709 CI47KZ 127708 Ki = 66 nM T78709 C9WG8X 131559 Ki = 24.8 nM T78709 C4PR2E 132564 IC50 = 8410 nM T78709 CC58NU 132955 Ki = 58 nM T78709 CY0O6P 151779 Ki = 831.76 nM T78709 C4VCM7 156372 Ki = 36000 nM T78709 CI80NA 160436 Ki = 10 nM T78709 CGT8R0 160510 Ki > 1670 nM T78709 C1ND9W 161665 Ki = 149 nM T78709 CK8RD5 168114 Ki = 11710 nM T78709 CJ34CF 168115 Ki = 3740 nM T78709 CLK7P3 169713 IC50 = 3 nM T78709 C3O4NA 179651 Ki > 100000 nM T78709 CZ0D8W 180707 Ki = 2290.87 nM T78709 CA91IX 185559 EC50 > 100000 nM T78709 COPZ85 188006 Ki = 20 nM T78709 C7ASC5 195252 Ki = 19 nM T78709 CQA75X 210165 IC50 = 15 nM T78709 CHLI84 210172 Ki = 1.738 nM T78709 CDA06R 211216 Ki = 181.97 nM T78709 CF72KY 211936 Ki = 1737.8 nM T78709 CJ8XZ3 211938 Ki = 50.12 nM T78709 CVI6X5 213046 Ki = 6.7 nM T78709 C5T7DJ 363353 Ki = 17.5 nM T78709 C2V5FA 398712 Ki = 1 nM T78709 CYV1R3 417052 Ki > 10000 nM T78709 CF7ZS4 417608 Ki = 1.7 nM T78709 C4O6RK 435595 Ki = 830 nM T78709 CFJ3R2 452533 Ki = 90 nM T78709 C0IH9E 688095 Ki = 110 nM T78709 CXQ6U0 735755 IC50 = 7600 nM T78709 C2VLP8 752521 Ki = 660 nM T78709 C5S3MB 785789 Ki > 1000 nM T78709 C1TV2F 1070749 IC50 > 1000 nM T78709 CJ30IQ 1248739 Ki = 3600 nM T78709 C9FI5L 1296368 Ki = 23740 nM T78709 C6VZT7 1984087 Ki = 4900 nM T78709 CGS9R7 2133793 Ki = 13490 nM T78709 CG9N3A 2136365 Ki = 4592 nM T78709 CA2OY6 2737389 Ki = 99 nM T78709 CE50LO 2756712 Ki = 72.1 nM T78709 C1C4LH 2843443 Ki = 26360 nM T78709 C1S8CM 2845719 IC50 > 100 nM T78709 CRA6F5 2853434 Ki = 10330 nM T78709 C3QRD6 2867758 Ki = 31400 nM T78709 CL2G3H 2870750 Ki = 21610 nM T78709 CC74QS 2872937 Ki = 20600 nM T78709 CRF65H 2880253 Ki = 41800 nM T78709 CET7C8 2921525 Ki = 15600 nM T78709 C2DE6R 2927683 Ki = 7100 nM T78709 CF01YE 2928642 Ki = 9100 nM T78709 CY8R6Q 2948971 Ki = 2450 nM T78709 CLXQ01 2950739 Ki = 6100 nM T78709 CO0C7J 2962174 Ki = 284100 nM T78709 CRQ30L 3025767 Ki = 11 nM T78709 CGMD76 3037048 EC50 = 2000 nM T78709 CB5Q2J 3037448 EC50 > 100000 nM T78709 C64CZV 3038494 Ki = 81 nM T78709 CVD51K 3039995 IC50 = 71 nM T78709 C6Z4QI 3050372 Ki = 25 nM T78709 C5NA6S 3069135 Ki = 24 nM T78709 C4X3VL 3073440 Ki = 16 nM T78709 CKB30E 3073449 Ki = 2.099 nM T78709 CAT54M 3074872 Ki = 25 nM T78709 C6SA2G 3132842 Ki = 36800 nM T78709 C82GMT 3246443 Ki = 908 nM T78709 CS8KE2 3649661 Ki = 714 nM T78709 CRUB15 4723431 Ki = 125 nM T78709 C7PX9E 4790508 Ki = 8 nM T78709 CW2C1I 5009938 Ki = 833 nM T78709 C9NKP1 5216959 Ki = 36 nM T78709 CG3Y4K 5221957 IC50 = 2700 nM T78709 C4BKS2 5242341 Ki = 5.3 nM T78709 CY67TC 5281073 Ki = 17 nM T78709 CLNI10 5281408 EC50 = 10300 nM T78709 CH50QK 5281643 Ki > 100000 nM T78709 CZM7D8 5281794 Ki = 18020 nM T78709 CRD82S 5318644 Ki > 100000 nM T78709 C4J3HP 5640104 Ki = 18490 nM T78709 CW34VC 6160690 Ki = 1.3 nM T78709 CCY85T 6442560 Ki = 13050 nM T78709 CFYP06 6442612 Ki = 5840 nM T78709 CWNZ35 6469693 Ki = 2200 nM T78709 CJTQ40 6469918 Ki = 1700 nM T78709 C5K4PX 6603808 Ki = 40.74 nM T78709 CXZ53N 6603866 Ki = 0.1 nM T78709 CP2QM5 6604000 Ki = 151 nM T78709 CR48ZF 6604840 IC50 = 16.9 nM T78709 CC6SM3 6618861 Ki = 354 nM T78709 C0QCK1 6918455 Ki = 398.11 nM T78709 CW0ZE5 6918542 Ki = 702 nM T78709 CC5PQ0 6918601 Ki > 5600 nM T78709 C1WXY3 6918603 Ki = 1000 nM T78709 CD0Z4I 6918648 Ki = 501.19 nM T78709 CX59ZP 6971167 Ki > 100000 nM T78709 C2F3BY 7125890 Ki = 13700 nM T78709 C2PL6S 8019695 IC50 = 9400 nM T78709 C6D0MA 8554729 Ki = 706 nM T78709 CUD06Z 9796627 Ki = 620 nM T78709 C57XYF 9798593 Ki = 0.69 nM T78709 CPG3J9 9798864 Ki = 35.1 nM T78709 CBG80E 9799121 Ki = 90.42 nM T78709 CFC9Y5 9799318 Ki = 512.86 nM T78709 CNE17Q 9799764 Ki = 23.9 nM T78709 CKM1U6 9800010 Ki = 0.2 nM T78709 CJ8SL4 9800133 Ki = 22.4 nM T78709 CSN81W 9801669 Ki = 18.9 nM T78709 CTUX42 9802369 EC50 = 2.138 nM T78709 CCV0M4 9802530 Ki = 40 nM T78709 C2VS1K 9802999 Ki > 1000 nM T78709 CE0DI5 9804612 Ki = 3.981 nM T78709 CNX4F0 9805456 Ki = 1000 nM T78709 CPZ05H 9805881 Ki = 61 nM T78709 CR8ET5 9814387 Ki = 44 nM T78709 CWOS30 9817810 Ki = 140 nM T78709 CX7N8J 9817881 IC50 = 12.59 nM T78709 CHQI10 9818448 Ki = 139 nM T78709 C8S6FJ 9819892 Ki = 1.622 nM T78709 C45QPU 9820163 Ki = 10.9 nM T78709 CS6KM1 9820536 Ki = 170 nM T78709 C1ZM6Q 9821397 IC50 = 2 nM T78709 CD30SC 9821838 Ki = 1.08 nM T78709 CZMK41 9822025 Ki = 5.012 nM T78709 CAX8D6 9822317 EC50 = 1.5 nM T78709 C2U3EZ 9822477 Ki = 69.55 nM T78709 CL2MG5 9822705 Ki = 91.86 nM T78709 CA2D7V 9822812 Ki > 1000 nM T78709 CF0J1A 9822814 Ki = 17.43 nM T78709 C6JN8C 9822942 Ki = 104.1 nM T78709 C5DB6G 9823115 Ki = 29.64 nM T78709 CL38GM 9826580 Ki = 23.4 nM T78709 CPXI10 9826761 Ki = 290 nM T78709 C0AU9L 9826801 Ki = 130 nM T78709 CLU54H 9827354 Ki = 273 nM T78709 CWS18C 9832057 Ki = 17.7 nM T78709 C2MN0P 9837094 Ki > 3521 nM T78709 C6I4QG 9841032 IC50 = 2951.21 nM T78709 C36NME 9842337 Ki = 71.6 nM T78709 C1LOQ2 9842682 Ki = 43.9 nM T78709 C53UPQ 9842861 Ki = 43.65 nM T78709 CXJ7Z3 9844300 Ki = 139.9 nM T78709 C8TE4O 9844321 Ki = 12.07 nM T78709 CFV1I3 9844747 Ki = 2.9 nM T78709 C96YOX 9844821 Ki = 22.2 nM T78709 C4YIM0 9845172 Ki = 248.19 nM T78709 C57TYA 9845202 Ki = 3.5 nM T78709 C5H7TG 9846057 Ki = 549.54 nM T78709 C5MHS3 9847013 Ki = 160 nM T78709 CNB65K 9848303 Ki = 29 nM T78709 CDOG70 9848876 Ki = 236 nM T78709 CYMP40 9851789 IC50 = 1.83 nM T78709 CM13ZV 9856041 EC50 > 10000 nM T78709 C7EZ2L 9859861 Ki > 1000 nM T78709 CZY34F 9860739 Ki = 1.33 nM T78709 C0ZR3E 9861687 IC50 > 100000 nM T78709 CNCK78 9862256 Ki = 170 nM T78709 CC0SQ3 9862968 Ki = 16.8 nM T78709 C8M5XK 9863333 Ki = 899 nM T78709 C6ERH9 9863540 Ki > 3000 nM T78709 CS7EY1 9863750 EC50 = 33.88 nM T78709 CKF2T8 9864325 Ki = 7.5 nM T78709 CTY02P 9865254 Ki = 55 nM T78709 CX3CQ2 9865576 Ki = 75.77 nM T78709 C5WYN4 9865858 Ki = 3.6 nM T78709 C0NV4T 9866094 Ki = 3.981 nM T78709 CHM4D6 9866320 Ki = 3.02 nM T78709 C1SOI8 9867138 Ki = 432.7 nM T78709 CB1F0C 9867475 Ki = 480 nM T78709 C57YPX 9867902 IC50 = 41 nM T78709 C2WB5T 9868306 Ki = 3.12 nM T78709 C8EG1K 9868735 Ki = 1.5 nM T78709 CDFP50 9868793 Ki = 3 nM T78709 C3GMU5 9868889 Ki = 0.2 nM T78709 C7AB8O 9870053 Ki < 3981.07 nM T78709 CHP5L7 9870809 Ki = 12.36 nM T78709 CK76MQ 9872238 Ki = 0.7 nM T78709 CS12TL 9873467 Ki = 18.7 nM T78709 CBF9T3 9879532 Ki = 69 nM T78709 C35LIA 9881324 EC50 = 35 nM T78709 C9NF3D 9881600 Ki = 16 nM T78709 C8L6GE 9882257 Ki > 1000 nM T78709 CY5HZ0 9882594 Ki = 345 nM T78709 C3DB5H 9884781 Ki = 540 nM T78709 CTAC24 9885114 Ki = 792 nM T78709 CW76OG 9885700 Ki = 0.7 nM T78709 COW86S 9886269 Ki = 19.95 nM T78709 CFW03P 9887458 Ki = 134.84 nM T78709 CJW1P5 9888494 Ki = 478.63 nM T78709 C9GB2M 9888555 Ki = 41 nM T78709 C6N8UE 9889681 Ki = 630.96 nM T78709 C1ANB8 9889726 Ki = 122.3 nM T78709 CM52WU 9890119 Ki = 158.49 nM T78709 C2R3PF 9890484 Ki = 214.1 nM T78709 CEG1K5 9891002 Ki = 251.19 nM T78709 C7QMK5 9891617 Ki = 794.33 nM T78709 CEL29O 9891618 Ki = 794.33 nM T78709 C6WY0D 9891901 Ki = 2040 nM T78709 C3J8GU 9892409 Ki = 630.96 nM T78709 CAY78Q 9892644 Ki = 62.22 nM T78709 CAM25C 9894665 Ki = 15 nM T78709 CFM67S 9897637 Ki = 1.66 nM T78709 C9J6KN 9901423 Ki = 4000 nM T78709 CFI97S 9904205 IC50 = 977.24 nM T78709 CUN81Q 9905249 Ki > 10000 nM T78709 CZ32BY 9906183 Ki = 0.54 nM T78709 CYWQ50 9906447 Ki = 432 nM T78709 C25XRA 9906677 Ki > 1000 nM T78709 C7JFZ5 9906978 Ki = 722.3 nM T78709 CWV8K4 9908283 Ki = 52.31 nM T78709 CY2I0L 9908478 Ki = 25 nM T78709 CA4B5Q 9908855 Ki = 5.3 nM T78709 CYZ5N4 9909089 Ki = 0.0631 nM T78709 CWD2G3 9909389 Ki = 0.33 nM T78709 CA0U4Y 9909471 Ki > 1000 nM T78709 CG80QK 9909555 Ki = 76.14 nM T78709 CO7BK6 9909648 Ki = 134 nM T78709 C3BR6W 9910451 Ki = 160 nM T78709 CUX71M 9910468 Ki = 2.9 nM T78709 C4L2CV 9911120 IC50 = 10.72 nM T78709 C9B3EA 9911844 Ki = 316 nM T78709 C78MDV 9913554 Ki = 125.89 nM T78709 CQ3YN1 9927016 IC50 = 12.59 nM T78709 C4UYZ7 9927441 Ki = 520 nM T78709 CY5L0E 9928161 Ki = 804.8 nM T78709 CID4Y2 9928432 Ki = 1.6 nM T78709 CJ6CF2 9928474 Ki = 920 nM T78709 CCX3F8 9929277 Ki = 258.1 nM T78709 CQX4W1 9929572 Ki = 78.3 nM T78709 C7SOT8 9929936 Ki = 275.44 nM T78709 C1C5KY 9931327 Ki = 360 nM T78709 CN3OW2 9932051 Ki = 0.91 nM T78709 CPB27K 9932697 EC50 = 135 nM T78709 C3L5MF 9932835 Ki = 127.84 nM T78709 CN6YW2 9933342 Ki = 0.8 nM T78709 C5V0UE 9933975 Ki = 0.7 nM T78709 C4L1GA 9934033 IC50 = 16.9 nM T78709 CYVZ47 9934284 Ki = 0.3981 nM T78709 CWO45F 9935387 Ki = 199.53 nM T78709 CYH3R7 9947817 Ki = 1000 nM T78709 C63EWV 9950390 Ki = 870 nM T78709 CXUC75 9950482 Ki = 1.6 nM T78709 CP5MQ0 9950538 EC50 = 26 nM T78709 CX6QW8 9952481 Ki = 154.85 nM T78709 C5W6RU 9953959 Ki = 136.45 nM T78709 C4G9VQ 9954092 Ki = 36 nM T78709 CK8NR2 9954121 Ki = 794.33 nM T78709 CU2C3V 9955072 Ki = 0.5 nM T78709 C9QPM4 9955522 Ki = 0.631 nM T78709 CSK1B2 9955819 Ki = 49.5 nM T78709 CHOJ30 9956365 Ki = 128.82 nM T78709 CFR41N 9957068 Ki = 3162.28 nM T78709 CZ9SC7 9957274 Ki = 1.259 nM T78709 CGO64P 9957376 Ki = 3.162 nM T78709 CBK3P7 9958160 Ki = 803.57 nM T78709 C2RU8Q 9966169 Ki = 1100 nM T78709 C9CT0V 9970622 Ki = 81 nM T78709 CR5XJ2 9975609 Ki = 21.6 nM T78709 CCZP34 9976750 IC50 = 5.012 nM T78709 C7JXL1 9976756 Ki = 3.548 nM T78709 C2XG1I 9977716 Ki = 3.162 nM T78709 CFN50J 9978683 Ki > 5000 nM T78709 CPX92V 9979309 Ki = 0.07943 nM T78709 CC6M7Z 9980998 Ki = 27.9 nM T78709 C09GVK 9981322 Ki = 0.75 nM T78709 C2PDI5 9982036 Ki = 2.799 nM T78709 CDG74Q 9983460 Ki = 40.3 nM T78709 CCR0T4 9984109 Ki = 20 nM T78709 CU2EB0 9991334 Ki = 152 nM T78709 CI1OT4 9991554 Ki = 49 nM T78709 CS1DG5 9992098 Ki = 66 nM T78709 CO9EM6 9992630 Ki > 1000 nM T78709 CK54BS 9992778 Ki = 33.9 nM T78709 CF0R6B 9995045 IC50 = 50.12 nM T78709 C3NHU1 9996500 Ki = 2.4 nM T78709 CWQ1K3 9999722 Ki = 10.4 nM T78709 C8A6EZ 10001971 Ki = 0.1259 nM T78709 CVWG72 10003116 Ki = 50.7 nM T78709 CHJ7C0 10003814 Ki = 24 nM T78709 CQL12P 10004545 Ki > 2000 nM T78709 CP54MB 10005122 Ki = 13 nM T78709 C4IG8L 10005161 EC50 = 2.512 nM T78709 CJ4SF5 10005953 Ki = 141 nM T78709 CV4T9U 10008868 Ki = 9.8 nM T78709 CM26VE 10014056 Ki = 54 nM T78709 CO39AR 10014057 Ki = 56 nM T78709 CUX43N 10014136 Ki = 0.1 nM T78709 CG8YK7 10014674 Ki = 1000 nM T78709 CYWH12 10014964 Ki = 5.4 nM T78709 C5MUC9 10015045 Ki = 49 nM T78709 CB32PO 10015338 Ki = 1.5 nM T78709 C3X4BD 10015438 Ki > 1000 nM T78709 C9A2SX 10015574 Ki = 0.12 nM T78709 CS40QN 10015688 Ki = 8.7 nM T78709 CF6OB5 10017429 Ki = 105 nM T78709 CV7R9F 10020040 Ki > 10000 nM T78709 C6XGV2 10020855 Ki = 0.028 nM T78709 CK18LT 10020895 Ki = 56 nM T78709 CQHW51 10023176 Ki = 100 nM T78709 CH6OC0 10024324 Ki = 3.7 nM T78709 CYB6X2 10024776 EC50 = 69.18 nM T78709 CM7W9G 10024936 Ki = 2.512 nM T78709 CR7Y9C 10025854 EC50 = 7.079 nM T78709 CNP9D7 10035788 Ki = 29 nM T78709 CM0Z7A 10036887 Ki > 470 nM T78709 CPXC69 10037436 Ki = 16 nM T78709 C2E1HD 10037437 Ki = 11 nM T78709 C6DT5M 10037522 Ki = 186 nM T78709 CWN9F2 10038106 Ki > 1000 nM T78709 C1IQ5D 10038966 Ki = 9.3 nM T78709 C2C1XS 10042602 Ki = 83.18 nM T78709 CA42DO 10047196 Ki = 9.2 nM T78709 C25WVJ 10047566 IC50 > 1000 nM T78709 C6EDO4 10047814 EC50 = 1.349 nM T78709 C4S0HI 10047915 Ki = 5.2 nM T78709 C2JZL1 10048222 Ki = 8.9 nM T78709 C2UI7F 10048252 Ki > 1000 nM T78709 CF84QJ 10048342 Ki = 0.5012 nM T78709 C8JLO2 10048343 Ki = 0.631 nM T78709 CBF02H 10048892 Ki = 0.247 nM T78709 C3MT0Y 10049499 Ki = 9.9 nM T78709 C4GHO2 10053476 Ki = 125 nM T78709 CFXB93 10059206 Ki = 92 nM T78709 C7CRY4 10059274 Ki = 31 nM T78709 C8KRW5 10059714 Ki = 5.9 nM T78709 C8FT2B 10059787 Ki = 3 nM T78709 C2G9HJ 10060349 Ki > 333 nM T78709 CB96PM 10061032 Ki = 10 nM T78709 CP9A6Q 10061694 IC50 = 63.1 nM T78709 CDA93R 10062435 IC50 = 199.53 nM T78709 C0KWB6 10062885 Ki = 17.3 nM T78709 CJ67EH 10062998 Ki > 1000 nM T78709 CFM51X 10063283 IC50 = 501.19 nM T78709 CUW74G 10064052 Ki = 1420 nM T78709 CR68SH 10064053 Ki = 1.8 nM T78709 C4PCO3 10065083 Ki = 30.5 nM T78709 C0I2RV 10065903 Ki = 3.715 nM T78709 CD0J3I 10067360 EC50 = 2.884 nM T78709 CIC0W2 10068815 Ki = 8.3 nM T78709 C2EG0W 10068933 Ki > 1000 nM T78709 C6HP2C 10069977 Ki = 13.6 nM T78709 C9KWT3 10071738 Ki = 0.3162 nM T78709 CJ50UM 10071897 Ki = 35.97 nM T78709 CT1U0X 10072874 Ki = 426 nM T78709 CV6R2F 10073139 Ki = 0.631 nM T78709 CN9B1F 10074286 Ki = 10.2 nM T78709 CVE2T1 10076176 IC50 = 100 nM T78709 CQ1YA4 10076876 Ki = 6.8 nM T78709 CJ92BN 10082834 Ki = 0.23 nM T78709 CWC26Y 10084026 Ki = 11 nM T78709 CKA5F4 10084076 Ki = 355 nM T78709 CJ16VZ 10084583 Ki = 2500 nM T78709 CD2RM6 10085260 Ki = 960 nM T78709 CQVJ58 10088453 Ki = 79.43 nM T78709 C6BDZ3 10089203 Ki = 460 nM T78709 C6KY5X 10090661 Ki = 29.2 nM T78709 C0IWD7 10091187 Ki = 0.21 nM T78709 C3XY4N 10091300 Ki = 1.023 nM T78709 CW9PL1 10091417 EC50 = 5.248 nM T78709 CR3D5E 10091430 IC50 = 6.31 nM T78709 CJXQ40 10092819 Ki = 17 nM T78709 C7BD6F 10093232 Ki = 39 nM T78709 CR17PA 10093856 Ki = 9.7 nM T78709 C9OXA7 10095692 Ki = 181.97 nM T78709 CLW53J 10097792 Ki = 741.31 nM T78709 CH5WC1 10105311 Ki = 36 nM T78709 C0XO1J 10105844 Ki = 0.2 nM T78709 CB4W8T 10105889 IC50 = 140 nM T78709 CJF84M 10105934 Ki = 1000 nM T78709 C5D2UI 10106412 IC50 = 25.12 nM T78709 C54EYD 10108561 IC50 < 1000 nM T78709 CKU06X 10108730 IC50 = 316.23 nM T78709 CC15UG 10111229 Ki = 83.3 nM T78709 C8CUX9 10112935 Ki = 2.692 nM T78709 CBW28F 10113692 Ki = 58.3 nM T78709 C2ISY6 10114480 Ki = 0.3981 nM T78709 C9PG3D 10115847 Ki = 39.81 nM T78709 CJZX05 10115848 Ki = 1.585 nM T78709 COWN03 10116877 Ki = 1.6 nM T78709 CP1CL5 10127149 Ki = 31.62 nM T78709 CLFA47 10127209 Ki < 10000 nM T78709 CKYQ52 10127424 Ki = 3.981 nM T78709 CRJ8M9 10127673 Ki = 15.85 nM T78709 C4SN0A 10127877 Ki = 2.512 nM T78709 C9J6KH 10128059 Ki = 125.89 nM T78709 CBT24S 10130700 Ki = 400 nM T78709 C8ZJ9G 10131066 Ki = 28 nM T78709 CW0E4F 10137577 Ki = 90 nM T78709 CWMT35 10138727 Ki = 0.7943 nM T78709 C4X9RB 10150658 Ki < 1258.93 nM T78709 CKGC73 10150796 Ki = 158.49 nM T78709 C6FEY0 10151426 Ki = 364 nM T78709 CJI9T7 10151492 Ki = 31.62 nM T78709 C4Q3UL 10154897 Ki > 100 nM T78709 CFL76R 10158326 Ki = 14.3 nM T78709 C3YK0R 10158884 Ki = 5.4 nM T78709 CSPG27 10159927 Ki = 1.585 nM T78709 C9JLX2 10161027 Ki = 19.95 nM T78709 CVA6N0 10161028 Ki = 0.5012 nM T78709 CQEB83 10163855 EC50 > 100000 nM T78709 C5E4SQ 10172853 Ki = 12.59 nM T78709 C3YT8A 10173169 Ki = 398.11 nM T78709 CJRV76 10173263 Ki = 25.12 nM T78709 CMP89S 10173443 Ki = 10 nM T78709 CT0CX5 10174078 Ki = 1.995 nM T78709 CQXI36 10174088 Ki = 2.512 nM T78709 C34ROH 10174199 Ki = 2.512 nM T78709 CG01HR 10178015 Ki = 111.2 nM T78709 CWK76Q 10179327 Ki = 549.54 nM T78709 C4W0PV 10180988 Ki = 6.026 nM T78709 C0NPG1 10180998 Ki = 6.5 nM T78709 COE73R 10183387 Ki = 819.8 nM T78709 CEDP29 10183895 Ki = 0.631 nM T78709 C6NA5G 10194297 Ki = 1000 nM T78709 CI76JU 10194809 Ki = 25.12 nM T78709 CLHY30 10194820 Ki = 251.19 nM T78709 CW1CM3 10195275 Ki = 1 nM T78709 CECA82 10203092 Ki = 1.585 nM T78709 C21MHR 10203336 Ki = 11.3 nM T78709 CE3S6M 10216160 Ki = 398.11 nM T78709 CRW49L 10216744 Ki = 63.1 nM T78709 C80QXD 10216873 Ki = 6.31 nM T78709 C1HF5Y 10222267 Ki = 295 nM T78709 C8LTG3 10223717 Ki = 1.259 nM T78709 C84CPM 10224961 Ki = 2.9 nM T78709 CO57AW 10226822 Ki = 694.2 nM T78709 CF4N1M 10237964 Ki = 1.995 nM T78709 C0Q2ZD 10238160 Ki = 79.43 nM T78709 CIR98N 10238565 Ki = 3.981 nM T78709 CK39BA 10238566 Ki = 2.512 nM T78709 C3L0WD 10238762 Ki = 19.95 nM T78709 CI9KH6 10238763 Ki = 7.943 nM T78709 CAC29B 10243514 IC50 > 1000 nM T78709 CL1K4S 10243702 Ki > 1000 nM T78709 CXD7O8 10244325 Ki = 1.8 nM T78709 CVF1E5 10246054 IC50 > 1000 nM T78709 CSE47M 10247171 IC50 = 5888.44 nM T78709 CG2B7I 10247701 Ki = 125.89 nM T78709 CFCP96 10247720 Ki = 45 nM T78709 C0NT8I 10248163 Ki = 0.31 nM T78709 C4Q2SH 10249573 Ki = 1000 nM T78709 CMA42P 10250834 Ki = 130 nM T78709 CD83JK 10251722 Ki = 390 nM T78709 CUSP67 10252256 IC50 = 17 nM T78709 C4FZ9V 10253106 Ki = 18 nM T78709 C2JDW3 10253939 Ki = 15.9 nM T78709 C4NYW7 10254142 Ki = 22 nM T78709 CX67OE 10254537 Ki = 12.8 nM T78709 CMRA02 10257042 Ki = 7943.28 nM T78709 CZW62U 10262307 Ki = 1000 nM T78709 CG71CB 10263220 Ki > 1000 nM T78709 CXB7U8 10264456 Ki = 721 nM T78709 CI5Z0M 10264555 Ki > 1000 nM T78709 CVT34Y 10264556 Ki > 1000 nM T78709 CC8PX4 10265905 IC50 = 630.96 nM T78709 C10YRB 10266873 Ki = 6.3 nM T78709 CH31DX 10267394 Ki = 2759.7 nM T78709 CR2J1V 10271949 Ki = 83.6 nM T78709 CB95IA 10272536 Ki = 37.15 nM T78709 CC56OL 10272986 Ki = 168.2 nM T78709 C0MVZ1 10273133 Ki = 13 nM T78709 CVC87R 10275633 Ki = 5.012 nM T78709 CL8DY9 10275767 Ki = 563.5 nM T78709 CE9Y8J 10276451 Ki = 198 nM T78709 CQ8N3F 10288132 Ki = 7.943 nM T78709 CWS2U4 10295406 Ki = 4.62 nM T78709 C8XKC0 10310103 Ki = 67 nM T78709 C3G8KJ 10310285 Ki = 5.012 nM T78709 C0WRV9 10310423 Ki = 5.012 nM T78709 CU89JD 10314060 Ki = 405.6 nM T78709 CA3E4W 10316297 Ki = 38.9 nM T78709 CHYJ47 10317514 Ki = 0.79 nM T78709 C5VC9X 10317939 Ki = 13.44 nM T78709 CUT3Y2 10318597 Ki = 24 nM T78709 C0OJ2C 10319235 Ki = 0.5012 nM T78709 CU12DB 10319570 IC50 = 2 nM T78709 CPH30X 10319737 Ki = 0.7943 nM T78709 CCXJ27 10321497 Ki = 42.6 nM T78709 C30CBI 10324625 Ki = 10.2 nM T78709 C3DB1Q 10332122 Ki = 0.5 nM T78709 CMFL49 10332127 Ki = 0.2 nM T78709 CP35VD 10332803 Ki = 19 nM T78709 CFL49K 10333305 IC50 = 125.89 nM T78709 C83GBY 10333405 Ki = 6.1 nM T78709 CE6IP1 10333670 Ki = 178 nM T78709 CRQN68 10333842 Ki = 45 nM T78709 CUY3O1 10340117 Ki = 7.8 nM T78709 CM10QP 10340549 Ki = 607 nM T78709 CXG6B1 10341129 Ki = 0.3981 nM T78709 C4ZI1X 10343002 Ki = 40 nM T78709 C5MH7Y 10343434 Ki = 6.8 nM T78709 C3ZN0F 10344705 Ki = 68.9 nM T78709 CIP38T 10344976 Ki < 1000 nM T78709 CV92JN 10345799 EC50 > 100000 nM T78709 C9IAV3 10346043 Ki > 3162.28 nM T78709 CI17PT 10348924 Ki = 2.2 nM T78709 CH6C8N 10353170 Ki = 11 nM T78709 CS24DU 10353268 IC50 = 287 nM T78709 CXO0J4 10353777 Ki = 4.9 nM T78709 COT48Q 10353846 Ki = 338 nM T78709 CJ6WS4 10354101 Ki = 84.5 nM T78709 C7DQA1 10354437 Ki = 4.7 nM T78709 CUYR47 10355219 Ki = 11 nM T78709 CK7E9M 10355252 Ki = 62.3 nM T78709 C4-DEC 10355779 IC50 = 199.53 nM T78709 CJO3F2 10355844 Ki = 15 nM T78709 CD4H6R 10361512 Ki = 4500 nM T78709 CA4R1B 10362715 Ki = 26.6 nM T78709 COC7M0 10363912 Ki = 0.6026 nM T78709 C72PTA 10364325 EC50 = 229.09 nM T78709 C8GR5I 10364994 Ki = 0.06761 nM T78709 CW41CF 10365352 IC50 = 12 nM T78709 CV0Y5B 10365638 Ki = 39 nM T78709 CR53YS 10365683 Ki = 77.8 nM T78709 C9QBP3 10367560 Ki = 78 nM T78709 CP43QS 10367835 Ki = 10.4 nM T78709 C6ZV2B 10368048 Ki = 7.8 nM T78709 C9LWG3 10369004 IC50 = 38 nM T78709 CD9PZ8 10369020 Ki = 47 nM T78709 CW7MQ0 10376578 Ki = 6.1 nM T78709 CPD3A2 10377136 Ki = 104 nM T78709 C2OWC5 10377224 Ki = 17 nM T78709 CFVW98 10377225 IC50 > 1000 nM T78709 CKMQ51 10377779 Ki = 66 nM T78709 CMJ0B7 10377872 Ki = 1 nM T78709 CIX51R 10378194 Ki = 270 nM T78709 CFT3C8 10378503 Ki = 9.4 nM T78709 CBI62Z 10378937 Ki = 9530 nM T78709 CUV0T8 10379049 IC50 = 316.23 nM T78709 CXQJ16 10379099 IC50 = 316.23 nM T78709 C5LPM8 10379100 IC50 = 316.23 nM T78709 CA7IM5 10379532 Ki = 16.9 nM T78709 CE1XW6 10380005 IC50 = 50.12 nM T78709 CDAC63 10381889 IC50 = 199.53 nM T78709 CMZA83 10383646 Ki > 5000 nM T78709 C69KIB 10385855 Ki = 7.7 nM T78709 CY59KH 10386049 Ki = 0.2884 nM T78709 C0XG9M 10387420 Ki = 0.2512 nM T78709 C8UI9F 10389173 Ki = 1.34 nM T78709 CG1IR6 10394346 Ki = 1.2 nM T78709 C64HBT 10398936 Ki > 470 nM T78709 C3RO4M 10398940 Ki = 174 nM T78709 C0D8HN 10399013 Ki = 4.8 nM T78709 C3LJV4 10400362 Ki = 384 nM T78709 CFEL74 10400539 Ki = 5 nM T78709 C2T0CR 10400849 IC50 = 158.49 nM T78709 CXU73R 10401626 IC50 = 501.19 nM T78709 CVQ9E8 10401691 IC50 = 316.23 nM T78709 CFM13B 10401705 Ki = 8.5 nM T78709 C4L5PQ 10404657 Ki = 499 nM T78709 CHW3Q9 10405775 EC50 = 6.026 nM T78709 CNV6P7 10406539 IC50 = 60 nM T78709 CX72MW 10407711 Ki = 5011.87 nM T78709 CDIZ70 10407753 Ki = 54.59 nM T78709 CU7V2W 10408477 IC50 = 20 nM T78709 CMBW49 10408880 Ki = 15 nM T78709 C8S3XE 10409556 IC50 = 0.1288 nM T78709 CY3O5W 10410577 Ki = 30.55 nM T78709 C01QDW 10411236 EC50 = 1.995 nM T78709 CSH4O3 10411600 Ki = 41.98 nM T78709 C4QJ8U 10412550 Ki = 56 nM T78709 C4TPN1 10413595 Ki = 501.19 nM T78709 CC4QS3 10420841 Ki = 37 nM T78709 C2B0IU 10421236 Ki = 684 nM T78709 C0HM5D 10421583 Ki = 80 nM T78709 CWD56M 10421850 IC50 = 63.1 nM T78709 CYB2Q9 10422079 Ki = 2 nM T78709 C13LGV 10422091 Ki = 2.9 nM T78709 C70IZX 10423337 Ki = 2.9 nM T78709 CR2D4Z 10424079 Ki = 642 nM T78709 CTG0F9 10429067 Ki = 347 nM T78709 CV49RW 10430183 EC50 = 0.78 nM T78709 CR4LS0 10430623 Ki = 573 nM T78709 CD7U5I 10433930 Ki = 3981.07 nM T78709 CK9QE0 10433973 Ki = 30.97 nM T78709 CCP0S9 10434440 Ki = 2.47 nM T78709 CDU91R 10434550 Ki = 257 nM T78709 CPK38Z 10435294 Ki = 46 nM T78709 C4UN0A 10436653 Ki = 69 nM T78709 C8KD1B 10438027 Ki = 130 nM T78709 CSM96F 10443274 Ki = 44 nM T78709 C0Z7FW 10444472 Ki = 145 nM T78709 CBM3X0 10444473 Ki = 69 nM T78709 CMEA74 10445202 Ki = 29 nM T78709 CQ1V2Z 10445845 IC50 = 158.49 nM T78709 CD1FO8 10445902 Ki = 4.1 nM T78709 CBAY90 10445946 Ki = 620 nM T78709 C7VOJ3 10445991 Ki = 15 nM T78709 C9-AUG 10446088 Ki > 1000 nM T78709 C5N8HO 10447116 Ki = 127 nM T78709 CF25ZL 10449555 Ki > 1000 nM T78709 C9WA5Q 10452875 Ki = 1.585 nM T78709 C94TVH 10452995 IC50 = 41686.94 nM T78709 C9YZI1 10453264 EC50 = 7943.28 nM T78709 CFK16Y 10454806 Ki = 0.2512 nM T78709 CYMS64 10454807 Ki = 1.259 nM T78709 C62WSQ 10456474 Ki = 15.1 nM T78709 C10NHR 10457710 Ki = 10 nM T78709 C8V6ZQ 10458087 Ki = 95 nM T78709 CQ4T7G 10458088 Ki = 5.1 nM T78709 CGS4E2 10466294 Ki > 1000 nM T78709 CP17RZ 10466368 Ki = 16 nM T78709 C1YS3M 10466454 Ki = 1000 nM T78709 CK3Q9O 10466960 Ki = 1 nM T78709 CL6FY4 10466962 Ki = 236 nM T78709 C3EH5D 10468253 IC50 = 63.1 nM T78709 COV85C 10472143 Ki = 0.45 nM T78709 C7GEB0 10474042 Ki = 0.08 nM T78709 CUFL05 10474089 EC50 = 2.818 nM T78709 CPI5M7 10476504 Ki = 24 nM T78709 CL63TF 10477223 Ki = 2.512 nM T78709 C8JCZ1 10477386 Ki = 24 nM T78709 CWY2J3 10478217 Ki = 3.981 nM T78709 CEF2O6 10478367 Ki = 641 nM T78709 CE0CF3 10479090 Ki = 100 nM T78709 CI6PN3 10495891 Ki = 19.1 nM T78709 CFQ8U6 10496827 Ki = 19.05 nM T78709 C0QR2H 10496957 IC50 > 100000 nM T78709 C3IY9P 10498554 IC50 = 50118.72 nM T78709 CQ9A2N 10498633 Ki = 1550 nM T78709 C4XWG7 10499348 IC50 = 0.2 nM T78709 C4IXZ5 10500422 Ki = 633 nM T78709 C6TQV3 10501785 IC50 = 0.8 nM T78709 CQE8U0 10502452 IC50 > 100000 nM T78709 CVO4H1 10503335 EC50 = 269.15 nM T78709 C1FV7A 10516340 IC50 = 117.49 nM T78709 CCPO93 10518850 Ki = 18 nM T78709 CTP65K 10519608 IC50 = 2290.87 nM T78709 CWH7R8 10521887 Ki = 90.33 nM T78709 C8WR5O 10522029 IC50 = 0.7 nM T78709 C7M0YQ 10523090 IC50 > 100000 nM T78709 C90TWP 10524876 IC50 = 0.2 nM T78709 CM0BI4 10525991 Ki = 363.08 nM T78709 CNE54K 10526362 IC50 = 389045.14 nM T78709 CDNJ39 10528303 EC50 = 162.18 nM T78709 C8NT2G 10528899 Ki = 5011.87 nM T78709 C5KOM9 10529394 Ki = 1000 nM T78709 C0ZM5P 10531639 Ki = 4 nM T78709 CI67OK 10535587 Ki > 3257 nM T78709 CYKP58 10539093 IC50 = 64565.42 nM T78709 C3N5MZ 10544888 Ki = 2754.23 nM T78709 C48BRW 10546334 Ki = 125.89 nM T78709 CFN8B5 10546440 IC50 = 5370.32 nM T78709 CFC5Z3 10546879 Ki = 109.65 nM T78709 CJ2T5R 10547091 IC50 = 0.3 nM T78709 CTLF72 10547809 IC50 = 102329.3 nM T78709 C1LV7P 10548259 IC50 = 10964.78 nM T78709 C32XGO 10549236 EC50 = 10 nM T78709 C4S7NI 10549573 Ki = 384.59 nM T78709 CJ30TE 10550097 EC50 = 20.42 nM T78709 C3P5VL 10550893 EC50 = 14 nM T78709 COF60K 10550911 EC50 = 8.318 nM T78709 CE59TG 10553922 IC50 > 100000 nM T78709 CYCT15 10562462 Ki = 40.7 nM T78709 CHOZ29 10567450 Ki = 575 nM T78709 C5JY4K 10568666 IC50 > 100000 nM T78709 CW6VX8 10568745 IC50 = 6165.95 nM T78709 CART26 10569395 IC50 = 4570.88 nM T78709 C7N1FY 10569470 IC50 = 257.04 nM T78709 CY37OI 10570263 Ki = 323.59 nM T78709 CQJ29H 10570535 Ki = 12.02 nM T78709 C5YH2I 10571274 Ki = 554 nM T78709 C9GSI8 10571450 IC50 = 12882.5 nM T78709 CN1UG2 10572945 Ki = 501.19 nM T78709 CY05PE 10573164 IC50 = 12589.25 nM T78709 CU63GA 10573576 IC50 = 0.8 nM T78709 CHE80N 10573876 Ki = 398.11 nM T78709 CBZP14 10574764 Ki = 89.13 nM T78709 CZ0IY9 10575934 EC50 = 5.754 nM T78709 CZC23D 10576554 EC50 = 309.03 nM T78709 C61SEA 10576618 IC50 = 17782.79 nM T78709 CM9N5S 10585117 Ki = 120 nM T78709 C69LZJ 10590206 IC50 = 120.23 nM T78709 C0DX7G 10590360 IC50 = 93.33 nM T78709 CCBU34 10590370 Ki = 2300 nM T78709 CV9LP1 10592579 Ki = 794.33 nM T78709 C7EN0K 10593348 Ki = 48.8 nM T78709 C5G1OF 10594234 Ki = 6.7 nM T78709 C9PKO0 10595710 Ki = 416.87 nM T78709 CBT12J 10596337 Ki = 5011.87 nM T78709 CO23YX 10597140 Ki = 1584.89 nM T78709 CW3TN5 10598044 IC50 = 31622.78 nM T78709 C85LBE 10600032 EC50 = 39.81 nM T78709 CO24RV 10600444 Ki = 446.68 nM T78709 CF74VT 10601619 Ki = 13.4 nM T78709 C49WAM 10610641 Ki = 14.4 nM T78709 CVYB63 10613373 Ki = 48 nM T78709 COB4F8 10616442 Ki = 15.85 nM T78709 C76HPC 10616443 Ki = 10 nM T78709 C42HFS 10616657 Ki > 1000 nM T78709 C2G4IR 10617200 Ki = 5.495 nM T78709 CRY9Q0 10617292 IC50 = 2570.4 nM T78709 C8GFT6 10618751 Ki = 27 nM T78709 C7KD2F 10619048 Ki = 18.2 nM T78709 C39FNQ 10619583 IC50 = 89125.09 nM T78709 C86KEZ 10620679 IC50 = 40738.03 nM T78709 CX3A0P 10620719 Ki = 967 nM T78709 CIV3M9 10621014 Ki = 501.19 nM T78709 CQH1X3 10621131 IC50 = 288.4 nM T78709 CD8KX9 10621491 Ki > 3356 nM T78709 CMV72H 10622257 IC50 = 25703.96 nM T78709 CFR74L 10623260 Ki = 19.95 nM T78709 CTA56W 10623356 Ki = 0.791 nM T78709 C6PXH9 10623459 Ki = 549.54 nM T78709 CUH0N7 10623740 Ki = 5011.87 nM T78709 CHO45W 10624365 Ki = 5011.87 nM T78709 CL8K0J 10624420 Ki = 257.04 nM T78709 CEWL87 10624604 Ki = 17.22 nM T78709 C0DZC5 10624695 Ki = 32.81 nM T78709 C01MLV 10637485 IC50 = 117.49 nM T78709 CAPO49 10638372 Ki > 1000 nM T78709 C1MYD5 10640199 Ki = 885 nM T78709 CQ1NJ0 10640504 Ki = 707.95 nM T78709 CER8L0 10640982 Ki = 0.8318 nM T78709 C2FH3S 10643939 Ki > 1000 nM T78709 C1A6ZO 10644514 IC50 = 3 nM T78709 C9XE8T 10645076 IC50 = 3000 nM T78709 CCS31Z 10645335 IC50 = 61659.5 nM T78709 CQD6R2 10645615 IC50 = 660.69 nM T78709 C8HO3D 10646854 Ki = 1584.89 nM T78709 CN5I9Q 10646934 EC50 = 30.9 nM T78709 CU50HJ 10647006 EC50 = 3.467 nM T78709 C6PBY1 10647387 Ki = 1 nM T78709 CPMS86 10647621 EC50 = 14.79 nM T78709 C5KNR9 10647622 EC50 = 2.754 nM T78709 CCA14X 10648046 Ki = 5011.87 nM T78709 CYDV92 10649124 Ki = 14.1 nM T78709 CH3V2L 10661560 Ki = 50.12 nM T78709 CQM6J9 10662302 Ki = 204 nM T78709 C07AKO 10663820 IC50 > 100000 nM T78709 CEVO29 10664203 Ki = 63 nM T78709 C87GYV 10664657 Ki = 199.53 nM T78709 C5W6PY 10665156 Ki = 9.3 nM T78709 CZN9V7 10665419 IC50 = 15488.17 nM T78709 C4PV2W 10666301 IC50 = 6760.83 nM T78709 CB3C9Z 10667071 IC50 = 40738.03 nM T78709 CH37WD 10669519 Ki = 501.19 nM T78709 CNFI24 10670050 EC50 = 6.607 nM T78709 C4D0QG 10671211 IC50 = 2 nM T78709 C4NOI8 10672566 Ki = 42.85 nM T78709 C0U6ZS 10672840 Ki = 114 nM T78709 CBC8N5 10674136 Ki = 5011.87 nM T78709 CC24YZ 10686563 Ki = 794.33 nM T78709 CCZ41N 10687440 Ki = 5011.87 nM T78709 CTS4A1 10687868 IC50 = 33884.42 nM T78709 CBEP65 10688604 Ki = 22.39 nM T78709 CTXW74 10688951 Ki = 33.88 nM T78709 CP45QK 10689339 IC50 = 43651.58 nM T78709 C26GSJ 10689888 Ki = 1000 nM T78709 C4I3YM 10690445 Ki = 50.12 nM T78709 C6YXC1 10691383 IC50 = 11 nM T78709 C5FQ9T 10691904 Ki = 23 nM T78709 C2LU1H 10692095 Ki > 3356 nM T78709 C48BQX 10692498 Ki = 851.14 nM T78709 C8SU4D 10692801 EC50 = 407.38 nM T78709 C0BOG6 10694238 EC50 = 33.11 nM T78709 CZLP81 10694239 EC50 = 3.715 nM T78709 CS35LF 10694660 EC50 = 0.7244 nM T78709 C4LM2C 10695395 EC50 = 8.913 nM T78709 CRB2A1 10695466 EC50 = 28.84 nM T78709 CV7D8G 10696202 Ki = 591.56 nM T78709 C9GR4O 10696705 Ki = 60.26 nM T78709 CM31PB 10696930 Ki = 8.6 nM T78709 CS4JW5 10698929 Ki > 10000 nM T78709 CSB3G8 10704251 Ki = 114 nM T78709 CLZ9F5 10706553 Ki = 31.1 nM T78709 CBE87R 10706626 Ki = 142 nM T78709 C61RTM 10709212 Ki = 371.54 nM T78709 CE7DB9 10710400 Ki = 800 nM T78709 C6M0GA 10711251 Ki = 5011.87 nM T78709 C7C9EY 10712619 Ki = 89.13 nM T78709 C9FAP1 10714457 IC50 = 11481.54 nM T78709 CIBU90 10714509 IC50 = 97723.72 nM T78709 CPW52V 10714712 Ki = 5011.87 nM T78709 CU32PG 10714877 Ki = 19.22 nM T78709 CVS29F 10715484 IC50 = 56234.13 nM T78709 CGO34D 10715991 Ki = 100 nM T78709 CX8K5B 10717072 IC50 = 1 nM T78709 C5NQX4 10717512 IC50 = 72.44 nM T78709 C4TV6C 10718220 EC50 = 12.3 nM T78709 CWV5A9 10718277 IC50 = 0.6 nM T78709 C0USP7 10718592 Ki = 3.4 nM T78709 CVK2T3 10718731 IC50 = 204173.79 nM T78709 CP7CE8 10718870 EC50 = 2.63 nM T78709 CI3V8M 10719425 EC50 = 12.02 nM T78709 CM7N9Q 10719857 IC50 = 7762.47 nM T78709 CUS3R0 10720301 Ki = 9.5 nM T78709 CZH1M4 10735345 Ki = 50.12 nM T78709 CZXG16 10735489 Ki = 199.53 nM T78709 CI0GE8 10737848 IC50 = 407.38 nM T78709 CQV9O7 10738182 Ki = 251.19 nM T78709 C1QJ2F 10738317 Ki > 1430 nM T78709 CY1M6L 10738329 IC50 > 100000 nM T78709 C1Y3KQ 10738599 Ki = 5011.87 nM T78709 C1ZH6B 10739272 IC50 = 1047.13 nM T78709 C7YXW0 10740939 EC50 = 3.631 nM T78709 C6SA9J 10742699 EC50 = 28.18 nM T78709 C96VMI 10743303 EC50 = 22.91 nM T78709 C8YQE1 10743835 Ki = 167.88 nM T78709 CX3FL8 10751317 Ki = 88 nM T78709 CZO1E3 10753377 IC50 = 64.57 nM T78709 C17OFU 10756517 IC50 = 67.61 nM T78709 C62VKE 10758083 Ki = 185 nM T78709 CPQ40M 10759541 IC50 = 3 nM T78709 C3TD1I 10762475 Ki = 173.78 nM T78709 CLJ74B 10764513 EC50 = 5.754 nM T78709 CQB52R 10765698 EC50 = 5.248 nM T78709 CWSA98 10777682 IC50 = 32359.37 nM T78709 C1RG2E 10780842 Ki = 716 nM T78709 C9PB7H 10782548 Ki = 794.33 nM T78709 CZJO64 10782681 Ki = 575 nM T78709 CQ12RP 10783275 Ki = 5011.87 nM T78709 CX70KH 10786335 Ki > 1000 nM T78709 CB7V4A 10787178 Ki = 3630.78 nM T78709 CN98JS 10787547 EC50 = 21.88 nM T78709 C6ISL1 10788207 IC50 = 0.7 nM T78709 C5H1DA 10789000 IC50 = 43 nM T78709 C8Y3OP 10789182 EC50 = 2.951 nM T78709 C2QBM4 10789419 EC50 = 3.02 nM T78709 C1XKJ8 10789756 EC50 = 10.72 nM T78709 COJ20B 10790813 IC50 > 100000 nM T78709 C8Y3TP 10791125 Ki = 117 nM T78709 CNUF06 10791244 Ki = 9.5 nM T78709 CK9O3B 10802304 Ki = 38 nM T78709 C5XKN1 10805222 Ki = 144.54 nM T78709 CZ7J1S 10805599 Ki = 1.84 nM T78709 CWA5J0 10807321 Ki = 139 nM T78709 C83RTC 10807421 Ki = 17.38 nM T78709 C2TDU4 10808641 Ki = 190.55 nM T78709 C8S4PF 10808909 IC50 = 14454.4 nM T78709 CPS68R 10809227 Ki = 10 nM T78709 CL12BA 10809238 IC50 = 40 nM T78709 C4K3SY 10809561 IC50 = 125892.54 nM T78709 CXY1Q0 10809674 Ki = 14.3 nM T78709 C5J4ND 10809876 IC50 = 0.2 nM T78709 CQN8A4 10811876 IC50 = 1348.96 nM T78709 CL0W3S 10812183 EC50 = 13.18 nM T78709 CQX1G6 10813526 Ki = 54.95 nM T78709 CE16DJ 10813865 EC50 = 5.012 nM T78709 C8QGX9 10813901 EC50 = 1.122 nM T78709 CCWH19 10814515 IC50 > 100000 nM T78709 CUI27T 10825325 Ki = 5.05 nM T78709 CT1I7H 10826076 IC50 = 52.48 nM T78709 CHMB58 10827788 Ki = 120.23 nM T78709 CF4KZ1 10827876 Ki = 154.88 nM T78709 CW2LK3 10828231 Ki = 1180 nM T78709 CVA26N 10830318 Ki = 114.82 nM T78709 CJ1D6P 10830587 Ki = 5011.87 nM T78709 CEW6J2 10831102 Ki = 5011.87 nM T78709 C2XE8D 10831313 Ki = 7.586 nM T78709 C5J1HW 10832055 IC50 = 0.7 nM T78709 CN0Z9Y 10833258 IC50 = 83.18 nM T78709 CL0BO9 10834414 IC50 = 63095.73 nM T78709 C8MHZ9 10835110 Ki = 316.23 nM T78709 C53KRN 10835365 EC50 = 20.89 nM T78709 C0MNA5 10836606 Ki = 1.8 nM T78709 C83QOA 10837858 Ki = 2.2 nM T78709 CC8XL5 10838063 Ki = 12.3 nM T78709 C4V3RT 10848041 Ki = 42 nM T78709 CIQS30 10852612 IC50 = 61.66 nM T78709 CBD60Q 10853821 IC50 > 100000 nM T78709 CU6T1Z 10854403 Ki = 5011.87 nM T78709 CM2TG7 10861457 Ki = 1.175 nM T78709 C3HT1X 10861511 Ki = 0.302 nM T78709 CZ31UD 10861880 Ki = 23.44 nM T78709 C9A8KN 10862425 Ki = 19 nM T78709 C8HN1F 10872581 Ki = 38 nM T78709 COHN31 10873456 Ki = 10.23 nM T78709 C70LSM 10880840 Ki = 37.15 nM T78709 CMV36C 10884046 Ki = 14 nM T78709 CRI50E 10885636 IC50 = 1020 nM T78709 C8OYI0 10891048 Ki = 780 nM T78709 C3I1CT 10892762 Ki = 3.77 nM T78709 CN8P5A 10893547 Ki = 67.61 nM T78709 CEUD36 10893672 Ki = 32.1 nM T78709 CB1HY3 10894144 IC50 = 1570 nM T78709 C2L5YE 10895387 Ki = 2.512 nM T78709 C84RHF 10896220 Ki = 3.3 nM T78709 C1RAP3 10904295 Ki = 17 nM T78709 CC74YP 10905186 Ki = 2.138 nM T78709 C0Q7GV 10915350 Ki = 100 nM T78709 CP7QR4 10915592 Ki = 316.23 nM T78709 CP32CE 10916460 Ki = 1000 nM T78709 CBH30I 10916771 Ki = 13.98 nM T78709 CD7QW2 10917316 Ki = 11.24 nM T78709 CL8AG5 10917920 Ki = 24 nM T78709 C2UZ8H 10917953 Ki = 49 nM T78709 C6D7JR 10924369 Ki = 800 nM T78709 CZN8J0 10925382 Ki = 560 nM T78709 C5X1OQ 10926112 Ki = 100 nM T78709 C3S0ND 10926737 Ki = 0.4365 nM T78709 C0N6KJ 10928520 Ki = 322.1 nM T78709 CD2GN7 10937803 Ki = 1.096 nM T78709 CWE3C9 10946905 Ki = 2000 nM T78709 CNB39C 10947658 Ki = 1.1 nM T78709 CE5XK3 10948133 Ki = 0.16 nM T78709 CGA29L 10948660 Ki = 11.48 nM T78709 CW6T1M 10949284 Ki = 0.5248 nM T78709 CTO4Z9 10949698 Ki = 1.48 nM T78709 CY7B6E 10959998 Ki < 1000 nM T78709 CAIJ61 10961351 Ki = 24.12 nM T78709 C86GIP 10971452 Ki = 5.1 nM T78709 CN6BC3 10972931 Ki = 35 nM T78709 C5NRU3 10973768 Ki = 55 nM T78709 CX5M6J 10974101 Ki = 1.6 nM T78709 CF91AG 10980986 Ki = 0.8318 nM T78709 C6IH1J 10990161 Ki = 550 nM T78709 C4QCY1 10992584 Ki = 0.4467 nM T78709 CF93PW 10992707 Ki = 2.188 nM T78709 CC2NG9 10994812 Ki = 1000 nM T78709 CB1ET0 11002686 Ki = 1.514 nM T78709 C7O5UG 11003379 Ki = 64 nM T78709 CJC9K4 11005810 IC50 = 985 nM T78709 CJS79L 11011968 Ki = 1400 nM T78709 CWU25O 11014017 EC50 > 100000 nM T78709 CLPB39 11014063 Ki = 1.288 nM T78709 C2BF0W 11014848 Ki = 13 nM T78709 CN63RC 11016395 Ki = 5.8 nM T78709 CH9GU5 11016418 Ki = 25 nM T78709 C4T8LY 11020695 IC50 = 8650 nM T78709 CSU4T7 11024618 Ki = 200 nM T78709 C14VMA 11025041 Ki = 26.92 nM T78709 C4Y9XK 11033734 Ki = 255 nM T78709 CX73TF 11035452 Ki = 106 nM T78709 CSK8N7 11037469 Ki = 10.47 nM T78709 C7BS5D 11038248 Ki = 40 nM T78709 C0ES3U 11038263 Ki = 51 nM T78709 CZM27Y 11039289 Ki = 7.2 nM T78709 C7ID8S 11043914 Ki = 2 nM T78709 C3G0FH 11046087 Ki = 400 nM T78709 CH9O0P 11046644 Ki = 0.38 nM T78709 CG0J7X 11047115 Ki = 130 nM T78709 C6EBF3 11048769 IC50 = 2080 nM T78709 CC1YO2 11049209 Ki = 33 nM T78709 C5N9GT 11056946 Ki = 350 nM T78709 CFJG64 11059058 IC50 = 4650 nM T78709 C60SDX 11066440 Ki = 520 nM T78709 C0FT4D 11067619 Ki = 72 nM T78709 CWK94J 11068036 Ki = 30 nM T78709 CL6Y9G 11068509 Ki = 98 nM T78709 C4IN6U 11069073 Ki = 4.898 nM T78709 CG41BK 11071079 IC50 = 1140 nM T78709 CUJ4W7 11071135 Ki = 64 nM T78709 C73PTF 11079090 Ki = 0.8511 nM T78709 C4LP9A 11079476 Ki = 17.38 nM T78709 CKVC23 11079928 Ki = 66.07 nM T78709 CUZ38C 11081136 Ki > 1000 nM T78709 CAJ24R 11090903 Ki = 79.43 nM T78709 CZE43W 11091176 Ki = 1.905 nM T78709 CM2BD4 11092112 Ki = 47 nM T78709 CE42CZ 11092142 Ki = 11 nM T78709 CF32NC 11092254 Ki = 76.23 nM T78709 CRU3M5 11110452 Ki = 41 nM T78709 CC3XK5 11110874 Ki = 22.91 nM T78709 C4VRT9 11111280 Ki = 20 nM T78709 C7DE0U 11113605 IC50 = 1110 nM T78709 CTBF50 11120893 Ki = 840 nM T78709 CVE8T3 11121216 Ki = 6.8 nM T78709 CDMI02 11121708 Ki = 42 nM T78709 C61OTF 11122212 Ki = 1.318 nM T78709 C16LCN 11123104 Ki = 3.02 nM T78709 C6G9KQ 11123573 Ki = 45 nM T78709 CJT65Y 11123606 Ki = 134.5 nM T78709 CF68CS 11133288 Ki = 10.72 nM T78709 C7MD3R 11133868 Ki = 10.23 nM T78709 C3ZJK1 11134424 Ki = 11.6 nM T78709 CC0HY8 11135150 Ki = 53.7 nM T78709 CWB0Z2 11138617 Ki = 3000 nM T78709 CJ63BK 11143175 Ki = 0.631 nM T78709 CA7Y5Z 11144555 Ki = 126.72 nM T78709 C73DFT 11145007 Ki = 1.39 nM T78709 CPA0G8 11145333 Ki = 12 nM T78709 C97CQD 11149594 Ki = 12.5 nM T78709 CYS2X0 11154079 Ki > 1000 nM T78709 C0W4OI 11154198 Ki = 0.54 nM T78709 CVS4I2 11154311 Ki > 1000 nM T78709 CCE1Z3 11156949 Ki = 3.4 nM T78709 CL3C0O 11164277 Ki = 190 nM T78709 C1JC7S 11164569 Ki = 12.9 nM T78709 C8CZQ9 11165409 Ki = 5.14 nM T78709 C8ZN3B 11166042 Ki = 272 nM T78709 CY67TG 11175450 Ki = 4.2 nM T78709 C75WKP 11176199 IC50 = 5 nM T78709 CUE3X2 11176459 Ki = 5.37 nM T78709 C0PHV3 11176648 Ki < 1000 nM T78709 C8KSG5 11177435 Ki = 17.6 nM T78709 CK2V3G 11177467 Ki = 86.25 nM T78709 CL49OC 11178730 IC50 < 10 nM T78709 C6CL1Y 11178830 Ki = 1.585 nM T78709 C4V7ZA 11188024 Ki = 67.8 nM T78709 C4PM2A 11188108 Ki = 300 nM T78709 C8SL0F 11189143 Ki = 17.6 nM T78709 C8FHB1 11189412 Ki = 8.22 nM T78709 C8WHY7 11190823 IC50 = 36.4 nM T78709 C0UQ5K 11191047 Ki > 1000 nM T78709 C6O5JF 11196186 Ki = 827 nM T78709 CCX87L 11200086 Ki = 5.25 nM T78709 C9N5QU 11200511 Ki = 170 nM T78709 C4DUK6 11201573 Ki > 10 nM T78709 CDMQ34 11202474 Ki = 196 nM T78709 COI73W 11206997 Ki = 94 nM T78709 CPX23W 11209208 IC50 > 10000 nM T78709 C36BUG 11210745 Ki > 1000 nM T78709 C4J8YG 11211017 Ki = 54 nM T78709 C41FWO 11213062 Ki = 17.7 nM T78709 C7Q4LE 11213399 IC50 < 10 nM T78709 CVXM03 11221557 Ki = 1.3 nM T78709 C6D1MZ 11223004 Ki = 552 nM T78709 CO58DX 11224478 Ki = 160.3 nM T78709 C0H3SU 11232913 Ki = 0.87 nM T78709 CG71SY 11233991 Ki = 40 nM T78709 C27PSA 11234042 Ki = 260 nM T78709 CLYZ97 11234093 Ki = 1.36 nM T78709 CR10CS 11234230 Ki = 1.06 nM T78709 C0UMB4 11234470 Ki > 1000 nM T78709 C6MI9K 11235335 Ki = 398.11 nM T78709 CNV7Y9 11235558 Ki = 26.27 nM T78709 C3NF5Z 11237443 Ki = 69.18 nM T78709 C1YUE4 11237863 Ki = 5.1 nM T78709 CX5TQ9 11245340 Ki = 248 nM T78709 CJCO91 11245732 Ki = 56.3 nM T78709 CNIC31 11245925 Ki = 125.3 nM T78709 CFC3D9 11246169 Ki = 10.7 nM T78709 C6PUQ7 11246478 Ki = 15.8 nM T78709 CCA7F9 11248217 IC50 = 40 nM T78709 CQ0WO7 11248650 Ki = 46.1 nM T78709 C90WSG 11248705 Ki = 2.512 nM T78709 CS5V2R 11249411 IC50 = 0.7 nM T78709 C7QN4J 11250167 Ki > 1000 nM T78709 CAPX71 11259254 Ki = 63.1 nM T78709 CPBA31 11260140 Ki = 19.2 nM T78709 CEWY47 11261072 Ki = 1.2 nM T78709 CIX25J 11268507 Ki = 65.8 nM T78709 CO25MT 11270107 Ki = 39.81 nM T78709 C2JP5V 11270594 Ki = 5.02 nM T78709 CKEJ43 11270912 Ki = 26.15 nM T78709 C8YKS1 11271864 Ki = 160.5 nM T78709 C5LK4Y 11272673 Ki = 1 nM T78709 C27GXZ 11277680 IC50 > 10000 nM T78709 CJ1S4F 11279872 Ki = 525.6 nM T78709 CW13FD 11280199 Ki = 17.1 nM T78709 CFX51L 11280207 Ki = 8.46 nM T78709 C74SDO 11281688 Ki = 234.4 nM T78709 C2CK8D 11291892 EC50 = 150 nM T78709 CHB4E7 11293380 IC50 = 4 nM T78709 CH4EN9 11293572 Ki = 9.3 nM T78709 C4U7GJ 11293591 IC50 > 2000 nM T78709 CR8ZB5 11295359 Ki = 9.2 nM T78709 C57GTA 11299968 IC50 > 10000 nM T78709 C1VNU0 11303180 Ki = 3.84 nM T78709 CE03YG 11303253 Ki = 2.33 nM T78709 CG0A3L 11303781 Ki = 22.4 nM T78709 C5IQV0 11304135 Ki = 11.27 nM T78709 C9BLC7 11304596 Ki = 0.3981 nM T78709 CJS9C0 11304851 IC50 > 3200 nM T78709 CWF6A1 11305391 IC50 < 10 nM T78709 CI79LV 11307899 Ki = 0.0631 nM T78709 CUXZ91 11311148 IC50 > 10000 nM T78709 C2GZD3 11311204 IC50 > 10000 nM T78709 C9E8WN 11311421 Ki = 252 nM T78709 CI5YQ9 11311820 Ki = 108 nM T78709 C2S0GP 11313610 Ki = 2.5 nM T78709 CCJF50 11313754 Ki = 7.7 nM T78709 CO6NX8 11315660 Ki = 19.97 nM T78709 C1CW4J 11316258 Ki > 10000 nM T78709 CP5E6Q 11316467 IC50 = 3 nM T78709 C0ZXF1 11325675 Ki > 1000 nM T78709 CJT02X 11326158 Ki > 1000 nM T78709 CKUG30 11327798 Ki = 330 nM T78709 CP4K5G 11328306 IC50 < 10 nM T78709 CTN62X 11328382 Ki = 2.512 nM T78709 CBO7W4 11329644 IC50 = 5.2 nM T78709 CH5NT3 11330481 Ki = 8.6 nM T78709 CT3V5I 11338314 Ki = 24 nM T78709 C3JBI0 11338418 Ki > 1000 nM T78709 CT3E6Q 11339067 Ki = 58 nM T78709 C3UA0O 11339351 Ki = 4.07 nM T78709 C4DV2B 11339853 IC50 < 10 nM T78709 CP6VZ2 11339973 Ki = 4.8 nM T78709 CG93PV 11348796 Ki = 25.9 nM T78709 CL7O2I 11349674 Ki = 54.2 nM T78709 C1EGH7 11350339 Ki = 1.68 nM T78709 C8V7GR 11350440 Ki = 717 nM T78709 CJT5E1 11350623 Ki = 26 nM T78709 CI2P0H 11350756 Ki = 19.82 nM T78709 CCY23Q 11351639 Ki = 388 nM T78709 CENY72 11360254 Ki > 1000 nM T78709 CGD42N 11361090 Ki = 97 nM T78709 C6OB5A 11361175 Ki = 29.2 nM T78709 C2HVQ5 11362047 IC50 = 1 nM T78709 CX6N8K 11368804 Ki = 350 nM T78709 CTB03C 11372228 Ki = 9.38 nM T78709 CY20HV 11372576 Ki > 1000 nM T78709 C6A9TH 11373342 Ki = 19.4 nM T78709 CV5XE3 11373704 Ki = 3.5 nM T78709 C1B8WJ 11374059 Ki > 1000 nM T78709 CU6CR4 11374124 IC50 < 10 nM T78709 C2N6CR 11374428 Ki = 2.1 nM T78709 CS9D3C 11374767 Ki = 17.8 nM T78709 CWV4P8 11375860 IC50 > 1000 nM T78709 C5X9JD 11381753 EC50 = 1.3 nM T78709 C6HFW9 11382841 EC50 = 0.34 nM T78709 CHQ9V1 11383270 Ki = 1.94 nM T78709 CBV52J 11384146 Ki = 200 nM T78709 CO1I8H 11384634 Ki = 7.5 nM T78709 CJQ71D 11384983 Ki = 1.29 nM T78709 C3IJD5 11385494 Ki = 73.8 nM T78709 C7XOK1 11394095 Ki = 8.5 nM T78709 CZ2GN9 11394353 Ki = 85.4 nM T78709 C6CAV8 11394411 Ki = 9.8 nM T78709 CU35HP 11395651 Ki = 2.4 nM T78709 CJLS45 11395842 Ki > 1000 nM T78709 CF4OX6 11397149 Ki = 3.981 nM T78709 C7GXP9 11397799 Ki = 6.05 nM T78709 C3V7NH 11405584 Ki = 172 nM T78709 C6WM2A 11406043 Ki > 1000 nM T78709 CMI90K 11407131 Ki > 1000 nM T78709 C7CX1Z 11407133 Ki = 445 nM T78709 CCA2X4 11407766 Ki < 10000 nM T78709 CGN10L 11408148 Ki = 58.8 nM T78709 C6GN7W 11416598 Ki = 36.1 nM T78709 CE5C4L 11418868 Ki = 7.3 nM T78709 C7W6OY 11418949 Ki = 399.2 nM T78709 CKL9J7 11419978 Ki = 1 nM T78709 CRH2D8 11428089 Ki = 1.5 nM T78709 CKPF10 11428376 Ki = 56.3 nM T78709 C13FKL 11429464 Ki > 1000 nM T78709 C0MRK1 11430182 Ki = 3.37 nM T78709 C85LYP 11430418 Ki = 0.7008 nM T78709 C7QX9L 11431037 Ki > 1000 nM T78709 C2B9FV 11440556 Ki = 57.2 nM T78709 CI6NJ2 11440679 Ki = 599.02 nM T78709 C9BNX8 11440979 Ki > 1000 nM T78709 CE79WO 11441652 Ki = 12.08 nM T78709 CGYC26 11442723 Ki = 372 nM T78709 CTD73K 11444410 Ki = 1.9 nM T78709 C6GXJ4 11451971 Ki > 1000 nM T78709 C59SDF 11452106 Ki = 10.1 nM T78709 CM6WJ3 11452107 Ki = 3.3 nM T78709 C6SVK9 11452692 Ki = 2.4 nM T78709 CZ6A2S 11453476 Ki > 1000 nM T78709 C5SJ8M 11459998 Ki = 102 nM T78709 CT73UV 11463955 Ki = 15.6 nM T78709 CG4ST6 11464355 Ki = 794.33 nM T78709 CN6F9K 11464531 IC50 < 10 nM T78709 C89FRU 11464777 Ki = 206.96 nM T78709 C74VWD 11464917 Ki = 107 nM T78709 C6OVE5 11474152 Ki = 25.35 nM T78709 CUOB81 11474564 Ki = 2363.1 nM T78709 C7ZYN5 11474777 Ki = 66.3 nM T78709 C6UBN9 11474937 Ki = 1.2 nM T78709 CQL2E8 11475828 Ki > 1000 nM T78709 CCGF98 11476072 Ki = 398.11 nM T78709 COMY40 11476372 IC50 < 10 nM T78709 CZ5SF1 11477432 IC50 = 91.5 nM T78709 C3QOL9 11484260 Ki = 48 nM T78709 C0GI9R 11484778 Ki = 91.4 nM T78709 CK54EC 11485068 Ki = 5.8 nM T78709 C51OVT 11485631 Ki = 259.34 nM T78709 CC7O5G 11485868 Ki = 2.3 nM T78709 C0XJ1E 11485956 Ki = 41.5 nM T78709 CH9QR1 11486099 Ki = 11 nM T78709 CVX8M3 11486499 Ki = 477.8 nM T78709 C8Q1LZ 11486511 Ki = 0.34 nM T78709 C3NF7L 11487449 Ki = 400.91 nM T78709 C8FN2P 11494093 Ki = 3 nM T78709 C9TU8S 11495769 Ki = 28 nM T78709 CASD80 11501253 Ki = 3 nM T78709 C16AXW 11501537 Ki = 36 nM T78709 CN63TR 11504230 Ki = 25 nM T78709 CE62TB 11511267 Ki = 8.9 nM T78709 CRG4D8 11515921 Ki = 9.31 nM T78709 C59SCV 11516033 Ki = 2300 nM T78709 CW68BJ 11518143 IC50 = 1000 nM T78709 C1KL7T 11518341 Ki = 1.3 nM T78709 CD03GT 11524646 Ki = 112 nM T78709 C38QFE 11530118 IC50 > 10000 nM T78709 CI8GN0 11532563 Ki = 30.9 nM T78709 C7DBO0 11537385 Ki = 52 nM T78709 C0MF3O 11539392 Ki = 11.22 nM T78709 C5ZY6N 11545813 Ki = 2332 nM T78709 C9VC7O 11551780 IC50 > 10000 nM T78709 CW17TM 11554167 Ki = 1.1 nM T78709 COC6U3 11554541 Ki = 11.75 nM T78709 C1V5CH 11559090 Ki > 10000 nM T78709 CY5I0U 11559581 Ki = 390 nM T78709 CVP1Q9 11567578 Ki = 8 nM T78709 CD3Z7J 11567928 Ki = 7.9 nM T78709 CNH1K4 11568826 Ki = 4.7 nM T78709 C8NMI4 11575479 Ki = 170 nM T78709 C6JC2T 11580039 IC50 > 10000 nM T78709 C8CU1X 11581237 Ki = 24 nM T78709 C2IE4D 11583392 Ki = 15.49 nM T78709 C6D1MA 11584660 Ki > 630.96 nM T78709 CU45DK 11595209 Ki > 10000 nM T78709 CGX8F6 11596869 Ki > 3020000 nM T78709 C6G7WS 11603119 Ki = 8 nM T78709 CGD62Y 11603486 Ki = 16 nM T78709 CJW9E6 11604548 Ki = 22.39 nM T78709 CCO15W 11609978 Ki = 218 nM T78709 C6JRN0 11619713 Ki = 23.99 nM T78709 CB7M8E 11625642 Ki = 17 nM T78709 C3IHP8 11626704 Ki = 6.607 nM T78709 C9VAI5 11633517 Ki = 18.2 nM T78709 C2YHQ0 11633739 Ki = 0.77 nM T78709 C2OU7Y 11638332 Ki > 10000 nM T78709 C19UMY 11638640 Ki = 85 nM T78709 CH89AK 11639248 Ki = 6 nM T78709 CI8PF4 11642083 Ki = 14.2 nM T78709 CO89VG 11646566 Ki = 385 nM T78709 C9YA0E 11647443 Ki = 6.3 nM T78709 C1HDM5 11653679 Ki = 117.4 nM T78709 CX7FR8 11655728 Ki = 0.1148 nM T78709 CE4FW0 11662306 Ki = 14 nM T78709 C4L7TV 11662592 Ki = 6.5 nM T78709 C9I7KB 11669646 Ki = 17.38 nM T78709 CB4J2V 11675876 Ki = 3.2 nM T78709 C4KUL7 11676638 Ki = 1.9 nM T78709 CMQX39 11676873 Ki = 34 nM T78709 CTK8R9 11678172 Ki = 22 nM T78709 CLV24Z 11682093 Ki = 258 nM T78709 CDV58J 11696813 Ki = 11.9 nM T78709 C1W8NR 11696910 Ki = 360 nM T78709 CKT7L2 11698732 Ki = 1513 nM T78709 CB4H2O 11699469 Ki = 190 nM T78709 CUVL17 11705133 Ki = 23.44 nM T78709 CJL61W 11706497 Ki = 660 nM T78709 C7RAS6 11712250 Ki = 4.786 nM T78709 C7PK3H 11712470 Ki = 20.89 nM T78709 CHK5I2 11712756 Ki = 0.1585 nM T78709 C46QYG 11720062 Ki = 1360 nM T78709 CGO56C 11720302 Ki = 290 nM T78709 CX9VH0 11720815 Ki = 0.3981 nM T78709 C18COQ 11722647 EC50 = 460 nM T78709 C3KU0D 11722772 Ki > 1000 nM T78709 CAF0J1 11725183 IC50 = 15.85 nM T78709 C2ML7T 11725312 IC50 = 5.012 nM T78709 C1N7MO 11725453 Ki = 142 nM T78709 CXYQ40 11725531 Ki = 2200 nM T78709 C3T9XB 11727140 Ki = 2000 nM T78709 C8YF2N 11728240 Ki = 0.5495 nM T78709 CR29GL 11729007 Ki = 0.7413 nM T78709 CP9TE7 11732304 Ki = 1584.89 nM T78709 CR1L6N 11732516 Ki > 1000 nM T78709 CMO0I9 11739679 Ki = 1670 nM T78709 CL7OG6 11739995 EC50 = 9.06 nM T78709 C57IKL 11740526 Ki = 776.25 nM T78709 CG02AK 11740935 Ki = 40 nM T78709 CJ60OP 11742834 Ki = 6.457 nM T78709 CPG15O 11743399 IC50 > 1000 nM T78709 CVP46J 11746122 Ki = 1000 nM T78709 CYV02C 11747350 Ki = 1800 nM T78709 CO8A3W 11750581 Ki = 9.12 nM T78709 C6IQ8O 11751072 Ki = 4.4 nM T78709 CZN37C 11751188 IC50 = 5 nM T78709 C2J7KO 11751611 Ki > 10000 nM T78709 CBNC94 11752512 IC50 < 10 nM T78709 CS68NX 11754336 Ki = 474.24 nM T78709 CG2WS6 11759467 Ki = 40 nM T78709 CR87JI 11773729 IC50 = 8 nM T78709 CJS7P8 11773878 Ki > 1000 nM T78709 CK1C4D 11774585 Ki = 501.19 nM T78709 C4Y6UC 11776081 Ki > 1000 nM T78709 C4KNX5 11777180 IC50 = 398.11 nM T78709 CJ82MT 11777192 Ki = 79 nM T78709 C2T3OV 11777228 IC50 = 316.23 nM T78709 CM9A7S 11777810 IC50 = 31.62 nM T78709 C06HZD 11782656 Ki = 0.86 nM T78709 CW41AO 11784471 Ki = 1.318 nM T78709 CGI2R8 11792032 IC50 = 4897.79 nM T78709 C2TC7F 11792177 Ki = 34.67 nM T78709 CYR2L7 11793287 IC50 = 346.74 nM T78709 CSLO73 11793877 Ki = 338.84 nM T78709 CW41PM 11793943 Ki = 12.88 nM T78709 CJ0R5E 11794066 Ki = 100 nM T78709 CGVY61 11794853 IC50 = 263.03 nM T78709 CC5DX7 11795765 EC50 = 12.59 nM T78709 C8AWF3 11796209 IC50 = 10232.93 nM T78709 CAMY96 11797158 Ki = 2.2 nM T78709 C90MLE 11797241 IC50 = 22908.68 nM T78709 CQRB24 11797416 Ki = 1584.89 nM T78709 C3U7IY 11797644 IC50 = 8.7 nM T78709 C1M3BY 11797762 IC50 = 54954.09 nM T78709 CN2BP0 11797998 Ki = 1.6 nM T78709 CY75KM 11797999 Ki = 4.3 nM T78709 CAI5J9 11798754 Ki = 5011.87 nM T78709 C3D2AU 11798958 Ki = 21.58 nM T78709 CS19AU 11800592 Ki = 4.06 nM T78709 CVM61S 11809531 Ki = 23 nM T78709 CCI4J0 11810279 Ki = 0.7079 nM T78709 CF9T0I 11810310 Ki = 135 nM T78709 C2R3GJ 11812916 Ki = 49 nM T78709 CLO4B9 11820595 Ki = 0.3 nM T78709 C47SPL 11824009 Ki = 660 nM T78709 CVW4B5 11824522 Ki = 31 nM T78709 CT5DQ9 11824789 Ki = 0.7762 nM T78709 C4WPI2 11825110 Ki = 11.75 nM T78709 CJ49VT 11826976 Ki = 13 nM T78709 CE1QZ8 11827039 Ki = 18 nM T78709 C3LKO9 11845453 Ki = 70.4 nM T78709 C0ZR7C 11845636 Ki = 2.14 nM T78709 CDTQ46 11845643 Ki = 266 nM T78709 CJ9D3N 11845645 Ki = 34.9 nM T78709 CO81MR 11845815 Ki = 1.5 nM T78709 CJ4TH0 11845817 Ki = 2.3 nM T78709 CVOC94 11845819 Ki = 2.1 nM T78709 C3L4QY 11845822 Ki = 1.2 nM T78709 CL0OH3 11845824 Ki = 253 nM T78709 CU39AH 11846005 Ki = 33.2 nM T78709 C58BSD 11846181 Ki = 45.2 nM T78709 CNVY54 11846183 Ki = 18.6 nM T78709 C7P8FK 11846185 Ki = 3.2 nM T78709 CX1B6K 11846187 Ki = 0.1 nM T78709 CXLW54 11948707 EC50 = 0.3 nM T78709 C8JQL7 11957735 IC50 > 10000 nM T78709 C8IFT7 11973922 Ki = 5000 nM T78709 C9IH7R 11973925 Ki = 5000 nM T78709 CS7U5H 11973926 Ki = 5000 nM T78709 C7RY5S 11983282 Ki = 37 nM T78709 CSFD67 11995339 Ki = 5000 nM T78709 CPY4W5 12004114 Ki = 276 nM T78709 C4R5OS 12004116 Ki = 1.2 nM T78709 CLN14H 12004141 Ki = 2 nM T78709 CTFA25 12004142 Ki = 0.4 nM T78709 CTAO18 12004197 Ki = 0.54 nM T78709 C16VZX 12004199 Ki = 0.46 nM T78709 C3QXZ6 12004200 Ki = 0.61 nM T78709 CQ4LI3 12004201 Ki = 0.63 nM T78709 CR9S2B 12004223 IC50 = 2.8 nM T78709 CR3F6P 12004224 Ki = 1.8 nM T78709 C8SVB9 12004226 Ki = 0.61 nM T78709 CI7UF0 12004227 Ki = 3.4 nM T78709 C79VMT 12004253 Ki = 2.1 nM T78709 C3AH4Q 12004254 Ki = 3.6 nM T78709 C2AWK9 12004255 Ki = 0.87 nM T78709 CB2O5M 12004280 Ki = 0.47 nM T78709 C1QY2P 12005903 Ki = 12200 nM T78709 CDNK26 12019526 Ki = 53.2 nM T78709 CCLH20 12313091 Ki > 5000 nM T78709 CLC82F 12374770 Ki = 3750 nM T78709 CQ4V3A 12737487 Ki = 180 nM T78709 CFN31J 12840734 Ki = 35.71 nM T78709 C6P7TB 12840735 Ki = 1.09 nM T78709 C3B8LI 12968865 Ki = 2.72 nM T78709 CB8V2N 12968873 Ki = 4.81 nM T78709 C72BFQ 12968875 Ki = 2.93 nM T78709 C8C5KI 12968876 Ki = 4.08 nM T78709 C13WPY 12968877 Ki = 1.34 nM T78709 C2V9FL 13091268 Ki = 27.7 nM T78709 C2VAE5 13091273 Ki = 37.6 nM T78709 CCG14E 13091356 Ki = 123 nM T78709 C1JW2Q 13091358 Ki = 123 nM T78709 CYN95Z 13091359 Ki = 20 nM T78709 C56TQR 13254321 IC50 = 205 nM T78709 CMA46J 13305910 Ki = 2.455 nM T78709 C0N7VC 13318472 Ki = 1 nM T78709 C2WY8Z 13361400 Ki = 24 nM T78709 C8ALK0 13608253 IC50 = 63 nM T78709 C4A9GO 14039979 Ki = 3.87 nM T78709 CV08GM 14378574 Ki > 5000 nM T78709 C4E7NH 14423371 Ki < 1000 nM T78709 C6E5IV 14576389 EC50 > 100000 nM T78709 CRE73S 14933735 Ki = 0.4 nM T78709 C1Y2UX 14944883 Ki = 1000 nM T78709 CTOY96 14944884 Ki = 0.3 nM T78709 CTQ83H 14944886 Ki = 1.4 nM T78709 C48XLF 14944887 Ki > 1000 nM T78709 CGF64U 14944894 Ki = 16 nM T78709 C47FIY 14950445 Ki = 7.6 nM T78709 C74OKN 14950446 Ki = 103 nM T78709 C8RE3J 14950447 Ki = 1.6 nM T78709 CG96YX 14950448 Ki = 1.9 nM T78709 CFS01M 14950449 Ki = 2.7 nM T78709 CY5P1M 14950450 Ki = 5.3 nM T78709 C0VPR6 14950455 Ki = 0.2 nM T78709 CDT8C1 14950456 Ki = 2.8 nM T78709 CJ16HE 15011385 IC50 = 562 nM T78709 C7VAI1 15011772 IC50 > 10000 nM T78709 CO5C4K 15029820 Ki = 3.2 nM T78709 C7X4LQ 15046233 Ki = 30 nM T78709 CBQY50 15057516 EC50 = 1395 nM T78709 CAF40B 15181802 IC50 = 40 nM T78709 CK21HZ 15226949 IC50 = 58.88 nM T78709 C2XUE8 15344574 Ki = 13 nM T78709 CD25UZ 15389642 Ki = 60.3 nM T78709 C8YB3I 15389644 Ki = 5.9 nM T78709 C8US7F 15410404 Ki = 21 nM T78709 CFTI13 15410410 Ki = 16 nM T78709 C4IB3W 15524005 Ki = 425 nM T78709 CPM16F 15548716 Ki = 1 nM T78709 CL6NC0 15548717 Ki = 6 nM T78709 CZ0A1R 15548718 Ki = 1.7 nM T78709 C06WRK 15548720 Ki = 2.2 nM T78709 C39CEG 15548721 Ki = 72 nM T78709 C0LO4Y 15548722 Ki = 2.3 nM T78709 C5Q8YL 15548723 Ki = 2.8 nM T78709 CRI1N9 15548724 Ki = 5.5 nM T78709 CN5XF4 15549328 Ki = 1.1 nM T78709 C1VWH5 15580747 Ki = 5500 nM T78709 CB6RG2 15654388 Ki = 2.9 nM T78709 CSD46O 15665503 Ki = 0.9 nM T78709 C98WHN 15665505 Ki = 1.2 nM T78709 CMK74C 15665506 Ki = 22 nM T78709 CU31EP 15665507 Ki = 17.8 nM T78709 CT6AY8 15665508 Ki = 0.3 nM T78709 CKQ42I 15665509 Ki = 3 nM T78709 C9SF4H 15665510 Ki = 1 nM T78709 CL2J4H 15665516 Ki = 1.6 nM T78709 C0NUO1 15665517 Ki = 0.6 nM T78709 CYC60K 15744955 Ki = 124 nM T78709 C9J5NY 15744956 Ki = 90 nM T78709 CE6J3A 15744957 Ki = 173 nM T78709 CYD2R7 15744959 Ki = 304 nM T78709 CAF6W2 15744960 Ki = 49 nM T78709 CS50LI 15744961 Ki = 933 nM T78709 CY9H7Z 15744962 Ki > 1000 nM T78709 C1T8UG 15744977 Ki = 12 nM T78709 CEZO41 15744985 Ki = 687 nM T78709 C3AXT9 15744989 Ki = 17 nM T78709 C1XKH0 15744991 Ki = 2.4 nM T78709 CD26OR 15744995 Ki = 31 nM T78709 C02THF 15744998 Ki = 3.2 nM T78709 CT2H9J 15745003 Ki = 105 nM T78709 CK8H9R 15745005 Ki = 109 nM T78709 C5S6ZU 15745006 Ki > 1000 nM T78709 CHQ9A5 15745007 Ki = 84 nM T78709 CY96DH 15745008 Ki = 95 nM T78709 C9LGI7 15745009 Ki > 1000 nM T78709 CU9QY8 15745011 Ki = 171 nM T78709 C74YVE 15745012 Ki > 1000 nM T78709 C90BKV 15745014 Ki = 4493 nM T78709 CCM64H 15786488 Ki = 47.86 nM T78709 CTPX97 15803947 Ki = 17 nM T78709 C1JYT9 15937766 Ki = 44 nM T78709 CT12KQ 15980807 Ki = 927 nM T78709 C5HQT6 15980808 Ki = 19 nM T78709 C4JT9L 15980809 EC50 = 54 nM T78709 C76PIS 15980810 Ki = 129 nM T78709 CF4Z2U 15980852 Ki = 966 nM T78709 CZ39MX 15980853 EC50 = 4 nM T78709 C0H7GI 15980854 Ki = 50 nM T78709 CTH2S5 15980895 Ki = 4 nM T78709 CXW37K 15987265 IC50 = 4800 nM T78709 C1LWZ6 16006605 Ki = 91 nM T78709 CK36NS 16006607 Ki = 265 nM T78709 CMZ69G 16007004 Ki = 4 nM T78709 C3M8GJ 16026344 Ki = 2745 nM T78709 C1SR0O 16071847 Ki > 5000 nM T78709 C4CZ6A 16091081 Ki = 0.4 nM T78709 C7UOM4 16092107 Ki = 24 nM T78709 CD3E8L 16093484 Ki = 181 nM T78709 CEW91O 16093485 Ki = 105 nM T78709 CTFM10 16109481 EC50 = 1412.54 nM T78709 C5RY7T 16109482 EC50 = 67.61 nM T78709 CTCG69 16109483 EC50 < 10000 nM T78709 C0HK1Y 16109484 EC50 = 46.77 nM T78709 CC1R5U 16109485 EC50 = 194.98 nM T78709 CO3HR8 16109486 EC50 = 6.457 nM T78709 C2JW4B 16109487 EC50 = 24.55 nM T78709 CS2QA9 16109488 EC50 = 112.2 nM T78709 C4GRY1 16109489 EC50 = 2.63 nM T78709 CQV32M 16109492 EC50 < 10000 nM T78709 CCOR68 16109496 EC50 = 69.18 nM T78709 CLFO01 16109508 EC50 = 1548.82 nM T78709 C4V8US 16109509 EC50 < 10000 nM T78709 CB8SI6 16109510 EC50 = 134.9 nM T78709 CF2A8R 16109511 EC50 = 32.36 nM T78709 CQS4V1 16112801 IC50 > 1000 nM T78709 CZ1WJ4 16117151 Ki = 455 nM T78709 CM32ZX 16117153 Ki = 4347 nM T78709 CXTB90 16117279 Ki = 859 nM T78709 C1F2LS 16118795 Ki > 5000 nM T78709 C69VDS 16118923 Ki = 3011 nM T78709 CZ2IS9 16660294 Ki > 10000 nM T78709 C3JV0P 16718827 IC50 > 1000 nM T78709 C3YN5S 16718917 IC50 = 1142 nM T78709 CJ8Y1H 16718919 IC50 > 10000 nM T78709 CB7G3R 16718920 IC50 > 1000 nM T78709 CM3FT4 16739258 Ki = 29 nM T78709 CT9GP4 16763549 Ki = 19890 nM T78709 CR63LE 17055181 Ki = 195600 nM T78709 C0QX5J 17374371 Ki = 4307 nM T78709 CF25CM 17449900 Ki = 6.8 nM T78709 C0T9ZY 17947861 Ki = 6.31 nM T78709 C42YEX 18133517 Ki = 52610 nM T78709 CI90UP 18133518 Ki = 38290 nM T78709 C7R1IG 18137015 Ki = 1285 nM T78709 C4I1FW 18137017 Ki = 1637 nM T78709 C07EOI 18137020 Ki = 3614 nM T78709 C9PV8A 18180076 IC50 = 57 nM T78709 CHXQ26 18366015 IC50 = 3548.13 nM T78709 C7G3UV 18694165 IC50 = 6.31 nM T78709 CIEM47 18694195 IC50 = 5.012 nM T78709 CZV26X 18694196 IC50 = 0.3981 nM T78709 CYOU05 18922713 EC50 = 0.13 nM T78709 CJH07D 18988813 Ki > 5000 nM T78709 C78NBQ 18988815 Ki > 1000 nM T78709 CVF4R7 18988817 Ki = 4.7 nM T78709 C08HLD 18988835 Ki > 1000 nM T78709 CV08LK 18988846 Ki = 4.4 nM T78709 C96KED 19023504 IC50 = 440 nM T78709 CU8TB3 19041559 Ki = 210 nM T78709 CYJ48A 19066163 Ki = 393 nM T78709 C0BE1M 19066188 Ki = 450 nM T78709 CV5FR6 19066200 Ki = 1000 nM T78709 C4RU6O 19066201 Ki = 700 nM T78709 CN96TB 19066203 Ki = 571 nM T78709 C60SWJ 19066205 Ki = 79 nM T78709 C5MS9T 19066235 Ki = 3000 nM T78709 C6AOE8 19426635 IC50 > 1000 nM T78709 C25YQI 19770958 IC50 > 10000 nM T78709 CQ3JL0 19956256 IC50 = 5754.4 nM T78709 C7T8JC 19958494 Ki > 10000 nM T78709 C6LI5E 19958507 Ki > 10000 nM T78709 CLVT08 19978038 IC50 = 97.72 nM T78709 CF34NC 19978059 IC50 = 9549.93 nM T78709 C7D0PH 20763915 Ki = 4 nM T78709 C10IHJ 21073216 Ki = 52.7 nM T78709 CH8EN1 21073533 Ki = 40.7 nM T78709 C1R0SA 21073563 Ki = 8.5 nM T78709 CBUG29 21073579 Ki = 1.7 nM T78709 C15NJA 21073584 Ki = 13.8 nM T78709 CXMG13 21073587 Ki = 0.95 nM T78709 C57EJD 21073595 Ki = 4.6 nM T78709 CR0D3H 21073606 Ki = 0.84 nM T78709 C60WIT 21073656 Ki = 1.2 nM T78709 C6CQO1 21073658 Ki = 8.4 nM T78709 C1OL3G 21073667 Ki = 3.3 nM T78709 CVT16Y 21073690 Ki = 2 nM T78709 C9GHF5 21073716 Ki = 3 nM T78709 CA24ZJ 21073731 Ki = 1.2 nM T78709 CGP56E 21073788 Ki = 0.78 nM T78709 C6ARE1 21073793 Ki = 1.1 nM T78709 C3KMW4 21073817 Ki = 3.9 nM T78709 CHM64K 21073872 Ki = 11.4 nM T78709 C5O8SN 21268191 Ki = 7.84 nM T78709 CJ63ET 21268208 Ki = 551 nM T78709 CLW5Z0 21268321 Ki = 32 nM T78709 CQ17TR 21460878 IC50 = 31.62 nM T78709 C2JT9X 21460905 IC50 = 1.995 nM T78709 C3T5HF 21509921 Ki = 596 nM T78709 CFN81Q 21527771 Ki = 74 nM T78709 CH59WN 21533446 Ki = 74 nM T78709 C4B0TN 21557475 Ki = 172 nM T78709 CUV0N3 21689040 EC50 = 1.2 nM T78709 CX45FW 21797090 EC50 = 14.79 nM T78709 CT7XG9 21830793 EC50 = 0.1 nM T78709 C9X8PI 22001618 Ki = 476 nM T78709 CYH4J9 22002244 Ki = 3 nM T78709 CBN84K 22065997 Ki = 990.7 nM T78709 C12QOJ 22113436 Ki = 10.6 nM T78709 CD7M8K 22113440 Ki = 6.82 nM T78709 CF8B0D 22113443 Ki = 28.6 nM T78709 CO32YX 22254068 Ki = 478 nM T78709 CNB53V 22321203 Ki = 6530 nM T78709 C2Z0BJ 22326660 Ki = 19.95 nM T78709 CD80PB 22326688 Ki = 0.2512 nM T78709 CJ3P6O 22326704 Ki = 50.12 nM T78709 C6UXL4 22330705 Ki = 19670 nM T78709 CZG9S2 22425072 Ki = 11860 nM T78709 C5SI3U 22464564 Ki = 93.4 nM T78709 CJ6WF3 22464606 Ki = 25.8 nM T78709 CA5BY9 22464614 Ki = 24.2 nM T78709 CQB94R 22464634 Ki = 9.1 nM T78709 CAZ23L 22464649 Ki = 0.7 nM T78709 CJCY98 22464720 Ki = 2.8 nM T78709 CB97XC 22464804 Ki = 11.8 nM T78709 C9MB7K 22464806 Ki = 429 nM T78709 C7DXE6 22464831 Ki = 2.9 nM T78709 C76FEA 22464842 Ki = 2.5 nM T78709 CPD8Q7 22549784 Ki = 12490 nM T78709 CRU1N2 22611622 Ki = 68 nM T78709 C49VCE 22675297 Ki = 0.82 nM T78709 CIC7F6 22675312 Ki = 15.9 nM T78709 CBCK13 22675339 Ki = 1.04 nM T78709 CPU6C8 22675347 Ki = 3.03 nM T78709 C85YGH 22675350 Ki = 0.89 nM T78709 CP41JS 22675387 Ki = 6.46 nM T78709 C5R7JT 22675398 Ki = 23.4 nM T78709 CA02UK 22849991 Ki = 18.7 nM T78709 C5DJR8 22849992 Ki = 2.9 nM T78709 C3RO8S 22864491 Ki = 106 nM T78709 C91NKL 22864495 Ki = 322 nM T78709 C0MZV7 22998900 Ki = 13 nM T78709 CQB20R 23155620 IC50 = 4.2 nM T78709 CZ25WJ 23155621 IC50 = 62.3 nM T78709 CM57CZ 23155625 IC50 = 5.6 nM T78709 CFB0G1 23155644 IC50 = 55.4 nM T78709 C7FQU2 23155650 IC50 < 10 nM T78709 C8Y7LC 23155667 IC50 < 10 nM T78709 C1PX5S 23155676 IC50 = 7.6 nM T78709 CC46FD 23155688 IC50 < 10 nM T78709 CAC0S3 23155689 IC50 = 4.3 nM T78709 C57WEZ 23155758 IC50 < 10 nM T78709 CXHB39 23155770 IC50 < 10 nM T78709 C1OVU4 23155818 IC50 = 1.3 nM T78709 CKQ2Y0 23155825 IC50 = 18 nM T78709 C2NOU7 23155834 IC50 < 1 nM T78709 C75GWQ 23155840 IC50 = 64.6 nM T78709 C1N6SD 23155860 IC50 = 24.4 nM T78709 CTC8Y5 23155869 IC50 = 90.4 nM T78709 CK3PM5 23155885 IC50 > 100 nM T78709 C8XYR2 23155900 IC50 = 13.5 nM T78709 CFG6D5 23155906 IC50 > 100 nM T78709 CQS93U 23155935 IC50 = 6.1 nM T78709 C3P1TG 23155946 IC50 = 66.6 nM T78709 C5LCT7 23155948 IC50 < 1 nM T78709 C6QCL8 23155950 IC50 > 100 nM T78709 C7DQ5C 23155951 IC50 < 1 nM T78709 C7PSB8 23155955 IC50 < 10 nM T78709 CXR3G9 23155963 IC50 = 96 nM T78709 CC1P4X 23155976 IC50 > 100 nM T78709 CJY62P 23155980 IC50 > 100 nM T78709 CH5C7X 23288790 Ki = 2463 nM T78709 C0NI3J 23290944 Ki = 1.21 nM T78709 CL3O0E 23290959 Ki = 33 nM T78709 C57MVP 23369416 Ki = 40 nM T78709 CL46OM 23625239 EC50 = 2041.74 nM T78709 CP47WR 23625381 EC50 = 3630.78 nM T78709 CFE62K 23625383 EC50 = 154.88 nM T78709 C3CJO8 23625384 EC50 = 309.03 nM T78709 C29WCH 23625533 EC50 = 85.11 nM T78709 CW63KP 23625534 EC50 = 42.66 nM T78709 C1N6WM 23625537 EC50 = 10 nM T78709 CMP38W 23625705 EC50 = 89.13 nM T78709 CXD3E6 23625925 Ki = 1513.56 nM T78709 C1YJ7D 23626001 EC50 = 239.88 nM T78709 CCQ4M1 23626164 EC50 = 446.68 nM T78709 CPZV02 23643663 Ki = 167 nM T78709 CX93TK 23643870 Ki = 112 nM T78709 CO4C6M 23653115 Ki = 36.31 nM T78709 CNU2X4 23725134 IC50 > 1000 nM T78709 CQE1N7 23906630 Ki = 23510 nM T78709 CZ0G9H 24069165 EC50 = 10200 nM T78709 CBXC05 24424330 IC50 = 0.6 nM T78709 CQ0KU9 24738459 Ki = 0.0504 nM T78709 C6GBU8 24762221 Ki = 0.7943 nM T78709 C6Z1PX 24768516 Ki = 79.2 nM T78709 C0HO5Q 24768517 Ki = 168 nM T78709 CX7E3K 24768518 Ki = 60 nM T78709 CW3PD4 24768519 Ki = 1196 nM T78709 C9G8ZH 24768520 Ki = 133 nM T78709 C0VPJ8 24768521 Ki = 415 nM T78709 C9UOG8 24768522 Ki = 2500 nM T78709 CSW50R 24768524 Ki = 29.2 nM T78709 CW8N2E 24768525 Ki = 36.4 nM T78709 CCT04Q 24768526 Ki = 194 nM T78709 C0I2HU 24769156 Ki = 99 nM T78709 CD7CV6 24771120 Ki = 8500 nM T78709 CEQY61 24781869 Ki = 1300 nM T78709 C3JSR4 24794436 IC50 > 1000 nM T78709 CJ4RO1 24804774 Ki = 0.631 nM T78709 CK84BF 24804775 EC50 = 0.03162 nM T78709 C1Z3OQ 24804941 Ki = 1.259 nM T78709 C6AE2U 24804942 Ki = 3.981 nM T78709 C1ZYM4 24804943 Ki = 3.981 nM T78709 C9K0CX 24805674 Ki = 97 nM T78709 CZY17F 24805675 Ki = 28 nM T78709 CT10CH 24805872 Ki = 2.6 nM T78709 C9DTE6 24805873 Ki = 0.2 nM T78709 C8L9WD 24805874 Ki = 0.5 nM T78709 C49EDA 24805875 Ki = 0.38 nM T78709 C58RUQ 24805876 Ki = 0.03 nM T78709 C36NFD 24806070 Ki = 22 nM T78709 CA9G8E 24806071 Ki = 0.2 nM T78709 C9QBV5 24806072 Ki = 2.1 nM T78709 C5I1BZ 24806073 Ki = 4.6 nM T78709 CL61TY 24806074 Ki = 0.54 nM T78709 C58AMS 24829343 Ki = 1610 nM T78709 CDC91N 24839550 Ki = 100 nM T78709 CY21RE 24841480 Ki = 1700 nM T78709 C93JWY 24865538 Ki = 25.12 nM T78709 C5F2VL 24865539 Ki = 5.012 nM T78709 CW9N1Z 24865540 Ki = 158.49 nM T78709 C8PXH7 24865541 Ki = 1258.93 nM T78709 CN5VB4 24865542 Ki = 6.31 nM T78709 CPF5E2 24865543 Ki = 25.12 nM T78709 CGDV58 24865724 Ki = 5.012 nM T78709 C3HK0J 24865725 Ki = 2.512 nM T78709 C5TX3M 24865726 Ki = 12.59 nM T78709 C0O6FX 24865727 Ki = 7.943 nM T78709 C98ZIV 24882509 IC50 = 500 nM T78709 C6L7KS 24887518 Ki < 3162.28 nM T78709 CI53SE 24893978 Ki = 38 nM T78709 CAOF91 24894071 IC50 > 10000 nM T78709 C3C0KP 24894134 EC50 > 50000 nM T78709 CX6R0P 24894141 Ki = 1.413 nM T78709 CMN75S 24901425 Ki = 158.49 nM T78709 C9OAG1 24906198 Ki = 28.18 nM T78709 CUY89J 24936155 Ki = 280 nM T78709 C0BP8C 24939244 IC50 > 10000 nM T78709 C8DJG7 24963860 Ki = 4826 nM T78709 C6DO4B 25032525 Ki = 1.1 nM T78709 CR5FX4 25059765 IC50 > 10000 nM T78709 CMVL70 25059766 IC50 > 1000 nM T78709 CED30A 25059770 IC50 > 1000 nM T78709 CJU9Y7 25060021 IC50 > 1000 nM T78709 C36PMH 25060023 IC50 > 1000 nM T78709 CHSB87 25060024 IC50 > 1000 nM T78709 CTI38U 25060119 Ki = 1310 nM T78709 CYJ5G1 25067564 Ki = 4730 nM T78709 C7O8YH 25068794 Ki = 0.149 nM T78709 CZ9SN8 25068797 Ki = 0.102 nM T78709 CL46IP 25068850 Ki = 0.204 nM T78709 CEH7D9 25068903 Ki = 0.243 nM T78709 CB03DL 25068905 Ki = 0.0152 nM T78709 C5ZHN9 25068906 Ki = 0.0447 nM T78709 C0ZJB7 25068907 Ki = 0.0141 nM T78709 C9G7EM 25068908 Ki = 1.54 nM T78709 CZBY61 25068962 Ki = 0.108 nM T78709 CP9G5Z 25068963 Ki = 0.269 nM T78709 CB3F0I 25068964 Ki > 4.04 nM T78709 CCO7B3 25068966 Ki = 1.46 nM T78709 C16ERI 25069015 Ki = 0.179 nM T78709 CZM94A 25069016 Ki = 0.0501 nM T78709 CYZ45N 25069072 Ki = 1.99 nM T78709 CEB96S 25069073 Ki = 1.92 nM T78709 CAI7V1 25069074 Ki = 0.279 nM T78709 C8A3HM 25069121 Ki = 0.74 nM T78709 CG5WX6 25069122 Ki = 6.88 nM T78709 CS8VK1 25069125 Ki = 1.45 nM T78709 CHZB81 25069180 Ki = 1.3 nM T78709 C3W1AX 25069181 Ki = 0.863 nM T78709 CPGZ03 25069239 Ki = 0.671 nM T78709 CT0R3H 25069240 Ki = 0.341 nM T78709 CX5JF4 25069241 Ki < 0.521 nM T78709 C1P4EC 25069242 Ki = 0.88 nM T78709 CCV27I 25069243 Ki = 0.637 nM T78709 C5BR0K 25069297 Ki = 1.77 nM T78709 CU34CX 25069298 Ki = 0.118 nM T78709 C0Z6YL 25069299 Ki = 2.71 nM T78709 C5Z9MA 25069300 Ki = 0.128 nM T78709 C1OGS2 25069301 Ki < 0.205 nM T78709 C53LJG 25069302 Ki < 0.14 nM T78709 CX74UK 25069353 Ki = 3.04 nM T78709 C8F6VC 25069354 Ki = 3.62 nM T78709 C56RCY 25069355 Ki = 4.56 nM T78709 CI7SM5 25069356 Ki = 5.01 nM T78709 C45AHR 25093400 Ki = 13 nM T78709 C0DFW8 25093401 Ki = 37 nM T78709 C67OHQ 25093402 Ki = 275 nM T78709 CXA09P 25107515 Ki = 2.04 nM T78709 CDW7J5 25107516 Ki = 3.7 nM T78709 C81QKN 25107517 Ki = 40 nM T78709 C1QE6A 25107519 Ki = 13 nM T78709 C3VY8O 25107520 Ki = 70 nM T78709 CYE53P 25107578 Ki = 325 nM T78709 CJO1X8 25107579 Ki = 94 nM T78709 C59IVO 25107580 Ki = 53 nM T78709 CMPG74 25107581 Ki = 10.3 nM T78709 CNW7A8 25107582 Ki = 57 nM T78709 CU71RN 25107583 Ki = 29 nM T78709 C8ZM2J 25107647 Ki = 124 nM T78709 CJF71U 25107648 Ki = 95 nM T78709 C6M9LD 25107649 Ki = 12 nM T78709 CEM90Y 25107650 Ki = 139 nM T78709 C2JW3O 25107651 Ki = 8.2 nM T78709 C7M1XT 25107652 Ki = 19 nM T78709 C4ASH8 25107717 Ki = 43 nM T78709 CQ71NR 25107718 Ki = 106 nM T78709 C3NGR5 25108474 Ki = 1.07 nM T78709 C8GW4P 25108475 Ki = 22 nM T78709 C2FY7C 25128757 Ki = 1720 nM T78709 C5NW4M 25129807 Ki > 10000 nM T78709 CAV81B 25130157 Ki = 1780 nM T78709 CF7P2A 25130875 Ki = 38.9 nM T78709 C7P1QS 25130876 Ki = 3.467 nM T78709 C6G5BO 25130877 Ki = 257.04 nM T78709 CL8GD3 25130878 Ki = 53.7 nM T78709 CT78MG 25130879 Ki = 4.169 nM T78709 C7WXA2 25131192 Ki > 1000 nM T78709 C3UVA0 25131193 Ki = 1.413 nM T78709 C0GM3L 25131196 Ki = 147.91 nM T78709 CCWO92 25131197 Ki = 7.586 nM T78709 CFUT35 25131198 Ki = 0.5888 nM T78709 C9P1ZV 25131523 Ki = 229.09 nM T78709 C1Y3TS 25131871 Ki = 416.87 nM T78709 C8CM1N 25131874 Ki = 37.15 nM T78709 CFJ6Y9 25131876 Ki = 0.6607 nM T78709 CNQX42 25132217 Ki = 25.7 nM T78709 C7WE4Y 25132564 Ki = 234.42 nM T78709 C6K1TB 25132565 Ki = 52.48 nM T78709 CJ19KC 25132566 Ki = 6.026 nM T78709 C67QCG 25132869 Ki > 10000 nM T78709 C0J3RD 25138742 Ki = 10.9 nM T78709 C8SPL6 25138902 Ki = 12.6 nM T78709 CSM12R 25138907 Ki = 0.81 nM T78709 CN13MI 25138912 Ki = 3.98 nM T78709 C3LHY5 25138913 Ki = 3.22 nM T78709 CTYC19 25139055 Ki = 6.21 nM T78709 C9JR6E 25139058 Ki = 1.75 nM T78709 C3VNW8 25139062 Ki = 14 nM T78709 C1QHJ5 25139063 Ki = 10.6 nM T78709 CAY54E 25139064 Ki = 5.44 nM T78709 CB8E6J 25139065 Ki = 19.25 nM T78709 C2L3OB 25139066 Ki = 10.78 nM T78709 C5PO7X 25139217 Ki = 1.32 nM T78709 C0A5NK 25139366 Ki = 2.64 nM T78709 C9RO2S 25139374 Ki = 17.35 nM T78709 CS14YK 25139517 Ki = 6.54 nM T78709 C5JWI0 25139643 Ki = 1.19 nM T78709 C6I9FN 25139645 Ki = 26.1 nM T78709 CJ63XC 25139652 Ki = 3.25 nM T78709 C6OCL8 25139785 Ki = 16.6 nM T78709 CA3E2B 25139914 Ki = 9.64 nM T78709 CD69BU 25140055 Ki = 12.83 nM T78709 CP57TN 25140057 Ki = 39.95 nM T78709 CG05CH 25140362 Ki = 1.88 nM T78709 CQO5P0 25140648 Ki = 5.35 nM T78709 CEF59R 25141218 Ki = 6.2 nM T78709 CL84YJ 25141534 Ki = 100 nM T78709 C4FXR9 25141535 Ki = 132 nM T78709 CW2PL7 25155850 Ki = 1130000 nM T78709 C4UXF6 25155851 Ki > 5000000 nM T78709 C65LWZ 25156129 Ki = 2874000 nM T78709 CS3Q4N 25156130 Ki = 1241000 nM T78709 CZ04VO 25156131 Ki = 756000 nM T78709 C6MXE3 25156132 Ki > 5000000 nM T78709 CU5C7V 25156133 Ki = 800000 nM T78709 C65FNY 25156411 Ki > 5000000 nM T78709 CKIH98 25156412 Ki = 656000 nM T78709 C35NHX 25156413 Ki = 558000 nM T78709 C94OIG 25156414 Ki > 5000000 nM T78709 C1IEF6 25156415 Ki > 5000000 nM T78709 CL1B2G 25156416 Ki = 1124000 nM T78709 CUX0F4 25156684 Ki = 1331000 nM T78709 CB4A2S 25156685 Ki > 5000000 nM T78709 CJO48V 25156686 Ki > 5000000 nM T78709 CF27EQ 25156688 Ki = 686000 nM T78709 C8U6PV 25156966 Ki > 5000000 nM T78709 C05TOB 25157253 Ki > 5000000 nM T78709 CYM3H9 25157257 Ki = 331000 nM T78709 CS0E3J 25157260 Ki > 5000000 nM T78709 CQI4S2 25157543 Ki > 5000000 nM T78709 C6Y4AJ 25157546 Ki = 1310000 nM T78709 CKP10W 25157549 Ki > 5000000 nM T78709 C9B0UR 25157845 Ki > 5000000 nM T78709 CX2CP8 25157848 Ki > 5000000 nM T78709 C1XP3Q 25157850 Ki > 5000000 nM T78709 C5J4ES 25158433 Ki = 1308000 nM T78709 COK46A 25158434 Ki = 1409000 nM T78709 CQRL83 25158435 Ki = 1092000 nM T78709 C26IMW 25158436 Ki = 783000 nM T78709 CNO83H 25181488 Ki = 0.6026 nM T78709 CEYF08 25181489 Ki = 0.5888 nM T78709 CI95EF 25192947 Ki > 10000 nM T78709 CDQ70A 25208878 IC50 > 1000 nM T78709 CJ1Z9H 25216680 Ki = 10100 nM T78709 C1T3LR 25218143 Ki = 8720 nM T78709 CPI03N 25218397 Ki = 8670 nM T78709 CL1R3Q 25218401 Ki = 12200 nM T78709 CW07GN 25256855 Ki = 454 nM T78709 CM2T9Y 25263297 Ki = 6400 nM T78709 CFJM71 25263302 Ki = 5600 nM T78709 C15QMB 25263320 IC50 > 1000 nM T78709 CYS8B2 25265257 EC50 = 18 nM T78709 C4MRQ0 27842480 Ki = 2108 nM T78709 CWT9F7 28918670 Ki = 562.34 nM T78709 CHJ35A 32354149 Ki = 2108 nM T78709 C9QGK3 34257212 Ki = 18 nM T78709 CDV36I 37219401 Ki = 1764 nM T78709 CA58DL 41305446 Ki = 9389 nM T78709 CN2CY7 42266246 Ki = 24.7 nM T78709 CI4Q3O 42266677 Ki = 54.3 nM T78709 CDP76A 42266865 Ki = 2.32 nM T78709 CO3LQ2 42267076 Ki = 50.7 nM T78709 CP54VF 42267840 Ki = 24.4 nM T78709 CWOL80 42273326 Ki = 17.8 nM T78709 CG56DF 42388639 IC50 = 4.6 nM T78709 CH5QX6 42389467 IC50 = 39 nM T78709 C32NKC 42605991 EC50 = 30 nM T78709 CX8L2W 42605992 EC50 = 46 nM T78709 CSY8H7 42605993 EC50 = 20 nM T78709 C0XMS9 42605994 EC50 = 17 nM T78709 CHRM07 42606101 EC50 = 30 nM T78709 C7FMV8 42606103 EC50 = 35 nM T78709 C2J3OV 42606104 EC50 = 20 nM T78709 CL7Q0T 42606105 EC50 = 42 nM T78709 CJ7P0D 42606106 EC50 = 54 nM T78709 CR7S3Z 42606222 EC50 = 12 nM T78709 CDEK82 42606334 EC50 = 99 nM T78709 CW30MB 42606335 EC50 = 50 nM T78709 CY10AG 42606336 EC50 = 62 nM T78709 C6VP2A 42606337 EC50 = 240 nM T78709 CD61JW 42606339 EC50 = 10 nM T78709 CJA90T 42606340 EC50 = 130 nM T78709 C83KBX 42606455 EC50 = 39 nM T78709 CB06ST 42606456 EC50 = 59 nM T78709 CEKO32 42606457 EC50 = 86 nM T78709 C3A6UH 42606458 EC50 = 63 nM T78709 C84YQR 42606459 EC50 = 15 nM T78709 CCZG96 42606461 EC50 = 240 nM T78709 C47AMD 42606572 EC50 = 34 nM T78709 C0TN5O 42606573 EC50 = 16 nM T78709 C1ZD2B 42606577 EC50 = 93 nM T78709 CO59TU 42606688 EC50 = 310 nM T78709 CA0B9F 42625181 Ki = 18.1 nM T78709 C3L0TN 42625183 Ki = 39 nM T78709 CW0OU4 42625185 Ki = 26 nM T78709 CHY12B 42625186 Ki > 1000 nM T78709 CP5X3K 42625188 Ki = 181 nM T78709 C8QSX3 42625267 Ki > 1000 nM T78709 CTM69J 42625269 Ki > 1000 nM T78709 CYM0J6 42625295 Ki = 58.3 nM T78709 CPDG98 42625353 Ki > 1000 nM T78709 CK3QD2 42625354 Ki = 360 nM T78709 CJ64FG 42625356 Ki = 11.5 nM T78709 C27KEF 42625359 Ki > 1000 nM T78709 CN81SE 42625440 Ki = 219 nM T78709 CF7DM0 42625445 Ki = 22 nM T78709 CJI51X 42625446 Ki = 16 nM T78709 CD9RN1 42626103 Ki = 193 nM T78709 CLH7Y0 42626289 Ki > 1000 nM T78709 C75QPL 42626291 Ki > 1000 nM T78709 C5VTZ6 42626293 Ki = 124 nM T78709 C70SWL 42626361 Ki > 1000 nM T78709 CV2X5B 42635027 IC50 = 44 nM T78709 CS9Q3H 42635204 IC50 = 29 nM T78709 CQ2M5S 42635387 IC50 = 215 nM T78709 CR3KM7 42635388 IC50 = 39 nM T78709 CJ3NP5 42636941 IC50 = 5011.87 nM T78709 C8A2VG 43066988 Ki = 30 nM T78709 C0AI7N 43229249 Ki = 707.95 nM T78709 CW2DP3 44123711 Ki = 5.129 nM T78709 C1YM3D 44131466 Ki = 24 nM T78709 CMTB93 44131470 Ki = 29 nM T78709 CYE20L 44131666 Ki = 3.7 nM T78709 CPR7L3 44133672 Ki = 71 nM T78709 CE3SD9 44133859 Ki = 37 nM T78709 CZ2VQ1 44133861 Ki = 37 nM T78709 C9P5XU 44133863 Ki = 5.5 nM T78709 C2G7AO 44134036 Ki = 10 nM T78709 C5YKI9 44134038 Ki = 11 nM T78709 C6DQJ3 44134039 Ki = 7.2 nM T78709 C8RZX0 44134041 Ki = 173 nM T78709 CXZH39 44138098 Ki = 0.2512 nM T78709 CUOD42 44138104 Ki = 0.1585 nM T78709 C8R1QU 44178224 Ki = 12.4 nM T78709 CW3X1D 44182545 Ki = 2.81 nM T78709 CI8SO3 44182695 Ki = 71.9 nM T78709 CQP5G0 44182696 Ki = 7.72 nM T78709 CYMQ43 44182839 Ki = 44.3 nM T78709 C6SG0O 44192200 Ki = 3.7 nM T78709 CMR7T1 44204999 EC50 = 50.12 nM T78709 CVG6X1 44209472 Ki = 3.6 nM T78709 CD5AB7 44209480 Ki = 1.1 nM T78709 CXR6K7 44212701 Ki = 6.5 nM T78709 C8ORL9 44212702 Ki = 9.2 nM T78709 CN71EI 44212703 Ki = 12 nM T78709 CSK83C 44213966 IC50 = 3.981 nM T78709 C69CVF 44213967 IC50 = 25.12 nM T78709 C34HLC 44213968 IC50 = 5.012 nM T78709 C8EDC7 44214579 Ki = 36.4 nM T78709 CIHS31 44219920 Ki = 20 nM T78709 CL0SN8 44219921 Ki = 32.9 nM T78709 C36ZRH 44219922 Ki = 17.2 nM T78709 CHY51E 44219923 Ki = 7.2 nM T78709 CC4RT6 44220111 Ki = 172 nM T78709 CL12NI 44220112 Ki = 47.3 nM T78709 C21PGV 44220113 Ki = 167 nM T78709 C4QOE7 44220114 Ki = 5.5 nM T78709 CTK38P 44220115 Ki = 2.8 nM T78709 C2M9DC 44220314 Ki = 6.8 nM T78709 C8I4KR 44220315 Ki = 2 nM T78709 CVW0O8 44220316 Ki = 1.5 nM T78709 C2FDB1 44250364 IC50 > 10000 nM T78709 C8MC0Q 44251387 IC50 > 10000 nM T78709 C5YEA8 44251388 IC50 > 10000 nM T78709 C0BSF6 44251389 IC50 > 10000 nM T78709 C2K0VZ 44253016 EC50 > 3162.28 nM T78709 CL09IQ 44263496 IC50 > 10000 nM T78709 C87MXH 44263497 IC50 > 10000 nM T78709 CT8MG3 44266611 Ki = 317 nM T78709 CFQ4L9 44266612 Ki = 338 nM T78709 C4QVN3 44266613 Ki = 49 nM T78709 C7AWM2 44266623 Ki = 10 nM T78709 CZ36NP 44266636 Ki = 16 nM T78709 CK0XI3 44266651 Ki = 4.9 nM T78709 CP52AC 44266663 Ki > 1000 nM T78709 C5RH3X 44266664 Ki < 1 nM T78709 C2Q4YJ 44266668 Ki = 16 nM T78709 CS6F3H 44266676 Ki = 1 nM T78709 CIO03X 44266677 Ki = 54 nM T78709 CW14OJ 44266678 Ki > 442 nM T78709 CN90JC 44266689 Ki = 252 nM T78709 CB2RF4 44266863 Ki = 4.5 nM T78709 CCP37Q 44267158 IC50 = 3019.95 nM T78709 CFEI56 44267161 IC50 = 512.86 nM T78709 CHU4L9 44267168 IC50 = 15848.93 nM T78709 CIZ5W7 44267181 IC50 = 234.42 nM T78709 CFE12G 44267205 IC50 = 15848.93 nM T78709 C5CPZ7 44267215 IC50 = 4168.69 nM T78709 CO65VL 44269006 Ki = 70.79 nM T78709 C0TP2Z 44269013 Ki = 79.43 nM T78709 CWR1Q3 44269487 Ki > 1000 nM T78709 CZ0YI5 44269492 Ki = 7 nM T78709 CLY2H7 44269511 Ki > 1000 nM T78709 C9QK2C 44269512 Ki = 611 nM T78709 CV0S8B 44269559 Ki = 12 nM T78709 CDC0H2 44269581 Ki = 28 nM T78709 C46WGB 44269582 Ki = 93 nM T78709 CE8NI2 44269606 Ki = 247 nM T78709 CGA1W5 44269820 Ki = 2000 nM T78709 C0C4QN 44269825 Ki = 1500 nM T78709 CIN1S4 44272400 IC50 = 4.571 nM T78709 C13QRS 44272402 IC50 = 72.44 nM T78709 CJ15FQ 44272419 IC50 = 9.12 nM T78709 CQ83VT 44274687 Ki = 2.2 nM T78709 C4MHT3 44274739 Ki = 470 nM T78709 CEY19W 44274740 Ki = 0.2 nM T78709 CD2KU5 44274871 Ki = 16 nM T78709 CNDU40 44274872 Ki = 1 nM T78709 C6U4TV 44274892 Ki = 1000 nM T78709 CC38DG 44274893 Ki = 317 nM T78709 CN01UL 44274899 Ki = 0.1 nM T78709 CLG10Y 44275015 Ki > 470 nM T78709 CU4KC2 44275016 Ki = 0.2 nM T78709 CBG61X 44275031 Ki = 236 nM T78709 C5SBH4 44275061 Ki = 1000 nM T78709 CSY7E4 44275135 Ki = 62 nM T78709 CVUE38 44275155 Ki = 54 nM T78709 CH3V9B 44275206 Ki = 442 nM T78709 CIRX69 44275207 Ki = 54 nM T78709 C86EDH 44275362 Ki = 105 nM T78709 CBV7O8 44275604 Ki = 6.4 nM T78709 CQ19YR 44275615 Ki = 304 nM T78709 CE60XZ 44275616 Ki = 80 nM T78709 C6JI7M 44275657 Ki = 104 nM T78709 CFA79L 44275658 Ki = 11 nM T78709 C1H0XC 44275766 Ki = 5.4 nM T78709 CNHE76 44276598 Ki = 170 nM T78709 CC2OD4 44278111 Ki > 10000 nM T78709 CRMA84 44278114 Ki > 10000 nM T78709 CF0Y4M 44278115 Ki = 3967.7 nM T78709 C08LZS 44279525 Ki = 0.96 nM T78709 C1OI7G 44279549 Ki = 5.8 nM T78709 CFWE96 44279550 Ki = 4 nM T78709 C7DR8P 44279889 Ki = 14 nM T78709 C51NLQ 44289248 Ki = 15.14 nM T78709 CWC49F 44289261 Ki = 6.31 nM T78709 C1JX5M 44289437 Ki = 10.96 nM T78709 CIM92E 44289525 Ki = 11.75 nM T78709 COQ53S 44290346 EC50 = 47.86 nM T78709 CU1S5W 44292309 IC50 = 46 nM T78709 C2C4UE 44292323 IC50 = 930 nM T78709 CM25WH 44292490 IC50 = 4 nM T78709 CGM6S1 44292505 IC50 = 710 nM T78709 C35JVN 44292507 IC50 = 840 nM T78709 CNKH68 44292523 IC50 = 64 nM T78709 C4KX1F 44292555 IC50 = 99 nM T78709 CM6A3I 44292629 IC50 = 460 nM T78709 CB0CD4 44292676 IC50 = 69 nM T78709 CLZ25G 44292706 IC50 = 210 nM T78709 C68SAH 44292707 IC50 = 1460 nM T78709 C0XYU8 44292776 IC50 = 87 nM T78709 CJK5G1 44292790 IC50 > 1000 nM T78709 CNQ82Z 44294182 Ki < 1000 nM T78709 C1IWT4 44296810 IC50 = 489.78 nM T78709 C8BXD4 44299396 Ki = 9.12 nM T78709 CV3PH7 44299504 Ki = 4.83 nM T78709 C0OX9M 44299511 Ki = 9.31 nM T78709 C59XUA 44299512 Ki = 29.4 nM T78709 C7U4DQ 44299513 Ki = 6.79 nM T78709 CJ0EQ1 44299524 Ki = 5.17 nM T78709 CWL48T 44299539 Ki = 7.64 nM T78709 C3QE4F 44299553 Ki = 6.07 nM T78709 CSTJ48 44299556 Ki = 7.21 nM T78709 COK1E4 44299569 Ki = 15.35 nM T78709 C14YCS 44299581 Ki = 7.5 nM T78709 CT48UN 44299643 Ki = 7.45 nM T78709 C2X0BS 44299664 Ki = 3.13 nM T78709 C0VXZ9 44299672 Ki = 1.44 nM T78709 CO6MJ9 44299681 Ki = 6.13 nM T78709 C2U0XO 44299682 Ki = 19.85 nM T78709 COCL75 44299716 Ki = 7.12 nM T78709 COI7M3 44299729 Ki = 1.89 nM T78709 C9K5QI 44299730 Ki = 4.7 nM T78709 CHZ3J7 44299764 Ki = 451.6 nM T78709 CH19QL 44299885 Ki = 14.15 nM T78709 CHD2X3 44299886 Ki = 27.83 nM T78709 C6T9BK 44299887 Ki = 22.6 nM T78709 CXYI48 44299888 Ki = 10.4 nM T78709 C9GX3Z 44299892 Ki = 12.66 nM T78709 CT74SG 44299914 Ki = 6.28 nM T78709 C89HGM 44299915 Ki = 3.09 nM T78709 CM8KV2 44300018 Ki = 4.24 nM T78709 CBSQ04 44300865 Ki = 790 nM T78709 CQ5A2E 44301054 Ki = 450 nM T78709 CEF72W 44305547 IC50 = 7762.47 nM T78709 CW07BA 44306007 IC50 = 457088.19 nM T78709 CKY68S 44309775 Ki = 941 nM T78709 C1TKV6 44309876 Ki = 540 nM T78709 C3L1OJ 44310701 Ki = 17 nM T78709 C8JP5T 44315098 Ki = 200 nM T78709 CN9ZV0 44315099 Ki = 17 nM T78709 C9BTW3 44315120 Ki = 130 nM T78709 CFB13Y 44315131 Ki = 41 nM T78709 CYVZ78 44315380 Ki = 32 nM T78709 C6AWP3 44315381 Ki = 26 nM T78709 C83WGQ 44315382 Ki = 49 nM T78709 CP9D6G 44315383 Ki = 85 nM T78709 CV4X1P 44315386 Ki = 15 nM T78709 C9G2KL 44315406 Ki = 7.6 nM T78709 C2HUA3 44315407 Ki = 21 nM T78709 CHJ1I7 44315426 Ki = 42 nM T78709 CFE15Q 44315427 Ki = 14 nM T78709 C8S5RH 44315436 Ki = 32 nM T78709 CL0Z3J 44315453 Ki = 23 nM T78709 CF3VK8 44315548 Ki = 7.9 nM T78709 C49OQD 44315568 Ki = 38 nM T78709 C7TCE9 44315569 Ki = 35 nM T78709 C1P0XE 44316740 Ki = 8.37 nM T78709 C62EYI 44316755 Ki = 14.45 nM T78709 CVKF37 44316789 Ki = 1.8 nM T78709 CFK6D0 44316790 Ki = 2.33 nM T78709 CGX14Y 44316815 Ki = 11.66 nM T78709 C2GKY9 44316828 Ki = 24.23 nM T78709 COM46U 44316963 Ki = 6.85 nM T78709 C65CRT 44316964 Ki = 0.98 nM T78709 C4M6VT 44316965 Ki = 11.75 nM T78709 C9TXA5 44316966 Ki = 16.48 nM T78709 C2PB8C 44317057 Ki = 2.98 nM T78709 C18BYV 44317081 Ki = 1.76 nM T78709 CLZH14 44317082 Ki = 5.67 nM T78709 CFY17P 44317084 Ki = 15.7 nM T78709 CXOP69 44317095 Ki = 5.26 nM T78709 C6E4UA 44317120 Ki = 4.23 nM T78709 CL78IT 44317121 Ki = 5.52 nM T78709 CTK8U7 44317134 Ki = 4.88 nM T78709 CBMS83 44317146 Ki = 3.09 nM T78709 C9Y4LX 44317147 Ki = 94.9 nM T78709 CV8WZ0 44318454 IC50 = 1584.89 nM T78709 CXJL56 44318842 IC50 > 1000 nM T78709 CHT83A 44320347 Ki = 3 nM T78709 C02LRC 44322770 Ki = 3.7 nM T78709 C40NAS 44322821 IC50 = 19.95 nM T78709 CZ7JF6 44322823 IC50 = 50.12 nM T78709 CSQT84 44322859 IC50 > 100 nM T78709 CR0DQ4 44322885 IC50 = 15.85 nM T78709 C5WL1J 44322886 IC50 = 1.585 nM T78709 C37UTX 44322916 IC50 = 1.995 nM T78709 C3C1OY 44322934 IC50 = 12.59 nM T78709 CJC37P 44322940 IC50 > 1000 nM T78709 C2LV3J 44322952 IC50 > 1000 nM T78709 C1MTR2 44322963 IC50 > 1000 nM T78709 C5R2NL 44322965 IC50 > 1000 nM T78709 C5UFN9 44323074 IC50 = 7.943 nM T78709 CTE2Y6 44323104 Ki = 1.84 nM T78709 CW2P4D 44323130 Ki = 1.43 nM T78709 CQ4C8I 44323137 Ki = 1.39 nM T78709 C3CZF1 44323147 IC50 = 7.943 nM T78709 CEH78W 44323156 IC50 = 125.89 nM T78709 CW7F6I 44323157 IC50 = 50.12 nM T78709 CLN5S4 44323161 IC50 = 15.85 nM T78709 CQI51B 44323162 IC50 = 5.012 nM T78709 CHG3F0 44323163 IC50 > 1000 nM T78709 CPB3U4 44323179 Ki = 1.82 nM T78709 CR14CB 44323200 IC50 > 1000 nM T78709 C9LUP6 44323231 IC50 = 3.981 nM T78709 CD26JI 44323253 IC50 = 1.259 nM T78709 CE7B0T 44323254 IC50 = 12.59 nM T78709 CE8VP0 44323267 IC50 > 1000 nM T78709 CW16JD 44324737 Ki > 1000 nM T78709 CA84SN 44324765 Ki > 1000 nM T78709 COA3H4 44324800 Ki = 475 nM T78709 CY04JW 44324972 Ki > 1000 nM T78709 CV56DM 44326256 Ki = 120 nM T78709 CV8A2N 44326257 Ki = 7.8 nM T78709 C2X9GN 44326324 Ki = 3.9 nM T78709 C2YZI8 44334603 Ki = 0.6 nM T78709 C1DH4T 44334637 Ki = 0.4 nM T78709 C6BJZ0 44335519 Ki = 92.6 nM T78709 C5JCR2 44335674 Ki = 19.6 nM T78709 CLG1Q8 44336170 EC50 = 0.78 nM T78709 C01UJW 44336554 EC50 > 100000 nM T78709 CS7NA2 44337678 Ki = 8 nM T78709 CU4F3W 44337731 Ki > 1000 nM T78709 CUT24A 44338900 Ki = 405 nM T78709 C03OMP 44342812 Ki = 6.7 nM T78709 C2VD8T 44342867 Ki = 32.9 nM T78709 CQ39UH 44342906 Ki = 45.4 nM T78709 C1LID6 44343052 Ki = 142 nM T78709 C7MLO1 44343055 Ki = 15.7 nM T78709 CMLA57 44343195 Ki = 391 nM T78709 CEA06L 44343196 Ki = 156 nM T78709 CD62CF 44345026 Ki = 860 nM T78709 C6N3XK 44345317 IC50 < 1000 nM T78709 CCU89V 44350664 Ki = 414.4 nM T78709 CJ14XP 44351290 Ki = 13.48 nM T78709 C2RU7Y 44351301 Ki = 9.42 nM T78709 CK0ME4 44351312 Ki = 9.2 nM T78709 C6NQ0M 44351330 Ki = 26.77 nM T78709 CT6Q4O 44351331 Ki = 4.06 nM T78709 C4Y6QD 44351334 Ki = 12.65 nM T78709 CHGF01 44351335 Ki = 12.35 nM T78709 CJX4D0 44351341 Ki = 23.15 nM T78709 CQ28XE 44351344 Ki = 15.65 nM T78709 C03RQI 44351345 Ki = 5.65 nM T78709 C43ZES 44351406 Ki = 7.11 nM T78709 C9Y8IW 44351426 Ki = 2.12 nM T78709 C5PZ7I 44351452 Ki = 20.2 nM T78709 CO5G7D 44351470 Ki = 14.35 nM T78709 CD0SK8 44351501 Ki = 10.52 nM T78709 C95TIX 44351508 Ki = 4.84 nM T78709 CZD3O8 44351509 Ki = 6.36 nM T78709 CS51MO 44351512 Ki = 28.1 nM T78709 C2D1RC 44351513 Ki = 19.38 nM T78709 CJ2ZT4 44351521 Ki = 104.63 nM T78709 CHGY49 44351527 Ki = 32 nM T78709 CIK31Q 44351535 Ki = 9.8 nM T78709 CX3ZL5 44351656 Ki = 71.7 nM T78709 CUXH48 44352308 Ki = 265 nM T78709 CH9F8G 44356232 Ki = 218.78 nM T78709 C3I9DE 44358574 Ki = 0.23 nM T78709 CJ80OW 44360984 Ki = 11 nM T78709 CS8K1A 44360992 Ki = 22 nM T78709 C3NZ7B 44361021 Ki = 15 nM T78709 CS3J6N 44363580 Ki > 100 nM T78709 C3LKN1 44364048 Ki = 1.995 nM T78709 C2MZ6D 44365404 Ki = 3.05 nM T78709 CSTQ01 44365426 Ki = 39 nM T78709 CFO5K8 44365439 Ki = 0.33 nM T78709 CV54RI 44365467 Ki = 16.7 nM T78709 CO4I2K 44365657 Ki = 5.87 nM T78709 CB0A1W 44365671 Ki = 0.81 nM T78709 C4AWE7 44365672 Ki = 1.53 nM T78709 C0RLY6 44365679 Ki = 1.6 nM T78709 CH26LQ 44365682 Ki = 127.7 nM T78709 CTE15U 44365700 Ki = 2.92 nM T78709 C40CAM 44365701 Ki = 61.6 nM T78709 C1M0OB 44365720 Ki = 307.1 nM T78709 CVU16E 44365728 Ki = 46 nM T78709 C10HST 44365811 Ki = 357 nM T78709 CPV96F 44367514 Ki = 1.5 nM T78709 C6CJ7S 44373641 Ki = 9.8 nM T78709 C1YIJ4 44373989 Ki = 3.8 nM T78709 CVL3U2 44374207 Ki = 41 nM T78709 CQ79MO 44374219 Ki = 11 nM T78709 CV8CP3 44374225 Ki = 2200 nM T78709 C04WKH 44374233 Ki = 37 nM T78709 CB2S7T 44374234 Ki = 1200 nM T78709 CH03ON 44374236 Ki = 7.6 nM T78709 CJ4A2U 44374299 Ki = 210 nM T78709 CD9QP8 44374649 Ki > 1786 nM T78709 C4BAI3 44374753 IC50 > 10000 nM T78709 CJ4KP3 44377759 Ki = 74 nM T78709 CE06VB 44377955 Ki = 0.89 nM T78709 C4VXQ1 44388858 Ki = 41 nM T78709 CTPG47 44388956 Ki = 115 nM T78709 CQ85AW 44389003 Ki > 2000 nM T78709 C8AG7U 44389016 Ki = 875 nM T78709 CV14HS 44389135 Ki = 194 nM T78709 CTZ7P5 44389374 Ki < 100 nM T78709 CC6XK1 44389508 Ki = 107.15 nM T78709 C6U3FH 44389522 Ki = 46.77 nM T78709 C74BRC 44389523 Ki = 16.6 nM T78709 C7DT6S 44391257 Ki = 0.5012 nM T78709 CV4PR8 44391267 Ki = 2.512 nM T78709 C0UEV5 44391270 Ki = 1.585 nM T78709 CL8G4N 44391284 Ki = 12.59 nM T78709 C35BYM 44391300 Ki = 1.259 nM T78709 C1PT7D 44391314 Ki = 1.585 nM T78709 CLZ83B 44391323 Ki = 1.995 nM T78709 C1XVH3 44391327 Ki = 10 nM T78709 C9P3WI 44391358 Ki = 7.943 nM T78709 C9XF0B 44391374 Ki = 100 nM T78709 CNO6S7 44391393 Ki = 6.31 nM T78709 C53UVJ 44393088 Ki > 100 nM T78709 C6WAK2 44393173 Ki = 87.1 nM T78709 CEO2W9 44393372 Ki = 27 nM T78709 CXP4Q7 44393393 Ki = 24 nM T78709 C6BZS0 44393403 Ki = 33 nM T78709 C86NED 44393411 Ki = 46 nM T78709 C9THO4 44393415 Ki = 10 nM T78709 CYOU64 44395296 Ki = 173.2 nM T78709 CECK89 44395347 Ki = 320 nM T78709 C3RV6T 44395741 Ki = 90.9 nM T78709 CN02LY 44395762 Ki = 240 nM T78709 CLH1T7 44395786 Ki = 160 nM T78709 C9K4SC 44395787 Ki = 310 nM T78709 C93XHA 44395809 Ki = 12 nM T78709 CTA27N 44395810 Ki = 860 nM T78709 C9A4NM 44395832 Ki = 11 nM T78709 C4B0OI 44397588 Ki = 794.33 nM T78709 C5FP0R 44397589 Ki = 1000 nM T78709 CE3G8U 44397670 Ki = 501.19 nM T78709 C1KA3F 44400359 Ki = 63.1 nM T78709 C0E5HY 44400500 Ki = 12 nM T78709 CO8EU5 44400519 Ki = 77 nM T78709 CRX12E 44400553 Ki = 14 nM T78709 CIU18E 44400585 Ki = 20 nM T78709 CV8K2W 44400594 Ki = 210 nM T78709 C84RNU 44400626 Ki = 27 nM T78709 CY94SF 44400674 Ki = 0.5 nM T78709 C9THQ3 44402868 Ki = 501.19 nM T78709 C1EI5Q 44402869 Ki = 79.43 nM T78709 CV0PC9 44402870 Ki = 50.12 nM T78709 CV15IH 44402871 Ki = 1584.89 nM T78709 CG1WU9 44402876 Ki = 12.59 nM T78709 C6WNI4 44402877 Ki = 501.19 nM T78709 CDL1F6 44402878 Ki = 1000 nM T78709 C1B4QL 44403095 Ki = 52.5 nM T78709 C1YL7Z 44403098 Ki = 1079 nM T78709 CFV98A 44403101 Ki = 405 nM T78709 C6OY9S 44403102 Ki = 382 nM T78709 CH4SX6 44403105 Ki = 882 nM T78709 C12FIH 44403106 Ki = 15.4 nM T78709 CQ4U2P 44403210 Ki = 15 nM T78709 CKE6T4 44403213 Ki = 60 nM T78709 CAJX39 44403214 Ki = 22 nM T78709 C61CNS 44403219 Ki = 28 nM T78709 C5AE9L 44403220 Ki = 24 nM T78709 CC6XM4 44403224 Ki = 30 nM T78709 C6JB4M 44403225 Ki = 51 nM T78709 CGE52H 44403232 Ki = 120 nM T78709 CI0WG5 44404225 Ki = 0.7943 nM T78709 C7FAW3 44404229 Ki = 1 nM T78709 C0MXR4 44404230 Ki = 10 nM T78709 C7OD6Q 44404236 Ki = 5.012 nM T78709 C5W2KR 44404240 Ki = 3.162 nM T78709 CI50CY 44404241 Ki = 3.981 nM T78709 CF69DU 44404244 Ki = 5.012 nM T78709 CE0NI6 44404245 Ki = 6.31 nM T78709 CLW3P7 44404249 Ki = 0.3162 nM T78709 CF8LN5 44404253 Ki = 1.259 nM T78709 C3LI6E 44404258 Ki = 3.162 nM T78709 C2NH8G 44404260 Ki = 6.31 nM T78709 C7R5HU 44404264 Ki = 31.62 nM T78709 CVTZ13 44404268 Ki = 1.585 nM T78709 C18ISW 44404272 Ki = 1.259 nM T78709 C4LKC1 44404394 Ki = 335 nM T78709 C3EJ4G 44404396 Ki = 315 nM T78709 C4Q2BS 44404551 Ki = 45 nM T78709 C7W3BP 44405573 Ki = 4.1 nM T78709 CV9IR7 44405574 Ki = 0.9 nM T78709 CFG72V 44405575 Ki = 1.9 nM T78709 C8WSZ2 44405586 Ki = 0.7 nM T78709 CEJ0C3 44405587 Ki = 2.5 nM T78709 C4DK0U 44405655 Ki = 5.6 nM T78709 C28WCH 44405665 Ki = 103.9 nM T78709 CS7ZD5 44405666 Ki = 0.6 nM T78709 CIH9J0 44405669 Ki = 0.4 nM T78709 CVZO38 44405677 Ki = 18.8 nM T78709 CMK32Z 44405701 Ki = 1.5 nM T78709 CZK5L6 44405702 Ki = 0.9 nM T78709 CO7G3W 44405725 Ki = 2.5 nM T78709 CU1VL9 44405726 Ki = 2.5 nM T78709 CO1P3W 44405730 Ki = 0.3 nM T78709 C65PBE 44405930 Ki = 113.4 nM T78709 CBGH16 44405935 Ki = 157.3 nM T78709 CF4S3Y 44405965 Ki = 1540 nM T78709 CT3Z8U 44405980 Ki = 1030 nM T78709 CQ7RI8 44405981 Ki = 19.1 nM T78709 C0BI5F 44405985 Ki = 64.9 nM T78709 C1FZE7 44405991 Ki = 295.1 nM T78709 C4NC8M 44405995 Ki = 1450 nM T78709 CVM1Y5 44406002 Ki = 333.34 nM T78709 C0R5VL 44406003 Ki = 1815 nM T78709 C90NQJ 44406012 Ki = 401.3 nM T78709 CL5C9T 44406077 Ki = 1070 nM T78709 CPNT73 44408681 Ki = 2.81 nM T78709 C81GYD 44408682 Ki = 7.25 nM T78709 C9J2VU 44408685 Ki = 30.21 nM T78709 CH9MC5 44408702 Ki = 12.76 nM T78709 C9IPV4 44408784 Ki = 103 nM T78709 C54EOX 44408852 Ki = 7.14 nM T78709 CCM7A1 44408853 Ki = 75.18 nM T78709 CM41IO 44408882 Ki = 8.15 nM T78709 CEM05A 44408883 Ki = 5.86 nM T78709 C5CKA7 44408888 Ki = 8.46 nM T78709 CUM50D 44408890 Ki = 6.91 nM T78709 C9R2BF 44408942 Ki = 15.31 nM T78709 CU15IW 44408946 Ki = 10.98 nM T78709 CG87PW 44409290 Ki > 720 nM T78709 CO4SX2 44412809 Ki = 230 nM T78709 C05FOC 44412810 Ki = 260 nM T78709 CILZ93 44412825 Ki = 63 nM T78709 CB1TC6 44412826 Ki = 69 nM T78709 C32NFQ 44412838 Ki = 40 nM T78709 CR5D1B 44412906 Ki = 40 nM T78709 C95HRZ 44412907 Ki = 480 nM T78709 CN02QD 44412913 Ki = 25 nM T78709 CHRS85 44412928 Ki = 170 nM T78709 CWD97B 44412932 Ki = 17 nM T78709 CC7Y5W 44412934 Ki = 24 nM T78709 COJ75S 44412935 Ki = 11 nM T78709 C9LS4E 44412965 Ki = 12 nM T78709 CS1GP5 44412966 Ki = 27 nM T78709 CFKI28 44412969 Ki = 4 nM T78709 CVDM51 44412991 Ki = 12 nM T78709 CHW6K9 44413006 Ki = 17 nM T78709 CFY4W8 44413015 Ki = 50 nM T78709 CAJI08 44413016 Ki = 17 nM T78709 CV8SQ0 44413025 Ki = 18 nM T78709 CC0UA4 44413026 Ki = 9 nM T78709 CR4Z8C 44413037 Ki = 15 nM T78709 CJN6P4 44427818 Ki = 6.71 nM T78709 CW3F5H 44427820 Ki = 29.7 nM T78709 CYLO03 44427821 Ki = 309 nM T78709 CJY9L5 44427822 Ki = 92 nM T78709 CO46HS 44427823 Ki = 60.6 nM T78709 CFG0S3 44427824 Ki = 666 nM T78709 C7PK0M 44427825 Ki = 21.7 nM T78709 CDV6A3 44427826 Ki = 71.8 nM T78709 C65ZXC 44427827 Ki = 34.3 nM T78709 CZ0X7U 44427829 Ki = 1810 nM T78709 C9U8YT 44427831 Ki = 36.2 nM T78709 C0C8AH 44427835 Ki = 117 nM T78709 C8EV3G 44427836 Ki = 15.1 nM T78709 CS9ND5 44427841 Ki = 59 nM T78709 COV6N3 44427842 Ki = 982 nM T78709 C6JK5A 44431532 Ki = 115 nM T78709 C5LNH6 44431533 Ki = 105 nM T78709 CLX73C 44431534 Ki = 307 nM T78709 C4P5XG 44431536 Ki = 26 nM T78709 CYPR70 44431537 Ki = 16 nM T78709 CVX7A6 44433249 Ki = 40.6 nM T78709 C5P4OW 44433250 Ki = 3.89 nM T78709 C3YV6I 44433251 Ki = 11.2 nM T78709 C0AT6Q 44433252 Ki = 26.1 nM T78709 C1SK2A 44433253 Ki = 18.3 nM T78709 COH61M 44433254 Ki = 1450 nM T78709 CPO7H6 44433255 Ki = 868 nM T78709 C8YPF6 44433257 Ki = 872 nM T78709 CZLT14 44433258 Ki = 125 nM T78709 CP0F4L 44433280 Ki > 3000 nM T78709 C4TN2F 44433281 Ki = 833 nM T78709 C6W8GQ 44433303 Ki = 76.1 nM T78709 CZK39E 44437329 Ki = 1.7 nM T78709 CKZF16 44439165 Ki = 2.512 nM T78709 CA4HZ3 44439167 Ki = 10 nM T78709 CT0C4I 44443093 Ki = 1.585 nM T78709 C8E1AC 44443094 Ki = 1.259 nM T78709 CZ6BK9 44443095 Ki = 0.2512 nM T78709 CV5T2C 44443096 Ki = 1.259 nM T78709 CT1S6L 44443097 Ki = 1.995 nM T78709 CF1V8O 44443098 Ki = 3.981 nM T78709 CHZ48Q 44443101 Ki = 1.259 nM T78709 CQ53TV 44443130 Ki = 7.943 nM T78709 CEZ6U8 44443131 Ki = 3.162 nM T78709 CN4XZ6 44443132 Ki = 2.512 nM T78709 C5RVE0 44446999 Ki = 4.9 nM T78709 C9E0FL 44447001 Ki = 2 nM T78709 CSJ4U5 44447002 Ki = 5 nM T78709 CL87PU 44447003 Ki = 5.5 nM T78709 CCD6B5 44447005 Ki = 12 nM T78709 CBH65G 44447007 Ki = 12 nM T78709 C8CF7X 44447008 Ki = 41.8 nM T78709 CN3EH7 44447010 Ki = 28.1 nM T78709 CYWP06 44447012 Ki = 56 nM T78709 C41KNM 44447013 Ki = 66.7 nM T78709 CE12BC 44447015 Ki = 4.5 nM T78709 CUD31L 44447018 Ki = 20.9 nM T78709 CNLX79 44447028 Ki = 37.2 nM T78709 CM8K1H 44447039 Ki = 7.9 nM T78709 C5IJW2 44447059 Ki = 6.5 nM T78709 CHXF10 44447061 Ki = 1 nM T78709 CG93OH 44447063 Ki = 2 nM T78709 C9KJR2 44447065 Ki = 2 nM T78709 C5QK8Z 44447067 Ki = 2 nM T78709 C7A6RP 44447068 Ki = 1 nM T78709 CM8P9A 44447070 Ki = 7.8 nM T78709 CK4HA6 44447072 Ki = 7.7 nM T78709 C2S6HQ 44448054 Ki = 373 nM T78709 C3Z7FI 44451927 IC50 = 960 nM T78709 C57SBC 44451980 IC50 = 120 nM T78709 CEST18 44451982 IC50 = 220 nM T78709 CRN4F8 44452007 IC50 = 370 nM T78709 CG1C6X 44452142 IC50 = 140 nM T78709 CVAU93 44452222 IC50 = 500 nM T78709 C0B3LC 44452327 IC50 = 400 nM T78709 CZL97F 44455426 Ki > 10000 nM T78709 CYS7T4 44455943 Ki = 765 nM T78709 C6BFI0 44456033 Ki = 95.2 nM T78709 CG91RD 44456395 Ki = 339 nM T78709 C12XGE 44456400 Ki > 10000 nM T78709 CZ1BM3 44461160 EC50 = 251.19 nM T78709 CD5L8N 44461162 EC50 = 12.59 nM T78709 CQ2IX7 44461606 IC50 > 1000 nM T78709 C4DL5C 44469677 IC50 = 1 nM T78709 CM5EY8 44474470 IC50 > 1000 nM T78709 C8UON6 44474625 IC50 > 1000 nM T78709 C6HVU1 44474629 IC50 > 10000 nM T78709 CE2Z8S 44474631 IC50 > 10000 nM T78709 C8LA4W 44474797 IC50 > 1000 nM T78709 CJ10OZ 44531812 Ki = 3090 nM T78709 C4SX7H 44537919 Ki = 105 nM T78709 CVD14L 44537925 Ki = 133 nM T78709 C3D4HR 44537940 Ki > 5000 nM T78709 CT85QK 44538690 Ki = 1330 nM T78709 C4LUK7 44549156 Ki = 7.244 nM T78709 CJ7U3K 44554227 Ki > 5000 nM T78709 CM0I1P 44554393 Ki > 5000 nM T78709 CNHA47 44554395 Ki = 1780 nM T78709 C6WV2P 44559406 IC50 > 10000 nM T78709 CB23PH 44560995 Ki = 19 nM T78709 C0N1LV 44561105 IC50 = 2.3 nM T78709 C7MAT0 44568331 Ki = 1.7 nM T78709 CVA67X 44568347 Ki = 450 nM T78709 CQF70H 44568357 Ki = 3 nM T78709 C6LK9P 44568358 Ki = 3.6 nM T78709 CIB94E 44568385 Ki = 8.3 nM T78709 COE94C 44568461 Ki = 9.1 nM T78709 CI0F2C 44568462 Ki = 42.6 nM T78709 CAR23X 44568818 Ki = 37.15 nM T78709 CAO31F 44568917 Ki = 7.586 nM T78709 CE3GV8 44568918 Ki = 229.09 nM T78709 C9LP7Z 44575219 EC50 = 9000 nM T78709 CZO5Y8 44580740 Ki = 3.162 nM T78709 C4N6PM 44580741 Ki = 1.585 nM T78709 C0XVL5 44580783 Ki = 125.89 nM T78709 C4SD7P 44580784 Ki = 0.2512 nM T78709 CNOU35 44581235 Ki = 7.943 nM T78709 CO6E5K 44581260 Ki = 5.012 nM T78709 CS6HG9 44581603 Ki = 6.31 nM T78709 C1HAQ2 44581604 Ki = 12.59 nM T78709 CRCH48 44582675 Ki > 10000 nM T78709 CEJ4R8 44582676 Ki = 1681 nM T78709 CZGP86 44582677 Ki > 10000 nM T78709 C5QB4K 44582678 Ki > 10000 nM T78709 C01RCI 44582705 Ki = 1883 nM T78709 CXL25V 44582706 Ki > 10000 nM T78709 C8MR1X 44582707 Ki = 1723 nM T78709 C4IT1N 44582708 Ki = 991 nM T78709 CSF39B 44588698 Ki = 630.96 nM T78709 C60NYB 44588704 Ki = 0.66 nM T78709 C7SKM1 44588720 Ki = 398.11 nM T78709 CI6SO1 44588721 Ki = 50.12 nM T78709 CB14UQ 44588722 Ki = 79.43 nM T78709 CNK64D 44588742 Ki = 158.49 nM T78709 CAT73D 44588743 Ki > 10000 nM T78709 C6DK3E 44588744 Ki > 1584.89 nM T78709 C9BO7K 44588745 Ki = 316.23 nM T78709 CD2CU8 44588771 Ki > 10000 nM T78709 CDIQ25 44588772 Ki = 501.19 nM T78709 CB27TM 44589076 Ki = 0.93 nM T78709 C34YST 44591228 Ki = 75.3 nM T78709 CKV67Q 44591229 Ki = 21.3 nM T78709 C6A2QJ 44591230 Ki = 7.4 nM T78709 CZKV93 44591244 Ki = 32 nM T78709 C1U2NH 44591245 Ki = 5.2 nM T78709 CF20JZ 44591246 Ki = 23.6 nM T78709 CB7QV5 44591259 Ki = 10.4 nM T78709 CQS54L 44591260 Ki = 26.6 nM T78709 CM72EB 44591261 Ki = 35.1 nM T78709 CS56IQ 44591262 Ki = 64.5 nM T78709 C5WRT1 44591263 Ki = 37.8 nM T78709 C1T0XN 44591280 Ki = 38.5 nM T78709 CIGM43 44591281 Ki = 42.5 nM T78709 C1EAR6 44591282 Ki = 40.2 nM T78709 C5E7HO 44591283 Ki = 3420 nM T78709 CZUX15 44591284 Ki = 780 nM T78709 C4VI7E 44591316 Ki = 4450 nM T78709 C3B0GO 44591317 EC50 = 51.4 nM T78709 CW9YA7 44591318 EC50 = 65 nM T78709 CK7XJ0 44591319 EC50 = 40.7 nM T78709 CB0S4Z 44592109 IC50 = 5248.07 nM T78709 C4EH6O 44592207 Ki = 0.2512 nM T78709 CZ5I1N 44592208 Ki > 3162.28 nM T78709 CKM8T7 44592209 Ki = 0.1259 nM T78709 CDJ32U 44592249 Ki = 0.631 nM T78709 CS2FL4 44592250 Ki = 0.1 nM T78709 CL17WU 44592251 Ki = 0.631 nM T78709 CJCL64 44592252 Ki = 0.5012 nM T78709 CM0I3E 44592294 Ki = 0.3162 nM T78709 CQ04EG 44592295 Ki = 0.3981 nM T78709 C65XQL 44592296 Ki = 0.1995 nM T78709 CEB2S1 44592297 Ki = 0.1995 nM T78709 CP51QS 44592332 Ki = 1.585 nM T78709 CD2Z4J 44592333 Ki = 1.995 nM T78709 C7NCT2 44592334 Ki = 6.31 nM T78709 CHY20X 44592335 Ki = 1.585 nM T78709 C5H7XK 44592371 Ki = 3.162 nM T78709 CR8T7B 44593415 Ki = 2.8 nM T78709 C1SN7Y 44593709 Ki = 0.25 nM T78709 CZ0W1I 44593711 Ki = 50.12 nM T78709 CHD0R7 44593712 Ki = 1.98 nM T78709 CPK6N9 44593714 Ki = 1.73 nM T78709 C5HSO3 44593715 Ki = 31.4 nM T78709 CAXK49 44593716 Ki = 7.34 nM T78709 C4WBK1 44593717 Ki = 9.48 nM T78709 CF4Q5M 44593729 Ki = 11.2 nM T78709 C4Y6SW 44598639 Ki = 44 nM T78709 CE9NU2 44598680 Ki = 116 nM T78709 C40ZMK 44598681 Ki = 6.8 nM T78709 CO7K4W 44598682 Ki = 0.67 nM T78709 C96QRP 44598683 Ki = 15 nM T78709 C62CAY 44598684 Ki = 0.47 nM T78709 C52QLW 44598685 Ki = 0.5 nM T78709 C5S3IT 44598725 Ki = 7.8 nM T78709 CXK8A2 44598726 Ki = 73 nM T78709 C0LS9C 44598727 Ki = 29 nM T78709 CL1J3B 44598728 Ki = 54 nM T78709 C67KZG 44608359 EC50 > 10000 nM T78709 CW0RU3 45102635 Ki = 1 nM T78709 C0DLU3 45109862 IC50 = 117 nM T78709 CGB2Z0 45113400 Ki = 7 nM T78709 CMJ1U7 45266443 EC50 > 100000 nM T78709 CEK5G3 45277221 Ki = 63.3 nM T78709 CL3I7B 45277224 Ki = 27 nM T78709 CI4O0A 45277387 Ki = 27.3 nM T78709 CHZ70D 45277559 Ki = 3.76 nM T78709 CZ71RN 45278805 IC50 = 54 nM T78709 CZN6M7 45278882 IC50 = 94 nM T78709 CC86HS 45481874 Ki = 799 nM T78709 C7MO3G 45481875 Ki = 85 nM T78709 CP4OS2 45481876 Ki = 98 nM T78709 CRL6D2 45481877 Ki = 648 nM T78709 C7S9HJ 45481888 Ki = 133 nM T78709 C0HPW1 45481889 Ki = 235 nM T78709 C47HZI 45481890 Ki = 457 nM T78709 CB7SG4 45481891 Ki = 381 nM T78709 C0CHF4 45482789 IC50 = 3600 nM T78709 CZ8G9V 45482876 Ki = 53.7 nM T78709 CX7BE9 45482877 Ki = 204.17 nM T78709 CR80QO 45482879 Ki = 10.96 nM T78709 C9E3JI 45482881 Ki = 100 nM T78709 C1I4FV 45482884 Ki = 416.87 nM T78709 C36LXH 45482890 Ki = 234.42 nM T78709 C6ILK5 45482891 Ki = 398.11 nM T78709 CEOX52 45482892 Ki = 50.12 nM T78709 C1SR9M 45482893 Ki = 30.2 nM T78709 C9LSN3 45482900 Ki = 42.66 nM T78709 C97JBX 45483401 Ki > 4570 nM T78709 C9K4XC 45483416 Ki = 2210 nM T78709 CZQ6H8 45483429 Ki > 1000 nM T78709 C3HAF8 45483430 Ki = 1160 nM T78709 CG2SM9 45483458 Ki = 9 nM T78709 CFM9P8 45483465 Ki = 4 nM T78709 C5DS3M 45483506 Ki = 101 nM T78709 CHCA47 45483511 Ki = 466 nM T78709 C05PBD 46176231 Ki = 66 nM T78709 CI3WX2 46176232 Ki = 279 nM T78709 C4XRY7 46176233 Ki = 35 nM T78709 C4WJ0Z 46176312 Ki = 45 nM T78709 CNW60S 46180190 Ki = 626 nM T78709 C5CET8 46180192 Ki = 12 nM T78709 CEW06P 46180193 Ki = 135 nM T78709 C9PBQ4 46180194 Ki = 6.7 nM T78709 CP8RF4 46180256 Ki = 14 nM T78709 CG8UK9 46180257 Ki = 29 nM T78709 CO7SA6 46180258 Ki = 66 nM T78709 CSY63N 46180259 Ki = 144 nM T78709 C64TDV 46180261 Ki = 373 nM T78709 CQNC52 46180262 Ki > 10000 nM T78709 CBM9O6 46180325 Ki = 149 nM T78709 CP7Y5E 46180326 Ki = 11 nM T78709 C1J3VH 46180327 Ki = 793 nM T78709 CUI5T0 46180329 Ki > 10000 nM T78709 C4Z5LD 46180330 Ki = 340 nM T78709 C73KNC 46180331 Ki = 630 nM T78709 CXQ7G5 46180393 Ki = 90 nM T78709 CHN09F 46180394 Ki = 55 nM T78709 CMS7T5 46180395 Ki = 125 nM T78709 C62FUY 46180396 Ki = 320 nM T78709 C10OKI 46180397 Ki = 510 nM T78709 CM4R8A 46180398 Ki = 3.1 nM T78709 CC7N8T 46180399 IC50 = 18 nM T78709 C62BEZ 46224739 Ki = 19 nM T78709 C34ZXM 46225029 Ki > 10000 nM T78709 C5LTG9 46225164 Ki = 1220 nM T78709 CQT3G4 46225165 Ki = 22 nM T78709 C5OC1A 46225166 Ki = 2 nM T78709 C1AM8J 46225207 Ki = 3 nM T78709 CNQ10M 46225208 Ki = 101 nM T78709 C8Z0DR 46225263 Ki = 85 nM T78709 CYE41P 46225264 EC50 = 22 nM T78709 C2H1PN 46225309 Ki = 4 nM T78709 CUR54A 46225310 Ki = 22 nM T78709 CY82LR 46227396 IC50 > 1000 nM T78709 C06QIT 46227754 EC50 = 25 nM T78709 C30ZIR 46227757 Ki = 23 nM T78709 C4YLZ1 46227762 Ki = 13 nM T78709 C08ZOG 46227770 Ki = 6 nM T78709 CN4HT2 46230756 Ki = 17 nM T78709 CGD6E4 46231118 Ki = 12 nM T78709 CEMB09 46231492 Ki = 12.7 nM T78709 C23JYW 46238348 Ki = 0.79 nM T78709 C42SVX 46700866 IC50 = 1200 nM T78709 CD0K6E 46700867 IC50 = 2100 nM T78709 C5TC2S 46830335 IC50 > 10000 nM T78709 C1K7FL 46830336 IC50 > 10000 nM T78709 C1N4KX 46842383 IC50 > 10000 nM T78709 C0ABR3 46846073 Ki = 2.188 nM T78709 CC62SX 46866711 IC50 = 298 nM T78709 C7ZEI6 46881382 Ki = 0.1288 nM T78709 CN0Q2A 46881443 Ki = 2.63 nM T78709 CGX02N 46881444 Ki = 7.943 nM T78709 C2MC4K 46881463 EC50 = 794.33 nM T78709 CSQ4C9 46881468 EC50 = 3162.28 nM T78709 C4U6RH 46881493 Ki = 8.318 nM T78709 CV7R9S 46881494 Ki = 1.023 nM T78709 C24QFO 46882032 Ki > 1000 nM T78709 C3GQW6 46882033 Ki = 28.84 nM T78709 CPG6U5 46882034 Ki = 1.698 nM T78709 CYB37P 46882085 Ki = 0.8913 nM T78709 CD8CX3 46882086 Ki > 1000 nM T78709 C57GAO 46882087 Ki = 97.72 nM T78709 CV3QW9 46882088 Ki = 7.586 nM T78709 CB8GE1 46884818 IC50 > 10000 nM T78709 C4MQ0A 46884856 IC50 > 10000 nM T78709 CCNT25 46884898 IC50 > 10000 nM T78709 C3MSG2 46885027 IC50 > 10000 nM T78709 CB7XI0 46885213 IC50 > 10000 nM T78709 COH48X 46886853 Ki = 371.54 nM T78709 CBG61I 46886861 Ki = 1445.44 nM T78709 C05KPX 46886862 Ki = 9.333 nM T78709 C1JSH9 46899637 Ki = 0.1259 nM T78709 C3MSL0 46899638 Ki = 0.1585 nM T78709 CV3LP2 46899639 Ki = 0.1259 nM T78709 CGHZ15 46899640 Ki = 0.3981 nM T78709 CN9FC3 46900150 Ki = 0.1259 nM T78709 C40ZJO 46900451 Ki = 0.1995 nM T78709 CNC02A 46900453 Ki = 0.1995 nM T78709 CTCH14 46900455 Ki = 0.1585 nM T78709 CP41AQ 46900457 Ki = 0.1995 nM T78709 CR3L4I 46900459 Ki = 0.07943 nM T78709 CK17PA 46900606 Ki = 0.07943 nM T78709 CQ2K1C 46900608 Ki = 0.5012 nM T78709 C5ZT1B 46900610 Ki = 0.631 nM T78709 C1NAX4 46900612 Ki = 0.3162 nM T78709 CT0SQ2 46900614 Ki = 1.585 nM T78709 CXD9S3 46900776 Ki = 0.1585 nM T78709 C8I7SJ 46900778 Ki = 1 nM T78709 C7QDM9 46900782 Ki = 0.1995 nM T78709 C15FMY 46900954 Ki = 0.1259 nM T78709 C8W1FU 46900956 Ki = 0.1585 nM T78709 CH35BV 46900958 Ki = 0.2512 nM T78709 CA75HK 46914485 Ki = 806 nM T78709 C9D7UW 46914486 Ki = 373 nM T78709 COB4R0 46914487 Ki = 2192 nM T78709 C4JZR8 46914620 Ki = 468 nM T78709 C4JIP7 46914621 Ki = 1720 nM T78709 CZ5TS4 46914771 Ki = 3339 nM T78709 C1LY6Z 46914772 Ki = 3251 nM T78709 C3XE4P 46914773 Ki = 469 nM T78709 C2E6UX 46914774 Ki = 2458 nM T78709 CT36AF 46914775 Ki = 774 nM T78709 CW74CK 46914776 Ki = 4722 nM T78709 CLC27S 46914777 Ki = 3383 nM T78709 CAT12G 46914926 Ki = 599 nM T78709 CE6SQ2 46914927 Ki = 3300 nM T78709 C7FX8L 46931072 Ki = 349 nM T78709 CZDN92 46934426 Ki = 54 nM T78709 C4VG2E 46934427 Ki = 9.62 nM T78709 CUTX67 46934428 IC50 > 1000 nM T78709 CI4XZ1 46934637 Ki = 5.129 nM T78709 CK1Z0M 46934639 Ki = 5.248 nM T78709 CU0TB9 46934641 Ki = 7.244 nM T78709 CR6JV7 46934643 Ki = 5.623 nM T78709 C14ZLO 46934645 Ki = 25.7 nM T78709 C2N9JZ 46934787 Ki = 5.129 nM T78709 CI4U0L 46934789 Ki = 44.67 nM T78709 C8HVG6 46934791 Ki = 3.162 nM T78709 CA51JI 46934793 Ki = 1.259 nM T78709 CB4Z7D 46934945 Ki = 2.63 nM T78709 C6J4TV 46946859 Ki = 0.151 nM T78709 C8V5MJ 46947455 Ki = 2 nM T78709 CY28OS 47556338 Ki = 1551 nM T78709 C4CL9S 49780599 EC50 = 13 nM T78709 C0F4ZA 49780600 EC50 = 8.6 nM T78709 CR61PL 49780603 EC50 = 6.6 nM T78709 CD42FE 49781265 EC50 = 270 nM T78709 C4TP1Q 49781928 EC50 = 52 nM T78709 C2YAD4 49781933 EC50 = 11 nM T78709 CVGW32 49782156 EC50 = 26 nM T78709 C2TGP4 49782388 EC50 = 36 nM T78709 CF2Z7T 49782389 EC50 = 100 nM T78709 C2LZJ0 49783209 Ki = 300 nM T78709 C57SMG 49783415 Ki > 10000 nM T78709 C0TG6I 49783419 Ki > 10000 nM T78709 COE79D 49836152 IC50 = 59.3 nM T78709 C6IN7B 49836154 IC50 > 100 nM T78709 C28CKM 49836301 Ki = 35.48 nM T78709 C5JO6E 49836302 Ki > 10000 nM T78709 C9TNO4 49836303 Ki = 6.026 nM T78709 CR40BA 49836386 IC50 = 1300 nM T78709 C0M5XC 49836496 IC50 = 1100 nM T78709 C8JQ4O 49837354 EC50 = 2.5 nM T78709 CN0MO8 49837461 IC50 < 10 nM T78709 CHB1I9 49837652 IC50 < 10 nM T78709 CG64FA 49837758 IC50 = 96.4 nM T78709 C3OHN0 49850566 Ki = 3.162 nM T78709 C4R2YS 49850567 Ki = 0.5012 nM T78709 CSGQ38 49850568 Ki = 0.7943 nM T78709 C8P5KH 49850569 Ki = 0.3981 nM T78709 C07JTU 49850570 Ki = 1.995 nM T78709 C6FP9W 49850571 Ki = 5.012 nM T78709 C3BVK5 49850668 Ki = 7.943 nM T78709 C6P3RH 49850669 Ki = 3.162 nM T78709 CGYT84 49850670 Ki = 3.981 nM T78709 C6Y3DW 49850671 Ki = 2.512 nM T78709 CK68QR 49850672 Ki = 0.3981 nM T78709 CI6O9A 49850673 Ki = 1.259 nM T78709 COFA76 49850768 Ki = 1.995 nM T78709 C4IX5R 49850769 Ki = 3.162 nM T78709 CXLT59 49850770 Ki = 2.512 nM T78709 C48DOX 49850771 Ki = 3.162 nM T78709 CN5XR1 49850772 Ki = 0.5012 nM T78709 CR4EZ0 49850870 Ki = 0.7943 nM T78709 C5K4EC 49850872 Ki = 1 nM T78709 C8AW0R 49850874 Ki = 1 nM T78709 CB2K6D 49850877 Ki = 0.631 nM T78709 C85KPE 49850980 Ki = 1.259 nM T78709 C5U3YD 49850982 Ki = 2.512 nM T78709 CV62IZ 49850984 Ki = 1.995 nM T78709 CED9V6 49852000 Ki = 1.585 nM T78709 CA0PW5 49852001 Ki = 1.995 nM T78709 C5S6BY 49852002 Ki = 1.995 nM T78709 C13ZTD 49852003 Ki = 6.31 nM T78709 CK17IE 49852105 Ki = 15.85 nM T78709 C6OQV2 49862237 Ki = 103 nM T78709 C6IW4Q 49862238 Ki > 1000 nM T78709 CDHY90 49864027 Ki = 2439 nM T78709 C9KIU1 49864289 IC50 = 672 nM T78709 CHO9C0 49864292 IC50 = 280 nM T78709 C8TB6G 49864336 Ki = 62 nM T78709 C5N8ML 49864359 Ki = 27.4 nM T78709 C15NIO 49864360 Ki = 102 nM T78709 C90MTG 49864602 IC50 = 3399 nM T78709 C5BCS4 49864722 IC50 = 95 nM T78709 CKZO79 49864723 IC50 = 3756 nM T78709 C74LZS 49864724 IC50 = 485 nM T78709 C2RY0J 50878551 Ki = 19 nM T78709 C1W6TV 50898777 Ki > 10000 nM T78709 CXMZ73 50898778 Ki > 10000 nM T78709 C67IRJ 50908804 Ki = 1.585 nM T78709 CLOB24 50908805 Ki = 1.259 nM T78709 CA89QH 50914389 Ki = 32.8 nM T78709 CX48AD 51002362 EC50 > 10000 nM T78709 C6LVM3 51003382 Ki = 3 nM T78709 CIW56N 51003383 Ki = 3 nM T78709 C8TA1J 51003550 IC50 = 1598 nM T78709 CQ1UJ7 51003551 IC50 = 1210 nM T78709 CGMI37 51003586 IC50 = 999 nM T78709 CE4KP1 51050257 Ki > 10000 nM T78709 C2HGK8 51122451 Ki = 30 nM T78709 CIWA18 52938727 Ki = 7.59 nM T78709 C6XY8V 52938728 Ki = 9.68 nM T78709 C9C0NB 52940734 Ki = 17.5 nM T78709 CLW3B0 52940951 Ki = 31.62 nM T78709 CWYS78 52941004 Ki = 5.012 nM T78709 CE0X9W 52941056 Ki = 7.943 nM T78709 C0UXM7 52941358 Ki = 2.09 nM T78709 CTM81E 52941423 Ki = 2.61 nM T78709 C40WVE 52941624 Ki = 2.512 nM T78709 CV7HZ6 52942047 Ki = 6.918 nM T78709 C5Y3VS 52942152 Ki = 15.85 nM T78709 CX9AF4 52942551 Ki = 0.3981 nM T78709 CE6R7D 52942615 Ki = 0.615 nM T78709 CR0G5U 52942644 Ki = 0.631 nM T78709 CX2E5H 52942854 Ki = 13.4 nM T78709 CU8WA5 52942916 Ki = 0.838 nM T78709 CO9J6M 52943356 Ki = 3.981 nM T78709 CLJ70C 52943589 EC50 = 32 nM T78709 CCF97B 52943811 Ki = 1 nM T78709 C2FG9O 52943861 Ki = 0.3981 nM T78709 C9G4CI 52943891 Ki = 1.259 nM T78709 C9RD4F 52944256 Ki = 35 nM T78709 CBU2Z6 52944379 Ki = 0.67 nM T78709 CRL3P0 52944615 Ki = 31.62 nM T78709 C4N6ET 52944674 Ki = 12.59 nM T78709 CCVP06 52944840 Ki = 3.162 nM T78709 C59ASG 52945060 Ki = 2.13 nM T78709 CDQ27E 52945156 Ki = 3.162 nM T78709 C7VQ5U 52945241 EC50 = 47 nM T78709 CHX9A2 52945310 Ki = 65.8 nM T78709 CPI9F4 52945803 Ki = 31.62 nM T78709 C4SH8M 52945840 Ki = 1.98 nM T78709 COM4R0 52946036 EC50 = 48 nM T78709 CJ49MX 52946290 Ki = 3.981 nM T78709 CRIV53 52946792 Ki = 1.08 nM T78709 C4S8JC 52946835 Ki = 0.803 nM T78709 CGZ1R7 52947088 Ki = 15.85 nM T78709 CS3OD1 52947342 Ki = 0.312 nM T78709 CCOQ59 52947343 Ki = 4.25 nM T78709 C6YB2T 52947380 Ki = 0.814 nM T78709 CK5ER0 52947414 Ki = 0.631 nM T78709 CNH57S 52947579 Ki = 15.85 nM T78709 CAVB03 52947615 Ki = 1 nM T78709 C1HRK4 52947622 Ki = 1 nM T78709 CS01XE 52947712 EC50 = 600 nM T78709 CD17LV 52948101 Ki = 1.44 nM T78709 CX04NC 52948119 Ki = 11.22 nM T78709 C7IR4Q 52948256 Ki = 0.517 nM T78709 CXR12O 52948486 EC50 = 18 nM T78709 CJ6OP5 52948620 Ki = 1.68 nM T78709 C4ZC1K 52948697 Ki = 0.631 nM T78709 C9YBJ3 52948823 Ki = 2.512 nM T78709 CLOB90 52949351 Ki = 3.61 nM T78709 CCQZ15 52949448 Ki = 15.14 nM T78709 C0RUM1 52949810 Ki = 2.34 nM T78709 CS6O4B 52949885 Ki = 3.22 nM T78709 CILY85 52950060 Ki = 0.786 nM T78709 CPVM58 52950169 Ki = 0.859 nM T78709 CT7A6Q 52952304 Ki = 50.12 nM T78709 CHC1S3 52952422 Ki = 3162.28 nM T78709 C4MZ1V 53237227 Ki = 1100 nM T78709 CBIL92 53237431 Ki = 2500 nM T78709 C7L6PJ 53237434 Ki = 2800 nM T78709 C9UX5B 53237437 Ki = 130 nM T78709 CMV78H 53237440 Ki = 39 nM T78709 CL73GJ 53237662 Ki = 240 nM T78709 CS02ZU 53237664 Ki = 2500 nM T78709 C5MLV8 53237666 Ki = 140 nM T78709 CLUD12 53237668 Ki = 100 nM T78709 C9P7KL 53237670 Ki = 59 nM T78709 C8T9OE 53237672 Ki = 14 nM T78709 COJM04 53237674 Ki = 160 nM T78709 C4TNP6 53237891 Ki = 68 nM T78709 C9RIJ7 53237893 Ki = 53 nM T78709 CBZX08 53237895 Ki = 68 nM T78709 C5ZT7N 53237897 Ki = 75 nM T78709 C4KRV8 53237899 Ki = 31 nM T78709 CNJ02E 53237901 Ki = 330 nM T78709 C0H6TR 53237903 Ki = 78 nM T78709 C8TDE6 53238121 Ki = 94 nM T78709 CN4R7I 53238123 Ki = 210 nM T78709 CIP64Q 53238125 Ki = 78 nM T78709 C70LGK 53238127 Ki = 420 nM T78709 C2WK6F 53238129 Ki = 2700 nM T78709 C6C0KM 53238131 Ki = 1400 nM T78709 CXN12U 53238133 Ki = 540 nM T78709 C9QXC8 53238134 Ki = 120 nM T78709 C9Z3FA 53238355 Ki = 310 nM T78709 C1Z8AH 53238357 Ki = 65 nM T78709 CMJ62D 53245590 Ki = 400 nM T78709 C4IV2J 53248158 Ki = 49 nM T78709 C03JEZ 53248159 Ki = 159 nM T78709 C2G0ZY 53248208 Ki = 37.9 nM T78709 C2UKM3 53248209 Ki = 1150 nM T78709 C8KW9J 53248210 Ki = 73 nM T78709 C87SLP 53248211 Ki = 501 nM T78709 CVD7E5 53248212 Ki = 101 nM T78709 CX6KG9 53248213 Ki = 223 nM T78709 C63MQD 53248256 Ki = 299 nM T78709 CG2O7F 53248257 Ki = 6000 nM T78709 CRK87G 53248258 Ki = 139 nM T78709 C73WQX 53248259 Ki = 2140 nM T78709 CKOV84 53248260 Ki = 1170 nM T78709 CGY45S 53248361 Ki = 1.11 nM T78709 CC9B3X 53248362 Ki = 1.11 nM T78709 CR4MN8 53248363 Ki = 0.87 nM T78709 CE9L8G 53248365 Ki = 0.64 nM T78709 C6KAR5 53248408 Ki = 1.95 nM T78709 CZG35A 53248409 Ki = 0.47 nM T78709 CGQJ07 53316788 Ki = 4 nM T78709 CZTW58 53317736 Ki = 22 nM T78709 CW70NZ 53318092 Ki = 30 nM T78709 C7PC1G 53318093 Ki = 8 nM T78709 CQ37BK 53318094 Ki = 19 nM T78709 C8RLQ9 53318095 Ki = 13 nM T78709 C5FRP2 53319428 Ki = 12 nM T78709 CY65NV 53319429 Ki = 6 nM T78709 C1MD0J 53319430 Ki = 16 nM T78709 C1E7BF 53319431 Ki = 90 nM T78709 C2OJW5 53319432 Ki = 1 nM T78709 CT0W3X 53319433 Ki = 203 nM T78709 C61DNP 53320009 IC50 = 672 nM T78709 C9ZDR5 53320010 IC50 = 333 nM T78709 CLQ85U 53322027 Ki = 8 nM T78709 C53HJK 53322028 Ki = 4 nM T78709 CQLK01 53322638 IC50 = 1226 nM T78709 CRUF31 53322954 Ki = 193 nM T78709 C2OB7G 53323389 Ki < 3 nM T78709 C4UBX5 53323390 Ki = 16 nM T78709 C1WU4E 53323391 Ki = 693 nM T78709 C32YWL 53324045 Ki = 481 nM T78709 CFJ1B0 53324709 Ki = 64 nM T78709 C35GJZ 53325137 Ki = 58 nM T78709 CRQF15 53325242 Ki = 1395 nM T78709 CZ69OW 53326010 Ki = 57 nM T78709 CZ1U9T 53326011 Ki = 14 nM T78709 C0UC1W 53326601 Ki = 7.5 nM T78709 C7MQZ6 53362652 Ki = 94 nM T78709 C4VW1I 53362653 Ki = 87 nM T78709 C24DBU 53362654 Ki = 89 nM T78709 CBF2P3 53362655 Ki = 96 nM T78709 C9MK6L 53362715 Ki = 124 nM T78709 C47KPJ 53362716 Ki = 90 nM T78709 C7PA6D 53362719 Ki = 276 nM T78709 CMB23T 53362720 Ki = 380 nM T78709 C7K0PH 53362779 Ki = 249 nM T78709 C8GC1B 53362840 Ki = 217 nM T78709 CU7W2I 53362841 Ki = 259 nM T78709 CH34LM 53362842 Ki = 137 nM T78709 CU4B6N 53370045 Ki = 489 nM T78709 CG24AT 53381002 Ki = 1354 nM T78709 C7WKR1 53387673 Ki > 10000 nM T78709 CFB1N5 53387674 Ki > 10000 nM T78709 CEIG81 53391632 Ki = 2540 nM T78709 CMOZ61 53475319 Ki = 708 nM T78709 C43VJF 54296648 Ki = 9.2 nM T78709 CEQ3M6 54579954 Ki = 2.15 nM T78709 C7WRB0 54579955 Ki = 1.68 nM T78709 C9VZ5P 54580443 Ki = 5 nM T78709 CQ4SI9 54580444 Ki = 9 nM T78709 C0R1QM 54581512 Ki = 851.14 nM T78709 C6PK2X 54582466 Ki = 15 nM T78709 CNW7S4 54582467 Ki = 7 nM T78709 C8V6BJ 54584468 Ki = 108 nM T78709 CY9QZ8 54584591 Ki = 0.6 nM T78709 CYX4S7 54585356 Ki = 11 nM T78709 CTQ08M 54586179 Ki = 3.5 nM T78709 CL5I1R 54753271 Ki = 1510 nM T78709 CG3UJ4 54758298 Ki = 6.7 nM T78709 COZ82F 55479093 Ki = 237 nM T78709 C8WHT5 56593934 Ki = 10000 nM T78709 CW89BT 56595402 Ki > 1000 nM T78709 C4C3XQ 56595529 Ki > 1000 nM T78709 CA54LD 56597090 Ki = 0.6 nM T78709 C6W1RA 56649648 Ki = 0.2 nM T78709 C2SW7J 56649649 Ki = 0.65 nM T78709 CQTR49 56649650 Ki = 0.86 nM T78709 CH37LU 56663451 IC50 > 10000 nM T78709 CR1OB6 56850389 EC50 = 16.3 nM T78709 CF63GQ 56850658 EC50 = 123 nM T78709 CJKO58 56852956 Ki = 40 nM T78709 CK7I9Z 56935084 Ki = 0.58 nM T78709 C20WGQ 56935085 Ki = 0.75 nM T78709 C17IZE 56935086 Ki = 0.74 nM T78709 CB0P9N 56944383 Ki = 110 nM T78709 C1ST9U 56944860 Ki = 4 nM T78709 CQKL90 56944861 Ki = 7 nM T78709 CS5J6Y 56944862 Ki = 10 nM T78709 CFLB40 56944863 Ki = 1.7 nM T78709 C53OTR 56944864 Ki = 6 nM T78709 C5T3RI 56944951 Ki = 5 nM T78709 CR6H7U 56944952 Ki = 12 nM T78709 C1Y2RP 56944953 Ki = 9 nM T78709 C1BH7I 56944954 Ki = 4 nM T78709 CTK9I8 56944955 Ki = 4 nM T78709 CCF1A5 56944956 Ki = 1 nM T78709 C2YVT8 56945042 Ki = 16 nM T78709 CNI2G3 56945043 Ki = 7.4 nM T78709 CCW38Z 56945164 Ki = 0.3236 nM T78709 CN6XE8 56945165 Ki = 0.5623 nM T78709 CPE6C7 56945166 Ki = 9.55 nM T78709 C4L7GW 56945167 Ki = 0.7943 nM T78709 CL68PZ 56946472 Ki = 1.995 nM T78709 CJ98DO 56946474 Ki = 0.8318 nM T78709 CB8J2F 56946573 Ki = 4.365 nM T78709 CCBY53 56946575 Ki = 10.47 nM T78709 CMO0U3 56946577 Ki = 3.467 nM T78709 CJZ3P4 56946579 Ki = 3.467 nM T78709 C1TC7Q 56963799 Ki > 10000 nM T78709 CUL4N1 56964693 Ki = 375 nM T78709 CQ5TP0 56964794 Ki = 19 nM T78709 CDGZ96 57326583 Ki = 266 nM T78709 C20ILW 57326584 Ki = 131 nM T78709 CD9I4N 57334553 IC50 = 11.8 nM T78709 C6H9UV 57345617 Ki = 102 nM T78709 CZU6L2 57345618 Ki = 73 nM T78709 CK9G8H 57345619 Ki = 91 nM T78709 C1US6F 57345626 Ki = 147.91 nM T78709 CD50GK 57345628 Ki = 10.47 nM T78709 C4FA1T 57345629 Ki = 14.79 nM T78709 C19DPJ 57381099 Ki = 711 nM T78709 CHD7U6 57381100 Ki = 10600 nM T78709 CL4Q2R 57381101 Ki = 776.5 nM T78709 C5ASK3 57381102 Ki = 1100 nM T78709 CZYV86 57381316 Ki = 221 nM T78709 C7U6SI 57381317 Ki = 2100 nM T78709 C0EW2L 57381318 Ki = 59000 nM T78709 C2F1UZ 57381319 Ki = 1400 nM T78709 CKIW81 57381320 Ki = 3200 nM T78709 CR9MZ4 57384073 Ki = 0.8 nM T78709 CATM39 57390694 Ki = 216 nM T78709 C6S0IE 57390695 Ki = 495 nM T78709 CCU1S2 57390881 Ki = 15 nM T78709 CV08WY 57391216 Ki = 93.1 nM T78709 CD75YK 57391306 Ki = 613 nM T78709 C07PMA 57391307 Ki = 80 nM T78709 CWT20M 57393083 Ki = 8.6 nM T78709 CDTG05 57393527 Ki = 22.91 nM T78709 CADH19 57394285 Ki = 168 nM T78709 C0WA3H 57394810 Ki = 454 nM T78709 CD4A3P 57396484 Ki = 23 nM T78709 C4EXS6 57396571 Ki = 154 nM T78709 C2ZWS1 57398007 Ki = 1.1 nM T78709 CR1Y7M 57398332 Ki > 10000 nM T78709 C3GW6L 57398351 Ki = 169 nM T78709 CO50ZB 57398352 Ki = 1080 nM T78709 CJ41PW 57399432 Ki = 263 nM T78709 CO3B4P 57399494 Ki = 415 nM T78709 C5GPJ0 57401515 Ki = 6.5 nM T78709 CG8MF3 57401516 Ki = 324 nM T78709 CZX05B 57401706 Ki = 6.2 nM T78709 CYN38R 57401819 Ki = 112 nM T78709 CO0XD2 57401820 Ki = 166 nM T78709 C8EFT7 57402251 Ki = 9.333 nM T78709 CL02EQ 57403172 Ki = 1.82 nM T78709 CX0B5M 57403525 Ki = 658 nM T78709 CWBG94 57403981 Ki = 274 nM T78709 CQB6F9 57456630 Ki = 85 nM T78709 C0M5PN 57873490 Ki > 1000 nM T78709 CH1BN8 57873491 Ki = 43 nM T78709 CI5UO1 57873492 Ki = 59 nM T78709 C2D9HA 57873499 Ki > 1000 nM T78709 C81MLX 57873504 Ki = 24 nM T78709 C7L9IE 57873508 Ki = 2 nM T78709 CZRL39 57873513 Ki > 1000 nM T78709 C98WTS 57873515 Ki = 2 nM T78709 C6BHT3 57873518 Ki = 94 nM T78709 CPX17D 57873520 Ki = 0.7 nM T78709 C54ROE 57873522 Ki = 26 nM T78709 CM7PI1 57873525 Ki = 9.9 nM T78709 CMUR21 57873527 Ki = 117 nM T78709 CO5Y9Q 57873531 Ki = 4 nM T78709 CZI37P 58760107 Ki = 10.91 nM T78709 CYSV60 60165411 Ki = 3.6 nM T78709 CB9GC6 60165412 Ki = 3.6 nM T78709 CI5PM3 60165413 Ki = 7.3 nM T78709 C2Q5VD 60165416 Ki = 90.5 nM T78709 C9JL3F 60165418 Ki = 6.6 nM T78709 C31PEN 60165535 Ki = 5.1 nM T78709 CP60YF 60165537 Ki = 111 nM T78709 CP1DR8 60165539 Ki > 10000 nM T78709 C85OTH 60165541 Ki = 85 nM T78709 CJO91V 60165543 Ki = 63 nM T78709 CJDC53 60165545 Ki = 214 nM T78709 C3K5JN 60165681 Ki = 28.3 nM T78709 C5RUP6 60167166 Ki = 312 nM T78709 CRH49P 60167309 Ki = 771 nM T78709 CX0NY3 60167310 Ki = 350 nM T78709 COHK72 60167451 Ki = 251.19 nM T78709 C30SVG 60167452 Ki = 102.33 nM T78709 CB4HT7 60195992 Ki = 63.2 nM T78709 C6VWY1 60196073 Ki = 31.4 nM T78709 C18AVJ 60196075 Ki = 14.9 nM T78709 CIN29U 60196077 Ki = 149 nM T78709 C5N3SG 60196080 Ki = 17.4 nM T78709 CI30FT 60204111 Ki = 10 nM T78709 CWSA08 60204112 Ki = 44 nM T78709 CLXS32 66561333 Ki = 226.8 nM T78709 CM24PO 66561413 Ki = 0.58 nM T78709 CN30YT 66800947 Ki = 1 nM T78709 CZ3MR6 66800959 Ki = 110 nM T78709 C92CMO 66800965 Ki = 3 nM T78709 C3K8DC 66801052 Ki = 21 nM T78709 C41VYW 66801295 Ki = 10 nM T78709 CR2N0J 66801344 Ki = 70 nM T78709 C3RX4C 66801425 Ki = 96 nM T78709 C7JD0I 66801429 Ki = 70 nM T78709 CN8OU1 66801430 Ki = 110 nM T78709 COR1H8 66801528 Ki = 36 nM T78709 C1F3YV 66801537 Ki = 18 nM T78709 C75WXP 66801561 Ki = 10 nM T78709 CC8JV6 66801624 Ki = 280 nM T78709 C3EI2F 66801625 Ki = 520 nM T78709 C0XG6B 66801701 Ki = 170 nM T78709 C42EBQ 66801837 Ki = 470 nM T78709 CW3AI2 66803474 Ki = 1.8 nM T78709 CPKH06 66803497 Ki = 11 nM T78709 CNJE57 66803500 Ki = 10 nM T78709 CN6FZ1 66803595 Ki = 6.1 nM T78709 C1LEH8 67268994 Ki > 10000 nM T78709 CD3U6K 68731121 Ki = 9720 nM T78709 C6IP8Q 69082816 Ki = 9040 nM T78709 CKM14W 69432471 Ki = 206 nM T78709 CP9V6A 69836292 Ki = 1995.26 nM T78709 CZ41VT 70683643 Ki = 125.8 nM T78709 C6EI2D 70684206 Ki = 730.02 nM T78709 CND4A2 70685780 Ki = 5.78 nM T78709 C6W9UK 70685781 Ki = 0.95 nM T78709 C4REJ6 70687910 Ki = 7.53 nM T78709 C4QNS1 70689942 Ki = 902.6 nM T78709 C0D7IM 70689943 Ki = 122.5 nM T78709 CY1BV3 70689944 Ki = 397.9 nM T78709 CBD3K8 70690497 Ki = 599.89 nM T78709 C8YMI5 70692100 Ki = 95.3 nM T78709 C9J3TO 70692655 Ki > 5000 nM T78709 CJQX48 70693375 Ki = 39.81 nM T78709 CIEG52 70694142 Ki = 159.8 nM T78709 CR7OD5 70694143 Ki = 4.73 nM T78709 C9HV4J 70694144 Ki = 1.39 nM T78709 CU4EK1 70694145 Ki = 2.26 nM T78709 C76JRL 70694146 Ki = 0.5 nM T78709 CET05I 70694683 Ki = 66 nM T78709 CTF76B 70694687 Ki > 1000 nM T78709 CST13M 70695474 Ki = 5.754 nM T78709 CQZ38N 70696271 Ki = 2264 nM T78709 CS7UT3 70697522 Ki = 569 nM T78709 CR5KY1 71061607 Ki = 877 nM T78709 C72XPZ 71061659 Ki = 1274 nM T78709 CKE2Y4 71061750 Ki = 614 nM T78709 CD1ET2 71061756 Ki = 918 nM T78709 C5KM2W 71061887 Ki = 239 nM T78709 C0D5SC 71062035 Ki = 35 nM T78709 CNQ65S 71062123 Ki = 80 nM T78709 CBF6Z8 71109804 Ki > 5000 nM T78709 C68NPQ 71109805 Ki = 208 nM T78709 CC43QK 71151588 Ki = 6.7 nM T78709 CJZ81X 71293954 Ki = 0.8 nM T78709 CZ35EN 71294092 Ki = 0.66 nM T78709 C6VL7X 71449080 Ki = 5.11 nM T78709 CKN5D4 71449120 Ki = 85.5 nM T78709 C91SZN 71449641 Ki = 290 nM T78709 C2GCN7 71449642 Ki = 65 nM T78709 CQN93U 71449643 Ki = 92 nM T78709 CEJ3B4 71449644 Ki = 10 nM T78709 C5SAJ1 71449645 Ki = 89 nM T78709 CG06AP 71449737 Ki = 2.48 nM T78709 C3XNC2 71450247 Ki = 8836 nM T78709 CDI84E 71450922 IC50 > 10000 nM T78709 CHT21G 71451454 Ki = 841 nM T78709 C2QZL4 71451455 Ki = 18 nM T78709 CXI5Q2 71451456 Ki = 456 nM T78709 CKJZ57 71451457 Ki = 21 nM T78709 C0F1HU 71451458 Ki = 5 nM T78709 CTZ24N 71451459 Ki = 49 nM T78709 C70JUP 71451460 Ki = 75 nM T78709 C9WLY7 71452692 Ki = 0.91 nM T78709 CUK2P5 71453252 Ki = 190 nM T78709 CKI58Z 71453278 Ki = 48 nM T78709 C1QM8D 71453279 Ki = 717 nM T78709 C6O4KT 71453280 Ki = 81 nM T78709 CL49VI 71453281 Ki = 31 nM T78709 CGXT64 71453282 Ki = 147 nM T78709 C7SQ0I 71453386 Ki = 14.01 nM T78709 CE0R9D 71454275 Ki = 5709 nM T78709 C0R2UV 71454458 Ki = 1.05 nM T78709 CGO13Q 71454997 Ki = 101 nM T78709 C0K1JV 71454998 Ki = 104 nM T78709 C3JF1D 71454999 Ki = 436 nM T78709 C2QZ1N 71455000 Ki = 313 nM T78709 C6FE5D 71455001 Ki = 230 nM T78709 C4L0JN 71455002 Ki = 22 nM T78709 CQSA61 71455082 Ki = 35.85 nM T78709 C8YH0J 71455083 Ki = 0.51 nM T78709 CAQF34 71455625 Ki = 4987 nM T78709 CD8O2C 71456208 Ki = 7.82 nM T78709 CWR40I 71456780 Ki = 283 nM T78709 CZUX67 71456781 Ki = 45 nM T78709 CZ17FC 71456782 Ki = 9 nM T78709 CKF09U 71456783 Ki = 22 nM T78709 CJKV72 71456784 Ki = 32 nM T78709 C82HSE 71456889 Ki = 1.89 nM T78709 C1PHO6 71456890 Ki = 16.29 nM T78709 C7MNB5 71457264 EC50 > 1000 nM T78709 CMJ1O9 71457409 Ki = 5629 nM T78709 C3GKR6 71458006 Ki = 4.45 nM T78709 CX06FZ 71458032 Ki = 24.55 nM T78709 CPO82B 71458050 Ki = 158.49 nM T78709 C84QJC 71458071 Ki = 510 nM T78709 C37EBC 71458647 Ki = 141 nM T78709 CM6OP1 71458648 Ki = 903 nM T78709 CRGE05 71458649 Ki = 270 nM T78709 CJN4S1 71458650 Ki = 28 nM T78709 CNT5J9 71458651 Ki = 23 nM T78709 C3NAM7 71458652 Ki = 10 nM T78709 CI6H3T 71458739 Ki = 1.61 nM T78709 CS83IF 71459269 Ki = 680 nM T78709 C3OR6K 71459910 Ki = 1.23 nM T78709 CG0WO9 71459954 Ki = 234 nM T78709 CT17XB 71460468 Ki = 30 nM T78709 CMOF94 71460561 Ki = 8.27 nM T78709 C63YLA 71461049 Ki > 10000 nM T78709 CJD96I 71461050 Ki > 10000 nM T78709 C6VL5X 71461632 Ki = 22.7 nM T78709 C0E9NL 71461634 Ki = 33.88 nM T78709 C7AX1Q 71462178 Ki = 45 nM T78709 C1CS0Z 71462179 Ki = 13 nM T78709 CHJ27Z 71462265 Ki = 36.19 nM T78709 CLP8D6 71462266 Ki = 8.36 nM T78709 C4P3JU 71462776 Ki > 10000 nM T78709 C3GUQ2 71462777 Ki > 10000 nM T78709 CD9G8B 71521478 Ki = 0.5495 nM T78709 CSV0G5 71521479 Ki = 0.309 nM T78709 CGN2M7 71521480 Ki = 0.3981 nM T78709 CT2ME3 71574204 Ki = 59 nM T78709 C3SXR5 71574206 Ki = 23 nM T78709 C2YRI9 71574208 Ki = 25 nM T78709 C62RWV 71574210 Ki = 14 nM T78709 CKC53S 71574212 Ki = 23 nM T78709 CNV42M 71574298 Ki = 88 nM T78709 C9PGQ1 71574300 Ki = 79 nM T78709 C2LXH5 71574302 Ki = 17 nM T78709 C2YPB8 71574304 Ki = 112 nM T78709 CK7GM0 71574306 Ki = 34 nM T78709 CI0GU8 71660496 IC50 > 48500 nM T78709 C0W2YA 71727193 Ki = 24 nM T78709 C79TLS 71727194 Ki = 15840 nM T78709 CFB10W 71727195 Ki = 1671 nM T78709 C6CIB5 71727196 Ki = 429 nM T78709 C7Z3JS 71727308 Ki = 117 nM T78709 CU5R1S 71758594 Ki = 243 nM T78709 C3ATN5 72197484 IC50 = 394.8 nM T78709 C20HSN 72197485 IC50 = 1252 nM T78709 CN8A5R 72197486 IC50 = 1057 nM T78709 CL3BF7 72197668 IC50 = 822.8 nM T78709 CWH6T3 72548703 IC50 = 0.43 nM T78709 C8Z0NM 72550642 Ki = 20 nM T78709 CL6W2Q 72550645 Ki = 11 nM T78709 C78LYM 72698087 Ki > 10000 nM T78709 C63HPK 72698088 Ki > 10000 nM T78709 C4AS0E 72699528 Ki = 1.3 nM T78709 CO20CN 72699532 Ki = 11 nM T78709 C8EVJ6 72699690 Ki = 3.9 nM T78709 CEAK86 72699692 Ki = 1.2 nM T78709 CIR7G1 72699716 EC50 = 590 nM T78709 CRMC07 72699718 Ki = 777.79 nM T78709 COH4F8 72699779 Ki = 15 nM T78709 C4X9AO 72699812 Ki = 997.7 nM T78709 C5K9JW 72699815 Ki = 553.1 nM T78709 CIDS43 72699817 EC50 = 850 nM T78709 C6J8GM 72699818 Ki = 175.32 nM T78709 CC8PL5 72699903 Ki = 285.33 nM T78709 C7YTK9 72699904 Ki = 654.64 nM T78709 C26STM 72700473 Ki = 0.69 nM T78709 CL96GC 72700475 Ki = 1.1 nM T78709 C45JKS 72700476 Ki = 5.6 nM T78709 C3TO8B 72700557 Ki = 1.7 nM T78709 CVA2X7 72700634 Ki = 2.1 nM T78709 C0KTL6 72734840 IC50 = 1200 nM T78709 CIO0W1 72734841 IC50 = 599 nM T78709 CTG91B 72734842 IC50 = 15 nM T78709 C49FUQ 72734843 IC50 = 16 nM T78709 C4E6PH 72734844 IC50 = 7200 nM T78709 CU9E5O 72734845 IC50 = 4500 nM T78709 CS48GA 72735019 IC50 = 5700 nM T78709 CB8CJ9 72735020 IC50 = 4900 nM T78709 C2WXK6 72735021 IC50 = 128 nM T78709 CC6Q5R 72771081 Ki < 100 nM T78709 C5L8NJ 72947314 Ki = 83.18 nM T78709 CE1JY2 72947315 Ki = 79.43 nM T78709 CC65OA 73213195 Ki = 371.54 nM T78709 CW83DK 73213196 Ki > 10000 nM T78709 C02FTM 73291731 Ki = 13.8 nM T78709 CCV91B 73346042 Ki = 0.1 nM T78709 CRG9J8 73346332 Ki > 10000 nM T78709 CM3IA6 73349341 EC50 = 45 nM T78709 C1MTL3 73350910 EC50 = 1195 nM T78709 CSCJ76 73350911 EC50 = 19 nM T78709 CD9Y0J 73350915 EC50 = 76 nM T78709 CL38VQ 73351112 Ki > 1000 nM T78709 CR0D1A 73356945 EC50 = 23 nM T78709 CVF5P0 73603034 IC50 = 4900 nM T78709 CUB97Z 74538690 Ki = 582 nM T78709 C2E7QW 75201901 Ki = 1200 nM T78709 C8IDL3 75306277 Ki = 39.81 nM T78709 CX17RZ 76280896 Ki = 203 nM T78709 C45OSP 76284193 Ki = 1055 nM T78709 C0CRJ1 76284452 Ki = 568 nM T78709 CS17IJ 76284453 Ki = 875 nM T78709 CH82JU 76284455 Ki = 272 nM T78709 CRO7Q9 76284721 Ki = 433 nM T78709 C4BIC2 76284724 Ki = 152 nM T78709 C0EKY7 76284725 Ki = 961 nM T78709 CS3HT5 76309671 Ki = 100 nM T78709 CXJG08 76314094 Ki = 387 nM T78709 CE5C2B 76319004 Ki = 25.7 nM T78709 C5F1XU 76321735 Ki = 700 nM T78709 C5TQ0X 76322648 Ki = 26.73 nM T78709 C94VNF 76324975 Ki = 537 nM T78709 CZ6P1E 76328545 Ki = 186 nM T78709 CGBE87 76335066 Ki = 90.2 nM T78709 CW3AK0 76335863 Ki = 743 nM T78709 C1UZ5J 76441180 Ki = 5.3 nM T78709 C28RIZ 76518514 Ki = 102 nM T78709 C8EWX5 85658088 Ki = 1805 nM T78709 C70ZVB 86221574 Ki = 5396 nM T78709 CJ9N5Q 86280005 Ki = 2.5 nM T78709 CJ92WR 86288399 Ki = 3.67 nM T78709 CMJA85 86288474 Ki = 1.1 nM T78709 C9S0XK 86288947 Ki = 121 nM T78709 CEPC94 86288948 Ki = 121 nM T78709 CJ9K3T 86290953 IC50 = 3800 nM T78709 CUA89I 86341962 Ki = 0.2 nM T78709 CWPH45 86341996 Ki = 1.4 nM T78709 CCR8X7 86342061 Ki = 12 nM T78709 CY2I8J 86342094 Ki = 5.2 nM T78709 CC47HJ 86342098 Ki = 5.3 nM T78709 CK03YC 86342156 Ki = 1.3 nM T78709 C5AQK2 86342192 Ki = 1.1 nM T78709 C9DZ2I 86342193 Ki = 0.52 nM T78709 CQP38R 86342194 Ki = 7.6 nM T78709 CE39OD 86342294 Ki = 1.1 nM T78709 C9T3LW 89638708 EC50 = 0.3 nM T78709 CHE2U4 90178632 Ki = 437 nM T78709 CD7R6P 90213677 Ki = 7.2 nM T78709 CWMU25 90644511 IC50 = 500 nM T78709 C37CYS 90654670 Ki = 122 nM T78709 C0IQ5R 90654671 Ki = 18 nM T78709 CVG2C1 90654672 Ki < 1 nM T78709 CU0ON1 90654673 Ki = 2 nM T78709 CJR3Y9 90654674 Ki = 122 nM T78709 CO1H4U 90654675 Ki = 107 nM T78709 CAY64Z 90654676 Ki = 12 nM T78709 CH0R8B 90654677 Ki = 77 nM T78709 CRFB56 90654678 Ki = 72 nM T78709 CPR21O 90654679 Ki = 236 nM T78709 C6YLV3 90654680 Ki = 499 nM T78709 CGUY51 90654681 Ki = 211 nM T78709 CK8X4O 90654682 Ki = 1914 nM T78709 CH8UQ9 90654683 Ki = 643 nM T78709 CTQ23Z 90654684 Ki = 16 nM T78709 C9Q2JW 90654685 Ki = 212 nM T78709 C98TJR 90654686 Ki = 377 nM T78709 CG3OI7 90654687 Ki = 230 nM T78709 CKTV83 90654688 Ki = 89 nM T78709 CVK85U 90654689 Ki = 47 nM T78709 CLG75D 90654690 Ki = 14 nM T78709 C7T9HW 90654691 Ki = 23 nM T78709 C92BZL 90654692 Ki = 313 nM T78709 C6CD9R 90654693 Ki = 214 nM T78709 C6H9NV 90654694 Ki = 44 nM T78709 CR74SD 90654695 Ki = 6307 nM T78709 C7VM4O 90654696 Ki = 52 nM T78709 CGFU53 90654697 Ki = 232 nM T78709 C7BEZ8 90654698 Ki = 141 nM T78709 CZ3IM2 90654699 Ki = 38 nM T78709 C8TMK5 90654700 Ki = 573 nM T78709 C7GK3C 90654701 Ki = 83 nM T78709 CN8BO1 90654702 Ki = 4 nM T78709 CHIW63 90654703 Ki = 2908 nM T78709 C1SAW2 90654704 Ki = 214 nM T78709 CJG31T 90654831 Ki = 5.5 nM T78709 CMU45O 90654832 Ki = 13.2 nM T78709 C14NPE 90654833 Ki = 135 nM T78709 C3C4BW 90654834 Ki = 124 nM T78709 C8QWR3 90654835 Ki = 23.3 nM T78709 C6ZR9L 90654837 Ki = 79 nM T78709 C0AC7R 90654839 Ki = 26 nM T78709 CKLG40 90654841 Ki = 45 nM T78709 C5JS8D 90654843 Ki = 76 nM T78709 C4VHZ6 90654845 Ki = 201 nM T78709 CG78PS 90654847 Ki = 235 nM T78709 CL39WP 90654849 Ki = 299 nM T78709 C0TVQ9 90654851 Ki = 305 nM T78709 C4I1CU 90654853 Ki = 88 nM T78709 CZ28YC 90654855 Ki = 301 nM T78709 CRO83N 90654857 Ki = 2178 nM T78709 CI91AM 90655807 Ki = 105 nM T78709 CY3L4T 90655808 Ki = 11.1 nM T78709 C2FG8Q 90655809 Ki = 2.62 nM T78709 C4R6CT 90655810 Ki = 14 nM T78709 CUQ8E6 90655811 Ki = 9.3 nM T78709 CU94HP 90655812 Ki = 7.55 nM T78709 CVY16X 90655813 Ki = 6.1 nM T78709 C12JSA 90655814 Ki = 33.5 nM T78709 CNB86Y 90655815 Ki = 42.5 nM T78709 C7NW4X 90655816 Ki = 221.4 nM T78709 CHG3S1 90655817 Ki = 31.6 nM T78709 C93XMI 90655818 Ki = 28.95 nM T78709 CANR17 90655819 Ki = 7.29 nM T78709 C58SPJ 90655820 Ki = 21 nM T78709 CB2ZL6 90655821 Ki = 8.06 nM T78709 CTZP78 90655822 Ki = 631 nM T78709 C23KCF 90655823 Ki = 425 nM T78709 CJSZ89 90655824 Ki = 496 nM T78709 CCOV98 90664359 Ki = 13340 nM T78709 C4MUI2 90664601 IC50 = 4.9 nM T78709 CXD5Q9 90664621 Ki = 4503 nM T78709 CKM05S 90664904 IC50 > 10000 nM T78709 CHT7D5 90664962 IC50 = 3.9 nM T78709 CACG19 90666899 Ki = 489.78 nM T78709 CODM50 90666903 Ki = 102.33 nM T78709 CSRU41 91242334 EC50 = 21.3 nM T78709 C0J5YH 91864602 Ki = 8.128 nM T78709 CRX16J 91884611 EC50 = 9.75 nM T78709 CDWS84 91937906 Ki < 1 nM T78709 CUQ6V0 92042918 Ki < 1000 nM T78709 CE0ZC6 101876962 Ki = 1174.9 nM T78709 C4DG3V 102364516 Ki > 1000 nM T78709 C4WDR8 109018769 Ki = 0.34 nM T78709 CF0XJ6 109018934 Ki = 938 nM T78709 CYB18Z 109027017 Ki = 272 nM T78709 CP6F4D 112815120 Ki = 305 nM T78709 CSH7K4 117949705 Ki = 118.7 nM T78709 C0M3CD 118051679 Ki = 13 nM T78709 CEMZ15 118464420 Ki = 320 nM T78709 CV2L6O 118464425 Ki = 116 nM T78709 CFNG86 118464427 Ki = 6764 nM T78709 CMSN80 118626035 Ki = 13 nM T78709 CT3AI0 118626042 Ki = 8 nM T78709 CKNJ72 118626045 Ki = 10 nM T78709 CGB42Y 118626088 Ki = 5 nM T78709 C0XJT5 118626089 Ki = 18 nM T78709 CIE4C7 118626101 Ki = 6 nM T78709 C1NYS5 118626120 Ki = 6 nM T78709 CPG04R 118626121 Ki = 13 nM T78709 C3S5LJ 118626129 Ki = 15 nM T78709 CY3F0N 118626140 Ki = 66 nM T78709 CE07IQ 118626142 EC50 = 11 nM T78709 C72OZY 118626161 Ki = 24 nM T78709 CY3E7S 118626169 Ki = 7 nM T78709 CHRB75 118626208 Ki = 6 nM T78709 C2Q4OP 118709739 Ki = 523 nM T78709 CZ68PL 118709740 Ki = 576 nM T78709 CSB25E 118709750 Ki = 13 nM T78709 CD4S9R 118709751 Ki = 8.2 nM T78709 CBP52O 118709752 Ki > 1000 nM T78709 CO72SF 118709753 Ki = 470 nM T78709 CJQR81 118709754 Ki = 491 nM T78709 CPW1D5 118709755 Ki > 1000 nM T78709 C1TMO7 118709756 Ki > 1000 nM T78709 CZDE01 118713090 Ki = 190 nM T78709 C1KR9C 118713091 Ki = 180 nM T78709 CI5U1R 118713092 Ki = 220 nM T78709 C4S7WD 118713093 Ki = 0.46 nM T78709 CB8Q2E 118713094 Ki = 0.835 nM T78709 CH9W0A 118713587 Ki = 913 nM T78709 CK43CN 118713588 Ki = 24.58 nM T78709 CL0TS7 118713589 Ki = 10.36 nM T78709 C4RD6F 118713590 Ki = 695.11 nM T78709 CIG13W 118713591 Ki = 83.33 nM T78709 CX5L1H 118713592 Ki = 6.13 nM T78709 CDWY84 118713593 Ki = 74.92 nM T78709 CO5S1I 118713594 Ki = 19.22 nM T78709 CI91US 118713595 Ki = 95.66 nM T78709 CW92LT 118713679 Ki = 11.86 nM T78709 C8P9YT 118713680 Ki = 7.13 nM T78709 CZ1K5R 118713681 Ki = 3.96 nM T78709 CH7ZE8 118713682 Ki = 0.91 nM T78709 CKX78H 118713683 Ki = 1.3 nM T78709 C5LSA7 118713684 Ki = 0.43 nM T78709 CPAI54 118713685 Ki = 29.78 nM T78709 C6U2LR 118713686 Ki = 0.27 nM T78709 CYA6E4 118713687 Ki = 0.19 nM T78709 CZ9UL2 118713688 Ki = 0.21 nM T78709 CUV5Y0 118715454 EC50 > 30000 nM T78709 CI7NQ9 118716698 Ki = 9.333 nM T78709 CGO9W4 118716699 Ki = 46.77 nM T78709 CVDI36 118716700 Ki = 14.45 nM T78709 C94AFL 118716701 Ki = 117.49 nM T78709 CTX92K 118716702 Ki = 81.28 nM T78709 CG02WP 118716703 Ki = 158.49 nM T78709 CTNL85 118716704 Ki = 15.85 nM T78709 CM1Y8W 118716705 Ki = 8.913 nM T78709 C42MOT 118716706 Ki = 58.88 nM T78709 C78ARU 118716707 Ki = 50.12 nM T78709 CO5TG3 118716708 Ki = 42.66 nM T78709 CNF78L 118716709 Ki = 20.42 nM T78709 C9CB1Q 118716710 Ki = 36.31 nM T78709 C3F6EQ 118716711 Ki = 64.57 nM T78709 C0L6YO 118716712 Ki = 323.59 nM T78709 CX2AC4 118716713 Ki = 52.48 nM T78709 CL1EU8 118716714 Ki = 26.92 nM T78709 C0V7GJ 118716715 Ki = 37.15 nM T78709 CRBI65 118716716 Ki = 69.18 nM T78709 C70IPZ 118716717 Ki = 24.55 nM T78709 CBI30N 118716718 Ki = 43.65 nM T78709 C7UBN8 118716719 Ki = 60.26 nM T78709 CV8HA2 118716720 Ki = 144.54 nM T78709 C30ZJB 118716721 Ki = 33.11 nM T78709 C58MND 118716722 Ki = 79.43 nM T78709 CO6T4G 118716723 Ki = 87.1 nM T78709 C8RVX4 118717455 Ki = 616.6 nM T78709 C5IM1N 118717456 Ki = 3467 nM T78709 CBCU90 118717457 Ki = 891 nM T78709 CN4LJ2 118717458 Ki = 1096 nM T78709 CZ35PU 118717459 Ki = 1380 nM T78709 C9BP7A 118717460 Ki = 1258.93 nM T78709 CFCM61 118717461 Ki = 2818 nM T78709 C8C6ZW 118717462 Ki = 602.56 nM T78709 CG0O3Q 118719795 Ki = 6 nM T78709 CUHT71 118719796 Ki = 5.8 nM T78709 CR0FM7 118719797 Ki = 7.4 nM T78709 CPX2Y1 118719798 Ki = 1.3 nM T78709 C0KH8S 118719799 Ki = 153 nM T78709 CWO13F 118719807 Ki = 9.4 nM T78709 CUH0A6 118719810 Ki = 3.9 nM T78709 CES97Y 118722639 Ki = 15 nM T78709 CM3P7R 118722912 Ki = 67 nM T78709 CP3QC2 118722913 Ki = 11 nM T78709 C1PG3C 118722914 Ki = 73 nM T78709 CR6E5D 118722915 Ki > 1000 nM T78709 CGA86P 118728506 Ki = 39.6 nM T78709 C9PGE7 118728507 Ki = 37.4 nM T78709 CR4GE1 118728510 Ki = 15.2 nM T78709 C14LZH 118728511 Ki = 363 nM T78709 C14RAC 118728513 Ki = 114 nM T78709 CQK04P 118728514 Ki = 53.9 nM T78709 CK9CG4 118728521 Ki = 28.9 nM T78709 C1N9JU 118728522 Ki = 268 nM T78709 C1UZ8G 118728523 Ki = 6.28 nM T78709 CPCE84 118728524 Ki = 51.5 nM T78709 CBN06J 118728525 Ki = 1.04 nM T78709 CF3QE0 118728526 Ki = 16.1 nM T78709 CJG4Q1 118728527 Ki = 211 nM T78709 C4NFW1 118728528 Ki = 3.23 nM T78709 CO8LF9 118728529 Ki = 26.4 nM T78709 CCN7R8 118728530 Ki = 1.03 nM T78709 C5O2NU 118729733 Ki = 3842 nM T78709 CTE58Z 118730369 Ki = 500 nM T78709 CB3Y2W 118731347 Ki = 16 nM T78709 CWZF06 118731348 Ki = 53 nM T78709 CA3O1H 118731349 Ki = 34 nM T78709 CU8P4W 118731350 Ki = 20 nM T78709 C8GKX6 118731351 Ki = 66 nM T78709 C2J4VC 118731352 Ki = 26 nM T78709 CF7NH5 118731353 Ki = 61 nM T78709 CQ8F6C 118731354 Ki = 1 nM T78709 CR9J0O 118731355 Ki = 17 nM T78709 CU12XM 118731356 Ki = 35 nM T78709 C4CEV7 118731357 Ki = 18 nM T78709 CU6T2D 118731358 Ki = 9 nM T78709 C95WKJ 118731359 Ki = 35 nM T78709 C20QAO 118731360 Ki = 16 nM T78709 CT6J8V 118731361 Ki = 14 nM T78709 C7QVJ4 118731362 Ki = 47 nM T78709 CA2X3O 118731363 Ki = 36 nM T78709 C4DV8I 118731364 Ki = 19 nM T78709 CHVY82 118731365 Ki = 40 nM T78709 CM5FG1 118731366 Ki = 16 nM T78709 C7W3EY 122178698 Ki = 506 nM T78709 CF8P1H 122178699 Ki = 153 nM T78709 C48MFR 122178700 Ki = 179 nM T78709 CZ72QS 122178701 Ki = 273 nM T78709 C4VY8A 122178702 Ki = 845 nM T78709 C2KF4Z 122178703 Ki = 563 nM T78709 CX6MJ2 122178704 Ki = 244 nM T78709 CA53KF 122178705 Ki = 117 nM T78709 C8XD3F 122178706 Ki = 152 nM T78709 CTRC59 122178707 Ki = 224 nM T78709 C5QV8D 122178708 Ki = 163 nM T78709 C84UED 122178709 Ki = 361 nM T78709 CV96JK 122178710 Ki = 92 nM T78709 CM89KS 122178711 Ki = 102 nM T78709 CXL5V3 122183764 Ki = 9 nM T78709 CK3VT8 122183765 Ki = 21 nM T78709 C12TRH 122183771 Ki = 84 nM T78709 C06GQO 122183778 Ki = 68 nM T78709 C3VDY7 122197403 Ki = 13 nM T78709 C1MFJ3 122197404 Ki = 13 nM T78709 CBHT01 122377930 Ki = 356 nM T78709 CLW53P 122483274 Ki = 22 nM T78709 CO63ET 122483280 Ki = 122 nM T78709 C4QM2E 124247485 Ki = 1866 nM T78709 CM57GR 126720252 Ki = 5650 nM T78709 CLWM12 126720394 Ki = 1354 nM T78709 C8Q1JB 126720403 Ki = 5934 nM T78709 C1U3SZ 126720425 Ki = 2277 nM T78709 C5G8FD 126720440 Ki = 2790 nM T78709 CD50YM 127024949 Ki = 23 nM T78709 C4GF2D 127024950 Ki = 46 nM T78709 CJ76IB 127024951 Ki = 206 nM T78709 CIHZ54 127025242 Ki = 142 nM T78709 CCY7P3 127025243 Ki = 98 nM T78709 CNJ4Z1 127025244 Ki = 99 nM T78709 CTBN56 127026052 Ki = 79.43 nM T78709 C26NMB 127026071 Ki = 1847 nM T78709 C1YD7M 127026119 Ki = 463 nM T78709 CUO7Y8 127026120 Ki = 197 nM T78709 CDU21O 127026131 Ki = 51 nM T78709 C9HDP8 127026132 Ki = 431 nM T78709 CTYP30 127026133 Ki = 254 nM T78709 C19BOM 127026141 Ki = 947 nM T78709 CZFB49 127026142 Ki = 199 nM T78709 C2FT3B 127026143 Ki = 148 nM T78709 CP4J5H 127026144 Ki = 591 nM T78709 C6BIU4 127026145 Ki = 190 nM T78709 C1FA2U 127026146 Ki = 718 nM T78709 CE43NR 127026147 Ki = 502 nM T78709 C1TV0X 127026296 Ki > 1000 nM T78709 CDAP16 127026434 Ki = 6147 nM T78709 C2XO3L 127026443 Ki = 4570 nM T78709 C80QHX 127026444 Ki = 556 nM T78709 CBF64M 127026450 Ki = 123 nM T78709 CO1FB4 127026451 Ki = 170 nM T78709 CC13RA 127026452 Ki = 74 nM T78709 CBE56W 127026514 Ki = 549 nM T78709 C0SZI4 127026515 Ki = 148 nM T78709 CS1WZ7 127026552 Ki > 1000 nM T78709 C67GCU 127026601 Ki = 7.586 nM T78709 C68ZHE 127026602 Ki = 7.244 nM T78709 C94PCX 127026603 Ki = 50.12 nM T78709 C03TAB 127026604 Ki = 125.89 nM T78709 C3MEP4 127026605 Ki = 416.87 nM T78709 C7P0YF 127026609 Ki > 1000 nM T78709 C1SV6Z 127026610 Ki > 1000 nM T78709 C3V1WR 127026611 Ki > 1000 nM T78709 CX6EI2 127026750 Ki = 545 nM T78709 CEG15O 127026751 Ki = 373 nM T78709 C1J4QY 127026752 Ki = 28 nM T78709 C0WB2U 127026753 Ki = 45 nM T78709 C9AWR7 127026894 Ki > 1000 nM T78709 CQC3H0 127026895 Ki > 1000 nM T78709 CSA2O0 127026896 Ki > 1000 nM T78709 CIG2V3 127027195 Ki > 1000 nM T78709 CC9O6J 127027196 Ki > 1000 nM T78709 C4R5SE 127027197 Ki > 1000 nM T78709 C0UOJ6 127027386 Ki = 371 nM T78709 C9IH1A 127027387 Ki = 407 nM T78709 C0TC7E 127027388 Ki = 536 nM T78709 CZ4W6I 127027389 Ki = 393 nM T78709 C4YR7A 127027390 Ki = 260 nM T78709 C3FA0I 127027391 Ki = 2667 nM T78709 CSHA70 127027488 Ki > 1000 nM T78709 CQJZ73 127027489 Ki > 1000 nM T78709 CZT84N 127027491 Ki > 1000 nM T78709 CNBO79 127027492 Ki > 1000 nM T78709 CJB98N 127027493 Ki > 1000 nM T78709 C3VO6E 127027494 Ki > 1000 nM T78709 CMT35D 127027495 Ki > 1000 nM T78709 CO21RS 127027496 Ki > 1000 nM T78709 CC71UE 127027715 Ki = 1068 nM T78709 CY2TW9 127028152 Ki = 2733 nM T78709 CAZJ04 127028153 Ki = 2969 nM T78709 CR48GO 127028154 Ki = 1646 nM T78709 C8MC1I 127028408 Ki = 750 nM T78709 CD8H7W 127028471 Ki = 397 nM T78709 C4EAY5 127028472 Ki = 98 nM T78709 CUS8R9 127028473 Ki = 319 nM T78709 CA10BY 127028634 Ki = 745 nM T78709 C7JD9S 127028726 Ki = 162.18 nM T78709 C31GSQ 127028730 Ki = 549.54 nM T78709 CZ26YR 127028797 Ki = 59 nM T78709 CI2R1N 127028798 Ki = 1304 nM T78709 CS8GJ5 127028799 Ki = 6862 nM T78709 CU0WQ3 127029375 Ki = 5298 nM T78709 CS1GX5 127029649 Ki = 9167 nM T78709 C9N3BE 127029650 Ki = 821 nM T78709 CQFS48 127029651 Ki = 1004 nM T78709 C7F3YE 127029652 Ki = 5570 nM T78709 CZ61LK 127034966 IC50 > 5011.87 nM T78709 CA0SN5 127034967 IC50 = 1995.26 nM T78709 CQ0ZT9 127035062 Ki = 821 nM T78709 CU49VE 127036186 Ki = 31.62 nM T78709 CG06BD 127036932 Ki = 58.88 nM T78709 CVW71O 127036953 Ki = 10 nM T78709 C7N5DF 127037679 Ki = 208 nM T78709 CD13VY 127037680 Ki = 455 nM T78709 CTE43C 127037681 Ki = 616 nM T78709 C0LGK6 127037682 Ki = 103 nM T78709 C2XBE8 127037921 Ki = 17770 nM T78709 CX0CN4 127037922 Ki = 342 nM T78709 CXR71M 127038002 Ki = 2.455 nM T78709 CDAE15 127038033 Ki = 232 nM T78709 CFA6Q8 127038034 Ki = 74 nM T78709 CERL85 127038035 Ki = 279 nM T78709 C8TC9G 127038281 Ki = 159 nM T78709 CPK2Z7 127038282 Ki = 5555 nM T78709 CL5N3P 127038713 Ki = 40.74 nM T78709 CYJ2D5 127039593 Ki = 214 nM T78709 CQED51 127039753 Ki = 159 nM T78709 CL4E2K 127039754 Ki = 368 nM T78709 CES26L 127039755 Ki = 234 nM T78709 CQ36LP 127039756 Ki = 183 nM T78709 C89SOL 127040060 Ki = 3.802 nM T78709 CQ3L8Z 127040156 Ki = 3.02 nM T78709 C7KA2C 127040443 Ki = 278 nM T78709 CKBZ01 127040444 Ki = 249 nM T78709 CFAB12 127040760 Ki = 178 nM T78709 CWQ47G 127040761 Ki = 373 nM T78709 C8D4AV 127040908 Ki = 180 nM T78709 CE12AY 127041106 Ki = 321 nM T78709 C71LGS 127041107 Ki = 74 nM T78709 C6RI9V 127041108 Ki = 102 nM T78709 C15BGV 127041244 Ki = 140 nM T78709 CU0J4S 127041258 Ki = 190 nM T78709 C20MZH 127041259 Ki = 346 nM T78709 CP16CZ 127041260 Ki = 2346 nM T78709 CZT53S 127041261 Ki = 4511 nM T78709 C0FJP2 127041563 Ki = 9054 nM T78709 CUC3F9 127041564 Ki = 9626 nM T78709 COG9D2 127041874 Ki = 62 nM T78709 CS4WH1 127042184 Ki = 30 nM T78709 C13AIN 127042185 Ki = 80 nM T78709 CR59TP 127042539 Ki = 158 nM T78709 C54IZC 127042540 Ki = 249 nM T78709 C8G1HF 127042841 Ki = 14030 nM T78709 C0V5YU 127048532 EC50 = 361 nM T78709 CHW0L2 127048533 EC50 = 120 nM T78709 C9QR6V 127048539 EC50 = 6 nM T78709 CU6K4P 127048540 EC50 = 8.2 nM T78709 CC7BU0 127049059 Ki = 380.19 nM T78709 C42FHY 127049060 Ki = 376 nM T78709 CF2QY9 127049061 Ki = 1162.5 nM T78709 CN2F1W 127049163 EC50 = 12 nM T78709 C1TI6J 127049515 EC50 = 7.2 nM T78709 CT16PL 127049516 EC50 = 122 nM T78709 C4QKS3 127049517 EC50 = 26 nM T78709 C03BLH 127049522 EC50 = 309 nM T78709 C2IX7Q 127049847 EC50 = 34.4 nM T78709 CRK8W3 127049848 EC50 = 97.2 nM T78709 C85PIF 127049849 EC50 = 137 nM T78709 CO2V5Z 127049850 EC50 > 10000 nM T78709 C27MWC 127049861 EC50 = 122 nM T78709 CZS1L6 127049862 EC50 = 13 nM T78709 CZD91J 127049863 EC50 = 13 nM T78709 C1S6EN 127049864 EC50 = 4.3 nM T78709 C2H0BQ 127049865 EC50 = 2.7 nM T78709 CUK1S9 127049866 EC50 = 5.1 nM T78709 CX53AC 127050632 Ki = 102 nM T78709 CP9UT4 127050764 EC50 > 100 nM T78709 C9T2VY 127050765 EC50 = 24 nM T78709 CIOZ65 127051038 EC50 = 26 nM T78709 C7XK3G 127051039 EC50 = 101 nM T78709 CR4TV6 127051040 EC50 = 464 nM T78709 CCTO35 127051041 EC50 = 74 nM T78709 CA2SJ6 127051340 EC50 = 301 nM T78709 CTL0S1 127051516 Ki = 194.98 nM T78709 CTL8J1 127051843 Ki = 295 nM T78709 CF6V9Q 127051844 Ki = 38 nM T78709 C8TNB1 127051845 Ki = 23 nM T78709 CT9O7G 127051863 Ki = 3153 nM T78709 C5ONG1 127051864 Ki = 251.19 nM T78709 CRF85X 127052458 Ki = 33.5 nM T78709 CCY71I 127052465 Ki = 533 nM T78709 C2E9VX 127052467 Ki = 1689 nM T78709 CPO4C3 127052468 Ki = 190.55 nM T78709 CSQ2N8 127052486 Ki = 611 nM T78709 CLU7C1 127052757 Ki = 141 nM T78709 C95KYT 127052758 Ki = 244 nM T78709 CYNR02 127052759 Ki = 217 nM T78709 C1JAS7 127052779 Ki = 33.88 nM T78709 C7MQK8 127053042 Ki = 40.74 nM T78709 C3WIA6 129103318 IC50 = 587.8 nM T78709 CBX2V6 129186527 EC50 > 10000 nM T78709 CV2K7I 129186528 EC50 = 24.22 nM T78709 CD9C1F 129186530 EC50 > 10000 nM T78709 C2F5YE 129186531 EC50 > 10000 nM T78709 C6GC0F 129186534 EC50 = 7.2 nM T78709 CTP0O3 129186549 EC50 = 34.1 nM T78709 C8KM6N 129186554 EC50 = 4.57 nM T78709 C7FR6U 129186558 EC50 = 899 nM T78709 CEZT92 129186564 EC50 = 7.09 nM T78709 C1CV2Y 129840786 Ki = 1.5 nM T78709 CJ5S2O 129840806 Ki = 809 nM T78709 C9K8MH 129840818 Ki = 6.7 nM T78709 C36AFR 129840841 Ki = 4.8 nM T78709 CUD71X 129840856 Ki = 33 nM T78709 CV4D2F 129840894 Ki = 250 nM T78709 C40HCZ 129840904 Ki = 8 nM T78709 CY7DS0 129840906 Ki = 1.7 nM T78709 CJX83W 129840907 Ki = 3500 nM T78709 C4PU0E 129840972 Ki = 1 nM T78709 C6K4NX 129840994 Ki = 60 nM T78709 C6Y7FB 129841007 Ki = 15 nM T78709 CKA0L7 129841015 Ki = 250 nM T78709 CK1G0Y 129841036 Ki = 0.7 nM T78709 CGUW90 129841059 Ki = 389 nM T78709 CV8SI7 129841063 Ki = 7 nM T78709 C10VDB 130431277 Ki = 70.3 nM T78709 CI1NF8 130431279 Ki = 3560 nM T78709 CS8O4E 130431287 Ki = 560 nM T78709 C85MOW 130431289 Ki = 910 nM T78709 C2OH7B 130431291 Ki = 2660 nM T78709 CEQ43Y 130431295 Ki = 9500 nM T78709 CK64GU 130431296 Ki = 117 nM T78709 CYW0X2 130431314 Ki = 248 nM T78709 CDN26V 130431316 Ki = 880 nM T78709 CL64UW 130431317 Ki = 27.6 nM T78709 C8HE2O 130431318 Ki > 7600 nM T78709 CZ6S4T 130431319 Ki = 131 nM T78709 C8ZHI7 130431325 Ki = 26 nM T78709 CF5SW8 130431328 Ki = 4980 nM T78709 CN9RZ3 130431329 Ki = 2800 nM T78709 CN70MW 130431337 Ki = 59 nM T78709 C4GF1U 130431342 Ki = 2410 nM T78709 C2WI5R 130431351 Ki = 2330 nM T78709 C50GOC 130442480 Ki = 6900 nM T78709 CM04RF 130442572 Ki = 2500 nM T78709 C1RI8Q 132060720 Ki = 2019 nM T78709 CY8B9L 132060743 Ki = 2609 nM T78709 C4VNA6 132060746 Ki = 2135 nM T78709 CGHO19 132060770 Ki = 335 nM T78709 CT81OY 132060776 Ki = 1201 nM T78709 CFXL21 132060812 Ki = 733 nM T78709 C4LJ2Y 132503215 Ki = 45 nM T78709 CM8B1L 132525569 Ki = 1501 nM T78709 CU5L0K 132525570 Ki = 637 nM T78709 CA10SQ 132547275 Ki = 17.4 nM T78709 C6E1GN 132547276 Ki = 6.96 nM T78709 C6VTW3 132547277 Ki = 8.21 nM T78709 CI70OP 132547278 Ki = 25.9 nM T78709 C3Q1LA 132547279 Ki = 2.99 nM T78709 CAVB41 132584404 Ki > 10000 nM T78709 CS0MB3 132938109 Ki = 1329 nM T78709 C8O2EP 134130246 Ki = 95 nM T78709 C8M9FH 134130379 Ki = 111 nM T78709 CA4GX3 134130447 Ki = 33.5 nM T78709 C7ZDA2 134130462 Ki = 18.6 nM T78709 CWL50Q 134130594 Ki = 167 nM T78709 C8TG2O 134130846 Ki = 100 nM T78709 CHP3J4 134131015 Ki = 90.3 nM T78709 CQ4IF8 134131147 Ki = 17.8 nM T78709 C6N5FS 134131151 Ki = 772 nM T78709 CH4XB2 134131159 Ki = 1032 nM T78709 CR32SP 134131265 Ki = 52.1 nM T78709 C0JKL5 134131283 Ki = 24.7 nM T78709 C3Z6SV 134131949 Ki = 4500 nM T78709 C0RQC6 134131976 Ki = 2870 nM T78709 C6D1HC 134132279 Ki > 1000 nM T78709 CQX4U3 134133064 Ki = 338.84 nM T78709 C2V8BH 134133118 Ki = 1.96 nM T78709 CCPI30 134133464 Ki = 2.3 nM T78709 CTS3J4 134133483 Ki = 105 nM T78709 C0J2ML 134133604 Ki = 15.49 nM T78709 CM4XE8 134133829 Ki = 2.239 nM T78709 C6QAF1 134133900 IC50 < 10 nM T78709 CM0TS6 134133967 Ki = 29 nM T78709 CC1DO8 134134456 Ki = 771 nM T78709 CR4F6X 134135492 Ki = 1.5 nM T78709 CM34TY 134135507 Ki = 3 nM T78709 C2Q3JY 134135516 Ki = 595 nM T78709 CJG3U0 134136134 Ki = 149 nM T78709 C3P9IJ 134136137 Ki = 9.4 nM T78709 CLA4R3 134136207 Ki = 2.27 nM T78709 CGX03A 134136246 Ki = 1096.48 nM T78709 C7L2SN 134136382 Ki = 6.04 nM T78709 CKH7W6 134137025 Ki = 5.012 nM T78709 C08ZBY 134137332 Ki = 1836 nM T78709 CD41CW 134137432 Ki = 2.9 nM T78709 CXF52V 134137560 Ki = 103 nM T78709 CN4LI8 134137732 Ki = 134 nM T78709 C5A6XO 134138438 Ki = 3.02 nM T78709 C90XZH 134138881 Ki = 15 nM T78709 CTP83K 134139510 Ki = 1.1 nM T78709 C7X6TJ 134139808 Ki = 5.4 nM T78709 CRC2V0 134139826 Ki = 2630 nM T78709 C8TC3Z 134140440 Ki = 2.12 nM T78709 CHK39T 134141166 Ki = 126 nM T78709 CLW86T 134141354 Ki = 1698.24 nM T78709 CXC80B 134142146 Ki = 1.3 nM T78709 C6PSI9 134142907 Ki = 3842 nM T78709 C46ZTY 134143085 Ki = 1.549 nM T78709 CVJ70S 134143778 Ki = 0.92 nM T78709 CR5L4K 134144303 Ki = 213.8 nM T78709 C80TGJ 134144864 Ki = 163 nM T78709 CWQG03 134145252 Ki = 0.81 nM T78709 CK37OV 134145259 Ki = 1.12 nM T78709 CK5RU9 134145903 Ki = 66 nM T78709 CLUV50 134145912 Ki = 1.4 nM T78709 C8AZ1F 134146083 Ki = 33 nM T78709 C8RI0E 134146106 Ki = 0.72 nM T78709 C2E0ID 134146185 Ki = 802 nM T78709 CC9P2T 134146194 Ki = 11 nM T78709 CV0QZ5 134147124 Ki = 365 nM T78709 C92WVK 134147870 Ki = 12.3 nM T78709 C41XSD 134147935 Ki = 6631 nM T78709 CL9RW7 134148069 Ki = 1.04 nM T78709 CBU81N 134149168 Ki > 10000 nM T78709 CEU53H 134149777 Ki = 0.9333 nM T78709 CA50EU 134150000 Ki = 29.3 nM T78709 CHK9J1 134150839 Ki = 1.56 nM T78709 CE6LN3 134151118 Ki = 74 nM T78709 CLU34D 134151427 Ki = 48.3 nM T78709 C2JN8Y 134151729 Ki = 202 nM T78709 CK23XB 134151891 Ki = 2.1 nM T78709 C76BZW 134151980 Ki = 160 nM T78709 CB14UF 134152029 Ki = 4 nM T78709 CIV4H5 134152583 Ki = 6064 nM T78709 CI0G7H 134153418 Ki = 39 nM T78709 CDWP64 134153527 Ki = 22.91 nM T78709 CB6M5Y 134153538 Ki = 41.69 nM T78709 CX4W7F 134153716 Ki = 109 nM T78709 C79TEI 134154068 Ki = 14.45 nM T78709 C9DQ4Y 134154208 Ki = 1.4 nM T78709 CMJ1U3 134154387 Ki = 138 nM T78709 CD80HF 134154490 Ki = 5 nM T78709 C4VGJ5 134154679 Ki = 9.9 nM T78709 C5SK4P 134154831 Ki = 0.36 nM T78709 CU6C4G 134154943 Ki = 5.3 nM T78709 C6QAY2 134155116 Ki = 18.62 nM T78709 C79QLN 134155460 Ki = 64.57 nM T78709 CIUZ94 134155476 Ki = 80 nM T78709 C90QNV 134155645 Ki = 101 nM T78709 CT5E7V 134155933 Ki = 2 nM T78709 CVR87Q 134156222 Ki = 122 nM T78709 CAB4K6 134156305 Ki = 147 nM T78709 C50XNE 134156520 Ki = 86 nM T78709 CUHE07 134157171 Ki = 160 nM T78709 C6S0VM 134157330 Ki = 3.02 nM T78709 CL6DN0 134157769 Ki = 152 nM T78709 C1GY2T 135156251 EC50 > 10000 nM T78709 C6N8GM 135367405 Ki > 10000 nM T78709 C6LU0C 135367816 Ki > 10000 nM T78709 CD2TH9 135367820 Ki > 10000 nM T78709 C5AMD9 135367857 Ki > 10000 nM T78709 CGBW93 135410312 Ki = 40.74 nM T78709 CVE08Y 135458392 Ki = 389 nM T78709 CP7HN4 135458393 Ki = 85 nM T78709 CS8XJ6 135458394 Ki = 246 nM T78709 C9B7XA 135458410 Ki = 124 nM T78709 CFV9A3 135458427 Ki = 240 nM T78709 CKX4N8 135458428 Ki = 53 nM T78709 C9ZCL5 135458672 Ki = 15560 nM T78709 C7DF4S 135464159 Ki = 323.59 nM T78709 CQDP70 135469307 Ki = 63 nM T78709 C7AGR0 135474338 Ki > 10000 nM T78709 CP9XN7 135500023 Ki = 11748.98 nM T78709 C34FXW 135501716 Ki = 2753 nM T78709 C6I9RK 135516645 Ki = 977.24 nM T78709 CQI23C 135516796 Ki = 1584.89 nM T78709 C3FV9I 135527031 Ki = 4168.69 nM T78709 CJF0P1 135600051 IC50 = 6.2 nM T78709 CD6L8Q 135895192 Ki = 1148 nM T78709 CA1M8B 135966709 Ki = 669 nM T78709 C6A8WK 136002690 IC50 = 46.6 nM T78709 C19GLK 136116062 Ki = 87 nM T78709 CA3JC8 136118613 Ki = 3445 nM T78709 CQ2GP6 136118614 Ki = 7361 nM T78709 C6R4IC 136118615 Ki = 7269 nM T78709 CS0JL5 136118616 Ki = 4608 nM T78709 C8RH6M 136118617 Ki = 2624 nM T78709 CHWC38 136118619 Ki > 10000 nM T78709 C5UDW3 136118620 Ki = 315 nM T78709 C8I6UN 136118621 Ki = 1812 nM T78709 C0W1TM 136118658 Ki = 6927 nM T78709 C40LYH 136118659 Ki = 2513 nM T78709 CZ7C3Y 136118660 Ki > 10000 nM T78709 C42FCS 136118661 Ki > 10000 nM T78709 CB12QP 136152964 Ki = 56 nM T78709 CFX06E 136152966 Ki = 348 nM T78709 C37YXA 136152971 Ki = 75 nM T78709 CY0C1X 136152972 Ki = 612 nM T78709 CSNE17 136179514 Ki = 478.63 nM T78709 CT0ZC8 136179515 Ki = 58.88 nM T78709 CX53NC 136180316 Ki = 36.6 nM T78709 CZ7WT9 136180317 Ki = 2.96 nM T78709 CQP2Y6 136180318 Ki = 75.3 nM T78709 CQT9H5 136180319 Ki = 43.5 nM T78709 CLPU18 136180320 Ki = 7.33 nM T78709 C0LO6Q 136180321 Ki = 116 nM T78709 C25RED 137631359 Ki = 0.5623 nM T78709 C9EIP8 137631570 EC50 = 30.8 nM T78709 CHM36P 137631892 Ki = 257 nM T78709 CVT4G8 137632024 Ki > 1000 nM T78709 CN1I7A 137634153 Ki > 20000 nM T78709 CC51JN 137635185 Ki > 10000 nM T78709 CNR82A 137635294 EC50 = 1300 nM T78709 C6DH9X 137635433 EC50 = 300 nM T78709 C0K3AP 137635725 EC50 > 10000 nM T78709 C94VXJ 137635884 Ki = 66 nM T78709 CFM92C 137636384 Ki > 10000 nM T78709 CF7KG5 137637817 Ki = 724 nM T78709 CDX39B 137637994 Ki = 370 nM T78709 C19JKQ 137638321 Ki = 1.122 nM T78709 CA03VC 137639125 Ki = 0.631 nM T78709 C1EK3W 137640451 Ki = 587 nM T78709 C3U5NF 137640522 EC50 = 680 nM T78709 CWQ80N 137640967 EC50 = 10.2 nM T78709 C3LYX9 137641832 Ki > 10000 nM T78709 C4I6QS 137641944 EC50 > 10000 nM T78709 C5WS6Q 137642134 Ki = 975 nM T78709 CU1O2P 137642386 Ki = 0.8913 nM T78709 CMJU75 137643395 EC50 = 28.6 nM T78709 CWUM83 137644521 Ki > 10000 nM T78709 CDA80E 137644790 Ki = 324 nM T78709 CHT42S 137645295 EC50 > 10000 nM T78709 CPCY48 137645406 Ki = 931 nM T78709 CZ8CU6 137645501 Ki = 40 nM T78709 CCP38D 137645926 Ki = 740 nM T78709 CVX74E 137646045 Ki = 5967 nM T78709 C96EAP 137646245 Ki = 0.6918 nM T78709 CPI68E 137646281 Ki = 0.22 nM T78709 C8PV0N 137646568 EC50 = 770 nM T78709 CO5U9A 137647674 EC50 = 1100 nM T78709 CMXI62 137649997 Ki = 749 nM T78709 CB4HG5 137650482 EC50 = 16.9 nM T78709 CWQF69 137650550 EC50 = 76.2 nM T78709 C52IRM 137650705 Ki = 54 nM T78709 CKG08R 137650961 Ki = 609 nM T78709 C47TWK 137651544 EC50 = 607 nM T78709 CW2L7Z 137651819 Ki = 0.7943 nM T78709 CU4S1W 137651887 Ki = 5 nM T78709 CVK26R 137652044 Ki = 543 nM T78709 CHFK13 137652210 Ki > 10000 nM T78709 C51CGJ 137652310 Ki = 759 nM T78709 C04XYN 137653567 EC50 = 10.5 nM T78709 C2E3FV 137653850 Ki = 32 nM T78709 C6N0DT 137654586 EC50 > 10000 nM T78709 CX82HS 137654666 Ki = 27 nM T78709 C0SKV1 137654850 Ki > 10000 nM T78709 C4VG0U 137655411 Ki = 29 nM T78709 CVEN03 137656381 EC50 = 69.7 nM T78709 CO3L7F 137656918 Ki > 10000 nM T78709 CEJ9L8 137657949 EC50 = 10.2 nM T78709 C3LHT5 137658253 EC50 = 32.9 nM T78709 C8G0HO 137658832 EC50 = 26.2 nM T78709 CFQ7C9 137659145 EC50 = 488 nM T78709 CLQX32 137659728 EC50 > 10000 nM T78709 CF9RZ5 137660385 EC50 = 450 nM T78709 CX4D7Y 137660741 Ki = 30 nM T78709 C9HPG8 137661516 IC50 = 600 nM T78709 C0R6XM 138691314 Ki = 1047 nM T78709 CU3Y7W 138691316 Ki = 1230 nM T78709 CH2W4P 138691317 Ki > 10000 nM T78709 CHSC40 138691321 Ki = 676 nM T78709 C18UZA 138691329 Ki = 9120 nM T78709 C1XWV0 138691338 Ki = 661 nM T78709 C6LE1A 138691362 Ki = 2138 nM T78709 CN9R4A 138691364 Ki = 123 nM T78709 C8H2KR 138691366 Ki = 2344 nM T78709 CJ43GI 139187858 Ki = 850 nM T78709 C47QCK 139187859 Ki = 3 nM T78709 C2Z9CD 139488518 Ki = 5623 nM T78709 CJK95T 139488527 Ki = 933 nM T78709 CZ6H9M 139488539 Ki = 316 nM T78709 CAF2H8 139488606 Ki = 589 nM T78709 C54CIL 139488740 Ki = 1738 nM T78709 CH7Y5D 141312275 Ki = 195 nM T78709 C4EU2S 141745651 Ki = 1.6 nM T78709 CCO6R0 141745657 Ki = 1.6 nM T78709 CO5DR9 145949220 Ki = 219 nM T78709 CWAF96 145949371 Ki = 85 nM T78709 CHG2W6 145950605 Ki = 305 nM T78709 COU57L 145950881 Ki = 140 nM T78709 CD4M6B 145951915 Ki = 18290 nM T78709 C5D1KR 145952639 EC50 = 1.2 nM T78709 C78AUI 145952711 Ki = 99 nM T78709 C8F3PN 145952866 EC50 > 10000 nM T78709 CA2J5S 145954503 Ki = 330400 nM T78709 C0JO8B 145954831 Ki = 421 nM T78709 CLJW61 145955880 Ki = 613 nM T78709 CHI1V8 145956064 Ki = 197 nM T78709 CSER68 145956892 Ki = 109 nM T78709 CLVI07 145957637 Ki = 18430 nM T78709 C91IDE 145958490 Ki = 341 nM T78709 C8VS7K 145959257 Ki = 2249 nM T78709 CSIZ31 145959706 Ki = 585 nM T78709 CD59BL 145960493 EC50 = 62.43 nM T78709 CXU82Q 145960544 EC50 = 93.37 nM T78709 CG8ZX0 145960719 EC50 < 0.14 nM T78709 CMO17A 145960744 Ki = 1.3 nM T78709 CQR07X 145960843 EC50 = 0.36 nM T78709 CDCS74 145960879 EC50 = 1563.21 nM T78709 CAJ7P6 145961144 Ki = 1 nM T78709 C59KNW 145961441 Ki = 2.2 nM T78709 CNF26K 145961458 EC50 = 34.98 nM T78709 CI4H8B 145961535 Ki = 92 nM T78709 C8PTZ7 145961730 Ki = 1 nM T78709 CP2M6G 145961773 EC50 = 0.58 nM T78709 CAE03F 145961788 EC50 = 28.8 nM T78709 CQ4RA7 145961842 Ki = 1.6 nM T78709 CBK15Q 145961968 EC50 = 0.35 nM T78709 C2TAU8 145962091 EC50 = 52 nM T78709 C1YE4Q 145962266 Ki = 1.5 nM T78709 CD6P4H 145962474 EC50 = 0.6 nM T78709 C8YS0D 145962581 EC50 = 0.75 nM T78709 C71HNB 145962633 Ki = 303 nM T78709 C7TM1V 145962678 EC50 = 146.01 nM T78709 C9G5YC 145962760 Ki = 253 nM T78709 C2A3DR 145962768 EC50 < 0.14 nM T78709 C56BKQ 145962801 Ki = 38 nM T78709 CVM9G4 145962946 Ki = 11 nM T78709 CFA09Q 145962985 Ki = 556 nM T78709 CO7P1B 145963059 Ki = 190 nM T78709 C4GS7B 145963079 EC50 = 0.72 nM T78709 CG94HV 145963146 EC50 = 1.55 nM T78709 C9B0SZ 145963169 Ki = 28 nM T78709 C2ZSA4 145963224 Ki = 1.6 nM T78709 CDTR93 145963270 Ki = 0.8 nM T78709 C4Y1PK 145963314 Ki = 100 nM T78709 CVM9W0 145963420 EC50 = 567 nM T78709 CHZ5I6 145963710 EC50 = 14.93 nM T78709 CNA8I5 145963810 Ki = 2 nM T78709 C7KC3T 145963830 IC50 > 10000 nM T78709 C5VWM7 145963860 Ki = 1169 nM T78709 CCK5G1 145963863 Ki = 1961 nM T78709 CEN94V 145963961 EC50 = 2.2 nM T78709 C3I6YP 145963975 EC50 > 100000 nM T78709 CV7YW9 145964086 Ki = 962 nM T78709 CE32PV 145964143 Ki = 5.4 nM T78709 CHDN35 145964150 IC50 > 10000 nM T78709 CR2B9G 145964154 Ki = 2058 nM T78709 C1KH2E 145964159 IC50 > 10000 nM T78709 C1B8QW 145964299 EC50 = 9 nM T78709 C7YKQ4 145964390 Ki = 8966 nM T78709 C95NZO 145964427 Ki = 32 nM T78709 C2P5NK 145964621 Ki = 1266 nM T78709 C0N8KC 145964622 EC50 = 28.1 nM T78709 CK0T1M 145964694 Ki = 742 nM T78709 C6T4RY 145964846 Ki = 20 nM T78709 C24NSP 145964857 Ki = 0.9 nM T78709 CE9K3L 145964944 Ki = 0.84 nM T78709 C7MBS0 145964982 EC50 > 100000 nM T78709 C7JS9I 145965041 EC50 = 117 nM T78709 C9D8IB 145965203 Ki = 2 nM T78709 C5DL3N 145965355 Ki = 14 nM T78709 C1MIR9 145965401 Ki = 496 nM T78709 CV07EO 145965433 EC50 > 100000 nM T78709 C9KXP6 145965474 Ki = 1350 nM T78709 CLP94W 145965668 Ki = 1096 nM T78709 C8TF9G 145965840 Ki = 13790 nM T78709 C53EFW 145966154 Ki = 388 nM T78709 CB05QA 145966199 Ki = 1322 nM T78709 CLM10C 145966333 EC50 = 1.2 nM T78709 C1T4DN 145966418 Ki = 2687 nM T78709 CRS7V6 145966748 Ki = 50 nM T78709 C5L4WF 145967359 EC50 = 17.6 nM T78709 CV03XA 145967457 Ki = 1951 nM T78709 CL58XS 145967572 Ki = 9.4 nM T78709 C58WSL 145967904 Ki = 272 nM T78709 C76SHX 145968149 Ki = 2.41 nM T78709 C3DZ7P 145968324 Ki = 42.8 nM T78709 C3D0LR 145968390 Ki = 11.3 nM T78709 CT09GI 145968506 Ki = 19.3 nM T78709 C9S8QE 145968791 Ki = 57.8 nM T78709 CB1FD8 145968810 Ki = 110 nM T78709 CM0Z9G 145968895 Ki = 2.25 nM T78709 CM6HG9 145968927 EC50 = 16.5 nM T78709 C2A0FO 145969167 EC50 > 100000 nM T78709 CVU49S 145969204 Ki = 19 nM T78709 CQ8EM6 145969402 Ki = 3755 nM T78709 CI5R8W 145969406 Ki = 0.5 nM T78709 CERC65 145969459 Ki = 69.9 nM T78709 CD3Z4I 145969495 Ki = 546 nM T78709 C48XNG 145969667 Ki = 15 nM T78709 CNZY06 145969934 Ki = 19 nM T78709 C3FNX8 145969978 Ki = 16 nM T78709 CRZN24 145970238 Ki = 251 nM T78709 CT2LQ4 145970743 Ki = 8.8 nM T78709 CQC6Y1 145970782 Ki = 1 nM T78709 C6FBU7 145970863 Ki = 43.1 nM T78709 C61MSO 145970938 Ki = 326 nM T78709 CF74MR 145971390 Ki = 1428 nM T78709 C1T7GL 145971527 Ki = 6100 nM T78709 CRC9T0 145971556 EC50 = 0.9 nM T78709 C8A2XG 145971561 Ki = 4054 nM T78709 CN64ZR 145971588 Ki = 770 nM T78709 CB43OV 145971604 Ki = 3.5 nM T78709 CQJ5O8 145971635 IC50 > 10000 nM T78709 C56RAO 145972025 Ki = 14900 nM T78709 C7BVC1 145972374 IC50 > 10000 nM T78709 CR06QO 145972382 EC50 > 100000 nM T78709 CWRM23 145972513 EC50 = 12.8 nM T78709 CJHI43 145972875 Ki = 1792 nM T78709 C1QY4E 145973003 Ki = 0.6 nM T78709 CS7WG8 145973438 Ki = 3198 nM T78709 C8KYV6 145973487 Ki = 2669 nM T78709 C0H1JO 145973539 Ki = 3168 nM T78709 CL74IP 145973853 Ki = 190 nM T78709 CT51VH 145974031 Ki = 0.9 nM T78709 CR0CX6 145974087 Ki = 184 nM T78709 C6AGN3 145974143 EC50 = 176 nM T78709 C8KZ5T 145974165 Ki = 6.3 nM T78709 C05IVJ 145974184 Ki = 8687 nM T78709 CW6EX3 145974189 Ki = 2081 nM T78709 C9L7EM 145974368 Ki = 2.5 nM T78709 CDOJ39 145974939 EC50 = 0.7 nM T78709 C3WG0J 145975106 Ki = 1630 nM T78709 CR83MU 145975214 EC50 = 23.6 nM T78709 C6PH4F 145975226 IC50 > 10000 nM T78709 CN8U3P 145975289 Ki = 1411 nM T78709 CJF4Z0 145975393 EC50 > 100000 nM T78709 CZ39GQ 145975595 EC50 > 100000 nM T78709 CSVR94 145975713 Ki = 4067 nM T78709 COY2P3 145975720 Ki = 14160 nM T78709 CL7EX5 145975776 Ki = 552 nM T78709 C1BI8E 145975778 Ki = 2368 nM T78709 C7R2MD 145975905 Ki = 6005 nM T78709 C71CYU 145975946 IC50 > 10000 nM T78709 C0V4AL 145975992 Ki = 52010 nM T78709 C2TN8W 145976085 IC50 > 10000 nM T78709 C8XFM7 145976120 Ki = 146 nM T78709 CF5B0W 145976158 Ki = 2211 nM T78709 CB2R6J 145976187 Ki = 1.5 nM T78709 C8BJI2 145976292 Ki = 1839 nM T78709 C90NFP 145976326 Ki = 1.48 nM T78709 CCDU50 145976348 EC50 = 42.3 nM T78709 CZ5XK2 145976408 Ki = 2891 nM T78709 C14OJW 145976618 Ki = 297 nM T78709 C0LRB2 145976686 Ki = 2677 nM T78709 C34XME 145976696 Ki = 5 nM T78709 CTCM92 145976698 Ki = 2349 nM T78709 CIZ69S 145976722 Ki = 462 nM T78709 C9FR7N 145976732 EC50 = 11.3 nM T78709 CNCS36 145976746 Ki = 3.7 nM T78709 CT7WO5 145976787 Ki = 4358 nM T78709 CI8AN3 145976890 Ki = 696 nM T78709 C81CSM 145976946 Ki = 1545 nM T78709 C8NW7Y 145977256 Ki = 3949 nM T78709 CHS96B 145977297 Ki = 2.4 nM T78709 C8DP4I 145977442 Ki = 11 nM T78709 C4L8EZ 145977467 Ki = 619 nM T78709 CC1DZ5 145977555 Ki = 2077 nM T78709 C0Y6QO 145977799 IC50 > 10000 nM T78709 CP8C6M 145978146 Ki = 506 nM T78709 C72SMR 145978208 EC50 = 6.2 nM T78709 C6HQI0 145978420 Ki = 509 nM T78709 C8VL3Y 145978472 Ki = 48240 nM T78709 C82NXP 145978482 Ki = 1456 nM T78709 C1Q2BR 145978965 EC50 = 17.4 nM T78709 C20XQJ 145979626 Ki = 6216 nM T78709 C2PK6X 145980101 Ki = 0.3 nM T78709 C87MSW 145980271 Ki = 1094 nM T78709 CW2CO4 145980458 Ki = 19 nM T78709 CD92WV 145980513 Ki = 1304 nM T78709 C8I7QL 145980875 Ki = 901 nM T78709 C6H7SC 145981004 Ki = 0.4 nM T78709 CC2UQ5 145981118 Ki = 186 nM T78709 C4AF0G 145981310 EC50 > 100000 nM T78709 C67AIW 145981408 EC50 = 2.4 nM T78709 CPK34X 145981875 Ki = 8.1 nM T78709 C7LBY5 145982138 Ki = 4 nM T78709 COY79P 145982165 Ki = 326 nM T78709 CO7WP6 145982353 EC50 = 10.5 nM T78709 CEK60A 145982506 Ki = 14 nM T78709 CI59TX 145983018 Ki = 23 nM T78709 CYC58R 145983059 Ki = 9 nM T78709 C4F5OT 145983128 Ki = 5 nM T78709 C5ZG9M 145983139 Ki = 179 nM T78709 CV2GU9 145983144 Ki = 146 nM T78709 C4PKM2 145983390 Ki = 50 nM T78709 C9LR8C 145983405 Ki = 18 nM T78709 CIAF74 145983468 Ki = 54 nM T78709 CE7MF4 145983751 Ki = 24 nM T78709 CDQ4U7 145983760 Ki = 12 nM T78709 CYW9B2 145983794 Ki = 12 nM T78709 C1DW4U 145983928 EC50 = 3.6 nM T78709 C8I1WG 145983961 Ki = 14 nM T78709 CP5H4D 145984065 Ki = 147 nM T78709 C58DHN 145984151 EC50 = 13.3 nM T78709 CJ35DM 145984299 Ki = 37 nM T78709 CU7E4M 145984511 Ki = 56 nM T78709 C6JUY0 145984737 Ki = 37 nM T78709 CID02G 145984807 Ki = 27 nM T78709 CP9D3A 145984902 Ki = 0.3 nM T78709 CM5X3V 145985050 Ki = 111 nM T78709 CG10LK 145985224 Ki = 48 nM T78709 CFJ9B3 145985233 Ki = 147 nM T78709 C5AOI6 145985289 Ki = 8 nM T78709 CW30NA 145985505 Ki = 86 nM T78709 C7ZRP1 145985527 Ki = 91 nM T78709 C2XY8Q 145985533 Ki = 25 nM T78709 C7NI4X 145985585 Ki = 96 nM T78709 C9LJ5T 145985692 Ki = 16 nM T78709 C7QIX0 145985718 Ki = 28 nM T78709 C6V5QS 145985823 Ki = 120 nM T78709 C07GKD 145985958 Ki = 36 nM T78709 CCM18E 145986031 Ki = 15 nM T78709 CR0XQ3 145986138 Ki = 16 nM T78709 CXC79K 145986552 EC50 = 47.9 nM T78709 COT25D 145986575 Ki = 468 nM T78709 CT37DW 145986720 Ki = 15150 nM T78709 CNJH37 145986752 Ki = 10000 nM T78709 C3VN5O 145987559 Ki = 5211 nM T78709 CZ5O8R 145987659 EC50 = 107 nM T78709 CI0PA9 145987771 Ki = 28 nM T78709 COS58J 145987942 EC50 = 10.6 nM T78709 C6MHU2 145988006 EC50 = 3.1 nM T78709 C9ZBE8 145988017 Ki = 3 nM T78709 CHOB70 145988038 EC50 = 1.6 nM T78709 CO4LK7 145988180 Ki = 12 nM T78709 CIS9P2 145988193 Ki = 62 nM T78709 C86XQR 145988313 Ki = 603 nM T78709 C9W1QA 145988497 EC50 = 8.8 nM T78709 CUGO10 145988693 Ki = 1262 nM T78709 C9D2OG 145988738 Ki = 129 nM T78709 C4C0YP 145988913 Ki = 21470 nM T78709 CDY48U 145989143 Ki = 0.53 nM T78709 CVC14L 145989181 EC50 = 91.3 nM T78709 CR2EV8 145989183 EC50 = 11.6 nM T78709 C39CSX 145989329 Ki = 154 nM T78709 CMJL94 145989451 EC50 = 6.1 nM T78709 CB6OP0 145989720 Ki = 8.76 nM T78709 C3GPR9 145990093 Ki = 377500 nM T78709 C41SBL 145990126 EC50 = 1.7 nM T78709 C2Q5UK 145990353 Ki = 128 nM T78709 CK5IA4 145990443 Ki = 6 nM T78709 CT7AB8 145990459 Ki = 5577 nM T78709 CE9PT1 145990482 EC50 = 3.3 nM T78709 C4GV8Q 145990586 Ki = 71 nM T78709 CKWF21 145990750 Ki = 1210 nM T78709 CMJ46R 145990794 EC50 = 6.9 nM T78709 CVBR36 145991084 Ki = 5.6 nM T78709 C5TNP0 145991127 EC50 = 1.1 nM T78709 CW14AE 145991244 EC50 > 100000 nM T78709 C7RJ4E 145991363 Ki = 11 nM T78709 CU6E1Z 145991746 EC50 = 13.8 nM T78709 C9TK6G 145991864 Ki = 15 nM T78709 CI1EQ3 145991900 Ki = 159 nM T78709 C9WME0 145992265 Ki = 0.4 nM T78709 CB8CM6 145992305 Ki = 1155 nM T78709 C5DVK4 145992403 Ki = 308 nM T78709 CCP2U1 145992489 Ki = 1363 nM T78709 CELG57 145992523 EC50 = 5.8 nM T78709 CLPU06 145992567 Ki = 413200 nM T78709 CB64KH 145992860 EC50 = 3.6 nM T78709 CBI94R 145992877 Ki = 13 nM T78709 C9PS8N 145993117 EC50 = 1.24 nM T78709 CT63XO 145993172 EC50 = 0.9 nM T78709 CI19KS 145993474 Ki = 25 nM T78709 C0Z6YX 145993493 EC50 = 7.7 nM T78709 C17HSV 145993577 EC50 = 1.2 nM T78709 C0TL8E 145993714 Ki = 1225 nM T78709 CX1N0L 145993740 Ki = 450 nM T78709 CO1BX3 145994087 Ki = 161 nM T78709 CS1LF2 145994186 Ki = 1.2 nM T78709 CC2G1V 146025727 Ki = 3700 nM T78709 C5ZOJ3 146680920 Ki = 5009 nM T78709 CG97ER 146709966 Ki = 2511.89 nM T78709 CF5B2L 147653864 Ki = 1000 nM T78709 C5PNX8 148302367 Ki = 1995.26 nM T78709 C9T0PS 153061504 Ki = 316.23 nM T78709 C1FA0K 153287541 Ki = 199.53 nM T78709 CEQ69Z 153287542 Ki = 199.53 nM T78709 C6P3SR 153287553 Ki > 10000 nM T78709 CW31CT 153287566 Ki = 199.53 nM T78709 CV9G7Z 153287572 Ki = 1995.26 nM T78709 CO85KL 153287574 Ki = 74 nM T78709 CZ1K4D 155510674 Ki = 4 nM T78709 CLX3D8 155510732 EC50 = 1180 nM T78709 CC3KP7 155510927 Ki > 10000 nM T78709 CM4RB0 155511262 Ki = 64 nM T78709 C0K7OA 155511383 EC50 > 100000 nM T78709 C9KX6O 155511928 Ki = 197 nM T78709 CZ7HP4 155512406 Ki = 993 nM T78709 C4OL0A 155512409 Ki = 5.15 nM T78709 C2H6LN 155512422 Ki = 52 nM T78709 CXF90M 155512487 Ki = 1010 nM T78709 C7N0VH 155512508 Ki > 1000 nM T78709 C1WG0H 155512850 EC50 = 100 nM T78709 CO68LC 155512944 Ki = 2344 nM T78709 C4Q5SY 155512981 Ki = 140 nM T78709 C90FST 155513438 Ki = 399 nM T78709 C36RDV 155513614 Ki = 327 nM T78709 C6DP0E 155513883 Ki = 218 nM T78709 C7W1OH 155513940 Ki = 1.549 nM T78709 C7FI9W 155514217 Ki = 84 nM T78709 CRP43D 155514341 IC50 > 1000 nM T78709 C95QOT 155514378 Ki = 2944 nM T78709 CK9YN0 155514430 Ki = 2260 nM T78709 CI4DT8 155514575 Ki = 126 nM T78709 CJUI87 155514774 Ki = 23 nM T78709 CM5A8F 155514858 Ki = 130 nM T78709 CQ84DA 155514889 Ki = 64 nM T78709 C21QLC 155515074 Ki = 63 nM T78709 CV8F7A 155515301 Ki = 12.02 nM T78709 C4X2RG 155515318 Ki = 431 nM T78709 C3NB0D 155515324 Ki > 1000000 nM T78709 C0Q8PR 155515407 Ki = 688 nM T78709 CWO56B 155515415 Ki > 10000 nM T78709 CU0PY6 155515687 Ki = 3.84 nM T78709 C2TN5D 155515890 Ki = 32 nM T78709 CW6O5J 155515898 Ki = 47 nM T78709 C7KT0D 155515919 Ki > 10000 nM T78709 C13LOV 155515942 Ki = 1872 nM T78709 CUM2N4 155515982 Ki = 17 nM T78709 C7OF4C 155516118 Ki = 6204 nM T78709 CG5M1O 155516282 Ki = 291 nM T78709 CG53LH 155516399 Ki = 40.4 nM T78709 C6X9UC 155516902 Ki = 76 nM T78709 CT4U8D 155517137 Ki = 28.18 nM T78709 CU8TC0 155517162 Ki = 12 nM T78709 CEA9D5 155517238 Ki = 157 nM T78709 CW0B5K 155518159 Ki > 10000 nM T78709 C87RWX 155518489 Ki = 431 nM T78709 CYB12O 155518974 Ki = 3569 nM T78709 CHVF41 155519045 Ki = 808 nM T78709 CCEZ93 155519102 Ki = 4540 nM T78709 CQD2J7 155519393 Ki = 1052 nM T78709 C2SXT1 155519515 Ki = 132 nM T78709 C0KLD8 155519559 Ki = 5036 nM T78709 CAV5Y1 155519565 Ki = 269.15 nM T78709 C07BTO 155519598 Ki = 54 nM T78709 CUSA24 155519891 Ki = 1000 nM T78709 C5FL7R 155520499 Ki = 482 nM T78709 C8OC3W 155520552 Ki = 149 nM T78709 CO1B0G 155520918 Ki = 233 nM T78709 CTV2F6 155521010 Ki > 1000 nM T78709 C17QKW 155521049 Ki = 134 nM T78709 CW0AM2 155521520 EC50 = 54400 nM T78709 CG2F9X 155521599 Ki = 261 nM T78709 CL07FB 155521817 Ki = 213.8 nM T78709 CWQ1D2 155521828 Ki = 378 nM T78709 CL20TG 155522125 EC50 > 100000 nM T78709 C98RDQ 155522218 Ki = 22 nM T78709 CAFT73 155522329 Ki = 68.7 nM T78709 CP6H1D 155522562 Ki = 46 nM T78709 CUQ61M 155522867 Ki = 21.2 nM T78709 CXEB36 155523275 Ki = 9.55 nM T78709 CD9QU6 155523519 Ki = 9 nM T78709 C2Y9CW 155523745 Ki = 220 nM T78709 C4NOD0 155524193 Ki = 1720 nM T78709 C5KYB4 155524228 Ki = 3.2 nM T78709 C7F2ZG 155524366 Ki = 240 nM T78709 CK4B0R 155524491 Ki = 8 nM T78709 CRF5T8 155524643 EC50 > 100000 nM T78709 CYZ60F 155524736 Ki = 70.79 nM T78709 CUO93F 155524808 Ki = 19 nM T78709 C65UZD 155524956 Ki = 106 nM T78709 CZQ5M2 155525523 Ki = 155 nM T78709 CR3DZ7 155525571 Ki = 203 nM T78709 CD5BI1 155525649 Ki = 5.248 nM T78709 C6MZJ9 155525703 Ki = 12 nM T78709 C81OCJ 155526014 Ki = 81.8 nM T78709 CZ81JA 155526026 Ki = 26 nM T78709 C68VNI 155526159 EC50 = 1600 nM T78709 CF7B3L 155526557 Ki = 50 nM T78709 CPCK60 155526570 Ki = 2860 nM T78709 C0MX4T 155526627 Ki = 66 nM T78709 C8GC1P 155526628 Ki = 0.5012 nM T78709 C1U2XO 155526651 Ki = 22 nM T78709 CXH79K 155526720 Ki = 38 nM T78709 CP76JX 155526977 Ki = 2511.89 nM T78709 C46NXV 155527302 Ki = 24.1 nM T78709 C6BHY8 155527304 Ki = 102 nM T78709 C3PS9Z 155527787 Ki = 290 nM T78709 CEQ8O4 155527891 Ki = 135 nM T78709 CL6XH7 155528009 Ki = 236 nM T78709 CIO6V1 155528183 Ki = 181.97 nM T78709 CHJ79N 155528236 Ki = 222 nM T78709 CRA6L0 155528255 Ki = 183 nM T78709 CW68KC 155528355 Ki > 10000 nM T78709 C7C1EF 155528967 Ki = 46 nM T78709 C7FR8Y 155529117 Ki = 11.48 nM T78709 C5J7AU 155529153 Ki = 5311 nM T78709 CF2DM6 155529314 Ki = 1.349 nM T78709 C9KS5C 155529450 Ki = 25 nM T78709 CEN90X 155529453 Ki = 125 nM T78709 CKZ25Y 155529679 Ki = 156 nM T78709 CD0C5A 155529797 Ki = 25 nM T78709 CGA7H6 155530006 Ki = 1074 nM T78709 C5T1OG 155530093 Ki = 239 nM T78709 C3X4IA 155530328 Ki = 21 nM T78709 C9PC3D 155530350 Ki = 989 nM T78709 C12AMJ 155530737 Ki = 321 nM T78709 CVLC03 155530779 Ki = 91 nM T78709 C98YQF 155531012 Ki = 54 nM T78709 C4W6VC 155531065 Ki = 292 nM T78709 C3ZL2V 155531279 Ki = 20.42 nM T78709 C5HWP4 155531362 Ki > 10000 nM T78709 CXOT20 155531661 Ki = 40 nM T78709 CKDE38 155531753 Ki = 1 nM T78709 C9YMR2 155531801 Ki = 194 nM T78709 CCT8V9 155531846 Ki = 8726 nM T78709 CLZY37 155531982 Ki = 24.1 nM T78709 CE3T7O 155532050 Ki = 52 nM T78709 C05KFL 155532137 Ki = 964 nM T78709 C3R4YM 155532148 Ki = 5.012 nM T78709 CS0L4A 155532204 Ki = 476 nM T78709 CX35QS 155532545 Ki > 10000 nM T78709 C3MXL6 155532834 Ki = 0.7762 nM T78709 CX6DV4 155533028 Ki = 9473 nM T78709 CTU64O 155533099 Ki = 7.244 nM T78709 C23GDV 155533534 Ki = 13 nM T78709 C3OEH2 155533648 Ki = 373 nM T78709 CZA89B 155533824 EC50 = 27.7 nM T78709 CY01GZ 155533850 Ki = 30 nM T78709 C3L0CP 155534184 Ki = 15 nM T78709 CG85SB 155534301 Ki = 94 nM T78709 CG8Y7W 155534312 Ki = 856 nM T78709 CSE59K 155534331 Ki = 336 nM T78709 C3VGT0 155534362 Ki = 42 nM T78709 CW7SV9 155534575 Ki = 24 nM T78709 CVWX57 155534647 Ki = 69 nM T78709 C8R2TB 155534729 Ki = 143.2 nM T78709 C75FSY 155534794 Ki > 10000 nM T78709 CTO4S9 155534839 Ki = 8.4 nM T78709 CU3YE7 155534933 Ki = 75.86 nM T78709 C6KF4E 155535154 Ki = 52 nM T78709 C1E7OC 155535162 Ki = 259 nM T78709 CGZ5T8 155535272 Ki = 37 nM T78709 C35NRU 155535386 Ki = 700 nM T78709 C8O4IQ 155535827 Ki = 17 nM T78709 C14JEX 155535878 Ki > 10000 nM T78709 C7YNR9 155535901 Ki = 142 nM T78709 CB79ZW 155536080 Ki = 630.96 nM T78709 C5I1JA 155536087 Ki = 12 nM T78709 CHMV76 155536112 Ki = 136 nM T78709 C72FLG 155536152 Ki = 1610 nM T78709 CQG68A 155536202 Ki = 60.26 nM T78709 CW2SC8 155536533 Ki = 40.4 nM T78709 CLZ01I 155536626 Ki = 132 nM T78709 CTB93R 155536809 Ki = 1684 nM T78709 C6LVS4 155536841 Ki = 122 nM T78709 C7FVE8 155537034 Ki = 220 nM T78709 C36FRH 155537074 Ki = 732 nM T78709 C6CFE2 155537427 Ki = 261 nM T78709 C1T8XW 155537724 Ki = 23 nM T78709 CVS04L 155537788 Ki = 369 nM T78709 CQ0WD1 155537995 Ki = 1780 nM T78709 CB8IC7 155538144 Ki = 3311 nM T78709 C5F2GI 155538236 Ki = 27 nM T78709 COYG20 155538350 Ki = 45 nM T78709 C9TIU2 155538367 Ki = 1698 nM T78709 CYC1P3 155538451 Ki = 28 nM T78709 CM08NT 155538716 Ki > 10000 nM T78709 CQ69UA 155538814 Ki = 7505 nM T78709 C0Q5NT 155538877 Ki = 489 nM T78709 CC89JF 155539461 Ki = 209 nM T78709 CAT98F 155539483 Ki = 7 nM T78709 C70SWG 155539596 Ki = 102 nM T78709 C6S8BA 155539600 Ki = 3384 nM T78709 CV9KY1 155539925 Ki = 204.1 nM T78709 C42GUK 155540147 Ki > 10000 nM T78709 C1X0IO 155540198 Ki = 350 nM T78709 C9J3BQ 155540635 Ki = 328 nM T78709 C1KA8C 155540755 Ki = 13.4 nM T78709 CR2K1T 155540795 Ki > 10000 nM T78709 CNU92V 155540807 Ki = 6.3 nM T78709 CUY87S 155540823 Ki = 15.2 nM T78709 COS2E7 155541072 Ki > 10000 nM T78709 C6B7QU 155541341 Ki = 333 nM T78709 C6SU1V 155541676 Ki > 10000 nM T78709 CP7UG2 155541866 Ki = 334 nM T78709 COZ46W 155541871 Ki = 43 nM T78709 CFH7K5 155542074 Ki = 724.44 nM T78709 CXCW81 155542321 Ki = 12530 nM T78709 C9FS3Y 155542461 Ki > 10000 nM T78709 C18OPI 155542619 Ki = 752 nM T78709 C9RV7W 155542678 Ki = 562 nM T78709 CT6HY4 155543250 Ki = 1230 nM T78709 C68MSK 155543653 Ki = 3438 nM T78709 C0QN3W 155543949 Ki = 48.7 nM T78709 CZ7O0A 155544139 Ki = 3584 nM T78709 CY57ZS 155544392 Ki = 139 nM T78709 C91VXF 155544397 Ki = 66.07 nM T78709 CR54LA 155544513 Ki = 3.162 nM T78709 CD84VK 155544810 Ki = 66 nM T78709 C3ZS0K 155544812 Ki = 294 nM T78709 C0YE6V 155544819 Ki = 78 nM T78709 C2XZD8 155545087 Ki = 79 nM T78709 CD39HU 155545397 IC50 > 1000 nM T78709 CI0YL8 155545625 Ki > 10000 nM T78709 CXI7S8 155545989 Ki = 50 nM T78709 C74GFO 155546189 Ki = 81 nM T78709 CCK3D7 155546303 Ki = 28 nM T78709 CH3W9N 155546350 Ki > 10000 nM T78709 C4C9NO 155546587 EC50 = 10100 nM T78709 C4UT5Z 155546595 Ki = 132 nM T78709 C98AIL 155546781 Ki = 128 nM T78709 C2KM3J 155547346 EC50 = 107 nM T78709 CD02EN 155547436 Ki = 47 nM T78709 CFL6E5 155547451 Ki = 42 nM T78709 COJ27N 155547693 Ki = 15070 nM T78709 CAT9X4 155548275 Ki > 10000 nM T78709 C87JGN 155549153 Ki > 10000 nM T78709 CGP8O5 155549315 Ki = 19 nM T78709 CXH9A8 155549493 Ki = 173.78 nM T78709 C3KXY1 155549528 Ki = 378 nM T78709 C52FRY 155549978 Ki = 20 nM T78709 C7YO2N 155550741 EC50 = 85000 nM T78709 C8HPN7 155551113 Ki = 64 nM T78709 C61IVC 155551353 Ki = 832 nM T78709 CHS71N 155551685 Ki = 58 nM T78709 CM26AV 155551704 Ki = 85 nM T78709 C6E9LK 155552054 Ki = 47 nM T78709 C3JEN6 155552089 Ki = 35.8 nM T78709 CX8JA1 155552185 Ki = 34 nM T78709 CQ48CS 155552188 Ki = 6.3 nM T78709 CA1WS9 155552212 Ki = 122 nM T78709 C38YJB 155552311 Ki = 142 nM T78709 C52FJU 155552469 Ki = 105 nM T78709 C0DQ3Z 155552695 Ki = 4400 nM T78709 C87PTM 155552707 Ki = 15 nM T78709 C92UAC 155552738 Ki = 62 nM T78709 CUXK56 155552760 Ki = 261 nM T78709 CDQ7C2 155552798 Ki = 536 nM T78709 C9XQ8H 155552820 Ki = 23.44 nM T78709 CPV35U 155552826 Ki > 10000 nM T78709 CBW52M 155553110 Ki = 486 nM T78709 CDV6B9 155554036 Ki = 5467 nM T78709 CFY5S4 155554150 Ki = 53 nM T78709 CKF75H 155554324 Ki = 181 nM T78709 CINW85 155554326 Ki = 91 nM T78709 C6ZSU3 155554462 Ki = 4389 nM T78709 C8JKT1 155555378 Ki = 16.4 nM T78709 C2E5TR 155555506 Ki = 775 nM T78709 CUNK28 155555525 Ki > 10000 nM T78709 CXM7C6 155555638 Ki = 246 nM T78709 C4LOH3 155555858 Ki = 15.49 nM T78709 CYP63A 155556311 Ki = 243 nM T78709 CO52HW 155556527 Ki > 10000 nM T78709 CO3G4A 155556672 Ki = 147 nM T78709 C1N5VF 155556756 Ki > 10000 nM T78709 C27JYZ 155556785 EC50 > 100000 nM T78709 CJCL47 155556806 Ki = 102 nM T78709 C5QYS0 155557134 Ki = 48 nM T78709 CXN47Z 155557425 Ki = 214 nM T78709 CD2L3K 155557443 Ki = 200 nM T78709 C8EM5K 155557592 Ki = 376 nM T78709 C0CV6O 155557695 Ki = 4.571 nM T78709 C2L0PC 155557720 Ki = 7 nM T78709 C3UCM2 155557792 Ki = 3.981 nM T78709 C9LA1I 155558180 EC50 > 500000 nM T78709 CF6H3V 155558408 Ki = 7688 nM T78709 C4I2OY 155558563 Ki = 2.1 nM T78709 C20QMI 155558704 Ki = 54.95 nM T78709 C4AG0H 155558726 Ki = 420 nM T78709 C9TB5D 155559092 Ki = 302 nM T78709 CI3G0A 155559625 Ki = 176 nM T78709 CE0HN5 155559841 Ki = 97.72 nM T78709 C3Y4RD 155560781 EC50 > 100000 nM T78709 COG70U 155560942 Ki > 10000 nM T78709 C75RMN 155561496 Ki = 1.2 nM T78709 C2HF6P 155561581 Ki = 3176 nM T78709 COL7N8 155561901 Ki = 263 nM T78709 CL45NV 155561914 Ki = 599 nM T78709 CJ57BI 155561978 Ki = 53 nM T78709 C0SDZ8 155561990 IC50 = 500 nM T78709 CW7M1D 155561995 Ki = 31 nM T78709 C8ZKT3 155562124 Ki = 1.862 nM T78709 C93KWN 155562202 Ki = 20 nM T78709 CO3C6L 155562423 Ki > 10000 nM T78709 C5AI0S 155562519 Ki = 4.9 nM T78709 C5BQ8U 155562652 Ki = 62 nM T78709 CF6B4W 155562834 Ki = 35 nM T78709 CZ6IA2 155562918 Ki = 14160 nM T78709 CYD62V 155562962 Ki = 281 nM T78709 CRCW25 155562997 Ki = 13 nM T78709 C71MOD 155563001 Ki = 1.995 nM T78709 CGC8W7 155563143 Ki = 80 nM T78709 CBH14K 155563164 Ki > 10000 nM T78709 CV9O7W 155563205 Ki > 5000 nM T78709 CG1L8E 155563286 Ki > 10000 nM T78709 C38WXS 155563374 Ki = 2467 nM T78709 C0INS4 155563826 Ki > 10000 nM T78709 CK0IW3 155563911 Ki = 37 nM T78709 C3OK2L 155565059 Ki = 160 nM T78709 CR12DI 155565189 Ki = 310 nM T78709 CQK8E3 155565209 Ki = 101 nM T78709 CE2YG1 155565215 Ki = 134 nM T78709 C3DK0P 155565218 Ki = 57.54 nM T78709 CESG75 155565298 EC50 = 11400 nM T78709 CVU9O2 155565448 Ki = 25.7 nM T78709 C19PZX 155565707 Ki = 213.8 nM T78709 CJ61GD 155565772 Ki = 257 nM T78709 C2MIU5 155565813 Ki = 202 nM T78709 C9C6WD 155565990 EC50 = 2200 nM T78709 C7P5VG 155566191 Ki = 120 nM T78709 C0D8ZO 155566396 Ki = 157 nM T78709 C5KDA9 155566405 Ki = 35.8 nM T78709 C7O6YP 155566439 Ki = 28510 nM T78709 C67LAG 155566854 Ki > 10000 nM T78709 CW1TN7 155566925 Ki = 1072 nM T78709 CRX52O 155567200 Ki = 1.622 nM T78709 C41UWT 155567307 Ki = 22 nM T78709 CBJ7M2 155567312 Ki = 50 nM T78709 CA8OE0 155567476 Ki = 2306 nM T78709 CC06FO 155567938 Ki = 38.7 nM T78709 CA68TK 155568224 Ki = 1680 nM T78709 C4EX7C 155568246 Ki = 2.3 nM T78709 C4POS3 155568373 Ki = 33.5 nM T78709 C67MIN 155568606 Ki = 0.2 nM T78709 CV5H3F 155568689 Ki = 320 nM T78709 CXP3E4 155568794 Ki = 146 nM T78709 CB5IP9 155569021 Ki = 161 nM T78709 C0CZK6 155569337 Ki > 10000 nM T78709 CP9V7M 155569396 Ki = 4365 nM T78709 C3ZNX6 155569414 Ki = 13 nM T78709 CZ8RV4 155569568 Ki = 218 nM T78709 C3N9VU 10251906 Ki > 500 nM T78709 CP9TR0 10324985 EC50 = 0.01 nM T78709 CQ1LV7 135508617 Ki = 527 nM T78709 CRKP76 136016509 Ki = 3215 nM T78709 C9J5HY 16105548 Ki = 16 nM T78709 C4ZD3A 16105549 Ki = 21 nM T78709 CFMK68 3246545 Ki = 64 nM T78709 CB2VD8 44241743 Ki = 1480 nM T78709 C13REG 44471685 Ki = 93.5 nM T78709 D00AVR 135476741 Ki > 10000 nM T78709 D00DEH 45483512 Ki = 5 nM T78709 D00FMX 46230706 Ki = 60 nM T78709 D00GSD 25107716 Ki = 188 nM T78709 D00HCC 12996705 Ki = 128 nM T78709 D00KRQ 23113096 Ki = 63 nM T78709 D00OBS 44559159 Ki > 10000 nM T78709 D00VHW 11152527 Ki = 226 nM T78709 D00YEB 25141414 Ki = 11.9 nM T78709 D01CGM 3033677 Ki = 1570 nM T78709 D01HRV 9847194 IC50 = 66 nM T78709 D01JXM 46222048 Ki > 1000 nM T78709 D01KAX 135453290 Ki = 141 nM T78709 D01KVG 9843179 Ki = 169 nM T78709 D01MBF 45483536 Ki = 156 nM T78709 D01TSX 9840090 Ki = 0.65 nM T78709 D01WWC 16573 Ki = 85 nM T78709 D01YNZ 45483529 Ki = 121 nM T78709 D02NNS 9845181 Ki = 300 nM T78709 D02RAY 16754 Ki = 171 nM T78709 D02UWB 1809 IC50 = 0.2951 nM T78709 D02YSX 197033 Ki > 100 nM T78709 D03DET 10287730 Ki = 316.23 nM T78709 D03DLZ 6089 Ki = 410 nM T78709 D03DQQ 45375938 Ki = 21 nM T78709 D03JOX 11311147 IC50 > 10000 nM T78709 D03LDH 10758200 Ki = 20.7 nM T78709 D03PYX 1219 Ki = 47 nM T78709 D03TDN 1342 Ki = 9.2 nM T78709 D03TSY 24825775 Ki = 700 nM T78709 D03XAE 10775128 Ki = 15 nM T78709 D03ZHB 44455973 Ki = 1081 nM T78709 D04AQE 1833 Ki = 3.2 nM T78709 D04DLR 128018 Ki = 842 nM T78709 D04JZJ 2838196 Ki = 120 nM T78709 D04LWD 11336800 Ki > 1000 nM T78709 D04NDO 45483400 Ki = 47 nM T78709 D04NKQ 22599992 Ki = 117 nM T78709 D04TPO 16006492 Ki = 192 nM T78709 D04TQF 11973927 Ki = 5000 nM T78709 D04TWX 9794475 IC50 > 20000 nM T78709 D04ZMS 11773145 Ki = 260 nM T78709 D04ZPF 45483409 Ki = 57 nM T78709 D05CGI 11245709 Ki = 297 nM T78709 D05EQG 5265 Ki = 17.2 nM T78709 D05GDP 599482 Ki > 10000 nM T78709 D05LJC 45483405 Ki = 606 nM T78709 D05XGR 6918647 Ki = 251.19 nM T78709 D05ZUX 44207909 Ki >= 1000 nM T78709 D06BWZ 68678 Ki = 430 nM T78709 D06DSX 12304178 Ki = 6000 nM T78709 D06FWM 44433247 Ki = 78.4 nM T78709 D06QGD 11357862 IC50 > 10000 nM T78709 D06QKW 2765 Ki = 34.67 nM T78709 D06UDU 45483520 Ki > 4570 nM T78709 D06VDN 443391 IC50 > 1000 nM T78709 D07DWS 45483446 Ki = 31 nM T78709 D07GQP 11477180 Ki = 85.4 nM T78709 D07LRJ 5312149 Ki = 340 nM T78709 D07ROK 44433248 Ki = 94.3 nM T78709 D07ZOP 11470616 IC50 > 10000 nM T78709 D08BCF 5011 Ki = 230 nM T78709 D08CKM 9863250 Ki = 1000 nM T78709 D08DOG 25130235 Ki = 42 nM T78709 D08EFH 36906 Ki = 4.6 nM T78709 D08JLB 45483406 Ki = 364 nM T78709 D08OFG 11177588 Ki > 10000 nM T78709 D08UQU 24766199 Ki = 258 nM T78709 D08VGJ 9904281 Ki = 1080 nM T78709 D08VUQ 10422832 Ki = 5.16 nM T78709 D09BNS 439280 Ki = 0.91 nM T78709 D09CKI 3037997 EC50 > 100000 nM T78709 D09HJL 10331436 IC50 > 10000 nM T78709 D09IIH 45483459 Ki = 20 nM T78709 D09MGF 11973811 Ki = 5000 nM T78709 D09OYA 2107 Ki = 12 nM T78709 D09PIN 3378093 Ki > 1000 nM T78709 D09RPR 16737207 Ki > 10000 nM T78709 D09WIL 10028436 Ki = 250 nM T78709 D0A7AK 11973810 Ki = 5000 nM T78709 D0C3EX 1797 Ki = 315 nM T78709 D0C5GF 6918515 Ki = 1470 nM T78709 D0C5XQ 1832 IC50 = 15 nM T78709 D0CA9H 25107518 Ki = 161 nM T78709 D0CG2Y 44133490 Ki = 101 nM T78709 D0CK9K 6918513 Ki = 170 nM T78709 D0DP8I 132266 Ki < 1000 nM T78709 D0E1PL 9865384 EC50 = 23.44 nM T78709 D0E3AL 56597938 Ki = 0.6 nM T78709 D0E6PQ 45483451 Ki = 128 nM T78709 D0F0IA 11301655 Ki = 1365 nM T78709 D0F6CD 5202 EC50 = 0.5 nM T78709 D0F6GB 44133853 Ki = 16 nM T78709 D0FF6S 16038374 IC50 = 10000 nM T78709 D0FU5E 10220053 Ki > 770 nM T78709 D0G2CP 10404144 Ki = 1400 nM T78709 D0G8CV 9954003 Ki = 5.012 nM T78709 D0H2TS 45483528 Ki > 1000 nM T78709 D0H3KU 172267 Ki = 344 nM T78709 D0H3WJ 44435193 Ki = 1100 nM T78709 D0H7PC 6918553 Ki > 6309.57 nM T78709 D0H9QG 5312148 Ki > 3000 nM T78709 D0I9KV 11220599 IC50 > 10000 nM T78709 D0IC4J 45375937 Ki = 11 nM T78709 D0J2UA 135433933 Ki > 10000 nM T78709 D0K3UL 9796720 Ki = 200 nM T78709 D0K6XD 44433256 Ki = 1772 nM T78709 D0K6ZT 44133851 Ki = 13 nM T78709 D0KT2M 44133674 Ki = 92 nM T78709 D0L3MJ 133538 Ki > 1000 nM T78709 D0L3XU 122187 Ki = 87 nM T78709 D0L7OM 6917970 Ki > 5000 nM T78709 D0LV7U 10667433 Ki > 1000 nM T78709 D0M2ZE 6604756 Ki = 168 nM T78709 D0M3PV 133633 Ki = 6300 nM T78709 D0M3TK 45483431 Ki = 8 nM T78709 D0N2RJ 45483432 Ki = 9 nM T78709 D0O3GF 1220 Ki = 0.17 nM T78709 D0PN8D 44351692 Ki = 2.8 nM T78709 D0Q6SH 45483408 Ki > 4570 nM T78709 D0QM3E 9870500 Ki = 3.981 nM T78709 D0R3GW 10296414 Ki = 0.3162 nM T78709 D0R3TA 45483407 Ki = 77 nM T78709 D0R5WX 11220953 Ki = 11.5 nM T78709 D0RQ8R 11973809 Ki = 5000 nM T78709 D0S0XK 9863146 IC50 = 398.11 nM T78709 D0S4JT 45483466 Ki = 189 nM T78709 D0T2RY 9948320 Ki = 280 nM T78709 D0U0VH 9904242 Ki = 0.1 nM T78709 D0V0PR 45483527 Ki > 1000 nM T78709 D0V7OO 10386282 IC50 = 5.4 nM T78709 D0W2HW 6090 Ki = 47 nM T78709 D0W8YO 46230654 Ki = 4.6 nM T78709 D0X1QW 122334 Ki = 410 nM T78709 D0X4PH 11224758 Ki = 52.7 nM T78709 D0X6MT 4106 Ki = 2.2 nM T78709 D0X8LG 11243002 IC50 > 10000 nM T78709 D0X9YS 23642275 Ki = 89.7 nM T78709 D0XX2U 16006606 Ki = 32 nM T78709 D0Y0SA 135399666 EC50 = 2890 nM T78709 D0Y1YR 442793 Ki > 100000 nM T78709 D0Y5CG 45483467 Ki = 116 nM T78709 D0Y9TL 13702393 Ki = 1701 nM T78709 D0Z1OF 23643664 Ki = 60.9 nM T78709 D0Z5GR 46230818 Ki = 4.5 nM T78709 D0ZU5W 22615724 Ki = 28 nM T12499 D00STL 644241 IC50 = 108.2 nM T12499 D03MNN 11341869 IC50 = 20 nM T12499 D03ZBT 11626560 IC50 < 1 nM T12499 D04AIT 5280445 IC50 = 10 ug.mL-1 T12499 D04LVK 57379345 IC50 = 560 nM T12499 D06XXH 11511120 IC50 = 94000 nM T12499 D09KTS 24821094 IC50 = 2.85 nM T12499 D0AZ3C 5291 IC50 = 320 nM T12499 D0E6XR 3062316 IC50 = 0.4 nM T12499 D0EG1I 9926791 IC50 = 3870 nM T12499 D0K8KX 5280343 IC50 = 40 ug.mL-1 T12499 D0OB0F 5328940 IC50 = 1.3 nM T12499 D0R0MW 5329102 IC50 = 8.9 nM T12499 D0W5HK 216239 IC50 = 60 nM T12499 D02RJY 11442891 IC50 = 155 nM T12499 D02UFQ 11620908 IC50 = 2400 nM T12499 D02XNW 5494449 Ki = 80 nM T12499 D03AND 11656518 IC50 > 6000 nM T12499 D03HUX 49792852 IC50 > 10000 nM T12499 D03LWG 53235510 IC50 = 2500 nM T12499 D07EHV 44814409 IC50 > 10000 nM T12499 D07HPJ 11476171 IC50 = 5600 nM T12499 D08AOZ 86582336 IC50 = 3800 nM T12499 D08HOM 46207586 IC50 = 3 nM T12499 D08UUL 46700756 IC50 > 10000 nM T12499 D0A5MC 11712649 IC50 = 3200 nM T12499 D0CY1B 6420138 Ki = 2800 nM T12499 D0E3TC 44259 IC50 = 1.01 nM T12499 D0G5XV 135565884 IC50 = 187 nM T12499 D0H2HZ 60194098 IC50 = 3981.07 nM T12499 D0HS5V 11234052 IC50 > 2500 nM T12499 D0LF1U 5287969 IC50 = 11000 nM T12499 D0M0XB 10302451 IC50 < 4 nM T12499 D0M9QZ 11485656 IC50 = 500000 nM T12499 D0N8RV 9868037 IC50 = 22 nM T12499 D0O0LS 25141092 IC50 > 1000 nM T12499 D0O6WV 24794418 IC50 = 120 nM T12499 D0P1CV 46191454 IC50 > 10000 nM T12499 D0Q7RE 16007391 Ki = 170 nM T12499 D0Q9UX 16718576 IC50 = 209 nM T12499 D0S4JK 24771867 IC50 = 320 nM T12499 D0S5RC 3025986 IC50 > 40000 nM T12499 D0U3EP 445154 IC50 = 112000 nM T12499 D0Z4RC 24756910 IC50 = 5910 nM T12499 D0LF0O 135441202 IC50 = 140 nM T12499 D00OWF 5280953 IC50 > 250000 nM T12499 D00PWQ 3820 IC50 = 470 nM T12499 D08DBE 10344820 Ki = 116 nM T12499 D09HEV 6539952 IC50 = 15 nM T12499 D0A9KI 9863367 IC50 > 10 nM T12499 D0F8DL 176155 IC50 = 3450 nM T12499 D0T3ME 156422 IC50 = 35000 nM T12499 D0U7OU 3220 IC50 = 5 ug.mL-1 T12499 CB1VW3 1400 IC50 = 5 nM T12499 CY58BM 1880 IC50 = 80 ug.mL-1 T12499 CZM9B7 2404 IC50 > 100000 nM T12499 CZ0T5U 2948 IC50 = 17 nM T12499 C1BE5N 3799 IC50 < 10000 nM T12499 C0W4UD 3896 IC50 = 10000 nM T12499 CBPM40 4878 Ki = 0.7943 nM T12499 CAME09 8512 IC50 > 800 ug.mL-1 T12499 C73JPZ 10639 IC50 > 800 ug.mL-1 T12499 C0RTM7 11796 IC50 = 20 ug.mL-1 T12499 C7H0NX 78630 IC50 = 2909000 nM T12499 C89ZVN 125519 IC50 = 1000 nM T12499 CWVL71 152444 IC50 = 1560000 nM T12499 CA5CO8 157820 IC50 = 18000 nM T12499 CPW0V2 165521 IC50 = 4 ug.mL-1 T12499 CV7W4J 176406 IC50 < 10000 nM T12499 C08RPS 177048 IC50 = 200000 nM T12499 CYE78A 182362 IC50 = 3 ug.mL-1 T12499 C75SNM 210813 IC50 = 5000 nM T12499 C7ER4A 229016 IC50 = 100 ug.mL-1 T12499 C2F4EP 332208 IC50 > 800 ug.mL-1 T12499 C1RBE6 368070 IC50 > 2927000 nM T12499 CHQ8V9 372421 IC50 > 2000000 nM T12499 CZH37Q 375454 IC50 = 26000 nM T12499 C0DI9H 375472 IC50 = 85000 nM T12499 C0M4OG 375473 IC50 = 1000 nM T12499 CQD2L7 380855 IC50 = 150000 nM T12499 CVJQ29 380856 IC50 = 42000 nM T12499 CCZW91 380857 IC50 = 65000 nM T12499 CA4FN2 380860 IC50 = 1000 nM T12499 CQO21P 383146 IC50 = 25000 nM T12499 C4MNG8 445840 IC50 = 2300 nM T12499 CIE63B 446044 IC50 > 200000 nM T12499 C1YNB7 447721 IC50 > 20000 nM T12499 C1ZG2U 449087 IC50 > 10000 nM T12499 C9L4RP 468132 IC50 = 5000 nM T12499 CMF14P 598873 IC50 = 1500000 nM T12499 CYC75Z 622510 IC50 > 2000000 nM T12499 C4G0QI 659323 IC50 = 260000 nM T12499 CIGS25 676030 IC50 = 80 ug.mL-1 T12499 CM2NR3 676310 IC50 = 50 ug.mL-1 T12499 C2XAH3 678080 IC50 = 999000 nM T12499 CQHO31 688662 IC50 = 40 ug.mL-1 T12499 CH5JI0 688813 IC50 > 800 ug.mL-1 T12499 C2RAL3 703616 IC50 = 622000 nM T12499 C2H5IE 735037 IC50 = 20 ug.mL-1 T12499 CA30WB 735606 IC50 > 3787000 nM T12499 C0G8LW 776222 IC50 = 307000 nM T12499 CPZV35 788949 IC50 = 205000 nM T12499 CWB7K2 814765 IC50 = 3097000 nM T12499 CYQ90E 1474874 IC50 > 100000 nM T12499 C3SGW1 1490236 IC50 = 10000 nM T12499 C7B3EF 1695774 IC50 > 800 ug.mL-1 T12499 CM8EJ4 2306385 IC50 > 2775000 nM T12499 CY32QZ 2488782 IC50 = 740 nM T12499 C9IWU0 2789324 IC50 = 50000 nM T12499 CI0P2J 2814562 IC50 = 38000 nM T12499 CHGP54 3035187 IC50 = 5000 nM T12499 CIU9K1 3049109 IC50 = 2117000 nM T12499 C2LIF3 3295701 IC50 = 619000 nM T12499 CYN03Q 3684055 IC50 > 2000000 nM T12499 CQ9YE2 3758644 IC50 = 2323000 nM T12499 CM49EB 5007981 IC50 > 2000000 nM T12499 CKWU34 5058788 IC50 > 2000000 nM T12499 CU6M8E 5280457 IC50 = 193000 nM T12499 C8ELV4 5281617 IC50 = 80 ug.mL-1 T12499 CN10FM 5281793 IC50 = 23500 nM T12499 CX4F7K 5281953 IC50 = 20 ug.mL-1 T12499 CTID76 5282335 IC50 > 40000 nM T12499 C0JX4D 5317038 IC50 > 800 ug.mL-1 T12499 CNB7Q3 5328796 IC50 = 1000000 nM T12499 C4RUV5 5329453 IC50 = 300 nM T12499 COX6Q3 5339689 IC50 = 2106000 nM T12499 CF24MP 5353259 IC50 = 60 nM T12499 CBC0E8 5374802 IC50 = 1229000 nM T12499 CJ3WR2 5381920 IC50 > 800 ug.mL-1 T12499 CVU01J 5388676 IC50 = 1500000 nM T12499 C0SO6F 5388678 IC50 = 100000 nM T12499 C9RAX0 5388679 IC50 = 500000 nM T12499 CMS0G9 5388680 IC50 = 2000000 nM T12499 CUX3A5 5388744 IC50 = 2285000 nM T12499 CA2GL7 5388745 IC50 = 516000 nM T12499 CB86MY 5391140 IC50 = 10 ug.mL-1 T12499 CR8AM5 5467796 IC50 > 2530000 nM T12499 CKX8Q5 5467800 IC50 > 2530000 nM T12499 CF0MC5 5467801 IC50 = 168000 nM T12499 CM34ED 5468835 IC50 = 74000 nM T12499 CDVG95 5481246 IC50 = 30 ug.mL-1 T12499 CDK3J0 5703619 IC50 = 3.3 nM T12499 C7H9VZ 5905112 IC50 = 2175000 nM T12499 CEZP52 6263849 IC50 > 50000 nM T12499 C03WIJ 6303920 IC50 = 615000 nM T12499 C4RVA6 6440397 IC50 = 118000 nM T12499 CA31PJ 6539953 IC50 = 40 nM T12499 C64ZJA 6539954 IC50 = 40 nM T12499 CBD1H7 6539955 IC50 = 110 nM T12499 CWHY29 6539956 IC50 = 93 nM T12499 CW76RA 6539957 IC50 = 4 nM T12499 C7K1QS 6539958 IC50 = 209 nM T12499 CJ7IL2 6539959 IC50 = 3120 nM T12499 CAE95J 6539960 IC50 = 167 nM T12499 CH86XJ 6539961 IC50 = 55 nM T12499 C41FUH 6539962 IC50 = 28 nM T12499 C7M2JP 6539963 IC50 = 92 nM T12499 CS5V1C 6539964 IC50 = 31 nM T12499 C10FYS 6539966 IC50 = 10 nM T12499 CIS1T3 6539967 IC50 = 50 nM T12499 CUPQ08 6539985 IC50 = 20000 nM T12499 CMEZ23 6540005 IC50 = 4500 nM T12499 CP0XI6 6603792 IC50 < 1 nM T12499 C3R5VW 9547983 IC50 = 3 nM T12499 CRK62A 9581370 IC50 > 3316000 nM T12499 CZDR80 9584504 IC50 > 3316000 nM T12499 C6MBQ4 9794567 IC50 = 19000 nM T12499 C2OL7K 9796455 IC50 = 1400 nM T12499 C01TAH 9802700 IC50 > 30000 nM T12499 CI80BK 9803350 IC50 = 200 nM T12499 CKT18P 9803404 IC50 > 20000 nM T12499 CSM34J 9804627 IC50 = 82 nM T12499 CR3Q2J 9818899 IC50 = 19.5 nM T12499 C2QX0O 9820995 IC50 = 1500 nM T12499 C6QBF8 9823235 IC50 = 4 nM T12499 CW8V0K 9864418 IC50 > 16000 nM T12499 CIEX48 9865315 IC50 = 3 nM T12499 C23BQG 9867983 IC50 = 650 nM T12499 C7RLN5 9867984 IC50 > 20000 nM T12499 CM5Z8X 9869943 IC50 = 0.5 nM T12499 C26LCM 9883941 IC50 = 58 nM T12499 C51QNA 9883977 IC50 = 86 nM T12499 CR2B8U 9888491 IC50 = 3300 nM T12499 CXA5C8 9893493 IC50 = 5100 nM T12499 C2Y3WG 9907612 IC50 = 300000 nM T12499 CAPU15 9908247 IC50 = 23 nM T12499 C13JNB 9917853 EC50 = 10000 nM T12499 CXD2Y6 9926586 IC50 = 3800 nM T12499 CL4TW5 9926914 IC50 = 153 nM T12499 CYW49X 9927718 IC50 = 35 nM T12499 CG6A1H 9927800 IC50 = 1100 nM T12499 C4OP1L 9932917 IC50 = 1400 nM T12499 CPQ13K 9933545 IC50 > 100000000 nM T12499 CRK63X 9933645 IC50 = 0.5 nM T12499 C6BZ2C 9934106 IC50 > 10000 nM T12499 CJO47T 9948405 IC50 > 10000 nM T12499 CJP49W 9949373 IC50 = 128 nM T12499 C54ZXH 9950678 IC50 = 2 nM T12499 CD63SU 9953450 IC50 = 290 nM T12499 CS35OC 9953741 IC50 = 27 nM T12499 CFC2E6 9954769 IC50 > 30000 nM T12499 CAH50Y 9970231 IC50 = 141000 nM T12499 CA8BC2 9976589 IC50 > 2000000 nM T12499 C37GXK 9983303 IC50 = 8000 nM T12499 C48VFS 9999126 IC50 = 2 nM T12499 CV8I5X 9999342 IC50 > 10000 nM T12499 CUY0F8 10005715 IC50 > 10000 nM T12499 CRY61O 10019770 IC50 = 102 nM T12499 C91VIF 10020232 IC50 > 2000000 nM T12499 C0IA4P 10037831 IC50 = 103000 nM T12499 CXL0R8 10038606 IC50 = 106000 nM T12499 C6AYQ3 10038709 IC50 = 7400 nM T12499 CN8T1M 10041189 IC50 > 2000000 nM T12499 C7YD1X 10048045 IC50 > 25000 nM T12499 CT4M1D 10056916 IC50 = 390 nM T12499 CG4IY8 10059651 IC50 = 17000 nM T12499 CUJR40 10062694 EC50 = 5 nM T12499 CVK3F1 10066999 IC50 = 20000 nM T12499 C7ZO6S 10073515 IC50 = 7 nM T12499 C1JUF8 10073832 IC50 = 18000 nM T12499 CF1D6Y 10075240 IC50 > 12500 nM T12499 CL9D6V 10084407 IC50 = 8500 nM T12499 C8A1TH 10085171 IC50 = 382000 nM T12499 C2C1BP 10089048 IC50 > 16000 nM T12499 C9S0TC 10104347 IC50 = 100000 nM T12499 C30CJT 10126524 IC50 = 149000 nM T12499 CL25BM 10138376 IC50 = 240 nM T12499 CREM37 10151881 IC50 = 710 nM T12499 C69DHW 10158652 IC50 < 16000 nM T12499 C5QHB6 10161543 IC50 = 170 nM T12499 CG2MT8 10176710 IC50 = 203000 nM T12499 CQU0G2 10198725 IC50 = 16000 nM T12499 CQU9K5 10200651 Ki > 5400 nM T12499 CEW30I 10217590 IC50 > 5000 nM T12499 C3UDT7 10217778 IC50 > 2030000 nM T12499 CVY59N 10244533 IC50 > 200000 nM T12499 C5TQ7X 10247543 IC50 > 10000 nM T12499 CI5N9U 10248746 IC50 = 1565000 nM T12499 C97GRN 10248747 IC50 = 26 nM T12499 C6G8NR 10264200 IC50 = 123000 nM T12499 C3HF6S 10264201 IC50 = 200000 nM T12499 CF81EM 10265006 IC50 = 502000 nM T12499 C6DC8Q 10275163 IC50 = 1600 nM T12499 C7SFI1 10296883 IC50 > 10000 nM T12499 C8RD3V 10301884 IC50 = 7 nM T12499 CDP39Q 10316258 IC50 > 2000000 nM T12499 CNS2K1 10318364 IC50 > 2030000 nM T12499 C5CBF9 10320381 IC50 = 100 nM T12499 C3JXP2 10323644 IC50 > 2030000 nM T12499 COC7P1 10333957 IC50 = 56000 nM T12499 CT7PD3 10336593 IC50 > 2000000 nM T12499 C40CWN 10343123 IC50 = 3 nM T12499 CA9L0O 10351200 IC50 = 100 nM T12499 CYCM39 10355659 IC50 = 326000 nM T12499 C37AMD 10356450 IC50 = 754000 nM T12499 C4DOQ9 10356451 IC50 = 46000 nM T12499 C50RSP 10365064 IC50 = 1.7 nM T12499 C52VFK 10366780 IC50 = 3 nM T12499 CVTI82 10377245 IC50 = 487000 nM T12499 C6NLD0 10381816 IC50 = 1876000 nM T12499 CUDE45 10397980 IC50 = 100000 nM T12499 CPS79C 10402283 IC50 = 0.62 ug.mL-1 T12499 C7WEF1 10404203 IC50 > 2000000 nM T12499 CQBD84 10410849 IC50 = 144 nM T12499 CLAX64 10413508 IC50 = 600 nM T12499 CY8H6P 10413576 IC50 > 2030000 nM T12499 CP6N2J 10423146 IC50 = 328000 nM T12499 C97TUR 10426617 IC50 > 2000000 nM T12499 C7HBP6 10429593 IC50 > 10000 nM T12499 CZ68BO 10436007 IC50 > 2030000 nM T12499 CEU25H 10445729 IC50 = 223000 nM T12499 C7ENZ5 10450419 IC50 = 2.4 nM T12499 CLP71R 10466312 IC50 = 58000 nM T12499 CW23SQ 10468973 IC50 = 1621000 nM T12499 C2WQ8M 10473563 IC50 > 10000 nM T12499 C1PB3U 10475630 IC50 > 2030000 nM T12499 C7PLI5 10478569 IC50 = 500 nM T12499 CRX6F0 10479082 IC50 = 10000 nM T12499 CJ5M1D 10482445 IC50 = 100 nM T12499 CXV6B7 10598533 IC50 = 79.7 ug.mL-1 T12499 CX64KP 10862285 IC50 = 170 nM T12499 CD62RJ 10864012 IC50 = 110 nM T12499 CFW87I 10867503 IC50 > 2000000 nM T12499 C7UP2S 10871490 IC50 = 150 nM T12499 CIQ49T 10885591 IC50 = 120 nM T12499 CEJ1S7 10893387 IC50 = 380 nM T12499 CYU8L6 10893773 IC50 > 40000 nM T12499 CBTD58 10894116 IC50 > 40000 nM T12499 C9AYL4 10909252 IC50 > 50000 nM T12499 CSU61K 10916861 IC50 = 730 nM T12499 CUZ74A 10928594 IC50 > 40000 nM T12499 CL9RB3 10939823 IC50 = 740 nM T12499 C8T7AZ 10948261 IC50 = 11000 nM T12499 CLU1O8 10950004 IC50 = 2 nM T12499 CZOF70 10951171 IC50 = 4 nM T12499 C7YX3I 10961937 IC50 = 30 nM T12499 C3C5EL 10962019 IC50 = 2000 nM T12499 CF9IZ1 10970293 IC50 > 40000 nM T12499 CT2N0F 10975200 IC50 = 33800 nM T12499 C0B6ZI 10979411 IC50 = 26000 nM T12499 CM8T6S 10981996 IC50 > 40000 nM T12499 CF7YV3 10982890 IC50 = 5100 nM T12499 CRZ3N4 10983330 IC50 = 2 nM T12499 C46KPJ 11003870 IC50 = 45 nM T12499 CMTX54 11014882 IC50 = 780 nM T12499 CIH8S7 11047384 IC50 = 460 nM T12499 CJ3G8F 11047824 IC50 = 18 nM T12499 CJV52R 11048780 IC50 = 460 nM T12499 C5MBH4 11051416 IC50 > 50000 nM T12499 CP0DG3 11058515 IC50 = 770 nM T12499 CP15QT 11060735 IC50 = 600 nM T12499 C91ZML 11070550 IC50 = 360 nM T12499 CK09XA 11073138 IC50 = 5020 nM T12499 C18KEF 11078754 IC50 > 40000 nM T12499 CPME05 11079939 IC50 = 9600 nM T12499 CO8H4W 11089354 IC50 = 460 nM T12499 C8GE1S 11090362 IC50 = 9600 nM T12499 CRY3O4 11091267 IC50 = 570 nM T12499 C96EUC 11111399 IC50 = 770 nM T12499 CIK0Z6 11113249 IC50 = 86 nM T12499 CE9W7F 11114178 IC50 = 10 nM T12499 C1R2VS 11123387 IC50 = 26 nM T12499 CN1CJ5 11124103 IC50 = 440 nM T12499 C97ISW 11134621 IC50 = 2 nM T12499 C03JWT 11135291 IC50 = 180 nM T12499 CFBH56 11144210 IC50 = 5900 nM T12499 C7I4RG 11147222 IC50 = 3800 nM T12499 CN2JQ0 11169051 IC50 = 23 nM T12499 CS9CK8 11186472 IC50 > 50000 nM T12499 CH3P1J 11186612 IC50 = 4800 nM T12499 CD9E2W 11188787 IC50 = 8 nM T12499 C0Y8TX 11192751 IC50 = 8 nM T12499 CEUR60 11192985 IC50 = 6 nM T12499 CBF04J 11197310 IC50 > 2000000 nM T12499 CO6K3J 11200510 IC50 < 0.2 nM T12499 CB06ZF 11204217 IC50 = 19 nM T12499 CT3K9Z 11213588 IC50 = 1 nM T12499 CEJ6F2 11214762 IC50 = 20 nM T12499 C4HUM2 11232168 IC50 = 10000 nM T12499 C2W5RC 11235063 IC50 > 50000 nM T12499 CVOW82 11238420 IC50 = 210 nM T12499 C02GWO 11245369 IC50 > 30000 nM T12499 CWD28N 11256035 IC50 > 50000 nM T12499 C8JK6G 11257376 IC50 = 98000 nM T12499 CLCW19 11260009 IC50 = 0.7 nM T12499 CC2L8U 11268003 IC50 > 50000 nM T12499 CNBX16 11270660 IC50 = 8 nM T12499 CEP0G1 11273105 IC50 = 10 nM T12499 C2HA7W 11283174 IC50 = 0.5 nM T12499 CBOP58 11293798 Ki > 10000 nM T12499 C9S8PK 11295293 IC50 = 96 nM T12499 CXS5E4 11316381 IC50 = 87 nM T12499 CGP80V 11328586 IC50 = 188 nM T12499 CDI42Q 11328827 IC50 < 0.5 nM T12499 CU5P8C 11331007 IC50 = 12 nM T12499 CC38HS 11336689 IC50 = 8.7 nM T12499 CW0JF9 11337764 IC50 = 121000 nM T12499 CEC31B 11351900 IC50 = 63 nM T12499 C0J2TB 11359024 IC50 = 10000 nM T12499 CFQ7J6 11361039 IC50 = 28000 nM T12499 C26BZX 11362471 Ki > 10000 nM T12499 CB45PJ 11362483 IC50 = 1200 nM T12499 C9B4XP 11363872 IC50 = 4 nM T12499 CGN8P2 11365768 IC50 = 6 nM T12499 C43NPS 11373886 IC50 > 10000 nM T12499 CP4ZO0 11375301 IC50 = 20 nM T12499 CT6Y9W 11376799 IC50 = 23 nM T12499 CEAR81 11381572 IC50 > 50000 nM T12499 CM30TC 11387552 IC50 = 240 nM T12499 CG9Y8F 11395429 IC50 = 5800 nM T12499 CWXB93 11397177 Ki > 10000 nM T12499 CV2IN9 11404920 IC50 = 10000 nM T12499 CMA4U9 11407465 IC50 = 0.2 nM T12499 CYW65I 11417763 IC50 = 380 nM T12499 C73PUW 11420344 IC50 = 18 nM T12499 C5O1RM 11421633 IC50 = 5 nM T12499 C71PYD 11427975 IC50 = 22000 nM T12499 C7AI2V 11432911 IC50 = 7800 nM T12499 C3AS8V 11439407 IC50 > 50000 nM T12499 CYD2A6 11440253 IC50 = 370 nM T12499 CFJ6B2 11441375 IC50 = 330 nM T12499 CO4F0R 11443738 IC50 = 350 nM T12499 CKM8E6 11444953 IC50 = 10 nM T12499 CJC95A 11454205 IC50 > 10000 nM T12499 CU50OG 11455909 IC50 = 12 nM T12499 CFN2C0 11466196 IC50 = 0.7 nM T12499 C4Q7XD 11474276 IC50 = 300 nM T12499 C6M9NC 11477626 IC50 = 4700 nM T12499 CDOF16 11484790 IC50 = 1900 nM T12499 C2Z7WP 11486459 IC50 = 1200 nM T12499 CLM98C 11487256 IC50 = 0.5 nM T12499 CPC9S5 11489476 IC50 = 190 nM T12499 C0H6QS 11495680 IC50 > 10000 nM T12499 C8RQD7 11501591 IC50 = 122 nM T12499 CIW9L5 11502867 IC50 > 10000 nM T12499 CU2OF8 11510392 IC50 = 0.6 nM T12499 C2T8YD 11511361 IC50 = 860 nM T12499 CK2Q0X 11516978 IC50 > 10000 nM T12499 C8AY3B 11518031 IC50 < 25 nM T12499 C87ARG 11519208 IC50 = 170 nM T12499 CHW13Q 11519350 IC50 = 8 nM T12499 CO70EZ 11526166 IC50 = 1480 nM T12499 CPE53F 11526238 IC50 > 10000 nM T12499 C7HMO6 11526786 IC50 > 30000 nM T12499 C5BM4T 11531799 IC50 > 10000 nM T12499 C53OSD 11532048 IC50 > 10000 nM T12499 CC4QM5 11532676 IC50 > 10000 nM T12499 C05FSE 11538753 IC50 = 35 nM T12499 CTG83F 11539329 Ki > 2700 nM T12499 CN1K3R 11545702 IC50 = 1 nM T12499 C01FVM 11546457 IC50 > 10000 nM T12499 C32PUD 11553058 IC50 = 210 nM T12499 CW43OA 11554885 IC50 = 14 nM T12499 CACS26 11561968 Ki > 2000 nM T12499 CNBM81 11562171 IC50 > 10000 nM T12499 CJ59WD 11562553 IC50 = 14 nM T12499 C9XI8Z 11574885 IC50 = 30 nM T12499 CO9KP5 11583459 IC50 > 10000 nM T12499 CA2KX0 11590078 IC50 = 11700 nM T12499 CMIL86 11590363 Ki > 2700 nM T12499 C3CS5K 11593704 IC50 > 3787000 nM T12499 C0NV9Y 11596881 IC50 > 10000 nM T12499 C45BMY 11603130 IC50 = 2100 nM T12499 C69FYK 11604142 Ki = 400 nM T12499 COW68T 11605551 IC50 > 100000 nM T12499 CU6T2L 11613133 IC50 = 30 nM T12499 C1BLZ5 11620055 IC50 > 10000 nM T12499 CUO43M 11620207 IC50 > 25000 nM T12499 CUQ4I5 11620266 IC50 = 27 nM T12499 C5B3XJ 11620410 IC50 = 1140 nM T12499 CG1JN5 11620467 IC50 = 54 nM T12499 C70LDZ 11625929 IC50 < 1 nM T12499 C9ZD2E 11626406 IC50 = 36 nM T12499 CX72ET 11626681 IC50 = 83 nM T12499 CPB48V 11626947 IC50 = 42 nM T12499 CWM80X 11627419 IC50 = 210 nM T12499 CK34LS 11632737 IC50 > 50000 nM T12499 CYL45U 11634544 IC50 = 200 nM T12499 C7CV8O 11634876 IC50 = 22 nM T12499 C1TZY3 11635079 IC50 = 22 nM T12499 C9T6SC 11640926 Ki > 2700 nM T12499 CVH29N 11642023 IC50 = 1920 nM T12499 CA80WI 11648745 IC50 = 11 nM T12499 C82TKN 11656437 IC50 = 11 nM T12499 C3L2HT 11656560 IC50 = 380 nM T12499 CX7C1T 11656606 IC50 = 29 nM T12499 C1AUX0 11661290 IC50 = 36 nM T12499 C24GRQ 11661959 IC50 > 10000 nM T12499 C60ASI 11663230 Ki = 138 nM T12499 C8RMT2 11663885 IC50 = 19 nM T12499 CCGO58 11669282 IC50 = 154 nM T12499 C1LV6H 11677453 IC50 = 11 nM T12499 CA4Q5F 11678465 IC50 = 22 nM T12499 CS72ED 11682843 IC50 > 10000 nM T12499 C5O6YX 11683692 IC50 = 0.4 nM T12499 CP3U0W 11684933 IC50 = 9 nM T12499 CYO6X9 11684994 Ki = 138 nM T12499 CCEY64 11689855 IC50 = 65 nM T12499 CU0E8O 11690457 Ki > 2000 nM T12499 CLC53E 11691173 IC50 > 10000 nM T12499 CI3EO4 11692100 IC50 = 1600 nM T12499 CB0AP2 11705863 Ki > 2000 nM T12499 C6EUQ9 11711497 IC50 = 10 nM T12499 C9ROB0 11713267 IC50 = 21 nM T12499 C1FTX3 11719305 IC50 > 10000 nM T12499 CZY05V 11719421 IC50 = 13 nM T12499 CQN04F 11723994 IC50 > 2000000 nM T12499 C0NVT9 11724908 IC50 > 2000000 nM T12499 C6N2AQ 11726550 IC50 = 2 nM T12499 CX21FQ 11727911 IC50 = 27 nM T12499 CGA26L 11729126 IC50 = 2500 nM T12499 C84LGZ 11730798 IC50 = 50 nM T12499 CA9HO6 11730954 IC50 = 120 nM T12499 CT7U6H 11731262 IC50 = 25 nM T12499 CPY1Z2 11740563 IC50 = 290 nM T12499 CS5QL4 11749561 IC50 = 700 nM T12499 CN8S1E 11752715 IC50 = 28 nM T12499 CE0KI4 11753519 IC50 = 110 nM T12499 CP7AH3 11755812 IC50 = 50000 nM T12499 CUKE53 11760559 IC50 = 1100 nM T12499 CMJ2Q9 11761204 IC50 > 2500 nM T12499 C28UON 11775143 IC50 = 1.3 nM T12499 C3J7MT 11777791 IC50 = 117000 nM T12499 C96TSA 11784426 IC50 = 2500 nM T12499 CL87KR 11785748 IC50 = 27 nM T12499 CCI6R5 11842847 IC50 = 1 nM T12499 CMO6N4 11842849 IC50 = 13 nM T12499 C9HT7B 11842850 IC50 = 49 nM T12499 CP6KY2 11843009 IC50 = 1 nM T12499 C8FHK9 11843010 IC50 = 1 nM T12499 C7D6MQ 11843012 IC50 = 1 nM T12499 C4T2WC 11843013 IC50 = 1 nM T12499 CS36BH 11843159 IC50 = 0.6 nM T12499 C7DU6T 11843160 IC50 = 2 nM T12499 CH6W3V 11844349 IC50 = 14 nM T12499 CI15NA 11844350 IC50 = 12 nM T12499 CUL2C8 11844485 IC50 = 10 nM T12499 C96ORQ 11844486 IC50 = 1 nM T12499 C4SK3L 11844487 IC50 = 1 nM T12499 C6KF8Z 11844488 IC50 = 1 nM T12499 C9ECK3 11844489 IC50 = 1 nM T12499 C83YRX 11844616 IC50 = 1 nM T12499 CV24WL 11844764 IC50 = 1 nM T12499 C9JT4S 11847343 IC50 > 10000 nM T12499 CAZS08 11848309 IC50 = 3614 nM T12499 C43IVN 11848567 IC50 = 1335 nM T12499 C9LAY8 11848825 IC50 > 10000 nM T12499 CHR92S 11858109 IC50 < 4 nM T12499 CHN2X6 11974313 IC50 = 3200 nM T12499 CTN38E 11974315 IC50 = 124 nM T12499 COFI19 11974316 IC50 = 47 nM T12499 CU4IJ6 12035491 IC50 = 700 nM T12499 CA4Z6H 12373545 IC50 > 2916000 nM T12499 C8YVD5 12381316 IC50 > 2000000 nM T12499 C5CPV2 12516472 IC50 > 10 ug.mL-1 T12499 CS0Y1J 12634029 IC50 = 18500 nM T12499 C1PI2A 12911686 IC50 > 50000 nM T12499 CU4C3V 12968172 IC50 = 11 nM T12499 CI8VE5 12968173 IC50 = 2290 nM T12499 CR75GZ 12968174 IC50 = 260 nM T12499 CEVY69 12968175 IC50 = 4 nM T12499 CL1PR6 12968176 IC50 = 17 nM T12499 CY5EA7 12968177 IC50 = 470 nM T12499 CZ98FV 12968178 IC50 = 310 nM T12499 C4SUK6 12968179 IC50 = 144 nM T12499 CGIZ84 12968180 IC50 = 20 nM T12499 C5MX8N 12968181 IC50 = 30 nM T12499 C0P5HT 13182760 IC50 > 800 ug.mL-1 T12499 CS6FK7 14304977 IC50 > 2000000 nM T12499 CQ29NJ 14304982 IC50 > 2000000 nM T12499 CA8E6W 14791361 IC50 = 1160000 nM T12499 CRED76 14791362 IC50 > 2000000 nM T12499 C8ZS9R 14791363 IC50 > 2000000 nM T12499 CH5RB9 14791364 IC50 > 2000000 nM T12499 C5UD8T 14791365 IC50 > 2000000 nM T12499 C25VAZ 14791366 IC50 > 2000000 nM T12499 CES4B9 14791367 IC50 > 2000000 nM T12499 C8R3IO 14791368 IC50 > 2000000 nM T12499 CLOA14 14791369 IC50 > 2000000 nM T12499 C9HLZ3 14791370 IC50 > 2000000 nM T12499 C5N6QA 14791371 IC50 > 2000000 nM T12499 CNB0F4 14791372 IC50 > 2000000 nM T12499 CM87DK 14791373 IC50 > 2000000 nM T12499 CR0J2L 14791374 IC50 > 2000000 nM T12499 CP2H9Y 14791375 IC50 > 2000000 nM T12499 CLXA81 14791376 IC50 > 2000000 nM T12499 CN3F5B 14791377 IC50 > 2000000 nM T12499 CRK9U6 14791378 IC50 > 2000000 nM T12499 CQ5F7V 14791379 IC50 > 2000000 nM T12499 C3RNU7 14791380 IC50 = 1595000 nM T12499 CI98LS 14791381 IC50 = 1032000 nM T12499 C9S7KU 14791382 IC50 = 439000 nM T12499 CWAV76 14791383 IC50 > 2000000 nM T12499 CGX9C2 14791384 IC50 > 2000000 nM T12499 C2YW0J 14791386 IC50 > 2000000 nM T12499 CM3Q7F 14791387 IC50 = 810000 nM T12499 CG10QR 14791388 IC50 > 2000000 nM T12499 C49FJH 14791389 IC50 > 2000000 nM T12499 CX8R7N 14791390 IC50 > 2000000 nM T12499 C0PRG2 14791391 IC50 > 2000000 nM T12499 CZ6WJ9 14791392 IC50 = 100000 nM T12499 CQ9Z0L 15550318 IC50 = 1200 nM T12499 CR7QG2 15550584 IC50 = 144 nM T12499 CF9S5H 15664638 IC50 = 234000 nM T12499 CARI31 15693660 IC50 = 40 ug.mL-1 T12499 CP9CD6 15693661 IC50 = 400 ug.mL-1 T12499 CDSL43 15693662 IC50 = 40 ug.mL-1 T12499 CWO05F 15693663 IC50 > 800 ug.mL-1 T12499 CER56U 15693664 IC50 = 40 ug.mL-1 T12499 C2Z1FO 15693665 IC50 = 40 ug.mL-1 T12499 CLG0Z7 15693666 IC50 = 200 ug.mL-1 T12499 CD7K9N 15693667 IC50 = 70 ug.mL-1 T12499 C0YWD7 15693668 IC50 > 800 ug.mL-1 T12499 C9M0SA 15693669 IC50 > 800 ug.mL-1 T12499 CUI6E5 15858664 IC50 = 200 nM T12499 CG07CP 15931492 IC50 = 1315000 nM T12499 CU9L0Z 15931493 IC50 > 3275000 nM T12499 C0M7TW 15948947 IC50 = 238 nM T12499 C1VNB4 15948949 IC50 = 7 nM T12499 CH8ZG5 15949048 IC50 = 11 nM T12499 CKNZ36 15949147 IC50 = 2090 nM T12499 CX9GH4 15949237 IC50 = 438 nM T12499 CK2Z6Y 15949521 IC50 = 32 nM T12499 CBZF29 15949522 IC50 = 132 nM T12499 C34MCY 15949523 IC50 = 11 nM T12499 CS3P9G 15949524 IC50 = 4 nM T12499 C1KPH2 15949525 IC50 = 1162 nM T12499 C5JG9R 15949617 IC50 = 4 nM T12499 C8FT6U 15949618 IC50 = 316 nM T12499 C30PVQ 15949619 IC50 = 120 nM T12499 C3PNO2 15949620 IC50 = 18 nM T12499 C4I5RS 15949621 IC50 = 2030 nM T12499 C8JLW2 15949711 IC50 > 2500 nM T12499 CVJ9A0 15949712 IC50 = 7 nM T12499 CD9IP6 15949713 IC50 > 2500 nM T12499 C2TAW9 15949714 IC50 > 2500 nM T12499 C5RI8G 15949799 IC50 = 789 nM T12499 CEI2K8 15949887 IC50 = 31 nM T12499 CAIN63 15949888 IC50 > 2500 nM T12499 C2VDI1 15949889 IC50 = 27 nM T12499 COC02T 15949890 IC50 = 881 nM T12499 CFQ6X3 15949974 IC50 = 29 nM T12499 CMKZ23 15949975 IC50 = 111 nM T12499 CWM5L4 15949976 IC50 = 6 nM T12499 CL1HO8 15950062 IC50 = 5 nM T12499 CA8S3R 15950063 IC50 = 119 nM T12499 CZ5F0K 15950065 IC50 = 583 nM T12499 CO7NG2 15950141 IC50 = 12 nM T12499 COIG45 15950224 IC50 = 7 nM T12499 C9V0TO 15950311 IC50 = 20 nM T12499 C9RQN8 15950748 IC50 = 14 nM T12499 CSK90Y 15991573 IC50 = 0.2 nM T12499 CPNW35 15991575 IC50 = 0.5 nM T12499 CFPW41 16007116 Ki > 2700 nM T12499 C09OWB 16015442 IC50 = 531 nM T12499 C0VF7Y 16037922 IC50 = 87 nM T12499 CN36QI 16043219 IC50 = 2 nM T12499 CFKE48 16064750 IC50 = 2000 nM T12499 CIHG50 16066841 IC50 = 3 nM T12499 CBU2X4 16066842 IC50 = 867 nM T12499 C3ZV2X 16086076 IC50 = 6 nM T12499 C0SO7D 16086077 IC50 = 0.6 nM T12499 C0WU9I 16086078 IC50 = 0.07 nM T12499 CVE6C8 16086088 IC50 = 0.27 nM T12499 CH1R8K 16086091 IC50 = 0.3 nM T12499 CT4RS8 16086092 IC50 = 8 nM T12499 CZ2QU1 16086093 IC50 = 297 nM T12499 C13OVU 16086099 IC50 = 0.01 nM T12499 C2YC0S 16086100 IC50 = 0.3 nM T12499 C28UZX 16086101 IC50 = 1 nM T12499 CKM8E4 16086102 IC50 = 0.5 nM T12499 CF0N4J 16086103 IC50 = 3 nM T12499 CKR57M 16086104 IC50 = 0.5 nM T12499 CI5HJ8 16086105 IC50 = 48 nM T12499 C68SBO 16086106 IC50 = 2 nM T12499 CAYV39 16086107 IC50 = 0.4 nM T12499 C06NOI 16086108 IC50 = 2 nM T12499 C6F2YX 16086109 IC50 = 150 nM T12499 CE71TI 16086110 IC50 = 0.5 nM T12499 CQ3UF2 16086111 IC50 = 0.9 nM T12499 CFXT05 16086112 IC50 = 200 nM T12499 C16NRY 16086114 IC50 = 0.2 nM T12499 C87TPW 16086115 IC50 = 3 nM T12499 CW35LJ 16086116 IC50 = 0.4 nM T12499 CA3BD7 16086117 IC50 = 14 nM T12499 C3EKF4 16086118 IC50 = 6 nM T12499 C0QCG4 16086142 IC50 = 1 nM T12499 C73MLJ 16108977 IC50 < 1 nM T12499 CQG45C 16109001 IC50 = 1100 nM T12499 C8P4ZK 16109016 IC50 = 19 nM T12499 CY1E3Q 16109017 IC50 = 42 nM T12499 CV7S6Z 16109018 IC50 = 370 nM T12499 CB98HV 16109019 IC50 = 780 nM T12499 C49VTS 16109020 IC50 = 620 nM T12499 C6FZ7A 16109023 IC50 = 1 nM T12499 CWS8D0 16109024 IC50 = 4 nM T12499 C1WS6E 16109034 IC50 = 410 nM T12499 C8IES6 16109035 IC50 = 150 nM T12499 C1U8XW 16109036 IC50 = 130 nM T12499 CNG5L6 16109037 IC50 = 1100 nM T12499 C34KRB 16109040 IC50 = 1 nM T12499 CZ5Y3V 16116847 IC50 = 5 nM T12499 CLO43V 16116849 IC50 = 48 nM T12499 C0HO6T 16118191 IC50 = 0.6 nM T12499 CT92BZ 16118192 IC50 = 1.4 nM T12499 CIZ6B4 16118193 IC50 = 0.3 nM T12499 C2CN5O 16118323 IC50 = 1.5 nM T12499 C4GTU3 16118324 IC50 = 1.3 nM T12499 CXC78K 16118603 IC50 = 63 nM T12499 CI4E6Y 16118605 IC50 = 72 nM T12499 C8LIW4 16118609 IC50 = 24 nM T12499 CGC34R 16118737 IC50 = 0.6 nM T12499 CAN2K6 16118739 IC50 = 1310 nM T12499 C5VPH9 16129448 IC50 = 2330 nM T12499 CZ08YH 16214904 IC50 = 81 nM T12499 CP3HS4 16220354 IC50 > 50000 nM T12499 CVZK29 16223008 IC50 > 50000 nM T12499 CZO8P2 16440205 IC50 = 50000 nM T12499 C6TQ2O 16664354 Ki = 11.7 nM T12499 C0H8UN 16730109 IC50 > 50000 nM T12499 C6S3YO 16731782 IC50 = 132 nM T12499 CK9CV4 16733534 IC50 = 405 nM T12499 CDZ31W 16747696 IC50 = 30963 nM T12499 C86UEN 16897096 IC50 = 160 nM T12499 CL9BQ6 17748275 IC50 = 146 nM T12499 C28TDB 17756743 IC50 = 81 nM T12499 CWH37T 17758574 IC50 = 4500 nM T12499 CUTS51 17960401 IC50 = 9 nM T12499 C1H7BJ 18007099 IC50 = 3700 nM T12499 C1V7AK 18007100 IC50 > 12500 nM T12499 C1V8BU 18007104 IC50 > 12500 nM T12499 C0Z6RE 18332602 IC50 = 800 nM T12499 C0NKJ2 18332605 IC50 = 1260 nM T12499 CRN5K7 18332650 IC50 = 1 nM T12499 CJ3TD7 18332663 IC50 = 46 nM T12499 CFL69G 18332667 IC50 = 242 nM T12499 CX6BH1 18332672 IC50 = 11 nM T12499 C9RHI4 18342784 IC50 = 1 nM T12499 CJK36Q 18354367 IC50 = 11.8 nM T12499 CP73AB 18354386 IC50 = 26.5 nM T12499 CU83MW 18354409 IC50 > 1000 nM T12499 C5RY6O 18375493 IC50 = 827 nM T12499 CA7T2W 18450829 IC50 = 380 nM T12499 CB2LF3 18450830 IC50 > 50000 nM T12499 CW0U4Z 18450843 IC50 = 140 nM T12499 C6E4YZ 18450934 IC50 = 9650 nM T12499 C0VWB3 18451020 IC50 = 290 nM T12499 C3J5HU 18451023 IC50 = 2950 nM T12499 CJA0D6 18451024 IC50 = 190 nM T12499 C0X9RC 18451029 IC50 = 230 nM T12499 CNBP94 18451030 IC50 = 6700 nM T12499 C6FQB7 18451036 IC50 = 290 nM T12499 CEI23S 18451044 IC50 = 770 nM T12499 CUZ1E0 18451049 IC50 = 1370 nM T12499 CGT10H 18451102 IC50 = 6850 nM T12499 CM9BN5 18451119 IC50 = 1520 nM T12499 CM1X8S 18451204 IC50 = 4810 nM T12499 CB84DI 18451225 IC50 = 20800 nM T12499 C45MTJ 18451346 IC50 = 5200 nM T12499 CYJ3M1 18451394 IC50 = 720 nM T12499 CHDY96 18770788 IC50 = 50000 nM T12499 C1GAJ2 18770840 IC50 = 500 nM T12499 CHI4W7 18770845 IC50 = 5000 nM T12499 C1C0EJ 18792861 IC50 = 360 nM T12499 C6HK0S 18792868 IC50 = 400 nM T12499 C4SPG1 19007057 Ki = 2800 nM T12499 C5WAV7 19597382 IC50 = 20 nM T12499 CU5CK6 19597400 IC50 = 140 nM T12499 CZQ92B 19597433 IC50 < 1 nM T12499 C02JLX 19597448 IC50 < 3 nM T12499 CYIX85 19597450 IC50 = 8 nM T12499 CFH4I2 19597457 IC50 < 3 nM T12499 CIBE65 19597460 IC50 = 130 nM T12499 C0JQ7H 19597465 IC50 < 1 nM T12499 CP01WN 19597468 IC50 < 1 nM T12499 CA09JB 19597476 IC50 = 5 nM T12499 CC78WA 19597518 IC50 = 390 nM T12499 CV0U1N 19597532 IC50 < 3 nM T12499 C1B3DX 19597536 IC50 < 1 nM T12499 C0E2OG 20579089 IC50 = 2200 nM T12499 CIC6E2 20703609 IC50 = 0.4 nM T12499 C5BS4H 20703624 IC50 = 2.6 nM T12499 CKE9O1 20703628 IC50 = 0.25 nM T12499 CX90RK 20703629 IC50 = 75.2 nM T12499 CRCY81 20703632 IC50 = 22.5 nM T12499 C4AZQ7 20703633 IC50 > 1000 nM T12499 C58WTF 20703634 IC50 = 501 nM T12499 CC1MJ6 20711999 IC50 = 40 nM T12499 CV7C2K 20817018 IC50 = 64 nM T12499 CQ5X7V 20817081 IC50 = 20 nM T12499 CEU1O0 20817327 IC50 = 341 nM T12499 CK1TF6 20817330 IC50 = 102 nM T12499 C6AN8E 20817403 IC50 = 23 nM T12499 C56HRP 20817416 IC50 = 106 nM T12499 CXCF38 20817425 IC50 = 30 nM T12499 CC1E7R 21078798 Ki > 5400 nM T12499 CH4B5K 21081523 IC50 > 5000 nM T12499 C25UKC 21081761 IC50 = 290 nM T12499 CU29EB 21137651 IC50 = 700 nM T12499 CBTS02 21137686 IC50 > 30000 nM T12499 CI82BH 21137692 IC50 = 12500 nM T12499 CA73LU 21137693 IC50 = 4400 nM T12499 CGB54O 21774685 IC50 = 92 ug.mL-1 T12499 C9RSY1 21911223 IC50 = 4.9 nM T12499 CAO1M7 21911235 IC50 = 180 nM T12499 C0D6BH 21911241 IC50 = 4470 nM T12499 CNTX42 21911266 IC50 = 1.2 nM T12499 CF9D4B 21911267 IC50 = 3 nM T12499 CQ2U0F 21911271 IC50 = 360 nM T12499 CC3UI5 21911283 IC50 = 1340 nM T12499 CEV1N5 21911286 IC50 = 18 nM T12499 CZ2K3O 21911293 IC50 = 5 nM T12499 CB5DO1 21911296 IC50 = 12080 nM T12499 CK06DT 21911324 IC50 = 3100 nM T12499 C6RM2E 21911333 IC50 = 6.3 nM T12499 C82VPK 21911338 IC50 = 4 nM T12499 C4FWH1 21911345 IC50 = 0.6 nM T12499 CQAW69 21911406 IC50 = 240 nM T12499 CCU5P6 21911412 IC50 = 130 nM T12499 CO36ZH 21911439 IC50 = 6.7 nM T12499 C0QTP8 21911457 IC50 = 50 nM T12499 C7ICY1 21911468 IC50 = 890 nM T12499 C1PTM5 21911491 IC50 = 620 nM T12499 CJV64F 21911517 IC50 = 800 nM T12499 CW81PU 21911520 IC50 = 9.4 nM T12499 CFW5Q4 21911536 IC50 = 17 nM T12499 CPN2M4 21911557 IC50 = 140 nM T12499 CXZ3J0 21911563 IC50 = 480 nM T12499 CK8AY5 21911573 IC50 = 2230 nM T12499 C01PAE 21911582 IC50 = 130 nM T12499 C4X9VW 21911584 IC50 = 390 nM T12499 CD91KJ 21911586 IC50 = 1.2 nM T12499 CL8V5Y 21911599 IC50 = 4 nM T12499 CLP84C 21911609 IC50 = 1400 nM T12499 CQWN07 21911611 IC50 = 710 nM T12499 CU59WY 21911623 IC50 = 0.5 nM T12499 C8EA6U 21911645 IC50 = 0.3 nM T12499 CX8Z1W 21985424 IC50 = 1200 nM T12499 CDS2B9 21985432 IC50 = 30 nM T12499 CP78LH 21985486 IC50 = 1300 nM T12499 C5WHN8 21994549 IC50 > 12500 nM T12499 CCPU92 21994552 IC50 = 2.4 nM T12499 CWZ8Y4 21994558 IC50 = 180 nM T12499 CKM54W 21994560 IC50 > 12500 nM T12499 C7JX0Z 21994562 IC50 = 4390 nM T12499 CEVT05 21994569 IC50 = 3 nM T12499 C6AQD0 21994570 IC50 = 820 nM T12499 CIO8H7 21994571 IC50 = 36 nM T12499 CI9D2L 21994591 IC50 = 2680 nM T12499 C6XQ1W 21994598 IC50 = 6 nM T12499 C1RUF7 21994601 IC50 = 1690 nM T12499 CRCD41 21994605 IC50 = 15 nM T12499 CJX07Q 21994606 IC50 = 890 nM T12499 C8ZN2J 21994630 IC50 > 12500 nM T12499 C21IJA 21994643 IC50 = 9.4 nM T12499 C86ONB 21994661 IC50 = 13 nM T12499 CA8B9K 21994707 IC50 = 16 nM T12499 CF35EU 21994709 IC50 = 9 nM T12499 C98IEP 21994713 IC50 = 3 nM T12499 CDIZ08 21994718 IC50 = 390 nM T12499 CBF70N 21994727 IC50 = 2 nM T12499 CDK0B1 21994742 IC50 = 3170 nM T12499 C43XZF 21994749 IC50 = 240 nM T12499 C71VCF 21994770 IC50 = 3 nM T12499 C1RV3C 21994777 IC50 = 10 nM T12499 CPFU26 21994778 IC50 = 14 nM T12499 CZ4CB9 21994781 IC50 = 100 nM T12499 C5FR4C 21994782 IC50 = 5520 nM T12499 CJV9A0 21994783 IC50 = 30 nM T12499 CQG8B4 21994786 IC50 = 60 nM T12499 CA5L3Q 21994789 IC50 = 1 nM T12499 CV78HM 21994811 IC50 > 12500 nM T12499 CLK0T6 21994850 IC50 = 11 nM T12499 C2RTU9 21994872 IC50 > 12500 nM T12499 CKA1C7 21994883 IC50 = 4 nM T12499 CZO46G 21994907 IC50 = 30 nM T12499 C2U5YF 21994914 IC50 = 4 nM T12499 C9XDA4 21994918 IC50 > 12500 nM T12499 CSEX73 21994919 IC50 = 360 nM T12499 CEPU70 21994926 IC50 = 9 nM T12499 CV06FC 21994930 IC50 = 3 nM T12499 CHN2Y3 21994942 IC50 = 100 nM T12499 C6DK9A 21994949 IC50 = 1330 nM T12499 CVA9P4 21994955 IC50 = 9 nM T12499 C1YF4W 21994961 IC50 = 9 nM T12499 C2BAM8 21994965 IC50 = 11 nM T12499 C8OBH7 21994981 IC50 = 6.2 nM T12499 CT17VP 21994984 IC50 = 240 nM T12499 C3C6FO 21994992 IC50 = 24 nM T12499 CA1CL8 21995003 IC50 = 26 nM T12499 CXJ26U 21995007 IC50 = 40 nM T12499 C12GPM 21995020 IC50 = 3170 nM T12499 CD7G2O 21995023 IC50 = 2.4 nM T12499 CEM56K 21995028 IC50 = 8 nM T12499 CP7R3X 21995029 IC50 = 18 nM T12499 CG35FE 21995041 IC50 = 3 nM T12499 CA16TP 21995049 IC50 = 4 nM T12499 C4NZJ6 21995088 IC50 = 50 nM T12499 CYR02Q 21995091 IC50 = 30 nM T12499 C7UQM9 21995099 IC50 > 12500 nM T12499 CXJI39 22022153 IC50 = 3000 nM T12499 CGX61W 22041319 IC50 = 65 nM T12499 CQ2XW6 22346679 IC50 = 74 nM T12499 CZRT79 22346947 IC50 = 50 nM T12499 C2AYF1 22634103 IC50 = 300 nM T12499 CZR4U0 22634116 IC50 = 90 nM T12499 CXP45U 22634145 IC50 = 80 nM T12499 C3CN7M 22634150 IC50 = 15 nM T12499 CUXV98 22634165 IC50 = 310 nM T12499 CMVL20 22634174 IC50 = 130 nM T12499 CCZ07D 22634175 IC50 = 700 nM T12499 C5E4BO 22634176 IC50 = 123 nM T12499 CT7MB6 22634192 IC50 = 55 nM T12499 C06DIG 22634197 IC50 = 565 nM T12499 CKX62Q 22634226 IC50 = 11 nM T12499 CWEL63 22634235 IC50 = 2010 nM T12499 C3CV5J 22634236 IC50 = 45 nM T12499 C5LXT1 22634281 IC50 = 337 nM T12499 C7H4DQ 22634288 IC50 = 100 nM T12499 CZE2U9 22634355 IC50 = 70 nM T12499 CEN7D5 22634359 IC50 = 7 nM T12499 CKOH73 22634360 IC50 = 1800 nM T12499 C68JBA 22634362 IC50 = 30 nM T12499 C54BIF 22634389 IC50 = 87 nM T12499 CH65IJ 22634393 IC50 = 1730 nM T12499 C6AE5O 22634424 IC50 = 330 nM T12499 C7OA9U 22634439 IC50 = 120 nM T12499 C7WX8F 22634450 IC50 = 39 nM T12499 C5P7OI 22634478 IC50 = 11 nM T12499 CAJ5E3 22634481 IC50 = 4 nM T12499 CD03MH 22634489 IC50 = 380 nM T12499 CI15AY 22634499 IC50 = 90 nM T12499 C1WRE8 22634507 IC50 = 7 nM T12499 CO4FX0 22634509 IC50 = 3120 nM T12499 CDQV06 22634522 IC50 = 19 nM T12499 CXSQ56 22634523 IC50 = 27 nM T12499 C4KY6D 22634526 IC50 > 12500 nM T12499 C5NP3B 22634530 IC50 = 85 nM T12499 C9P3CF 22634544 IC50 > 3125 nM T12499 CTWJ81 22634553 IC50 = 20 nM T12499 CNJ78C 22634560 IC50 = 15070 nM T12499 CSIO14 22634565 IC50 = 666 nM T12499 CLOR96 22736225 IC50 = 46 nM T12499 CT39NL 22736235 IC50 < 1 nM T12499 CAU62I 22736238 IC50 = 890 nM T12499 CV1OI5 22736332 IC50 = 42 nM T12499 C5ONK2 22736361 IC50 = 120 nM T12499 CT57UR 23075146 IC50 = 829000 nM T12499 CGV8M7 23375461 IC50 = 200 nM T12499 CG12OL 23518511 IC50 = 600 nM T12499 CE7K3W 23532567 IC50 > 10000 nM T12499 C5AZ7B 23536770 IC50 = 6 nM T12499 CW6OB1 23627212 IC50 = 260 nM T12499 CR3M1N 23644582 Ki = 20 nM T12499 C70VCY 23646368 IC50 = 20 nM T12499 CG6D4M 23647319 IC50 > 10000 nM T12499 CY8Z7X 23647330 IC50 > 10000 nM T12499 C4XD8H 23647348 IC50 > 10000 nM T12499 CI6C1R 23658582 IC50 = 75 nM T12499 CBXC05 24424330 IC50 = 31 nM T12499 C3RVK4 24750458 IC50 > 800 ug.mL-1 T12499 CA3I4T 24753787 IC50 > 50000 nM T12499 CHU49V 24757938 IC50 = 38 nM T12499 C7YG1N 24759534 IC50 = 19 nM T12499 CAJ4T2 24762205 IC50 = 22 nM T12499 CQNP54 24764449 IC50 = 1000 nM T12499 C2UOE0 24766030 IC50 = 46 nM T12499 C31EHS 24767187 IC50 > 100000 nM T12499 C4Z9CN 24769780 IC50 = 33 nM T12499 CJUK39 24770517 IC50 > 10000 nM T12499 CLBP72 24798571 IC50 = 4440 nM T12499 C9PA0M 24807809 IC50 > 30000 nM T12499 C0JUN4 24812717 IC50 = 19 nM T12499 CP6N9M 24812718 IC50 = 1900 nM T12499 CW0G8H 24812719 IC50 = 1700 nM T12499 CO9Z0H 24822598 IC50 = 1100 nM T12499 C51IZL 24822599 IC50 = 1300 nM T12499 CA90EF 24822600 IC50 = 1800 nM T12499 CCP2M3 24822704 IC50 > 50000 nM T12499 C4A6LB 24823090 IC50 = 2000 nM T12499 C2B4JP 24823091 IC50 = 4300 nM T12499 C14FLQ 24823250 IC50 = 25000 nM T12499 C3KPO7 24823251 IC50 = 1000 nM T12499 C3A2BF 24823416 IC50 = 4600 nM T12499 CYBI02 24823426 IC50 = 15 nM T12499 C45UGH 24823586 IC50 = 0.5 nM T12499 CFA3T8 24823588 IC50 = 14 nM T12499 C51ZTV 24823589 IC50 = 5 nM T12499 CX0QC1 24823590 IC50 = 0.8 nM T12499 CR7CH6 24823736 IC50 = 10 nM T12499 C26KXV 24823738 IC50 = 6 nM T12499 CO3K7R 24823740 IC50 = 1.8 nM T12499 CBLJ48 24823898 IC50 = 6 nM T12499 CG0K1Z 24824046 IC50 = 239 nM T12499 CDT3L2 24824050 IC50 = 27 nM T12499 CLN48F 24824051 IC50 = 90 nM T12499 C0NXE2 24824052 IC50 = 1500 nM T12499 CWTI12 24824188 IC50 = 500 nM T12499 CQ1A8W 24824189 IC50 = 19 nM T12499 C8RE5C 24824190 IC50 > 4000 nM T12499 C3K1FM 24824191 IC50 > 4000 nM T12499 CV0S5L 24824318 IC50 = 2200 nM T12499 CUK14T 24824319 IC50 > 4000 nM T12499 CZ09ID 24824320 IC50 = 2400 nM T12499 CM28KX 24824321 IC50 = 1000 nM T12499 CD57UN 24824322 IC50 = 150 nM T12499 CNI50G 24824323 IC50 = 78 nM T12499 C84VZK 24824448 IC50 = 1000 nM T12499 C6OC4K 24824449 IC50 = 1300 nM T12499 C5BA7V 24824452 IC50 = 21 nM T12499 CR49SP 24824453 IC50 > 4000 nM T12499 CG64EL 24824454 IC50 > 4000 nM T12499 CM28WD 24825721 IC50 > 10000 nM T12499 CX0S9L 24854902 IC50 = 6048 nM T12499 C1SVT2 24854903 IC50 > 5000 nM T12499 C61KPI 24856363 IC50 > 16000 nM T12499 CS82HN 24856408 IC50 = 37 nM T12499 CZ5Y4H 24856498 IC50 = 23 nM T12499 CC10FW 24857629 IC50 = 92 nM T12499 CCS58O 24863072 IC50 = 21 nM T12499 C6C2GX 24863500 IC50 = 23 nM T12499 CYVB83 24863584 IC50 = 210 nM T12499 CQ15ML 24863670 IC50 = 78 nM T12499 C4XZ3N 24863671 IC50 = 110 nM T12499 CSW5V3 24865437 IC50 = 24000 nM T12499 CE3IW4 24879184 IC50 = 340 nM T12499 C7V8BA 24879242 IC50 = 480 nM T12499 CT76XV 24879243 IC50 = 740 nM T12499 CGD8J5 24879244 IC50 = 230 nM T12499 C1XWO7 24879245 IC50 = 110 nM T12499 CA21RX 24879305 IC50 = 580 nM T12499 COF05N 24879306 IC50 = 1700 nM T12499 C6NIQ2 24879307 IC50 = 7.2 nM T12499 C45HIT 24879308 IC50 = 1200 nM T12499 CM6G7A 24879309 IC50 = 150 nM T12499 C0KW5Y 24879310 IC50 = 410 nM T12499 C7M9FB 24879311 IC50 = 25000 nM T12499 C0ZJX6 24879366 IC50 = 570 nM T12499 C5NA4Z 24879367 IC50 = 1800 nM T12499 CDJE41 24879368 IC50 = 7800 nM T12499 C4MG3B 24882476 IC50 = 0.6 nM T12499 C43HWQ 24883287 IC50 = 300 nM T12499 C8DA5Q 24883334 IC50 < 100 nM T12499 C0P6AU 24894017 IC50 < 1 nM T12499 CY8L7E 24896769 IC50 > 10000 nM T12499 C5ZM4T 24936119 IC50 = 7 nM T12499 C8DG1Y 24941253 IC50 > 10000 nM T12499 CLZ23U 24951610 IC50 > 30000 nM T12499 CU7I2E 24963046 IC50 = 122 nM T12499 CD5HQ0 24969301 IC50 > 10000 nM T12499 CT8OF0 24983254 IC50 = 25 nM T12499 CVF62Q 24983255 IC50 = 80 nM T12499 CX6FR3 24983298 IC50 = 4799 nM T12499 CEQ1F2 24983299 IC50 = 269 nM T12499 CQ46VT 24983495 IC50 = 292 nM T12499 C4EG8R 24993189 IC50 > 10000 nM T12499 CS3Q8B 24995659 IC50 > 2000 nM T12499 C6P1CX 25066843 IC50 = 28 nM T12499 C2KY1G 25094210 IC50 = 468 nM T12499 CTG49K 25110690 IC50 = 14 nM T12499 CG3XC9 25124150 IC50 = 1200 nM T12499 CO2IR5 25124816 IC50 > 3000 nM T12499 CF7C5B 25129829 IC50 > 10000 nM T12499 CXNM84 25129830 IC50 = 3814 nM T12499 CY2S1P 25129831 IC50 > 10000 nM T12499 C36FXD 25138012 IC50 = 14 nM T12499 CQMU82 25138148 IC50 = 0.4 nM T12499 CD9O6K 25138149 IC50 = 7 nM T12499 CO6N7P 25138154 IC50 > 25000 nM T12499 CGT1W6 25144294 IC50 = 12 nM T12499 CU7VR0 25144732 IC50 <= 1 nM T12499 C65YQG 25145144 IC50 = 384 nM T12499 C6BWZ8 25145145 IC50 = 2353 nM T12499 C78YWA 25145716 IC50 = 271 nM T12499 CL47VI 25145718 IC50 = 45 nM T12499 CSO82D 25154877 Ki = 0.04 nM T12499 CR0S2O 25195244 IC50 = 6 nM T12499 CNG96H 25210579 IC50 > 10000 nM T12499 CNQ9G5 25218180 IC50 < 1000 nM T12499 CRO8T9 25263033 Ki = 11 nM T12499 CC71QJ 27666048 IC50 = 10900 nM T12499 CXG02H 42226845 IC50 = 10000 nM T12499 CWS37O 42618140 IC50 > 25118.86 nM T12499 C2JV3O 42618143 IC50 = 15848.93 nM T12499 CG01BO 42618144 IC50 = 19952.62 nM T12499 CI9DK5 42628614 IC50 = 1300 nM T12499 CU9E4P 42629114 IC50 > 10000 nM T12499 CO42DC 44138048 IC50 > 10000 nM T12499 CL65QV 44138049 IC50 > 10000 nM T12499 CLW80F 44160269 IC50 = 2900 nM T12499 CO6HU7 44178069 IC50 = 731 nM T12499 CCFQ29 44187005 IC50 = 505 nM T12499 CEL61X 44229839 IC50 = 1700 nM T12499 CG1C9E 44269392 IC50 > 250000 nM T12499 CAT6W7 44269404 IC50 > 250000 nM T12499 C4SA3Y 44269518 IC50 > 250000 nM T12499 CVE17U 44271480 IC50 = 22000 nM T12499 CMZD96 44276805 IC50 > 2000 nM T12499 CDM14R 44277152 IC50 = 7.4 nM T12499 CFKY97 44277389 IC50 = 170 nM T12499 CP4Z9O 44277406 IC50 = 7700 nM T12499 C7AMH2 44277415 IC50 = 2800 nM T12499 CDSK68 44277416 IC50 = 30 nM T12499 CX0R6Z 44277458 IC50 = 400 nM T12499 CT03HW 44277459 IC50 = 17000 nM T12499 CP3FK1 44277464 IC50 > 12500 nM T12499 C6ILO7 44277479 IC50 = 1900 nM T12499 C54EAR 44277500 IC50 = 350000 nM T12499 CY9S4U 44277503 IC50 = 10000 nM T12499 CTOR69 44277507 IC50 = 1100 nM T12499 CM4QB2 44277523 IC50 = 1600 nM T12499 CTUE56 44277530 IC50 = 810 nM T12499 C94XTC 44277552 IC50 = 1900 nM T12499 C25XAV 44277553 IC50 = 6000 nM T12499 CM8ZU1 44277554 IC50 = 8500 nM T12499 CH70ZJ 44277555 IC50 = 2000 nM T12499 CT2C8Y 44277556 IC50 = 100 nM T12499 C7GVH2 44277568 IC50 = 1600 nM T12499 C0R5LM 44277575 IC50 = 1200 nM T12499 C48NAJ 44277576 IC50 = 1100 nM T12499 CC09ZV 44277619 IC50 = 1800 nM T12499 CF39VK 44277620 IC50 = 1200 nM T12499 CN26TB 44277621 IC50 = 1800 nM T12499 CUCN89 44277736 IC50 = 10 nM T12499 CHOA91 44277745 IC50 = 69 nM T12499 CNZR96 44277759 IC50 = 238 nM T12499 CQ2Y5R 44277762 IC50 = 53 nM T12499 CZ9NX1 44277837 IC50 = 60 nM T12499 COPF86 44277899 IC50 = 1600 nM T12499 CA74WK 44277900 IC50 = 1500 nM T12499 C6EJ0W 44278090 IC50 = 665 nM T12499 CG84EI 44278256 IC50 = 6.2 nM T12499 CZFQ76 44291533 IC50 = 19 nM T12499 CTX6L9 44293106 IC50 = 242000 nM T12499 CZ8W0T 44293432 IC50 > 2094000 nM T12499 CH3J2E 44299176 IC50 = 80 nM T12499 C27GVO 44299203 IC50 = 800 nM T12499 CY6WC0 44299236 IC50 = 400 nM T12499 C3RG0C 44299304 IC50 = 700 nM T12499 CJM26I 44299321 IC50 = 300 nM T12499 C9UGL3 44299325 IC50 = 700 nM T12499 CJEZ96 44299338 IC50 = 500 nM T12499 CNH34G 44299354 IC50 = 400 nM T12499 C82MSD 44299360 IC50 = 700 nM T12499 CF1N4E 44307877 IC50 = 178000 nM T12499 CD9J2B 44308029 IC50 = 638000 nM T12499 CC07XF 44308301 IC50 > 12500 nM T12499 CPK13M 44308362 IC50 = 110 nM T12499 C5P1AZ 44308363 IC50 > 12500 nM T12499 C5KA1C 44308378 IC50 > 12500 nM T12499 CM3O2B 44308391 IC50 = 3230 nM T12499 CWJ3T4 44308408 IC50 = 7250 nM T12499 C2X3TN 44308485 IC50 = 4400 nM T12499 CG8U6C 44308486 IC50 = 200 nM T12499 CG47MH 44308503 IC50 > 12500 nM T12499 C0M1IY 44308504 IC50 > 12500 nM T12499 C6PEF5 44308506 IC50 > 12500 nM T12499 C0XY4O 44308544 IC50 = 272 nM T12499 CP76DF 44308560 IC50 > 12500 nM T12499 C1S6MR 44308561 IC50 = 5600 nM T12499 C8MN4Y 44308567 IC50 > 12500 nM T12499 CB85WM 44308568 IC50 = 90 nM T12499 CMZI25 44308570 IC50 = 70 nM T12499 C13DBO 44308571 IC50 > 12500 nM T12499 C46QFM 44308664 IC50 > 12500 nM T12499 C2ZJH7 44308683 IC50 > 12500 nM T12499 CE5T3I 44308684 IC50 = 23000 nM T12499 CS1W5Z 44308685 IC50 > 12500 nM T12499 CEU2W4 44308690 IC50 < 2 nM T12499 C8EVZ0 44308700 IC50 > 12500 nM T12499 CWY9N5 44308701 IC50 = 4270 nM T12499 CIYE50 44308712 IC50 > 12500 nM T12499 C4U1MP 44308728 IC50 > 12500 nM T12499 CPA69W 44308729 IC50 = 3 nM T12499 CY6ZB5 44308830 IC50 = 220 nM T12499 C1I6RG 44308968 IC50 < 3 nM T12499 C1I0LN 44308993 IC50 < 3 nM T12499 CKVZ38 44308994 IC50 = 40 nM T12499 CF9I2S 44309110 IC50 = 1490 nM T12499 C8VX1L 44309229 IC50 = 942 nM T12499 CZQ4S0 44309230 IC50 < 3 nM T12499 CHF28G 44309494 IC50 = 131 nM T12499 CE9Z6L 44319231 IC50 = 820 nM T12499 CRWF80 44319232 IC50 = 2680 nM T12499 CF3QW5 44319234 IC50 = 3170 nM T12499 CFQ2L8 44319256 IC50 = 3170 nM T12499 CEL1H2 44319376 IC50 = 24 nM T12499 C4M6VJ 44319377 IC50 = 26 nM T12499 C7PS2Z 44319406 IC50 = 9 nM T12499 C9AT6W 44319420 IC50 = 4 nM T12499 C61ISW 44319421 IC50 = 2 nM T12499 CE1XR0 44319422 IC50 = 5 nM T12499 C6A0ZG 44319438 IC50 = 7 nM T12499 CIK71G 44319439 IC50 = 10 nM T12499 C3DXJ2 44319445 IC50 = 3 nM T12499 CIP4B3 44319451 IC50 = 9.4 nM T12499 CW5AR2 44319455 IC50 = 21 nM T12499 CUC1O5 44319479 IC50 = 4 nM T12499 CTKI85 44319593 IC50 = 100 nM T12499 C3Y4AS 44319618 IC50 = 15 nM T12499 CY5WL6 44319619 IC50 = 70 nM T12499 CKN3C5 44319631 IC50 = 26 nM T12499 C8ZF6H 44320538 IC50 > 3100 nM T12499 C4KS5N 44320732 IC50 = 1.1 nM T12499 CI6W3R 44320738 IC50 = 6 nM T12499 CC6YI7 44320769 Ki = 0.54 nM T12499 CBN1H4 44320801 IC50 = 403 nM T12499 C2USC1 44320802 IC50 > 3100 nM T12499 CTI86J 44320812 IC50 = 1890 nM T12499 C38YXS 44320815 IC50 = 2 nM T12499 C16ATL 44320820 IC50 > 3100 nM T12499 C6XRM9 44320821 IC50 = 1740 nM T12499 CMJ4Y2 44320829 IC50 = 1 nM T12499 CN7MI0 44320840 IC50 > 3100 nM T12499 CIQ1Y8 44320841 IC50 > 3100 nM T12499 C0WNK8 44320856 IC50 > 3100 nM T12499 C2C3HQ 44320857 IC50 > 3100 nM T12499 CL86PD 44320858 IC50 > 3100 nM T12499 C5WA0P 44320868 IC50 = 13 nM T12499 C9E2WN 44320869 IC50 = 10 nM T12499 C2B9QV 44320870 IC50 = 138 nM T12499 CKHP01 44320871 IC50 = 180 nM T12499 CCBU40 44320872 IC50 = 72 nM T12499 CP64WV 44320885 IC50 = 32 nM T12499 CJZ26I 44320905 IC50 = 8 nM T12499 C5JBP7 44320912 IC50 = 6 nM T12499 CE4OA6 44320964 IC50 > 3100 nM T12499 CR8Q1U 44320965 IC50 = 15 nM T12499 CK2X4T 44321004 IC50 = 5 nM T12499 CTJ69K 44321005 IC50 = 8 nM T12499 CD72YE 44321008 IC50 = 27 nM T12499 C29TOE 44321009 IC50 = 84 nM T12499 CI9U1O 44321055 IC50 = 20 nM T12499 CO0E8Y 44321057 IC50 = 17 nM T12499 CC68EY 44321060 IC50 = 1590 nM T12499 CBZ15Y 44321061 IC50 = 9 nM T12499 C14SKY 44321062 IC50 = 9 nM T12499 CO6T2M 44321063 IC50 = 403 nM T12499 CMX7N1 44321092 IC50 = 31 nM T12499 C7RE2Q 44321105 IC50 = 20 nM T12499 C3V4CY 44321106 IC50 = 5 nM T12499 CGNQ90 44321109 IC50 = 35 nM T12499 C1UE2V 44321110 IC50 = 13 nM T12499 CL6TY5 44321118 IC50 = 77 nM T12499 C9UTH8 44321136 IC50 = 21 nM T12499 CJ4Q9Z 44321140 IC50 = 20 nM T12499 C6OJ7A 44321151 IC50 = 3 nM T12499 C5TNF7 44321155 IC50 = 53 nM T12499 CLV2C0 44321167 IC50 = 7 nM T12499 C1LFI2 44321182 IC50 = 6 nM T12499 C74NLZ 44321198 IC50 = 10 nM T12499 C0PX6H 44321252 IC50 = 2 nM T12499 C3XB0U 44321258 IC50 = 6 nM T12499 C82NIY 44321259 IC50 = 8 nM T12499 CXM61A 44321260 IC50 = 2 nM T12499 CLAS90 44321316 IC50 = 235 nM T12499 CQX6F9 44321339 IC50 > 3100 nM T12499 CFD31S 44321340 IC50 = 327 nM T12499 C2Y3NE 44321361 IC50 = 1 nM T12499 C2FST3 44324647 IC50 = 81 nM T12499 CI8YR0 44324649 IC50 = 3800 nM T12499 C7JYP4 44324728 IC50 = 27000 nM T12499 CY69SU 44324769 IC50 = 18000 nM T12499 C3PED0 44331665 IC50 = 36000 nM T12499 CLG7Q6 44337120 IC50 = 6 nM T12499 CCGB45 44337122 IC50 = 2 nM T12499 CVW4D1 44337132 IC50 = 10 nM T12499 CE2AV7 44337155 IC50 = 5 nM T12499 CW4Q0X 44337161 IC50 = 7 nM T12499 CLB03R 44337267 IC50 = 3 nM T12499 C3LO9F 44337272 IC50 = 26 nM T12499 CC3BV7 44337290 IC50 = 7 nM T12499 CG7I6O 44337337 IC50 = 10 nM T12499 C7S6FQ 44337369 IC50 = 70 nM T12499 CQ2W7M 44337378 IC50 = 9 nM T12499 CP64NY 44337501 IC50 = 5 nM T12499 CSC40Y 44337509 IC50 = 5.4 nM T12499 CVP9L5 44337524 IC50 = 10 nM T12499 CH26ZA 44343296 IC50 > 10000 nM T12499 C2OMC0 44343708 IC50 > 500000 nM T12499 CQZM34 44355143 IC50 > 100000 nM T12499 CX1I0D 44355168 IC50 > 50000 nM T12499 C2F9DZ 44355323 IC50 > 100000 nM T12499 C4LKS3 44355443 IC50 = 10000 nM T12499 CJWK61 44355456 IC50 > 50000 nM T12499 C9YI1R 44355486 IC50 = 2500 nM T12499 CO5S7X 44379379 IC50 > 2000000 nM T12499 C6LSB4 44381409 IC50 = 340 nM T12499 C6LC8M 44381556 IC50 = 620 nM T12499 CC35RY 44386906 IC50 = 9650 nM T12499 C7PBJ8 44405918 IC50 = 2350 nM T12499 C0GR5F 44405919 IC50 = 3480 nM T12499 CO5WU8 44405977 IC50 = 8960 nM T12499 C9LX5Q 44406001 IC50 = 23200 nM T12499 CQ4U7T 44406037 IC50 = 106 nM T12499 CEVF48 44406058 IC50 = 9180 nM T12499 CF46WP 44406078 IC50 = 318 nM T12499 CUQ6R8 44406079 IC50 = 54 nM T12499 CG2W4V 44406138 IC50 > 50000 nM T12499 CV09DY 44410717 IC50 > 10000 nM T12499 CP3CI1 44410720 IC50 > 10000 nM T12499 C8W7AD 44410723 IC50 > 10000 nM T12499 CAT5X4 44410829 IC50 > 10000 nM T12499 CC6Y5P 44410844 IC50 > 10000 nM T12499 CG34TY 44410851 IC50 > 10000 nM T12499 C41EIA 44410869 IC50 > 10000 nM T12499 CB6AE8 44410948 IC50 > 10000 nM T12499 CXZG12 44410949 IC50 > 10000 nM T12499 CS7IE9 44410953 IC50 > 10000 nM T12499 CA9M4X 44410954 IC50 > 10000 nM T12499 C3SP5H 44410955 IC50 > 10000 nM T12499 C5D6YP 44410956 IC50 > 10000 nM T12499 C5W1VC 44410959 IC50 > 10000 nM T12499 CM1C2G 44410960 IC50 > 10000 nM T12499 CVSI80 44411048 IC50 > 10000 nM T12499 CN72BR 44411161 IC50 > 10000 nM T12499 C4AW0O 44411183 IC50 > 10000 nM T12499 C0WQ2A 44412535 IC50 > 10000 nM T12499 C9EL3N 44412536 IC50 > 10000 nM T12499 CCP34J 44412547 IC50 = 971 nM T12499 C0JW3X 44412548 IC50 = 2350 nM T12499 C71GSY 44412549 IC50 > 10000 nM T12499 C8YIO7 44412564 IC50 = 229 nM T12499 CD0XK4 44412565 IC50 = 1450 nM T12499 C45MBP 44412566 IC50 = 5990 nM T12499 C2Z9QT 44412568 IC50 = 32 nM T12499 CUAQ42 44412569 IC50 = 149 nM T12499 CIF8K3 44412570 IC50 = 52 nM T12499 C6IUQ8 44412571 IC50 = 3 nM T12499 C7C2NQ 44412577 IC50 = 708 nM T12499 CRHK90 44412586 IC50 = 28 nM T12499 C8WX2G 44412587 IC50 = 96 nM T12499 CRA02Z 44412602 IC50 = 418 nM T12499 C42YIW 44412603 IC50 > 10000 nM T12499 CR18DN 44412728 IC50 = 4 nM T12499 C7LBS4 44412754 IC50 > 10000 nM T12499 C6P9LY 44412768 IC50 > 10000 nM T12499 C4KR2P 44412769 IC50 = 2580 nM T12499 CSL1C7 44412787 IC50 > 10000 nM T12499 CV12PJ 44412788 IC50 = 155 nM T12499 CO0R3U 44412789 IC50 = 3 nM T12499 CT1EU9 44412790 IC50 = 4 nM T12499 C5JQ0S 44412804 IC50 > 10000 nM T12499 CZE9H2 44412805 IC50 = 4490 nM T12499 C1XOC5 44412806 IC50 = 230 nM T12499 CFB16V 44412829 IC50 = 1820 nM T12499 CA6GK9 44412842 IC50 = 3130 nM T12499 CLS5H6 44412843 IC50 = 301 nM T12499 CP9KT1 44412856 IC50 = 190 nM T12499 CNJS19 44412857 IC50 = 4290 nM T12499 CS05HP 44412870 IC50 = 6 nM T12499 C50CHI 44412871 IC50 = 9 nM T12499 C4TD2F 44412992 IC50 = 3860 nM T12499 C0F3NI 44414305 IC50 = 143 nM T12499 C6FY3V 44414306 IC50 = 26 nM T12499 C3E4AR 44414321 IC50 = 43 nM T12499 C7KZV2 44414322 IC50 = 21141 nM T12499 CJM06T 44414347 IC50 > 50000 nM T12499 C8R4PT 44414468 IC50 = 182 nM T12499 CXR08Z 44414469 IC50 = 2814 nM T12499 CE1V5J 44414487 IC50 = 71 nM T12499 CBSJ78 44414580 IC50 = 21 nM T12499 C3Z7VW 44414581 IC50 = 3 nM T12499 CC8R6T 44414609 IC50 = 4802 nM T12499 CRB78V 44414623 IC50 = 2837 nM T12499 C8ED2X 44414624 IC50 = 10 nM T12499 CXTJ75 44414636 IC50 = 179 nM T12499 CH0VO6 44414656 IC50 = 7269 nM T12499 CCF69N 44414657 IC50 = 285 nM T12499 C8G5YN 44415111 IC50 = 1 nM T12499 CHJ7T1 44415158 IC50 = 1 nM T12499 C5TQ4F 44415291 IC50 = 1 nM T12499 C32UJZ 44419930 IC50 = 7700 nM T12499 CR2WY4 44419931 IC50 > 10000 nM T12499 C9Y1FS 44419937 IC50 > 10000 nM T12499 CAP2D3 44419938 IC50 = 1286 nM T12499 C2I3LY 44419942 IC50 = 294 nM T12499 CC31RB 44419943 IC50 = 79 nM T12499 CCV9U5 44419947 IC50 = 384 nM T12499 CXUV94 44419948 IC50 = 71 nM T12499 C76LAG 44419953 IC50 = 137 nM T12499 C3C0SW 44419954 IC50 = 3 nM T12499 CSFI82 44419961 IC50 = 17 nM T12499 CB47IS 44419962 IC50 = 65 nM T12499 C6W7YQ 44419967 IC50 = 44 nM T12499 CX1U0E 44419972 IC50 = 130 nM T12499 CSH8I0 44419973 IC50 = 45 nM T12499 CS83YT 44419977 IC50 = 165 nM T12499 C2SZ3E 44419978 IC50 = 519 nM T12499 CL4O8E 44419981 IC50 = 43 nM T12499 C25NUJ 44419988 IC50 = 333 nM T12499 CA9K5Y 44419989 IC50 = 193 nM T12499 CKWI23 44419990 IC50 > 10000 nM T12499 CTC09S 44419991 IC50 = 4.2 nM T12499 CK93IX 44419994 IC50 = 5564 nM T12499 C3N6EX 44419995 IC50 = 8640 nM T12499 CCS6L8 44419998 IC50 > 10000 nM T12499 C9RBH4 44419999 IC50 = 24 nM T12499 C26YUL 44420000 IC50 = 6.8 nM T12499 C8HOG7 44422489 IC50 = 20 nM T12499 CBS5K2 44432304 IC50 = 17600 nM T12499 CFJX63 44432305 IC50 = 240 nM T12499 C54URN 44432306 IC50 = 541 nM T12499 C57FJN 44432307 IC50 = 130 nM T12499 C0PHT6 44432309 IC50 = 4470 nM T12499 CA9SP2 44432315 IC50 = 31 nM T12499 CL05KJ 44438314 IC50 = 1210 nM T12499 C3XQK1 44438318 IC50 = 6 nM T12499 CSB51N 44438320 IC50 = 6 nM T12499 CGV37F 44440254 IC50 = 16038 nM T12499 C5JUV3 44440256 IC50 > 50000 nM T12499 CFB56S 44440259 IC50 = 21382 nM T12499 CEW9G2 44440261 IC50 = 26529 nM T12499 CI9W8E 44447914 IC50 = 3310 nM T12499 CUB12D 44449577 IC50 = 185 nM T12499 CDV6X9 44454507 IC50 = 7 nM T12499 C6SMY7 44454538 IC50 = 53 nM T12499 CZI92T 44454651 IC50 = 84 nM T12499 CIA39D 44454676 IC50 = 45 nM T12499 C7DGA2 44454678 IC50 = 19 nM T12499 C1F3LT 44454702 IC50 = 22 nM T12499 CCW57R 44454703 IC50 = 101 nM T12499 CFS7W2 44454728 IC50 = 25 nM T12499 CTL43P 44454729 IC50 = 41 nM T12499 CZC95J 44454731 IC50 = 44 nM T12499 CIB24G 44457163 IC50 > 12500 nM T12499 CN8HV0 44457164 IC50 = 60 nM T12499 C3I6ZY 44457241 IC50 = 810 nM T12499 C67VXQ 44457503 IC50 = 1 nM T12499 C71EPS 44460198 IC50 = 7.5 ug.mL-1 T12499 C3PAD4 44460222 IC50 > 10 ug.mL-1 T12499 CLNZ91 44460237 IC50 > 10 ug.mL-1 T12499 C9Z8XJ 44460238 IC50 = 1.2 ug.mL-1 T12499 CH9F0N 44460247 IC50 > 10 ug.mL-1 T12499 CV1Q0D 44460258 IC50 = 0.62 ug.mL-1 T12499 CF9Z3W 44461749 IC50 = 710 nM T12499 C84RLC 44461768 IC50 = 1500 nM T12499 C3WV2D 44461769 IC50 = 310 nM T12499 C5KD6H 44461778 IC50 = 5000 nM T12499 CGR15K 44461807 IC50 = 1400 nM T12499 CW5QX9 44461811 IC50 = 470 nM T12499 COK3T6 44461852 IC50 = 1700 nM T12499 CN0P6M 44461863 IC50 = 5000 nM T12499 CNW9M3 44461865 IC50 = 110 nM T12499 CEDL98 44461873 IC50 = 880 nM T12499 CXDB59 44461880 IC50 = 600 nM T12499 C24SNH 44461881 IC50 > 5000 nM T12499 CFJ28C 44461889 IC50 = 1000 nM T12499 CH7M6G 44461919 IC50 = 1700 nM T12499 CF08CB 44462184 IC50 > 5000 nM T12499 CJ3QZ6 44462200 IC50 = 32 nM T12499 CQ3PB5 44462201 IC50 = 5000 nM T12499 C5WL1F 44473009 IC50 = 1200 nM T12499 CEG1S5 44473011 IC50 = 600 nM T12499 C46OMR 44473016 IC50 = 47000 nM T12499 C7N2AQ 44473101 IC50 = 280 nM T12499 C4MG3F 44473102 IC50 = 12 nM T12499 CA85NJ 44473103 IC50 = 150 nM T12499 CYH6P3 44520205 IC50 = 566 nM T12499 CWPT02 44555415 IC50 = 0.12 nM T12499 C3VRO9 44557921 IC50 > 10000 nM T12499 CF16QB 44560451 IC50 = 546 nM T12499 C0U8DH 44560546 IC50 = 2760 nM T12499 C3XTA7 44562721 Ki = 13 nM T12499 CO3SK5 44563262 IC50 = 220 nM T12499 C3HW7L 44570553 IC50 > 30000 nM T12499 C17PVE 44570554 IC50 > 30000 nM T12499 CLOY92 44570599 IC50 = 500 nM T12499 CK06LT 44570600 IC50 = 7000 nM T12499 CJY8S0 44570884 IC50 = 38000 nM T12499 CWFB42 44571820 IC50 = 710 nM T12499 CW8P9Y 44576189 IC50 = 7000 nM T12499 C9VXN3 44578709 IC50 > 10000 nM T12499 C3J9AT 44578884 IC50 = 1167 nM T12499 CA7R2X 44579356 EC50 = 14400 nM T12499 CNS6A4 44579357 EC50 = 23300 nM T12499 C31TFG 44579358 EC50 = 18400 nM T12499 C53ZVU 44579359 IC50 = 50000 nM T12499 CM9TC5 44579360 EC50 > 150000 nM T12499 CV01SB 44579361 EC50 = 4400 nM T12499 C7Q1VU 44580077 IC50 = 6000 nM T12499 CL90SE 44580358 IC50 = 2000 nM T12499 CK1VE7 44580420 IC50 = 8000 nM T12499 CH2R7X 44580449 IC50 = 3000 nM T12499 C1VH0C 44580532 IC50 > 16000 nM T12499 CXC52J 44580649 IC50 = 3000 nM T12499 CE32BQ 44580689 IC50 = 70 nM T12499 C8Z5AX 44580778 IC50 = 1000 nM T12499 C6RJZ5 44581565 IC50 = 48 nM T12499 CV5GD1 44589002 IC50 = 180 nM T12499 C83KEG 44589022 IC50 = 590 nM T12499 CL3DO5 44593603 IC50 = 100 ug.mL-1 T12499 C4EP8N 44593604 IC50 > 800 ug.mL-1 T12499 C3KS6C 44593605 IC50 = 700 ug.mL-1 T12499 C8WX5D 44593606 IC50 > 800 ug.mL-1 T12499 CU3RF1 45139989 IC50 > 10000 nM T12499 CQGZ06 45139991 IC50 > 10000 nM T12499 C6F8UE 45261965 IC50 = 10000 nM T12499 C0T2MQ 45262036 IC50 = 20000 nM T12499 CKQ5U9 45266326 IC50 > 1936000 nM T12499 C5Q4DT 45266328 IC50 > 2088000 nM T12499 COE8U0 45267045 IC50 = 41000 nM T12499 CY83PR 45267327 IC50 = 300 nM T12499 C84QFJ 45269074 IC50 > 1000 nM T12499 C3DH8I 45273358 IC50 > 1000 nM T12499 C6E2SC 45482700 IC50 > 10000 nM T12499 CZXH74 45482750 IC50 > 10000 nM T12499 C5S8MA 45485083 IC50 = 520 nM T12499 CZ8GR7 45486752 IC50 = 2073 nM T12499 C0D5TG 45486762 IC50 = 1770 nM T12499 CD40LR 45486763 IC50 = 1.5 nM T12499 C2D7YJ 45486771 IC50 = 47 nM T12499 CH4VY9 45486772 IC50 = 243 nM T12499 CP5YK9 45486775 IC50 = 0.06 nM T12499 CPC7I2 45486776 IC50 = 0.07 nM T12499 CG7RM9 45486777 IC50 = 1 nM T12499 CNC7M3 45486780 IC50 = 106 nM T12499 CZN60P 45486785 IC50 = 203 nM T12499 C1BMI3 45486789 IC50 > 1000 nM T12499 CPJD02 45486792 IC50 = 0.4 nM T12499 CB49PG 45486793 IC50 = 0.07 nM T12499 CR41JA 45486794 IC50 = 0.2 nM T12499 C4NTY8 45486795 IC50 = 1.8 nM T12499 CT4IR9 45486796 IC50 = 0.2 nM T12499 CXC03L 45486797 IC50 = 0.45 nM T12499 C3W9RC 45486798 IC50 = 115 nM T12499 CSK69U 45486806 IC50 > 20000 nM T12499 CTU89Y 45486814 IC50 = 110 nM T12499 CW2Q6T 45486815 IC50 = 10 nM T12499 CW42YX 45487634 IC50 > 1000 nM T12499 CG92CF 46175112 IC50 = 9200 nM T12499 C96BNW 46179972 IC50 = 35 nM T12499 CZBL95 46220496 IC50 = 18 nM T12499 CY3HW5 46224684 IC50 = 4600 nM T12499 C2P9QO 46228508 IC50 = 584 nM T12499 C6E5PY 46228822 IC50 > 10000 nM T12499 C3T8AM 46228951 IC50 = 5020 nM T12499 CYT37A 46232443 IC50 > 50000 nM T12499 C48ZVW 46232555 IC50 = 14000 nM T12499 CS9B1U 46232556 IC50 = 28000 nM T12499 C7ON5A 46233287 IC50 > 10000 nM T12499 CQW97N 46846072 IC50 = 790 nM T12499 COTJ39 46863083 IC50 = 1000 nM T12499 C7H4YM 46865419 IC50 > 10000 nM T12499 CC2O9R 46865656 IC50 = 5011.87 nM T12499 CX43UQ 46871756 IC50 = 7 nM T12499 CLS29B 46872626 IC50 > 10000 nM T12499 CRS61F 46879438 IC50 = 702 nM T12499 C27JEF 46879439 IC50 = 22 nM T12499 CF0T8P 46879440 IC50 = 406 nM T12499 C12RMW 46879441 IC50 = 38 nM T12499 CH2D7N 46879442 IC50 = 19 nM T12499 CI6OD8 46879443 IC50 = 38 nM T12499 C7YD4Q 46879444 IC50 = 11 nM T12499 C8MN5Q 46879445 IC50 = 18 nM T12499 CX6SW2 46879446 IC50 = 275 nM T12499 CNF3V6 46879447 IC50 = 4456 nM T12499 CW46VY 46879448 IC50 = 12 nM T12499 CLK6X3 46879907 IC50 = 58 nM T12499 CRPU47 46879908 IC50 = 7 nM T12499 C1TIE9 46880013 IC50 = 715 nM T12499 C2A8KO 46880066 IC50 = 230 nM T12499 CBRP80 46880067 IC50 = 23 nM T12499 C3FY2B 46880068 IC50 = 13 nM T12499 CX89TY 46880069 IC50 = 5 nM T12499 CB0XY1 46880070 IC50 = 26 nM T12499 CUD81V 46880071 IC50 = 38 nM T12499 CZP58Q 46880072 IC50 = 71 nM T12499 CC8OF9 46880073 IC50 = 204 nM T12499 CF41HG 46880098 IC50 = 132 nM T12499 C6O2YG 46880099 IC50 = 83 nM T12499 CI78DM 46880100 IC50 = 7 nM T12499 CU04ZK 46880101 IC50 = 16 nM T12499 C4E0MF 46880133 IC50 = 17 nM T12499 COJ16A 46880134 IC50 = 43 nM T12499 C71MGJ 46880135 IC50 = 63 nM T12499 C3R6TL 46880213 IC50 = 90 nM T12499 CT8BQ4 46880214 IC50 = 2280 nM T12499 C0JTO4 46880215 IC50 = 616 nM T12499 CAFN49 46880216 IC50 > 2500 nM T12499 CMVZ46 46886319 Ki = 39.81 nM T12499 C2O8RZ 46886323 IC50 = 71 nM T12499 CM02UJ 46890253 IC50 = 387 nM T12499 CB7VI8 46890254 IC50 = 10000 nM T12499 C7V3IA 46890314 IC50 = 4087 nM T12499 CHE6A1 46890315 IC50 = 1856 nM T12499 C1YS5A 46890918 IC50 = 28 nM T12499 CJ5S3N 46890968 IC50 = 4 nM T12499 CAGE32 46890969 IC50 = 23 nM T12499 C3A7BP 46890970 IC50 = 24 nM T12499 CTV73J 46890971 IC50 = 16 nM T12499 CUX9B4 46891024 IC50 = 8 nM T12499 CG35WP 46891025 IC50 = 6 nM T12499 C3FBH0 46891026 IC50 = 8 nM T12499 CYOU90 46891080 IC50 = 4 nM T12499 CJ16KH 46891081 IC50 = 106 nM T12499 C7DOF4 46891082 IC50 = 14 nM T12499 CM14YO 46891147 IC50 = 5 nM T12499 CRPL41 46891148 IC50 = 128 nM T12499 C6FJ7G 46891184 IC50 = 116 nM T12499 C1B2UZ 46891185 IC50 = 546 nM T12499 CYM5B2 46891226 IC50 > 1000 nM T12499 C2DZE0 46891227 IC50 = 209 nM T12499 C1W0JX 46891228 IC50 = 7 nM T12499 CI3VZ0 46891275 IC50 = 699 nM T12499 C28ELR 46912278 Ki = 100 nM T12499 CD4L7V 46912279 Ki = 63.1 nM T12499 C7S2HO 46913757 Ki = 79.43 nM T12499 CT46HI 46913758 Ki = 100 nM T12499 C9PAT7 46927672 IC50 = 10 nM T12499 C60GAV 46929544 IC50 = 385 nM T12499 CHSF07 49806372 IC50 > 1000 nM T12499 C9L3XR 49838879 IC50 = 7000 nM T12499 CRA74I 49842779 IC50 > 10000 nM T12499 CF91RS 49843531 IC50 > 10000 nM T12499 CQ3KU9 50899556 IC50 = 430 nM T12499 C2Y6QS 50938552 IC50 > 10000 nM T12499 C6XYT1 50941838 IC50 > 100000 nM T12499 C61DVY 50990961 IC50 = 610 nM T12499 CV3UP9 50992247 IC50 = 170 nM T12499 CAZQ43 51003133 IC50 = 61 nM T12499 C9NYP4 51036677 IC50 > 10000 nM T12499 C4WRY3 51037112 IC50 > 10000 nM T12499 CRI28Z 51037948 IC50 > 10000 nM T12499 CXA03W 52920796 IC50 = 470 nM T12499 CEQN27 52936621 Ki = 490 nM T12499 C3LB5V 52941849 IC50 = 970 nM T12499 CC42PX 52942070 IC50 = 568 nM T12499 CW2X5E 52944268 IC50 = 20 nM T12499 C9PX2J 52945752 IC50 = 94 nM T12499 CL4ED3 52945753 IC50 = 440 nM T12499 CIR3Q0 52947964 IC50 > 10000 nM T12499 C6OTY5 53251320 IC50 > 19000 nM T12499 CE8OY2 53317913 IC50 < 1 nM T12499 CZ0BV7 53320342 IC50 > 10000 nM T12499 C2W9OA 53324451 IC50 = 4700 nM T12499 CD4H3S 53354074 Ki > 1000 nM T12499 C8NA4L 53384644 IC50 > 30000 nM T12499 CZ1CI3 53469824 IC50 = 741 nM T12499 CXA92G 53484170 IC50 > 20000 nM T12499 C7UK2N 53484181 IC50 > 20000 nM T12499 CKD9H6 53484182 IC50 > 20000 nM T12499 CH05EO 53484183 IC50 = 14114 nM T12499 CAR45T 53484184 IC50 > 20000 nM T12499 CE1ZK6 54759168 IC50 > 10000 nM T12499 C8AB1J 54759606 Ki = 2000 nM T12499 CM8JX1 56604907 IC50 = 10 nM T12499 CN9QD7 56643097 IC50 > 10000 nM T12499 C8GJ9S 56658692 IC50 = 330 nM T12499 CK3A4Z 56658700 IC50 = 3417 nM T12499 C1JD6Z 56658841 IC50 = 603 nM T12499 C98WRJ 56658842 IC50 = 169 nM T12499 C2Z9YO 56662177 IC50 = 4648 nM T12499 CR50XZ 56662178 IC50 = 3208 nM T12499 C8NGC7 56662179 IC50 = 597 nM T12499 C3H0VQ 56662180 IC50 = 945 nM T12499 CWM35E 56662181 IC50 > 20000 nM T12499 CB0VE5 56662182 IC50 > 20000 nM T12499 CEI39Q 56665634 IC50 = 284 nM T12499 CG5K2Q 56665635 IC50 = 365 nM T12499 CVEM27 56665636 IC50 > 20000 nM T12499 CDT3K4 56665637 IC50 > 20000 nM T12499 C9ZTL3 56669088 IC50 > 20000 nM T12499 CC8F0R 56669218 IC50 = 2000 nM T12499 CXW95K 56669219 IC50 = 2262 nM T12499 C8R9TW 56672548 IC50 = 476 nM T12499 C0ROQ7 56672549 IC50 = 10400 nM T12499 CI6K1R 56672550 IC50 > 20000 nM T12499 CC5NQ4 56672551 IC50 = 420 nM T12499 CY0PA7 56672679 IC50 = 722 nM T12499 CP6AE8 56672680 IC50 = 1200 nM T12499 C0GUO4 56672681 IC50 = 70 nM T12499 CWT5X6 56674974 IC50 = 2000 nM T12499 CJA2N4 56675924 IC50 = 1830 nM T12499 C95JAC 56681742 IC50 = 660 nM T12499 CLKP65 56682548 IC50 = 722 nM T12499 CW2YZ7 56682555 IC50 = 539 nM T12499 C1JWN7 56682556 IC50 = 1501 nM T12499 CS9YF2 56682557 IC50 > 20000 nM T12499 COM56E 56682674 IC50 = 3710 nM T12499 CG2A4M 56682676 IC50 = 10 nM T12499 CBOD63 56835089 IC50 > 30000 nM T12499 CI5ZJ7 56835161 IC50 > 100000 nM T12499 CJBL48 56925034 IC50 = 81 nM T12499 CR16SD 56947170 IC50 = 110 nM T12499 CJ47MX 56963907 IC50 = 120 nM T12499 C9L6FD 56963908 IC50 = 3300 nM T12499 CE50IB 56963909 IC50 > 10000 nM T12499 CPHX64 57325478 IC50 > 50000 nM T12499 CQ9BW4 57325479 IC50 > 50000 nM T12499 CE1A9V 57394653 IC50 = 755 nM T12499 CNV76Z 57394656 IC50 = 2790 nM T12499 CD6Y9Z 57395116 IC50 > 30000 nM T12499 C8W6IG 57395117 IC50 > 30000 nM T12499 CG7S0D 57396882 IC50 > 30000 nM T12499 C0UDY9 57401151 IC50 > 30000 nM T12499 CZSM95 57412684 IC50 > 10000 nM T12499 CVK0G4 58056356 IC50 > 50000 nM T12499 CH7L5N 58172700 IC50 = 1448 nM T12499 CWXC70 58180596 IC50 = 1800 nM T12499 C6BPR2 58985201 IC50 > 30000 nM T12499 CZ3TG1 59375154 IC50 = 108 nM T12499 CP9A8T 59503659 IC50 = 271 nM T12499 C1MA6J 59503711 IC50 > 3000 nM T12499 CX29EU 59503744 IC50 = 579 nM T12499 CXJ63M 59603829 IC50 = 37 nM T12499 CQEU96 59603842 IC50 = 3.9 nM T12499 CLH49Z 59790029 IC50 = 3 nM T12499 COH62U 60097413 IC50 > 5000 nM T12499 C1MR8Q 60097495 IC50 > 10000 nM T12499 C9QRX3 60098131 IC50 = 200 nM T12499 CUBL90 66545750 IC50 = 1380 nM T12499 C1HSE0 67035086 IC50 = 690 nM T12499 CWI6K5 67035106 IC50 > 10000 nM T12499 C38RGB 67035556 IC50 = 8900 nM T12499 CV3HW2 67035568 IC50 = 7400 nM T12499 C37NKO 67129970 IC50 = 7790 nM T12499 CK80LJ 67130050 IC50 = 7510 nM T12499 CV63UL 67240318 IC50 > 10000 nM T12499 CZC9M5 67469084 IC50 = 12600 nM T12499 C8I7GC 68293638 IC50 = 8900 nM T12499 CD56XK 68293660 IC50 = 4900 nM T12499 C7GRV2 68755406 IC50 = 3700 nM T12499 C0HA8V 68783839 IC50 = 7 nM T12499 CAIO65 68796885 IC50 = 69 nM T12499 C5DGR9 69036886 IC50 = 818 nM T12499 C7VJ6A 70647728 IC50 = 150 nM T12499 C82FIP 70686752 IC50 = 52 nM T12499 C0QX3Y 70688829 IC50 = 79 nM T12499 CSOT12 70693058 IC50 = 620 nM T12499 CS6NW3 70693059 IC50 = 960 nM T12499 CWM62Q 70694846 Ki = 79.43 nM T12499 C1IEJ2 70789254 IC50 = 113000 nM T12499 C8T7ZP 70789255 IC50 = 20000 nM T12499 COU73Y 71226944 IC50 = 11 nM T12499 C40JOZ 71235465 IC50 = 28 nM T12499 C91HPI 71300299 IC50 > 5000 nM T12499 C2HBG8 71450398 IC50 = 2.35 ug.mL-1 T12499 CKOE90 71451677 IC50 = 1023 nM T12499 CEBO91 71452977 IC50 = 1300 nM T12499 C8AH1B 71454033 IC50 = 12.76 ug.mL-1 T12499 CI37UR 71454035 IC50 = 0.94 ug.mL-1 T12499 CX3AN8 71454037 IC50 > 50 ug.mL-1 T12499 C9ZVW4 71459442 IC50 = 7.91 ug.mL-1 T12499 CO9PR0 71459445 IC50 > 50 ug.mL-1 T12499 CB9V6C 71461186 IC50 = 7.17 ug.mL-1 T12499 CJ6T0K 71462927 IC50 = 4.52 ug.mL-1 T12499 CMV23P 71462929 IC50 = 11.88 ug.mL-1 T12499 C6HF8S 71521082 IC50 = 44620 nM T12499 C9Z3AI 71521083 IC50 = 11050 nM T12499 C5ZKU7 71546969 IC50 = 493 nM T12499 C7ARI9 71547113 IC50 = 617 nM T12499 CCN01X 71547862 IC50 > 10000 nM T12499 C1NPL0 71552941 IC50 > 30000 nM T12499 CA4PS8 71552942 IC50 > 30000 nM T12499 C3UA9C 71553011 IC50 = 15020 nM T12499 CEZ15Y 71553012 IC50 = 1360 nM T12499 CVIA91 71553085 IC50 = 610 nM T12499 C1TR3O 71553152 IC50 = 3680 nM T12499 C7ZR4F 71555873 IC50 = 5 nM T12499 CRX81Q 71575642 IC50 > 10000 nM T12499 CZ31PU 71583657 IC50 = 3200 nM T12499 C3OS8U 71714087 IC50 = 140 nM T12499 C92AZQ 71714088 IC50 = 6050 nM T12499 CN1Y9I 71714230 IC50 = 390 nM T12499 CM6NE9 71714231 IC50 = 50 nM T12499 CG28AP 71714232 IC50 = 120 nM T12499 C91CRY 71714233 IC50 = 1100 nM T12499 C67HDT 71714234 IC50 = 180 nM T12499 CRS05F 71714235 IC50 = 7 nM T12499 CVC19T 71714373 IC50 = 330 nM T12499 CD5C8J 71714374 IC50 = 1100 nM T12499 C51ISR 71714375 IC50 = 360 nM T12499 C5HJK2 71714376 IC50 = 120 nM T12499 C70SJV 71714377 IC50 = 1000 nM T12499 C7E6YV 71720026 IC50 = 264 nM T12499 CF04BD 71765399 IC50 = 6400 nM T12499 CZM1K4 71765510 IC50 = 412 nM T12499 C4KV0T 71765585 IC50 = 1300 nM T12499 C98LKV 71777716 Ki = 440 nM T12499 C3MI4O 71777717 Ki = 55 nM T12499 CD28XR 71816087 IC50 = 2.3 nM T12499 CS10DX 72544168 Ki = 150 nM T12499 CQH45K 72544389 Ki = 110 nM T12499 CMS5O0 72544619 Ki = 1700 nM T12499 CFTK59 72705466 Ki > 25118.86 nM T12499 C1CU0H 72705467 Ki = 15848.93 nM T12499 CX2AW3 72705468 Ki = 100 nM T12499 CVK4Z3 72705469 Ki = 501.19 nM T12499 C4ND6R 72705470 Ki = 100 nM T12499 CT67YO 72706106 Ki = 199.53 nM T12499 C3L2WD 73292576 Ki = 1800 nM T12499 C52LFH 73292907 Ki = 1400 nM T12499 C4FY5U 73346554 Ki = 79.43 nM T12499 CPGD07 73348027 Ki = 2511.89 nM T12499 C05XEV 73348028 Ki = 3162.28 nM T12499 CUW70Y 73348034 Ki = 251.19 nM T12499 CFEU95 73348035 Ki = 501.19 nM T12499 C6K0UL 73348036 Ki = 316.23 nM T12499 CD7X5Q 73348645 IC50 = 360 nM T12499 CD6KE7 73349574 Ki = 19.95 nM T12499 CV8UR4 73351136 Ki = 50.12 nM T12499 CAS60G 73352600 Ki = 125.89 nM T12499 CX75YR 73352604 Ki = 100 nM T12499 C5YKB4 73352605 Ki = 501.19 nM T12499 C03YUP 73355623 Ki = 251.19 nM T12499 CSUZ81 73356106 IC50 = 120000 nM T12499 C6UA4K 73356522 IC50 > 3000 nM T12499 C1A9PR 73357167 Ki = 316.23 nM T12499 CMEV76 74983355 Ki = 340 nM T12499 C0RP9Y 76309810 Ki = 46 nM T12499 C2A7SL 76320747 Ki = 890 nM T12499 CPG3A5 86302574 IC50 > 30000 nM T12499 C1HW4B 89735655 IC50 = 5000 nM T12499 CFB75T 90479825 IC50 = 136 nM T12499 CN7CG9 90644798 IC50 = 142 nM T12499 CLZ71J 90644800 IC50 = 7 nM T12499 C19HKY 90644801 IC50 = 16 nM T12499 C3MU1B 90644802 IC50 = 4 nM T12499 CI0VF7 90644803 IC50 = 4 nM T12499 COA7S0 90644804 IC50 = 4 nM T12499 CY5Z3V 90644805 IC50 = 7 nM T12499 CGIL57 90644806 IC50 = 0.9 nM T12499 CUDB61 90644807 IC50 = 287 nM T12499 CY0UC4 90645194 IC50 > 10000 nM T12499 CE3OV2 90645543 Ki = 1800 nM T12499 CLBC06 90663203 IC50 > 10000 nM T12499 CI8XJ4 90663933 IC50 = 6.24 nM T12499 CMH6T8 90664306 IC50 = 83 nM T12499 CYHR27 91664373 IC50 = 52 nM T12499 C6J0GR 91809511 IC50 = 5900 nM T12499 CAU45T 91971978 IC50 > 30000 nM T12499 CWF97Y 92045039 IC50 = 1220 nM T12499 CY7BI2 118706214 IC50 > 10000 nM T12499 CTP2E8 118737132 Ki = 210 nM T12499 C5GTM2 118737133 Ki = 240 nM T12499 C7MJ5H 118737134 Ki = 640 nM T12499 C3XF2A 118737135 Ki = 600 nM T12499 CNP5K8 118737136 Ki = 660 nM T12499 C8FDR1 118737137 Ki > 2500 nM T12499 C37DUM 121293882 IC50 > 2000 nM T12499 CXQR89 121294143 IC50 > 2000 nM T12499 C08KEM 122179540 IC50 = 2000 nM T12499 CG0RP7 122179547 IC50 = 3000 nM T12499 C1A0SQ 122179548 IC50 = 5200 nM T12499 CLPI09 122180346 IC50 = 13000 nM T12499 CFKD32 122191637 IC50 = 569 nM T12499 C4X7SD 122192466 IC50 > 10000 nM T12499 C8F0DQ 129909860 IC50 = 36 nM T12499 C71KMN 130429150 IC50 = 337 nM T12499 CSG8J3 130429224 IC50 = 77 nM T12499 C5PT1M 130429242 IC50 = 468 nM T12499 C0UNO3 130429244 IC50 = 18 nM T12499 CGFK71 130429248 IC50 = 44 nM T12499 CEX8D1 130429250 IC50 = 137 nM T12499 C9J6ZK 130429255 IC50 = 106 nM T12499 C6OMB1 132204257 IC50 = 425 nM T12499 CV89JM 132231876 IC50 = 420 nM T12499 C6ROQ3 132546210 IC50 = 12 nM T12499 C54FXD 134957362 IC50 > 10000 nM T12499 C1GY2T 135156251 EC50 > 10000 nM T12499 C73DLE 135399258 IC50 = 610000 nM T12499 C1UZW9 135400585 IC50 > 2000000 nM T12499 C6RDV7 135402873 IC50 > 50000 nM T12499 COH41B 135403151 IC50 > 2514000 nM T12499 CR3XN0 135408977 IC50 > 1000000 nM T12499 C7LI1N 135408978 IC50 = 1000 nM T12499 CMB3F6 135409035 IC50 = 200 nM T12499 CHS5X0 135409466 IC50 = 2 ug.mL-1 T12499 C2DH1R 135412832 IC50 = 20 ug.mL-1 T12499 CUI1B3 135417010 IC50 = 1000 nM T12499 CU60YC 135431661 IC50 = 2550 nM T12499 C4VH8I 135438239 IC50 = 600000 nM T12499 C8GZ2B 135449326 Ki = 1200 nM T12499 C5G9XP 135452204 IC50 > 2000000 nM T12499 CX35PB 135468746 IC50 = 500 nM T12499 C9BK5Y 135469311 IC50 = 750000 nM T12499 CWPK94 135478626 IC50 = 40000 nM T12499 CRTS92 135484881 IC50 = 1900000 nM T12499 CZ9L3S 135499405 IC50 = 105000 nM T12499 CTJ48K 135524085 IC50 = 4300 nM T12499 CUT1W7 135524168 IC50 = 6000 nM T12499 CCHD04 135533486 IC50 = 1005000 nM T12499 C3CRI9 135546620 IC50 = 162000 nM T12499 CJ03PU 135566610 IC50 = 162.1 nM T12499 CQ9A5I 135566611 IC50 = 3178.4 nM T12499 C42TOW 135566612 IC50 = 39.2 nM T12499 CN48IF 135566613 IC50 = 203.2 nM T12499 C67IYS 135566618 IC50 = 63.9 nM T12499 CZFA70 135611366 IC50 = 1360 nM T12499 CP54JV 135752285 IC50 = 352000 nM T12499 CX4ZB3 135863110 IC50 > 30000 nM T12499 CYDM01 135891431 IC50 = 0.72 nM T12499 CGI34T 135971386 IC50 = 2.3 nM T12499 CI5U7F 135971387 IC50 = 0.94 nM T12499 CKPA94 135971389 IC50 = 4.8 nM T12499 C3H9ZQ 135971390 IC50 = 2.3 nM T12499 CFT9R7 135971391 IC50 = 0.3 nM T12499 CSO65Z 135971392 IC50 = 1.2 nM T12499 CDS3V4 135971394 IC50 = 0.51 nM T12499 C4X0AQ 135971395 IC50 = 1.5 nM T12499 C45RKA 135971396 IC50 > 100 nM T12499 C36UAJ 135971397 IC50 = 1.5 nM T12499 CR5B1S 135971404 IC50 = 1 nM T12499 C0XP6W 135971405 IC50 = 3.9 nM T12499 C05MXR 135971406 IC50 = 8.2 nM T12499 CNT07W 135971407 IC50 = 0.77 nM T12499 CYZT63 135971410 IC50 = 0.55 nM T12499 C8RV2Z 135971411 IC50 = 0.41 nM T12499 C5HTQ7 135971412 IC50 = 1 nM T12499 CK5Y8N 135971414 IC50 = 0.75 nM T12499 CAKJ23 135971415 IC50 = 1.2 nM T12499 CQ8ZL5 135971416 IC50 = 5.4 nM T12499 CU2V3A 135971417 IC50 = 2.8 nM T12499 CMW4A0 135971418 IC50 = 10 nM T12499 CT8FK6 135971419 IC50 = 0.56 nM T12499 CG2YB1 135971420 IC50 = 1.1 nM T12499 C2K8XA 135971421 IC50 = 0.44 nM T12499 C4GWD2 135971422 IC50 = 3.9 nM T12499 C34CFS 135971423 IC50 = 0.8 nM T12499 C8BJM6 135971424 IC50 = 1 nM T12499 CQ1V2X 135971425 IC50 = 2 nM T12499 CSGD27 135972425 IC50 = 2400 nM T12499 CHA4N2 136013680 IC50 > 10 nM T12499 CP5SD0 136016241 IC50 = 1101.3 nM T12499 C5XIE8 136026041 IC50 = 18000 nM T12499 CIVJ39 136056094 IC50 = 144000 nM T12499 CVIC49 136069671 IC50 = 4800 nM T12499 C48DLS 136123445 IC50 > 1500 nM T12499 CD48LY 136185992 IC50 = 3.75 ug.mL-1 T12499 CPE2B1 136185998 IC50 > 20 ug.mL-1 T12499 CR9XE0 136185999 IC50 = 5 ug.mL-1 T12499 C1I8LC 136186000 IC50 = 5 ug.mL-1 T12499 C40HWO 136186001 IC50 > 20 ug.mL-1 T12499 CK5VW8 136186003 IC50 > 10 ug.mL-1 T12499 C7V1YL 136186004 IC50 > 10 ug.mL-1 T12499 CGP04W 136186009 IC50 = 20 ug.mL-1 T12499 CS5QE7 136186010 IC50 > 20 ug.mL-1 T12499 C1YUD0 136219394 IC50 > 10 nM T12499 CIU8W3 136254389 IC50 > 10 nM T12499 CXC69T 137321158 IC50 = 43 nM T12499 C90FJW 137365215 IC50 = 22 nM T12499 C7ZYL2 137365217 IC50 = 12130 nM T12499 CRKO38 137365218 IC50 = 106 nM T12499 C6K5WV 137365221 IC50 = 1860 nM T12499 C07TXV 137365226 IC50 = 39 nM T12499 CB7N3X 137365228 IC50 = 11600 nM T12499 CMX1A3 137365229 IC50 = 33.5 nM T12499 C42HOT 137365231 IC50 = 54 nM T12499 C1QZH5 137365233 IC50 = 3170 nM T12499 C1OQ7V 137365243 IC50 = 6.5 nM T12499 C5CZ2A 137365245 IC50 = 6 nM T12499 CZOD53 137633880 IC50 = 74 nM T12499 CI1E8V 137634241 IC50 = 699 nM T12499 C7BJY5 137636807 IC50 = 21 nM T12499 CO89DX 137649100 IC50 = 7 nM T12499 CINE03 137652514 IC50 = 100 nM T12499 C28QUP 137652864 IC50 = 194.7 nM T12499 CN0X5D 138454787 IC50 = 860 nM T12499 CLJH31 139209093 IC50 = 42 nM T12499 CI1D9F 139600335 IC50 = 27 nM T12499 CVI30A 139600340 IC50 = 260 nM T12499 C9ZYG8 141366083 IC50 = 910 nM T12499 C6RT5B 142749651 IC50 > 100000 nM T12499 CON17J 142749653 IC50 = 10300 nM T12499 CZ2K6B 142749654 IC50 = 58400 nM T12499 CX2Q5T 142749655 IC50 = 5480 nM T12499 CITW53 142749657 IC50 = 7970 nM T12499 C0TYX5 142749658 IC50 > 100000 nM T12499 CV9WM8 142749660 IC50 > 100000 nM T12499 CF5X8A 142749661 IC50 = 41400 nM T12499 CD1EC9 142749662 IC50 = 17450 nM T12499 CSC02Q 142749664 IC50 > 100000 nM T12499 CNU4M3 145704714 IC50 = 31600 nM T12499 C82RKW 145756290 IC50 = 62 nM T12499 CLU0G7 145756294 IC50 = 225 nM T12499 C6VB3O 145925651 IC50 >= 5000 nM T12499 C9N2TO 145950233 IC50 = 71150 nM T12499 CPZR56 145950296 IC50 = 110 nM T12499 CXQT26 145950509 IC50 = 312 nM T12499 CZ8JC7 145952422 IC50 = 510 nM T12499 C57XVG 145954817 IC50 = 22150 nM T12499 C7AIW6 145957749 IC50 = 130 nM T12499 CDA08X 145957845 IC50 = 502 nM T12499 C9NBS5 145959808 IC50 > 100000 nM T12499 CDNC31 145967951 IC50 < 1 nM T12499 CLUS34 145971460 IC50 = 3300 nM T12499 CF27EG 155511610 IC50 = 1183 nM T12499 C0ZAN6 155512322 IC50 = 250 nM T12499 C0AN1O 155512752 IC50 = 1497 nM T12499 C8TL1A 155513050 IC50 = 26000 nM T12499 C2MD1Q 155513187 IC50 > 10000 nM T12499 CI23DH 155516489 IC50 = 74 nM T12499 CEDI24 155516854 IC50 = 300 nM T12499 C3NA2I 155519537 IC50 = 31 nM T12499 C70NHV 155523393 IC50 > 31000 nM T12499 CS69CA 155532132 IC50 = 40.9 nM T12499 C3LC9I 155536820 IC50 = 1000 nM T12499 C2CG1A 155537016 IC50 > 10000 nM T12499 CKOC12 155537703 IC50 = 10000 nM T12499 CB6AN2 155537880 IC50 = 3980 nM T12499 C3V4LG 155538413 IC50 = 515 nM T12499 CGDJ81 155539793 IC50 = 3100 nM T12499 CDW9G6 155541623 IC50 = 31000 nM T12499 CM8E5L 155548006 IC50 = 3160 nM T12499 CLJ80U 155548662 IC50 = 110 nM T12499 CGTR28 155552797 IC50 = 230 nM T12499 CCV06Q 155554126 IC50 = 120 nM T12499 CZQM57 155554194 IC50 = 3156 nM T12499 CJL3D2 155555429 IC50 = 7940 nM T12499 C3DQI8 155557074 IC50 = 24000 nM T12499 CTR18O 155557674 IC50 = 10000 nM T12499 CVS68Y 155558083 IC50 > 50000 nM T12499 CWD8X0 155558928 IC50 > 31000 nM T12499 CV7H5S 155559048 IC50 = 1000 nM T12499 CT8VX1 155562023 IC50 = 26 nM T12499 CY42EB 155566265 IC50 > 31000 nM T12499 CR6EL3 155568078 IC50 = 34000 nM T12499 C12HQW 155568509 IC50 = 43000 nM T12499 D00DNY 3213 IC50 = 18500 nM T12499 D00ERW 44444843 Ki > 2701 nM T12499 D00HVA 11624601 Ki > 2700 nM T12499 D00RIX 5280443 IC50 = 4 ug.mL-1 T12499 D01IZN 44312289 IC50 = 50000 nM T12499 D01KKU 5281894 IC50 = 80 ug.mL-1 T12499 D01NTW 5328768 IC50 = 7000 nM T12499 D01UYI 5281607 IC50 = 5 ug.mL-1 T12499 D02BUW 2061 IC50 = 3000 nM T12499 D02NNT 53232451 IC50 = 215 nM T12499 D02SRA 44312288 IC50 > 800000 nM T12499 D03AER 9549185 IC50 = 20 nM T12499 D03DZO 11715767 IC50 > 10000 nM T12499 D03NPX 447077 IC50 < 5 nM T12499 D04PEI 11467730 IC50 = 2400 nM T12499 D05FXD 44478401 IC50 = 1.3 nM T12499 D05PTT 5281792 IC50 = 24000 nM T12499 D06HVH 54613583 IC50 > 10000 nM T12499 D06WGX 9549184 IC50 = 147 nM T12499 D07ADX 54764565 IC50 = 333 nM T12499 D07AIB 712152 IC50 < 8 nM T12499 D07ERV 44312580 IC50 = 11000 nM T12499 D07IHM 9823787 IC50 > 10000 nM T12499 D07OXC 11650194 IC50 = 8 nM T12499 D08HFG 24809764 IC50 > 10000 nM T12499 D08LYB 5166 IC50 = 18 nM T12499 D08RZB 11153014 IC50 = 1 nM T12499 D08WOG 9948853 IC50 = 1000 nM T12499 D09DVB 44312287 IC50 = 260000 nM T12499 D09HVH 135566652 IC50 > 10 nM T12499 D09HXU 16086113 IC50 = 94 nM T12499 D09QBA 23378546 IC50 = 6400 nM T12499 D09RYV 9911652 IC50 > 100000000 nM T12499 D09ZNV 447682 IC50 = 11000 nM T12499 D0A2LX 44312363 IC50 = 11000 nM T12499 D0B4PI 44312309 IC50 = 470000 nM T12499 D0B8DE 135469328 IC50 > 10000 nM T12499 D0BS6R 9549183 IC50 = 37 nM T12499 D0D5EW 5311104 IC50 < 5 nM T12499 D0D5KZ 11540659 IC50 = 5 nM T12499 D0D9TU 3894 IC50 = 8000 nM T12499 D0E7VO 59627005 IC50 < 100 nM T12499 D0FH3M 18770833 IC50 > 100000 nM T12499 D0GW4Q 5330524 IC50 < 5 nM T12499 D0H1OK 11562302 Ki = 29.4 nM T12499 D0IR6U 5494425 IC50 > 8000 nM T12499 D0IZ8M 56675928 IC50 = 180 nM T12499 D0M4SY 135440466 IC50 = 341 nM T12499 D0ME9B 46868971 IC50 = 510 nM T12499 D0MF5Y 5281614 IC50 = 4 ug.mL-1 T12499 D0N4LR 53469448 IC50 = 1250 nM T12499 D0O0VZ 667639 IC50 = 20 ug.mL-1 T12499 D0O6OH 71553154 IC50 = 220 nM T12499 D0OH3J 5330526 IC50 < 5 nM T12499 D0OZ2S 11785878 IC50 = 1600 nM T12499 D0P0WT 3139 IC50 > 10000 nM T12499 D0P3JW 447700 IC50 < 5 nM T12499 D0Q2UZ 44312307 IC50 = 260000 nM T12499 D0Q3EW 9549303 IC50 = 131 nM T12499 D0Q3NG 11715520 Ki > 2700 nM T12499 D0QN6U 9806182 IC50 > 10000 nM T12499 D0R2WK 16038120 EC50 > 1000 nM T12499 D0S1KJ 5328733 IC50 < 5 nM T12499 D0S7IE 11658882 Ki > 2700 nM T12499 D0SY6C 5282073 IC50 = 200 ug.mL-1 T12499 D0T8NU 16757525 IC50 > 4000 nM T12499 D0T9FQ 10061448 IC50 > 10000 nM T12499 D0V2LK 10244983 IC50 > 2000000 nM T12499 D0W7LW 44312308 IC50 = 220000 nM T12499 D0Y0BK 11524144 IC50 = 16 nM T12499 D0Y1SR 11844351 IC50 = 2 nM T12499 D0Y4BL 11676971 IC50 = 88 nM T12499 D0Y7HG 5281616 IC50 = 80 ug.mL-1 T12499 D0YZ7H 9797370 IC50 = 100 nM T12499 D0Z4HV 10354294 IC50 > 10000 nM T12499 D0Z7GH 5330525 IC50 < 5 nM T12499 D0Z7TM 22273644 IC50 > 2000 nM T25362 D00SUC 74766595 IC50 = 2300 nM T25362 CI03VK 934 IC50 = 25000 nM T25362 CEQ4V8 2723716 IC50 > 100000 nM T25362 CCYF63 9942424 IC50 = 1258.93 nM T25362 CF47JU 25138011 IC50 = 1100 nM T25362 C68RKH 76310231 IC50 = 31000 nM T25362 CO1EN3 76317452 IC50 = 140 nM T25362 CT5FZ8 76321184 IC50 = 12000 nM T25362 C6XRT0 76321186 IC50 = 37000 nM T25362 CKB5O9 76328366 IC50 = 9100 nM T25362 CUNK03 76335652 IC50 = 9700 nM T25362 CX23ZP 78426670 IC50 > 2500 nM T25362 CKXW73 78427224 IC50 > 2500 nM T25362 CIG3E9 83672127 IC50 = 43000 nM T25362 C2NA5I 91801131 IC50 = 19952.62 nM T25362 CP3DK0 96607511 IC50 = 57 nM T25362 C10RDJ 101882871 IC50 > 100000 nM T25362 C6YT2Q 118598059 IC50 > 4000 nM T25362 C5IZD1 122181577 IC50 > 100000 nM T25362 CRM93S 122181583 IC50 > 100000 nM T25362 CU57QX 122181584 IC50 > 100000 nM T25362 C9QVZ5 122181587 IC50 > 100000 nM T25362 CJQ91K 122181588 IC50 > 100000 nM T25362 C75JVN 122191451 IC50 = 25118.86 nM T25362 C3YX7W 122191453 IC50 = 7943.28 nM T25362 C3IBR8 122191455 IC50 = 7943.28 nM T25362 C59KNQ 122191457 IC50 = 12589.25 nM T25362 CM5X8J 122191459 IC50 = 3162.28 nM T25362 C7ASR0 122191460 IC50 = 10000 nM T25362 CRI6J4 122191461 IC50 = 19952.62 nM T25362 CAS4H6 122191462 IC50 = 50118.72 nM T25362 C9J6LX 122191463 IC50 > 100000 nM T25362 C75NJO 122191464 IC50 > 100000 nM T25362 C50VYK 122191465 IC50 = 31622.78 nM T25362 CSKY20 122191466 IC50 > 100000 nM T25362 CS3L8H 122191467 IC50 = 50118.72 nM T25362 CZ2NV1 122191468 IC50 > 100000 nM T25362 CYTW93 122191469 IC50 > 100000 nM T25362 CZV45H 122191470 IC50 = 31622.78 nM T25362 CF6I2N 122191471 IC50 = 100000 nM T25362 CZU02B 122191472 IC50 > 100000 nM T25362 CE27AS 122191473 IC50 > 100000 nM T25362 CAJ28B 122191475 IC50 = 63095.73 nM T25362 C36PDK 122191476 IC50 = 100000 nM T25362 CQ04FW 122191477 IC50 = 39810.72 nM T25362 C12OHA 122191478 IC50 = 63095.73 nM T25362 CL2K0J 122191479 IC50 = 31622.78 nM T25362 CT6HG3 122191480 IC50 = 50118.72 nM T25362 CK7LD6 122191481 IC50 = 25118.86 nM T25362 CMJ72N 122191482 IC50 = 50118.72 nM T25362 C6H2YQ 122383780 IC50 = 191000 nM T25362 CT2UZ4 125377518 IC50 > 100000 nM T25362 CT4O5U 135567037 IC50 = 11000 nM T25362 CC4H1N 135567038 IC50 = 5700 nM T25362 CQBH95 135567040 IC50 = 33000 nM T25362 CP6IH9 135567041 IC50 = 2300 nM T25362 C8HMG2 135567042 IC50 = 9000 nM T25362 CIW61V 135567106 IC50 = 26200 nM T25362 CL9ZD4 135567108 IC50 = 13900 nM T25362 C1VAI3 135567112 IC50 = 4800 nM T25362 C8LFY7 135567115 IC50 = 6100 nM T25362 C34LUV 137175094 IC50 = 5300 nM T25362 C93YUK 137175210 IC50 = 8300 nM T25362 CYG29R 138393334 IC50 = 2020 nM T25362 CNG82D 138393336 IC50 = 5780 nM T25362 CARJ34 138753212 IC50 = 6130 nM T25362 C4M1EO 155519111 IC50 = 6420 nM T25362 CP8K5E 155540290 IC50 = 5680 nM T25362 CFR06L 155551969 IC50 = 50000 nM T25362 C3SQ4A 155569285 IC50 = 1850 nM T25362 D07IOY 10365 IC50 = 3300 nM T25362 D08IZY 3080614 IC50 = 1995.26 nM T25362 D0S3DD 56963315 IC50 = 39810.72 nM T25362 D0X5US 459617 IC50 = 158.49 nM T16902 D0U2BH 65064 IC50 = 60000 nM T16902 D05HSW 3218 IC50 = 7200 nM T16902 C9XI4U 5703 IC50 = 6100 nM T16902 CL80QG 11820 IC50 = 70000 nM T16902 CHU6D4 343829 IC50 = 221000 nM T16902 C6BCK4 393160 IC50 = 2990 nM T16902 CH6RY3 393161 IC50 = 4430 nM T16902 CSP97B 393162 IC50 = 860 nM T16902 C3Q9OD 393163 IC50 = 4100 nM T16902 C1KX0Y 393164 IC50 = 11800 nM T16902 CT5J0P 393165 IC50 = 12900 nM T16902 CXCB27 393166 IC50 = 5300 nM T16902 COJA52 393167 IC50 = 5710 nM T16902 C2JB3F 393168 IC50 = 1830 nM T16902 CWD08M 393169 IC50 = 15900 nM T16902 CM1L3Q 394797 IC50 = 2720 nM T16902 CCHK53 394798 IC50 = 6510 nM T16902 CHR5Q8 395862 IC50 = 6640 nM T16902 CK69TC 462934 IC50 = 67000 nM T16902 CTIN45 463831 IC50 = 13600 nM T16902 CN7WA6 615185 IC50 = 5400 nM T16902 CEW57U 703058 IC50 = 7660 nM T16902 CO8HA9 832572 IC50 = 12000 nM T16902 C6CQG0 1519964 IC50 = 3690 nM T16902 CJWR09 1561807 IC50 = 67200 nM T16902 CS05BM 1600566 IC50 = 97700 nM T16902 C8E9HY 2221149 IC50 = 34700 nM T16902 C4T8OV 2325816 IC50 = 6190 nM T16902 C1YZ8I 2327942 IC50 = 5770 nM T16902 CS62ZV 2327945 IC50 = 5820 nM T16902 CTVG84 2328663 IC50 = 6010 nM T16902 CNM3K2 2328664 IC50 = 4550 nM T16902 COTE61 2408437 IC50 = 13600 nM T16902 C1LNM0 2467794 IC50 = 6950 nM T16902 CZE13I 2816786 IC50 = 9300 nM T16902 CRIH61 2829592 IC50 = 145900 nM T16902 C5F2BD 2854538 IC50 > 100000 nM T16902 C28JDY 3581192 IC50 = 5000 nM T16902 C2M0BI 5271649 IC50 = 22960 nM T16902 CJ32NW 5276854 IC50 = 1600 nM T16902 C2D4HQ 5337613 IC50 = 5100 nM T16902 C13OPQ 5352088 IC50 = 5000 nM T16902 CK4GM7 7574135 IC50 = 3800 nM T16902 C2FM4R 9875131 IC50 = 1000000 nM T16902 CH41UK 9992116 IC50 = 720 nM T16902 CP96LW 10148995 IC50 > 10000 nM T16902 CY67TD 10197845 IC50 = 3000 nM T16902 CDA2X7 10355152 IC50 = 5030 nM T16902 CUD8X4 10355367 IC50 = 3530 nM T16902 CQMG50 10631053 IC50 = 19952.62 nM T16902 C2QTW8 11052198 IC50 = 28000 nM T16902 CA6X8S 11184436 IC50 = 2200 nM T16902 C61TAS 11230373 IC50 = 203600 nM T16902 C2QXV8 11252989 IC50 = 5400 nM T16902 CR39BD 11253617 IC50 = 5900 nM T16902 C2LGY7 11277137 IC50 = 215100 nM T16902 CC9N1I 11288052 IC50 = 10800 nM T16902 CR0ZW2 11345613 IC50 = 180000 nM T16902 C2NM3S 11357323 IC50 = 34900 nM T16902 C9SOZ5 11379279 IC50 = 125600 nM T16902 C61VWH 11380016 IC50 = 102700 nM T16902 CTL4F6 11390927 IC50 = 77800 nM T16902 CCW1Q4 11402704 IC50 = 7200 nM T16902 C9SLU8 11436521 IC50 = 1600 nM T16902 C0WTI5 12889060 IC50 = 2400 nM T16902 C8XM5J 13017443 IC50 > 10000 nM T16902 CK2NM8 13017478 IC50 > 10000 nM T16902 C7U9KW 13099766 IC50 = 17450 nM T16902 CKF7Z1 13169715 IC50 = 12589.25 nM T16902 C29QHR 13374635 IC50 = 7100 nM T16902 C5S2UI 13554995 IC50 = 4630 nM T16902 C1JO9C 15294640 IC50 > 200000 nM T16902 C1DM9I 18783165 IC50 > 500000 nM T16902 C1XN4F 19425176 IC50 > 10000 nM T16902 CQ14MA 19425177 IC50 = 2500 nM T16902 C4K8PQ 19876167 IC50 = 19800 nM T16902 CBS63Q 21879398 IC50 > 10000 nM T16902 CEOI61 22514828 IC50 = 15100 nM T16902 CPQ68C 33287028 IC50 = 15848.93 nM T16902 C89IXD 33323919 IC50 = 6309.57 nM T16902 C46RLS 42609873 IC50 = 1500 nM T16902 CBJS60 42609916 IC50 = 1800 nM T16902 C31WGD 42609917 IC50 = 5600 nM T16902 CS0D7W 42609918 IC50 = 4900 nM T16902 CNR26A 42609919 IC50 > 10000 nM T16902 C8KC5T 44564008 IC50 > 200000 nM T16902 C6Q7IJ 44564009 IC50 = 19000 nM T16902 C4MOV8 44564010 IC50 = 58000 nM T16902 C8ZBL0 44564011 IC50 > 200000 nM T16902 CC9AP5 44564012 IC50 = 32000 nM T16902 CSN6W0 44564013 IC50 = 102000 nM T16902 CG39PD 44564014 IC50 = 42700 nM T16902 C3KD1U 44564054 IC50 > 200000 nM T16902 CZ1WM3 44564055 IC50 = 3100 nM T16902 CH02PI 44564426 IC50 = 2900 nM T16902 CDV70K 44564427 IC50 = 2900 nM T16902 CN60YA 44564428 IC50 = 2800 nM T16902 CU6I4V 44564429 IC50 = 3200 nM T16902 C2NZU6 44564430 IC50 = 2000 nM T16902 CIA7Q6 44564431 IC50 = 2500 nM T16902 CNKG68 44564432 IC50 = 2600 nM T16902 C3Z9BQ 44564469 IC50 > 10000 nM T16902 CO3UF4 44564514 IC50 = 7500 nM T16902 CL40BF 44564515 IC50 = 109000 nM T16902 CRK2E6 44564516 IC50 = 6500 nM T16902 CT39LN 44564517 IC50 = 162000 nM T16902 C52BJH 44571034 IC50 = 108300 nM T16902 C52ONY 44612934 IC50 > 10000 nM T16902 CFC40W 44612935 IC50 > 10000 nM T16902 C60CBK 44612936 IC50 > 10000 nM T16902 CQZ14C 44612937 IC50 > 10000 nM T16902 CRZ81U 44612938 IC50 > 10000 nM T16902 CSB75V 44612939 IC50 > 10000 nM T16902 CNQL69 44613061 IC50 > 10000 nM T16902 C4VQ2K 44613062 IC50 > 10000 nM T16902 C90VFZ 44613063 IC50 > 10000 nM T16902 C8JL5A 44613064 IC50 > 10000 nM T16902 CX39TE 45256553 IC50 = 11800 nM T16902 CJB6E8 45482638 IC50 = 2600 nM T16902 CYL3P6 45494068 IC50 = 9410 nM T16902 C8K7NG 45882522 IC50 = 6309.57 nM T16902 CC7SL5 46927927 IC50 = 662000 nM T16902 CA80ZD 49653721 IC50 = 41800 nM T16902 C4C0GT 49654128 IC50 = 10700 nM T16902 CG3PR6 52912222 IC50 > 7943.28 nM T16902 C4XCJ0 53257845 IC50 = 25500 nM T16902 C3LX0K 53315396 IC50 = 27900 nM T16902 CQK43N 56662996 IC50 = 86300 nM T16902 C3QZ4C 56666477 IC50 = 4570 nM T16902 C94ZFM 56666478 IC50 = 5900 nM T16902 CBOE48 56669892 IC50 = 6940 nM T16902 CFM97A 56676691 IC50 = 4800 nM T16902 CZH49U 56683381 IC50 = 101000 nM T16902 C2WB3X 56683382 IC50 = 22200 nM T16902 CIPN50 71760902 IC50 > 1000 nM T16902 CO2A1X 71812233 IC50 = 900 nM T16902 CBX37Z 72201043 IC50 = 35000 nM T16902 CX7LT6 76320951 IC50 = 1700 nM T16902 CA7P3H 76320952 IC50 = 2800 nM T16902 CS3W6O 90667751 IC50 = 28800 nM T16902 CZBD29 90667752 IC50 = 78200 nM T16902 CF4W8Q 90667754 IC50 = 63700 nM T16902 C2B4NA 90667755 IC50 = 41800 nM T16902 C9WB3G 95828281 IC50 > 20000 nM T16902 CIX5V3 113222223 IC50 = 15848.93 nM T16902 CX9J1Q 113231872 IC50 = 7943.28 nM T16902 CB5O8P 115579930 IC50 = 31622.78 nM T16902 CVA75B 115611029 IC50 = 1258.93 nM T16902 C21EWV 115611032 IC50 = 15848.93 nM T16902 CM6CX7 118928793 IC50 = 19 nM T16902 CKF18M 118928795 IC50 = 19 nM T16902 CDH8M4 121373418 IC50 > 20000 nM T16902 C47QXT 121376807 IC50 > 20000 nM T16902 C38ERO 121472643 IC50 = 6309.57 nM T16902 C1OIJ9 121476448 IC50 = 501.19 nM T16902 C07JLO 121476460 IC50 = 13 nM T16902 CD3AJ2 126797002 IC50 = 4200 nM T16902 CG9S7A 126961735 Ki = 1.259 nM T16902 CV4D8T 127030247 IC50 = 5000 nM T16902 C0VEM9 131698638 IC50 = 36 nM T16902 CA0P5D 131953422 IC50 = 300 nM T16902 CK1O5N 132153759 IC50 = 70 nM T16902 CGDN94 132275066 IC50 > 20000 nM T16902 CHL8K4 132941768 IC50 = 10000 nM T16902 CU2F1G 135566900 Ki < 3340 nM T16902 CW94QO 136226511 Ki < 3340 nM T16902 C5I9TL 137634095 IC50 = 10000 nM T16902 C2IHE8 137635251 IC50 = 25118.86 nM T16902 CQT3A9 137636309 IC50 > 100000 nM T16902 CULX38 137646779 IC50 = 79.43 nM T16902 CN7V5T 137648161 IC50 = 39810.72 nM T16902 CV7G1I 137654127 IC50 = 6309.57 nM T16902 CSI4V8 137661043 IC50 = 1000 nM T16902 C6C7ZM 138105961 IC50 = 7 nM T16902 C8ZQ2U 141736359 IC50 > 20000 nM T16902 C5VNM4 141736367 IC50 > 20000 nM T16902 C3YGJ5 145948689 IC50 = 300 nM T16902 C96NCH 145950955 IC50 > 20000 nM T16902 C3ZV1O 145952497 IC50 > 20000 nM T16902 CTE74G 145954441 IC50 > 20000 nM T16902 C5WX1Y 145954899 IC50 = 200000 nM T16902 C3D8LO 145955588 IC50 = 160000 nM T16902 CN5YO3 145957310 IC50 > 20000 nM T16902 C8JI5E 145957556 IC50 > 500000 nM T16902 C7C5WL 145958595 IC50 > 20000 nM T16902 C8Z9OM 146205579 IC50 > 20000 nM T16902 CL2SN9 154641364 IC50 = 41 nM T16902 CAN03S 155510571 IC50 = 10 nM T16902 C1E8WH 155513683 IC50 = 17 nM T16902 CAF7V6 155520495 IC50 = 14 nM T16902 C70MDA 155522763 IC50 = 25 nM T16902 C5C6SH 155523656 IC50 = 32 nM T16902 CP4UN7 155523768 IC50 = 35 nM T16902 C98TUC 155526102 IC50 = 47 nM T16902 C5BL1C 155535313 IC50 = 125 nM T16902 C95OQP 155536635 IC50 > 50000 nM T16902 C73HGS 155544332 IC50 = 30 nM T16902 CMON16 155545209 IC50 = 73 nM T16902 C07OQG 155553182 IC50 = 22 nM T16902 C4Z5KF 155562459 IC50 = 30 nM T16902 D03XXT 72201027 IC50 > 20000 nM T16902 D07MTM 403 IC50 > 500000 nM T16902 D07UCF 615184 IC50 = 4200 nM T16902 D08XXD 17815 IC50 = 3600 nM T16902 D09HBR 135566899 Ki = 5520 nM T16902 D0E6JS 167551 IC50 = 5000 nM T16902 D0P0IE 10205 IC50 = 50000 nM T16902 D0W3NA 87642 IC50 = 41910 nM T95736 D0E3TC 44259 IC50 = 2300 nM T95736 D0Z5DM 5081913 IC50 > 100000 nM T95736 CC1PI7 90469 IC50 > 100000 nM T95736 CZ34CV 349435 IC50 = 51000 nM T95736 CFBU18 400433 IC50 = 41000 nM T95736 CYN49L 575802 IC50 = 61100 nM T95736 CU73ST 599501 IC50 > 100000 nM T95736 CL3X6Q 1508801 IC50 > 100000 nM T95736 CMC16L 2782960 IC50 > 100000 nM T95736 CS6VL5 6539018 IC50 > 80000 nM T95736 CK4W6A 8891610 IC50 > 50000 nM T95736 CGRY94 10777396 IC50 > 100000 nM T95736 CACS26 11561968 Ki > 10000 nM T95736 CU0E8O 11690457 Ki > 10000 nM T95736 CB0AP2 11705863 Ki > 10000 nM T95736 CG7X9F 12330558 IC50 > 100000 nM T95736 C78ADF 16751210 IC50 = 1800 nM T95736 C6OY4H 16751569 IC50 = 150 nM T95736 CF0H3L 17229016 IC50 > 100000 nM T95736 CJM4C7 24219848 IC50 > 100000 nM T95736 CC9V2Y 24882562 IC50 = 480 nM T95736 C56VHY 25219675 IC50 > 100000 nM T95736 C90BUF 43157763 IC50 > 100000 nM T95736 CJ7D5T 43157843 IC50 > 100000 nM T95736 C6Z2SA 43560957 IC50 > 100000 nM T95736 CT8P3E 46911431 IC50 = 90000 nM T95736 CVYL83 54768752 IC50 = 24000 nM T95736 CLAQ16 57525824 IC50 = 4.2 nM T95736 C12VDY 58221397 IC50 = 100 nM T95736 C96JRL 58221549 IC50 = 41 nM T95736 CV7E3R 58221661 IC50 = 190 nM T95736 CJS4Y6 58221760 IC50 = 550 nM T95736 C1MR8Q 60097495 IC50 > 10000 nM T95736 CL36SQ 61992242 IC50 > 100000 nM T95736 CNP85L 61992815 IC50 > 100000 nM T95736 CU28AB 62900145 IC50 > 100000 nM T95736 C5L0SQ 68388404 IC50 = 76 nM T95736 CXV8G4 71560537 IC50 = 16000 nM T95736 C57CZF 71560538 IC50 = 4000 nM T95736 CVNT74 71560539 IC50 = 310 nM T95736 CEHS93 71560540 IC50 = 300 nM T95736 C53UOG 71560541 IC50 = 89 nM T95736 CPN3M1 71560660 IC50 = 42000 nM T95736 CLY84V 71560661 IC50 > 80000 nM T95736 CGVE29 71560662 IC50 > 80000 nM T95736 CG9KZ7 71560663 IC50 = 110 nM T95736 C0E9CU 71560664 IC50 = 30000 nM T95736 CB56LM 71560665 IC50 = 70 nM T95736 CW57HX 71560666 IC50 = 2600 nM T95736 C3A1WL 71560667 IC50 = 1200 nM T95736 CG3H8S 71560783 IC50 = 21000 nM T95736 CVBN17 71560784 IC50 = 30000 nM T95736 C7PTA0 71560785 IC50 = 30000 nM T95736 CQ25SH 71580632 IC50 = 63 nM T95736 C1GQE5 71714612 Ki = 41 nM T95736 CPW42O 71714613 Ki = 35.5 nM T95736 C2ZBV7 71714614 Ki = 201 nM T95736 C4GF6B 71714694 Ki = 310 nM T95736 CV50MB 71714695 Ki = 28 nM T95736 CP2LG8 71714710 Ki = 36 nM T95736 CF2U3Z 71714711 Ki = 0.3 nM T95736 C54OCN 71714717 Ki = 101 nM T95736 C3S8AL 71714722 Ki = 20.2 nM T95736 CN31CF 71714729 Ki = 7.5 nM T95736 CUQ0T6 71714731 Ki = 40 nM T95736 CQ8KM1 71715050 Ki = 7 nM T95736 CJ9YX0 71715393 Ki = 3.2 nM T95736 C63JAT 71715396 Ki = 1.5 nM T95736 CK0MZ9 71717636 IC50 = 15000 nM T95736 CE8V7C 71720042 IC50 = 24000 nM T95736 C1XJ2W 71720688 IC50 = 63 nM T95736 CB04OD 82482456 IC50 > 100000 nM T95736 C0ZXY3 86693116 Ki > 250 nM T95736 C0ZOK6 86693155 Ki = 14 nM T95736 CBJ1P2 86693157 Ki = 10 nM T95736 CMY4D7 86693162 Ki = 3.1 nM T95736 CT23XM 86693188 Ki = 0.47 nM T95736 C1H0AG 86693196 Ki = 986 nM T95736 CK8UX7 86693200 Ki = 3 nM T95736 CSKY40 86693215 Ki = 8.7 nM T95736 CAX6M8 86693217 Ki = 4282 nM T95736 CPFS76 86693462 Ki = 9.9 nM T95736 CU78DC 86693540 Ki = 1.7 nM T95736 CWLV65 89754409 Ki = 2503 nM T95736 CU7P5O 89754494 Ki = 2.9 nM T95736 CAO58E 89754729 Ki = 1164 nM T95736 CT04ER 89754780 Ki = 0.9 nM T95736 C2ONT4 89754889 Ki = 405 nM T95736 C2FUO8 89754902 Ki = 0.8 nM T95736 CL4QV3 89754913 Ki = 547 nM T95736 CEI14Q 89754914 Ki = 2 nM T95736 CDEW02 89755037 Ki > 1250 nM T95736 CX0G7V 89755117 Ki = 20 nM T95736 C6Z7ID 89759863 Ki = 0.4 nM T95736 CH75AV 89759865 Ki = 0.8 nM T95736 C1H6FV 117901716 Ki = 68 nM T95736 C0BQS1 117901834 Ki = 1.3 nM T95736 CK8LF5 117902000 Ki = 0.23 nM T95736 CEZW47 117902083 Ki = 0.42 nM T95736 C2GNU7 117902249 Ki = 2 nM T95736 CO5TN3 117902279 Ki = 0.59 nM T95736 C1HX2O 117902381 Ki = 0.07 nM T95736 CYO59C 117902575 Ki = 0.07 nM T95736 CP01MU 117911529 Ki = 4.7 nM T95736 CIOG01 117911755 Ki = 0.86 nM T95736 C1TCH6 117911819 Ki = 16 nM T95736 C98YHE 117911843 Ki = 9.4 nM T95736 C58YIP 117912362 Ki = 0.23 nM T95736 C6TND8 117912488 Ki = 0.18 nM T95736 CPAF91 117923520 Ki = 28 nM T95736 CSY13U 117923525 Ki = 0.08 nM T95736 C5E9JC 117923543 Ki = 0.17 nM T95736 C7WB2P 117923580 Ki = 0.27 nM T95736 CXJ98Z 117923582 Ki = 0.13 nM T95736 CL10MC 117923585 Ki = 0.23 nM T95736 C8LZ6Y 117923640 Ki = 0.05 nM T95736 CB57TM 123132912 Ki = 1280 nM T95736 C3UH2V 129202507 IC50 = 45 nM T95736 C0RE4Q 130270547 IC50 = 1.8 nM T95736 C9G1PS 130270628 IC50 = 21.4 nM T95736 C50DYF 130270664 IC50 = 5.5 nM T95736 C2BE5F 130270736 IC50 = 1.8 nM T95736 CJ1F4A 130270771 IC50 = 4.1 nM T95736 CRV6D7 130270775 IC50 = 2.3 nM T95736 CW5KC8 130270952 IC50 = 1.3 nM T95736 CMX40O 130270954 IC50 = 6.6 nM T95736 CUN4V6 130271143 IC50 = 7.4 nM T95736 C1R6WD 130271145 IC50 = 1.2 nM T95736 CS7ME6 130271227 IC50 = 1.3 nM T95736 C6MZL2 134145793 Ki >= 1250 nM T95736 CQDC40 134151887 Ki = 582 nM T95736 CCH37I 134163557 Ki > 1250 nM T95736 C2AN7T 134611886 IC50 = 8400 nM T95736 CSV6O4 134817242 Ki = 0.3 nM T95736 CKOD92 141758865 IC50 = 189.8 nM T95736 CQJ70P 141758871 IC50 = 85.5 nM T95736 CL04BH 141758877 IC50 = 120 nM T95736 C9S2EO 141758879 IC50 = 2290 nM T95736 CK6E5G 141758883 IC50 = 319 nM T95736 CR0UO6 141758884 IC50 > 10000 nM T95736 CGH4R2 141758885 IC50 = 10910 nM T95736 C01BVU 141758886 IC50 > 10000 nM T95736 CS4W5N 141758888 IC50 = 87.3 nM T95736 CI4AL6 141758890 IC50 = 410 nM T95736 C5REB0 141758892 IC50 = 215 nM T95736 CC1V0S 141758895 IC50 = 11700 nM T95736 CU78RH 141758898 IC50 = 290 nM T95736 CV95IH 141758900 IC50 = 85.2 nM T95736 C4LB2Z 141758901 IC50 = 234 nM T95736 CFH3E1 141758902 IC50 = 2484 nM T95736 C4W8YB 141758903 IC50 = 120 nM T95736 CFW67Y 141758907 IC50 = 641 nM T95736 CCJ30F 141758909 IC50 > 10000 nM T95736 C4Z2HP 141758910 IC50 = 25830 nM T95736 C0EIJ7 141758911 IC50 > 10000 nM T95736 C4J3VR 141758912 IC50 = 3837 nM T95736 C79ZXF 141758918 IC50 > 10000 nM T95736 C69HLJ 141758920 IC50 = 475 nM T95736 CEYA72 141758926 IC50 = 25.7 nM T95736 CVFR90 141758928 IC50 = 2030 nM T95736 C3RO7M 141758929 IC50 = 303 nM T95736 CCIU75 141758930 IC50 = 2204 nM T95736 C0JW8Z 141758931 IC50 = 335 nM T95736 CZH9V1 141758932 IC50 = 219 nM T95736 C1RFW5 141758933 IC50 = 1750 nM T95736 C0OSR6 141758938 IC50 = 204 nM T95736 C4V8EF 141758940 IC50 = 26.1 nM T95736 CH3QM6 141758943 IC50 = 1570 nM T95736 C6JYI1 141758946 IC50 = 468 nM T95736 CC3P2D 141758947 IC50 = 748 nM T95736 C7FYT5 141758948 IC50 = 2060 nM T95736 CE93LI 141758949 IC50 = 22.4 nM T95736 CMWV78 141758951 IC50 = 218 nM T95736 CUV3E7 141758953 IC50 = 2481 nM T95736 C80DZI 141758956 IC50 > 10000 nM T95736 CVBT03 141758957 IC50 > 10000 nM T95736 CZB6J5 141758959 IC50 = 216 nM T95736 CV8YQ9 141758960 IC50 = 290 nM T95736 CEG6I9 141758961 IC50 > 10000 nM T95736 CQT4K6 141758963 IC50 = 720 nM T95736 CDR2I6 141758964 IC50 = 1860 nM T95736 CKXA01 141758965 IC50 = 6160 nM T95736 C3FJN2 141758966 IC50 = 1640 nM T95736 C71BDY 141758967 IC50 = 388 nM T95736 CWF92L 141758969 IC50 = 2061 nM T95736 CJDN92 141758978 IC50 = 6380 nM T95736 CT89FP 145952913 IC50 > 100000 nM T95736 CE6T2K 145965917 Ki = 5.9 nM T95736 C91BHP 145971744 IC50 > 100000 nM T95736 CR73ZD 145976166 Ki = 350 nM T95736 CURX24 145976657 IC50 = 0.8 nM T95736 CML8O0 145979124 IC50 > 100000 nM T95736 CQLH68 145979774 IC50 > 100000 nM T95736 C5YR8W 145979893 IC50 > 100000 nM T95736 CGL48D 145980076 IC50 > 100000 nM T95736 C5LK9A 145980083 IC50 > 100000 nM T95736 CCSY15 145980681 IC50 = 58200 nM T95736 CY80PH 145981483 IC50 = 39600 nM T95736 CN3U5W 145981500 IC50 > 100000 nM T95736 CFSQ94 145981688 IC50 > 100000 nM T95736 CI3P2B 145981824 IC50 > 100000 nM T95736 CVRZ23 145984375 IC50 > 100000 nM T95736 CGE7B8 145987124 IC50 > 100000 nM T95736 C86HGI 145987159 IC50 = 41000 nM T95736 CU3J8R 145987461 IC50 > 100000 nM T95736 CRJQ18 145988918 IC50 > 100000 nM T95736 C8QH2W 145989390 IC50 > 100000 nM T95736 CFAK86 145989643 IC50 > 100000 nM T95736 CHWR01 145989760 IC50 > 100000 nM T95736 C3EIA1 145990026 IC50 > 100000 nM T95736 CBZ94U 145990465 IC50 = 3300 nM T95736 C8M5AU 145990524 IC50 > 100000 nM T95736 C4FQ0C 145990918 IC50 > 100000 nM T95736 CN38UG 145990988 IC50 = 2900 nM T95736 CGSZ75 145991182 IC50 = 24300 nM T95736 C2SY4M 145991367 IC50 > 100000 nM T95736 C0CJ9I 145991401 IC50 > 100000 nM T95736 CI60XK 145991710 IC50 > 100000 nM T95736 C17TOS 145991715 IC50 = 27400 nM T95736 C68ZYI 145991820 IC50 > 100000 nM T95736 C3HIB8 145992014 IC50 = 23000 nM T95736 CF28WP 145992122 IC50 > 100000 nM T95736 C85OWM 145992355 IC50 > 100000 nM T95736 CD54KY 145992596 IC50 > 100000 nM T95736 CQI81V 145992947 IC50 > 100000 nM T95736 C3NU7C 145993088 IC50 > 100000 nM T95736 C0CJ9B 145993626 IC50 = 12500 nM T95736 C2GH5C 145993662 IC50 > 100000 nM T95736 CMJ6G4 145993951 IC50 > 100000 nM T95736 CS61OX 147007484 IC50 = 5.9 nM T95736 CXN9Z8 155510685 IC50 = 2230 nM T95736 C7H5XM 155517858 IC50 = 9.1 nM T95736 CJP09I 155520168 Ki = 0.16 nM T95736 CS29GT 155528718 Ki > 1250 nM T95736 C0FAD1 155540387 Ki > 1250 nM T95736 CLA0I9 155552645 Ki = 634 nM T95736 D07MQC 9949093 IC50 > 100000 nM T95736 D0J3LR 11634725 Ki > 5000 nM T95736 D0LE7J 58221375 IC50 = 20 nM T95736 D0P0IE 10205 IC50 > 100000 nM T65721 C43DAY 68635 IC50 = 4600 nM T65721 C5KW4H 72311 IC50 = 7000 nM T65721 CYUH56 363208 IC50 = 31000 nM T65721 CWJ43S 443767 IC50 = 34000 nM T65721 CORM47 1849091 IC50 = 21300 nM T65721 C9N5XB 2026662 IC50 = 8700 nM T65721 CD8BS4 2999946 IC50 = 46100 nM T65721 CYZ0U7 4891910 IC50 = 5300 nM T65721 CAK90T 4893331 IC50 = 27900 nM T65721 CU8LQ0 4893774 IC50 = 24200 nM T65721 CF9QP2 9076354 IC50 = 24100 nM T65721 CT8RA9 9099810 IC50 = 57200 nM T65721 CK7N4D 9880653 IC50 = 2700 nM T65721 CD57RY 24344410 IC50 = 28300 nM T65721 CN3Y9K 25138381 IC50 = 9300 nM T65721 CDU76N 25164618 IC50 = 54000 nM T65721 C4OP0C 25165019 IC50 = 58000 nM T65721 C51DAH 45272995 IC50 = 12200 nM T65721 CP57CD 45483073 IC50 = 13000 nM T65721 CURM73 51031035 IC50 = 1100 nM T65721 C0EQA8 90655048 IC50 = 95000 nM T65721 C1KBS9 135431654 IC50 = 1800 nM T65721 C9PY6U 135959764 IC50 = 37000 nM T23984 CG3PR6 52912222 IC50 > 1.259 nM T23984 CIPN50 71760902 IC50 > 1000 nM T23984 COZ8S1 78319129 IC50 > 1000 nM T23984 CYX7T2 117072549 IC50 = 3410 nM T23984 C87ZPY 118796358 IC50 = 117 nM T23984 CC14FI 118933132 IC50 = 82 nM T23984 C9MQF0 119098887 IC50 = 240 nM T23984 C0QX4D 119098889 IC50 = 108 nM T23984 CGA71L 127048256 IC50 = 3283 nM T23984 CH6T5J 127048257 IC50 = 2976 nM T23984 C60SZQ 127048258 IC50 = 4307 nM T23984 C50BMV 127049279 IC50 = 230 nM T23984 CTF4N2 127051087 IC50 = 188 nM T23984 CLSZ47 127051725 IC50 = 41 nM T23984 CMY93U 127051726 IC50 = 3725 nM T23984 CY8V1A 127051727 IC50 = 1565 nM T23984 CXZT48 127052023 IC50 = 2475 nM T23984 CV4X7R 135566898 Ki = 3540 nM T23984 CU2F1G 135566900 Ki < 1430 nM T23984 CW94QO 136226511 Ki < 1430 nM T23984 CQT3A9 137636309 IC50 > 100000 nM T23984 CQ6XB7 139030526 IC50 = 63095.73 nM T23984 D08LXU 91827372 IC50 = 3300 nM T23984 D09HBR 135566899 Ki = 2720 nM T23984 D0O6XT 91827373 IC50 = 140 nM T17067 C4DQ7P 11222830 IC50 = 3000 nM T17067 C3Z5CV 46830074 IC50 > 200000 nM T17067 D0N6BC 950368 Ki = 100000 nM T17067 D0Y7OI 11563133 Ki = 4000 nM T07663 D05MQK 110635 IC50 = 1.2 nM T07663 D0C9SY 135400189 Ki = 0.7 nM T07663 D0F9GE 3108 IC50 = 574 nM T07663 D0NJ3V 4680 IC50 = 8800 nM T07663 D0Y5JC 9869929 Ki = 5 nM T07663 D0Y9ZE 4197 IC50 = 740 nM T07663 D0Z7ZM 135398744 Ki = 1.6 nM T07663 D03QJL 3671 IC50 = 103000 nM T07663 D05OQG 5318997 IC50 = 5900 nM T07663 D09OCK 135430955 IC50 = 4.2 nM T07663 D0A9IY 135564558 IC50 > 10000 nM T07663 D0L0BX 5318980 IC50 = 2200 nM T07663 D0M9FQ 11465695 IC50 = 0.5012 nM T07663 D0T5PO 5092 IC50 = 720 nM T07663 D05VBJ 71295299 IC50 > 10000 nM T07663 D0WS3T 72706254 IC50 = 260 nM T07663 D00SPK 23665864 IC50 = 3.7 nM T07663 D00YPW 135399235 Ki = 130 nM T07663 D01QUF 9842576 Ki > 100000 nM T07663 D02EMR 151170 IC50 > 10000 nM T07663 D05VLN 55690 IC50 = 58000 nM T07663 D0BK6B 3021729 IC50 > 10000 nM T07663 D0F0CS 5723 IC50 > 10000 nM T07663 D0K2BQ 71356 Ki = 7500 nM T07663 D0N5SC 135536943 IC50 = 1.23 nM T07663 D0W8OH 135529458 IC50 = 80 nM T07663 CVQ0G5 1348 IC50 = 500 nM T07663 C03NGJ 1713 IC50 = 230 nM T07663 CH8J2B 4977 Ki = 600000 nM T07663 CCJ8F0 5353 IC50 = 21000 nM T07663 C3B8VG 5369 IC50 = 1 nM T07663 CAMB41 100554 IC50 = 5500 nM T07663 C9T3FB 105007 IC50 = 1580 nM T07663 CGA17S 127779 Ki = 6500 nM T07663 C1H8NR 155248 IC50 > 50000 nM T07663 CH2P8A 158961 Ki = 600000 nM T07663 CVN23X 158962 Ki = 600000 nM T07663 CL27HC 160179 IC50 = 9300 nM T07663 CYWS98 185848 IC50 > 40000 nM T07663 C78DLE 205964 IC50 = 360 nM T07663 C1B6ZL 662965 IC50 > 50000 nM T07663 C3A4HW 675226 IC50 = 8600 nM T07663 CA56MW 675227 IC50 = 3900 nM T07663 CHAB75 696516 IC50 = 1900 nM T07663 CW2U6N 698956 IC50 = 420 nM T07663 CYBA13 719250 IC50 = 4700 nM T07663 C1HM0K 832282 IC50 = 4300 nM T07663 C9KVI7 832283 IC50 = 22000 nM T07663 CM6Q1D 869895 IC50 = 2400 nM T07663 C6QBR5 874599 IC50 = 540 nM T07663 CR7A3U 930420 IC50 = 1200 nM T07663 CWIA36 987187 IC50 = 5600 nM T07663 CT62PH 987189 IC50 = 3100 nM T07663 CO0Z8N 1002275 IC50 = 1700 nM T07663 CXQ4P8 1183964 IC50 = 860 nM T07663 CZQ09F 1204882 IC50 = 7200 nM T07663 CHP0S3 1204883 IC50 = 570 nM T07663 C0JM2Q 1215407 IC50 = 700 nM T07663 CZ2XI5 1271431 IC50 = 3100 nM T07663 COW58U 1277329 IC50 = 190 nM T07663 C6VF0S 1490272 IC50 = 840 nM T07663 CQ69OY 1490552 IC50 = 1100 nM T07663 CD0G9E 1553819 IC50 = 14000 nM T07663 CYD6E3 1553838 IC50 = 190 nM T07663 CXP17G 1604254 IC50 = 4600 nM T07663 C8JLO0 2243267 IC50 = 370 nM T07663 CTQ23N 2452792 IC50 = 800 nM T07663 CLNU08 2456309 IC50 = 740 nM T07663 CYP23V 2465033 IC50 = 800 nM T07663 CE70KT 2471983 IC50 = 1200 nM T07663 CE4D1W 2789492 IC50 = 5600 nM T07663 CFC30O 2789499 IC50 = 1000 nM T07663 C4LSR7 2886111 IC50 > 10000 nM T07663 C6AT3L 2930929 IC50 = 6300 nM T07663 CD70ZG 3119958 IC50 = 8700 nM T07663 C4MSC9 3120507 IC50 = 3000 nM T07663 CPX4V3 4352680 IC50 = 130620 nM T07663 C5IZS9 4636426 IC50 = 746450 nM T07663 CC3LA4 4672917 IC50 = 8500 nM T07663 C5P0LU 4672918 IC50 = 29300 nM T07663 C3JHM8 4687521 IC50 = 1.2 nM T07663 C0JVX6 4867627 IC50 = 4900 nM T07663 CN0Z3D 4880961 IC50 = 11000 nM T07663 C0C9HP 6610310 IC50 = 19 nM T07663 CAYS61 6918354 IC50 = 4000 nM T07663 CB40PM 6918356 IC50 = 200 nM T07663 CI7K0P 6918667 IC50 = 69800 nM T07663 CP1GO7 6918668 IC50 > 84900 nM T07663 CA05PF 6918674 IC50 = 700 nM T07663 C87WYR 6918795 IC50 > 67300 nM T07663 CRGE51 6918796 IC50 > 101000 nM T07663 CUP4M8 6918797 IC50 > 50700 nM T07663 C0LRO8 6918798 IC50 > 101000 nM T07663 C53ESK 6918799 IC50 > 91000 nM T07663 CU1E0G 6918800 IC50 > 101000 nM T07663 CRU46D 7161211 IC50 = 3250 nM T07663 CQ41MA 8055545 IC50 = 2300 nM T07663 CZF0N3 8055573 IC50 = 2400 nM T07663 CN86QP 8078832 IC50 = 2500 nM T07663 CI15SH 9797222 IC50 = 14000 nM T07663 CNC2F4 9798336 IC50 > 1000000 nM T07663 CFJ62Y 9799389 IC50 > 10000 nM T07663 CZH08Y 9802738 IC50 = 7.2 nM T07663 CDV76T 9803328 Ki = 0.29 nM T07663 CR09LM 9805655 IC50 = 0.3 nM T07663 CB57DJ 9807085 IC50 = 72 nM T07663 CXF0J7 9818343 IC50 = 10 nM T07663 C1CXA5 9818702 IC50 = 5000 nM T07663 CSOX21 9819114 IC50 = 2.8 nM T07663 C1MN3A 9821924 IC50 = 2 nM T07663 C7FY1U 9824408 IC50 = 1.1 nM T07663 C4J2XE 9836643 IC50 > 101000 nM T07663 C4YB1S 9844037 IC50 = 5.3 nM T07663 C5YQB0 9859898 IC50 = 78000 nM T07663 CZGM43 9864862 IC50 = 22000 nM T07663 CEI5P4 9868140 IC50 = 440 nM T07663 C92GMV 9879320 IC50 = 13000 nM T07663 C0Q5VN 9880010 IC50 > 101000 nM T07663 CWD1F6 9880288 IC50 > 101000 nM T07663 C2NK8E 9888568 IC50 = 0.56 nM T07663 C0P8ZH 9892886 Ki = 0.21 nM T07663 CC05QE 9901606 IC50 = 101000 nM T07663 CMBO89 9912467 IC50 = 2000 nM T07663 CBA29H 9922545 IC50 > 101000 nM T07663 CKF4C2 9922691 IC50 = 73200 nM T07663 CY17NM 9922999 IC50 = 8400 nM T07663 C70AMC 9924305 IC50 = 7270 nM T07663 CKI6N2 9924468 IC50 > 88000 nM T07663 C6AZ5F 9924709 IC50 > 101000 nM T07663 C54ICU 9927654 IC50 = 3500 nM T07663 C60BWM 9933503 IC50 = 0.8 nM T07663 CX1UV7 9946954 IC50 = 20160 nM T07663 C7OP5A 9947052 IC50 = 3970 nM T07663 C04HAV 9949594 IC50 = 225 nM T07663 C53AVJ 9951793 IC50 = 2.3 nM T07663 CE8ZD7 9954790 IC50 = 0.93 nM T07663 CH46TF 9954942 Ki = 0.23 nM T07663 C8X7RN 9956576 IC50 = 0.1 nM T07663 C2OYA1 9957043 IC50 = 0.55 nM T07663 CJO0X4 9966737 IC50 = 10940 nM T07663 CFP1Y5 9966830 IC50 > 101000 nM T07663 C9NKY4 9967652 IC50 = 74000 nM T07663 CI6AX1 9968005 IC50 > 101000 nM T07663 C7PCS8 9968050 IC50 = 40350 nM T07663 CFB48Q 9968370 IC50 = 98000 nM T07663 CU73AJ 9968471 IC50 > 101000 nM T07663 C0AP8O 9969020 IC50 = 17880 nM T07663 C9X7PF 9972372 IC50 = 8800 nM T07663 CL6V2I 9973407 IC50 = 770 nM T07663 CCDX84 9973586 IC50 = 0.53 nM T07663 C5AE2I 9973597 IC50 > 200000 nM T07663 CTQ59Y 9975543 IC50 = 3600 nM T07663 CW3S7O 9977675 IC50 > 1000000 nM T07663 C05RPA 9977814 IC50 = 2700 nM T07663 C20XIY 9985391 IC50 = 2200 nM T07663 CHG4K5 9992525 IC50 = 64000 nM T07663 CO87TV 9994528 IC50 = 100 nM T07663 CC86WM 9995163 IC50 = 6800 nM T07663 CB9EY5 9995187 IC50 = 90 nM T07663 CWJ0K5 9995367 IC50 = 210 nM T07663 CZR07N 9995467 IC50 = 930 nM T07663 C3GHJ7 9996490 IC50 = 105 nM T07663 CH70VI 9996675 IC50 = 1100 nM T07663 CE5O4D 9998316 IC50 = 350 nM T07663 CYS20P 10004422 IC50 = 38000 nM T07663 CB41WF 10017397 IC50 = 3000 nM T07663 CKE92N 10017795 IC50 = 3600 nM T07663 CHJ73C 10018556 IC50 = 8700 nM T07663 CI9WK7 10021158 IC50 = 1300 nM T07663 C6MUC5 10024867 IC50 = 2500 nM T07663 C5E4QJ 10030897 Ki = 0.24 nM T07663 C1G5XC 10032458 IC50 = 6500 nM T07663 CE25WO 10039122 IC50 = 4400 nM T07663 CUYW65 10039809 IC50 = 20000 nM T07663 C0SZB8 10039848 IC50 = 36300 nM T07663 CJ1Q7Z 10040540 IC50 = 50 nM T07663 CJ05CZ 10040882 IC50 = 15000 nM T07663 CK5VB0 10041530 IC50 = 14000 nM T07663 C9FD1X 10041853 IC50 = 7500 nM T07663 CT6Y9J 10043209 IC50 > 1000000 nM T07663 CY6FQ4 10053217 IC50 = 3 nM T07663 CD1N4K 10062262 IC50 = 1000 nM T07663 CHCJ86 10065791 IC50 = 810 nM T07663 CC6PO8 10066654 IC50 > 40000 nM T07663 C3MA2L 10067044 IC50 > 1000000 nM T07663 C5FCT6 10070215 IC50 = 0.6 nM T07663 COSV65 10074226 Ki = 0.23 nM T07663 CG39NX 10083598 IC50 = 40000 nM T07663 C5P7AS 10083609 IC50 = 6000 nM T07663 C7YBR0 10083610 IC50 = 33000 nM T07663 CAX67L 10084334 IC50 = 3000 nM T07663 CP6W8T 10086869 IC50 = 18500 nM T07663 CLB5S6 10087203 IC50 = 11000 nM T07663 CNA75V 10087755 IC50 = 1400 nM T07663 CJ16FV 10087963 IC50 > 1000000 nM T07663 CSP05N 10088555 IC50 = 730 nM T07663 CRW6E1 10088941 IC50 > 40000 nM T07663 C09ZNQ 10088960 IC50 = 2.6 nM T07663 C0O6MQ 10089225 IC50 = 2300 nM T07663 C13QUP 10089597 IC50 = 65000 nM T07663 CARY56 10091146 IC50 > 200000 nM T07663 CP8I5O 10093297 IC50 = 9800 nM T07663 CS4QG0 10095269 IC50 = 900 nM T07663 C61QRH 10096810 IC50 = 49000 nM T07663 CN23KJ 10105662 IC50 = 18000 nM T07663 CP3D7N 10108060 IC50 = 6000 nM T07663 C12LED 10109572 IC50 > 101000 nM T07663 CT0A4J 10113055 IC50 = 9 nM T07663 CPWL59 10113972 IC50 = 8 nM T07663 C5GRV3 10117157 IC50 = 56 nM T07663 C2PBD6 10131447 IC50 = 19300 nM T07663 C3AOI5 10138533 IC50 = 134 nM T07663 C8XPO7 10145438 Ki = 0.2 nM T07663 C4F3SH 10151707 IC50 = 1.585 nM T07663 C3H1IG 10161792 IC50 = 750 nM T07663 C89DXP 10181676 IC50 = 6 nM T07663 C5HC2X 10182563 IC50 = 52400 nM T07663 CK3TY8 10187239 IC50 = 2.089 nM T07663 CJZK81 10195399 IC50 = 1.9 nM T07663 C3GN8K 10200432 IC50 > 101000 nM T07663 CK81LJ 10203901 Ki = 4 nM T07663 CEY6F7 10205437 IC50 = 10.96 nM T07663 CLW92Y 10205894 IC50 = 65 nM T07663 CULN70 10206649 Ki = 0.31 nM T07663 C8JR4W 10221093 IC50 = 44000 nM T07663 CFGO46 10221904 IC50 = 60000 nM T07663 C8V6FE 10225063 IC50 = 2 nM T07663 CX35CL 10244508 IC50 = 6200 nM T07663 CGA50J 10244709 IC50 = 230 nM T07663 CT7RC0 10245770 IC50 = 15000 nM T07663 CC80XO 10247363 IC50 = 620 nM T07663 CP4YR0 10248176 IC50 > 1000000 nM T07663 C8G3BJ 10249105 IC50 = 3.5 nM T07663 C7MQZ1 10249183 IC50 > 1000000 nM T07663 C3AFN6 10250999 IC50 = 8300 nM T07663 CRK1U0 10252045 IC50 = 53000 nM T07663 C7GTC0 10264205 IC50 = 3020 nM T07663 C5VQL9 10264224 IC50 = 26000 nM T07663 CP70US 10267904 IC50 = 13800 nM T07663 CQ61CV 10268304 IC50 = 68400 nM T07663 C1QU2B 10268305 IC50 = 9470 nM T07663 C1VL9A 10269511 IC50 = 0.48 nM T07663 CH9C4K 10269859 IC50 = 23600 nM T07663 CR92JY 10270352 IC50 > 101000 nM T07663 C7CHR0 10270536 IC50 = 12600 nM T07663 C1VH6L 10279632 Ki = 8 nM T07663 C1FA4P 10288830 IC50 = 1.6 nM T07663 C3YO7N 10289243 IC50 = 1.288 nM T07663 CISQ36 10291967 IC50 = 63000 nM T07663 CKR74B 10292282 IC50 = 840 nM T07663 CA54BI 10294138 IC50 = 4 nM T07663 CKQ8I4 10313609 IC50 = 860 nM T07663 CUE72P 10314633 IC50 = 16 nM T07663 CJO72N 10315684 IC50 = 14 nM T07663 CIPN48 10316358 IC50 = 22000 nM T07663 C36AGZ 10321525 IC50 = 240 nM T07663 C90QZM 10324834 IC50 = 2.1 nM T07663 CRJW04 10334696 IC50 = 4000 nM T07663 C5K1LH 10336744 IC50 = 480 nM T07663 C6AQ0U 10338401 IC50 > 200000 nM T07663 C4GB5L 10338602 IC50 = 38 nM T07663 C52EPV 10339653 IC50 > 1000000 nM T07663 CMJG73 10342601 IC50 = 1200 nM T07663 CK05FV 10343476 IC50 = 68000 nM T07663 C32IUF 10344870 IC50 = 40000 nM T07663 CHZL20 10345264 IC50 = 1.6 nM T07663 CA18KO 10347662 IC50 = 20000 nM T07663 CC4W3M 10349233 IC50 = 24000 nM T07663 CQD9O7 10355498 IC50 = 6000 nM T07663 C4BL9Q 10358104 IC50 = 20000 nM T07663 CG8V6F 10358836 IC50 = 9000 nM T07663 CEIW08 10359077 IC50 = 175000 nM T07663 CP5S1A 10359273 IC50 = 165 nM T07663 C7QYK3 10359377 IC50 = 2150 nM T07663 CR35FX 10378878 IC50 = 15000 nM T07663 C2H9SE 10380126 IC50 = 4000 nM T07663 C6E5OY 10380621 IC50 = 5900 nM T07663 C5EVH3 10381520 IC50 = 380 nM T07663 C0J7OV 10382041 IC50 = 11000 nM T07663 C9IK3H 10382413 IC50 = 120 nM T07663 C52DNX 10384462 IC50 = 5500 nM T07663 CF6A1Q 10385088 IC50 > 200000 nM T07663 CZ6X9Y 10391444 IC50 = 3100 nM T07663 CQOX84 10393352 IC50 = 3.5 nM T07663 C9-APR-07 10394586 IC50 = 34000 nM T07663 CI8B3P 10401473 IC50 = 1000 nM T07663 C6E0PG 10401818 IC50 = 2000 nM T07663 C7X4EW 10402019 IC50 = 630 nM T07663 C78SRU 10403787 IC50 = 72 nM T07663 CUF0X6 10404302 IC50 > 1000000 nM T07663 C0ADP3 10404378 IC50 = 56000 nM T07663 CV3I5E 10405045 IC50 = 380 nM T07663 CP8ZV5 10408375 IC50 = 140 nM T07663 C4BF5Y 10411270 IC50 = 1.4 nM T07663 CQUE27 10413015 IC50 = 37000 nM T07663 CS7J4V 10414339 IC50 = 16 nM T07663 C0ZLB5 10423102 IC50 = 1000 nM T07663 C5ZQG3 10426854 IC50 = 5500 nM T07663 C5HMX2 10428149 IC50 = 32000 nM T07663 CB2X9W 10429802 IC50 = 110 nM T07663 CAW23H 10434818 IC50 > 1000000 nM T07663 CH76CS 10443650 IC50 = 42000 nM T07663 CBH5V4 10445800 IC50 = 24000 nM T07663 CZ8IC4 10448177 IC50 > 1000000 nM T07663 CYU38H 10448853 IC50 = 1600 nM T07663 C1RZ9E 10449000 IC50 > 1000000 nM T07663 C18EHX 10449737 IC50 = 1300 nM T07663 CU2HN6 10450290 IC50 > 200000 nM T07663 C9IF7Y 10451065 IC50 = 4.8 nM T07663 CY4O0K 10452443 IC50 = 38000 nM T07663 CI1H7F 10452463 IC50 = 0.05 nM T07663 C4LOK1 10454517 IC50 = 3600 nM T07663 CR04LJ 10456913 IC50 = 54000 nM T07663 CASV91 10466228 IC50 = 34000 nM T07663 C6IP3N 10468291 IC50 = 24000 nM T07663 C6PXC2 10471556 IC50 = 31 nM T07663 C2FYT6 10471617 IC50 = 2300 nM T07663 C2DEO3 10472374 IC50 > 200000 nM T07663 CBMI84 10473521 IC50 = 810 nM T07663 CF0I6O 10479155 IC50 = 13000 nM T07663 C5CI3G 10479468 IC50 = 53000 nM T07663 CZ92DR 10481735 IC50 = 9 nM T07663 CE2RJ7 10499713 IC50 = 420 nM T07663 C0N5LU 10504068 IC50 = 0.53 nM T07663 C71AJB 10520277 IC50 = 19 nM T07663 CSZ7L0 10520799 IC50 = 19 nM T07663 CPWU60 10524067 IC50 = 8000 nM T07663 CG1QK8 10542139 IC50 = 6200 nM T07663 C7LG4O 10543051 IC50 = 26000 nM T07663 C7K5PG 10544204 IC50 = 26 nM T07663 C0Z1CT 10546352 IC50 = 63 nM T07663 CCK5F8 10549901 IC50 = 120 nM T07663 CMK39Q 10553487 IC50 = 200 nM T07663 CQW79N 10554042 IC50 = 10000 nM T07663 CTYQ03 10565296 IC50 = 7500 nM T07663 C1DO9H 10573238 IC50 = 275 nM T07663 CI8GS1 10574005 IC50 = 590 nM T07663 CY9P5W 10575733 IC50 = 30000 nM T07663 CFY5J3 10576937 IC50 = 305 nM T07663 CYD4Z2 10592106 IC50 = 140 nM T07663 C4HVR8 10595830 IC50 = 5600 nM T07663 CRKT15 10597744 IC50 = 43 nM T07663 C71YLE 10598277 IC50 = 4 nM T07663 CJ7CU4 10603606 IC50 = 1000 nM T07663 CR9H4Z 10617782 IC50 = 4500 nM T07663 CK3GR5 10624131 IC50 = 20000 nM T07663 C25WRZ 10627119 IC50 = 9000 nM T07663 CC68NQ 10636956 IC50 = 100 nM T07663 CE57IW 10639502 IC50 = 3300 nM T07663 C0U8KD 10642598 IC50 = 10000 nM T07663 CX61NW 10642809 IC50 = 810 nM T07663 CNK65G 10646809 IC50 = 100000 nM T07663 CKNA14 10648008 IC50 = 20000 nM T07663 C32TRJ 10659857 IC50 = 240 nM T07663 C9GJ5K 10660011 IC50 = 13000 nM T07663 C8KWM5 10663015 IC50 = 34 nM T07663 CP13SC 10663562 IC50 = 80 nM T07663 COQ17R 10666144 IC50 = 9200 nM T07663 CBQ24O 10668762 IC50 = 4000 nM T07663 C1R9VY 10669652 IC50 = 110 nM T07663 CB9Y7A 10669693 IC50 = 40000 nM T07663 CWYZ15 10670833 IC50 = 2 nM T07663 C2Y5HF 10675032 IC50 = 800 nM T07663 CW12SY 10690095 IC50 = 510 nM T07663 CV6WT3 10692240 IC50 > 30000 nM T07663 C29YKI 10692613 IC50 = 1200 nM T07663 C0FPL8 10692684 IC50 = 800 nM T07663 CI6ON5 10698519 IC50 = 4000 nM T07663 C2JTX7 10715358 IC50 = 400 nM T07663 C1I8VM 10716045 IC50 = 1500 nM T07663 CDMP96 10717370 IC50 = 30000 nM T07663 CCI8R7 10729204 IC50 > 100000 nM T07663 C2P5VY 10731865 IC50 = 610 nM T07663 CSQG30 10741916 IC50 = 0.55 nM T07663 CTCS25 10753773 IC50 = 100 nM T07663 C3X8UM 10754735 IC50 = 800 nM T07663 C4EG9Z 10759241 IC50 = 19 nM T07663 CEIZ87 10761565 IC50 = 54 nM T07663 CINX82 10763354 IC50 = 20000 nM T07663 COVG15 10764868 IC50 = 120 nM T07663 C51XRM 10776762 IC50 = 2400 nM T07663 CR4O8B 10781567 IC50 = 16000 nM T07663 C7O8WB 10787783 IC50 = 180 nM T07663 CLM42P 10788651 IC50 = 20000 nM T07663 C7U2NT 10808382 IC50 = 140 nM T07663 CEI0J8 10809340 IC50 = 49 nM T07663 CDF43L 10810826 IC50 = 66 nM T07663 CTMX70 10815441 IC50 = 58000 nM T07663 CA9UW6 10816539 IC50 = 200 nM T07663 C5V1AY 10828080 IC50 = 60 nM T07663 C0SEG5 10830345 IC50 = 6000 nM T07663 CI0XH5 10833134 IC50 = 98 nM T07663 CT6VP3 10834312 IC50 = 560 nM T07663 C8HY0A 10835448 IC50 = 11 nM T07663 CZY5K8 10836947 IC50 = 600 nM T07663 CG2O1B 10836974 IC50 = 200 nM T07663 CR50XV 10841036 IC50 = 40000 nM T07663 CJ0TR9 10854527 IC50 = 100 nM T07663 CW3T1L 10863491 Ki = 154 nM T07663 C9TH7M 10863695 Ki = 1.75 nM T07663 CH0B6V 10885231 Ki = 188 nM T07663 CQ8YB7 10897309 Ki = 1.78 nM T07663 C0RTU9 10897531 EC50 = 9.5 nM T07663 CG0LM2 10907083 Ki = 0.4 nM T07663 CB6U4L 10929261 Ki = 0.47 nM T07663 CL1RW3 10929391 Ki = 0.21 nM T07663 C0BS9L 10939795 Ki = 0.71 nM T07663 C4KLI7 10951390 Ki = 1.14 nM T07663 C9UXZ6 10951441 Ki = 1.01 nM T07663 CP59RB 10968191 IC50 = 22300 nM T07663 C3GAM5 10973079 IC50 = 0.03 nM T07663 C96GWI 10983515 IC50 = 0.7 nM T07663 C84LQY 10983963 Ki = 2.59 nM T07663 CJCO78 10992580 Ki = 1.08 nM T07663 CKX30W 10994934 Ki = 0.61 nM T07663 C3EH8D 11006014 Ki = 24.7 nM T07663 CF7RW4 11016445 Ki = 2.64 nM T07663 CX1GO8 11016581 Ki = 2.71 nM T07663 CR7C1N 11017676 EC50 = 12 nM T07663 CO05WV 11024165 IC50 = 3900 nM T07663 CJMS98 11025421 Ki = 1.2 nM T07663 C3QT7I 11028215 Ki = 0.53 nM T07663 C98IUO 11039211 Ki = 0.76 nM T07663 CF6BL1 11049430 Ki = 62.8 nM T07663 C7B4MG 11071221 Ki = 1.71 nM T07663 CIO28H 11092703 Ki = 0.99 nM T07663 CG74CI 11093245 EC50 = 130 nM T07663 CW2AS4 11103879 Ki = 0.29 nM T07663 CRV32I 11114031 Ki = 3.74 nM T07663 C72TWL 11123617 Ki = 246 nM T07663 CX3N0E 11123630 Ki = 0.31 nM T07663 C24VFA 11125005 EC50 = 37 nM T07663 CL3DT7 11145432 Ki = 0.73 nM T07663 CU5C3E 11145600 Ki = 0.61 nM T07663 C3B1QP 11161553 IC50 = 21000 nM T07663 C6OH2Y 11212743 Ki = 0.22 nM T07663 CA8E0W 11212836 Ki = 0.58 nM T07663 C0FSV9 11225074 IC50 = 0.07 nM T07663 C8TD3U 11247946 IC50 = 0.14 nM T07663 C01VJK 11270159 Ki = 23.3 nM T07663 CF7R3Y 11270592 Ki = 1.06 nM T07663 C26HWL 11270869 IC50 = 0.78 nM T07663 C4R1UG 11270952 Ki = 11 nM T07663 CRZ9V8 11293623 Ki = 3.48 nM T07663 CGO29X 11318932 IC50 = 7600 nM T07663 CY9O2K 11351010 Ki = 0.35 nM T07663 CY71CZ 11351116 Ki = 4.53 nM T07663 C1YTA6 11351932 Ki = 118 nM T07663 CREQ98 11373312 IC50 = 95000 nM T07663 C4H9WX 11375723 IC50 = 320 nM T07663 CVT52P 11385644 Ki = 113 nM T07663 CPJ0Z3 11396900 Ki = 601 nM T07663 C4V6DZ 11418838 Ki = 12.5 nM T07663 C45VZC 11438405 IC50 > 16000 nM T07663 CKZ43J 11496164 IC50 = 0.08 nM T07663 CO9WX8 11497051 IC50 = 1.7 nM T07663 CS5P1N 11502459 IC50 = 2.1 nM T07663 C7S4QZ 11539946 IC50 = 1.01 nM T07663 C4ZYH9 11547485 IC50 = 2.5 nM T07663 C50BPN 11554196 IC50 = 0.65 nM T07663 CJ41RB 11560313 IC50 = 0.4 nM T07663 CJ1R6X 11568346 IC50 = 0.007 nM T07663 CL83VR 11574797 IC50 = 0.65 nM T07663 C86YZS 11575452 IC50 = 0.78 nM T07663 C53ARX 11582654 IC50 = 9.52 nM T07663 C1TOQ3 11583812 IC50 = 6.48 nM T07663 CY5JK4 11589901 IC50 = 34 nM T07663 CI6AW2 11590842 IC50 = 0.09 nM T07663 C58OXQ 11596704 IC50 = 3.3 nM T07663 CG5LT6 11605112 IC50 = 3.15 nM T07663 C7JLT3 11611915 IC50 = 0.07 nM T07663 CLU3G9 11639525 IC50 = 10 nM T07663 CO6XA4 11647832 IC50 = 0.72 nM T07663 CRK10B 11669288 IC50 = 67 nM T07663 C0B7RV 11675647 IC50 = 1.5 nM T07663 C1WV4T 11682414 IC50 = 0.5 nM T07663 C5LPU2 11690391 IC50 = 0.76 nM T07663 C5PHZ0 11710213 IC50 = 1300 nM T07663 CT69CO 11718514 IC50 = 2.6 nM T07663 C1RX0I 11720166 IC50 = 0.35 nM T07663 C7BAC0 11724504 IC50 = 4300 nM T07663 CM5T9U 11724564 IC50 = 35000 nM T07663 CNL0G1 11725859 IC50 = 10 nM T07663 C0AKJ4 11742456 IC50 > 100000 nM T07663 CA1E6R 11754694 Ki = 0.53 nM T07663 C26CKE 11754697 IC50 = 300 nM T07663 C6ERQ9 11755313 Ki = 18 nM T07663 CMP35Y 11762536 Ki = 0.15 nM T07663 C57BPZ 11763070 Ki = 1.3 nM T07663 C1K3JX 11764545 IC50 = 37000 nM T07663 CF23VJ 11775013 IC50 = 0.5012 nM T07663 C23DSJ 11782534 IC50 = 9300 nM T07663 C5EFC7 11793221 IC50 = 1000 nM T07663 CGA1F8 11794425 IC50 = 3000 nM T07663 CUM8A9 11795949 IC50 = 4300 nM T07663 C3LO2Q 11799196 IC50 = 3.1 nM T07663 C0GP6R 11812647 Ki = 0.35 nM T07663 C1J9UP 11813138 Ki = 0.52 nM T07663 CMU6W8 11826705 Ki = 1.74 nM T07663 CB4RS5 11826881 Ki = 2.09 nM T07663 C29HOL 11828590 EC50 = 44 nM T07663 CT5C0K 11849942 IC50 = 100 nM T07663 CS42FO 11849943 IC50 = 240 nM T07663 C2FZY3 11850012 IC50 = 470 nM T07663 CRY1U7 11850013 IC50 = 140 nM T07663 CVJ1X4 11850014 IC50 = 50 nM T07663 CAPF41 11850015 IC50 = 180 nM T07663 C4GQ2P 11850016 IC50 = 38 nM T07663 C4YP5D 11850079 IC50 = 40 nM T07663 C8VUW0 11850080 IC50 = 23 nM T07663 CJ6ZX9 11850081 IC50 = 8.3 nM T07663 CQ2JU9 11850082 IC50 = 79 nM T07663 CSI25Y 11850083 IC50 = 95 nM T07663 CW6D5J 11850144 IC50 = 370 nM T07663 CT9LD7 11850145 IC50 = 1500 nM T07663 C14ZXU 11850147 IC50 = 390 nM T07663 CU7X9W 11850294 IC50 = 71 nM T07663 C8ZM2F 11850366 IC50 = 220 nM T07663 CLI6G9 11850367 IC50 = 100 nM T07663 CC59AF 11850439 IC50 = 1400 nM T07663 CUK49V 11988837 Ki = 600 nM T07663 CFIO49 11988967 Ki = 1600 nM T07663 C2D0NG 11989101 Ki = 590 nM T07663 C65ABT 11989102 Ki = 1200 nM T07663 C05CLB 11992443 IC50 = 0.68 nM T07663 C0Z3KV 11992527 IC50 = 0.9 nM T07663 CXW57M 11992528 IC50 = 0.26 nM T07663 CH86SQ 11992529 IC50 = 0.11 nM T07663 CIX0V4 11992531 IC50 = 1.05 nM T07663 C7X4LC 11992631 IC50 = 0.78 nM T07663 C1B4XD 11992634 IC50 = 0.05 nM T07663 CAG1U6 11992635 IC50 = 0.1 nM T07663 CHT82G 11992739 IC50 = 0.09 nM T07663 CR4CA6 11992740 IC50 = 0.14 nM T07663 CIOU94 11992741 IC50 = 0.25 nM T07663 C95DJC 11992742 IC50 = 0.24 nM T07663 C0KM5I 11992827 IC50 = 1.1 nM T07663 CM57ID 11992831 IC50 = 0.07 nM T07663 CPX16N 11993169 IC50 = 0.07 nM T07663 C0Q4KT 11993170 IC50 = 0.04 nM T07663 C3HOV8 11993171 IC50 = 0.05 nM T07663 CZ7YR6 11993243 IC50 = 2.59 nM T07663 C4VY3X 11993244 IC50 = 0.34 nM T07663 CP4J1S 11993342 IC50 = 0.14 nM T07663 C0QZ6W 11993365 IC50 = 0.15 nM T07663 COQ5N2 11993435 IC50 = 0.43 nM T07663 C39KLP 11993437 IC50 = 1.17 nM T07663 CL8TM7 11993463 IC50 = 0.13 nM T07663 C1ZDC4 11993465 IC50 = 0.08 nM T07663 CK63SM 11993560 IC50 = 1.65 nM T07663 CIRM68 11993561 IC50 = 0.07 nM T07663 C6W2LU 11993562 IC50 = 0.13 nM T07663 C6VI5Z 12020635 Ki = 126 nM T07663 C48IYW 12020642 Ki = 24 nM T07663 CJC01W 12020645 Ki > 1000 nM T07663 CJ4H1G 12020670 Ki = 123 nM T07663 C6D0MG 12069381 IC50 = 1.4 nM T07663 C6S8LD 12355883 IC50 = 1500 nM T07663 CX0C7I 12993019 Ki = 543 nM T07663 CNR05L 12993020 Ki = 126 nM T07663 CO3G0B 12993027 Ki = 0.98 nM T07663 C09OJP 12993038 Ki = 2.07 nM T07663 CI18JL 13026433 IC50 = 1610 nM T07663 C51CKG 14583584 IC50 = 45500 nM T07663 C2ZX8H 14756622 IC50 = 1000 nM T07663 CVT43Z 15473392 IC50 = 60 nM T07663 C2RT6A 15500912 IC50 = 1.9 nM T07663 C8E4IH 15524307 IC50 = 11 nM T07663 C12BUL 15524308 IC50 = 19 nM T07663 CAC5H0 15606258 IC50 = 91000 nM T07663 C3BI9R 15951010 IC50 > 2000 nM T07663 CW6MV8 15981426 IC50 = 26 nM T07663 CYE3L9 16038477 IC50 = 2.6 nM T07663 C9OF5R 16038616 IC50 = 3.7 nM T07663 C8FJM7 16038617 IC50 = 4.5 nM T07663 C4T6CP 16038618 IC50 = 1.2 nM T07663 CIR42U 16038756 IC50 = 12 nM T07663 CF3UG1 16066664 IC50 = 0.04 nM T07663 CG1V8D 17799315 IC50 = 2.7 nM T07663 C1PZ8C 18734933 IC50 > 16000 nM T07663 C6OJI9 18796635 IC50 = 8900 nM T07663 C1FJL6 18796640 IC50 > 100000 nM T07663 CRJO82 18796649 IC50 = 4000 nM T07663 CA16YO 18796653 IC50 = 780 nM T07663 CKCM70 18796657 IC50 = 2200 nM T07663 C36LEN 18796668 IC50 = 1300 nM T07663 C0L8NR 18796689 IC50 = 1900 nM T07663 CBF8M6 18796697 IC50 = 1000 nM T07663 C3RH7V 18796719 IC50 = 11000 nM T07663 CC2WD9 18796725 IC50 > 100000 nM T07663 CNSH93 18796735 IC50 = 2000 nM T07663 CHK4Z7 18796752 IC50 = 32000 nM T07663 CNZ3I1 18796756 IC50 = 4600 nM T07663 CC1LP2 18796767 IC50 = 1000 nM T07663 C2FN9A 18796769 IC50 = 26000 nM T07663 CUE4A2 18796773 IC50 = 2000 nM T07663 C02JXD 18796791 IC50 = 1700 nM T07663 CQ8I5K 18796795 IC50 = 3500 nM T07663 CDC76R 20299686 IC50 = 26 nM T07663 CNX2D5 20646826 IC50 = 0.86 nM T07663 C36XCM 20646828 IC50 = 4.4 nM T07663 C1H2WT 20709323 IC50 = 1.8 nM T07663 C58VPG 21212519 IC50 = 2100 nM T07663 CXM8E3 21704212 IC50 = 0.79 nM T07663 CRY9Z1 21704213 IC50 = 0.32 nM T07663 CS09OZ 21704217 IC50 = 0.5 nM T07663 CH53WM 21704221 IC50 = 14 nM T07663 C7RK1W 21920272 IC50 = 5180 nM T07663 CH7N9S 21920275 IC50 = 7000 nM T07663 CV04DH 21920370 IC50 > 101000 nM T07663 C97JPF 22004355 IC50 = 6.7 nM T07663 C7DJ9E 22004357 IC50 = 2.6 nM T07663 CY6QT7 22004369 IC50 = 1.7 nM T07663 C2STP3 22004386 IC50 = 6.8 nM T07663 C7ZH2R 22004388 IC50 = 0.3 nM T07663 COM30K 22004392 IC50 = 0.7 nM T07663 C37JNS 22004412 IC50 = 0.7 nM T07663 C64YFT 22226537 IC50 = 553 nM T07663 C5G6BS 22226562 IC50 = 30 nM T07663 C70JWO 22226563 IC50 = 94 nM T07663 C8TEV5 22601583 IC50 = 0.4 nM T07663 C2FMU0 22601651 IC50 = 1.3 nM T07663 CNGD52 22744443 IC50 = 1.2 nM T07663 CMIO49 23527107 IC50 = 100 nM T07663 CZD94A 23527108 IC50 = 19 nM T07663 CW96SI 23624262 IC50 = 561 nM T07663 CXB78L 23624298 IC50 > 5000 nM T07663 C4S6VD 23654252 IC50 > 50000 nM T07663 CAJ57O 24751843 IC50 = 79000 nM T07663 CR0D6X 24751988 IC50 > 400000 nM T07663 CL79TD 24751991 IC50 = 65000 nM T07663 C51ZNR 24774842 IC50 > 5000 nM T07663 CQ19ZC 24775191 IC50 = 3500 nM T07663 C9WGI4 24802717 IC50 = 919 nM T07663 C4Y3FK 24883368 IC50 = 1.6 nM T07663 C5F6SD 24956185 IC50 = 26 nM T07663 CA9PN0 24957913 IC50 = 17 nM T07663 C6EQG2 24963293 IC50 = 0.2 nM T07663 CJ43BX 24963638 IC50 = 0.18 nM T07663 CLDO78 24963639 IC50 = 0.72 nM T07663 CG1BJ3 24965774 IC50 = 0.21 nM T07663 CDC01R 24965775 IC50 = 0.33 nM T07663 CDF34R 24966125 IC50 = 0.22 nM T07663 CNO40A 24966126 IC50 = 0.3 nM T07663 CY0G1A 24966127 IC50 = 0.23 nM T07663 CS56UN 24966128 IC50 = 1.08 nM T07663 CA25UL 24969619 IC50 = 0.31 nM T07663 C3AFU0 25093775 IC50 = 3.28 nM T07663 C93DZI 25147798 IC50 > 50000 nM T07663 CPC08B 25179287 IC50 > 50000 nM T07663 COB03R 25179478 IC50 = 40000 nM T07663 C1AV7L 30105766 IC50 = 8 nM T07663 C43UKE 42628078 IC50 = 2.4 nM T07663 CICF39 42629702 IC50 = 1850 nM T07663 CM3X9S 42629827 IC50 > 1000 nM T07663 CQN26J 42629945 IC50 = 1240 nM T07663 C6O5FX 42630062 IC50 = 2080 nM T07663 C71ZNR 42630180 IC50 = 1440 nM T07663 C4RHY0 42630191 IC50 > 5000 nM T07663 CT6RS9 42630192 IC50 = 5165 nM T07663 CYZL43 42630317 IC50 = 8780 nM T07663 CH42OZ 42630318 IC50 > 5000 nM T07663 C7X5AH 42630437 IC50 = 2050 nM T07663 CEPY38 43826154 IC50 = 200000 nM T07663 CQU19I 44180409 IC50 = 30300 nM T07663 CW8OB3 44243146 Ki = 10600 nM T07663 C19SIQ 44249786 IC50 = 14.5 nM T07663 C03DAV 44249787 IC50 = 2.3 nM T07663 CJ1GS3 44249944 IC50 = 0.9 nM T07663 CAL8X3 44264943 IC50 = 1 nM T07663 C59QCJ 44274690 IC50 = 3.89 nM T07663 C9KV6Y 44274762 IC50 = 6.457 nM T07663 CXA6Y3 44274773 IC50 = 0.61 nM T07663 CF4H9A 44274775 IC50 = 0.8913 nM T07663 CW7J4K 44274797 IC50 = 1.995 nM T07663 C9VK6M 44274798 IC50 = 5.012 nM T07663 CTP4O5 44274817 IC50 = 2.818 nM T07663 CA6J8T 44274920 IC50 = 3000 nM T07663 CV1ZA7 44280486 IC50 = 3.6 nM T07663 CG8R0W 44280487 IC50 = 4 nM T07663 CS0FX4 44280546 IC50 = 2.7 nM T07663 C05SIA 44280556 IC50 = 12.8 nM T07663 CA9KV4 44280558 IC50 = 8.4 nM T07663 CY74KE 44280614 IC50 = 19.8 nM T07663 C4RO9D 44280635 IC50 = 2.5 nM T07663 CH7W2T 44280722 IC50 = 1.2 nM T07663 CTO54N 44280723 IC50 = 0.7 nM T07663 CXRU70 44280792 IC50 = 13.2 nM T07663 CO7NV0 44280794 IC50 = 164 nM T07663 CG8I6M 44280801 IC50 = 57 nM T07663 CDQ8B2 44280847 IC50 = 1.5 nM T07663 C0N3JE 44280911 IC50 = 2 nM T07663 C3DHJ2 44280985 IC50 = 1.9 nM T07663 CA3GF6 44280994 IC50 = 127 nM T07663 CXB40D 44281036 IC50 = 28.6 nM T07663 CA1HN8 44281061 IC50 = 15.7 nM T07663 C7TKW4 44281095 IC50 = 7.1 nM T07663 CK3W1B 44281096 IC50 = 4 nM T07663 CC81DV 44281265 IC50 = 132 nM T07663 CNO94A 44281273 IC50 > 1000 nM T07663 CO1L0H 44282267 IC50 = 160 nM T07663 C79RGL 44282685 IC50 = 270 nM T07663 CK8Y4F 44286951 IC50 = 160 nM T07663 CNW8B7 44287071 IC50 = 73 nM T07663 CDHP47 44287318 IC50 = 0.6 nM T07663 C2O0JN 44307127 IC50 = 530 nM T07663 C2FW1A 44310350 IC50 = 2900 nM T07663 COP54Y 44318505 IC50 = 1.5 nM T07663 CK0N6P 44318516 IC50 = 0.95 nM T07663 C4AWN5 44318518 IC50 = 1.23 nM T07663 CP30VE 44318806 IC50 = 0.73 nM T07663 CH4T3J 44318846 IC50 = 0.7 nM T07663 CKLM51 44318862 IC50 = 150 nM T07663 CX5SO4 44320719 IC50 = 77 nM T07663 C1SI7O 44320739 IC50 = 551 nM T07663 C3TZ6O 44320740 IC50 = 105 nM T07663 CH18VT 44320762 IC50 = 135 nM T07663 C45ZJD 44320781 IC50 = 130 nM T07663 CF1DO2 44320804 IC50 = 160 nM T07663 CLBV45 44320831 IC50 = 28 nM T07663 C6RS5T 44320847 IC50 = 1360 nM T07663 CVS5D1 44320863 IC50 = 20 nM T07663 C0GM7F 44320900 IC50 = 315 nM T07663 C13WMT 44320988 IC50 = 12 nM T07663 CP78QN 44320989 IC50 = 26 nM T07663 CP34EA 44321012 IC50 = 63 nM T07663 CN8Z1I 44321013 IC50 = 24 nM T07663 CDP87G 44321026 IC50 = 3.5 nM T07663 C9G0OQ 44321064 IC50 = 19 nM T07663 CWMD23 44321111 IC50 = 5.5 nM T07663 CPEB60 44321112 IC50 = 10 nM T07663 CX9L7V 44321135 IC50 = 11 nM T07663 C51CET 44321137 IC50 = 5 nM T07663 CD0QO6 44321152 IC50 = 93 nM T07663 C69MZC 44321154 IC50 = 5420 nM T07663 CUV0W1 44321156 IC50 > 10000 nM T07663 CP71YV 44321172 IC50 = 16 nM T07663 CXNO48 44321173 IC50 > 10000 nM T07663 C7NE6Q 44321175 IC50 > 10000 nM T07663 C81WUS 44321176 IC50 = 1500 nM T07663 C4QO0A 44321178 IC50 > 10000 nM T07663 CZWA59 44321202 IC50 = 60 nM T07663 C4B1WH 44321204 IC50 = 73 nM T07663 CIAN09 44321224 IC50 = 1810 nM T07663 C86ATM 44321229 IC50 = 100 nM T07663 CR54IA 44321231 IC50 > 10000 nM T07663 C4VFQ5 44321253 IC50 = 91 nM T07663 CYVA51 44321254 IC50 > 10000 nM T07663 CUQ3R1 44321255 IC50 = 100 nM T07663 C7BM6I 44321261 IC50 = 59 nM T07663 CZ16IY 44324251 IC50 = 30000 nM T07663 CCX9Z3 44324252 IC50 = 24000 nM T07663 CG6UT1 44324296 IC50 = 20000 nM T07663 C8M4WJ 44324373 IC50 = 22000 nM T07663 CY5HZ7 44324390 IC50 = 9000 nM T07663 C5KYV6 44324391 IC50 = 8000 nM T07663 C5C4QX 44324507 IC50 = 22000 nM T07663 CNK2F8 44331802 IC50 = 270 nM T07663 CGFP09 44336826 IC50 = 0.82 nM T07663 C98VIX 44336827 IC50 = 0.69 nM T07663 C1L6SG 44336834 IC50 = 1.1 nM T07663 CH8RY1 44336844 IC50 = 1.8 nM T07663 C1AC3Z 44336847 IC50 = 0.3 nM T07663 C0NT4K 44336855 IC50 = 0.33 nM T07663 C9WLD8 44336856 IC50 = 2 nM T07663 CUME98 44336924 IC50 = 0.58 nM T07663 CM1BO3 44348247 IC50 = 32000 nM T07663 CY5L6J 44348257 IC50 = 11000 nM T07663 CD5ZW3 44348484 IC50 = 650 nM T07663 C80PGJ 44348564 IC50 = 1500 nM T07663 CY0T1M 44348625 IC50 = 9600 nM T07663 CG98RE 44358477 Ki = 3.32 nM T07663 C3H4MR 44358478 Ki = 2.49 nM T07663 CBD52Z 44358886 Ki = 4.66 nM T07663 C7LN0W 44363056 IC50 = 50 nM T07663 C71YUD 44363183 IC50 = 3000 nM T07663 CF0IB6 44377834 IC50 = 105 nM T07663 CWO45S 44377842 Ki = 145 nM T07663 C27ZVC 44377867 Ki = 132 nM T07663 C7TXQ3 44377869 Ki = 179 nM T07663 CSW1J4 44377881 Ki = 219 nM T07663 C27TDG 44377933 Ki > 100 nM T07663 C8XM3I 44377988 IC50 = 100 nM T07663 C5IOH4 44378004 IC50 = 95 nM T07663 C85XCK 44378015 Ki = 850 nM T07663 C0H7KF 44378030 Ki > 5000 nM T07663 CU29OZ 44378056 Ki = 130 nM T07663 CLV13K 44378110 Ki > 10000 nM T07663 CL3SI5 44378121 Ki = 50.6 nM T07663 CYA76O 44378142 IC50 > 10000 nM T07663 C6IOU8 44378149 Ki = 8.11 nM T07663 CBQ5W3 44378155 IC50 = 67 nM T07663 CR30BD 44378165 Ki = 32.3 nM T07663 CHL5D9 44378187 Ki = 77.5 nM T07663 CV5Y1A 44378199 Ki = 64.2 nM T07663 CT8NH9 44383851 IC50 > 10000 nM T07663 C19CRH 44383901 IC50 = 19700 nM T07663 CR9O3I 44383902 IC50 > 30000 nM T07663 CW47HV 44383906 IC50 = 17700 nM T07663 CL86MY 44383907 IC50 > 10000 nM T07663 CW63HQ 44383912 IC50 > 10000 nM T07663 CF98LG 44384286 IC50 > 10000 nM T07663 CN1WS7 44384345 IC50 = 66700 nM T07663 C01XPL 44384404 IC50 = 22700 nM T07663 CWPR87 44384405 IC50 = 2900 nM T07663 C59SDR 44384406 IC50 = 3900 nM T07663 C7WT4G 44384540 IC50 = 18200 nM T07663 C4RQB0 44384541 IC50 = 21200 nM T07663 CRZ5G8 44384546 IC50 > 100000 nM T07663 C6W4GY 44384713 IC50 = 56100 nM T07663 CKH7M8 44384714 IC50 > 30000 nM T07663 C0ZGU6 44385109 IC50 = 12100 nM T07663 CE80VB 44385244 IC50 = 1700 nM T07663 CH5GU8 44385282 IC50 = 14900 nM T07663 CL50UE 44385283 IC50 = 9700 nM T07663 CSN56E 44386916 IC50 = 3.981 nM T07663 C13HPW 44393651 IC50 > 101000 nM T07663 CJ6GB5 44393709 IC50 = 11600 nM T07663 CQP01D 44393950 IC50 = 18770 nM T07663 CU1CQ8 44394047 IC50 = 80000 nM T07663 CJYC83 44397324 IC50 = 2070 nM T07663 CZUY06 44397327 IC50 = 5620 nM T07663 CB64FY 44397328 IC50 = 1690 nM T07663 CDJ87T 44397345 IC50 = 6190 nM T07663 C5CTF6 44397346 IC50 = 140 nM T07663 C2T7BQ 44397347 IC50 = 680 nM T07663 C39VBJ 44397348 IC50 = 3350 nM T07663 CU3BF4 44397365 IC50 = 1840 nM T07663 CRTY10 44397366 IC50 = 2930 nM T07663 CYFD01 44397379 IC50 = 1510 nM T07663 C4VS1H 44397382 IC50 = 74 nM T07663 C8YCU6 44397384 IC50 = 3190 nM T07663 CQD8Z7 44397386 IC50 = 13 nM T07663 CCL9D6 44397387 IC50 = 620 nM T07663 CSAQ43 44397397 IC50 = 3190 nM T07663 C7MZ8J 44397413 IC50 = 5990 nM T07663 C8KA6R 44397415 IC50 = 920 nM T07663 CR8P4T 44397447 IC50 = 3280 nM T07663 C9TK8I 44397448 IC50 = 5150 nM T07663 CF2AP3 44397474 IC50 = 230 nM T07663 CQT12O 44397490 IC50 = 2720 nM T07663 C6FJV7 44397494 IC50 = 1280 nM T07663 CZ5QV6 44397495 IC50 = 2130 nM T07663 CAP7W0 44397504 IC50 = 1210 nM T07663 CU13ES 44397515 IC50 = 96 nM T07663 CQY79V 44397539 IC50 = 8900 nM T07663 CTAI27 44397548 IC50 = 1470 nM T07663 C98ZCS 44397556 IC50 = 270 nM T07663 CMC12S 44397573 IC50 = 6490 nM T07663 CL15YW 44397574 IC50 = 3810 nM T07663 C6GIS2 44397576 IC50 = 10000 nM T07663 C65PLD 44397577 IC50 = 4520 nM T07663 C8MFC2 44397582 IC50 = 3300 nM T07663 C3PN4D 44397598 IC50 = 790 nM T07663 CE2GZ3 44397599 IC50 = 6680 nM T07663 CY0KB5 44397600 IC50 = 2660 nM T07663 C86IAQ 44397602 IC50 = 1900 nM T07663 CR0D6I 44397603 IC50 = 8760 nM T07663 CD67XW 44397612 IC50 = 6090 nM T07663 C1ISA5 44397619 IC50 = 7820 nM T07663 CG2XI7 44397621 IC50 = 6250 nM T07663 C1HBU8 44397622 IC50 = 3160 nM T07663 CA1FG3 44397627 IC50 = 9070 nM T07663 C1FJH9 44397640 IC50 = 74 nM T07663 CV2Q1K 44397643 IC50 = 17 nM T07663 C69WZC 44397646 IC50 = 130 nM T07663 CC8Z3A 44397647 IC50 = 3680 nM T07663 C1VB8P 44397694 IC50 = 630 nM T07663 CV2M0A 44397708 IC50 = 3500 nM T07663 C8MZF1 44397709 IC50 = 4580 nM T07663 C2OA3Y 44397724 IC50 = 9460 nM T07663 CJIK26 44397727 IC50 = 320 nM T07663 CFP7S8 44397728 IC50 = 350 nM T07663 CERQ57 44397746 IC50 = 2640 nM T07663 C2PJ6R 44397748 IC50 = 10000 nM T07663 CAQD83 44397749 IC50 = 1100 nM T07663 C5GLC2 44397761 IC50 = 40 nM T07663 CUZY95 44397764 IC50 = 8620 nM T07663 CQCN29 44397781 IC50 = 770 nM T07663 C0B2YM 44397782 IC50 = 830 nM T07663 CWL0A9 44397785 IC50 = 3410 nM T07663 CSN79W 44397799 IC50 = 1800 nM T07663 C20BLM 44397801 IC50 = 1830 nM T07663 CJG87Q 44397802 IC50 = 500 nM T07663 CP1CU7 44397810 IC50 = 650 nM T07663 CI7HS1 44397811 IC50 = 6070 nM T07663 C9SQ1V 44397814 IC50 = 1450 nM T07663 CZF29N 44397816 IC50 = 190 nM T07663 CIVF18 44397836 IC50 = 890 nM T07663 CP18FI 44397837 IC50 = 2580 nM T07663 CRMN86 44397859 IC50 = 3200 nM T07663 CC7B3S 44397860 IC50 = 460 nM T07663 C01CAI 44397871 IC50 = 10000 nM T07663 C8Y0WF 44397874 IC50 = 7650 nM T07663 CJ6B1W 44397876 IC50 = 2420 nM T07663 C28ERI 44397877 IC50 = 2490 nM T07663 C6Y9XN 44397888 IC50 = 520 nM T07663 CIOM21 44397889 IC50 = 430 nM T07663 CVQ8C1 44397891 IC50 = 1240 nM T07663 CX3M5J 44397892 IC50 = 270 nM T07663 CYX72U 44397904 IC50 = 3100 nM T07663 C5JS4T 44397906 IC50 = 8910 nM T07663 CVB7K2 44397908 IC50 = 2200 nM T07663 CP8CW5 44397940 IC50 = 9430 nM T07663 CFHR09 44397941 IC50 = 9280 nM T07663 CP62TK 44397956 IC50 = 4990 nM T07663 C6UY9Z 44397957 IC50 = 4250 nM T07663 C23GTH 44397958 IC50 = 8430 nM T07663 CG36QI 44397976 IC50 = 10000 nM T07663 CDK84C 44397977 IC50 = 7560 nM T07663 CB3ZG1 44397979 IC50 = 1030 nM T07663 C4AO1D 44397980 IC50 = 9870 nM T07663 CW65CR 44397987 IC50 = 5470 nM T07663 C1DQW5 44397991 IC50 = 40 nM T07663 CP8F9A 44397992 IC50 = 8580 nM T07663 CM1ZW4 44401687 IC50 = 230 nM T07663 C0YZV7 44401690 IC50 = 33 nM T07663 C7CDY2 44401692 IC50 = 74 nM T07663 CT8R0Q 44401694 IC50 = 81 nM T07663 CDSE04 44401695 IC50 = 90 nM T07663 CB3RC6 44401705 IC50 = 60 nM T07663 CA59PR 44401708 IC50 = 81 nM T07663 CXA4D6 44401724 IC50 = 23 nM T07663 C17ODM 44401727 IC50 = 430 nM T07663 CX0AZ7 44401742 IC50 = 270 nM T07663 C3G2RU 44401767 IC50 = 350 nM T07663 C4BJ3U 44401771 IC50 = 38 nM T07663 C0F9ZD 44401772 IC50 = 2.3 nM T07663 CM45YT 44401790 IC50 = 33 nM T07663 CA1SR3 44401812 IC50 = 29 nM T07663 CN63AH 44401816 IC50 = 30 nM T07663 CVOW53 44401827 IC50 = 32 nM T07663 CVCN36 44401831 IC50 = 920 nM T07663 C59TYU 44401851 IC50 = 200 nM T07663 C78VHO 44401870 IC50 = 13000 nM T07663 CSM4X8 44401879 IC50 = 20 nM T07663 CZU4T7 44401880 IC50 = 3.3 nM T07663 C01BEI 44401886 IC50 = 100 nM T07663 CU4AR1 44401892 IC50 = 5.3 nM T07663 C14LNK 44401904 IC50 = 60 nM T07663 CVPZ92 44401905 IC50 = 28 nM T07663 C0BRH8 44401908 IC50 = 450 nM T07663 CN4T6Z 44401928 IC50 = 145 nM T07663 CV17OM 44401929 IC50 = 14 nM T07663 CK9VN7 44401931 IC50 = 320 nM T07663 C9Q1ET 44401943 IC50 = 40 nM T07663 CB98IX 44401972 IC50 = 130 nM T07663 CD51UN 44401977 IC50 = 100 nM T07663 C19QCE 44401981 IC50 = 48 nM T07663 C04BTX 44401982 IC50 = 15 nM T07663 C7MY1S 44402027 IC50 = 59 nM T07663 C6XA7P 44402060 IC50 = 3100 nM T07663 CTZ52C 44402073 IC50 = 28 nM T07663 C4P8RN 44402077 IC50 = 35 nM T07663 C6S8KA 44402114 IC50 = 40 nM T07663 CDNZ52 44402130 IC50 = 180 nM T07663 CP78NL 44402133 IC50 = 1100 nM T07663 CWVH96 44402149 IC50 = 100 nM T07663 C9BN6H 44402168 IC50 = 6.5 nM T07663 CQM65U 44402195 IC50 = 160 nM T07663 CM90NL 44402196 IC50 = 980 nM T07663 C6IY5O 44402213 IC50 = 39 nM T07663 C4O7QE 44402239 IC50 = 22 nM T07663 C4P0AC 44402278 IC50 = 75 nM T07663 C1GPC2 44402295 IC50 = 7.8 nM T07663 CCZ2E8 44438552 IC50 = 462 nM T07663 CB1C2M 44438553 IC50 = 25 nM T07663 C7RV5Q 44438554 IC50 = 20 nM T07663 CCOJ06 44438555 IC50 = 28 nM T07663 CB93RX 44438557 IC50 = 33 nM T07663 C9AO2Z 44438558 IC50 = 42 nM T07663 C50ZMB 44438560 IC50 = 5 nM T07663 C39ZMJ 44438561 IC50 = 26 nM T07663 CBQN25 44438563 IC50 = 10000 nM T07663 CJH70L 44438564 IC50 = 34 nM T07663 CE4S8J 44438565 IC50 = 51 nM T07663 CK1JU3 44459193 IC50 = 1.288 nM T07663 CZFU59 44459332 IC50 = 43 nM T07663 CJ0Q4D 44459333 IC50 = 2.2 nM T07663 CT39RH 44459469 IC50 = 2.8 nM T07663 CG4AI3 44459482 IC50 = 2.089 nM T07663 CZ6IU2 44459494 IC50 = 6.457 nM T07663 C68RBI 44459495 IC50 = 5.37 nM T07663 CNJ16Q 44459505 IC50 = 4.5 nM T07663 C0FQ1O 44459535 IC50 = 5 nM T07663 CT9R7K 44459542 IC50 = 46 nM T07663 CP97OV 44459564 IC50 = 57.54 nM T07663 C49NWP 44459572 IC50 = 550 nM T07663 C5G2JO 44459598 IC50 = 19.95 nM T07663 C8MBD9 44459599 IC50 = 158.49 nM T07663 C0W4VT 44459622 IC50 = 39.81 nM T07663 C18EJF 44459640 IC50 = 1.8 nM T07663 C7RGD3 44459641 IC50 = 2.089 nM T07663 CQ95TO 44459661 IC50 = 128.82 nM T07663 CRH7N1 44459687 IC50 = 6.31 nM T07663 C8JS2X 44459694 IC50 = 18 nM T07663 CO3F9K 44459713 IC50 = 8.3 nM T07663 CF4C3P 44459717 IC50 = 7 nM T07663 C1W5OG 44459718 IC50 = 21.88 nM T07663 C31SQM 44459720 IC50 = 2.291 nM T07663 CS17XE 44459751 IC50 = 6.761 nM T07663 C85QDR 44459752 IC50 = 13 nM T07663 CI2V6T 44459760 IC50 = 1.096 nM T07663 CJN91Z 44459761 IC50 = 0.8913 nM T07663 CQ01TE 44459776 IC50 = 3.09 nM T07663 C24BGR 44459782 IC50 = 1.514 nM T07663 CB37LV 44459783 IC50 = 6.3 nM T07663 C1V3CW 44459848 IC50 = 3.02 nM T07663 C52JOE 44459875 IC50 = 47.86 nM T07663 CZ1DJ8 44459876 IC50 = 55 nM T07663 CWXV09 44459906 IC50 = 0.3 nM T07663 CJ4L3O 44459907 IC50 = 7.943 nM T07663 CZ0DN5 44572149 IC50 > 10000 nM T07663 C6U8QW 44572150 IC50 > 10000 nM T07663 C9XD8C 44572789 IC50 = 5200 nM T07663 C72XEI 44572984 IC50 > 10000 nM T07663 CIX5Q0 44572985 IC50 > 10000 nM T07663 C7UXN8 44572986 IC50 > 10000 nM T07663 CRBQ49 44572987 IC50 = 6500 nM T07663 C0WXB4 44580020 IC50 = 1.585 nM T07663 CHA63L 44580021 IC50 = 6.31 nM T07663 CX3L1P 44587252 IC50 = 160 nM T07663 CI3K8T 44605342 IC50 = 87100 nM T07663 CV8RY3 45260952 IC50 = 3 nM T07663 CLEU14 45260983 IC50 = 12 nM T07663 C48QSY 45261659 IC50 = 1700 nM T07663 CC5Z7N 45261660 IC50 = 2300 nM T07663 C26IBG 45261674 IC50 = 5000 nM T07663 CTG0D9 45261728 IC50 = 2800 nM T07663 CS7GA3 45264997 IC50 = 760 nM T07663 C3IOB7 45265000 IC50 = 360 nM T07663 CKW39R 45267744 IC50 = 4.571 nM T07663 C9PC5S 45267756 IC50 = 223.87 nM T07663 CR7QN3 45267764 IC50 = 0.3 nM T07663 C1KTZ3 45267771 IC50 = 33.9 nM T07663 C6WLB4 45268626 IC50 = 2.5 nM T07663 CE0U3W 45268639 IC50 = 13.49 nM T07663 CR8JH9 45268646 IC50 = 33.3 nM T07663 CM8OP3 45268652 IC50 = 0.3 nM T07663 CD6A0O 45269469 IC50 = 20.3 nM T07663 CL42XG 45269481 IC50 = 3.467 nM T07663 CRWE76 45269493 IC50 = 0.4 nM T07663 CHN4F0 45269499 IC50 = 2.9 nM T07663 C6DQU1 45269515 IC50 = 534 nM T07663 CB4IO3 45269516 IC50 = 51 nM T07663 CD47UP 45270308 IC50 = 28.18 nM T07663 C4VPC6 45270320 IC50 = 1 nM T07663 CMF3T7 45270338 IC50 = 36.5 nM T07663 C1XZ4Q 45270704 IC50 = 1.21 nM T07663 C89NBL 45270705 IC50 = 1.21 nM T07663 CDWX76 45271142 IC50 = 147.91 nM T07663 C62LVH 45272043 IC50 = 52.5 nM T07663 C0AO8K 45272078 IC50 = 43 nM T07663 CN7GR1 45272848 IC50 = 1.995 nM T07663 C8RZ7H 45272849 IC50 = 2.692 nM T07663 CQ34VM 45272857 IC50 = 3 nM T07663 C5H9RX 45272874 IC50 = 22.4 nM T07663 C7X2VE 45272888 IC50 = 0.9 nM T07663 CN8G9K 45272901 IC50 = 26.7 nM T07663 C2MW1C 45272908 IC50 = 25 nM T07663 C3X7RV 45273795 IC50 = 1.288 nM T07663 C74IXB 45273827 IC50 = 0.3 nM T07663 CLZ39M 45379958 IC50 = 2.38 nM T07663 C98KFA 45486490 IC50 = 1.17 nM T07663 CGA65L 45486496 IC50 = 0.17 nM T07663 CZ8JD0 45486497 IC50 = 0.28 nM T07663 CYF73X 45486498 IC50 = 0.38 nM T07663 C86XSZ 45486501 IC50 = 0.55 nM T07663 CDYO49 45486504 IC50 = 0.06 nM T07663 CNW0I9 45486505 IC50 = 0.71 nM T07663 CWQ6Y5 45486511 IC50 = 16.3 nM T07663 CSG37U 45486513 IC50 = 2.59 nM T07663 CEX01M 45486514 IC50 = 0.32 nM T07663 C58IWJ 45486519 IC50 = 0.25 nM T07663 CE3PK0 45486527 IC50 = 0.68 nM T07663 C1ZYT9 45486549 IC50 = 2.95 nM T07663 CHE56F 45486550 IC50 = 0.34 nM T07663 C84NHX 45486564 IC50 = 0.54 nM T07663 CLMZ68 45486571 IC50 = 4 nM T07663 CB2MG1 45486572 IC50 = 0.32 nM T07663 C0MWV4 45486574 IC50 = 0.88 nM T07663 C9SI3E 45486581 IC50 = 0.36 nM T07663 C51CUF 46193118 IC50 = 640 nM T07663 CTP8R1 46193119 IC50 = 38 nM T07663 CDT4U1 46193239 IC50 = 29000 nM T07663 C0W3LE 46193243 IC50 = 100 nM T07663 CKUN01 46193244 IC50 = 88000 nM T07663 CHU8I7 46193370 IC50 = 2800 nM T07663 C7NC9V 46193371 IC50 = 60 nM T07663 CY49DB 46193372 IC50 = 320 nM T07663 CN05XT 46193373 IC50 = 41000 nM T07663 C1Q6WV 46193374 IC50 = 32000 nM T07663 C60KFT 46193375 IC50 = 50 nM T07663 C2J9IH 46193486 IC50 = 260 nM T07663 CJ86KO 46193489 IC50 = 50 nM T07663 CPYK94 46193490 IC50 = 3400 nM T07663 CHUN05 46193595 IC50 = 40 nM T07663 C5IMB2 46239424 Ki = 6400 nM T07663 CKR9P7 46239425 Ki = 8900 nM T07663 C7SLP0 46239531 Ki = 5000 nM T07663 CI1F5C 46239840 Ki > 100000 nM T07663 C26XVS 46240044 Ki = 17324 nM T07663 CC3UF9 46830325 IC50 = 0.15 nM T07663 CE4JU7 46842025 IC50 = 0.27 nM T07663 CR8JC2 46842169 IC50 = 0.27 nM T07663 CF23CG 46842171 IC50 = 0.27 nM T07663 CWY45O 46842322 IC50 = 4.1 nM T07663 CY9UB1 46842324 IC50 = 0.27 nM T07663 CVP3F6 46886964 IC50 = 0.94 nM T07663 CF49HM 46886965 IC50 = 3.92 nM T07663 CQ91ZP 46887034 IC50 = 2.96 nM T07663 CDI09L 46887035 IC50 = 0.38 nM T07663 C8X6IR 46887483 IC50 = 0.3 nM T07663 C51BJT 46887484 IC50 = 0.86 nM T07663 CB3F2M 46887522 IC50 = 1.84 nM T07663 CVX57Z 46887568 IC50 = 3.28 nM T07663 C3GW8T 46887569 IC50 = 9.79 nM T07663 C13VUK 46888519 IC50 = 0.07 nM T07663 C7G5PM 46888541 IC50 = 0.66 nM T07663 C6NIG0 46888542 IC50 = 1.4 nM T07663 CPM4S1 46888559 IC50 = 5.5 nM T07663 CV53IU 46888560 IC50 = 0.89 nM T07663 C9UY1R 46888576 IC50 = 2.5 nM T07663 CE79JU 46888577 IC50 = 1.2 nM T07663 CQ5B2F 46888578 IC50 = 2.3 nM T07663 C8ITU7 46888595 IC50 = 0.2 nM T07663 C0IQ2C 46888596 IC50 = 2 nM T07663 CS6F1J 46888597 IC50 = 0.087 nM T07663 C7B3ZY 46888631 IC50 = 0.42 nM T07663 C8FW5K 46888632 IC50 = 2.3 nM T07663 C57KWS 46888633 IC50 = 0.35 nM T07663 CS27GK 46888659 IC50 = 0.011 nM T07663 C38INP 46888660 IC50 = 0.07 nM T07663 C6WQ5Y 46888661 IC50 = 1.2 nM T07663 CZ3SO4 46888707 IC50 = 0.19 nM T07663 C02RDT 46888708 IC50 = 0.08 nM T07663 CUN72Y 46888738 IC50 = 0.05 nM T07663 C3P2IN 46933992 IC50 = 11000 nM T07663 CHA5Z0 49821469 IC50 > 1000 nM T07663 C1AYP0 49821627 IC50 > 500 nM T07663 C85AXR 49821714 IC50 > 1000 nM T07663 CZS03D 50902030 Ki > 4274 nM T07663 CH2Z1E 50902289 Ki > 7100 nM T07663 C4HJL2 50902291 Ki > 7950 nM T07663 C6A1IU 50902549 Ki > 2000 nM T07663 C3Y2AV 50903255 Ki > 2000 nM T07663 CN41YJ 50925469 IC50 = 2 nM T07663 CQ3RG5 50925470 IC50 = 7 nM T07663 C2E5JK 50940516 IC50 = 850 nM T07663 CEB5T9 50940517 IC50 = 50 nM T07663 C2C0IA 50940656 IC50 = 850 nM T07663 C4I9OJ 50940659 IC50 = 8750 nM T07663 C6F5RK 50940660 IC50 = 300 nM T07663 C9O4LE 50940680 IC50 = 590 nM T07663 CT3H4X 50940682 IC50 = 4140 nM T07663 CN4S0D 50940686 IC50 = 2310 nM T07663 CT8V2L 50940687 IC50 = 12 nM T07663 CP3G6K 50940690 IC50 = 2300 nM T07663 C7MV1Y 50940692 IC50 = 380 nM T07663 CUM0O5 50940699 IC50 = 730 nM T07663 C9IFA6 50940700 IC50 = 50 nM T07663 C7TF6Q 50940701 IC50 = 1200 nM T07663 CI3AG0 50941259 IC50 = 260 nM T07663 CCUK19 50941260 IC50 = 990 nM T07663 CY37HL 50941261 IC50 = 10 nM T07663 CC0QW5 50941262 IC50 = 1340 nM T07663 C5Q9YU 50941264 IC50 = 3300 nM T07663 C7Y8HK 50941365 IC50 = 270 nM T07663 C8WQX5 50941366 IC50 = 1110 nM T07663 C3NK7Q 50941367 IC50 = 4460 nM T07663 C3QEV9 50941368 IC50 = 290 nM T07663 CA3HQ6 50941461 IC50 = 2040 nM T07663 C8LSY4 50941462 IC50 = 190 nM T07663 C4GBV9 50941463 IC50 = 1260 nM T07663 CYL8N5 50941464 IC50 = 1350 nM T07663 C10WDU 50941465 IC50 = 260 nM T07663 C6YM0P 50941551 IC50 = 1270 nM T07663 C6R4YN 50993785 IC50 = 10000 nM T07663 C0M6XL 50993786 IC50 = 10000 nM T07663 C0OR7K 53248667 IC50 > 100000 nM T07663 CS3R1I 53248669 IC50 = 28900 nM T07663 C30RNE 53248670 IC50 = 6400 nM T07663 C1RJ7M 54580520 IC50 > 400000 nM T07663 CCXF36 54580521 IC50 = 145000 nM T07663 CZG36N 54580522 IC50 > 400000 nM T07663 C0NPM8 54580523 IC50 = 225000 nM T07663 C25VSX 54580524 IC50 > 400000 nM T07663 CBT56Y 54581676 IC50 = 5200 nM T07663 C0MN3D 54582527 IC50 = 156000 nM T07663 C6T1QX 54582528 IC50 = 350000 nM T07663 CP4N1Q 54582529 IC50 > 400000 nM T07663 CW1X3G 54583497 IC50 > 400000 nM T07663 CN96IQ 54585432 IC50 > 400000 nM T07663 CH25CO 54586393 IC50 > 400000 nM T07663 C82LED 54586394 IC50 > 400000 nM T07663 CQ1H3C 54587403 IC50 > 400000 nM T07663 C28GAC 54587404 IC50 > 400000 nM T07663 CFX89L 54587804 IC50 = 5700 nM T07663 CGF65A 54670110 IC50 > 30000 nM T07663 C90ZLC 54670399 IC50 > 30000 nM T07663 CLK61N 56587955 IC50 = 0.1 nM T07663 C4TGL7 56648496 IC50 > 1000 nM T07663 CH6C3L 56648679 IC50 > 10000 nM T07663 CCY79V 56648680 IC50 = 3110 nM T07663 CNE96P 56648857 IC50 > 10000 nM T07663 CX86AQ 56648859 IC50 > 1000 nM T07663 CPC3T4 56654131 IC50 > 10000 nM T07663 C0YD3P 56928304 IC50 > 5000 nM T07663 C8RO6A 56929788 IC50 > 1000 nM T07663 CD52CA 57391118 IC50 = 0.02 nM T07663 C7Y4BX 57391119 IC50 = 1.47 nM T07663 C4PSK2 57391120 IC50 = 0.04 nM T07663 CA1TE7 57391121 IC50 = 0.01 nM T07663 CN60KE 57391196 IC50 = 0.09 nM T07663 CM7N8I 57391197 IC50 = 0.05 nM T07663 C7VXN9 57391198 IC50 = 1.3 nM T07663 C7SC4E 57392888 IC50 = 0.44 nM T07663 CG3DF1 57392948 Ki > 10000 nM T07663 CQT1G9 57392966 IC50 = 1.38 nM T07663 CR28IN 57394623 IC50 = 0.38 nM T07663 CHZ67R 57394624 IC50 = 0.27 nM T07663 CE36TV 57394695 Ki = 24400 nM T07663 CLEY35 57396379 IC50 = 0.64 nM T07663 C7W6TP 57396380 IC50 = 0.05 nM T07663 C80CVX 57396381 IC50 = 0.01 nM T07663 C86YCU 57396469 IC50 = 0.1 nM T07663 C3M6EL 57396470 IC50 = 1.64 nM T07663 CPQ91V 57396471 IC50 = 0.22 nM T07663 CP0AB6 57396472 IC50 = 0.28 nM T07663 CNY5Z8 57398261 IC50 = 0.35 nM T07663 CH57NZ 57398879 IC50 = 15.8 nM T07663 CTYR07 57399826 IC50 = 0.04 nM T07663 CL5UP7 57401597 IC50 = 0.36 nM T07663 C37KMA 57401598 IC50 = 0.13 nM T07663 CHQ79W 57401599 IC50 = 0.02 nM T07663 CWG70K 57401600 IC50 = 0.06 nM T07663 CU5KP3 57401601 IC50 = 0.1 nM T07663 C8GD5N 57402376 IC50 = 8.2 nM T07663 CLU6J0 57403348 IC50 = 2.43 nM T07663 CD73NJ 57403349 IC50 = 0.02 nM T07663 CPA3D1 57403394 Ki = 20800 nM T07663 CEN5Z8 57403417 IC50 = 0.08 nM T07663 CY75FP 57403418 IC50 = 0.05 nM T07663 CA4KZ8 57403419 IC50 = 1.31 nM T07663 C4XMB6 58547809 IC50 > 30000 nM T07663 CEB3G9 58547814 IC50 > 30000 nM T07663 C08QVG 58547833 IC50 > 30000 nM T07663 CFVG67 58547863 IC50 > 30000 nM T07663 CYZA38 58548077 IC50 > 30000 nM T07663 CN57ZH 67426178 IC50 > 10000 nM T07663 CO8C0Z 67453423 IC50 > 2000 nM T07663 CY8J3O 68181896 IC50 = 26000 nM T07663 CUGH78 68654838 IC50 = 1000 nM T07663 CH2X0Z 69394992 IC50 = 2.884 nM T07663 CC43LF 71074083 IC50 = 437 nM T07663 C4P0XT 71092344 IC50 = 4610 nM T07663 C6DAG4 71092519 IC50 = 13900 nM T07663 C2HGI7 71153408 IC50 > 10000 nM T07663 C9GR3L 71153436 IC50 > 10000 nM T07663 CHLQ31 71530755 IC50 = 160 nM T07663 CN8KP5 71575273 IC50 = 0.27 nM T07663 C4GNJ3 71598545 IC50 > 1000 nM T07663 C0M9IA 71666277 IC50 = 21.6 nM T07663 C3O9KX 71666278 IC50 = 0.59 nM T07663 CU0M5P 71666433 IC50 = 0.19 nM T07663 CZC74T 71666437 IC50 = 1.55 nM T07663 C68SDB 71719394 IC50 = 1995.26 nM T07663 CF2W4Z 71738037 IC50 = 240 nM T07663 C95QWN 71765666 IC50 = 17 nM T07663 CZ0G2X 72165213 IC50 > 10000 nM T07663 C7XRY6 72190879 IC50 > 30000 nM T07663 CQ3GD7 72704434 Ki = 630 nM T07663 C9JE6M 75815419 IC50 = 54.3 nM T07663 C65ZBN 76323083 IC50 = 537.03 nM T07663 CZ3P5K 89706867 IC50 = 0.056 nM T07663 CF03DW 90168772 IC50 > 20000 nM T07663 CM6J9K 90168778 IC50 > 20000 nM T07663 C45QVJ 91668196 IC50 = 2300 nM T07663 C1JPD6 91844700 IC50 = 5400 nM T07663 CYQV05 92471958 IC50 = 410 nM T07663 C6TD3W 117685212 IC50 = 337 nM T07663 CVUC27 117685328 IC50 = 1.5 nM T07663 C71BEL 117824219 IC50 = 1.7 nM T07663 CFAG87 117824250 IC50 = 0.059 nM T07663 C62NZT 117824353 IC50 = 64 nM T07663 C3WT5R 117824368 IC50 = 0.29 nM T07663 CGH1Z4 117824420 IC50 = 333 nM T07663 CX12RS 117824489 IC50 = 3.8 nM T07663 CS97IT 117830474 IC50 = 45.2 nM T07663 C60ADH 117830507 IC50 = 57 nM T07663 CMJR74 117830513 IC50 = 0.32 nM T07663 CSCY01 117949009 IC50 = 9800 nM T07663 CYQ74R 118479645 IC50 > 10000 nM T07663 CVYK24 118556943 IC50 > 50000 nM T07663 CM6XW1 118724093 IC50 = 520 nM T07663 C46LFG 118724094 IC50 > 10000 nM T07663 CYM21X 118724095 IC50 = 2900 nM T07663 C4HI1Q 118729758 IC50 = 3000 nM T07663 CKBG19 118729759 IC50 = 3100 nM T07663 C8LRQ7 121370930 IC50 = 110 nM T07663 CRJE23 122185011 IC50 > 30000 nM T07663 CS6M9C 122193679 IC50 > 100000 nM T07663 CVX7U9 127029185 IC50 = 3810 nM T07663 C9OVF8 127029366 IC50 = 5.2 nM T07663 C4UR7D 127038167 IC50 > 1000 nM T07663 C4H2TJ 127038168 IC50 > 1000 nM T07663 CL9JT8 127038169 IC50 = 606 nM T07663 CJPX60 127038509 IC50 = 232 nM T07663 C26EAG 127038511 IC50 = 201 nM T07663 CTM9E4 127038512 IC50 = 279 nM T07663 C6AQ2U 127038513 IC50 = 195 nM T07663 CV1FM0 127038868 IC50 = 228 nM T07663 CADU23 127038869 IC50 = 91.6 nM T07663 CACJ46 132489333 IC50 = 5.6 nM T07663 C2P1IU 134129996 IC50 > 100000 nM T07663 CLE03O 134130328 IC50 > 100000 nM T07663 CSN6J0 134130563 IC50 > 100000 nM T07663 C0A1CZ 134131162 IC50 > 100000 nM T07663 C23CYE 134814217 IC50 = 1.41 nM T07663 CHX5W7 134908214 IC50 = 91200 nM T07663 C1QMI8 135401477 IC50 = 26.92 nM T07663 C1BA7R 135406502 IC50 = 2 nM T07663 CIC0M9 135406542 IC50 = 3 nM T07663 CL6W5K 135406554 IC50 = 5.3 nM T07663 CL6YK2 135406621 IC50 = 1.1 nM T07663 C1LG3R 135406622 IC50 = 27 nM T07663 C9S5CV 135406637 IC50 = 1.4 nM T07663 C17YXR 135406983 IC50 = 5 nM T07663 C41TDB 135413523 IC50 = 3.5 nM T07663 C5JYM4 135415122 IC50 = 3 nM T07663 CN7LX8 135415142 IC50 = 1.5 nM T07663 CJG93Q 135415214 IC50 = 3.2 nM T07663 CQOL86 135417284 IC50 = 30 nM T07663 CG96MZ 135419216 IC50 = 2 nM T07663 COD5W1 135419220 IC50 = 2000 nM T07663 CBA1Q7 135419269 IC50 = 5 nM T07663 CP4HN6 135419318 IC50 = 7 nM T07663 CCXB28 135419329 IC50 = 2 nM T07663 CL8U1V 135419421 IC50 = 3.5 nM T07663 CN1CE4 135423930 IC50 = 2 nM T07663 C1GPZ3 135423938 IC50 = 0.2 nM T07663 C7A2NS 135427992 IC50 = 7.1 nM T07663 C6UFD4 135430871 IC50 = 10 nM T07663 C1Z3WH 135430893 IC50 = 8 nM T07663 CAJU63 135430952 IC50 = 50 nM T07663 CNP87H 135433645 IC50 = 330 nM T07663 C2DAG7 135433829 IC50 = 50 nM T07663 CHD03R 135433867 IC50 = 80 nM T07663 CJ0B6N 135438524 IC50 = 9.5 nM T07663 CJ9IE8 135438525 IC50 = 21 nM T07663 C94RVJ 135438569 IC50 = 0.7 nM T07663 C1A4MY 135439488 IC50 = 100 nM T07663 C0IE4A 135443738 IC50 = 200 nM T07663 C5U1NW 135444771 IC50 = 0.48 nM T07663 CF1U2Y 135451848 IC50 = 0.52 nM T07663 C0DBS7 135452901 IC50 = 1.905 nM T07663 CFKO84 135455980 IC50 = 5.7 nM T07663 CQW8U9 135456038 IC50 = 1 nM T07663 C9LD5N 135456042 IC50 = 2.089 nM T07663 C0BQH8 135456061 IC50 = 10 nM T07663 CA83SQ 135456100 IC50 = 1 nM T07663 C4ZQ1W 135456180 IC50 = 1.3 nM T07663 CM1K9A 135456702 IC50 = 150 nM T07663 C3R8SE 135457869 IC50 = 5200 nM T07663 C6TO5S 135462289 IC50 = 4 nM T07663 CUX8S3 135462319 IC50 = 70 nM T07663 C7HC3R 135462338 IC50 = 2.5 nM T07663 CA8X3R 135462413 IC50 = 1.7 nM T07663 CY3A0S 135462886 IC50 = 2.89 nM T07663 CA9V7D 135463722 IC50 = 10 nM T07663 C4C3JV 135467743 IC50 = 6 nM T07663 CTN73W 135467948 IC50 = 1 nM T07663 CHSI34 135469671 IC50 = 10 nM T07663 CAR9X0 135474505 IC50 = 0.62 nM T07663 CADL53 135475879 IC50 = 40 nM T07663 C3IT7F 135477808 IC50 = 13 nM T07663 C9E5KR 135480166 IC50 = 20 nM T07663 CZ9HT7 135480403 IC50 = 1.7 nM T07663 CJS37E 135482260 IC50 > 101000 nM T07663 CUNL35 135484025 IC50 = 10 nM T07663 C95GLJ 135484081 IC50 = 0.69 nM T07663 CVTR78 135484097 IC50 = 1.04 nM T07663 CKP9T0 135485820 IC50 = 5.3 nM T07663 CUV8L0 135485839 IC50 = 1.1 nM T07663 C23SWA 135485841 IC50 = 1.6 nM T07663 C4ILF7 135487662 IC50 = 1.7 nM T07663 CEHK47 135487696 IC50 = 2.6 nM T07663 CEZ5P3 135487732 IC50 = 5 nM T07663 C18DSI 135489339 IC50 = 34 nM T07663 CHO1Z5 135489408 IC50 = 7 nM T07663 CBW5A9 135491781 IC50 = 3.6 nM T07663 CG82XZ 135491934 IC50 = 18.2 nM T07663 CMNE87 135491938 IC50 = 8.2 nM T07663 CLFQ43 135493551 IC50 = 3 nM T07663 C8L1NK 135494369 IC50 = 3 nM T07663 C7FM8V 135494393 IC50 = 2 nM T07663 C3D4IY 135496441 IC50 = 3 nM T07663 C2MTZ8 135497265 IC50 = 2 nM T07663 CS4NM0 135501101 IC50 = 2 nM T07663 CJ3XM0 135503009 IC50 = 14.7 nM T07663 C86THJ 135503803 IC50 = 1 nM T07663 CN4BY1 135503843 IC50 = 2 nM T07663 C7BM8D 135504134 IC50 = 70 nM T07663 CK0S3E 135505670 IC50 = 0.9 nM T07663 C4ZNY0 135505809 IC50 = 7 nM T07663 C78CIT 135505815 IC50 = 12 nM T07663 CM27YS 135506900 IC50 = 40 nM T07663 CC87SI 135510018 IC50 = 53 nM T07663 CVM2R1 135513834 IC50 = 50 nM T07663 C6GNF4 135513951 IC50 = 0.1 nM T07663 CC9N6X 135513970 IC50 = 1 nM T07663 CL1W4B 135513981 IC50 = 5 nM T07663 CYS04P 135514690 IC50 = 0.9 nM T07663 C4NSC9 135515154 IC50 = 4 nM T07663 C9IU6B 135515212 IC50 = 2.5 nM T07663 CEV79B 135515565 IC50 = 5.5 nM T07663 C0STP6 135518654 IC50 = 2.5 nM T07663 CKDH83 135518785 IC50 = 0.2 nM T07663 C8VT4S 135520162 IC50 = 6.4 nM T07663 CKD97I 135520170 IC50 = 13 nM T07663 CL0HD1 135520500 IC50 = 18 nM T07663 C5EBI4 135525517 IC50 = 44 nM T07663 CD84SI 135528161 IC50 = 35 nM T07663 CYF17I 135528172 IC50 = 3.3 nM T07663 CB6H4I 135528567 IC50 = 13 nM T07663 C6KQV1 135528758 IC50 = 5 nM T07663 CFN34H 135528775 IC50 = 4 nM T07663 CLU8A5 135529022 IC50 = 1.53 nM T07663 C6YF2L 135529725 IC50 = 8 nM T07663 CJIA83 135529861 IC50 = 20 nM T07663 CTX70E 135530119 IC50 = 2.7 nM T07663 CCM89A 135530700 IC50 = 8.5 nM T07663 C43HNQ 135531347 IC50 = 1.1 nM T07663 CV34FU 135532825 IC50 = 5.2 nM T07663 CM3GD7 135532874 IC50 = 10 nM T07663 CGWS52 135532916 IC50 = 2.47 nM T07663 CEF96L 135536692 IC50 = 30 nM T07663 CKC9M0 135536718 IC50 = 40 nM T07663 C6E0BM 135536759 IC50 = 7 nM T07663 CWRQ95 135536783 IC50 = 4 nM T07663 C1Z7AY 135536802 IC50 = 0.8 nM T07663 CSO34W 135536977 IC50 = 0.78 nM T07663 CR0VL3 135543052 IC50 = 3.7 nM T07663 C45LHQ 135543089 IC50 = 2.76 nM T07663 CX4H6D 135544114 IC50 = 9.1 nM T07663 C4ASW0 135544141 IC50 = 0.6 nM T07663 CYE4C5 135544159 IC50 = 8 nM T07663 CW53FT 135545949 IC50 = 0.31 nM T07663 CK5F9W 135546517 IC50 = 1000 nM T07663 C9VKC6 135547908 IC50 = 10.8 nM T07663 C3HTJ7 135548164 IC50 = 3 nM T07663 C2CXY7 135559102 IC50 = 17 nM T07663 C8HW0M 135565273 IC50 = 8.9 nM T07663 C6J2FV 135566412 IC50 = 110 nM T07663 CHDC83 135566745 IC50 = 1.6 nM T07663 C5S7PD 135566746 IC50 > 1000 nM T07663 C3H1QO 135566795 IC50 = 18.2 nM T07663 CN1OH0 135566796 IC50 = 77 nM T07663 C9IJK1 135566935 IC50 = 90.6 nM T07663 C7M1TE 135604959 IC50 = 5 nM T07663 C6I3HM 135678134 IC50 = 20 nM T07663 CCB89G 135723513 IC50 = 20 nM T07663 CZP1J0 135731499 IC50 = 100 nM T07663 C7VBI4 135740146 IC50 = 82 nM T07663 CIQ83H 135744761 IC50 = 300 nM T07663 C97IUH 135750162 IC50 = 37000 nM T07663 CG1AN3 135790070 IC50 = 200 nM T07663 CD5J1S 135790088 IC50 = 1.76 nM T07663 C0M1LQ 135790105 IC50 = 0.31 nM T07663 CH13EW 135832627 IC50 = 4466.84 nM T07663 C31VFB 135832642 IC50 = 4400 nM T07663 C3PO9K 135856789 IC50 = 7560 nM T07663 C7KDO8 135874585 IC50 = 150 nM T07663 C51XVI 135874586 IC50 = 60 nM T07663 CWT6F3 135890114 IC50 = 5.8 nM T07663 C1EP3X 135890118 IC50 = 6.6 nM T07663 C25PUK 135890126 IC50 = 41 nM T07663 CI4DB0 135890131 IC50 = 4.5 nM T07663 CO07ZA 135890143 IC50 = 1.23 nM T07663 CBI80F 135890150 IC50 = 1.61 nM T07663 CQ8CT6 135890151 IC50 = 4 nM T07663 C8I2XR 135890178 IC50 = 1.01 nM T07663 CTX54Z 135896326 IC50 = 1500 nM T07663 CK4X2F 135898900 IC50 = 100 nM T07663 CPNJ62 135898901 IC50 = 50 nM T07663 C43ZKU 135898902 IC50 = 320 nM T07663 CSO02I 135898910 IC50 = 200 nM T07663 C30ZQG 135898911 IC50 = 510 nM T07663 CJQ74U 135898912 IC50 = 38 nM T07663 C4TRA9 135898925 IC50 = 70 nM T07663 CM2T5C 135898926 IC50 = 140 nM T07663 CH5R6Y 135898941 IC50 = 70 nM T07663 CYJ07O 135898942 IC50 = 530 nM T07663 CR30YL 135898943 IC50 = 500 nM T07663 C0MUP5 135898944 IC50 = 310 nM T07663 CT1H3Q 135898959 IC50 = 370 nM T07663 CU3MH0 135964375 IC50 = 381 nM T07663 CI46LV 135964379 IC50 = 1050 nM T07663 C61SDR 135964388 IC50 > 10000 nM T07663 C42FTR 135964389 IC50 = 116 nM T07663 CZ5UD9 135964390 IC50 = 710 nM T07663 CUQ41O 135964394 IC50 = 2100 nM T07663 C7NRJ6 135964396 IC50 = 849 nM T07663 CY6LT4 135964400 IC50 = 4870 nM T07663 C8UT0J 135964407 IC50 = 634 nM T07663 C04IQT 135964410 IC50 = 2160 nM T07663 C98BHJ 135964418 IC50 = 3340 nM T07663 CS4FT5 135964421 IC50 = 80 nM T07663 CO51CW 135964422 IC50 = 146 nM T07663 CC3HS1 135964423 IC50 = 15 nM T07663 C7KI6V 135964424 IC50 = 1330 nM T07663 C1WB6M 135964425 IC50 = 112 nM T07663 CKSO87 135964426 IC50 = 48 nM T07663 CY24DM 135964428 IC50 = 33 nM T07663 CMYW62 135964429 IC50 = 9 nM T07663 CPL92J 135964430 IC50 = 1570 nM T07663 CLX28E 135964433 IC50 = 38 nM T07663 C6D0FX 136026515 IC50 > 10000 nM T07663 CL7BE5 136032221 IC50 = 1.7 nM T07663 C9OQ5U 136032222 IC50 = 2.1 nM T07663 C6OU3Z 136034782 IC50 = 10 nM T07663 CWPB32 136034783 IC50 = 878 nM T07663 C3KCA0 136042216 IC50 = 0.69 nM T07663 CO4FS2 136042217 IC50 = 0.75 nM T07663 C5MCV8 136042218 IC50 = 2.44 nM T07663 C0EZ4B 136042219 IC50 = 0.74 nM T07663 CX1L3V 136042220 IC50 = 0.86 nM T07663 CS32WP 136042221 IC50 = 0.26 nM T07663 C21HJT 136042222 IC50 = 1.27 nM T07663 C4DP9X 136042223 IC50 = 1.83 nM T07663 CMH5B3 136042224 IC50 = 1.36 nM T07663 CMW86G 136042225 IC50 = 1.01 nM T07663 CJ5X4O 136042226 IC50 = 1.66 nM T07663 CM1TU5 136042227 IC50 = 4.35 nM T07663 C4A6JD 136043740 IC50 = 3.1 nM T07663 CS38OR 136044186 IC50 = 0.58 nM T07663 C6LT3U 136053630 IC50 = 0.29 nM T07663 C9OTF5 136053631 IC50 = 0.28 nM T07663 C5ZIU7 136056125 IC50 = 1000 nM T07663 C70DJG 136056126 IC50 = 2.1 nM T07663 C9Q3BW 136056127 IC50 = 81.28 nM T07663 C4U1SF 136056128 IC50 = 954.99 nM T07663 CI8E5F 136056129 IC50 = 780 nM T07663 CJ43ZC 136059652 IC50 = 3 nM T07663 CZT97J 136059653 IC50 = 77 nM T07663 C2DQ4L 136059654 IC50 = 100 nM T07663 CJ1TW7 136059659 IC50 = 80 nM T07663 CE75BO 136059660 IC50 = 100 nM T07663 C58IEH 136059684 IC50 = 1.1 nM T07663 CG6E8F 136059685 IC50 = 7.7 nM T07663 C97HLB 136059686 IC50 = 5.6 nM T07663 CZQ84P 136059687 IC50 = 0.62 nM T07663 CV6PU2 136059688 IC50 = 0.89 nM T07663 C12UMG 136059728 IC50 = 370 nM T07663 C6WH2S 136078534 IC50 = 10 nM T07663 CE51KZ 136079586 IC50 = 4 nM T07663 CRP24A 136087045 IC50 = 417 nM T07663 C7SUX4 136087050 IC50 = 141 nM T07663 C8UF7G 136087052 IC50 = 3300 nM T07663 C6U2FG 136104505 IC50 = 0.18 nM T07663 CB1GP4 136104506 IC50 = 0.28 nM T07663 CIC08H 136104509 IC50 = 0.41 nM T07663 C0LRM5 136104510 IC50 = 0.34 nM T07663 CNRF74 136104512 IC50 = 0.7 nM T07663 C5LXO8 136104513 IC50 = 0.32 nM T07663 C9UK1F 136132272 IC50 = 100 nM T07663 CBO5H3 136132273 IC50 = 50 nM T07663 CPY6I0 136132274 IC50 = 500 nM T07663 CDE2S8 136132275 IC50 = 300 nM T07663 CPL26N 136132276 IC50 = 1 nM T07663 C4ZBT6 136132277 IC50 = 300 nM T07663 CJ9QG1 136132278 IC50 = 5 nM T07663 C23BTX 136132279 IC50 = 20 nM T07663 C1BFD5 136132280 IC50 = 40 nM T07663 C21FVA 136180322 IC50 = 1.5 nM T07663 C41CAD 136180323 IC50 = 1.7 nM T07663 CC42DB 136180324 IC50 = 1.9 nM T07663 CGJX71 136180325 IC50 = 3.4 nM T07663 C0W3NC 136180326 IC50 = 3.9 nM T07663 CYC9Z6 136180327 IC50 = 12 nM T07663 C5EJ0K 136180328 IC50 = 32 nM T07663 CZ1JH2 136180329 IC50 = 14 nM T07663 C9OM5D 136180330 IC50 = 2.6 nM T07663 CMF1V6 136180331 IC50 = 1.6 nM T07663 C01TYU 136180332 IC50 = 16 nM T07663 CXT68L 136180333 IC50 = 13 nM T07663 CY0T8W 136180334 IC50 = 3.3 nM T07663 C1WHX6 136197281 IC50 = 0.83 nM T07663 CQW7T0 136197286 IC50 = 0.62 nM T07663 CPA8E7 136197297 IC50 = 1.21 nM T07663 CS8TV5 136197304 IC50 = 1.7 nM T07663 COTY62 136197323 IC50 = 8.8 nM T07663 C5HIL8 136197357 IC50 = 9.6 nM T07663 CE0F5T 136197398 IC50 = 1.46 nM T07663 CK2FL9 136197415 IC50 = 5.33 nM T07663 CS16YF 136197417 IC50 = 1.86 nM T07663 CN0G6U 136197445 IC50 = 0.92 nM T07663 C8TQ7A 136217455 IC50 = 3300 nM T07663 C4JCZ7 136219297 IC50 = 272 nM T07663 CE32YG 136219298 IC50 = 21.3 nM T07663 CXOM76 136236320 IC50 = 12.6 nM T07663 C65BFU 136236321 IC50 = 58 nM T07663 C96WPH 136236322 IC50 = 8.5 nM T07663 CY2NJ1 136236323 IC50 = 4.8 nM T07663 CUS40O 136236324 IC50 = 13.7 nM T07663 CS9Z1P 136236325 IC50 = 3 nM T07663 CRZ58U 136236326 IC50 = 4.8 nM T07663 C9PIO3 136236327 IC50 = 34.3 nM T07663 CSU3J2 136236328 IC50 = 7.2 nM T07663 C5KF0V 136236329 IC50 > 2000 nM T07663 CDNI42 136236330 IC50 = 312 nM T07663 CI0M5R 136236331 IC50 = 104 nM T07663 CF43SC 136236332 IC50 = 88 nM T07663 CMGK71 136236333 IC50 = 31.5 nM T07663 C9R6HE 136236334 IC50 = 65 nM T07663 C7ZU0K 136236335 IC50 = 71 nM T07663 C2BCV9 136236336 IC50 = 450 nM T07663 CO4S8B 136236337 IC50 > 2000 nM T07663 C6N2KA 136236338 IC50 = 12.5 nM T07663 CN69OZ 136239327 IC50 = 6.2 nM T07663 C63FEW 136239328 IC50 = 29.3 nM T07663 CQZR23 136244112 IC50 = 48 nM T07663 CO9M4H 136244113 IC50 = 10.2 nM T07663 CK6GB7 136244114 IC50 = 74 nM T07663 CF5BV2 136244123 IC50 = 25.5 nM T07663 C5VT4W 136244124 IC50 = 11.1 nM T07663 CZD04T 136244125 IC50 = 2.8 nM T07663 CUQA38 136244132 IC50 = 17.4 nM T07663 CILG36 136286746 IC50 = 3 nM T07663 C39WRP 136286747 IC50 = 3 nM T07663 C7ZX5O 136286761 IC50 = 48 nM T07663 C9SV6G 136645392 IC50 = 65 nM T07663 CANQ56 136645396 IC50 = 53 nM T07663 C9TGH1 136645397 IC50 = 14 nM T07663 C1F7JV 136645401 IC50 = 144 nM T07663 C32LNQ 136645404 IC50 = 149 nM T07663 C4W0IE 136645405 IC50 = 27 nM T07663 CMIU28 136645406 IC50 = 40 nM T07663 C3K2WL 136645410 IC50 = 79 nM T07663 CC1D0X 136645415 IC50 = 20 nM T07663 C02RIK 136645417 IC50 = 12 nM T07663 C8CT0Z 136645422 IC50 = 20 nM T07663 CAWT82 136645431 IC50 = 10 nM T07663 CBZ8Q1 136645433 IC50 = 22 nM T07663 C21EJD 136645435 IC50 = 2 nM T07663 C1KTV3 136645436 IC50 = 36 nM T07663 CK1B9W 136645438 IC50 = 1 nM T07663 C6QOP7 136645441 IC50 = 7 nM T07663 CMZ71T 136645444 IC50 = 10 nM T07663 CL47WS 136645445 IC50 = 3 nM T07663 C64BZR 136645447 IC50 = 44 nM T07663 C7X1UL 136645449 IC50 = 5 nM T07663 CI9ZO7 136645454 IC50 = 13 nM T07663 CA3I8S 136645455 IC50 = 2 nM T07663 CRN16W 136645457 IC50 = 1 nM T07663 CGQ92L 136645458 IC50 = 2 nM T07663 CO5DN2 136645462 IC50 = 2 nM T07663 CRPN39 136645466 IC50 = 11 nM T07663 CL5X3G 136645467 IC50 = 3 nM T07663 C48HNY 136959539 IC50 = 74 nM T07663 C1P8ZW 136959550 IC50 = 5 nM T07663 CKU95F 136966187 IC50 = 17 nM T07663 CFRG19 136985286 IC50 = 15 nM T07663 CE7F4O 136985287 IC50 = 10 nM T07663 CFPT21 136985288 IC50 = 0.5 nM T07663 CBH5Y0 136985291 IC50 = 24 nM T07663 CDAK28 136985292 IC50 = 0.6 nM T07663 CQ9XW7 136985295 IC50 = 122 nM T07663 C1M6NW 136985296 IC50 = 31 nM T07663 CJOA28 136985302 IC50 = 3 nM T07663 C8HG0E 137051684 IC50 = 2.02 nM T07663 CANS59 137136982 IC50 = 47 nM T07663 C5AE3Q 137283418 IC50 = 19 nM T07663 C0KM1X 137288419 IC50 = 2439 nM T07663 C5QIX1 137289788 IC50 = 17 nM T07663 C5X0YR 137289866 IC50 = 7 nM T07663 CU70ZB 137289868 IC50 = 207 nM T07663 CV6AN7 137289892 IC50 = 57 nM T07663 CB14CI 137289900 IC50 = 5 nM T07663 CLY69S 137289946 IC50 = 13 nM T07663 CC5HA4 137290225 IC50 = 121 nM T07663 C4RBC7 137290234 IC50 = 4 nM T07663 CKJ6Q4 137290238 IC50 = 46 nM T07663 CR53GQ 137290273 IC50 = 34 nM T07663 C8DYG6 137290344 IC50 = 13 nM T07663 C9G3JB 137292402 IC50 = 7 nM T07663 C6MXL3 137292504 IC50 = 57 nM T07663 CAZ49O 137300702 IC50 = 4 nM T07663 CGE0J6 137300703 IC50 = 165 nM T07663 CDU43L 137300704 IC50 = 11 nM T07663 CK0QG6 137300705 IC50 = 303 nM T07663 C91IPL 137300706 IC50 = 70 nM T07663 C5UYP8 137300707 IC50 = 5 nM T07663 CHSG63 137300708 IC50 = 23 nM T07663 CX57MR 137300709 IC50 = 39 nM T07663 C54KGS 137300710 IC50 = 10 nM T07663 CQD07Z 137300711 IC50 = 20 nM T07663 C3I1CB 137300712 IC50 = 38 nM T07663 C2N9VT 137348687 IC50 > 10000 nM T07663 C14DWB 137631637 IC50 = 157510 nM T07663 CML1E3 137631792 IC50 > 100 nM T07663 CA92EX 137632005 IC50 = 31 nM T07663 C5HM3W 137632322 IC50 = 17600 nM T07663 C0SGD8 137633727 IC50 = 77 nM T07663 CTRF70 137634642 IC50 > 100 nM T07663 CO7J5T 137635211 IC50 > 100 nM T07663 CF6EZ1 137635781 IC50 > 1000000 nM T07663 CKB51U 137637339 IC50 = 100000 nM T07663 CU17GD 137637935 IC50 = 5.4 nM T07663 C8RG2S 137638853 IC50 > 100 nM T07663 CA3BX6 137639488 IC50 > 100 nM T07663 C49UCG 137642312 IC50 > 100 nM T07663 C8R1GD 137644106 IC50 > 100 nM T07663 CSQ7P5 137644148 IC50 = 16 nM T07663 CM57EI 137646989 IC50 = 3.1 nM T07663 CPLM78 137647044 IC50 = 56 nM T07663 C18JOP 137647693 IC50 = 30 nM T07663 C4V8QP 137648482 IC50 = 50000 nM T07663 CSW42J 137651273 IC50 = 50 nM T07663 CH6EC3 137653604 IC50 > 100 nM T07663 CPK1J0 137654639 IC50 > 100 nM T07663 C93WRT 137655765 IC50 > 100 nM T07663 CDQ8B5 137657724 IC50 > 100 nM T07663 CY57JX 137658794 IC50 = 21 nM T07663 C2ITK1 137660715 IC50 > 100 nM T07663 CJA7I0 137662139 IC50 = 100000 nM T07663 C6KYD7 137700754 IC50 = 4010 nM T07663 CM3UF7 137700779 IC50 > 20000 nM T07663 CPTE92 138319693 IC50 = 0.32 nM T07663 C2QLX3 138393292 IC50 > 5000 nM T07663 CF3B2O 141492937 IC50 = 0.52 nM T07663 CEK54I 141492938 IC50 = 1.2 nM T07663 CMJW70 141492939 IC50 = 3.28 nM T07663 CKB05G 141492943 IC50 = 0.53 nM T07663 CU6A0R 141492944 IC50 = 2.85 nM T07663 CW7NV6 141492945 IC50 = 0.6 nM T07663 C2NW6Y 141492955 IC50 = 0.67 nM T07663 C13PVI 141492968 IC50 = 0.6 nM T07663 C42GOU 141492970 IC50 = 26.9 nM T07663 CGNK49 141492971 IC50 = 0.82 nM T07663 CXN3U7 141492981 IC50 = 86 nM T07663 CZ0M1Y 141492988 IC50 = 1.25 nM T07663 C2T8GE 141492992 IC50 = 6.45 nM T07663 C5XTB1 141492998 IC50 = 2.5 nM T07663 C93ZIQ 141492999 IC50 = 0.39 nM T07663 CUXZ06 141493000 IC50 = 0.97 nM T07663 C7RTX9 141493002 IC50 = 3.14 nM T07663 CQV0B4 141737648 IC50 = 155 nM T07663 C0JV6Y 141737649 IC50 = 39.7 nM T07663 CSOF52 141737655 IC50 = 19.9 nM T07663 C7SRA2 141737657 IC50 = 7.02 nM T07663 CE1H7F 141737660 IC50 = 97.5 nM T07663 CA5UL8 141737663 IC50 = 61 nM T07663 C6ZA7D 141737664 IC50 = 36.9 nM T07663 CMIY07 141737666 IC50 = 21.4 nM T07663 CC61SD 141737667 IC50 = 30.3 nM T07663 C14CZJ 141737668 IC50 = 8.44 nM T07663 CTNG49 141737674 IC50 = 36.4 nM T07663 CJ38IC 141737676 IC50 = 12.7 nM T07663 C1MC5Z 141737681 IC50 = 8.68 nM T07663 CK34HF 141737682 IC50 = 50.2 nM T07663 CQCM72 141737683 IC50 = 177 nM T07663 C2MEL1 141737684 IC50 = 56.4 nM T07663 CTUL23 141737690 IC50 = 5.24 nM T07663 CMW20N 141737696 IC50 = 3.87 nM T07663 CZWD98 141737697 IC50 = 80.2 nM T07663 C7GBH6 141737698 IC50 = 52.5 nM T07663 CVQJ85 141737699 IC50 = 383 nM T07663 CO1C4S 141737703 IC50 = 27.6 nM T07663 CX9N1P 141737704 IC50 = 10.5 nM T07663 C8HEG7 141737705 IC50 = 2.92 nM T07663 C8OWX3 145964082 IC50 = 2.64 nM T07663 C0P7CN 145964738 IC50 = 3.04 nM T07663 CZ1M5C 145964966 IC50 = 1.58 nM T07663 C07GTQ 145966108 IC50 = 0.79 nM T07663 C38QXR 145966233 IC50 = 251.19 nM T07663 CUM0Y5 145968257 IC50 = 6.82 nM T07663 CO4N2T 145968939 IC50 = 2.09 nM T07663 CDHG23 145971317 IC50 = 9.63 nM T07663 CMNV65 145973708 IC50 = 1.05 nM T07663 CC7HN2 145974174 IC50 > 100000 nM T07663 CIFW03 145974279 IC50 = 0.52 nM T07663 CWM49T 145974605 IC50 = 1.63 nM T07663 C2JF3R 145974856 IC50 = 2.64 nM T07663 C8BEH3 145975382 IC50 = 2.38 nM T07663 C5C6NR 145976885 IC50 = 2.37 nM T07663 CTJ6L8 145977069 IC50 = 0.39 nM T07663 C6M5ZW 145977440 IC50 = 19.95 nM T07663 CDB1E7 145977898 IC50 = 4.38 nM T07663 CK1BR0 145978345 IC50 > 100000 nM T07663 CJD7B2 145978603 IC50 = 4.03 nM T07663 CU5VD3 145978669 IC50 = 3.82 nM T07663 C9LGT4 145979889 IC50 = 235 nM T07663 CKZ1Y6 145979895 IC50 = 170 nM T07663 C50DFR 145982956 Ki = 8 nM T07663 CKTF58 145987769 IC50 = 227 nM T07663 CJA1B0 145991631 IC50 = 81.2 nM T07663 CHJ79V 145997874 IC50 = 3390 nM T07663 CM7TX2 148279038 IC50 = 1530 nM T07663 CYPW78 155510908 IC50 = 1.55 nM T07663 C6VZ5O 155514730 IC50 = 1.69 nM T07663 CL8CU6 155521936 IC50 > 200000 nM T07663 CAUO07 155524955 IC50 = 0.54 nM T07663 CT85RG 155530589 IC50 > 200000 nM T07663 CXMU51 155537188 IC50 = 0.79 nM T07663 C1IP4D 155556194 IC50 = 3.9 nM T07663 C2DA1W 155561694 IC50 > 500000 nM T07663 CQ2R0W 155568588 IC50 > 500000 nM T07663 CV07RN 44579973 IC50 = 0.6166 nM T07663 D00REK 5712 IC50 = 31900 nM T07663 D01RLF 105078 IC50 = 794.33 nM T07663 D01TOR 667555 IC50 = 450 nM T07663 D02NWF 2573787 IC50 = 720 nM T07663 D02VRN 6442679 IC50 = 1470 nM T07663 D03BWH 44587253 IC50 = 360 nM T07663 D06NIT 135564899 IC50 = 349 nM T07663 D06TLQ 5488822 IC50 = 1700 nM T07663 D09AUL 10266864 IC50 = 260 nM T07663 D09RKU 46239428 Ki = 9700 nM T07663 D09WUP 25058047 IC50 = 74 nM T07663 D0I6XA 149784 Ki > 200000 nM T07663 D0J0CB 2753 IC50 = 7150 nM T07663 D0J7GF 780643 IC50 = 320 nM T07663 D0O3QI 10356247 IC50 = 4200 nM T07663 D0R6MT 3758 IC50 = 63000 nM T07663 D0S8AV 509245 IC50 = 16230 nM T07663 D0U8YQ 921562 IC50 = 310 nM T07663 D0V1CL 37015 IC50 = 180 nM T07663 D0V4WB 149790 IC50 > 16000 nM T07663 D0W2BI 9799499 IC50 = 700 nM T07663 D0X7SR 10246505 IC50 = 1290 nM T07663 D0YZ0L 44605341 IC50 = 12600 nM T61657 D02DGU 444795 Ki = 0.4 nM T61657 D0BM5G 5381 EC50 = 0.8 nM T61657 D0G3PI 449171 Ki = 0.5 nM T61657 D0JC9N 60164 EC50 = 2 nM T61657 D0N0RU 82146 Ki = 50 nM T61657 D02GTY 108143 Ki = 30 nM T61657 D06FOU 11518241 EC50 = 125 nM T61657 D06QXI 9863342 EC50 = 340 nM T61657 D09YFJ 135411 EC50 = 226 nM T61657 D0M5EC 1714884 EC50 = 125.89 nM T61657 D08GRF 5287705 Ki = 0.7 nM T61657 D0YO4D 3922 Ki > 1000 nM T61657 C7QAB1 2418 EC50 = 1650 nM T61657 CZBJ59 119342 Ki = 3 nM T61657 CX90MS 128016 Ki = 680 nM T61657 CWZY65 135754 Ki = 13 nM T61657 CRJ7K2 164456 Ki = 26 nM T61657 CF61YU 2063335 EC50 = 15.85 nM T61657 CE8H3O 2757304 EC50 = 63.1 nM T61657 CLY2T6 2802556 EC50 = 100 nM T61657 CI8NO1 3025917 EC50 = 570 nM T61657 C4ZB0M 3086355 EC50 = 25.12 nM T61657 C81XYO 3092138 EC50 = 15.85 nM T61657 C0D8UF 3563820 EC50 = 31.62 nM T61657 C7AJR4 4433908 EC50 = 63.1 nM T61657 CUL8F1 5354022 EC50 = 2200 nM T61657 C8ES5G 6366138 EC50 = 190 nM T61657 C5EOB6 6366685 EC50 > 5 nM T61657 CGL71X 6366726 EC50 = 23 nM T61657 C5EON6 6366727 EC50 > 0.001 nM T61657 C62YGF 6366732 EC50 > 0.001 nM T61657 CK4UA6 6366733 EC50 = 1080 nM T61657 CLF4M5 6366734 EC50 = 21 nM T61657 CA5GS8 6438168 EC50 > 0.001 nM T61657 C7C9SR 6439768 EC50 > 10000 nM T61657 CV6S9Y 6439770 EC50 = 0.4 nM T61657 C8WU1N 6440217 EC50 = 15 nM T61657 CG1S2D 6440346 EC50 = 0.5 nM T61657 C5LH2R 6441236 EC50 = 2 nM T61657 CJHW10 6441985 EC50 = 74 nM T61657 CHA3C2 6447986 EC50 = 43 nM T61657 C3F4GD 6447987 EC50 = 72 nM T61657 CEV62Y 6450532 EC50 = 40 nM T61657 C31YCL 9797765 Ki = 36 nM T61657 CBE62R 9799320 EC50 > 1000 nM T61657 CRK31P 9799442 EC50 = 436 nM T61657 COP9S7 9799477 EC50 = 220 nM T61657 CENQ29 9799532 IC50 = 22 nM T61657 CSNI93 9799841 EC50 > 10000 nM T61657 CX2HY4 9801929 EC50 > 10000 nM T61657 CCUE13 9802971 Ki = 4064 nM T61657 CW7D0R 9810431 EC50 = 2068 nM T61657 CUJ14W 9819890 EC50 > 10000 nM T61657 CEK1O4 9820039 EC50 = 46 nM T61657 CQI49S 9820393 EC50 > 10000 nM T61657 C7R9JM 9820462 Ki = 90 nM T61657 C2X3PS 9822318 EC50 = 8.6 nM T61657 C9SQ7J 9825106 Ki > 10000 nM T61657 CIWO37 9843061 EC50 = 25 nM T61657 CI1P9A 9844563 Ki = 156 nM T61657 CQFA96 9845057 Ki = 4687 nM T61657 CE7D1J 9845382 IC50 = 6.5 nM T61657 CQ1ZH6 9847065 Ki = 2270 nM T61657 C4W3MR 9864378 EC50 = 200 nM T61657 CA74MZ 9864886 IC50 = 40 nM T61657 C2ZY0W 9865875 EC50 > 1000 nM T61657 CZVA73 9866726 Ki > 10000 nM T61657 C8F3DE 9867254 Ki > 10000 nM T61657 CAE0R3 9868664 Ki = 6008 nM T61657 CRC51S 9869157 Ki = 5325 nM T61657 CA0TS6 9884959 EC50 = 139 nM T61657 CSK5B8 9885521 EC50 > 1000 nM T61657 CH0PV4 9885573 IC50 = 1000000 nM T61657 C3CS9R 9886082 EC50 > 10000 nM T61657 C5AD1H 9886137 Ki > 10000 nM T61657 C41JUL 9887430 EC50 = 115 nM T61657 CG3JR4 9887949 EC50 > 10000 nM T61657 CRA64P 9888023 Ki > 10000 nM T61657 CU2OI0 9888037 Ki = 8269 nM T61657 C8V1ON 9888385 IC50 = 7.5 nM T61657 C90UXQ 9889347 Ki = 5681 nM T61657 C8MK1Y 9889522 Ki = 320 nM T61657 C2WFX1 9905729 EC50 = 304 nM T61657 C2D9WJ 9906413 EC50 = 2238 nM T61657 C9AJZ7 9906514 EC50 = 17 nM T61657 C7E0IO 9907433 EC50 > 10000 nM T61657 CK9Z7I 9907650 IC50 = 230 nM T61657 CVG53F 9910801 Ki = 8000 nM T61657 C0A3UZ 9911319 Ki = 2112 nM T61657 CSW2Y8 9929026 EC50 = 339 nM T61657 C9WZ1S 9930650 Ki = 5623 nM T61657 CTXK14 9932151 Ki > 10000 nM T61657 CX7U3M 9932436 Ki = 8064 nM T61657 CIS1Z0 9948900 EC50 = 355 nM T61657 C9VEF0 9949645 EC50 = 1388 nM T61657 C6CI3S 9950957 EC50 > 10000 nM T61657 CS8M7V 9953061 EC50 = 26 nM T61657 CU46RB 9953712 Ki = 71 nM T61657 C6JLI1 9973307 EC50 > 10000 nM T61657 CV1A3K 9974457 EC50 > 1000 nM T61657 C63OUJ 9976842 EC50 > 1000 nM T61657 CT7YJ8 9977495 EC50 > 1000 nM T61657 C05EXS 9998870 EC50 > 10000 nM T61657 CL7X4Y 9999621 EC50 > 10000 nM T61657 CM1BQ5 10003577 Ki = 3927 nM T61657 CZP71W 10022432 EC50 = 310 nM T61657 CN6LP5 10022568 EC50 > 10000 nM T61657 C4K5OP 10026035 Ki = 4742 nM T61657 C6L0XH 10044201 Ki = 36 nM T61657 CN0Y1P 10044591 EC50 = 45 nM T61657 CC4MF5 10045395 EC50 = 92 nM T61657 CE60FI 10065757 EC50 = 287 nM T61657 C2C0GJ 10066739 EC50 = 29 nM T61657 CVMD62 10069273 EC50 = 41 nM T61657 C4VU6T 10087372 EC50 > 10000 nM T61657 CC8R9M 10093918 Ki = 320 nM T61657 C8MG7C 10094345 IC50 > 3000 nM T61657 CSG68Q 10127015 IC50 = 22 nM T61657 C72HLB 10172878 IC50 = 21 nM T61657 C15HAE 10194688 IC50 = 15 nM T61657 C9XS2G 10203771 Ki = 288 nM T61657 CVL1Q6 10227224 Ki = 89 nM T61657 C3IHN5 10251128 IC50 = 25 nM T61657 CSE96Y 10292425 IC50 = 250000 nM T61657 CY1J5M 10308975 Ki > 1000 nM T61657 C9D7QC 10314719 EC50 = 0.3 nM T61657 C7G6XH 10315687 EC50 = 3 nM T61657 CVQ7Z6 10316839 EC50 > 10000 nM T61657 C6C5GP 10320109 Ki = 810 nM T61657 C5LV9X 10358286 EC50 = 1200 nM T61657 CUEF37 10362997 IC50 = 150 nM T61657 CG01ED 10383375 EC50 = 337 nM T61657 CIK6T7 10384337 EC50 = 256 nM T61657 CW39AL 10384413 IC50 = 53 nM T61657 CJCA73 10385620 Ki = 1245 nM T61657 C25HLM 10389354 Ki = 158 nM T61657 CTO46Q 10405813 IC50 = 140 nM T61657 CXQ9S4 10450790 EC50 = 395 nM T61657 CXA0N9 10458226 Ki = 500 nM T61657 CV7C4F 10478196 IC50 = 2 nM T61657 C0KZT7 10519016 Ki = 105 nM T61657 CY62NU 10523459 Ki = 70 nM T61657 CQR8K0 10524574 IC50 = 4.5 nM T61657 C5BXE0 10543210 EC50 > 1000 nM T61657 CUO1I2 10543981 Ki = 12 nM T61657 C6CWZ1 10545954 EC50 = 110 nM T61657 C26NJB 10547547 IC50 = 2.5 nM T61657 C9EBZ0 10572606 IC50 = 36 nM T61657 CKBI92 10619546 IC50 = 39 nM T61657 CS96IV 10619935 EC50 = 31 nM T61657 C2HXP8 10641611 Ki = 90 nM T61657 CMH87P 10643692 EC50 > 10000 nM T61657 CZ2C5K 10663499 Ki > 3000 nM T61657 C92TJP 10666483 Ki = 17 nM T61657 CSC54U 10687664 EC50 > 1000 nM T61657 C89VQU 10690943 IC50 = 290 nM T61657 C9K4YM 10709275 EC50 > 1000 nM T61657 C1SNV6 10760998 Ki = 660 nM T61657 C9UFH8 10763649 Ki = 105 nM T61657 C2TJY4 10788561 Ki > 10000 nM T61657 CTI5N7 10789247 Ki = 21 nM T61657 CMXI39 10804037 EC50 = 770 nM T61657 C4U5ZQ 10906425 Ki = 2056 nM T61657 C8UG3F 10926235 EC50 > 500 nM T61657 C13TFH 10938920 Ki > 10000 nM T61657 C75PWJ 10961406 Ki > 10000 nM T61657 CL9QM1 11070809 Ki > 10000 nM T61657 CV38KY 11167904 EC50 = 13 nM T61657 CW14SH 11253452 EC50 > 100000 nM T61657 C27ERO 11279584 IC50 = 90000 nM T61657 CX24ON 11317250 EC50 = 7700 nM T61657 CT4HL6 11340230 IC50 = 32000 nM T61657 CZ8IT7 11349121 IC50 = 175000 nM T61657 CUY07B 11382535 IC50 = 500000 nM T61657 CCL2D4 11472545 EC50 > 100000 nM T61657 CY6PJ9 11504066 EC50 = 40 nM T61657 CJH04T 11510627 EC50 = 35 nM T61657 CM34CL 11518525 EC50 = 14 nM T61657 C9NH8Y 11547131 EC50 = 25 nM T61657 CQAF21 11554936 EC50 = 17 nM T61657 CLID54 11569584 EC50 = 9.5 nM T61657 CQ8S3K 11627002 EC50 = 60 nM T61657 C41AJB 11634244 EC50 > 10000 nM T61657 C3RMA0 11718697 EC50 = 248 nM T61657 C34NCO 11724776 EC50 > 1000 nM T61657 C0S9KJ 11740691 EC50 = 1004 nM T61657 CFC0X5 11751490 IC50 < 1 nM T61657 C7H2KQ 11784536 EC50 = 17600 nM T61657 C0WA5F 11793407 EC50 = 8 nM T61657 CD5K4U 11799011 Ki > 10000 nM T61657 C7UWV3 12112296 EC50 = 21 nM T61657 CIQJ20 12112298 EC50 = 21 nM T61657 CQ9YE5 12358678 EC50 = 3.3 nM T61657 C97MLN 13554588 EC50 = 50.12 nM T61657 CL23YP 13765519 EC50 = 1000 nM T61657 C7JSH9 13833722 EC50 = 140 nM T61657 C1M8SC 13833726 EC50 = 430 nM T61657 C7Z0YT 13833727 EC50 = 320 nM T61657 CT41DZ 14557465 EC50 = 1900 nM T61657 CN7CX1 14726558 IC50 = 100 nM T61657 C8DP6M 14776682 EC50 = 18 nM T61657 CQI17S 15160092 EC50 = 5 nM T61657 CNS9T8 15434197 Ki > 1000 nM T61657 CS2B4X 15951828 EC50 = 100 nM T61657 CU8LV5 15951923 EC50 = 39.81 nM T61657 CDA7J9 15951925 EC50 = 63.1 nM T61657 C4LRI8 15951927 EC50 = 63.1 nM T61657 C9S5XT 15952013 EC50 = 79.43 nM T61657 CCZ8Y4 15952016 EC50 = 125.89 nM T61657 CKW7N6 15952017 EC50 = 125.89 nM T61657 C0AZ9Q 15952019 EC50 = 100 nM T61657 CX2CS8 15952020 EC50 = 251.19 nM T61657 C3U7WJ 15952211 EC50 = 630.96 nM T61657 C5J3ZE 16661643 EC50 = 6.8 nM T61657 CX6L0G 16661644 EC50 = 3.8 nM T61657 C5GTA2 18507967 EC50 = 250 nM T61657 CQYD01 18768139 EC50 = 5 nM T61657 CX3Q7D 20243100 EC50 = 0.4 nM T61657 C5MHX3 21217837 Ki > 3000 nM T61657 CV1C4A 22226112 EC50 > 1000 nM T61657 CLV67T 22971725 EC50 = 10 nM T61657 CTE1N2 24748569 EC50 > 10000 nM T61657 C26ZLQ 25259039 EC50 < 10000 nM T61657 C1TH9L 25259040 EC50 < 10000 nM T61657 CSTR97 25259041 EC50 = 39.81 nM T61657 CP6OG5 25259262 EC50 < 10000 nM T61657 C7FLT0 25259263 EC50 < 10000 nM T61657 CT2B1Z 25259265 EC50 = 19.95 nM T61657 C2G6QF 25259266 EC50 = 56.7 nM T61657 C4HJ5Z 25259267 EC50 < 10000 nM T61657 CO7M0D 44285104 EC50 = 1100 nM T61657 CS7U6L 44285287 EC50 = 20 nM T61657 CFTB98 44313143 Ki > 3000 nM T61657 C4E1OW 44313513 Ki > 3000 nM T61657 C8W6JP 44314319 Ki = 11 nM T61657 C17LMT 44314320 Ki > 1100 nM T61657 C7U3IB 44316094 EC50 = 1000 nM T61657 CRY69X 44316095 EC50 = 36 nM T61657 COX51B 44316155 EC50 = 280 nM T61657 C92VTZ 44316277 EC50 = 170 nM T61657 C8RM3G 44316292 EC50 = 4 nM T61657 C90NSH 44316354 EC50 = 4 nM T61657 CIVH74 44316525 Ki > 1000 nM T61657 CAP68W 44316543 EC50 = 809 nM T61657 CAI2Z5 44316544 Ki > 1000 nM T61657 C0YQ8H 44316756 Ki > 1000 nM T61657 C6Q1CA 44316796 EC50 = 637 nM T61657 CLK5H0 44316811 EC50 = 559 nM T61657 CK48CT 44321880 EC50 = 3200 nM T61657 CID72B 44321881 EC50 = 2000 nM T61657 CXV0B4 44321951 EC50 = 1500 nM T61657 C1KUN0 44325759 Ki > 1000 nM T61657 CLB6X7 44325767 EC50 = 809 nM T61657 CW0T6K 44353336 Ki = 2112 nM T61657 C8K0AB 44353347 Ki = 4623 nM T61657 C3DYE9 44353422 Ki = 3597 nM T61657 C5DTY3 44353441 Ki = 1956 nM T61657 C2M8TN 44353456 Ki > 10000 nM T61657 CVKA40 44353466 Ki = 2612 nM T61657 C8J5SA 44353480 Ki = 1984 nM T61657 CIB15X 44353481 Ki > 10000 nM T61657 C3MY4C 44364348 Ki = 210 nM T61657 CY9XP2 44366042 EC50 > 10000 nM T61657 CT3S5O 44377822 EC50 = 8 nM T61657 COX1B7 44397758 EC50 = 5300 nM T61657 C5QRI4 44401302 IC50 = 7 nM T61657 CJVG73 44459626 EC50 = 1800 nM T61657 CR5SI0 44476535 EC50 > 10000 nM T61657 CP4DM5 44581289 EC50 = 10 nM T61657 C8UHG5 45270032 IC50 = 40 nM T61657 CUD91T 49862248 EC50 > 10000 nM T61657 C5ZX4B 54597874 EC50 > 10000 nM T61657 C9G4IT 60729785 EC50 = 77.8 nM T61657 CZ38NM 69588033 EC50 = 40 nM T61657 CN03UB 71568951 EC50 = 136.3 nM T61657 CX9EA0 71568952 EC50 = 12.1 nM T61657 C4GRK9 71571262 EC50 = 11 nM T61657 C6TBD2 121345502 EC50 > 20000 nM T61657 CQZ9W3 121414283 EC50 = 2.05 nM T61657 C6L4GM 135949402 EC50 = 26 nM T61657 C5L6AU 136126668 EC50 = 820 nM T61657 CN5MO3 136126669 EC50 > 1000 nM T61657 CJ5EH7 136126670 EC50 > 1000 nM T61657 CI4CG1 136126671 EC50 > 1000 nM T61657 C1J4DV 145965542 EC50 = 2.5 nM T61657 CRKW68 145966900 EC50 > 10000 nM T61657 C4MY5N 145967331 EC50 = 26 nM T61657 CC05VW 145970742 EC50 > 10000 nM T61657 CDBR75 145976745 EC50 = 40 nM T61657 C2A1UC 10429766 Ki > 1000 nM T61657 D09RRF 11530459 EC50 = 7.943 nM T61657 D0F8CC 10090192 EC50 = 140 nM T61657 D0F8JO 9951075 IC50 = 175000 nM T61657 D0G6JM 5289501 Ki = 0.5 nM T61657 D0P0PP 10044792 IC50 = 135 nM T61657 D0Q0IR 177238 IC50 = 20 nM T61657 D0Q9FZ 6442223 EC50 = 10 nM T61657 D0RD0R 2126 EC50 = 8.6 nM T61657 D0X5WP 10410894 Ki = 220 nM T37541 D00STL 644241 Ki = 99 nM T37541 D01MUR 68844 Ki = 2.8 nM T37541 D01WLC 4170 Ki = 2.1 nM T37541 D02PJA 24841 Ki = 250000 nM T37541 D03QGM 5355 Ki = 3.6 nM T37541 D03RTS 2662 Ki = 2170 nM T37541 D03UOT 785 Ki = 883000 nM T37541 D04AIT 5280445 Ki = 4.7 nM T37541 D05OFX 219078 Ki = 4446 nM T37541 D05UYW 5284549 Ki = 3.5 nM T37541 D07HBX 338 Ki = 82100 nM T37541 D07INV 3295 Ki = 0.78 nM T37541 D07MGA 72281 Ki = 3.3 nM T37541 D07VDZ 5284627 Ki = 0.87 nM T37541 D09NIA 2732 Ki = 2.8 nM T37541 D09VAZ 5565 Ki = 45000 nM T37541 D0AZ3C 5291 Ki = 109 nM T37541 D0AZ8C 5213 Ki = 4710 nM T37541 D0C2II 4100 Ki = 2.1 nM T37541 D0C8FX 3005837 Ki = 7760 nM T37541 D0E1SW 1986 Ki = 2 nM T37541 D0H8FH 3702 Ki = 0.23 nM T37541 D0J4GO 3038 Ki = 6 nM T37541 D0J7RK 36811 Ki = 4300 nM T37541 D0K0OZ 5702160 Ki = 3 nM T37541 D0K1QD 3998 Ki = 75 nM T37541 D0K8KX 5280343 Ki = 4840 nM T37541 D0L4JT 5333 Ki = 70 nM T37541 D0L6DA 119607 Ki = 3900 nM T37541 D0OT0O 44561 Ki = 560000 nM T37541 D0PQ3G 3440 Ki = 513 nM T37541 D0SH3I 387447 Ki = 6940 nM T37541 D0U5QK 1983 Ki = 9100 nM T37541 D0W5HK 216239 Ki = 8136.4 nM T37541 D0Y2IZ 5560 Ki = 7.9 nM T37541 D0Z3EI 6038 Ki = 420 nM T37541 D04IIU 216468 Ki = 122 nM T37541 D04PBH 5280804 Ki = 3.8 nM T37541 D05NJI 5287541 Ki = 23 nM T37541 D08BXT 1102 Ki = 1230 nM T37541 D0I7MT 5281807 Ki = 452.6 nM T37541 D0L6HN 996 Ki > 500000 nM T37541 D0U3EP 445154 Ki = 4350 nM T37541 D0V0UK 82267 Ki = 6800 nM T37541 D03SLR 445858 Ki = 7410 nM T37541 D0NH9P 135 Ki = 4080 nM T37541 D0X2AU 23427 Ki > 100000 nM T37541 D0LD9S 1103 Ki = 710 nM T37541 CI0WH9 72 Ki = 7870 nM T37541 CUT2V4 260 Ki = 1060000 nM T37541 COV5W3 402 Ki = 1240000 nM T37541 CSZ43B 540 Ki = 15200000 nM T37541 C97QXH 767 Ki = 160000 nM T37541 C39CTO 768 Ki = 9200000 nM T37541 C1QDT0 781 Ki = 170000 nM T37541 CW0R2L 944 Ki = 190000 nM T37541 CQV86E 1100 Ki = 7300000 nM T37541 C8W7BZ 1118 Ki = 1380000 nM T37541 CU12QE 1203 Ki = 450 nM T37541 C6O0MZ 1491 Ki = 72000 nM T37541 C5L7VX 2871 Ki = 4680 nM T37541 CQ0D8J 3469 Ki = 68000 nM T37541 CJ2F6P 5056 Ki = 8980 nM T37541 CDJ4K6 5987 Ki = 9500 nM T37541 CUP2F4 7043 Ki = 7250 nM T37541 C1CVT7 7121 Ki = 7150 nM T37541 C6NC4O 7414 Ki = 5740 nM T37541 C6QYD8 8434 Ki = 8700 nM T37541 CHP7I1 9016 Ki = 3880 nM T37541 CLYZ50 9338 Ki = 6600 nM T37541 CV5PC3 11568 Ki = 5900 nM T37541 CUA0L6 14917 Ki = 1240000 nM T37541 CNI85U 15109 Ki = 3220 nM T37541 CQ4C5U 16523 Ki = 850 nM T37541 CNGB21 20098 Ki = 900 nM T37541 C3LA1Z 20161 Ki = 940 nM T37541 C3NG2U 24529 Ki = 1780000 nM T37541 CFM9L6 24530 Ki = 1410000 nM T37541 C3F1OY 25502 Ki = 670000 nM T37541 C4OU6D 35703 Ki = 7800 nM T37541 CN94KU 65008 Ki = 8870 nM T37541 C1NQ8E 65188 Ki = 9180 nM T37541 CT6YO0 66548 Ki = 6270 nM T37541 C0ZK7U 67284 Ki = 3700 nM T37541 CVI38F 69809 Ki = 410 nM T37541 CTMF08 75076 Ki = 780 nM T37541 C0I4UT 75077 Ki = 8300 nM T37541 CE5RZ1 76509 Ki = 730 nM T37541 C9V0ME 77547 Ki = 750 nM T37541 C6TS8J 77548 Ki = 830 nM T37541 CX79KD 78297 Ki = 273.1 nM T37541 CX47BZ 78479 Ki = 58000 nM T37541 C5BFK4 87432 Ki = 700 nM T37541 C6K3MG 101424 Ki > 100000 nM T37541 CN19UT 129695 Ki = 100 nM T37541 C2P0RH 139584 Ki = 36540000 nM T37541 CJ0FR9 155148 Ki = 9310 nM T37541 C8AO0Z 165323 Ki = 5.4 nM T37541 CU3WG6 179620 Ki = 8850 nM T37541 CSMP84 219987 Ki = 470 nM T37541 C3QV5H 287064 Ki = 810 nM T37541 C26HNY 289493 Ki = 9030 nM T37541 C96DKW 310360 Ki = 8550 nM T37541 CT3ZU4 388776 Ki = 1090 nM T37541 CH21KA 389641 Ki = 107000 nM T37541 C6CQO3 389642 Ki = 108000 nM T37541 CNPZ40 394897 Ki = 35 nM T37541 C7HME8 439246 Ki = 4.3 nM T37541 CA8C5N 439514 Ki = 9110 nM T37541 C5HM8E 474578 Ki = 465.8 nM T37541 C49CNT 519869 Ki = 710 nM T37541 CJ7FR6 533728 Ki = 1470000 nM T37541 CYGK68 676946 Ki = 850 nM T37541 CMO61A 694792 Ki = 7.1 nM T37541 CF93TC 821388 Ki = 810 nM T37541 C8SN5L 889524 Ki = 51 nM T37541 CEN67I 897592 Ki = 861 nM T37541 C4QX1Z 1146666 Ki = 2.6 nM T37541 C6T0NU 1230924 Ki = 9.5 nM T37541 C9IBF8 1241259 Ki = 0.74 nM T37541 CF1N3S 1277269 Ki = 4 nM T37541 C40CKN 1316238 Ki = 3.2 nM T37541 C9DY2L 1488548 Ki = 380 nM T37541 CDQR23 2049187 Ki = 9.8 nM T37541 C2O9YS 2196398 Ki = 6.5 nM T37541 C4TD8M 2388085 Ki = 1.3 nM T37541 C8QGL9 2760606 Ki > 10000 nM T37541 CE2GR3 2900806 Ki = 1240 nM T37541 CME74N 2904589 Ki = 605 nM T37541 C61OTP 2991092 Ki = 21 nM T37541 CN2Y5M 3083616 Ki = 5560 nM T37541 C9GT5Z 3083928 Ki = 9280 nM T37541 CL6E2Y 3426384 Ki = 5122 nM T37541 CQ5F9P 3724005 Ki = 9.5 nM T37541 CV0KG3 3950536 Ki = 4.3 nM T37541 C4E5VQ 4447263 Ki = 5.8 nM T37541 C96LCZ 4476238 Ki = 65 nM T37541 CDK4L0 4608376 Ki = 600000 nM T37541 CLSY09 4626049 Ki = 760 nM T37541 C3GDR0 4634582 Ki = 62 nM T37541 CCB9Z5 4656684 Ki = 71 nM T37541 C7JBU0 5019114 Ki = 161 nM T37541 C4OAL9 5070078 Ki = 6400 nM T37541 CI8JY0 5172475 Ki = 4.3 nM T37541 CY9IV8 5223338 Ki = 5 nM T37541 CEBD92 5272990 Ki = 4600 nM T37541 CP09FG 5272997 Ki = 5900 nM T37541 C4SV5T 5273568 Ki = 3870 nM T37541 CU4E5S 5273569 Ki = 4320 nM T37541 CN10FM 5281793 Ki = 71.4 nM T37541 CA18OQ 5316302 Ki = 4530 nM T37541 CTJ01E 5317485 Ki = 8110 nM T37541 CI58XK 5319562 Ki = 820 nM T37541 CNO53D 5321265 Ki = 650 nM T37541 C8PS4E 5358858 Ki = 3690 nM T37541 CXEW32 5491996 Ki = 14500 nM T37541 CK0M4A 5910585 Ki = 7820 nM T37541 C2JTF7 6432768 Ki = 5010 nM T37541 CS4KQ6 6482974 Ki = 7010 nM T37541 C9L8AX 6537802 Ki = 840 nM T37541 C65FRB 6852128 Ki = 6.4 nM T37541 CKCM96 7463376 Ki = 7950 nM T37541 CDCP43 7766335 Ki = 630 nM T37541 CY47OI 9998322 Ki = 6.5 nM T37541 CNKD31 10016330 Ki = 620.3 nM T37541 C5X7GY 10059582 Ki = 1899 nM T37541 CY8F0E 10076040 Ki = 58300 nM T37541 C0P5XV 10081897 Ki = 956 nM T37541 CD58EL 10083644 Ki = 720 nM T37541 C7WU0A 10107532 Ki = 467.8 nM T37541 CJV68L 10220266 Ki = 389.3 nM T37541 CQ8A0I 10328097 Ki = 26.6 nM T37541 CN40WD 10331524 Ki = 1178 nM T37541 C3HBY6 10375558 Ki = 66 nM T37541 CVIN94 10439991 Ki = 4.7 nM T37541 CWQY26 10535227 Ki > 10000 nM T37541 C73KXU 10586607 Ki = 14500 nM T37541 C9TSQ6 10632698 Ki = 31400 nM T37541 C6D2TJ 10712038 Ki = 35 nM T37541 C36BAC 11034581 Ki > 100000 nM T37541 C8C6ER 11069133 Ki = 2.9 nM T37541 CMK4Y0 11096006 Ki = 435.5 nM T37541 CIL4M9 11183499 Ki > 100000 nM T37541 CHC42Y 11245700 Ki = 19 nM T37541 CF15AS 11287957 Ki = 4965 nM T37541 CHA0V5 11321514 Ki = 910 nM T37541 C8PM3Z 11353795 Ki = 18 nM T37541 CM8P2L 11609292 Ki = 23 nM T37541 C9QL2F 11615432 Ki = 7507 nM T37541 C9JR2I 11674590 Ki = 8580 nM T37541 CV7HN1 11795548 Ki = 15 nM T37541 CNHD71 12051191 Ki > 200000 nM T37541 CMPA32 12066940 Ki > 500000 nM T37541 CB15KR 12066941 Ki > 500000 nM T37541 C60EFT 12354987 Ki = 300 nM T37541 C5RS4H 12528487 Ki = 975.3 nM T37541 CM8TP6 12528490 Ki = 1364 nM T37541 CK90BP 12765315 Ki = 320 nM T37541 CF2BM7 13177311 Ki = 2.1 nM T37541 C8VM1A 13201770 Ki = 720 nM T37541 CC25BI 13927398 Ki = 1100000 nM T37541 C7K4JV 14024589 Ki = 1282 nM T37541 C4UG2O 14057643 Ki > 100000 nM T37541 CHOG93 14611919 Ki = 89 nM T37541 C76ASY 14787919 Ki > 200000 nM T37541 CH5YR2 15014351 Ki > 200000 nM T37541 C7XD2T 15118768 Ki = 8980 nM T37541 CK8GE9 15230629 Ki = 1790 nM T37541 C8PMQ9 15729847 Ki > 200000 nM T37541 C8PER5 15938557 Ki > 500000 nM T37541 C3W2MB 15939939 Ki = 3.9 nM T37541 CC0Z4V 16119626 Ki = 730 nM T37541 CDWU20 17537594 Ki = 39.4 nM T37541 CK7D2I 17748220 Ki = 10 nM T37541 CLY1N4 17757567 Ki = 170 nM T37541 C6SFI8 18268734 Ki = 4.7 nM T37541 CR9VF3 18668331 Ki = 9.9 nM T37541 CQE5K4 18710120 Ki > 200000 nM T37541 C60NAV 18971452 Ki = 86.4 nM T37541 C2K5BX 19374444 Ki = 8.3 nM T37541 C62PKT 19838794 Ki = 7.8 nM T37541 CDU40W 20184392 Ki > 200000 nM T37541 CKR8T2 20970546 Ki = 10.5 nM T37541 C61KUX 21726402 Ki = 1.7 nM T37541 CJ4O2E 21806575 Ki = 5.8 nM T37541 C02IPY 21978067 Ki = 10.1 nM T37541 C9U4TE 22313850 Ki = 135 nM T37541 C9KMP4 23275795 Ki = 7.7 nM T37541 C7V6YP 23665706 Ki = 0.24 nM T37541 C01LHS 24640776 Ki = 13.3 nM T37541 CT8O2Z 24643222 Ki = 9.5 nM T37541 CISH83 25186263 Ki = 1.5 nM T37541 CU14KG 25258358 Ki = 68700 nM T37541 CQ1WE2 25258360 Ki > 200000 nM T37541 CL5EZ6 25258361 Ki > 200000 nM T37541 COU19V 25258363 Ki > 200000 nM T37541 CRP6F5 25335375 Ki = 62.9 nM T37541 CPN2T5 25392418 Ki = 6.9 nM T37541 C5EC2T 26535209 Ki = 10.4 nM T37541 CLNR46 26598995 Ki = 3238 nM T37541 CA9UZ7 26773685 Ki = 6.9 nM T37541 CI0K1J 36865965 Ki = 8.3 nM T37541 C6WU8M 42609905 Ki = 2.7 nM T37541 CYJ0H4 43089860 Ki = 16.5 nM T37541 CIM4Z8 43132043 Ki = 5.4 nM T37541 CXJY80 43235186 Ki = 4.6 nM T37541 C7EO2A 43329592 Ki = 8.9 nM T37541 CA0DX4 43342474 Ki = 9.7 nM T37541 C2HY4R 43342475 Ki = 9.4 nM T37541 CBK0M6 43342481 Ki = 0.9 nM T37541 C82MRL 44144383 Ki = 73.2 nM T37541 CI3O9B 44395149 Ki = 45 nM T37541 CMSJ40 44395790 Ki = 3.7 nM T37541 CZ4DF9 44399462 Ki = 8.3 nM T37541 CD5MJ6 44399571 Ki = 9.4 nM T37541 C2T7MB 44399654 Ki = 84 nM T37541 CA90GQ 44424362 Ki = 160 nM T37541 C5HB4P 44424363 Ki > 200000 nM T37541 CK8S7Y 44424364 Ki > 200000 nM T37541 C28QYE 44424366 Ki = 320 nM T37541 CM3J0U 44430517 Ki = 24 nM T37541 C9LT7Y 44430518 Ki = 41 nM T37541 C1VTB6 44430520 Ki = 79 nM T37541 C2L5MB 44430521 Ki = 18 nM T37541 CVEO17 44430523 Ki = 23 nM T37541 C8MFL1 44430524 Ki = 25 nM T37541 CFW8V2 44520897 Ki = 7 nM T37541 CR4NZ3 44520898 Ki = 6.9 nM T37541 CI78UO 44520899 Ki = 7.2 nM T37541 CQUC34 44520900 Ki = 6.9 nM T37541 CNC1D8 44520905 Ki = 8.5 nM T37541 CR43NP 44520906 Ki = 6.1 nM T37541 CXD9V3 44590306 Ki > 200000 nM T37541 COE8U0 45267045 Ki = 35.5 nM T37541 C23MVW 45269009 IC50 = 27900 nM T37541 C0RG8K 45269749 Ki = 8500 nM T37541 CSW5V6 45378228 Ki = 6.4 nM T37541 CV5RQ3 45484187 Ki = 98 nM T37541 CTG20B 45485271 Ki = 8900 nM T37541 CK4U0V 45485283 Ki = 3200 nM T37541 C6ION5 46236927 Ki = 49 nM T37541 C7SFG3 46236928 Ki = 8370 nM T37541 CC82QE 46237039 Ki = 556 nM T37541 CBCK34 46237040 Ki = 60 nM T37541 CSD29O 46237041 Ki = 581 nM T37541 CEB1X9 46237042 Ki = 54 nM T37541 C1VIK9 46237043 Ki = 53 nM T37541 C3RJ5M 46237044 Ki = 5150 nM T37541 CU5Y9E 46237045 Ki = 6.5 nM T37541 CM7N6J 46237172 Ki = 64 nM T37541 CP15GJ 46237173 Ki = 54 nM T37541 CT65RE 46868356 Ki = 3.9 nM T37541 CNEO10 46871889 Ki = 4.6 nM T37541 C93AIR 46899573 Ki = 108000 nM T37541 CJ0R2O 46911381 Ki = 48 nM T37541 C0NUM6 53386724 Ki = 60.2 nM T37541 C54FGU 53386866 Ki = 12.1 nM T37541 CRI54V 53386867 Ki = 34.9 nM T37541 CUX7S4 53386868 Ki = 91.7 nM T37541 CCFP92 53516400 IC50 > 50000 nM T37541 C6SM5T 54613427 Ki = 7 nM T37541 C0ZJ2L 55629711 Ki = 310 nM T37541 CIJ9V0 56684131 Ki = 912 nM T37541 CH52DA 56921864 Ki = 6750 nM T37541 CTFL92 56928044 Ki = 10.2 nM T37541 C4VGE9 57047254 Ki = 8.3 nM T37541 CP7YR5 57345662 Ki = 270 nM T37541 C1M0LS 57394809 Ki = 690 nM T37541 CW1TU4 57412422 Ki = 4.8 nM T37541 CT4BV9 57412423 Ki = 5.9 nM T37541 C31NWX 57412424 Ki = 13.9 nM T37541 CD86ER 57412425 Ki = 6.5 nM T37541 CB94YU 57412426 Ki = 8 nM T37541 C2K8YJ 57412507 Ki = 5.7 nM T37541 CSF4V6 57412508 Ki = 5.8 nM T37541 CHAO86 57412509 Ki = 8.2 nM T37541 C3U6TH 57412510 Ki = 34.7 nM T37541 C40LOS 57412511 Ki = 23.4 nM T37541 CZ47VT 57412512 Ki = 17.8 nM T37541 C28WRD 57412600 Ki = 61.7 nM T37541 C2XPG5 57413583 Ki = 7.9 nM T37541 CM2AY7 57413584 Ki = 50.8 nM T37541 C9V6EY 60446869 Ki = 911.3 nM T37541 CGF3W6 66586679 Ki = 890 nM T37541 CN84CU 66586879 Ki = 840 nM T37541 C2Y5KV 70682044 Ki = 73.3 nM T37541 CXJ16H 71450117 Ki = 873 nM T37541 CB8JA3 71455488 Ki = 628 nM T37541 C02UHX 71455489 Ki = 609 nM T37541 CICJ97 71457274 Ki = 602 nM T37541 CMHG14 71521493 Ki = 6300 nM T37541 CHN53G 71521494 Ki = 7100 nM T37541 CZJ5M6 71521495 Ki = 5800 nM T37541 CFBE53 71521496 Ki = 4900 nM T37541 CME27W 71521497 Ki = 9000 nM T37541 C24XWU 71521575 Ki = 9500 nM T37541 CJF68W 71521576 Ki = 9300 nM T37541 C19OIY 71579130 Ki = 730 nM T37541 CGO24R 71584196 Ki = 465 nM T37541 CV0LU6 71602117 Ki = 540 nM T37541 CZL96Y 71602476 Ki = 3.1 nM T37541 C50LSJ 71714068 Ki = 24900 nM T37541 CM4T1R 71717003 Ki = 78400 nM T37541 CG4I1X 71718239 Ki = 7200 nM T37541 C0LYX1 71718858 Ki = 4300 nM T37541 CM24ND 71719433 Ki = 800 nM T37541 CT3D5S 71719441 Ki = 6800 nM T37541 CJG34A 71720036 Ki = 6920 nM T37541 CIU4L2 71720670 Ki = 8700 nM T37541 C0ROQ1 71770179 Ki = 3.5 nM T37541 C8W6DJ 71770180 Ki = 3.5 nM T37541 CB3Y0X 71770181 Ki = 46.9 nM T37541 CKHM42 71770182 Ki = 1.3 nM T37541 CBL41T 71770183 Ki = 4.7 nM T37541 C30EYH 71770184 Ki = 2.2 nM T37541 C5IU0Y 72163201 Ki = 54 nM T37541 CNP42E 72163326 Ki = 4 nM T37541 C2KE5D 72163327 Ki = 55 nM T37541 C0Q5XL 72163343 Ki = 59 nM T37541 C63MIX 72163344 Ki = 77 nM T37541 CL3WV2 72163345 Ki = 80 nM T37541 C4T9DA 72163346 Ki = 175 nM T37541 CTK07O 72163347 Ki = 84 nM T37541 CE32BF 72163348 Ki = 72 nM T37541 CBN48K 72163465 Ki = 65 nM T37541 CGB02D 72163466 Ki = 199 nM T37541 CVFN85 72163467 Ki = 41 nM T37541 C82RDA 72163468 Ki = 245 nM T37541 CA1X6Z 72163476 Ki = 68 nM T37541 C7TKJ4 72163610 Ki = 368 nM T37541 C70OBD 72163611 Ki = 264 nM T37541 CA0Q4T 72163612 Ki = 152 nM T37541 C96GMR 72163613 Ki = 127 nM T37541 CJ2K8R 72163743 Ki = 498 nM T37541 CPY81U 72163744 Ki = 334 nM T37541 CC1D3Y 72163745 Ki = 225 nM T37541 CYH0G5 72163746 Ki = 375 nM T37541 CEZM40 72163861 Ki = 5 nM T37541 CMBR85 72163862 Ki = 14 nM T37541 CZ9IE5 72163863 Ki = 22 nM T37541 CZM75P 72163975 Ki = 142 nM T37541 CPT0C9 72163976 Ki = 46 nM T37541 CX82JD 72696463 Ki = 6.2 nM T37541 COCV73 72696591 Ki = 21.9 nM T37541 C5KHD7 72696592 Ki = 8.5 nM T37541 C4FBA6 72696593 Ki = 6.7 nM T37541 CO1JM5 72696594 Ki = 6.5 nM T37541 CUF61Q 72696595 Ki = 8.3 nM T37541 CO1JT3 73054728 Ki = 30 nM T37541 CU9I6V 82078731 Ki = 125.5 nM T37541 C5TB6O 82080973 Ki = 690.9 nM T37541 C6UZR9 82911195 Ki = 9.6 nM T37541 C3AYZ5 91811067 Ki = 2796 nM T37541 CQF98O 91827503 Ki = 8.5 nM T37541 C3I6NV 91827505 Ki = 9.2 nM T37541 CW1P4E 91827506 Ki = 819 nM T37541 C28QRZ 101564149 Ki > 100000 nM T37541 CDGZ03 101879106 Ki = 24 nM T37541 CY6ER7 101879108 Ki = 17.7 nM T37541 CB1PK8 102151146 Ki > 100000 nM T37541 C0A6FY 102151151 Ki = 7800 nM T37541 C1XV9H 102311866 Ki = 8900 nM T37541 C0CVO4 102480165 Ki > 100000 nM T37541 CUR4V8 114816322 Ki = 0.27 nM T37541 CKV43U 118710106 Ki = 303.5 nM T37541 CBAQ59 118710108 Ki = 269 nM T37541 C0D1SQ 118724328 Ki = 50.6 nM T37541 C89YTC 118724329 Ki = 253.5 nM T37541 CBT87C 118724330 Ki = 28.7 nM T37541 C49AWZ 118724331 Ki = 21.9 nM T37541 CHE1K4 118729473 Ki = 8.9 nM T37541 C9V8MA 118729474 Ki = 97.2 nM T37541 C8GJP5 118729475 Ki = 70.7 nM T37541 C4MEZ0 118729476 Ki = 73.8 nM T37541 CE3IV5 118729477 Ki = 8.6 nM T37541 CUQ7H9 119082247 Ki = 40.5 nM T37541 CN16RY 122189300 Ki = 2.4 nM T37541 CYN3T8 122189301 Ki = 878 nM T37541 CSW9D1 122189302 Ki = 3.1 nM T37541 C6USQ7 122189303 Ki = 2.8 nM T37541 CQ4X1G 122189304 Ki = 4 nM T37541 CH1N0C 122193189 Ki = 730 nM T37541 C19HVL 122193190 Ki = 820 nM T37541 C5TQJ1 122193251 Ki = 520 nM T37541 C8XCL0 122193252 Ki = 710 nM T37541 CC1UO6 122226187 Ki = 660 nM T37541 C7T0FH 122226188 Ki = 1800 nM T37541 C3EG2B 122226189 Ki = 6500 nM T37541 C26IUP 122386532 Ki > 100000 nM T37541 CV4GW7 126961712 Ki = 0.21 nM T37541 C0FD4E 126961713 Ki = 0.19 nM T37541 CS2K4U 127034999 Ki = 0.24 nM T37541 CFG39M 127035855 Ki = 0.43 nM T37541 C6MH2V 127035856 Ki = 0.45 nM T37541 CVO4B6 127035857 Ki = 2.2 nM T37541 CQC6P9 127035858 Ki = 0.31 nM T37541 C7YA3N 127035859 Ki = 0.3 nM T37541 CXZI89 127035860 Ki = 0.28 nM T37541 C5KLP8 127035861 Ki = 0.37 nM T37541 CL76JS 127037630 Ki = 0.39 nM T37541 CY1JU3 127037755 Ki = 5.1 nM T37541 C0UQ7W 127037756 Ki = 3.3 nM T37541 CQUE67 127037757 Ki = 3.5 nM T37541 CG8B3V 127039153 Ki = 0.46 nM T37541 CIO74C 127039154 Ki = 0.35 nM T37541 C0L8NH 127039155 Ki = 0.31 nM T37541 CS96GU 127039479 Ki = 4.4 nM T37541 C3J8ET 127040041 Ki = 2.9 nM T37541 CQC6A4 127042329 Ki = 14.5 nM T37541 C5EX6R 127048632 Ki = 48.2 nM T37541 CK1X5H 127048994 Ki = 2 nM T37541 C2XK0I 127048995 Ki = 1.3 nM T37541 CY4P2X 127048996 Ki = 5.7 nM T37541 C6JB5S 127048997 Ki = 90.7 nM T37541 C1T3WG 127049310 Ki = 39 nM T37541 CKO03S 127049970 Ki = 44.6 nM T37541 CP8KG9 127049971 Ki = 10.4 nM T37541 C9EJ6L 127050230 Ki = 22.4 nM T37541 C7MI5Q 127050568 Ki = 29.6 nM T37541 C1RGQ6 127050569 Ki = 28.9 nM T37541 CB5W0L 127050570 Ki = 10.9 nM T37541 CUG58A 127050571 Ki = 35 nM T37541 C9FZ4E 127050900 Ki = 8.1 nM T37541 CUWE95 127051804 Ki = 50.5 nM T37541 COBU26 127051805 Ki = 60.7 nM T37541 C7SIY6 127051806 Ki = 50 nM T37541 CJ7WT3 127052106 Ki = 35.5 nM T37541 C26TUM 127052712 Ki = 8.5 nM T37541 C7PS8D 127052713 Ki = 54.8 nM T37541 C32ART 127052714 Ki = 54.6 nM T37541 C9D6CB 127053004 Ki = 22.6 nM T37541 CHN5K6 127567366 Ki = 198.5 nM T37541 C4JC3W 127573780 Ki = 801.2 nM T37541 CXN16P 132495328 Ki = 0.8 nM T37541 CKLY32 132502995 Ki = 1881.2 nM T37541 C5O1JE 132547793 Ki > 100000 nM T37541 CKYC42 132547798 Ki > 100000 nM T37541 CRL24F 132596304 Ki > 50000 nM T37541 C4K1YW 132961363 Ki = 6.7 nM T37541 CQ64ZM 132961364 Ki = 3.8 nM T37541 C5LGV6 132961365 Ki = 4.5 nM T37541 C69NDK 133107891 Ki = 0.27 nM T37541 C2AIR8 134129901 Ki = 0.81 nM T37541 C1Y9AL 134130029 Ki = 0.68 nM T37541 CU10DE 134130177 Ki = 9.1 nM T37541 CP8XK0 134130364 Ki = 4 nM T37541 C83LZE 134130471 Ki = 1.8 nM T37541 C5N8AO 134130483 Ki = 7.2 nM T37541 C9V3LX 134130512 Ki = 6.4 nM T37541 CO7G6J 134130566 Ki = 0.91 nM T37541 C69IZA 134130639 Ki > 10000 nM T37541 C8MGN3 134130817 Ki = 65.3 nM T37541 C52IRH 134131086 Ki = 0.7 nM T37541 C9HVL2 134131189 Ki = 0.73 nM T37541 C7GBW5 134131361 Ki = 9.1 nM T37541 C3WJR8 134131535 Ki = 3.6 nM T37541 CQ0K5P 134131567 Ki = 1.4 nM T37541 C8Q5JZ 134131574 Ki = 7.6 nM T37541 CZQ3T2 134132041 Ki > 10000 nM T37541 C89TVU 134132755 Ki = 9.6 nM T37541 CFQG76 134133776 Ki = 8 nM T37541 CT8Z2Q 134133785 Ki = 7.4 nM T37541 CHR23F 134137004 Ki > 10000 nM T37541 C2X1UG 134137145 Ki = 51.9 nM T37541 CHM19B 134139215 Ki = 26.8 nM T37541 CRNF42 134140829 Ki = 62 nM T37541 C1T9JU 134140936 Ki = 52.2 nM T37541 CG4NU1 134141378 Ki = 5.7 nM T37541 CIK25S 134142323 Ki = 67.1 nM T37541 CIRG86 134142877 Ki = 7.8 nM T37541 CWT6O9 134142989 Ki = 29 nM T37541 C5BD1C 134143174 Ki > 10000 nM T37541 CWQ62J 134144541 Ki = 1000 nM T37541 CG7X9K 134144756 Ki = 49.1 nM T37541 CJ5QD3 134144926 Ki = 602.5 nM T37541 CR5F8T 134145685 Ki = 423.5 nM T37541 C8FV5Y 134147016 Ki > 10000 nM T37541 C0TV9S 134147261 Ki = 308.3 nM T37541 C85ABV 134147911 Ki = 54.6 nM T37541 CGBZ05 134148709 Ki = 4.1 nM T37541 CS7K8C 134149271 Ki = 701.1 nM T37541 CD5TI1 134149815 Ki = 628.7 nM T37541 CZ2C3J 134149835 Ki = 3.8 nM T37541 CIL4H9 134151823 Ki > 10000 nM T37541 C9GF7L 134152087 Ki = 7 nM T37541 CZ4WI8 134152920 Ki = 86.3 nM T37541 CD4EN0 134153199 Ki = 45.3 nM T37541 CH6OT4 134153506 Ki = 27.4 nM T37541 CZ9T6I 134153525 Ki > 10000 nM T37541 CWSI54 134154346 Ki = 376.2 nM T37541 CQZU97 134154945 Ki > 10000 nM T37541 C52UTP 134156470 Ki = 4.3 nM T37541 C7OV6T 134156655 Ki = 88.9 nM T37541 CR3Q5U 134159783 Ki = 2 nM T37541 CV9W6N 134159784 Ki = 0.24 nM T37541 CJT9W0 135393499 Ki = 0.45 nM T37541 CK8FP3 135393500 Ki = 2.6 nM T37541 CRL4V7 135393501 Ki = 7.8 nM T37541 CPW4T3 135530880 Ki = 28 nM T37541 C4KH2F 136138702 Ki = 53.6 nM T37541 CYKW91 136728963 Ki = 665.3 nM T37541 CRK6Y9 137631731 Ki = 2614 nM T37541 CZ5GQ4 137631746 Ki > 100 nM T37541 CFQ5W2 137631798 Ki = 490 nM T37541 CBJ75C 137632178 Ki = 536.5 nM T37541 CYD0E3 137632442 Ki = 6.8 nM T37541 CL5K3D 137632743 Ki > 100 nM T37541 C9YKD5 137633039 Ki = 27.8 nM T37541 C5J3AX 137633409 Ki = 121.4 nM T37541 C9AD2H 137633797 Ki = 188 nM T37541 C7N0ER 137634525 Ki > 100000 nM T37541 CP0EC3 137635051 Ki = 281.6 nM T37541 CY1HI4 137635059 Ki = 892.1 nM T37541 C1ZKU2 137635320 Ki = 15.2 nM T37541 CV12YX 137636350 Ki > 100 nM T37541 C7YKB0 137636981 Ki > 50000 nM T37541 C2Z7GO 137637071 Ki = 3.8 nM T37541 C0H2CK 137637173 Ki = 10.1 nM T37541 CWO5Z6 137637365 Ki > 100 nM T37541 CGV9M8 137637508 Ki = 8683 nM T37541 CG0N8K 137637564 Ki = 408.1 nM T37541 C80KCO 137637736 Ki = 79.3 nM T37541 C2HY8G 137637767 Ki = 64.5 nM T37541 CHQ3P9 137638456 Ki = 28.6 nM T37541 CK6OW4 137638637 Ki = 0.77 nM T37541 C6V8ED 137638882 Ki = 5.4 nM T37541 C64JQN 137639095 Ki = 0.53 nM T37541 C4LB2X 137639339 Ki = 100.4 nM T37541 C0IQ1U 137639377 Ki = 4200 nM T37541 COE61G 137639833 Ki = 5800 nM T37541 C2OT9R 137640310 Ki > 50000 nM T37541 CX3JI9 137640517 Ki = 55.2 nM T37541 C6B0CQ 137641198 Ki = 0.51 nM T37541 C0HER8 137641290 Ki > 50000 nM T37541 CMOZ57 137641425 Ki = 203 nM T37541 C53ZAF 137641717 Ki > 10000 nM T37541 CR5JZ8 137642047 Ki > 10000 nM T37541 CCSN50 137642054 Ki > 100 nM T37541 CN6WS9 137642180 Ki = 8.9 nM T37541 CEOC90 137642331 Ki = 9388 nM T37541 CSY67B 137642513 Ki = 3198 nM T37541 C61TSP 137642864 Ki > 100000 nM T37541 C3Y2GU 137643607 Ki = 9.4 nM T37541 C1BW5I 137643671 Ki > 100000 nM T37541 C0B8QA 137643949 Ki > 100 nM T37541 CF31BQ 137644307 Ki = 13.2 nM T37541 CFA3R0 137644914 Ki = 605 nM T37541 C6UAB5 137645654 Ki = 5001 nM T37541 CDZ6T8 137645734 Ki = 267.6 nM T37541 CBRK83 137645944 Ki = 9.3 nM T37541 C7E6NL 137646223 Ki = 299 nM T37541 C10YVU 137646329 Ki > 50000 nM T37541 C5WG2P 137646543 Ki = 16.2 nM T37541 C0YFX2 137646956 Ki > 10000 nM T37541 CRP78K 137647221 Ki > 100 nM T37541 CXD9A0 137647636 Ki = 0.4 nM T37541 CR2H7M 137647845 Ki > 50000 nM T37541 CCD71U 137648259 Ki = 1907.3 nM T37541 C49PLO 137648279 Ki = 694.3 nM T37541 CW8CL7 137648379 Ki = 55.5 nM T37541 CK14XO 137648525 Ki = 3343 nM T37541 C21TVD 137648644 Ki = 707.1 nM T37541 C6RIM2 137648717 Ki = 67.2 nM T37541 CEZT03 137649001 Ki = 8.5 nM T37541 CI9LS2 137649321 Ki = 43.6 nM T37541 CSWR71 137649376 Ki = 911.9 nM T37541 C4N1MP 137650156 Ki = 84.4 nM T37541 CD08YK 137650293 Ki = 138.4 nM T37541 CKJ36G 137650647 Ki = 1897.6 nM T37541 CD7S5L 137650698 Ki > 100000 nM T37541 CV89IF 137651491 Ki = 90.9 nM T37541 CSTP12 137651755 Ki = 0.35 nM T37541 C01BXO 137651769 Ki > 100 nM T37541 CY0C6Z 137652226 Ki > 100 nM T37541 C6GWB1 137652305 Ki > 100 nM T37541 CN3RQ8 137652373 Ki > 10000 nM T37541 C9UGN4 137653309 Ki = 58.5 nM T37541 C8Y7XR 137653485 Ki = 85.6 nM T37541 CIV3E9 137653528 Ki = 1.7 nM T37541 CTP0U2 137654343 Ki = 91 nM T37541 CXC7I2 137655261 Ki = 88.6 nM T37541 C2P5FH 137655445 Ki = 404 nM T37541 C3DT7S 137655450 Ki > 100 nM T37541 CASB61 137655528 Ki > 100 nM T37541 CAZ27T 137655913 Ki = 54.7 nM T37541 C27ALW 137655946 Ki = 3.2 nM T37541 CC0OY9 137655984 Ki = 177.6 nM T37541 C8TJN9 137656061 Ki = 553.5 nM T37541 COEY05 137656447 Ki = 16.7 nM T37541 C0CK7G 137656796 Ki > 10000 nM T37541 C8RNZ6 137657759 Ki > 100 nM T37541 C0KI6G 137657917 Ki = 583.3 nM T37541 C41MLN 137658275 Ki > 10000 nM T37541 CKX78V 137658314 Ki = 1885.2 nM T37541 CL2H0T 137658375 Ki > 100 nM T37541 CT98MV 137658877 Ki > 100 nM T37541 C8YV5D 137659052 Ki = 0.33 nM T37541 CXO9Y7 137659205 Ki > 100 nM T37541 CJ5O8M 137659269 Ki = 360 nM T37541 C5AM2K 137659383 Ki > 10000 nM T37541 C60DEN 137660288 Ki > 10000 nM T37541 CMS92X 137660799 Ki = 1.8 nM T37541 C0TZD5 137661006 Ki > 100000 nM T37541 C0PIE6 137661027 Ki = 78.1 nM T37541 CQ56MJ 137661167 Ki = 347.5 nM T37541 C62QWK 137661307 Ki = 5065 nM T37541 CRC92Y 137661359 Ki = 0.77 nM T37541 C1Z8KG 137661675 Ki = 0.2 nM T37541 C74YSR 137661914 Ki = 37.8 nM T37541 CEAR56 137662187 Ki = 318 nM T37541 CMP8S7 137662201 Ki = 9.2 nM T37541 CFR73V 137662256 Ki = 84.5 nM T37541 CIX41M 138393379 Ki = 0.8 nM T37541 CBOM51 138753317 Ki = 0.8 nM T37541 CB83JY 139593608 Ki = 5.7 nM T37541 C8BZI0 145949366 Ki = 0.84 nM T37541 CHVR98 145949393 Ki = 74.2 nM T37541 C7X0DZ 145949728 Ki = 462.8 nM T37541 C20RXT 145949974 Ki = 1.9 nM T37541 C9QUL0 145951028 Ki = 36.2 nM T37541 CPD05I 145951366 Ki = 0.38 nM T37541 C86DBE 145951463 Ki = 6.8 nM T37541 C38QHU 145951654 Ki = 0.93 nM T37541 CIM8X0 145951670 Ki = 7.4 nM T37541 CJ2W6V 145951720 Ki = 0.25 nM T37541 C2OTU3 145951886 Ki = 3.8 nM T37541 C4N3QL 145952239 Ki = 0.77 nM T37541 CM30EN 145952365 Ki = 311.8 nM T37541 C75RDX 145952490 Ki = 4.6 nM T37541 C26OLK 145952634 Ki = 37.4 nM T37541 CW42HX 145952649 Ki = 0.97 nM T37541 C56QVF 145952880 Ki = 0.85 nM T37541 CAS8M7 145952940 Ki = 0.83 nM T37541 C5DJY9 145953324 Ki = 3.5 nM T37541 CVNE29 145954045 Ki = 86 nM T37541 CD52IH 145954185 Ki = 0.96 nM T37541 C0XO6A 145954770 Ki = 17.4 nM T37541 C1LFA9 145954917 Ki = 3.4 nM T37541 C0UG3K 145955383 Ki = 0.87 nM T37541 C89HDL 145956309 Ki = 7.2 nM T37541 CYJ3N0 145956346 Ki = 0.31 nM T37541 C2KV9S 145956347 Ki = 9.4 nM T37541 CWPZ94 145956803 Ki = 0.93 nM T37541 C7K2DA 145957040 Ki = 0.97 nM T37541 CAMD59 145957136 Ki = 7.1 nM T37541 CM07ZF 145958200 Ki = 6.6 nM T37541 CXVC18 145959110 Ki = 0.84 nM T37541 CU8J0M 145959118 Ki = 645 nM T37541 CWNS89 145959524 Ki = 0.77 nM T37541 CPL41Z 145959905 Ki = 0.71 nM T37541 CGZ1K8 145959957 Ki = 0.35 nM T37541 C2SI5J 145960220 Ki = 1.8 nM T37541 C6JND4 145960287 Ki = 0.68 nM T37541 C6JG2V 145961631 Ki = 0.28 nM T37541 CD9I1U 145971467 Ki = 27.1 nM T37541 CGE23X 145972719 Ki = 295.6 nM T37541 CSPH69 145979414 Ki = 11.4 nM T37541 CQDB02 145979430 Ki = 49.6 nM T37541 CUDO01 145979473 Ki = 135.3 nM T37541 CIF72X 145979737 Ki = 125.9 nM T37541 CLFJ74 145980146 Ki = 6.2 nM T37541 C9S0WG 145983404 Ki = 132.2 nM T37541 CB5G4W 145983664 Ki = 750.9 nM T37541 C8C0AB 145984626 Ki = 118.2 nM T37541 CN56XE 145986933 Ki = 147.7 nM T37541 CZPA17 145987454 Ki = 78.8 nM T37541 CJ1P5W 145988462 Ki = 127.4 nM T37541 C1LV0U 145988936 Ki = 606.7 nM T37541 C9RVK0 145989853 Ki = 17.8 nM T37541 CHMR39 145990191 Ki = 41.5 nM T37541 CYOD69 145990290 Ki = 98.4 nM T37541 CZB2X3 145990392 Ki = 121.5 nM T37541 CB63XC 145990519 Ki = 180.8 nM T37541 C3QXL4 145991981 Ki = 94.7 nM T37541 C7RYJ4 145992796 Ki = 147.1 nM T37541 CE34YK 145992956 Ki = 72 nM T37541 C48CZD 146160385 Ki = 16.1 nM T37541 C6FD2N 147348395 Ki = 2565 nM T37541 C1PG9M 155511036 Ki = 2.7 nM T37541 CN6DW9 155511075 Ki = 25 nM T37541 CJA94W 155512108 Ki = 0.72 nM T37541 CZ5W1M 155514230 Ki = 3589.4 nM T37541 CM5J3L 155514471 Ki = 18.1 nM T37541 CDM78Q 155514660 Ki = 18.9 nM T37541 CCQB03 155515285 Ki = 37.2 nM T37541 CT2ZB0 155515980 Ki = 1 nM T37541 CZN16J 155516304 Ki = 69 nM T37541 COP4Q6 155516517 Ki = 5.4 nM T37541 C2E0ZF 155517026 Ki = 56.4 nM T37541 CAG9L4 155517430 Ki = 3.6 nM T37541 C1VNX3 155518220 Ki = 31.4 nM T37541 CEH62Y 155518447 Ki = 5.6 nM T37541 CP7UI1 155518510 Ki = 6.2 nM T37541 C8MYG2 155519248 Ki = 12.2 nM T37541 CO6D1Y 155519288 Ki = 41.5 nM T37541 CC47MV 155519432 Ki = 85.4 nM T37541 CO4V0B 155519627 Ki = 44.4 nM T37541 CIV68R 155520019 Ki = 38.2 nM T37541 CP49HE 155520274 Ki = 4.7 nM T37541 C8E0SN 155520671 Ki = 4900 nM T37541 C4LPA1 155520806 Ki = 792.4 nM T37541 CQ0OR1 155520930 Ki > 10000 nM T37541 C2J1YG 155521041 Ki = 15.4 nM T37541 CCGT71 155521462 Ki = 3.1 nM T37541 CF7HE1 155521700 Ki = 5.8 nM T37541 CZ7WI8 155521830 Ki = 23.5 nM T37541 C6AWP0 155522679 Ki = 4.8 nM T37541 C3HGK6 155523328 Ki = 5.5 nM T37541 CSC58M 155524279 Ki > 10000 nM T37541 C9PV5X 155524649 Ki > 100000 nM T37541 CS21YC 155524712 Ki = 86.3 nM T37541 C70ZPH 155524915 Ki = 5.3 nM T37541 CA02GS 155526086 Ki = 85.5 nM T37541 CWGS97 155526825 Ki = 609 nM T37541 CAMY18 155527145 Ki = 4.3 nM T37541 CDE96Y 155527673 Ki = 55.2 nM T37541 CLF2V0 155528496 Ki = 28.6 nM T37541 C38SKR 155528605 Ki = 68.1 nM T37541 CB08MU 155528753 Ki > 100000 nM T37541 C2LF1H 155528761 Ki = 69.3 nM T37541 CN27OU 155528858 Ki = 488.1 nM T37541 CECZ45 155529036 Ki = 363.3 nM T37541 C8DN2F 155529373 Ki = 304.1 nM T37541 CG3J0Q 155529984 Ki = 55 nM T37541 CKO2V5 155530358 Ki = 71.3 nM T37541 CIGQ50 155530440 Ki = 30.4 nM T37541 CTJ3I7 155530506 Ki = 4.7 nM T37541 CO7P5W 155531268 Ki = 0.68 nM T37541 CLMZ93 155531382 Ki = 9.3 nM T37541 CW6TC5 155531936 Ki = 3100 nM T37541 C5H8QF 155532861 Ki = 893 nM T37541 C0BNY7 155533528 Ki = 52.2 nM T37541 C78ZFI 155534074 Ki = 11.9 nM T37541 CT5NG1 155534179 Ki = 0.2 nM T37541 CS0FK9 155534753 Ki = 78.7 nM T37541 CE1I8S 155535343 Ki = 273 nM T37541 CVU5P6 155535355 Ki = 1.5 nM T37541 CV0N9I 155535382 Ki > 10000 nM T37541 CKR07J 155535598 Ki > 10000 nM T37541 CNFR72 155535756 Ki > 100000 nM T37541 CFYA23 155535780 Ki = 33.9 nM T37541 CD2O3A 155535852 Ki = 810 nM T37541 CZPY79 155536184 Ki = 210.1 nM T37541 C0EDQ2 155536876 Ki = 65.1 nM T37541 CZ0T6A 155537018 Ki = 3949 nM T37541 COP2R4 155537042 Ki = 48.3 nM T37541 C4K0MB 155537772 Ki = 870 nM T37541 CYM0A3 155538069 Ki = 70.2 nM T37541 C5RV9W 155538073 Ki = 81.7 nM T37541 COX74J 155538083 Ki = 62.8 nM T37541 C9AP8F 155538224 Ki = 20.8 nM T37541 C9K2TL 155539730 Ki = 1690 nM T37541 CS1G5V 155539783 Ki = 75.5 nM T37541 CS1UR7 155539868 Ki = 78.8 nM T37541 CSAD81 155540401 Ki = 13.5 nM T37541 CZ8FJ3 155540422 Ki = 58 nM T37541 C8RV6T 155541805 Ki = 3.7 nM T37541 CW96ES 155541807 Ki = 1.1 nM T37541 C4MW9Q 155541811 Ki = 79.2 nM T37541 CZ2CT0 155542259 Ki = 534 nM T37541 CW61DF 155542555 Ki = 46.6 nM T37541 CT9GZ2 155542660 Ki = 1034.1 nM T37541 CDK2W5 155542691 Ki = 34.6 nM T37541 C75TVG 155542954 Ki = 261.9 nM T37541 C2AEH6 155543096 Ki = 355 nM T37541 CN2SJ7 155543228 Ki = 48.1 nM T37541 C19DJA 155543271 Ki = 647 nM T37541 CI2T8N 155544664 Ki = 49.4 nM T37541 CY6SX5 155545800 Ki > 100000 nM T37541 C83ZIS 155547526 Ki = 36 nM T37541 CW19PC 155547551 Ki = 94.5 nM T37541 C73YLV 155547628 Ki = 0.8 nM T37541 C61MSB 155547730 Ki = 0.78 nM T37541 CQG5F9 155548326 Ki = 15.7 nM T37541 CU1NE7 155549031 Ki = 3 nM T37541 CA25QH 155549266 Ki = 43.3 nM T37541 CR79SY 155549354 Ki = 705 nM T37541 C4O6TN 155550616 Ki = 17 nM T37541 CMWQ79 155550618 Ki = 916.3 nM T37541 C6XPV0 155550626 Ki = 85.4 nM T37541 C4S0JZ 155551334 Ki = 100.8 nM T37541 COC4Z9 155551784 Ki = 18.9 nM T37541 CZ0T3C 155551786 Ki = 3.5 nM T37541 CG9PN8 155552113 Ki = 3 nM T37541 CW8S7L 155552594 Ki = 96.4 nM T37541 C0OG8P 155553361 Ki = 0.38 nM T37541 CP15VC 155553400 Ki > 50000 nM T37541 C1R7CJ 155553759 Ki = 34 nM T37541 CMEP40 155554179 Ki = 30.5 nM T37541 CZU9Y7 155554800 Ki = 46.3 nM T37541 C5YA7C 155555084 Ki = 46.8 nM T37541 CWB82E 155555878 Ki = 5.1 nM T37541 CD4K6H 155556521 Ki = 0.55 nM T37541 CJF9O7 155557300 Ki > 100000 nM T37541 C40MOH 155557452 Ki = 2.9 nM T37541 CH1Z2S 155558695 Ki = 910 nM T37541 CXE2R9 155561928 Ki = 63.7 nM T37541 C6KD7C 155563215 Ki = 761.5 nM T37541 CP85AZ 155563623 Ki = 41.3 nM T37541 C07GFY 155564664 Ki = 80.6 nM T37541 C0E4QV 155565149 Ki = 6.1 nM T37541 CNL8B7 155565372 Ki = 584.9 nM T37541 CJ7I6Z 155565419 Ki = 7.7 nM T37541 COA9F8 155566222 Ki = 8700 nM T37541 CCW3L7 155566305 Ki = 735 nM T37541 CJQP47 155566378 Ki = 9.5 nM T37541 CI8U3W 155566755 Ki = 174.5 nM T37541 CDB8T4 155568445 Ki = 4.4 nM T37541 C94QKZ 155568447 Ki = 3323 nM T37541 CH5VU6 155568899 Ki = 4.4 nM T37541 C1C2GI 155569076 Ki = 0.63 nM T37541 C83MGT 155569151 Ki = 46.3 nM T37541 C1A7IN 155569676 Ki = 4.4 nM T37541 D00FGB 11414131 Ki = 10 nM T37541 D00GVA 44520904 Ki = 7.9 nM T37541 D00IUB 13019 Ki = 777000 nM T37541 D00RNZ 910172 Ki = 15300 nM T37541 D00XIB 11680415 Ki = 1.7 nM T37541 D00XJA 711717 Ki = 50500 nM T37541 D00YEF 148885 Ki = 92.3 nM T37541 D01BUB 94952 Ki = 554000 nM T37541 D01ISX 670786 Ki = 7.6 nM T37541 D01STY 9861037 Ki = 150 nM T37541 D01UYI 5281607 Ki = 171.41 nM T37541 D02DBP 5054 Ki = 644000 nM T37541 D02QGI 273 Ki = 420 nM T37541 D03DAM 2725651 Ki = 7200 nM T37541 D03NBX 637308 Ki = 620 nM T37541 D03ZMQ 323 Ki = 3300 nM T37541 D04CVC 4687472 Ki = 75 nM T37541 D04HRS 404195 Ki = 46 nM T37541 D04NSN 169682 Ki = 80 nM T37541 D05QOR 5280460 Ki = 8710 nM T37541 D05QUG 45485279 Ki = 44500 nM T37541 D05TLB 11117301 Ki = 76.6 nM T37541 D05WQF 637540 Ki > 1000000 nM T37541 D05XZM 10081162 Ki = 60 nM T37541 D06ALC 6441498 Ki = 268.3 nM T37541 D06DYP 234562 Ki = 32400 nM T37541 D06XNT 4119643 Ki = 6.8 nM T37541 D07CYN 20347846 Ki = 1.6 nM T37541 D07LYW 11537386 Ki = 9.3 nM T37541 D07MTM 403 Ki = 1359000 nM T37541 D07PNA 11660633 Ki = 1.9 nM T37541 D07QJJ 289 Ki = 714000 nM T37541 D07TAJ 914298 Ki = 9700 nM T37541 D07YDN 5281654 Ki = 4.4 nM T37541 D08AIJ 440735 Ki = 4.3 nM T37541 D08AOA 11543564 Ki = 3.9 nM T37541 D08BFU 5282102 Ki = 423.7 nM T37541 D09JPC 16402 Ki = 440 nM T37541 D09LWR 3433937 Ki = 5.5 nM T37541 D09PWX 8739 Ki = 52 nM T37541 D09TES 44395768 Ki = 7.1 nM T37541 D09WSJ 19772348 Ki = 88.9 nM T37541 D09WVV 8111 Ki = 12100 nM T37541 D0A0YX 5143 Ki = 10 nM T37541 D0A1CM 5281855 Ki = 6320 nM T37541 D0A3JR 3051968 Ki = 6.9 nM T37541 D0A8HW 44395685 Ki = 1.5 nM T37541 D0AU0M 637542 Ki = 5230 nM T37541 D0C4QB 44395769 Ki = 8 nM T37541 D0C7LR 313 Ki = 1840000 nM T37541 D0D4OV 20043772 Ki = 79.6 nM T37541 D0D5XC 101753 Ki = 36150000 nM T37541 D0D6UR 12394434 Ki = 3700 nM T37541 D0E0RW 69894 Ki = 23800 nM T37541 D0E8CC 18794 Ki = 0.45 nM T37541 D0EJ9B 66827 Ki = 8300 nM T37541 D0G0FJ 11206245 Ki = 68 nM T37541 D0G3BI 25090 Ki = 32 nM T37541 D0G3TK 5280863 Ki = 25 nM T37541 D0G9NE 11659798 Ki = 8.2 nM T37541 D0H3NS 10752 Ki = 6200 nM T37541 D0HN0R 11623958 Ki = 0.78 nM T37541 D0IB3K 5320686 Ki = 4.6 nM T37541 D0J3SP 11718391 Ki = 6.8 nM T37541 D0KZ2D 11638641 Ki = 1.7 nM T37541 D0L5TZ 20195365 Ki = 17100 nM T37541 D0LC0F 96876 Ki = 5.1 nM T37541 D0LU4S 156219 Ki = 4100 nM T37541 D0M3PO 69561 Ki = 100 nM T37541 D0M6RM 7365 Ki = 12500 nM T37541 D0N1AW 45485270 Ki = 9000 nM T37541 D0N7WP 44520903 Ki = 7.7 nM T37541 D0NN3Q 78105 Ki = 89 nM T37541 D0O0UE 729977 Ki = 4.7 nM T37541 D0O4KL 11640067 Ki = 1.9 nM T37541 D0O8WV 11536481 Ki = 4.5 nM T37541 D0O9VU 44520901 Ki = 5.4 nM T37541 D0OI1H 72894 Ki = 45 nM T37541 D0OT5L 1631814 Ki = 7100 nM T37541 D0P6AM 3526523 Ki = 61 nM T37541 D0Q7DJ 10742 Ki = 7810 nM T37541 D0RB0D 44268050 Ki = 30100 nM T37541 D0S9YX 5280373 Ki = 371.5 nM T37541 D0SF3B 11529486 Ki = 6.5 nM T37541 D0SY2M 5281708 Ki = 4.2 nM T37541 D0T3NP 7456 Ki = 780 nM T37541 D0TY8X 31036 Ki = 6.8 nM T37541 D0U4BB 10748 Ki = 2400 nM T37541 D0V9EN 689043 Ki = 6420 nM T37541 D0VD7H 84724 Ki = 5.2 nM T37541 D0W1OR 7424 Ki = 7170 nM T37541 D0W9VC 670143 Ki = 6.2 nM T37541 D0X5HL 15107 Ki = 360 nM T37541 D0X6IE 4422372 Ki = 5.6 nM T37541 D0XL5K 67944 Ki = 4 nM T37541 D0Y3TZ 370 Ki = 6070 nM T37541 D0Y7HG 5281616 Ki = 24.5 nM T37541 D0YU8J 1502014 Ki = 120 nM T37541 D0Z1HY 67136 Ki = 210 nM T37541 D0Z5GE 44520902 Ki = 5.3 nM T37541 D0ZC3W 6269 Ki = 88 nM T59626 D09JUG 60490 IC50 = 420 nM T59626 D0O4NR 5280492 Ki = 0.12 nM T59626 D0S0WN 114999 IC50 = 1 nM T59626 D0DK4I 4534 IC50 = 85 nM T59626 D0NS6I 10037501 Ki = 100000 nM T59626 D00GNK 177941 Ki = 25 nM T59626 D01XMO 192617 Ki = 0.04 nM T59626 D04JJE 132425 IC50 = 60 nM T59626 D05LYL 196905 IC50 = 1.5 nM T59626 D09LQP 132379 Ki = 0.14 nM T59626 D0B6JV 6435820 Ki = 7.1 nM T59626 D0C0EO 9867257 IC50 = 8.4 nM T59626 D0G7SP 6441619 Ki = 0.78 nM T59626 D0JY4Y 443292 IC50 = 210 nM T59626 D0NK8D 204058 Ki = 1.3 nM T59626 D0OP7B 6450158 Ki = 5.9 nM T59626 D0U9JL 6444688 IC50 = 1.9 nM T59626 D0Y2IH 122023 Ki = 77 nM T59626 D0Z0OT 6438358 Ki = 3.7 nM T59626 D0Z1TF 9850974 Ki = 1 nM T59626 CPVH47 129065 IC50 = 30 nM T59626 CY35ZC 178581 IC50 = 20 nM T59626 C6E7UC 192624 Ki = 3.467 nM T59626 C2DP3F 195214 IC50 = 210 nM T59626 C4JBN5 204055 IC50 = 3.2 nM T59626 CLJ1V0 3083459 Ki = 4.677 nM T59626 CLG18V 6439436 Ki = 4.7 nM T59626 CBM47Q 6852392 Ki = 700 nM T59626 COF3U8 9800998 Ki = 38000 nM T59626 CQ94JS 9805394 IC50 = 2.4 nM T59626 CVP13O 9807782 Ki = 4 nM T59626 C92QAN 9826485 Ki = 280 nM T59626 CS4D7L 9829619 Ki = 14 nM T59626 C4GI1E 9845585 Ki = 33.88 nM T59626 CF04AP 9845587 Ki = 61.66 nM T59626 CM76TV 9849151 IC50 = 610 nM T59626 CRS48K 9850643 Ki = 1 nM T59626 CVP79S 9865985 IC50 = 1 nM T59626 C78PTA 9872540 Ki = 42 nM T59626 CMGA15 9911868 IC50 = 7 nM T59626 CF7Y2J 9912012 Ki = 3.51 nM T59626 C67CBX 9930128 IC50 = 15.9 nM T59626 C5NBC4 9934323 IC50 = 43 nM T59626 CX38IE 9934500 IC50 = 800 nM T59626 CJSG78 9955657 IC50 = 4 nM T59626 CHY6Q3 9958441 Ki = 1.5 nM T59626 CFP2X1 9959228 Ki = 80 nM T59626 CLH47O 9976757 IC50 = 4 nM T59626 C0JM4I 9976891 IC50 = 8000 nM T59626 CHV5W2 9978895 IC50 = 6 nM T59626 CKLU93 9980059 IC50 = 1200 nM T59626 CDN4R5 9984593 Ki = 15.4 nM T59626 CGJ5W3 9985159 IC50 = 1150 nM T59626 C2JAZ3 9999718 IC50 = 40 nM T59626 CZ21UT 9999755 IC50 = 10 nM T59626 CI9NV6 10001576 IC50 = 5 nM T59626 CPJ5S8 10007005 IC50 = 25 nM T59626 CHF5J3 10019853 IC50 = 700 nM T59626 CH4U8L 10021622 IC50 = 2000 nM T59626 CV2HL3 10022413 IC50 = 45 nM T59626 CGL59Z 10023244 IC50 = 5 nM T59626 CCT4B7 10024190 IC50 = 110 nM T59626 CZ79EA 10032156 IC50 = 5800 nM T59626 CPUH04 10046386 IC50 = 2500 nM T59626 CC18QV 10046878 IC50 = 4 nM T59626 CYFS74 10047140 IC50 = 5 nM T59626 CFGB01 10050724 Ki = 4.8 nM T59626 C1CZP6 10052488 IC50 = 1100 nM T59626 COIH64 10052575 IC50 = 93 nM T59626 C8S0KE 10053028 IC50 = 320 nM T59626 CH5J9D 10053662 IC50 = 12.3 nM T59626 CD1O6X 10068808 IC50 = 400 nM T59626 C9CP2E 10069416 IC50 = 15 nM T59626 CNW4B1 10069417 IC50 = 1100 nM T59626 CIQS13 10071290 IC50 = 10000 nM T59626 CD7AP1 10090758 IC50 = 40 nM T59626 C85COL 10091738 IC50 = 13 nM T59626 CR45PL 10092630 IC50 = 9.5 nM T59626 C4A1IL 10120811 Ki = 0.14 nM T59626 CK4UL8 10159791 Ki = 58.88 nM T59626 C0K3FJ 10179915 Ki = 3.02 nM T59626 C5DH9M 10182429 Ki = 20.42 nM T59626 CI8DY3 10247237 IC50 = 550 nM T59626 CQ2R1G 10248148 IC50 = 183 nM T59626 COX86A 10250881 IC50 = 150 nM T59626 C7IR8W 10257351 Ki = 8 nM T59626 C73LQM 10314767 IC50 = 300 nM T59626 CK0W8I 10315808 IC50 = 1800 nM T59626 CYK46J 10318241 IC50 = 5 nM T59626 C1B8HI 10319829 IC50 = 22 nM T59626 C7XK2U 10324028 Ki = 28 nM T59626 CAES31 10325873 Ki = 240 nM T59626 CC1UF0 10335738 IC50 < 100 nM T59626 CFHI60 10337448 IC50 = 700 nM T59626 CHU5F0 10339300 IC50 = 68.2 nM T59626 C5X4IP 10340408 IC50 = 500 nM T59626 CMR45D 10341135 IC50 = 50 nM T59626 CV1KW5 10341242 IC50 = 2 nM T59626 CC3VK8 10342316 Ki = 38.02 nM T59626 CKH19Z 10343923 IC50 = 2 nM T59626 CB58OJ 10346127 Ki = 9.2 nM T59626 CCYB57 10347709 IC50 = 890 nM T59626 CH71MO 10349070 IC50 = 750 nM T59626 CQZ6S3 10362331 IC50 = 30 nM T59626 C2UW4Y 10363485 Ki = 38000 nM T59626 CP7IQ1 10363959 IC50 = 600 nM T59626 CZIL76 10364772 IC50 = 4.2 nM T59626 C6FS8B 10371282 Ki = 53 nM T59626 C5XYM3 10385899 IC50 = 10 nM T59626 CF9RH8 10386030 IC50 = 200 nM T59626 C2X5KM 10387303 IC50 = 300 nM T59626 CR9Q0B 10387480 IC50 = 30 nM T59626 CN1KZ9 10390056 IC50 = 150 nM T59626 C6M8ZS 10391552 IC50 = 520 nM T59626 CD05VJ 10406292 IC50 = 3 nM T59626 C2SCY7 10407131 IC50 = 300 nM T59626 CN0WY3 10407251 IC50 = 100 nM T59626 CZ1PY3 10415106 IC50 = 44500 nM T59626 C25MYB 10425738 IC50 < 100 nM T59626 C6V2ZW 10427789 IC50 = 50 nM T59626 C2PRE8 10430674 IC50 = 18 nM T59626 CJM40K 10430678 IC50 = 300 nM T59626 C2DHB5 10430946 IC50 = 2000 nM T59626 C8G7SN 10436331 IC50 = 5.2 nM T59626 C1HD2M 10451768 IC50 = 30 nM T59626 CE5VO0 10455429 IC50 = 300 nM T59626 C59MAC 10474073 IC50 > 1000 nM T59626 C5CQU8 10474602 IC50 = 15 nM T59626 C16TRD 10475503 IC50 = 5 nM T59626 C0CD8E 10475982 Ki = 16000 nM T59626 CU7FJ6 10477988 IC50 = 20 nM T59626 C6OV4L 10481412 IC50 = 770 nM T59626 C7WUL1 10482767 IC50 = 26 nM T59626 CQ23JE 10483151 IC50 = 2800 nM T59626 CWS3I5 10507666 Ki = 36 nM T59626 CK9MR2 10529082 Ki = 1.2 nM T59626 CK1X4N 10529241 Ki = 1.3 nM T59626 CJ9OI2 10554820 Ki = 33 nM T59626 CS65WD 10600128 Ki = 66.07 nM T59626 CEYL09 10625086 IC50 > 300 nM T59626 CH3FV2 10648186 Ki = 1.4 nM T59626 CSAF60 10670634 Ki = 63.1 nM T59626 CQ4S9P 10692884 Ki = 9.5 nM T59626 C3YMX7 10694814 Ki = 2.8 nM T59626 C5FXV6 10737187 IC50 = 900 nM T59626 CGT19D 10741106 IC50 = 80 nM T59626 C35FCG 10745069 Ki = 25 nM T59626 C35LWJ 10745838 Ki = 0.11 nM T59626 CMV5O6 10793277 Ki = 5.9 nM T59626 CO36IA 10812265 Ki = 16.22 nM T59626 CKH76L 11725988 IC50 = 500 nM T59626 C5WMJ9 11726048 IC50 = 150 nM T59626 CRDS63 11740566 IC50 = 800 nM T59626 CAO1X6 11741184 IC50 = 1000 nM T59626 CJP4L1 11756030 IC50 = 100 nM T59626 C24LXS 11798329 Ki = 12 nM T59626 CG1TE6 11798848 Ki = 1.5 nM T59626 C4EZ9M 11799000 IC50 = 60 nM T59626 CSR1I5 11800543 Ki = 12 nM T59626 C7HA8C 14282627 IC50 = 26200000 nM T59626 CS8T7E 14946858 IC50 = 100 nM T59626 C5MO7U 14977894 Ki = 429 nM T59626 CRH1W3 14977898 Ki = 165 nM T59626 C8VTF9 14977907 Ki = 1130 nM T59626 C1G0DR 14977911 Ki = 338 nM T59626 CK6B9V 14977913 Ki = 150 nM T59626 CWNE34 14977916 Ki = 478 nM T59626 C4WAQ7 14977920 Ki = 252 nM T59626 C76KWU 14977924 Ki = 151 nM T59626 C5IT0Y 14977927 Ki = 284 nM T59626 CZCJ15 14977931 Ki = 34 nM T59626 CL46SC 14977933 Ki = 36 nM T59626 C1VS5J 14977939 Ki = 74 nM T59626 CPR26X 14977943 Ki = 72 nM T59626 CDPY62 14977946 Ki = 148 nM T59626 CT59OE 14977948 Ki = 609 nM T59626 CC42FK 14977952 Ki = 147 nM T59626 CV70FZ 14977955 Ki = 789 nM T59626 C8RJ2H 14977957 Ki = 36 nM T59626 C81AXN 14977959 Ki = 11 nM T59626 C45IKJ 14977961 Ki = 43 nM T59626 C73MEH 14977963 Ki = 14 nM T59626 CPQ5E3 14977965 Ki = 12 nM T59626 CK79ZP 15227776 Ki = 3.53 nM T59626 C8JPS3 15658097 Ki = 900 nM T59626 CAX32C 15658098 Ki = 1400 nM T59626 CRZV56 15658099 Ki = 2800 nM T59626 CJ5R9F 15658119 Ki = 600 nM T59626 C80ROL 15658122 Ki = 140 nM T59626 CT83ZJ 15658147 Ki = 1 nM T59626 C2KPE8 15666575 IC50 = 10000 nM T59626 CH1QG8 15666577 IC50 = 1000 nM T59626 C5Z7NC 15666578 IC50 = 1000 nM T59626 C9FEK1 15666579 IC50 = 1000 nM T59626 CT4IA8 15666581 IC50 = 5000 nM T59626 C1EG6H 15666582 IC50 = 3000 nM T59626 CBC62V 15666586 IC50 = 700 nM T59626 CV67IJ 15666588 IC50 = 300 nM T59626 CEDG15 15666597 IC50 = 10000 nM T59626 C9WXO4 15666601 IC50 = 3500 nM T59626 C83QOF 15666603 IC50 = 1000 nM T59626 CH07PD 15666610 IC50 = 4500 nM T59626 C2CSJ4 15666613 IC50 = 1500 nM T59626 C9BL8Z 15666614 IC50 = 300 nM T59626 CFQ59K 15666615 IC50 = 200 nM T59626 CX1UQ4 15666618 IC50 = 110 nM T59626 CL86KV 15666621 IC50 = 1000 nM T59626 C8PU5J 15666623 IC50 = 800 nM T59626 C5LOM8 15666630 IC50 = 3000 nM T59626 C3N8MR 15666631 IC50 = 6000 nM T59626 CSH98I 15718079 IC50 = 1766 nM T59626 C0R7QD 15718082 IC50 = 2097 nM T59626 CV0YI1 15718085 IC50 = 832 nM T59626 CC2ER7 15839729 IC50 = 39.6 nM T59626 CJMU02 15839731 Ki = 4.96 nM T59626 CO70YW 15839732 Ki = 18.5 nM T59626 C7T8QY 15839733 Ki = 15.5 nM T59626 CCSA24 15839735 IC50 = 190 nM T59626 C0IX4S 15839751 Ki = 1.2 nM T59626 C0HRV3 18373300 IC50 = 500 nM T59626 C5GXB8 18373357 IC50 = 400 nM T59626 CDM6Q7 18373405 IC50 = 400 nM T59626 C9HF6C 18963032 Ki = 1.93 nM T59626 C7NL1V 19600933 Ki = 0.073 nM T59626 C8W2UP 21765772 Ki = 5.7 nM T59626 CD4K3V 21765774 Ki = 161 nM T59626 CMZU98 21765776 Ki = 112 nM T59626 CIF6K8 23257866 Ki = 129 nM T59626 CTBZ01 23257882 Ki = 245 nM T59626 CG0XA7 23257889 Ki = 192 nM T59626 CRG1H3 23257891 Ki = 232 nM T59626 CE2NF8 23257894 Ki = 37 nM T59626 C3TVL7 23501721 IC50 = 0.48 nM T59626 C90URE 23672801 Ki = 100 nM T59626 C3AP9Q 23672802 Ki = 50 nM T59626 CB9CM0 23672803 Ki = 9000 nM T59626 C2V8OU 23672804 Ki = 500 nM T59626 CZM4J7 23672805 Ki = 1 nM T59626 CGW18L 23672806 Ki = 60 nM T59626 CM9FX3 23672807 Ki = 3 nM T59626 CJ34EX 23672808 Ki = 1000 nM T59626 CC6PW9 23682552 IC50 = 300 nM T59626 C3A8CU 23699208 Ki = 10.3 nM T59626 CJMZ37 25174150 IC50 = 0.07 nM T59626 CVB0H8 25191879 IC50 = 0.18 nM T59626 C3JX1S 25191880 IC50 = 0.2 nM T59626 CV3TA6 25192021 IC50 = 0.21 nM T59626 C9WI6J 25192023 IC50 = 0.22 nM T59626 C2W9JA 25192174 IC50 = 0.36 nM T59626 CGV6N8 25192175 IC50 = 0.39 nM T59626 C7E8AM 25192176 IC50 = 0.38 nM T59626 CX3P6J 25192325 IC50 = 0.57 nM T59626 CO1E8H 25192326 IC50 = 0.58 nM T59626 CC6OR8 25192327 IC50 = 0.58 nM T59626 C9UL8Y 25192468 IC50 = 0.61 nM T59626 C7A8UE 25192471 IC50 = 1.19 nM T59626 CYK6X5 44213761 IC50 = 300 nM T59626 CP1F9I 44270188 Ki = 15.4 nM T59626 CA73JM 44275225 IC50 > 2000 nM T59626 CRM07V 44290966 Ki = 65.7 nM T59626 CZ8S4B 44291011 IC50 = 6.6 nM T59626 C7VKX3 44291012 IC50 = 35.6 nM T59626 CY5Q3Z 44291013 IC50 = 30.8 nM T59626 C24UOY 44291014 IC50 = 41.5 nM T59626 CG39HS 44291030 IC50 = 12 nM T59626 CM2A0S 44291031 Ki = 4.75 nM T59626 CDO50G 44296838 IC50 = 3800 nM T59626 CRGM38 44302134 Ki = 6.8 nM T59626 CP81YA 44302954 Ki = 5.53 nM T59626 C2GA3P 44302962 Ki = 28.4 nM T59626 C07QMJ 44302965 Ki = 3.2 nM T59626 C3MJH6 44302966 Ki = 320 nM T59626 CGQ38X 44302971 Ki = 5.14 nM T59626 C9XI2B 44302983 Ki = 6.51 nM T59626 CLT39P 44315538 IC50 = 70000 nM T59626 CE06WF 44315582 IC50 = 8000 nM T59626 CFU18I 44315784 IC50 = 1000 nM T59626 CQ0U2I 44317392 IC50 = 319 nM T59626 CAIE35 44337707 IC50 = 1200 nM T59626 CKL2R3 44340786 Ki = 10 nM T59626 C5E9JY 44341073 Ki = 27000 nM T59626 CY3XG6 44341107 Ki = 19000 nM T59626 CXJ7K3 44341141 Ki = 225 nM T59626 C1JQ9S 44341265 Ki = 9000 nM T59626 C1QIP7 44341318 Ki = 2400 nM T59626 CA39XW 44348541 IC50 = 50 nM T59626 CS9G0A 44356239 IC50 = 4700 nM T59626 C35ENC 44357534 IC50 = 50 nM T59626 C2S4FU 44357546 IC50 = 7 nM T59626 CLIK19 44359651 IC50 = 400 nM T59626 CE5Z1Q 44379572 IC50 = 6000 nM T59626 CS7I2Y 44379573 IC50 = 2000 nM T59626 C6PUO7 44379592 IC50 = 2000 nM T59626 CI2VA5 44379910 IC50 > 10000 nM T59626 C3JC5B 44381856 IC50 = 15.5 nM T59626 CL8B3S 44382275 Ki = 330 nM T59626 C4HZU0 44382276 Ki = 5200 nM T59626 C4N9UJ 44382378 IC50 = 220 nM T59626 CU8SD4 44382384 Ki = 3300 nM T59626 CEU1A0 44382463 Ki = 39000 nM T59626 C05WVE 44382468 Ki = 1900 nM T59626 CAOW45 44384957 IC50 = 784 nM T59626 CJT8L2 44384958 IC50 = 276 nM T59626 C93RQX 44385131 IC50 = 1180 nM T59626 CQ3AK6 44385159 IC50 = 1220 nM T59626 C8Y5RF 44385160 IC50 = 4570 nM T59626 C4M3OJ 44385199 IC50 = 1510 nM T59626 C1TZE0 44385218 IC50 = 1180 nM T59626 CA9FK0 44385257 IC50 > 10000 nM T59626 CQ5HY6 44385258 IC50 = 190 nM T59626 CAT57Z 44385920 IC50 = 830 nM T59626 CJQM34 44385966 IC50 = 932 nM T59626 C7X2YA 44386171 IC50 = 908 nM T59626 CRDA84 44386172 IC50 = 16.7 nM T59626 COL05K 46888195 IC50 = 8.5 nM T59626 CK20OJ 46888196 IC50 = 31.1 nM T59626 CXNZ90 46888197 IC50 = 5.35 nM T59626 CLK29W 46888198 IC50 = 5.39 nM T59626 C24FWR 46888199 IC50 = 139.7 nM T59626 C5A4PJ 46888200 IC50 = 13.98 nM T59626 C3BSZ4 46888201 IC50 = 3.27 nM T59626 CS6CR7 46888202 IC50 = 60.2 nM T59626 C62DUR 135401173 IC50 = 12 nM T59626 C8GIO2 135430350 IC50 = 738 nM T59626 C8YS2G 135457469 IC50 = 9.3 nM T59626 CV6YJ0 135500104 IC50 = 87 nM T59626 C1GON6 135503765 IC50 = 11 nM T59626 C1A9MF 135507183 IC50 = 54 nM T59626 C72JDF 135507225 IC50 = 55 nM T59626 CVB8W3 135507252 IC50 = 28 nM T59626 C84SWJ 135507273 IC50 = 834 nM T59626 C4V2EX 135516891 IC50 = 6.4 nM T59626 CCSR81 135531245 IC50 = 107 nM T59626 C6WFG1 135543741 IC50 = 82 nM T59626 C7MEH5 135543742 IC50 = 5.7 nM T59626 C4XA8E 135543808 IC50 = 4.5 nM T59626 D00HYO 20704716 Ki = 5300 nM T59626 D05HNB 9893718 Ki = 1.2 nM T59626 D06IJI 44379678 IC50 = 0.1 nM T59626 D07EGC 15817161 IC50 = 0.85 nM T59626 D09QJS 9958915 IC50 = 8.5 nM T59626 D0C2GW 44379453 IC50 = 0.15 nM T59626 D0F4EL 10021742 Ki = 1300 nM T59626 D0H6YL 44403368 IC50 = 8 nM T59626 D0L8VT 44403823 IC50 = 54 nM T59626 D0R9ED 15237280 IC50 = 5.3 nM T59626 D0V3ZG 25192022 IC50 = 114 nM T59626 D0ZB8S 44379679 IC50 < 0.1 nM T15571 D01AZG 5073 Ki = 1000 nM T15571 D01TSI 8223 Ki = 14 nM T15571 D03WEX 9966051 Ki = 220 nM T15571 D08VRO 3822 Ki = 20000 nM T15571 D0CQ0Z 33630 Ki = 1000 nM T15571 D0G8NN 119570 Ki > 10000 nM T15571 D0H3HM 60795 Ki = 1000 nM T15571 D0H7KF 5002 Ki > 1000 nM T15571 D0V4QS 135398745 Ki > 1000 nM T15571 D0W5HK 216239 Ki = 3296 nM T15571 D0Z1RV 135398737 Ki = 1000 nM T15571 D0Z6UC 5358 IC50 = 501.19 nM T15571 D0N1HW 5311200 Ki > 10000 nM T15571 D00OWF 5280953 Ki > 10000 nM T15571 D08AWI 11430856 Ki > 5000 nM T15571 D0M7LV 5761 Ki = 9 nM T15571 D0YP7L 6604889 Ki = 63.1 nM T15571 CUQ05A 3564 Ki > 10000 nM T15571 C2QLD4 3565 Ki > 10000 nM T15571 C5H9CN 9287 Ki > 10000 nM T15571 C6WDL7 49756 Ki = 10450 nM T15571 CHKO01 91522 Ki > 10000 nM T15571 CX1GC4 108182 Ki = 16000 nM T15571 CP9D2L 151142 Ki < 10 nM T15571 C6RSI8 159809 Ki > 10000 nM T15571 CGT8R0 160510 Ki = 845 nM T15571 CYV1R3 417052 Ki > 10000 nM T15571 CAH9F5 656705 Ki > 10000 nM T15571 C2VLP8 752521 Ki = 389 nM T15571 COG8R1 2058916 Ki > 10000 nM T15571 CA2OY6 2737389 Ki = 76 nM T15571 CS8KE2 3649661 Ki = 457 nM T15571 C6SHA4 4713248 Ki = 5000 nM T15571 C8HQN1 5376026 Ki > 10000 nM T15571 C3MA1N 9819150 IC50 = 794.33 nM T15571 CM13ZV 9856041 Ki > 10000 nM T15571 CJW1P5 9888494 Ki = 1479.11 nM T15571 CUN81Q 9905249 Ki > 10000 nM T15571 CYWQ50 9906447 Ki > 10000 nM T15571 CWC69L 9998879 IC50 = 501.19 nM T15571 CV7R9F 10020040 Ki > 10000 nM T15571 C86UFO 10021702 IC50 = 125.89 nM T15571 C2EUY0 10035109 Ki > 10000 nM T15571 C92UGJ 10043491 IC50 = 125.89 nM T15571 CH25VX 10245588 IC50 = 630.96 nM T15571 CH31DX 10267394 Ki > 10000 nM T15571 CU89JD 10314060 Ki > 10000 nM T15571 CAS0N1 10315894 IC50 = 199.53 nM T15571 C7M5TZ 10337965 IC50 = 251.19 nM T15571 C6C3HX 10340828 IC50 = 79.43 nM T15571 C8FB4S 10382508 Ki = 13 nM T15571 CP3OG2 10383252 IC50 = 1000 nM T15571 C9MXP8 10404070 IC50 = 1995.26 nM T15571 CHD23R 10404770 IC50 = 125.89 nM T15571 CYM5R8 10412397 IC50 = 199.53 nM T15571 C2B0IU 10421236 IC50 > 10000 nM T15571 C5RH4N 10471382 IC50 = 794.33 nM T15571 CY0EK4 10471383 IC50 = 794.33 nM T15571 COV85C 10472143 Ki = 27 nM T15571 CP8WN3 10872812 Ki = 200 nM T15571 CXP8H3 10881882 Ki = 930 nM T15571 CI9Z8E 10882775 Ki = 200 nM T15571 CRI50E 10885636 IC50 = 3380 nM T15571 CGI03V 10893866 Ki = 250 nM T15571 C1BF4J 10924201 Ki = 1920 nM T15571 CXFH06 10926167 Ki = 350 nM T15571 CNB39C 10947658 Ki = 16 nM T15571 C3X5OI 11035049 Ki = 190 nM T15571 C3AJ7L 11074351 Ki > 10000 nM T15571 CM9KX0 11088692 Ki = 1080 nM T15571 CVE8T3 11121216 Ki = 13 nM T15571 CS3YK5 11352884 Ki = 25.12 nM T15571 CF1O2M 11364267 Ki = 31.62 nM T15571 C85LYP 11430418 IC50 > 1000 nM T15571 C5C6ZJ 11443218 Ki = 125.89 nM T15571 CNH1K4 11568826 Ki > 10 nM T15571 CGX8F6 11596869 Ki > 6900000 nM T15571 C4L7TV 11662592 Ki > 1 nM T15571 C9X7EK 11722814 IC50 = 630.96 nM T15571 CE5C1J 11726973 Ki = 620 nM T15571 C7PVL8 11730467 IC50 = 5520 nM T15571 C7X4KL 11759441 Ki > 10000 nM T15571 CO9YM4 11808247 Ki = 400 nM T15571 CXLW54 11948707 Ki > 10000 nM T15571 C8JQL7 11957735 IC50 > 10000 nM T15571 C20RFT 14935215 Ki > 10000 nM T15571 C7VAI1 15011772 IC50 > 10000 nM T15571 C1LWZ6 16006605 Ki = 6.5 nM T15571 CK36NS 16006607 Ki = 10 nM T15571 CD3E8L 16093484 Ki = 2 nM T15571 CEW91O 16093485 Ki = 4.7 nM T15571 CZ2IS9 16660294 Ki > 10000 nM T15571 C7T8JC 19958494 Ki > 10000 nM T15571 C6LI5E 19958507 Ki > 10000 nM T15571 C3T5HF 21509921 Ki = 741.31 nM T15571 CT7XG9 21830793 Ki > 10000 nM T15571 CBN84K 22065997 Ki > 10000 nM T15571 CZ7J4B 22857296 Ki = 630 nM T15571 CDC91N 24839550 Ki < 10000 nM T15571 CY21RE 24841480 Ki = 2200 nM T15571 C3HK0J 24865725 Ki = 1258.93 nM T15571 C0O6FX 24865727 Ki = 1584.89 nM T15571 CUY89J 24936155 Ki = 3000 nM T15571 CJ3NP5 42636941 IC50 > 10000 nM T15571 CCP07F 44275750 Ki = 3 nM T15571 CC2OD4 44278111 Ki > 10000 nM T15571 CRMA84 44278114 Ki > 10000 nM T15571 CF0Y4M 44278115 Ki > 10000 nM T15571 CER86D 44327952 Ki = 200 nM T15571 CN3QX1 44351063 Ki = 1775 nM T15571 C57PAS 44351077 Ki = 285 nM T15571 C4WY3Z 44351100 Ki = 185 nM T15571 CR85QU 44351102 Ki = 174 nM T15571 CI47MT 44351116 Ki = 1120 nM T15571 C2J6RG 44351139 Ki = 100 nM T15571 CTF6U8 44351140 Ki = 100 nM T15571 CD1JZ2 44351180 Ki = 225 nM T15571 CP92MG 44351183 Ki = 1395 nM T15571 C7H6ZS 44351184 Ki = 165 nM T15571 CSW4B9 44351193 Ki = 270 nM T15571 CYO3S8 44351342 Ki = 168 nM T15571 CD5E1G 44374431 Ki = 287 nM T15571 CK28HY 44374637 Ki > 3448 nM T15571 C8EK9X 44374648 Ki = 3067 nM T15571 CA0W9E 44397360 Ki = 31.62 nM T15571 CL96VK 44397361 Ki = 79.43 nM T15571 C7YV9X 44397363 Ki = 25.12 nM T15571 C1AVF4 44397364 Ki = 5.012 nM T15571 CE2ZW4 44397426 Ki = 501.19 nM T15571 CO8J2L 44397428 Ki = 6309.57 nM T15571 CD85BN 44397430 Ki = 1000 nM T15571 CK7DX8 44397432 Ki = 630.96 nM T15571 CJ1UF5 44397434 Ki = 398.11 nM T15571 CS2E6D 44397486 Ki = 199.53 nM T15571 CODE60 44397510 Ki = 3162.28 nM T15571 C4K0MN 44397512 Ki = 251.19 nM T15571 C4B0OI 44397588 Ki = 25.12 nM T15571 C5FP0R 44397589 Ki = 50.12 nM T15571 C6GSJ1 44397592 Ki = 251.19 nM T15571 CYJF09 44397618 Ki = 12.59 nM T15571 C2AGC5 44397667 Ki = 199.53 nM T15571 CA46QM 44397668 Ki = 79.43 nM T15571 CE3G8U 44397670 Ki = 6.31 nM T15571 CG87PW 44409290 Ki > 720 nM T15571 CZL97F 44455426 Ki > 10000 nM T15571 CYS7T4 44455943 Ki = 26.5 nM T15571 CPJ16W 44455962 Ki = 415 nM T15571 CO7TM5 44455963 Ki = 122 nM T15571 C4DAW2 44455980 Ki = 1172 nM T15571 CGBA20 44455982 Ki > 10000 nM T15571 CY7B1J 44455985 Ki = 38 nM T15571 C6BFI0 44456033 Ki = 1.6 nM T15571 CCE8Z7 44456170 Ki = 1990 nM T15571 CBU1G5 44456207 Ki = 97 nM T15571 CTF4X6 44456246 Ki = 463 nM T15571 C5SYI3 44456251 Ki = 1375 nM T15571 C45ELH 44456253 Ki = 647 nM T15571 C1WX4S 44456284 Ki = 274 nM T15571 CB34EP 44456286 Ki = 911 nM T15571 CG91RD 44456395 Ki = 22.9 nM T15571 C4X0ZV 44456398 Ki = 882 nM T15571 C12XGE 44456400 Ki = 466 nM T15571 CYUQ72 44456443 Ki = 550 nM T15571 C6NE3T 44456487 Ki = 145 nM T15571 C4DL5C 44469677 IC50 = 1 nM T15571 CRCH48 44582675 Ki = 6814 nM T15571 CEJ4R8 44582676 Ki = 1584 nM T15571 CZGP86 44582677 Ki > 10000 nM T15571 C5QB4K 44582678 Ki > 10000 nM T15571 C01RCI 44582705 Ki = 1684 nM T15571 CXL25V 44582706 Ki > 10000 nM T15571 C8MR1X 44582707 Ki > 10000 nM T15571 C4IT1N 44582708 Ki > 10000 nM T15571 CVJ04W 45263888 Ki = 99 nM T15571 CZOG43 45266001 Ki = 347 nM T15571 C2LZJ0 49783209 Ki = 8589 nM T15571 C57SMG 49783415 Ki > 10000 nM T15571 C0TG6I 49783419 Ki > 10000 nM T15571 CR40BA 49836386 IC50 > 1000 nM T15571 C2RY0J 50878551 Ki = 3311.31 nM T15571 C1W6TV 50898777 Ki > 10000 nM T15571 CXMZ73 50898778 Ki > 10000 nM T15571 CE4KP1 51050257 Ki > 10000 nM T15571 CRQF15 53325242 Ki = 894 nM T15571 CG24AT 53381002 Ki = 1525 nM T15571 CH37LU 56663451 IC50 > 10000 nM T15571 C1TC7Q 56963799 Ki > 10000 nM T15571 C1LEH8 67268994 Ki > 10000 nM T15571 C3XNC2 71450247 Ki > 10000 nM T15571 C9VZ8J 71450550 Ki > 10000 nM T15571 CYK20Z 71452384 Ki > 10000 nM T15571 C7UCP8 71452650 Ki = 208 nM T15571 CAQF34 71455625 Ki > 10000 nM T15571 CMJ1O9 71457409 Ki > 10000 nM T15571 CS83IF 71459269 Ki = 1700 nM T15571 CK5T4P 71459604 Ki = 7815 nM T15571 C63YLA 71461049 Ki > 10000 nM T15571 CJD96I 71461050 Ki > 10000 nM T15571 C4P3JU 71462776 Ki = 5805 nM T15571 C3GUQ2 71462777 Ki > 10000 nM T15571 CWH6T3 72548703 IC50 = 106 nM T15571 C8Z0NM 72550642 Ki = 1178 nM T15571 CL6W2Q 72550645 Ki = 517 nM T15571 C78LYM 72698087 Ki > 10000 nM T15571 C63HPK 72698088 Ki > 10000 nM T15571 CC6Q5R 72771081 Ki < 100 nM T15571 CC65OA 73213195 Ki > 10000 nM T15571 CW83DK 73213196 Ki > 10000 nM T15571 CCV91B 73346042 Ki = 2128 nM T15571 C1NJ0R 73353884 Ki = 6060 nM T15571 C4F7VK 73355415 Ki = 7502 nM T15571 C2E7QW 75201901 Ki > 10000 nM T15571 C8IDL3 75306277 Ki = 199.53 nM T15571 CEMZ15 118464420 Ki = 227 nM T15571 CV2L6O 118464425 Ki = 595 nM T15571 CFNG86 118464427 Ki = 994 nM T15571 CLW53P 122483274 Ki = 337 nM T15571 CO63ET 122483280 Ki = 5 nM T15571 C4QM2E 124247485 Ki > 10000 nM T15571 CTBN56 127026052 Ki = 4265.8 nM T15571 C0SZI4 127026515 Ki = 933 nM T15571 CU49VE 127036186 Ki = 3235.94 nM T15571 CG06BD 127036932 Ki = 2089.3 nM T15571 CVW71O 127036953 Ki = 2398.83 nM T15571 C50GOC 130442480 Ki = 9500 nM T15571 CM04RF 130442572 Ki = 7400 nM T15571 C1RI8Q 132060720 Ki = 875 nM T15571 CGHO19 132060770 Ki > 10000 nM T15571 CT81OY 132060776 Ki = 1747 nM T15571 CAVB41 132584404 Ki > 10000 nM T15571 CBU81N 134149168 Ki > 10000 nM T15571 C6N8GM 135367405 Ki > 10000 nM T15571 C6LU0C 135367816 Ki > 10000 nM T15571 CD2TH9 135367820 Ki = 1231 nM T15571 C5AMD9 135367857 Ki = 1135 nM T15571 CVE08Y 135458392 Ki = 10.72 nM T15571 CP7HN4 135458393 Ki = 6.31 nM T15571 CS8XJ6 135458394 Ki = 6.3 nM T15571 C9B7XA 135458410 Ki = 5.7 nM T15571 CFV9A3 135458427 Ki = 22.2 nM T15571 CKX4N8 135458428 Ki = 28.2 nM T15571 CTE23K 135464118 Ki = 89 nM T15571 C7AGR0 135474338 Ki = 5355 nM T15571 C1CZ9M 135514796 Ki = 101 nM T15571 CA1M8B 135966709 Ki = 25.4 nM T15571 CUKO20 136020617 Ki > 10000 nM T15571 COF0U5 136020618 Ki > 10 nM T15571 CF89JI 136030596 Ki > 10000 nM T15571 CE8GB9 136030693 Ki > 10000 nM T15571 C65VFI 136030744 Ki > 10000 nM T15571 COIX80 136054961 Ki > 10000 nM T15571 C7JHO0 136100333 Ki = 1791 nM T15571 C19GLK 136116062 Ki = 33.4 nM T15571 CA3JC8 136118613 Ki = 1282 nM T15571 CQ2GP6 136118614 Ki = 2332 nM T15571 C6R4IC 136118615 Ki = 1550 nM T15571 CS0JL5 136118616 Ki = 1454 nM T15571 CHWC38 136118619 Ki = 1425 nM T15571 C5UDW3 136118620 Ki = 7828 nM T15571 CLH0V9 136118648 Ki = 3372 nM T15571 CR72MQ 136118651 Ki = 3324 nM T15571 C0W1TM 136118658 Ki = 5080 nM T15571 C40LYH 136118659 Ki = 9118 nM T15571 CZ7C3Y 136118660 Ki = 4681 nM T15571 C42FCS 136118661 Ki = 6913 nM T15571 CR3DK1 136118716 Ki = 123 nM T15571 CON04G 136118728 Ki = 184 nM T15571 COX1F8 136118729 Ki = 112 nM T15571 C0R5PV 136118732 Ki = 1323 nM T15571 CB7N0X 136152962 Ki = 103 nM T15571 C01THU 136152963 Ki = 1472 nM T15571 CB12QP 136152964 Ki = 6.8 nM T15571 CRK8C7 136152965 Ki = 124 nM T15571 CFX06E 136152966 Ki = 22.2 nM T15571 C1UKM5 136152967 Ki = 96 nM T15571 CX0R8L 136152968 Ki = 163 nM T15571 CB8A6N 136152969 Ki = 279 nM T15571 C1JQG9 136152970 Ki = 37 nM T15571 C37YXA 136152971 Ki = 1.8 nM T15571 CY0C1X 136152972 Ki = 504 nM T15571 CFQR93 136152973 Ki = 241 nM T15571 CTW8Y5 136152974 Ki = 176 nM T15571 C0WP1E 136152976 Ki = 488 nM T15571 CQXB23 136152977 Ki = 87 nM T15571 CD81KX 136152978 Ki = 397 nM T15571 CP2M7N 136152980 Ki = 189 nM T15571 C26MKZ 136152981 Ki = 153 nM T15571 C90OMK 136179599 Ki = 196 nM T15571 CAE39V 136188797 Ki > 10000 nM T15571 CLAP52 136259032 Ki > 10000 nM T15571 C7KC3T 145963830 Ki = 4700 nM T15571 CHDN35 145964150 Ki > 10000 nM T15571 C1KH2E 145964159 Ki > 10000 nM T15571 C12OVL 145965034 Ki > 10000 nM T15571 C5W4LM 145965940 Ki > 10000 nM T15571 C81VUO 145967771 Ki > 10 nM T15571 CJS56K 145967795 Ki = 8200 nM T15571 CQJ5O8 145971635 Ki > 10000 nM T15571 C79TNE 145972796 Ki > 10000 nM T15571 C6XIN0 145974114 Ki > 10000 nM T15571 CD8ZL6 145974750 Ki > 10 nM T15571 C6PH4F 145975226 Ki > 10000 nM T15571 C71CYU 145975946 Ki > 10000 nM T15571 C2TN8W 145976085 Ki > 10000 nM T15571 C6BFY7 145977338 Ki > 10000 nM T15571 C0Y6QO 145977799 Ki = 6800 nM T15571 C3BI1R 145978113 Ki > 10000 nM T15571 CQU8R0 145978665 Ki > 10000 nM T15571 C6AV9G 145978819 Ki > 10000 nM T15571 C87MSW 145980271 Ki = 4152 nM T15571 CNJH37 145986752 Ki = 4973 nM T15571 CC2G1V 146025727 Ki = 6200 nM T15571 CV9G7Z 153287572 Ki > 10000 nM T15571 CO85KL 153287574 Ki > 10000 nM T15571 CB79ZW 155536080 Ki = 1995.26 nM T15571 C0OK3E 155551348 Ki = 8690 nM T15571 C3N9VU 10251906 Ki > 500 nM T15571 CP9TR0 10324985 Ki = 228.6 nM T15571 CQ1LV7 135508617 Ki = 6725 nM T15571 D00CRA 1574 Ki > 10000 nM T15571 D00GSD 25107716 Ki = 178 nM T15571 D00OBS 44559159 Ki > 10000 nM T15571 D00VRV 10171 Ki < 10 nM T15571 D01HRV 9847194 IC50 > 10000 nM T15571 D01KAX 135453290 Ki > 10000 nM T15571 D01WWC 16573 Ki = 566 nM T15571 D02UWB 1809 Ki = 20 nM T15571 D03DET 10287730 Ki = 3162.28 nM T15571 D03LPH 107838 Ki = 3200 nM T15571 D03TDN 1342 Ki = 40 nM T15571 D03XKU 44455986 Ki = 24 nM T15571 D03ZHB 44455973 Ki = 84.4 nM T15571 D04TPO 16006492 Ki = 5.012 nM T15571 D04UTQ 12683497 Ki = 2800 nM T15571 D05EQG 5265 Ki = 63000 nM T15571 D05GDP 599482 Ki > 10000 nM T15571 D07XTU 1229 Ki > 1000 nM T15571 D08OFG 11177588 Ki > 10000 nM T15571 D08VGJ 9904281 Ki = 43 nM T15571 D09HJL 10331436 Ki > 10000 nM T15571 D09RPR 16737207 Ki > 10000 nM T15571 D09WIL 10028436 Ki = 168 nM T15571 D0C3AR 44456244 Ki = 892 nM T15571 D0C5GF 6918515 Ki = 5160 nM T15571 D0CK9K 6918513 Ki = 4620 nM T15571 D0D1PE 169339 Ki > 10000 nM T15571 D0EA7Z 44455983 Ki = 805 nM T15571 D0F6CD 5202 Ki = 82 nM T15571 D0FF6S 16038374 IC50 > 10000 nM T15571 D0I6II 45263885 Ki = 658 nM T15571 D0J2UA 135433933 Ki = 9621 nM T15571 D0L5MW 181743 Ki = 2224 nM T15571 D0M2ZE 6604756 Ki = 168 nM T15571 D0O3GF 1220 Ki = 1000 nM T15571 D0W2YN 2760172 Ki = 2100 nM T15571 D0X1QW 122334 Ki = 2331 nM T15571 D0X6MT 4106 Ki = 1 nM T15571 D0X9YS 23642275 Ki = 98.5 nM T15571 D0XX2U 16006606 Ki = 6.3 nM T15571 D0Y9TL 13702393 Ki = 99 nM T12241 D08HZC 5852 IC50 = 270000 nM T12241 CVQR28 168091 IC50 = 40000 nM T12241 CE7M6K 269624 IC50 = 6300 nM T12241 CKFD03 439742 IC50 = 14000 nM T12241 C89ZER 2746654 IC50 = 6000 nM T12241 C8O4KD 5281599 IC50 > 400000 nM T12241 C3ZJ8U 5281609 IC50 > 400000 nM T12241 CDBE15 5947235 IC50 > 100000 nM T12241 CGH12F 6436272 IC50 = 1100 nM T12241 CU6W4G 6789060 IC50 = 6000 nM T12241 CX8V7B 6832311 IC50 = 5000 nM T12241 C1JGO8 9557956 IC50 = 40000 nM T12241 CSJ73Q 10347674 IC50 > 400000 nM T12241 CG56QX 13128573 IC50 = 50000 nM T12241 CS56LP 49822436 IC50 > 400000 nM T12241 CX1Y4Q 135517155 IC50 > 100000 nM T12241 CYCK69 145950009 IC50 > 100000 nM T12241 CY0CA3 145950025 IC50 = 2000 nM T12241 CBJE91 145950525 IC50 = 15000 nM T12241 CQ7TR0 145950586 IC50 = 6000 nM T12241 C7HIR2 145950806 IC50 = 15000 nM T12241 C09VKF 145951046 IC50 = 6000 nM T12241 CMD12Q 145951265 IC50 > 100000 nM T12241 CN8O3L 145951907 IC50 = 30000 nM T12241 CE0LR1 145952322 IC50 = 12000 nM T12241 CG5IR7 145952829 IC50 = 3000 nM T12241 CFYH93 145952906 IC50 = 12000 nM T12241 CID02M 145953955 IC50 = 3500 nM T12241 CYA18C 145954124 IC50 = 2100 nM T12241 CID9L8 145954253 IC50 = 40000 nM T12241 C9EV7T 145954518 IC50 > 100000 nM T12241 CU0N7F 145954660 IC50 = 6000 nM T12241 CWT0C2 145954999 IC50 = 10000 nM T12241 C4A7EB 145955194 IC50 = 2000 nM T12241 CC34VO 145955249 IC50 = 2500 nM T12241 CV6JN2 145955896 IC50 = 2700 nM T12241 CU0I6G 145956477 IC50 > 100000 nM T12241 CQN7K8 145956633 IC50 = 1900 nM T12241 CY5OA8 145957277 IC50 = 7000 nM T12241 CVJ8Q7 145957412 IC50 = 2000 nM T12241 C21RHB 145957746 IC50 = 2000 nM T12241 CP74VC 145958243 IC50 = 25000 nM T12241 C2Q9PB 145958460 IC50 = 10000 nM T12241 CD0L9T 145958807 IC50 > 400000 nM T12241 C8AK7F 145959104 IC50 = 6000 nM T12241 C7EX3J 145959358 IC50 = 15000 nM T12241 COW3Z4 145959534 IC50 = 1200 nM T12241 C8PQC2 145959639 IC50 > 100000 nM T12241 CDQ90E 145959869 IC50 = 6000 nM T12241 C1WQP3 145971246 IC50 = 3000 nM T12241 CU61TX 145972452 IC50 = 6000 nM T12241 CK05FS 145974829 IC50 = 5000 nM T12241 D01BTV 286 IC50 = 570 nM T57278 D03ZBT 11626560 IC50 > 1000 nM T57278 D09KTS 24821094 IC50 > 1000 nM T57278 D0E6XR 3062316 IC50 = 137 nM T57278 D03HUX 49792852 IC50 > 10000 nM T57278 D04AHQ 71721540 IC50 = 20 nM T57278 D04SLF 9903 IC50 = 50000 nM T57278 D0E3TC 44259 IC50 = 74.5 nM T57278 D03BNU 59604787 IC50 > 10000 nM T57278 D0T3ME 156422 IC50 = 160 nM T57278 CT52XN 92997 IC50 = 39810.72 nM T57278 CXQ5O3 115245 IC50 = 48977.88 nM T57278 CY13FW 644243 IC50 = 760 nM T57278 C4RUV5 5329453 IC50 = 250 nM T57278 C5GE7T 9917045 IC50 = 5200 nM T57278 CSGD16 10246246 IC50 > 7000 nM T57278 CBOP58 11293798 Ki > 10000 nM T57278 C26BZX 11362471 Ki > 10000 nM T57278 CWXB93 11397177 Ki > 10000 nM T57278 C35EIU 11698847 IC50 > 316227.77 nM T57278 C45EWD 11723489 IC50 > 7000 nM T57278 CP7AH3 11755812 IC50 = 35 nM T57278 CFPW41 16007116 Ki > 8000 nM T57278 C6JV7W 23400934 IC50 > 7000 nM T57278 CD5S7O 23401001 IC50 > 7000 nM T57278 CA3I4T 24753787 IC50 > 50000 nM T57278 CY8L7E 24896769 IC50 > 10000 nM T57278 C6W5LZ 25081574 IC50 = 4100 nM T57278 CA98KR 44432441 IC50 > 10000 nM T57278 C3VRO9 44557921 IC50 > 10000 nM T57278 C3HW7L 44570553 IC50 > 30000 nM T57278 C17PVE 44570554 IC50 > 30000 nM T57278 CLOY92 44570599 IC50 = 3000 nM T57278 CK06LT 44570600 IC50 > 30000 nM T57278 CY3HW5 46224684 IC50 > 10000 nM T57278 CYT37A 46232443 IC50 > 50000 nM T57278 C48ZVW 46232555 IC50 = 4400 nM T57278 CS9B1U 46232556 IC50 = 5200 nM T57278 CLS29B 46872626 IC50 > 10000 nM T57278 C2O8RZ 46886323 IC50 = 370 nM T57278 C0WYM1 46898022 IC50 = 10000 nM T57278 CF91RS 49843531 IC50 > 10000 nM T57278 CQ3KU9 50899556 IC50 = 260 nM T57278 C2Y6QS 50938552 IC50 > 10000 nM T57278 C61DVY 50990961 IC50 = 18 nM T57278 CV3UP9 50992247 IC50 = 11 nM T57278 CS9G6E 50997096 IC50 > 10000 nM T57278 C9NYP4 51036677 IC50 > 10000 nM T57278 C4WRY3 51037112 IC50 > 10000 nM T57278 CRI28Z 51037948 IC50 > 10000 nM T57278 C3LB5V 52941849 IC50 > 10000 nM T57278 CW2X5E 52944268 IC50 = 740 nM T57278 C9PX2J 52945752 IC50 = 300 nM T57278 CL4ED3 52945753 IC50 = 840 nM T57278 CIR3Q0 52947964 IC50 = 5600 nM T57278 C09SDH 53257410 IC50 > 10000 nM T57278 CBK9Q6 53357848 IC50 > 10000 nM T57278 C8NA4L 53384644 IC50 = 16000 nM T57278 CPHX64 57325478 IC50 > 50000 nM T57278 CQ9BW4 57325479 IC50 > 50000 nM T57278 CVK0G4 58056356 IC50 > 50000 nM T57278 CT3EW2 59292007 IC50 > 1000 nM T57278 C9ZCT2 62705065 IC50 > 1000 nM T57278 C10AMI 66553589 IC50 = 6180 nM T57278 CV63UL 67240318 IC50 > 10000 nM T57278 C23UCM 70946730 IC50 = 300 nM T57278 CKT60L 71455860 Ki > 2800 nM T57278 CCN01X 71547862 IC50 > 10000 nM T57278 CVIA91 71553085 IC50 = 30000 nM T57278 C1TR3O 71553152 IC50 = 30000 nM T57278 CF8Z9P 71604568 IC50 = 19952.62 nM T57278 CP5T7A 71604569 IC50 = 30902.95 nM T57278 CG6SI4 71604570 IC50 = 23988.33 nM T57278 CD1PS3 71604720 IC50 = 17378.01 nM T57278 CN3FH0 71604721 IC50 = 101000 nM T57278 C13PNG 71604722 IC50 = 60255.96 nM T57278 CB8KL7 71604723 IC50 > 316227.77 nM T57278 C01POC 71604724 IC50 > 316227.77 nM T57278 C24DHJ 71604873 IC50 > 316227.77 nM T57278 CR4D9H 71604874 IC50 = 26000 nM T57278 CUGT42 71604875 IC50 = 27542.29 nM T57278 CJDA65 71604876 IC50 = 6606.93 nM T57278 CEK72C 71604877 IC50 = 7585.78 nM T57278 CW6NK4 71605036 IC50 = 50118.72 nM T57278 CX3E8O 71605037 IC50 = 100000 nM T57278 C60QZJ 71605038 IC50 = 20417.38 nM T57278 CZHF09 71716449 IC50 >= 100000 nM T57278 C7H6GC 71717050 IC50 = 6300 nM T57278 CV2HP0 71717673 IC50 >= 100000 nM T57278 CN56HF 71718279 IC50 >= 100000 nM T57278 C9E3XT 71718280 IC50 = 14000 nM T57278 CQL9G2 71718885 IC50 = 24000 nM T57278 CSEQ21 71719490 IC50 > 100000 nM T57278 CQ36JS 71719491 IC50 = 13000 nM T57278 CN6CA9 71720086 IC50 = 94000 nM T57278 C46ONG 71720087 IC50 = 29000 nM T57278 C4TRW2 71720468 IC50 > 316227.77 nM T57278 CR97JV 71720738 IC50 = 71000 nM T57278 CBX0N9 71720739 IC50 = 15000 nM T57278 C60TUV 72737208 IC50 > 10000 nM T57278 CJ3WA6 72737404 IC50 > 10000 nM T57278 CVNW01 73386831 IC50 > 1000 nM T57278 CCJ43A 86302281 IC50 > 10000 nM T57278 CB5NJ4 86302541 IC50 > 10000 nM T57278 CPG3A5 86302574 IC50 > 30000 nM T57278 CY0UC4 90645194 IC50 > 10000 nM T57278 CX29IY 90655145 IC50 > 10000 nM T57278 CAPB10 91666638 IC50 = 160 nM T57278 CY7BI2 118706214 IC50 > 10000 nM T57278 CKM13G 118710440 IC50 = 1190 nM T57278 CVJ7A8 118710441 IC50 = 1470 nM T57278 CSRQ30 118710442 IC50 = 2500 nM T57278 C4E0UV 118710443 IC50 = 750 nM T57278 CA1ZY6 118710444 IC50 = 2310 nM T57278 COJ3U8 118710445 IC50 = 680 nM T57278 CDTF80 118710446 IC50 = 580 nM T57278 C0D1PA 118710447 IC50 = 730 nM T57278 C6BH8K 118710448 IC50 = 720 nM T57278 CDLQ85 118710449 IC50 = 620 nM T57278 C9M5ZO 118710451 IC50 = 960 nM T57278 C28ABH 118710452 IC50 = 3210 nM T57278 CO8C6F 118710453 IC50 = 200 nM T57278 CR4S3Y 118710454 IC50 = 170 nM T57278 C7E0VG 118710455 IC50 = 450 nM T57278 C78JUP 118710456 IC50 = 230 nM T57278 CC70YB 118710457 IC50 = 320 nM T57278 CQCX41 118737057 IC50 = 16 nM T57278 C8KXV1 127025843 IC50 > 1000 nM T57278 C40DLR 127035199 IC50 = 4265.8 nM T57278 CN3F9G 127035350 IC50 = 89125.09 nM T57278 C0OM1N 127035351 IC50 = 6309.57 nM T57278 CEV2H1 127035714 IC50 = 8912.51 nM T57278 CO7SQ1 127035899 IC50 > 100000 nM T57278 C9WGB8 127035904 Ki = 1400 nM T57278 CCLF46 127035905 IC50 > 100000 nM T57278 C06KQV 127035906 IC50 = 22387.21 nM T57278 CVU98P 127035907 Ki = 2400 nM T57278 CDI68C 127035908 IC50 = 47863.01 nM T57278 C6TJF3 127036098 IC50 > 100000 nM T57278 CD98XV 127036099 IC50 = 50118.72 nM T57278 CFSP72 127036100 IC50 = 5011.87 nM T57278 CKIA98 127036101 IC50 = 4073.8 nM T57278 CKX40V 127037812 IC50 > 10000 nM T57278 C70RUP 127038480 IC50 > 10000 nM T57278 C3WCN8 127041777 IC50 > 10000 nM T57278 CHK16Q 127045929 IC50 > 1000 nM T57278 CY3J0C 127047591 IC50 > 1000 nM T57278 CERS64 132937256 IC50 > 30000 nM T57278 CN35SO 134146628 IC50 > 1000 nM T57278 CYL5V1 134694986 IC50 > 30000 nM T57278 CDT7E4 136211077 IC50 > 100 nM T57278 CXC69T 137321158 IC50 = 341 nM T57278 C25ERN 137631967 IC50 > 100 nM T57278 C06JRX 137637094 IC50 > 10 nM T57278 CTD9I4 137637448 Ki > 15000 nM T57278 C1DK0P 137651391 IC50 > 100 nM T57278 CSB0L1 137654726 IC50 = 5000 nM T57278 CV5H3Z 137657932 IC50 > 10 nM T57278 CSRI06 138547901 IC50 > 1000 nM T57278 CUXO19 138617501 IC50 > 1000 nM T57278 CO9P7G 145351804 IC50 > 1000 nM T57278 C29XUO 145945978 IC50 > 1000 nM T57278 C4OD9Q 145967187 IC50 > 1000 nM T57278 CUJS82 145969463 IC50 = 4900 nM T57278 COD32L 145970693 IC50 = 4100 nM T57278 C2MD1Q 155513187 IC50 > 10000 nM T57278 CS69CA 155532132 IC50 = 13.5 nM T57278 D00ERW 44444843 Ki > 8000 nM T57278 D02BXJ 46864270 IC50 = 0.6 nM T57278 D05FXD 44478401 IC50 = 2.3 nM T57278 D0C2GE 67161540 IC50 = 1700 nM T57278 D0O6OH 71553154 IC50 = 2430 nM T57278 D0X8BU 71718651 IC50 = 2041.74 nM T57278 D0Y0BK 11524144 IC50 = 11 nM T01385 D09GOS 2812 IC50 = 1400 nM T01385 D08OOJ 73051434 IC50 = 11 nM T01385 D0F6NT 1162727 IC50 > 30000 nM T01385 C05ZPG 397069 IC50 > 100000 nM T01385 C86FWD 470278 IC50 > 100000 nM T01385 C5EY0V 672872 IC50 = 80 nM T01385 CHXJ51 697280 IC50 = 190 nM T01385 CR98CN 704363 IC50 = 230 nM T01385 C1IV9D 704494 IC50 = 290 nM T01385 C4X1BC 704553 IC50 = 300 nM T01385 CYF9E1 720920 IC50 > 30000 nM T01385 C1QRW7 768027 IC50 = 2000 nM T01385 C30HYZ 788482 IC50 = 1290 nM T01385 C34XJV 793670 EC50 = 90 nM T01385 C9M6JL 863286 IC50 > 30000 nM T01385 C1KQL0 864171 IC50 > 30000 nM T01385 C8KUR0 865869 IC50 = 9920 nM T01385 C3FX5T 865870 IC50 = 2690 nM T01385 C7MLU1 877530 IC50 > 10000 nM T01385 CHX2D5 877815 IC50 = 430 nM T01385 CA0J3M 906598 IC50 > 100000 nM T01385 CD7O0J 935549 IC50 = 4800 nM T01385 CPL20I 973124 IC50 = 1300 nM T01385 CZ32JI 2249447 IC50 = 8300 nM T01385 C5Q0HK 2975404 IC50 > 37000 nM T01385 CX3JD7 3556408 IC50 = 760 nM T01385 CEM5C8 25100438 IC50 = 360 nM T01385 C07VAB 25100440 IC50 = 670 nM T01385 CDXT96 30869108 IC50 = 990 nM T01385 C1M5SP 45019715 IC50 > 30000 nM T01385 CH2V5M 46865782 IC50 = 120 nM T01385 C9P6UC 46880290 IC50 > 20000 nM T01385 CGIA46 46880328 IC50 = 2700 nM T01385 C3VKZ8 46880369 IC50 = 180 nM T01385 CZHM28 46880414 IC50 = 91 nM T01385 CAU6O0 46880464 IC50 = 120 nM T01385 CXDK90 46880466 IC50 = 140 nM T01385 CVEC92 46880467 IC50 = 170 nM T01385 CHW21A 46880468 IC50 = 190 nM T01385 C2YWI1 46880469 IC50 = 330 nM T01385 CBQ49H 46880502 IC50 = 130 nM T01385 CA6IV3 46880503 IC50 = 230 nM T01385 CZPV27 49830258 IC50 = 110 nM T01385 C7EY1H 49852176 IC50 > 5000 nM T01385 C4VIP1 50918580 IC50 = 425 nM T01385 C9OJG1 52374396 IC50 > 30000 nM T01385 CCR7O0 54670937 IC50 > 5000 nM T01385 CM59RJ 56928016 IC50 > 5000 nM T01385 CH65ZE 57328756 IC50 = 22000 nM T01385 C1XBG6 58523937 IC50 > 5000 nM T01385 C07XGU 71520305 IC50 = 88 nM T01385 CWZ27A 71520306 IC50 = 90 nM T01385 C5WQ8Z 71520307 IC50 = 100 nM T01385 CN4O3X 71520308 IC50 = 134 nM T01385 C5OK4Z 71520309 IC50 = 150 nM T01385 C6SRU5 71520310 IC50 = 184 nM T01385 C82ATI 71520425 IC50 = 225 nM T01385 C2B9KN 71520426 IC50 = 257 nM T01385 CQ1JY3 71520427 IC50 = 443 nM T01385 CZ80NI 71520429 IC50 = 43 nM T01385 CB4JG8 71520430 IC50 = 48 nM T01385 C13YPQ 71520540 IC50 = 71 nM T01385 CO2QT1 71520541 IC50 = 41 nM T01385 CI8B7L 71520542 IC50 = 42 nM T01385 CKQL06 71520543 IC50 = 63 nM T01385 CY6PL1 71520544 IC50 = 65 nM T01385 CE4Q0T 71520634 IC50 = 112 nM T01385 CMQ68E 71520635 IC50 = 162 nM T01385 CP9UY2 71520818 IC50 > 30000 nM T01385 C7HFN3 71520819 IC50 = 960 nM T01385 CS90CX 71520820 IC50 = 720 nM T01385 CPB6S5 71520821 IC50 = 960 nM T01385 C4K1AN 71520822 IC50 = 1150 nM T01385 C45XQJ 71520919 IC50 > 30000 nM T01385 C7V2LX 71520920 IC50 = 3790 nM T01385 C0F5TW 71520926 IC50 = 172 nM T01385 CBO1H8 71520927 IC50 = 262 nM T01385 C1BSM0 71520928 IC50 = 523 nM T01385 CR42SU 71520929 IC50 = 683 nM T01385 C6I0OW 71520930 IC50 = 976 nM T01385 COYE37 71520931 IC50 = 1236 nM T01385 CEHQ96 71521025 IC50 > 30000 nM T01385 C4KCX9 71521026 IC50 > 30000 nM T01385 CEYG08 71521027 IC50 > 30000 nM T01385 CU10JB 71521028 IC50 = 2250 nM T01385 C1YF8L 71521029 IC50 = 1960 nM T01385 CIG40P 71521030 IC50 = 19430 nM T01385 C5IH4G 71521031 IC50 > 30000 nM T01385 CT4O1M 71521032 IC50 = 2031 nM T01385 CH97TQ 71521033 IC50 = 536 nM T01385 CXG73H 71521034 IC50 = 379 nM T01385 CZMO73 71521035 IC50 = 1394 nM T01385 C8F3AT 71521036 IC50 = 451 nM T01385 C9YN6X 71521037 IC50 = 908 nM T01385 C27VGT 71521131 IC50 = 1880 nM T01385 CT7IQ3 71521132 IC50 = 2060 nM T01385 C1N0IP 71521133 IC50 = 2320 nM T01385 C9EJZ4 71521134 IC50 = 16220 nM T01385 C8AR7M 71521135 IC50 > 30000 nM T01385 CG1XD3 71521136 IC50 = 19600 nM T01385 C3H7PS 71521137 IC50 > 30000 nM T01385 C6X8OQ 71521138 IC50 = 71 nM T01385 C10NRW 71521139 IC50 = 58 nM T01385 C7H1ME 71521140 IC50 = 25 nM T01385 CK6M1Y 71521141 IC50 = 54 nM T01385 CI0DC4 71521236 IC50 = 2690 nM T01385 C4R3FX 71521237 IC50 = 740 nM T01385 C3AJ2W 71521238 IC50 = 960 nM T01385 CS5E0K 71521239 IC50 = 2780 nM T01385 CVSF75 71521240 IC50 = 53 nM T01385 CIY79B 71521241 IC50 = 67 nM T01385 C0K3FZ 71521347 IC50 = 2810 nM T01385 CDR29I 71521348 IC50 > 30000 nM T01385 C4P1OI 71521349 IC50 > 30000 nM T01385 C2FU7P 71521350 IC50 > 30000 nM T01385 CSP46C 71521351 IC50 > 30000 nM T01385 C2F8TA 71521352 IC50 = 470 nM T01385 CVYJ16 71521353 IC50 > 30000 nM T01385 CR1LF6 71521458 IC50 = 1290 nM T01385 CDF30Z 71521459 IC50 = 2400 nM T01385 CU9D2H 71521460 IC50 = 7730 nM T01385 C2H9UV 71521461 IC50 = 11780 nM T01385 CG8Z3S 71521462 IC50 = 26720 nM T01385 C7CF8N 71521463 IC50 > 30000 nM T01385 CM7UB5 71521536 IC50 = 440 nM T01385 C46IZM 71521537 IC50 = 18640 nM T01385 C21MUO 71521538 IC50 = 2860 nM T01385 CS43JP 71521539 IC50 = 1940 nM T01385 CMUZ53 71521540 IC50 = 8720 nM T01385 CE1FJ6 71521541 IC50 = 11170 nM T01385 CQ0BK1 71521542 IC50 > 30000 nM T01385 CBJM79 71521620 IC50 > 30000 nM T01385 CY8RF0 71521621 IC50 = 1970 nM T01385 CV4Q5F 71521622 IC50 = 4300 nM T01385 CJ9B0Z 71521623 IC50 > 30000 nM T01385 CS84PN 71521624 IC50 = 2850 nM T01385 CX6Z8C 71521625 IC50 = 3450 nM T01385 CTK92X 71521626 IC50 = 5560 nM T01385 CPF75N 71521709 IC50 = 1277 nM T01385 CPJ3Q1 71521710 IC50 = 279 nM T01385 CP82UW 71521711 IC50 = 283 nM T01385 CXRZ18 71521712 IC50 = 379 nM T01385 C3W9KG 71521713 IC50 = 524 nM T01385 CN96LY 71521714 IC50 = 3129 nM T01385 CLD68Y 71521715 IC50 = 375 nM T01385 C5WV4I 71521791 IC50 = 140 nM T01385 C93NYA 71521792 IC50 = 168 nM T01385 CSH67K 71521793 IC50 = 604 nM T01385 C7KRB8 71521794 IC50 = 220 nM T01385 C7IU9X 71521795 IC50 = 609 nM T01385 C23LYC 71521796 IC50 = 587 nM T01385 CRO46G 71521797 IC50 = 71 nM T01385 CH1KQ4 71604308 IC50 = 760 nM T01385 CEA94U 71604309 IC50 = 1100 nM T01385 CC1V2S 71607189 IC50 = 370 nM T01385 C4TG6V 72721010 IC50 = 43 nM T01385 C2R9LK 73051132 IC50 = 445 nM T01385 C1M0KD 73051133 IC50 = 153 nM T01385 CG71JS 73051280 IC50 = 47 nM T01385 C1NQ8H 73051924 IC50 = 98 nM T01385 C7IMZ0 73052240 IC50 = 3134 nM T01385 C4HM1G 73052241 IC50 = 76 nM T01385 C4FWO9 73052243 IC50 > 5000 nM T01385 C3VLG0 73052401 IC50 = 95 nM T01385 C79HDC 73052716 IC50 = 1790 nM T01385 CEG8R1 73052718 IC50 = 192 nM T01385 CTR3G9 73052878 IC50 = 6 nM T01385 C0VA6M 73053029 IC50 = 304 nM T01385 C95DXT 82192375 IC50 > 37000 nM T01385 C46GEV 89927846 IC50 = 370 nM T01385 C9W7GE 89927907 IC50 = 3000 nM T01385 CBC03Z 89927958 IC50 = 152 nM T01385 CRX36D 89927984 IC50 = 145 nM T01385 CC36BE 89928011 IC50 = 233 nM T01385 C0XAP3 89928021 IC50 = 248 nM T01385 CMI21Z 89928023 IC50 = 68 nM T01385 CYEC61 89928082 IC50 > 5000 nM T01385 C0J7BI 89928094 IC50 = 149 nM T01385 CE81KH 89928101 IC50 = 144 nM T01385 CTGD01 89928106 IC50 = 2075 nM T01385 C6WS8V 89928107 IC50 = 632 nM T01385 CK7GM3 89928109 IC50 = 795 nM T01385 CDP70Y 89928159 IC50 = 227 nM T01385 C29ART 89928200 IC50 = 342 nM T01385 C7PH3D 89928222 IC50 = 180 nM T01385 C8AZT1 89928224 IC50 = 1068 nM T01385 CBK1W6 89941289 IC50 > 5000 nM T01385 CB8IQ2 90031714 IC50 > 5000 nM T01385 CN91SG 90032051 IC50 = 651 nM T01385 CJZS64 90032070 IC50 = 367 nM T01385 CY5TU6 90032147 IC50 = 3912 nM T01385 C9ISK1 90032171 IC50 = 215 nM T01385 CNE9B5 90032547 IC50 = 8908 nM T01385 C2XC7V 90032634 IC50 = 648 nM T01385 CBTL19 101907906 IC50 = 26300 nM T01385 CA6E9Y 101910775 IC50 = 61 nM T01385 CMY30U 101910777 IC50 = 74 nM T01385 C1A8JZ 114286471 IC50 = 70 nM T01385 CMA84J 117094775 IC50 = 907 nM T01385 CF2RD3 118322226 IC50 = 4832 nM T01385 CQBG03 118724369 IC50 = 21600 nM T01385 CD71XN 118724370 IC50 = 20500 nM T01385 CEC71H 118724371 IC50 > 37000 nM T01385 CF53BA 118724372 IC50 > 37000 nM T01385 C5RFT0 118724373 IC50 = 15400 nM T01385 CH8PF1 118724374 IC50 > 37000 nM T01385 C9C4WZ 118724375 IC50 = 2600 nM T01385 C9SLR5 118724376 IC50 = 8700 nM T01385 CYX0K4 118724377 IC50 > 37000 nM T01385 COE61I 118724378 IC50 > 37000 nM T01385 CS8YZ3 118724379 IC50 = 11400 nM T01385 C9RJV7 118724380 IC50 = 4800 nM T01385 CA3LT6 118724381 IC50 > 37000 nM T01385 CE43MW 118724382 IC50 = 2700 nM T01385 CH42TP 118724383 IC50 = 2600 nM T01385 CQFZ65 118724384 IC50 = 8400 nM T01385 CYV7T4 118724385 IC50 > 37000 nM T01385 C2SV1M 118724386 IC50 = 300 nM T01385 CYLT37 118724387 IC50 = 673 nM T01385 CA93NZ 118724388 IC50 = 141 nM T01385 CV56WG 118724389 IC50 = 700 nM T01385 C7LCP1 118724390 IC50 = 3041 nM T01385 C7XV4F 118724391 IC50 = 578 nM T01385 CD2WN1 118724392 IC50 = 552 nM T01385 C9FVI6 118724393 IC50 = 483 nM T01385 C0O3AC 118724394 IC50 = 543 nM T01385 C82IQE 118724395 IC50 = 116 nM T01385 CO9R3I 118724396 IC50 = 201 nM T01385 CRF7Z9 118724397 IC50 = 879 nM T01385 C5N1SJ 118724762 IC50 = 577 nM T01385 CG01LE 118724763 IC50 = 742 nM T01385 CA39KG 118724764 IC50 = 221 nM T01385 C1JTS3 118724765 IC50 = 921 nM T01385 CK7Y9N 118724766 IC50 = 1091 nM T01385 CCM3X6 118724767 IC50 = 2189 nM T01385 CAMZ23 118724768 IC50 = 112 nM T01385 CHZ6K1 118724769 IC50 = 60 nM T01385 C5T1RV 118724770 IC50 = 150 nM T01385 CZKE26 118724771 IC50 = 570 nM T01385 CGP36N 118724772 IC50 = 1201 nM T01385 C3YPM4 118724773 IC50 = 1667 nM T01385 C3K2BJ 118724774 IC50 = 2188 nM T01385 CYJR42 118724775 IC50 = 27 nM T01385 CF5X3Y 118724776 IC50 = 36 nM T01385 C7UZ5H 118724777 IC50 = 4313 nM T01385 CO6GN4 118724778 IC50 > 10000 nM T01385 CPK72W 118724779 IC50 = 127 nM T01385 CGO35H 118724780 IC50 = 448 nM T01385 C96YAG 118724781 IC50 = 133 nM T01385 CJ1UK5 118724782 IC50 = 264 nM T01385 C8DX9G 118724783 IC50 = 986 nM T01385 CN49SF 118724784 IC50 = 9288 nM T01385 CA78KC 118724785 IC50 = 1691 nM T01385 CL25HP 118724786 IC50 = 6939 nM T01385 CEG6T2 118724787 IC50 = 7108 nM T01385 C32LRP 118724788 IC50 = 8860 nM T01385 C43QNY 118724789 IC50 = 1679 nM T01385 CCDH40 118724790 IC50 = 474 nM T01385 CA6F9K 118724791 IC50 = 2762 nM T01385 CV5P0J 118724792 IC50 = 5645 nM T01385 CWQ61D 118724793 IC50 = 4608 nM T01385 CKM04D 118724794 IC50 = 7610 nM T01385 CTRV82 118724795 IC50 = 2181 nM T01385 C69HKQ 118724796 IC50 = 2433 nM T01385 CO9W1I 118724797 IC50 = 3473 nM T01385 CLVO02 118724798 IC50 = 5036 nM T01385 CACB18 118724799 IC50 = 5165 nM T01385 C8LJ1X 118724800 IC50 > 10000 nM T01385 CCK45Q 118724801 IC50 = 46 nM T01385 C6B1FX 118724802 IC50 = 87 nM T01385 CY50JH 118724803 IC50 = 106 nM T01385 CS8O9F 118724804 IC50 = 135 nM T01385 C4SU7T 118724805 IC50 = 149 nM T01385 CW9E3Z 118724806 IC50 = 183 nM T01385 CY6C3R 118724807 IC50 = 237 nM T01385 C6H9CJ 118724808 IC50 = 59 nM T01385 CX7FM5 118724809 IC50 = 89 nM T01385 CE54NW 118724810 IC50 = 102 nM T01385 CXJ43Z 118724811 IC50 = 106 nM T01385 CVKT57 118724812 IC50 = 222 nM T01385 CZV40N 118724813 IC50 = 246 nM T01385 C4YH3Q 118724814 IC50 = 299 nM T01385 C0F8VX 118724815 IC50 = 82 nM T01385 C6QRS2 118724816 IC50 = 109 nM T01385 C3NK9E 118724817 IC50 = 452 nM T01385 C2DSR3 118724818 IC50 = 491 nM T01385 C4UJ7V 127031857 IC50 = 50 nM T01385 CT0F5Y 127032127 IC50 = 710 nM T01385 C3VG0W 127032128 IC50 = 3800 nM T01385 CGU32Y 127032429 IC50 = 4700 nM T01385 CVXR24 127032715 IC50 = 21500 nM T01385 CRN4B7 127032716 IC50 = 240 nM T01385 CKGU65 127039986 IC50 > 5000 nM T01385 CRB4C1 127039987 IC50 > 5000 nM T01385 C2GX8Z 127039988 IC50 > 5000 nM T01385 CV81YZ 127039989 IC50 = 3860 nM T01385 C6OQ4W 127039990 IC50 > 5000 nM T01385 CB2AR3 127040617 IC50 > 5000 nM T01385 CJ4FQ3 127040618 IC50 > 5000 nM T01385 CX0P2U 127040619 IC50 > 5000 nM T01385 C82QOL 127040620 IC50 > 5000 nM T01385 CWC4M7 127040621 IC50 > 5000 nM T01385 CWA09O 127040622 IC50 > 5000 nM T01385 CQ6KV5 127041309 IC50 = 15 nM T01385 CI0X6E 127041536 IC50 > 5000 nM T01385 CQ2VO1 127041608 IC50 = 71 nM T01385 CGN9I7 127041609 IC50 = 23 nM T01385 C3TUR2 127041878 IC50 > 5000 nM T01385 CR8PG7 127041879 IC50 > 5000 nM T01385 CV92NA 129073433 IC50 = 180 nM T01385 C3IN1Q 132561319 IC50 = 7900 nM T01385 C1LN3T 132570328 IC50 = 160 nM T01385 C3H6DA 132570329 IC50 = 44 nM T01385 C6H9BZ 132570331 IC50 = 31400 nM T01385 CEZ9B2 139035043 IC50 = 7200 nM T01385 CEX63L 139298248 IC50 = 7 nM T01385 C10RBQ 140939034 IC50 = 90 nM T01385 CKW53D 140939044 IC50 = 100 nM T01385 C8CQT0 140939054 IC50 = 280 nM T01385 C7TX2S 140939070 IC50 = 190 nM T01385 COWD30 140939079 IC50 = 20 nM T01385 C4V7CI 140939088 IC50 = 2610 nM T01385 C2C9PG 140939100 IC50 = 1130 nM T01385 C6PN5R 140939111 IC50 = 200 nM T01385 C0ZH4R 140939116 IC50 = 800 nM T01385 CTJ0U5 140939119 IC50 = 19000 nM T01385 CGLY18 140939126 IC50 = 210 nM T01385 CUC3P9 140939138 IC50 = 1060 nM T01385 CW8U7Q 140939163 IC50 = 4760 nM T01385 CZ0XI5 140939170 IC50 = 1050 nM T01385 CX7F5D 140939178 IC50 = 50 nM T01385 CP7Q2G 140939185 IC50 = 330 nM T01385 C4JAX8 145988686 IC50 = 380 nM T01385 C7LGD3 154730745 Ki = 33.2 nM T01385 CDN0B5 155068296 IC50 = 82.8 nM T01385 C9YQ7I 155510447 Ki = 20.8 nM T01385 C43MSR 155510502 Ki = 28.1 nM T01385 CQV4H6 155513260 Ki = 32.8 nM T01385 C3K1VZ 155513650 IC50 = 119.7 nM T01385 CSB62H 155515179 Ki = 24.5 nM T01385 CN98ID 155517954 IC50 = 922.1 nM T01385 CD0A2C 155518618 Ki = 40.8 nM T01385 CM48LB 155522046 IC50 = 34.6 nM T01385 CR34KJ 155522981 Ki = 26.6 nM T01385 C0CA1Z 155524986 Ki = 43 nM T01385 CWTP12 155527743 Ki = 32.3 nM T01385 CZA90T 155528495 IC50 = 36.4 nM T01385 C0HU1L 155528572 IC50 = 134.9 nM T01385 CG8Z9A 155530177 Ki = 30.6 nM T01385 C69LKC 155530248 Ki = 37.3 nM T01385 CBQ3N1 155533126 IC50 = 192.6 nM T01385 C80XHD 155536273 IC50 = 387.1 nM T01385 CWZS75 155538655 IC50 = 8 nM T01385 C9KO2J 155545885 IC50 = 129.4 nM T01385 C3VHG0 155547513 Ki = 42.4 nM T01385 CYFP96 155547774 Ki = 24.1 nM T01385 CLV2Z5 155555002 Ki = 26.9 nM T01385 C42ONM 155556308 IC50 = 448.7 nM T01385 C1QNZ5 155557365 Ki = 18.6 nM T01385 CGYS98 155557471 Ki = 37.9 nM T01385 CL28DA 155561627 IC50 = 160.9 nM T01385 C2M7QB 155561797 IC50 = 447.2 nM T01385 C3FXR6 155563226 IC50 = 100.9 nM T01385 C4LU8S 155563972 IC50 = 5104.5 nM T01385 CPU5R9 155564364 IC50 = 308.1 nM T01385 CIYS74 155565460 Ki = 31.4 nM T01385 D00YNY 753704 EC50 < 1200 nM T01385 D0D8SU 71521142 IC50 = 24 nM T57818 D0RA5Q 72172 IC50 = 160000 nM T57818 CK8VJ3 5311145 Ki > 1000000 nM T57818 CP4VT2 13633258 Ki = 51 nM T57818 CT3L5Q 14542146 Ki = 130000 nM T57818 CP4OT8 14542149 Ki = 170 nM T57818 CE1P6J 15719279 Ki = 1500 nM T57818 CD28WR 15719282 Ki = 3200 nM T57818 CYR87Z 15719283 Ki = 6500 nM T57818 CMWK71 44276411 Ki = 11 nM T57818 CS75VD 44360285 Ki > 300000 nM T57818 CVS46P 54394267 IC50 = 3500 nM T57818 D02BLC 20384324 Ki = 0.9 nM T57818 D0A7GO 44309732 Ki = 39000 nM T84117 D01AZG 5073 Ki > 1000 nM T84117 D0G8NN 119570 Ki > 10000 nM T84117 D0H3HM 60795 Ki > 1000 nM T84117 D0H7KF 5002 Ki > 1000 nM T84117 D0V4QS 135398745 Ki > 1000 nM T84117 D0Z1RV 135398737 Ki = 1000 nM T84117 D0Z6UC 5358 IC50 = 5500 nM T84117 D0N1HW 5311200 Ki > 10000 nM T84117 D0X2XF 177336 Ki < 10000 nM T84117 D02ZSO 6426760 IC50 > 10000 nM T84117 D03YPJ 5163 Ki < 5011.87 nM T84117 D0M7LV 5761 Ki = 93 nM T84117 D0Q2JS 10436045 Ki = 6.31 nM T84117 D0YP7L 6604889 Ki < 6309.57 nM T84117 C5H9CN 9287 Ki = 1905.46 nM T84117 C6WDL7 49756 Ki = 1800 nM T84117 CTB26S 52899 Ki > 10000 nM T84117 CKP25M 121881 Ki < 10000 nM T84117 C2VLP8 752521 Ki > 10000 nM T84117 CS8KE2 3649661 Ki > 10000 nM T84117 C0QCK1 6918455 Ki < 10000 nM T84117 CW0ZE5 6918542 Ki = 4220 nM T84117 CD0Z4I 6918648 Ki = 2511.89 nM T84117 CYMP40 9851789 IC50 = 99 nM T84117 CJW1P5 9888494 Ki < 10000 nM T84117 C3J8GU 9892409 Ki < 1000 nM T84117 CUN81Q 9905249 Ki > 10000 nM T84117 CYWQ50 9906447 Ki > 10000 nM T84117 C78MDV 9913554 Ki = 1584.89 nM T84117 CWO45F 9935387 Ki = 1000 nM T84117 CYH3R7 9947817 Ki = 770 nM T84117 C3S7XA 10009042 IC50 = 392 nM T84117 CV7R9F 10020040 Ki > 10000 nM T84117 CK18LT 10020895 Ki = 660 nM T84117 C4Q2SH 10249573 Ki < 10000 nM T84117 CMRA02 10257042 Ki < 6309.57 nM T84117 CH31DX 10267394 Ki > 10000 nM T84117 CU89JD 10314060 Ki > 10000 nM T84117 C9IAV3 10346043 Ki > 10000 nM T84117 C4TPN1 10413595 Ki > 10000 nM T84117 CD7U5I 10433930 Ki > 10000 nM T84117 COV85C 10472143 Ki = 280 nM T84117 CHE80N 10573876 Ki < 2511.89 nM T84117 CO23YX 10597140 Ki < 10000 nM T84117 C8MHZ9 10835110 Ki = 2511.89 nM T84117 CNB39C 10947658 Ki = 200 nM T84117 CVE8T3 11121216 Ki = 140 nM T84117 C9ZT5F 11536299 Ki > 10000 nM T84117 CGX8F6 11596869 Ki > 5370000 nM T84117 CXLW54 11948707 Ki > 10000 nM T84117 C8JQL7 11957735 IC50 > 10000 nM T84117 CZ2IS9 16660294 Ki > 10000 nM T84117 C7T8JC 19958494 Ki > 10000 nM T84117 C6LI5E 19958507 Ki > 10000 nM T84117 C3T5HF 21509921 Ki = 4045 nM T84117 CBN84K 22065997 Ki > 10000 nM T84117 CDC91N 24839550 Ki = 380.19 nM T84117 C3HK0J 24865725 Ki = 2511.89 nM T84117 C0O6FX 24865727 Ki > 10000 nM T84117 CI53SE 24893978 Ki > 10000 nM T84117 CA58DL 41305446 Ki > 10000 nM T84117 CC2OD4 44278111 Ki > 10000 nM T84117 CRMA84 44278114 Ki > 10000 nM T84117 CF0Y4M 44278115 Ki > 10000 nM T84117 CPWJ26 44343212 Ki < 10000 nM T84117 CUXH48 44352308 Ki > 4830 nM T84117 C4B0OI 44397588 Ki < 10000 nM T84117 C5FP0R 44397589 Ki < 10000 nM T84117 CE3G8U 44397670 Ki < 10000 nM T84117 CZL97F 44455426 Ki > 10000 nM T84117 C12XGE 44456400 Ki > 10000 nM T84117 C5ZML8 44457907 IC50 > 1000 nM T84117 CM3IR1 44457909 IC50 > 1000 nM T84117 CAS01K 44458044 IC50 > 1000 nM T84117 CGD04W 44458045 IC50 > 1000 nM T84117 C94DNM 44458229 IC50 > 1000 nM T84117 CM9YD2 44458486 IC50 > 1000 nM T84117 CRCH48 44582675 Ki > 10000 nM T84117 CEJ4R8 44582676 Ki > 10000 nM T84117 CZGP86 44582677 Ki > 10000 nM T84117 C5QB4K 44582678 Ki > 10000 nM T84117 C01RCI 44582705 Ki > 10000 nM T84117 CXL25V 44582706 Ki > 10000 nM T84117 C8MR1X 44582707 Ki > 10000 nM T84117 C4IT1N 44582708 Ki > 10000 nM T84117 C5ZDY3 46915370 Ki = 2900 nM T84117 C2LZJ0 49783209 Ki = 10000 nM T84117 C57SMG 49783415 Ki > 10000 nM T84117 C0TG6I 49783419 Ki > 10000 nM T84117 C2RY0J 50878551 Ki = 413 nM T84117 C1W6TV 50898777 Ki > 10000 nM T84117 CXMZ73 50898778 Ki > 10000 nM T84117 CE4KP1 51050257 Ki > 10000 nM T84117 C1TC7Q 56963799 Ki > 10000 nM T84117 C1LEH8 67268994 Ki = 1366 nM T84117 C3XNC2 71450247 Ki > 10000 nM T84117 CAQF34 71455625 Ki > 10000 nM T84117 CMJ1O9 71457409 Ki > 10000 nM T84117 C63YLA 71461049 Ki > 10000 nM T84117 CJD96I 71461050 Ki > 10000 nM T84117 C4P3JU 71462776 Ki > 10000 nM T84117 C3GUQ2 71462777 Ki > 10000 nM T84117 CC6Q5R 72771081 Ki < 100 nM T84117 CC65OA 73213195 Ki > 10000 nM T84117 CW83DK 73213196 Ki > 10000 nM T84117 C2E7QW 75201901 Ki = 9800 nM T84117 C8IDL3 75306277 Ki = 2511.89 nM T84117 C70ZVB 86221574 Ki > 10000 nM T84117 CEMZ15 118464420 Ki > 10000 nM T84117 CV2L6O 118464425 Ki > 10000 nM T84117 CFNG86 118464427 Ki > 10000 nM T84117 C7ODW3 122195524 Ki > 900 nM T84117 C4QM2E 124247485 Ki = 793 nM T84117 CTBN56 127026052 Ki = 478.63 nM T84117 CU49VE 127036186 Ki = 489.78 nM T84117 CG06BD 127036932 Ki = 354.81 nM T84117 CVW71O 127036953 Ki = 512.86 nM T84117 C50GOC 130442480 Ki = 8900 nM T84117 CM04RF 130442572 Ki = 9900 nM T84117 CY8B9L 132060743 Ki = 403 nM T84117 C7FM0U 132060763 Ki = 1242 nM T84117 CGHO19 132060770 Ki = 1666 nM T84117 CAVB41 132584404 Ki > 10000 nM T84117 CBU81N 134149168 Ki > 10000 nM T84117 C6N8GM 135367405 Ki = 890 nM T84117 C6LU0C 135367816 Ki > 10000 nM T84117 CD2TH9 135367820 Ki > 10000 nM T84117 C5AMD9 135367857 Ki = 1787 nM T84117 C8WL0I 135449090 Ki > 10000 nM T84117 C03HVY 135846955 Ki > 10000 nM T84117 CE4QG5 135846981 Ki > 10000 nM T84117 C3UB7L 135846982 Ki > 10000 nM T84117 CUKO20 136020617 Ki > 10000 nM T84117 COF0U5 136020618 Ki > 10 nM T84117 CF89JI 136030596 Ki > 10000 nM T84117 CE8GB9 136030693 Ki > 10000 nM T84117 C65VFI 136030744 Ki > 10000 nM T84117 COIX80 136054961 Ki > 10000 nM T84117 C6R4IC 136118615 Ki > 10000 nM T84117 CHWC38 136118619 Ki > 10000 nM T84117 C5UDW3 136118620 Ki > 10000 nM T84117 C8I6UN 136118621 Ki > 10000 nM T84117 CCHM67 136118657 Ki > 10000 nM T84117 C0W1TM 136118658 Ki > 10000 nM T84117 CON04G 136118728 Ki > 10000 nM T84117 COX1F8 136118729 Ki > 10000 nM T84117 C0R5PV 136118732 Ki > 10000 nM T84117 CAE39V 136188797 Ki > 10000 nM T84117 CC6OP7 136244089 Ki > 10000 nM T84117 CLAP52 136259032 Ki > 10000 nM T84117 C7KC3T 145963830 Ki = 2400 nM T84117 CHDN35 145964150 Ki > 10000 nM T84117 C1KH2E 145964159 Ki > 10000 nM T84117 C12OVL 145965034 Ki > 10000 nM T84117 C5W4LM 145965940 Ki > 10000 nM T84117 C81VUO 145967771 Ki > 10 nM T84117 CJS56K 145967795 Ki > 10000 nM T84117 CQJ5O8 145971635 Ki > 10000 nM T84117 C7BVC1 145972374 Ki = 1400 nM T84117 C79TNE 145972796 Ki > 10000 nM T84117 C6XIN0 145974114 Ki > 10000 nM T84117 CD8ZL6 145974750 Ki > 10 nM T84117 C6PH4F 145975226 Ki = 4600 nM T84117 C71CYU 145975946 Ki > 10000 nM T84117 C2TN8W 145976085 Ki > 10000 nM T84117 C6BFY7 145977338 Ki > 10000 nM T84117 C0Y6QO 145977799 Ki = 4000 nM T84117 C3BI1R 145978113 Ki > 10000 nM T84117 CQU8R0 145978665 Ki > 10000 nM T84117 C6AV9G 145978819 Ki > 10000 nM T84117 C86XQR 145988313 Ki > 10000 nM T84117 CC2G1V 146025727 Ki = 7800 nM T84117 C6P3SR 153287553 Ki > 10000 nM T84117 CV9G7Z 153287572 Ki > 10000 nM T84117 CO85KL 153287574 Ki > 10000 nM T84117 CUSA24 155519891 Ki > 10000 nM T84117 CB79ZW 155536080 Ki > 10000 nM T84117 C3N9VU 10251906 Ki > 500 nM T84117 CRKP76 136016509 Ki > 10000 nM T84117 D00CRA 1574 Ki > 10000 nM T84117 D01HRV 9847194 IC50 > 10000 nM T84117 D03DET 10287730 Ki < 10000 nM T84117 D04AZE 3277600 Ki < 100000 nM T84117 D05XGR 6918647 Ki = 1584.89 nM T84117 D07LRJ 5312149 Ki < 10000 nM T84117 D08CKM 9863250 Ki < 10000 nM T84117 D09OYA 2107 Ki > 10000 nM T84117 D09PIN 3378093 Ki > 10000 nM T84117 D09RPR 16737207 Ki > 10000 nM T84117 D09WIL 10028436 Ki < 5011.87 nM T84117 D0C5GF 6918515 Ki > 10000 nM T84117 D0CK9K 6918513 Ki = 520 nM T84117 D0F6CD 5202 Ki = 4 nM T84117 D0H7PC 6918553 Ki > 10000 nM T84117 D0H9QG 5312148 Ki < 15848.93 nM T84117 D0L5MW 181743 Ki > 10000 nM T89879 D04AIT 5280445 IC50 = 20000 nM T89879 D07EXH 359 IC50 > 200000 nM T89879 D07MGA 72281 IC50 = 8300 nM T89879 D0J9ZR 4477 IC50 = 40000 nM T89879 D0K8KX 5280343 IC50 = 8100 nM T89879 C5H9TY 14697 IC50 = 207000 nM T89879 C3I7VB 102678 IC50 = 24500 nM T89879 CL5Y4J 159516 Ki = 3100 nM T89879 CV0B7W 442027 IC50 = 49600 nM T89879 C1E2FR 442048 IC50 = 283500 nM T89879 CZ3MD8 647122 IC50 = 16100 nM T89879 C2C8QU 948801 Ki = 27500 nM T89879 CXA4P6 1265413 IC50 = 90720 nM T89879 CUD4A1 1328543 IC50 = 58350 nM T89879 C3ZP4U 2131972 Ki = 9110 nM T89879 CA1N3H 2131982 Ki = 9930 nM T89879 CKL8B2 2219105 IC50 = 29900 nM T89879 CN43XQ 2806068 IC50 = 160 nM T89879 C5J6MO 2849659 IC50 = 28800 nM T89879 CN3P7A 2911959 IC50 = 74500 nM T89879 CZDG23 2947583 IC50 = 186000 nM T89879 CBIP72 2986413 IC50 = 76700 nM T89879 CCU3P7 3635406 IC50 = 2200 nM T89879 CZF0R5 4004950 IC50 = 500 nM T89879 C3AN7C 4117477 IC50 = 1180 nM T89879 CS2WB7 4236803 IC50 = 29800 nM T89879 C0AW3N 4378077 IC50 = 13860 nM T89879 CO3Y0T 4614896 IC50 = 9910 nM T89879 CY68ZT 4788586 IC50 = 940 nM T89879 CTR4Q1 5320532 IC50 = 13300 nM T89879 CVG47I 5958938 IC50 = 10500 nM T89879 CD8ZT2 6026688 IC50 > 50000 nM T89879 C3LZX9 8027611 IC50 = 12660 nM T89879 CJ4C5K 9180583 IC50 = 10800 nM T89879 CYQ8Z4 9882716 IC50 > 50000 nM T89879 C8K2NO 10062715 IC50 = 800000 nM T89879 C49CMU 10411574 IC50 = 21700 nM T89879 C6GN2F 11642725 IC50 = 870000 nM T89879 CHYP53 12310492 IC50 = 233400 nM T89879 C65EOH 15949840 IC50 = 7500 nM T89879 C9V8EM 15956553 IC50 = 300000 nM T89879 C3WYR4 16061499 IC50 = 2000 nM T89879 CTO43V 16085283 Ki = 116000 nM T89879 CU35DQ 21582568 IC50 = 220800 nM T89879 CN45FL 23427055 IC50 = 164700 nM T89879 CK3AF8 25256829 IC50 = 5400 nM T89879 C2SZ7L 42624533 IC50 = 14000 nM T89879 CYP8V1 44404067 IC50 > 50000 nM T89879 CD20PF 44433696 IC50 = 80000 nM T89879 CI4P2V 44433697 IC50 = 10000 nM T89879 CW7B0J 44433698 IC50 = 15000 nM T89879 C8DWL3 44433699 IC50 = 200000 nM T89879 C0ZPE2 44517748 IC50 = 2700 nM T89879 C0OH2T 44584893 IC50 = 5400 nM T89879 C0NZ5E 44584944 IC50 = 7300 nM T89879 CT70DZ 44590821 IC50 = 22500 nM T89879 C0SW2K 45266425 IC50 = 2500 nM T89879 C5WBP2 45266482 IC50 = 3800 nM T89879 CA4K8F 45266488 IC50 = 6600 nM T89879 C3BHZ4 45268445 IC50 > 50000 nM T89879 CC05NI 45268452 IC50 = 15400 nM T89879 C6QD9E 45269292 IC50 > 50000 nM T89879 CY7RV4 45269761 Ki = 21000 nM T89879 CO80TH 45269762 Ki = 297000 nM T89879 CU34ZK 45269763 Ki = 584000 nM T89879 C9P3LZ 45269764 Ki = 478000 nM T89879 CXS19V 45269765 Ki = 45200 nM T89879 C3DY4T 45270971 IC50 > 50000 nM T89879 CR4WA8 45270979 IC50 = 20900 nM T89879 CM78GO 45271412 Ki = 462000 nM T89879 CC90BU 45271826 IC50 = 5200 nM T89879 C0B6KX 45271831 IC50 = 9300 nM T89879 CN85IQ 45271832 IC50 = 8100 nM T89879 C7IF2O 45272299 Ki = 363000 nM T89879 CZRV73 45272304 Ki = 34100 nM T89879 CGV14L 45272305 Ki = 112000 nM T89879 CVTL97 45272306 Ki = 2200 nM T89879 CAM89I 45273174 Ki = 135000 nM T89879 CZT67B 45273179 Ki = 614000 nM T89879 CHF4M5 45273180 Ki = 49300 nM T89879 CND1R3 45273184 Ki = 159000 nM T89879 C0V5WT 45273625 IC50 > 50000 nM T89879 C6OE7V 46784066 IC50 = 28300 nM T89879 C6LH5I 46881919 Ki = 800 nM T89879 CI2FO1 49870840 IC50 = 5500 nM T89879 CF2D0I 49870841 IC50 = 8400 nM T89879 CM52SZ 49870842 IC50 = 6800 nM T89879 C8Q2CZ 50885062 IC50 > 50000 nM T89879 CJ6KV7 52941131 IC50 = 13900 nM T89879 C8M2QD 52943127 IC50 = 24300 nM T89879 CQ84MD 52945913 IC50 = 12000 nM T89879 CJ1LG2 52945915 IC50 = 42000 nM T89879 CZ35DX 52945977 IC50 = 128900 nM T89879 CAB1Y3 52946772 IC50 = 163200 nM T89879 CO4R1B 52947200 IC50 = 18000 nM T89879 CC4X1O 52948928 IC50 = 137700 nM T89879 CMG4U7 52949213 IC50 = 10800 nM T89879 C0X5BL 58589722 IC50 = 76740 nM T89879 CY3CL6 71544384 IC50 = 610 nM T89879 CV3P2U 71544385 IC50 = 230 nM T89879 CJS60O 71571220 IC50 = 49000 nM T89879 C1AY0M 71571221 IC50 = 49000 nM T89879 CY21XB 71571222 IC50 = 4600 nM T89879 C1DX9H 71571223 IC50 = 39000 nM T89879 CKE2C3 73056463 IC50 > 100000 nM T89879 C9S8ZH 73056464 IC50 > 100000 nM T89879 CK9OI0 73056465 IC50 = 31710 nM T89879 C4D8LK 73056466 IC50 = 32080 nM T89879 CRY86G 73056467 IC50 = 34910 nM T89879 C3VS4F 73056760 IC50 = 10070 nM T89879 CYH1F4 73056761 IC50 = 51330 nM T89879 C2CRZ8 73056762 IC50 = 2250 nM T89879 CD4YR3 73056763 IC50 = 11830 nM T89879 C3P2OZ 73056764 IC50 = 67200 nM T89879 C1H8PX 73056765 IC50 = 82910 nM T89879 C8JO7B 73056766 IC50 = 13860 nM T89879 CCYE63 73057087 IC50 = 5520 nM T89879 C54JWM 73057088 IC50 = 39870 nM T89879 C8RBU6 73057089 IC50 = 1040 nM T89879 CEBH65 73057090 IC50 = 1690 nM T89879 C8M2DX 73057091 IC50 = 17820 nM T89879 CQ42AZ 73057092 IC50 = 2820 nM T89879 CPLJ64 73057388 IC50 = 4700 nM T89879 CIN5V0 76320984 IC50 = 4300 nM T89879 C05AYV 102341658 IC50 = 16400 nM T89879 C8S3CR 102341659 IC50 = 37500 nM T89879 C2G9CP 127043455 IC50 = 20200 nM T89879 CVZ4I3 127043641 IC50 = 6000 nM T89879 C7BST4 127043642 IC50 = 5800 nM T89879 CGO01F 127043643 IC50 > 50000 nM T89879 C2TU5A 127043644 IC50 = 6400 nM T89879 C0Y9IT 127043645 IC50 = 41200 nM T89879 CF3B1Z 127045220 IC50 = 11700 nM T89879 CIXJ94 127045221 IC50 = 8600 nM T89879 CQ1CT5 127045222 IC50 = 18700 nM T89879 CKRX04 127045227 IC50 = 30700 nM T89879 CDZ2E1 127045228 IC50 > 50000 nM T89879 CG3E9B 127045229 IC50 = 6700 nM T89879 CG6VR3 127045386 IC50 = 15700 nM T89879 CK9JE3 127045387 IC50 > 50000 nM T89879 CY1E4Z 127045392 IC50 > 50000 nM T89879 CK5PA4 127045393 IC50 = 44700 nM T89879 C34TWD 127045394 IC50 > 50000 nM T89879 C97MQC 127048409 IC50 = 20000 nM T89879 C41VRM 127048410 IC50 = 7500 nM T89879 CZ0B1R 127052510 IC50 = 10000 nM T89879 CRW05E 127052511 IC50 > 50000 nM T89879 CC3TX0 127052512 Ki = 72000 nM T89879 CIQ1U9 127052513 Ki = 41000 nM T89879 CI13JZ 135452883 IC50 = 10000 nM T89879 CG1KW5 135470831 IC50 = 77090 nM T89879 CH4Q6A 145964401 IC50 = 5500 nM T89879 CHU61S 145964420 IC50 = 42100 nM T89879 C6YCA8 145964710 IC50 = 28800 nM T89879 CV6F7L 145966788 IC50 = 2100 nM T89879 CBWX17 145967285 IC50 = 4300 nM T89879 COR9X3 145972736 IC50 = 3900 nM T89879 CQ0M2X 145972809 IC50 = 4100 nM T89879 CF95RZ 145972878 IC50 = 3200 nM T89879 CXI0D1 145975081 IC50 = 6300 nM T89879 CG84ZR 145975487 IC50 = 5100 nM T89879 C91FOT 145976006 IC50 = 5200 nM T89879 C3F4UH 145978039 IC50 = 8800 nM T89879 CL7FB0 2919450 IC50 = 62790 nM T89879 D00RIX 5280443 IC50 = 280800 nM T89879 D01XMM 4117383 IC50 = 4450 nM T89879 D08MZY 145937 Ki = 8200 nM T89879 D08UYP 3008868 Ki = 2400 nM T89879 D09BUG 10207 IC50 = 132000 nM T89879 D0L7AT 10480940 Ki = 19300 nM T89879 D0S0BN 130976 Ki = 10600 nM T89879 D0SY2M 5281708 IC50 = 105000 nM T89879 D0UQ6U 10569 IC50 = 189100 nM T89879 D0WA9S 10429214 IC50 = 146500 nM T88752 C43DAY 68635 IC50 = 4600 nM T88752 C5KW4H 72311 IC50 = 7000 nM T88752 CYUH56 363208 IC50 = 31000 nM T88752 CWJ43S 443767 IC50 = 34000 nM T88752 CORM47 1849091 IC50 = 21300 nM T88752 C9N5XB 2026662 IC50 = 8700 nM T88752 CD8BS4 2999946 IC50 = 46100 nM T88752 CYZ0U7 4891910 IC50 = 5300 nM T88752 CAK90T 4893331 IC50 = 27900 nM T88752 CU8LQ0 4893774 IC50 = 24200 nM T88752 CF9QP2 9076354 IC50 = 24100 nM T88752 CT8RA9 9099810 IC50 = 57200 nM T88752 CK7N4D 9880653 IC50 = 2700 nM T88752 CD57RY 24344410 IC50 = 28300 nM T88752 CN3Y9K 25138381 IC50 = 9300 nM T88752 CDU76N 25164618 IC50 = 54000 nM T88752 C4OP0C 25165019 IC50 = 58000 nM T88752 C51DAH 45272995 IC50 = 12200 nM T88752 CP57CD 45483073 IC50 = 13000 nM T88752 CURM73 51031035 IC50 = 1100 nM T88752 C0EQA8 90655048 IC50 = 95000 nM T88752 C1KBS9 135431654 IC50 = 1800 nM T88752 C9PY6U 135959764 IC50 = 37000 nM T12581 CS1QX6 125545 EC50 = 210 nM T12581 CYPF58 443266 IC50 = 430 nM T12581 CVJZ65 12068910 IC50 = 6.1 nM T12581 C7R4XW 44458634 IC50 = 44 nM T12581 D0MH9X 107758 IC50 = 2.9 nM T12581 D0W1GH 121920 IC50 = 620 nM T84133 D05MQK 110635 IC50 > 10000 nM T84133 D06BCB 443955 IC50 > 10000 nM T84133 D0C9SY 135400189 IC50 = 790 nM T84133 D0F9GE 3108 Ki = 1000 nM T84133 D0NJ3V 4680 IC50 = 21 nM T84133 D0Z7ZM 135398744 IC50 = 3100 nM T84133 D01LCC 17754438 IC50 = 2700 nM T84133 D0EY0A 42636350 IC50 = 5500 nM T84133 D0OH2W 11581936 IC50 = 0.37 nM T84133 D0T5PO 5092 IC50 > 16000 nM T84133 D0X0PP 59351313 IC50 = 0.1 nM T84133 D01ITP 71295652 IC50 = 9 nM T84133 D03GTM 118485599 IC50 > 10000 nM T84133 D05VBJ 71295299 IC50 = 1760 nM T84133 D07EUB 46200734 IC50 = 9.83 nM T84133 D09BDD 56933838 IC50 = 506 nM T84133 D0J1LK 118485649 IC50 = 1200 nM T84133 D0WS3T 72706254 IC50 = 690 nM T84133 D00YPW 135399235 IC50 = 22000 nM T84133 D01FXD 9802841 IC50 > 10000 nM T84133 C0NP3E 7195 Ki = 500000 nM T84133 C4IQ1D 11829 Ki = 590000 nM T84133 CX06SW 11830 Ki = 94000 nM T84133 CBU72A 13021 Ki = 1300000 nM T84133 C67CJL 29872 Ki = 210000 nM T84133 CBIG84 66593 Ki = 500000 nM T84133 CIN2O4 67432 Ki = 410000 nM T84133 CL51WY 76081 Ki = 16000 nM T84133 C03JPW 76143 Ki = 1200000 nM T84133 C3YI1T 217632 Ki > 1000 nM T84133 C09RTL 243166 Ki = 300000 nM T84133 CG5QY2 305345 IC50 > 1000 nM T84133 C9LH4S 371187 IC50 = 48.8 nM T84133 C1B6ZL 662965 IC50 > 50000 nM T84133 CN9WF3 700124 IC50 = 851000 nM T84133 CM1XC0 735871 IC50 < 10000 nM T84133 CA5R2Z 866356 IC50 > 10000 nM T84133 CRW0V2 1122713 IC50 = 35 nM T84133 CHPF20 1188002 IC50 = 39 nM T84133 CNZ6L4 1366773 Ki = 87 nM T84133 CR94IK 1415219 IC50 = 210 nM T84133 C8JLO0 2243267 IC50 = 3500 nM T84133 C38ELQ 2776174 Ki = 940000 nM T84133 C7MYP8 2884317 IC50 = 68 nM T84133 CCL7M3 3685273 IC50 = 1000 nM T84133 CK12OT 3814427 IC50 = 84 nM T84133 CZ71SC 4080937 IC50 > 10000 nM T84133 CF95QS 4195078 IC50 = 3000 nM T84133 CVQ8G9 4259342 IC50 = 380 nM T84133 CW7AM9 4458268 IC50 = 4500 nM T84133 C2LMB4 5151485 IC50 = 310 nM T84133 CMK39Q 10553487 IC50 > 10000 nM T84133 C4BC0Z 10680968 IC50 = 1800 nM T84133 CF4SN3 11074154 Ki = 24000 nM T84133 C45VZC 11438405 IC50 > 16000 nM T84133 CIM6H8 11504190 IC50 = 16 nM T84133 CE0XC8 11512099 IC50 = 22 nM T84133 CJH21A 11517420 IC50 = 41.5 nM T84133 CI15RY 11525659 IC50 = 7 nM T84133 CLI15E 11533673 IC50 = 120 nM T84133 C4ZYH9 11547485 IC50 = 2200 nM T84133 CI95DB 11576116 IC50 = 6 nM T84133 C53ZEH 11590899 IC50 = 3 nM T84133 C3G1BO 11604203 IC50 = 0.28 nM T84133 C5S1WA 11613446 IC50 = 3 nM T84133 CQ6Z7B 11634505 IC50 = 4 nM T84133 CS3J8Z 11635020 IC50 = 2 nM T84133 C6GY9D 11635241 IC50 = 1900 nM T84133 C40YUX 11637556 IC50 = 16300 nM T84133 CB2G3L 11641069 IC50 = 2 nM T84133 C2J7OE 11641566 IC50 = 34 nM T84133 CU2RN6 11648276 IC50 = 0.3 nM T84133 C94GTK 11655421 IC50 = 4 nM T84133 CR8CQ7 11669507 IC50 = 0.29 nM T84133 C3XYS6 11698194 IC50 = 6 nM T84133 COU75F 11710344 IC50 = 3 nM T84133 CC1S6V 11720710 IC50 = 2 nM T84133 CA26IK 11742611 IC50 > 10000 nM T84133 CL6F4C 11955614 Ki = 4 nM T84133 CUK49V 11988837 Ki = 2700 nM T84133 CFIO49 11988967 Ki = 7900 nM T84133 C2D0NG 11989101 Ki = 5400 nM T84133 C65ABT 11989102 Ki = 19000 nM T84133 CY20HE 14943631 IC50 = 890 nM T84133 CSX70H 15991588 Ki = 12 nM T84133 C08TUE 16102593 Ki = 811 nM T84133 C7GDQ8 16102594 Ki = 240 nM T84133 CHAL10 16102596 Ki = 130 nM T84133 C6Z7GM 16102598 Ki = 54 nM T84133 C4JVF5 16102599 Ki = 136 nM T84133 CMR3A7 16102600 Ki = 68 nM T84133 CX1B4L 16102601 Ki = 44 nM T84133 CC0DP8 16102602 Ki = 123 nM T84133 CLH34A 16102603 Ki = 112 nM T84133 CK06QM 16102604 Ki = 210 nM T84133 C4TH8R 16102605 Ki = 17 nM T84133 C6X1VB 16102606 Ki = 18 nM T84133 C04SBT 16102607 Ki = 19 nM T84133 C9IK5Y 16102620 Ki = 326 nM T84133 CL6Y7J 16102621 Ki = 198 nM T84133 CNAW90 16102622 Ki = 56 nM T84133 C1GD3A 16102623 Ki = 100 nM T84133 CA52VZ 16102625 Ki = 94 nM T84133 CH25WX 16102626 Ki = 67 nM T84133 C5V1LM 16102627 Ki = 128 nM T84133 CC21RZ 16102628 Ki = 18 nM T84133 C5SN6Y 16102629 Ki = 12 nM T84133 C3S2KA 16102630 Ki = 12 nM T84133 C9XNR3 16419285 IC50 = 2400 nM T84133 C1L2MA 16582132 IC50 = 2500 nM T84133 COG39H 16727125 IC50 = 1500 nM T84133 C0MA2Z 17437959 IC50 = 15 nM T84133 C6J4OB 17454842 IC50 = 110 nM T84133 CXFT59 17757146 IC50 = 823 nM T84133 C1PZ8C 18734933 IC50 > 16000 nM T84133 C25GCV 19935268 Ki = 380000 nM T84133 CGJH45 21002944 IC50 = 1800 nM T84133 C7YT4G 21259157 IC50 = 324000 nM T84133 CW96SI 23624262 IC50 = 7 nM T84133 CJ0ZF1 24180492 IC50 = 430 nM T84133 C8MU9Q 24745788 IC50 = 21.4 nM T84133 CW2US9 24746467 IC50 = 125 nM T84133 C6LV1F 24802716 IC50 = 12.4 nM T84133 C9WGI4 24802717 IC50 = 7.28 nM T84133 CC25EQ 24802718 IC50 = 15.7 nM T84133 COM21S 24802719 IC50 = 81.2 nM T84133 C08NUH 24802721 IC50 = 51.3 nM T84133 C2OB3S 24802722 IC50 = 2.84 nM T84133 C7NVY6 24802884 IC50 = 223 nM T84133 C7CAQ3 24802885 IC50 = 116 nM T84133 C01PNE 24802891 IC50 = 8.32 nM T84133 C2QV8Z 24803049 IC50 = 32.5 nM T84133 CE4SQ3 24803050 IC50 = 25.1 nM T84133 CGT60I 24803051 IC50 = 13.2 nM T84133 COTR52 24803223 IC50 = 22.9 nM T84133 C3NKC1 24803224 IC50 = 206 nM T84133 CDEK56 24803227 IC50 = 535 nM T84133 CC6XU8 24803383 IC50 = 55.4 nM T84133 C67TRL 24803384 IC50 = 381 nM T84133 CVZ1G5 24803385 IC50 = 15.3 nM T84133 CO6ZN3 24803386 IC50 = 39.2 nM T84133 C9DSN4 24803387 IC50 = 64.7 nM T84133 C2TR8E 24803388 IC50 = 53.4 nM T84133 CN7GJ6 24803389 IC50 = 617 nM T84133 CI54GC 24803543 IC50 = 132 nM T84133 CFG52I 24804535 IC50 = 24.8 nM T84133 C0GY4W 24804536 IC50 = 92.2 nM T84133 CJ1U3Z 24804537 IC50 = 63 nM T84133 C4O0IX 24804538 IC50 = 270 nM T84133 CJ40AC 24804539 IC50 = 2270 nM T84133 CKR97Z 24804540 IC50 = 731 nM T84133 C5XFP1 24804699 IC50 = 149 nM T84133 C05DQY 24804701 IC50 = 391 nM T84133 CFC7X5 24804871 IC50 = 383 nM T84133 CZ4R9U 24805030 IC50 = 962 nM T84133 C8B5LM 24805034 IC50 = 617 nM T84133 CS0I7F 24805035 IC50 = 209 nM T84133 CE6QM4 24805036 IC50 = 2390 nM T84133 C76DWZ 24805199 IC50 = 10.9 nM T84133 CXB7H2 24805200 IC50 = 36.4 nM T84133 C07XUR 24805202 IC50 = 23.3 nM T84133 C6GIQ3 24805203 IC50 = 89.6 nM T84133 C10ADY 24805204 IC50 = 284 nM T84133 C79SXK 24805205 IC50 = 33.9 nM T84133 C20VHK 24871823 IC50 = 85 nM T84133 C0E9RA 24983496 IC50 = 9.7 nM T84133 C9WX7I 25195576 IC50 = 1.5 nM T84133 CG4HU9 25195579 IC50 = 7 nM T84133 CL1S8F 25195685 IC50 = 1.1 nM T84133 C0R2EF 25195686 IC50 = 17.3 nM T84133 CL1N8C 25195687 IC50 = 16.3 nM T84133 CQ64SM 25196602 IC50 = 4.9 nM T84133 CGZP65 25196603 IC50 = 13.2 nM T84133 CD35KE 25196606 IC50 = 1.2 nM T84133 C9BQI5 25196607 IC50 = 2.6 nM T84133 C9GIO4 25196715 IC50 = 3.2 nM T84133 CV0F2B 25196716 IC50 = 5.8 nM T84133 C4J0YD 25196719 IC50 = 1.52 nM T84133 CAR7F0 25197023 IC50 = 1.3 nM T84133 C64KEG 25218869 IC50 = 400 nM T84133 C4I8XH 42623946 IC50 = 472 nM T84133 CD4NM7 42623948 IC50 = 175 nM T84133 C14KMP 42624027 IC50 = 1050 nM T84133 CEJ67W 42624216 IC50 = 246 nM T84133 CJ6UR1 42624218 IC50 = 482 nM T84133 CMI41E 42624219 IC50 = 146 nM T84133 CS7RC9 42629350 IC50 = 13.3 nM T84133 C7SGR9 42629353 IC50 = 14.4 nM T84133 C9CE2J 42629699 IC50 = 13.9 nM T84133 CP9TE3 42629700 IC50 = 14.9 nM T84133 CICF39 42629702 IC50 = 11 nM T84133 CIFO36 42629821 IC50 = 65.3 nM T84133 CMIX45 42629822 IC50 = 173 nM T84133 CM3X9S 42629827 IC50 = 7.4 nM T84133 C29JFA 42629944 IC50 = 186 nM T84133 CQN26J 42629945 IC50 = 7.4 nM T84133 CRX87A 42629953 IC50 = 11 nM T84133 C6O5FX 42630062 IC50 = 1.8 nM T84133 CR2VK6 42630063 IC50 = 24 nM T84133 C1A4UY 42630064 IC50 = 20.5 nM T84133 CWT8E7 42630065 IC50 = 14.4 nM T84133 C70YVS 42630068 IC50 = 79.5 nM T84133 CTS74L 42630069 IC50 = 22 nM T84133 C3P1XN 42630071 IC50 = 3.9 nM T84133 C2O1WH 42630072 IC50 = 11.7 nM T84133 CGU0S3 42630073 IC50 = 1.5 nM T84133 C71ZNR 42630180 IC50 = 2.8 nM T84133 C7T8DM 42630184 IC50 = 46 nM T84133 C9UZW3 42630188 IC50 = 2.9 nM T84133 CX9ZT6 42630190 IC50 = 2 nM T84133 C4RHY0 42630191 IC50 = 0.7 nM T84133 CT6RS9 42630192 IC50 = 0.55 nM T84133 CYLS05 42630193 IC50 = 0.35 nM T84133 C7J0PY 42630314 IC50 = 1.5 nM T84133 CJC7B8 42630315 IC50 = 0.85 nM T84133 CCPV45 42630316 IC50 = 63.9 nM T84133 CYZL43 42630317 IC50 = 0.5 nM T84133 CH42OZ 42630318 IC50 = 0.2 nM T84133 C7X5AH 42630437 IC50 = 0.14 nM T84133 C8L7XT 42630438 IC50 = 7.5 nM T84133 C0ZFQ8 42630439 IC50 = 102 nM T84133 C5IVS3 42630440 IC50 = 1.9 nM T84133 CKE04L 42630684 IC50 = 9.62 nM T84133 CGV5A0 42630796 IC50 = 6 nM T84133 C18ZNC 42630799 IC50 = 21.4 nM T84133 C5Q0IN 42647289 IC50 = 388 nM T84133 CNIE98 44143458 IC50 = 632 nM T84133 CW8OB3 44243146 Ki = 1 nM T84133 CE8CL6 44440359 IC50 = 140 nM T84133 CWV38B 44440363 IC50 = 45 nM T84133 C6XB2I 44440367 IC50 = 30 nM T84133 C4Q1AZ 44440369 IC50 = 35 nM T84133 CG04FU 44440370 IC50 = 35 nM T84133 COCF81 44440373 IC50 = 7 nM T84133 CR25KM 44440389 IC50 = 5 nM T84133 CMAD80 44440391 IC50 = 0.3 nM T84133 C4RTA8 44440392 IC50 = 10 nM T84133 C9G1QE 44440395 IC50 = 1 nM T84133 CT7Q2I 44440397 IC50 = 4 nM T84133 CI87NE 44440399 IC50 = 2 nM T84133 CS07MP 44440400 IC50 = 18 nM T84133 CH0KB2 44440401 IC50 = 3 nM T84133 CF80NI 44440403 IC50 = 6 nM T84133 CJQP98 44440404 IC50 = 21 nM T84133 CS6W5I 44440405 IC50 = 1900 nM T84133 CM0PA2 44440406 IC50 > 4000 nM T84133 CVR47J 44440407 IC50 = 100 nM T84133 CX0LW3 44440408 IC50 = 18 nM T84133 CVK5U4 44440409 IC50 = 120 nM T84133 CJCX12 44440410 IC50 = 160 nM T84133 C4UD9G 44440415 IC50 = 79 nM T84133 C8JDH7 44440416 IC50 = 4000 nM T84133 CA0E7D 44440418 IC50 = 1300 nM T84133 C1NZE3 44441802 IC50 = 2800 nM T84133 CM13IX 44441825 IC50 = 130 nM T84133 CSD1Q8 44441827 IC50 = 1100 nM T84133 CG49SA 44441829 IC50 = 600 nM T84133 C8FK0V 44441831 IC50 = 120 nM T84133 CTI03C 44441833 IC50 = 20 nM T84133 CZYW49 44441837 IC50 = 760 nM T84133 CQ0N7Y 44441840 IC50 = 1700 nM T84133 C98UBL 44452447 Ki = 185 nM T84133 CPOZ04 44452603 Ki = 171 nM T84133 CK9NU0 44537944 IC50 = 7.2 nM T84133 CUO2D3 44539913 IC50 < 50 nM T84133 CCVO04 44546588 IC50 < 50 nM T84133 CS2A4J 44547515 IC50 = 0.32 nM T84133 CY41QP 44547965 IC50 = 0.32 nM T84133 C7GNE3 44548113 IC50 = 67 nM T84133 CGP02T 44555440 IC50 < 50 nM T84133 CDQP73 44608934 IC50 = 7.2 nM T84133 CM83YD 46174637 IC50 = 0.0033 nM T84133 CI68SV 46178283 IC50 = 0.44 nM T84133 C6LZJ3 46185994 IC50 < 50 nM T84133 CC0OM2 46185995 IC50 < 50 nM T84133 C0D2MN 46186792 IC50 = 13.1 nM T84133 CR1K5E 46198523 IC50 = 9.6 nM T84133 C58BSW 46198541 IC50 = 2430 nM T84133 C1BIJ2 46198546 IC50 = 388 nM T84133 CC42ER 46198694 IC50 = 45.5 nM T84133 C0WRO9 46198713 IC50 = 45.9 nM T84133 CON1M4 46199019 IC50 = 91.3 nM T84133 C5AND7 46199167 IC50 = 114 nM T84133 CKX1A6 46199301 IC50 = 23.7 nM T84133 CZU0H7 46199329 IC50 = 51.5 nM T84133 CD9LN1 46199458 IC50 = 77.2 nM T84133 CXG34R 46199487 IC50 = 47.6 nM T84133 CAL85J 46199794 IC50 = 12.4 nM T84133 CZF5C0 46199795 IC50 = 42.4 nM T84133 CI9EA4 46199799 IC50 = 10.1 nM T84133 C26RJV 46200090 IC50 = 3.3 nM T84133 C5WND9 46200233 IC50 = 1.48 nM T84133 CKIC45 46200238 IC50 = 4.16 nM T84133 CS46AE 46200399 IC50 = 2.06 nM T84133 C1S3BK 46200706 IC50 = 1.53 nM T84133 C4P5QJ 46200709 IC50 = 2.41 nM T84133 CV8Y6W 46200711 IC50 = 3.99 nM T84133 CK1N4X 46200728 IC50 = 15 nM T84133 CH9FU8 46200877 IC50 = 8.33 nM T84133 CEZ3V4 46200878 IC50 = 9.43 nM T84133 C10HQS 46207696 IC50 < 25 nM T84133 C5N9FO 46207938 IC50 = 4.5 nM T84133 CF8UT3 46207939 IC50 = 24.4 nM T84133 CNHS37 46208071 IC50 = 2.8 nM T84133 COGX29 46208072 IC50 = 4.1 nM T84133 CRBA01 46208073 IC50 = 7.2 nM T84133 CJKH84 46208209 IC50 = 20.6 nM T84133 CIJ62X 46208210 IC50 = 5.1 nM T84133 CRXN04 46208214 IC50 = 5.1 nM T84133 C6IRP8 46208470 IC50 = 1.7 nM T84133 CF6Z5P 46208937 IC50 = 168 nM T84133 CAO2U6 46208939 IC50 = 1.1 nM T84133 C8DY5G 46209045 IC50 = 4.3 nM T84133 C36XLQ 46209046 IC50 = 4.2 nM T84133 C2Q4YT 46209162 IC50 = 138 nM T84133 CJOE41 46209386 IC50 = 0.199 nM T84133 C3P4SJ 46209520 IC50 = 1 nM T84133 C7ZY8O 46219578 IC50 = 14 nM T84133 C4UL5T 46238926 IC50 < 100 nM T84133 CU73QW 46238927 Ki = 130 nM T84133 CB9S1L 46239023 Ki = 3 nM T84133 C0V6EL 46239024 Ki = 280 nM T84133 C1HNK7 46239025 IC50 < 100 nM T84133 CYQ09Z 46239122 Ki = 5 nM T84133 CH8B1X 46239123 Ki = 15 nM T84133 C8WI1G 46239124 Ki = 29 nM T84133 CLG7K1 46239125 Ki = 14 nM T84133 CAE91W 46239126 Ki = 409 nM T84133 CV5DO7 46239228 Ki = 52 nM T84133 CED8X2 46239234 Ki = 3.3 nM T84133 CZQ5T9 46239329 Ki = 1 nM T84133 C7N8FR 46239331 Ki = 202 nM T84133 CIEM75 46239333 Ki = 871 nM T84133 CI7EX8 46239423 Ki = 32 nM T84133 C5IMB2 46239424 Ki = 3 nM T84133 CKR9P7 46239425 Ki = 3 nM T84133 CJB81K 46239426 Ki = 49 nM T84133 CEP91S 46239427 Ki = 24 nM T84133 CZV29L 46239429 Ki = 57 nM T84133 CZ5G3P 46239530 Ki = 30 nM T84133 C7SLP0 46239531 Ki = 0.6 nM T84133 CNI1U7 46239532 Ki = 37 nM T84133 CS64WE 46239728 Ki = 104 nM T84133 C95RNE 46239731 IC50 < 100 nM T84133 CAK37R 46239835 Ki = 70 nM T84133 CGBT01 46239836 Ki = 3.6 nM T84133 C08FHG 46239839 Ki = 41 nM T84133 CI1F5C 46239840 Ki = 11 nM T84133 C7P3HS 46239939 Ki = 23 nM T84133 C0X8CQ 46239940 Ki = 363 nM T84133 C0GJN1 46239943 Ki = 15 nM T84133 C26XVS 46240044 Ki = 12 nM T84133 C15QIP 46240135 Ki = 196 nM T84133 C8XFU6 46240137 Ki = 55 nM T84133 CO17GN 46683800 IC50 = 1300 nM T84133 CWB30P 46831671 IC50 = 81.5 nM T84133 C5C0KQ 46831672 IC50 = 486 nM T84133 C8TJ7K 46831673 IC50 = 1195 nM T84133 CY91XU 46831931 IC50 = 1.43 nM T84133 CKE4T9 46831932 IC50 = 7.33 nM T84133 C7TL2F 46831933 IC50 = 45.8 nM T84133 C8BWX3 46831934 IC50 = 285 nM T84133 C8RAC0 46831935 IC50 = 326 nM T84133 CE4JU7 46842025 IC50 > 10000 nM T84133 CR8JC2 46842169 IC50 > 10000 nM T84133 C6WM0L 46848741 IC50 = 0.79 nM T84133 CE6FK9 46848917 IC50 = 0.94 nM T84133 CJ4R0P 46849078 IC50 < 10 nM T84133 C9VW5F 46872031 IC50 = 27 nM T84133 C7QXI6 46873747 IC50 = 9 nM T84133 C3P2IN 46933992 IC50 >= 43000 nM T84133 COKU43 46937608 IC50 < 10 nM T84133 C3DH7C 49821302 IC50 = 5.7 nM T84133 C9Q6KE 49821304 IC50 = 3.5 nM T84133 CE8Y6Q 49821305 IC50 = 5.5 nM T84133 C94YDM 49821342 Ki = 6.1 nM T84133 C3WO9Y 49821343 Ki = 0.1 nM T84133 CAWZ34 49821394 IC50 = 0.05 nM T84133 C3TVS5 49821396 IC50 = 0.06 nM T84133 CHA5Z0 49821469 IC50 = 0.7 nM T84133 CL1BK9 49821500 Ki = 2 nM T84133 CD3C4H 49821501 Ki = 20 nM T84133 CE7GI8 49821502 Ki = 219 nM T84133 CHE15O 49821503 Ki = 0.072 nM T84133 C1ZGA8 49821582 Ki = 0.37 nM T84133 C1AYP0 49821627 IC50 = 0.09 nM T84133 C85AXR 49821714 IC50 = 0.8 nM T84133 CE41RK 49821911 Ki = 0.9 nM T84133 C5KU8W 49821931 Ki = 0.15 nM T84133 CEH5A1 49821987 Ki = 0.63 nM T84133 CF49WN 49821989 Ki = 0.92 nM T84133 C15XPB 49821991 Ki = 1 nM T84133 C29WPI 49822075 Ki = 135 nM T84133 C09BVO 49822155 Ki = 14 nM T84133 C0B8JE 49843464 IC50 < 10 nM T84133 C7Z0UN 50901948 Ki = 186 nM T84133 C3TR2P 50901952 Ki = 508 nM T84133 CMN05G 50901953 Ki = 31 nM T84133 CO4XK6 50901954 Ki = 861 nM T84133 C7V0OZ 50902028 Ki = 199 nM T84133 C9GT3X 50902029 Ki = 121 nM T84133 CZS03D 50902030 Ki = 29 nM T84133 C5I0LT 50902031 Ki = 101 nM T84133 CXT78Y 50902034 Ki = 40 nM T84133 C18FIN 50902113 Ki = 212 nM T84133 CPL5E6 50902114 Ki = 30 nM T84133 C6P8UV 50902116 Ki = 114 nM T84133 CK62ML 50902118 Ki = 628 nM T84133 CAD40F 50902119 Ki = 33 nM T84133 CD98UC 50902202 Ki = 32 nM T84133 CXB85R 50902203 Ki = 6.4 nM T84133 C9QLF2 50902206 Ki = 8 nM T84133 CH2Z1E 50902289 Ki = 20 nM T84133 C4HJL2 50902291 Ki = 25 nM T84133 C7EQ9Y 50902548 Ki = 10 nM T84133 C6A1IU 50902549 Ki = 8.7 nM T84133 CVM28N 50902550 Ki = 1.5 nM T84133 CN1P7Q 50902632 Ki = 4.3 nM T84133 C17RSC 50902804 IC50 < 10 nM T84133 C3Y2AV 50903255 Ki = 35 nM T84133 CDXL06 50942847 Ki = 15 nM T84133 CUI54F 50944015 Ki = 47.9 nM T84133 C6R4YN 50993785 IC50 = 12 nM T84133 C0M6XL 50993786 IC50 = 16 nM T84133 CSG76C 50993859 IC50 = 50 nM T84133 C6PQ3C 51000508 IC50 < 0.1 nM T84133 C2CK4X 51033482 IC50 = 0.2 nM T84133 CSNM30 51034710 IC50 = 0.1 nM T84133 C5Z3KH 51034712 IC50 = 0.1 nM T84133 C58OLQ 51304060 IC50 = 1300 nM T84133 C0IQM5 53232478 Ki = 17 nM T84133 CV35MO 53236526 IC50 = 1 nM T84133 CVRM83 53250985 IC50 = 6.7 nM T84133 CM48WF 53317312 IC50 = 76 nM T84133 CYBI97 53317313 IC50 = 50 nM T84133 C4YEK3 53317314 IC50 = 31 nM T84133 CJDV81 53318548 IC50 = 110 nM T84133 CLOI58 53319920 IC50 = 78 nM T84133 C3TI4S 53321175 IC50 = 83 nM T84133 CV3OG4 53322495 IC50 = 0.18 nM T84133 CBHF42 53323878 IC50 = 100 nM T84133 C40SMX 53323879 IC50 = 160 nM T84133 C9IVN4 53323880 IC50 = 16 nM T84133 C5JN2O 53323881 IC50 = 430 nM T84133 C5SY0C 53325113 IC50 = 130 nM T84133 C5XSA2 53325521 IC50 = 37 nM T84133 C8GH0Z 53326417 IC50 = 48 nM T84133 CZU82C 53326418 IC50 = 73 nM T84133 CZ48TX 53326461 IC50 = 52 nM T84133 CSD57U 53329353 IC50 < 1 nM T84133 COX9K5 53330053 IC50 = 2 nM T84133 CND92B 53363484 IC50 < 1000 nM T84133 CQL2P8 53378114 IC50 < 1000 nM T84133 CV3K8C 53467809 IC50 = 35 nM T84133 C7ZT0S 53468024 IC50 = 6 nM T84133 CX9Z8Q 53492734 IC50 < 100 nM T84133 CXCN02 54575101 IC50 < 100 nM T84133 CD5BR2 54575103 IC50 < 100 nM T84133 CX42VW 54575159 IC50 < 100 nM T84133 C94QRU 54576233 IC50 = 39 nM T84133 CHLA42 54576311 IC50 = 49 nM T84133 C6DEG8 54576313 IC50 = 58.5 nM T84133 CJF0K2 54576315 IC50 = 55 nM T84133 CNW81G 54576317 IC50 = 55 nM T84133 CA4I3X 54576449 IC50 = 15 nM T84133 C9WEO5 54576525 IC50 = 28 nM T84133 C3Y4WG 54576665 IC50 = 17 nM T84133 C4XM9U 54580514 IC50 = 14 nM T84133 CMG4F7 54580515 IC50 = 65 nM T84133 CE12AP 54581526 IC50 = 55 nM T84133 C19DVI 54581527 IC50 = 150 nM T84133 C9T4HK 54581943 IC50 = 1300 nM T84133 CAG1V9 54581955 IC50 = 1100 nM T84133 CV49PU 54582523 IC50 = 250 nM T84133 C2P3JM 54582524 IC50 > 10000 nM T84133 CMJ01N 54582525 IC50 = 120 nM T84133 C2RXU9 54582878 IC50 = 460 nM T84133 C59NEO 54582879 IC50 = 1000 nM T84133 CAL7N2 54582880 IC50 = 1900 nM T84133 C8ZDG9 54583877 IC50 = 320 nM T84133 CRY06I 54584473 IC50 = 130 nM T84133 C61CGS 54584474 IC50 = 790 nM T84133 CKBN97 54584475 IC50 = 190 nM T84133 CPG8Y9 54584829 IC50 > 10000 nM T84133 CL8N6Q 54585783 IC50 > 10000 nM T84133 C8XMH0 54585784 IC50 = 1600 nM T84133 C7GSO3 54585785 IC50 = 460 nM T84133 CRH83J 54585786 IC50 = 170 nM T84133 C8MGS6 54585797 IC50 = 2300 nM T84133 C8AI1O 54586387 IC50 = 8900 nM T84133 CCPD21 54586388 IC50 = 990 nM T84133 CKEP52 54586389 IC50 = 160 nM T84133 C7Z1YC 54586766 IC50 = 1500 nM T84133 CI4CO0 54587803 IC50 = 450 nM T84133 CFX89L 54587804 IC50 = 35 nM T84133 C0M5CY 54595731 Ki = 8700 nM T84133 CGF65A 54670110 IC50 = 29 nM T84133 CN4XU7 54670394 IC50 = 4100 nM T84133 C90ZLC 54670399 IC50 = 6.8 nM T84133 CAEJ46 54670484 IC50 = 7800 nM T84133 CSVE57 54670488 IC50 = 11000 nM T84133 C2JF8C 54670489 IC50 = 5700 nM T84133 C6AF1J 54671050 IC50 = 166000 nM T84133 CMT5R1 54671051 IC50 = 45000 nM T84133 C0UA1I 54674275 IC50 = 21.9 nM T84133 C5CZF9 54755130 IC50 < 500 nM T84133 CI91NY 54759276 IC50 = 140 nM T84133 C0K7YN 54760757 IC50 = 13.7 nM T84133 CJLD10 54769120 IC50 = 112 nM T84133 CKP39D 54769350 IC50 = 198 nM T84133 CWQ7S3 54769351 IC50 = 244 nM T84133 CR62YP 54769352 IC50 = 237 nM T84133 CVL03F 54769353 IC50 = 500 nM T84133 C97ACM 54769354 IC50 = 872 nM T84133 CX8P1B 54769355 IC50 = 248 nM T84133 C79BUR 54769575 IC50 = 303 nM T84133 CRA91G 54769784 IC50 = 469 nM T84133 CM96AK 54769785 IC50 = 246 nM T84133 CDRM84 56587975 IC50 = 12 nM T84133 CXI6G8 56596127 IC50 = 16 nM T84133 C1AC8K 56596128 IC50 = 93 nM T84133 CJ06ML 56596176 IC50 = 130 nM T84133 CI48VY 56596177 IC50 = 240 nM T84133 CJI54S 56596178 IC50 = 400 nM T84133 C7LF6A 56596179 IC50 = 170 nM T84133 C9NH1J 56596227 IC50 = 110 nM T84133 C7LPG5 56596228 IC50 = 31 nM T84133 CQY73S 56596229 IC50 = 61 nM T84133 C7G4FQ 56596230 IC50 = 250 nM T84133 C8FVQ1 56596231 IC50 = 12 nM T84133 COHX27 56648495 IC50 = 1.9 nM T84133 C4TGL7 56648496 IC50 = 4.3 nM T84133 C43WOF 56648497 IC50 = 60 nM T84133 CM3OI5 56648498 IC50 = 44 nM T84133 CM09EW 56648583 IC50 = 102 nM T84133 CIT68E 56648584 IC50 = 87 nM T84133 C9U0JW 56648585 IC50 = 114 nM T84133 C8O9PD 56648586 IC50 = 197 nM T84133 C52KXF 56648587 IC50 = 7.3 nM T84133 C9NC5E 56648588 IC50 = 18.2 nM T84133 CSZ6J1 56648589 IC50 = 14.2 nM T84133 CH6C3L 56648679 IC50 = 6.1 nM T84133 CCY79V 56648680 IC50 = 3.7 nM T84133 CL6Q1H 56648681 IC50 = 4.2 nM T84133 C4PH0I 56648682 IC50 = 73.4 nM T84133 CR0C8I 56648683 IC50 = 7.9 nM T84133 C15YZK 56648684 IC50 = 5.2 nM T84133 C9Z8TP 56648763 IC50 = 3.6 nM T84133 CNTL59 56648764 IC50 = 113 nM T84133 CT7QP0 56648765 IC50 = 158 nM T84133 CF95SJ 56648766 IC50 = 49.2 nM T84133 C0HX6Z 56648767 IC50 = 28.9 nM T84133 C85VDI 56648768 IC50 = 24.2 nM T84133 C0Y1RV 56648769 IC50 = 46 nM T84133 CNE96P 56648857 IC50 = 8.3 nM T84133 CU95MC 56648858 IC50 = 35.7 nM T84133 CX86AQ 56648859 IC50 = 7.4 nM T84133 CLV5E3 56648860 IC50 = 6.8 nM T84133 C6QG0A 56648861 IC50 = 11.4 nM T84133 CL8QN3 56648862 IC50 = 1.7 nM T84133 C16DEO 56648951 IC50 = 0.1 nM T84133 CG9DR0 56651641 IC50 = 0.08 nM T84133 CCM2A1 56654130 IC50 = 0.81 nM T84133 CPC3T4 56654131 IC50 = 0.76 nM T84133 CY04IO 56658425 IC50 = 200 nM T84133 CQZ4U7 56675681 IC50 = 262 nM T84133 CNX6T3 56834947 Ki = 14 nM T84133 C0YD3P 56928304 IC50 > 5000 nM T84133 C8RO6A 56929788 IC50 > 1000 nM T84133 CB5TR6 56949351 Ki = 0.01 nM T84133 CHL1C5 56949449 Ki = 0.02 nM T84133 C71JRF 56949451 Ki = 0.0082 nM T84133 CEU98Q 56949473 Ki = 9 nM T84133 CG0A3Z 56949475 Ki = 2 nM T84133 C9D8GO 56949508 Ki = 0.04 nM T84133 CP6AS2 56952795 Ki = 9.2 nM T84133 CZK51H 57328384 IC50 = 1 nM T84133 C0ZF1L 57328385 IC50 = 1 nM T84133 C8C1EW 57334262 Ki = 3 nM T84133 CLI7H6 57390414 Ki = 585 nM T84133 C9F7UR 57390415 Ki = 0.6 nM T84133 CWD1J3 57390416 Ki = 3.1 nM T84133 CZ2V5R 57390439 IC50 = 92.8 nM T84133 CJ0TI1 57390440 IC50 = 16.4 nM T84133 C94ZPA 57391164 Ki = 50 nM T84133 CD07RK 57391165 Ki = 2 nM T84133 CC76GU 57391166 Ki = 39 nM T84133 C4G1ZM 57391317 IC50 = 65 nM T84133 CC9N2A 57391318 IC50 = 22 nM T84133 C7T6XA 57391319 IC50 = 8 nM T84133 C9B5VW 57391320 IC50 = 67 nM T84133 C4QFY6 57392208 Ki = 550 nM T84133 C3TY1C 57392228 IC50 = 5.8 nM T84133 C31CEX 57392229 IC50 = 7.5 nM T84133 CZ09KG 57392230 IC50 = 13 nM T84133 C9TE7C 57392231 IC50 = 1.9 nM T84133 CR0GQ3 57392232 IC50 = 4 nM T84133 C4EGB7 57392860 IC50 = 12.9 nM T84133 C9JYK4 57392932 Ki = 12 nM T84133 CG2V1L 57392939 Ki = 26 nM T84133 CP0U1L 57392947 Ki = 153 nM T84133 CG3DF1 57392948 Ki = 8 nM T84133 CZ7X3C 57392949 Ki = 19 nM T84133 C7D3LX 57392950 Ki = 1200 nM T84133 C03TGV 57393096 IC50 = 561 nM T84133 C7GNB1 57393097 IC50 = 315 nM T84133 CZFH10 57393098 IC50 = 13 nM T84133 C6Q2PY 57393099 IC50 = 2 nM T84133 C2Z0ND 57393100 IC50 = 1770 nM T84133 CN0M9Y 57393928 IC50 = 6.2 nM T84133 CF1S9B 57393964 Ki = 0.5 nM T84133 C3R8KN 57393977 IC50 = 12.2 nM T84133 CW61NE 57394681 Ki = 171 nM T84133 CE36TV 57394695 Ki = 1 nM T84133 CMGZ76 57394696 Ki = 41 nM T84133 C9BMF8 57394826 IC50 = 21 nM T84133 C4NZS8 57395703 Ki = 419 nM T84133 CGZB82 57395734 IC50 = 124 nM T84133 C4WIC9 57395735 IC50 = 36.9 nM T84133 CF8UW0 57395736 IC50 = 10.9 nM T84133 CYV61E 57395737 IC50 = 18.6 nM T84133 CJ1UO3 57395738 IC50 = 2.6 nM T84133 C1MB4C 57395739 IC50 = 1.6 nM T84133 CE75UA 57396432 Ki = 2 nM T84133 C9K7YS 57396433 Ki = 4 nM T84133 CWE8N9 57396434 Ki = 21 nM T84133 CS0XU5 57396444 Ki = 353 nM T84133 C9L0ID 57396451 Ki = 9 nM T84133 C7VA8P 57396452 Ki = 229 nM T84133 C62JOU 57396592 IC50 = 746 nM T84133 CI25UB 57396593 IC50 = 27 nM T84133 CB71KN 57396814 Ki = 21 nM T84133 CTJN91 57397492 Ki = 35 nM T84133 CPI4V0 57397493 Ki = 27 nM T84133 C0TPH2 57397516 IC50 = 320 nM T84133 C5TJQ7 57397517 IC50 = 7.6 nM T84133 C5LNO0 57397518 IC50 = 40.6 nM T84133 CDWI58 57398224 Ki = 0.4 nM T84133 CG8B2K 57398367 IC50 = 144 nM T84133 C58IAE 57398368 IC50 = 97 nM T84133 CWQI09 57398380 IC50 = 608 nM T84133 CDSH51 57398573 Ki = 0.6 nM T84133 C7WH5G 57398574 Ki = 2 nM T84133 C8H2CI 57399125 IC50 = 3 nM T84133 CK85OQ 57399182 Ki = 6 nM T84133 CJT6U2 57399198 IC50 = 590 nM T84133 CU9XL6 57399199 IC50 = 4.4 nM T84133 C0LVB6 57399872 Ki = 83 nM T84133 C1U7LP 57399873 Ki = 1 nM T84133 CYC7S5 57399874 Ki = 0.2 nM T84133 CR9L0Z 57400027 IC50 = 9 nM T84133 CZAG81 57400035 IC50 = 13 nM T84133 C2GO5M 57400235 Ki = 54 nM T84133 CSE92V 57400886 IC50 = 1.8 nM T84133 CSQ5K8 57400960 IC50 = 10.1 nM T84133 CF7X2D 57400961 IC50 = 3 nM T84133 C7PY8W 57400962 IC50 = 2.4 nM T84133 CI0PX2 57401662 Ki = 804 nM T84133 C4PBS1 57401836 IC50 = 108 nM T84133 C3MB2N 57401837 IC50 = 31 nM T84133 CMS98N 57402038 Ki = 0.07 nM T84133 COMK36 57402700 Ki = 9.6 nM T84133 C09BLM 57402720 IC50 = 181 nM T84133 C6DI8T 57402721 IC50 = 24.4 nM T84133 CU14SI 57402722 IC50 = 9.7 nM T84133 C6B3IK 57403377 Ki = 0.3 nM T84133 CW54GL 57403378 Ki = 11 nM T84133 CI9A1D 57403379 Ki = 1 nM T84133 CPA3D1 57403394 Ki = 2 nM T84133 CQVZ29 57403395 Ki = 46 nM T84133 CU7OS0 57403396 Ki = 60 nM T84133 C14ASM 57403543 IC50 = 3 nM T84133 CR43CG 57403544 IC50 = 456 nM T84133 CJZ62H 57403545 IC50 = 52 nM T84133 C4EWA9 57403779 Ki = 0.06 nM T84133 C1H5LA 57403780 Ki = 10 nM T84133 C8HW7P 57523648 IC50 = 5.7 nM T84133 CZM4V5 58072466 IC50 < 10 nM T84133 CU8K2W 58074722 IC50 < 10 nM T84133 CRCT63 58368041 IC50 < 1 nM T84133 CSH3D7 58432081 IC50 < 1000 nM T84133 CFY5X9 58432151 IC50 < 1000 nM T84133 C7VFY2 58446918 IC50 = 1.9 nM T84133 C8I4YF 58547692 IC50 = 11000 nM T84133 C1ARH3 58547740 IC50 = 12000 nM T84133 CY7T1P 58547742 IC50 = 13000 nM T84133 CX1RJ5 58547786 IC50 = 29000 nM T84133 C7N2CL 58547789 IC50 = 147000 nM T84133 CV40CE 58547801 IC50 = 32000 nM T84133 C4XMB6 58547809 IC50 = 4700 nM T84133 CEB3G9 58547814 IC50 = 2.6 nM T84133 CYDO80 58547818 IC50 = 350000 nM T84133 CSAK24 58547819 IC50 = 46000 nM T84133 C08QVG 58547833 IC50 = 2.4 nM T84133 CP9N4A 58547845 IC50 = 54000 nM T84133 CFVG67 58547863 IC50 = 6500 nM T84133 CKR02G 58547875 IC50 = 43000 nM T84133 COD7Z3 58547879 IC50 = 38000 nM T84133 C2S8LJ 58547883 IC50 = 343000 nM T84133 C26PHF 58547902 IC50 = 41000 nM T84133 C02IVH 58547942 IC50 = 10300 nM T84133 C1GR4Z 58547944 IC50 = 64000 nM T84133 C57KYU 58547951 IC50 = 30000 nM T84133 CW82DY 58547956 IC50 = 36000 nM T84133 CYG43X 58548001 IC50 = 107000 nM T84133 C35JZX 58548005 IC50 = 45000 nM T84133 CUM63O 58548012 IC50 = 30000 nM T84133 CS80ZD 58548016 IC50 = 32000 nM T84133 CM8SN3 58548022 IC50 = 125000 nM T84133 CY5R2D 58548040 IC50 = 103000 nM T84133 CU85ZP 58548075 IC50 = 18000 nM T84133 CYZA38 58548077 IC50 = 6.8 nM T84133 C62WUD 58548080 IC50 = 39000 nM T84133 CCXW43 58548107 IC50 = 8500 nM T84133 CCHM36 58548113 IC50 = 38000 nM T84133 C91KHW 58548143 IC50 = 98000 nM T84133 C2IDR8 58548163 IC50 = 12 nM T84133 C4O5QX 58548370 IC50 = 31.5 nM T84133 C1GD9K 58578146 Ki < 1000 nM T84133 C2D4WV 58578164 Ki < 1000 nM T84133 CX7ZO2 58578167 Ki < 1000 nM T84133 CWX3N7 59320301 IC50 = 432 nM T84133 C7PB1U 59321218 IC50 = 53.1 nM T84133 CS32XI 59321284 IC50 = 1.48 nM T84133 C23WQA 59321310 IC50 = 7 nM T84133 CX45HS 59321315 IC50 = 0.7 nM T84133 CZ6C9L 59321318 IC50 = 5.11 nM T84133 C1OHZ0 59321339 IC50 = 1.85 nM T84133 C31ZBU 59326858 IC50 = 0.1 nM T84133 CHP92T 59326873 IC50 = 0.21 nM T84133 C16BHM 59326903 IC50 = 0.05 nM T84133 C6LF8T 59327006 IC50 = 0.1 nM T84133 CFL10E 59327126 IC50 = 45 nM T84133 C80VMG 59327176 IC50 = 0.96 nM T84133 C0EP5I 59341847 IC50 > 10000 nM T84133 CHQ28A 59341978 IC50 > 10000 nM T84133 CWF0O7 59351198 IC50 = 0.8 nM T84133 CJ0YB8 59351288 IC50 = 2.4 nM T84133 CZI6T1 59351366 IC50 = 7.4 nM T84133 CCA1H6 59351376 IC50 = 19.3 nM T84133 CX46SN 59351424 IC50 = 12.5 nM T84133 CEJX65 59370073 IC50 = 6 nM T84133 C64YEX 59373996 IC50 = 36.6 nM T84133 C2JW6Y 59436207 IC50 < 10 nM T84133 CMQH82 59453408 IC50 = 7 nM T84133 C0AFM6 60150358 IC50 = 0.28 nM T84133 CE0Q1S 60152740 IC50 > 1000 nM T84133 CJK53Q 60152741 IC50 = 45 nM T84133 CI3GJ1 66678348 Ki = 8.4 nM T84133 C6C8RD 66802145 IC50 = 4010 nM T84133 CU1SJ4 67075100 IC50 < 50 nM T84133 CC7B0L 67124352 IC50 = 13 nM T84133 C0SU4O 67257897 IC50 = 4.6 nM T84133 CF4A3M 67259323 IC50 = 0.27 nM T84133 CREP31 68014633 IC50 = 0.11 nM T84133 C9K8HT 68014634 IC50 = 0.13 nM T84133 CB04EH 68014656 IC50 = 0.22 nM T84133 CI68ER 68014850 IC50 = 170 nM T84133 CY8J3O 68181896 IC50 = 3900 nM T84133 C4ZEH9 68578314 IC50 = 1.82 nM T84133 CTJ46X 68594477 IC50 = 13.1 nM T84133 CV4X6K 68595169 IC50 = 64.5 nM T84133 C8E0XY 68596001 IC50 = 1.65 nM T84133 CJ80VI 68596013 IC50 = 13.1 nM T84133 CL2H4T 68596452 IC50 = 6.53 nM T84133 C93IHS 68596628 IC50 = 25.4 nM T84133 CDZ01B 68596639 IC50 = 3.55 nM T84133 C1CD9S 68596902 IC50 = 0.85 nM T84133 C7PCW0 68597211 IC50 = 9.11 nM T84133 CGJB21 68597401 IC50 = 11.7 nM T84133 CHK4S0 68597804 IC50 = 7.84 nM T84133 C10TGO 68598825 IC50 = 7.2 nM T84133 C8OD2Z 68853786 IC50 = 5.52 nM T84133 C3THF9 69568791 IC50 = 1.7 nM T84133 CFS2Z3 69569103 IC50 = 438 nM T84133 C15RXG 70169344 IC50 < 100 nM T84133 CBL8K3 70643905 Ki < 1000 nM T84133 CFPY14 70648748 IC50 < 500 nM T84133 COI2P3 70679302 IC50 = 0.097 nM T84133 CU9GQ0 70681149 Ki = 26 nM T84133 CIB7J9 70681150 Ki = 264 nM T84133 CNLD61 70681151 Ki = 183 nM T84133 CI9G8L 70683261 Ki = 3.8 nM T84133 COB1T8 70683262 Ki = 240 nM T84133 CAB45C 70684642 IC50 = 0.8 nM T84133 C6BN5J 70685361 Ki = 40 nM T84133 CM3OP8 70686796 IC50 = 5.13 nM T84133 CHBT91 70686797 IC50 = 3.35 nM T84133 CF6O3T 70687501 Ki = 6.6 nM T84133 CX6J1I 70695878 Ki = 12 nM T84133 CIBQ16 70810145 IC50 < 10 nM T84133 CC43LF 71074083 IC50 = 0.062 nM T84133 C4P0XT 71092344 IC50 = 810 nM T84133 C6DAG4 71092519 IC50 = 4030 nM T84133 CLU1S6 71151948 IC50 = 33 nM T84133 C7WD8I 71151969 IC50 = 0.1 nM T84133 C34XNL 71151981 IC50 = 20 nM T84133 C82AUP 71152059 IC50 = 20 nM T84133 C5VUO9 71152240 IC50 = 41 nM T84133 CY3RW6 71152297 IC50 = 29 nM T84133 C1M0EN 71153110 IC50 = 33 nM T84133 CZ4B9M 71153166 IC50 = 0.16 nM T84133 CG9C3J 71153201 IC50 = 29 nM T84133 C74BDZ 71153260 IC50 = 20 nM T84133 CYC05R 71153264 IC50 = 0.16 nM T84133 CCY3I0 71153278 IC50 = 41 nM T84133 CH51WI 71153284 IC50 = 33 nM T84133 C40HNF 71153309 IC50 = 29 nM T84133 C9GR3L 71153436 IC50 = 33 nM T84133 CZN5H8 71450204 IC50 = 0.34 nM T84133 CDJQ59 71450205 Ki < 1000 nM T84133 C8FEU2 71450432 Ki = 63 nM T84133 C4K1BM 71450433 Ki = 0.6 nM T84133 C8SXU3 71450486 Ki = 868 nM T84133 C2WZ8K 71450487 Ki = 156 nM T84133 CKAJ45 71450488 Ki = 864 nM T84133 CR5NQ6 71450591 IC50 = 0.941 nM T84133 CGD56M 71450592 IC50 = 6210 nM T84133 C06PTK 71452031 IC50 = 5.3 nM T84133 C06EHV 71452032 Ki = 2.19 nM T84133 CD50FS 71452033 IC50 = 3.3 nM T84133 CY6FZ1 71452252 Ki = 247 nM T84133 C1EFD6 71452326 Ki = 117 nM T84133 C9ADT4 71452327 Ki = 94 nM T84133 CZ1YN2 71452430 IC50 = 0.056 nM T84133 CI1M8Q 71452431 IC50 = 2.82 nM T84133 C6C2JD 71453832 IC50 = 0.89 nM T84133 CL6AT2 71454111 Ki = 186 nM T84133 CM6I9V 71454112 Ki = 500 nM T84133 C98ZEN 71454113 Ki = 4340 nM T84133 CX5D2O 71454197 IC50 = 422 nM T84133 C3EW1B 71455564 Ki < 1000 nM T84133 CR7Z6K 71455565 Ki < 1000 nM T84133 C5SH1U 71455566 IC50 = 0.61 nM T84133 CE3T7F 71455795 Ki = 1 nM T84133 C1JK6L 71455843 Ki = 522 nM T84133 CJV1G2 71455939 IC50 = 0.092 nM T84133 CVJ60C 71457356 IC50 = 0.22 nM T84133 CS54CU 71457642 Ki = 223 nM T84133 C1SWR4 71457643 Ki = 122 nM T84133 C8A9RD 71457644 Ki = 512 nM T84133 C8A4ME 71457746 IC50 = 0.075 nM T84133 CVY1U6 71459478 Ki = 4.5 nM T84133 CD3OM7 71459535 Ki = 93 nM T84133 COG41D 71459536 Ki = 98 nM T84133 C0YE2G 71459537 Ki = 422 nM T84133 C5HK3M 71459538 Ki = 121 nM T84133 C3VKH8 71459650 IC50 = 0.521 nM T84133 CHS8O5 71460995 Ki = 0.1 nM T84133 CH61LY 71461213 Ki = 3 nM T84133 CD3R9I 71461214 Ki = 8 nM T84133 C8B9OL 71461280 Ki = 7.9 nM T84133 CY9W5C 71461281 Ki = 843 nM T84133 CT6A8W 71461282 Ki = 991 nM T84133 CT2D6E 71461384 IC50 = 0.513 nM T84133 C73BXI 71462690 IC50 < 10 nM T84133 CS61KO 71520599 IC50 = 33 nM T84133 CT3IN6 71520691 IC50 = 33 nM T84133 C1D7QX 71520692 IC50 = 41 nM T84133 C1ADI4 71578082 IC50 < 100 nM T84133 C4GNJ3 71598545 IC50 > 1000 nM T84133 C9ASX2 71625031 IC50 = 991 nM T84133 CX7MY5 71680558 IC50 = 0.8 nM T84133 C68SDB 71719394 IC50 = 501.19 nM T84133 CU4RD3 71934591 IC50 = 530 nM T84133 CI6H0M 72163876 IC50 = 750 nM T84133 CMB3E6 72163877 IC50 = 660 nM T84133 CM57IJ 72163878 IC50 = 660 nM T84133 C8MIQ4 72163990 IC50 = 460 nM T84133 CUTR32 72163991 IC50 = 88 nM T84133 C7GO9N 72163992 IC50 = 87 nM T84133 CQV3Y9 72163993 IC50 = 24 nM T84133 CC2Q8Z 72164107 IC50 = 1600 nM T84133 CG9KC1 72164108 IC50 = 1600 nM T84133 CMH8P7 72164109 IC50 = 920 nM T84133 CP57OH 72164110 IC50 = 950 nM T84133 CZ0G2X 72165213 IC50 > 10000 nM T84133 C7XRY6 72190879 IC50 > 30000 nM T84133 COL24U 72193890 IC50 = 92 nM T84133 CKGQ16 72194628 IC50 = 0.15 nM T84133 CQ3GD7 72704434 Ki = 1800 nM T84133 CPIO30 72706193 IC50 > 10000 nM T84133 C1CQG9 72706253 IC50 = 1700 nM T84133 CF4W8Z 72706442 IC50 = 1600 nM T84133 C1H6MG 72724772 IC50 = 351.2 nM T84133 C98ESL 72724774 IC50 = 666.4 nM T84133 CPW50Y 72724856 IC50 = 4.85 nM T84133 C8O1UV 72724923 IC50 = 8.73 nM T84133 CWQ9G1 72724924 IC50 = 13.85 nM T84133 C9TQB6 72724925 IC50 = 0.9 nM T84133 CS4P2W 72724926 IC50 = 7.45 nM T84133 C2GUI0 72724927 IC50 = 18.48 nM T84133 C06ETS 72724928 IC50 = 5.12 nM T84133 CDOA38 72724979 IC50 = 6.88 nM T84133 CDTV07 72724982 IC50 = 157.1 nM T84133 CVC17O 72724984 IC50 = 6.73 nM T84133 CQ2S1U 72725040 IC50 = 8.96 nM T84133 CBM61I 73293715 IC50 = 403 nM T84133 CHR7D0 73334611 IC50 = 43 nM T84133 CQ9B4J 73387632 IC50 = 1590 nM T84133 CIE2C3 73387739 IC50 = 1790 nM T84133 C9ODB8 73387740 IC50 = 5 nM T84133 C5X6GJ 73387742 IC50 = 23 nM T84133 CT1E6V 73387743 IC50 = 21 nM T84133 C7D1SJ 73387744 IC50 = 83 nM T84133 CG89ET 73387745 IC50 = 25 nM T84133 CX65SQ 73387860 IC50 = 298 nM T84133 C3HSE2 73387863 IC50 = 171 nM T84133 CXOT45 73387957 IC50 = 1800 nM T84133 C74MPW 73387958 IC50 = 535 nM T84133 C3R0TC 73387959 IC50 = 11 nM T84133 CAL1N4 73387960 IC50 = 555 nM T84133 CHFG14 73425856 IC50 = 115 nM T84133 CEL2P4 73425857 IC50 = 639 nM T84133 C74TSX 73425972 IC50 = 87 nM T84133 CWX3M6 73425973 IC50 = 83 nM T84133 CEH2R6 73425974 IC50 = 20 nM T84133 CK5SA7 73425975 IC50 = 125 nM T84133 CPV3X9 73659152 Ki = 1100 nM T84133 C2FK6C 73659153 Ki = 5500 nM T84133 CVL07C 74049853 IC50 = 210 nM T84133 CT9Z7W 74049854 IC50 = 92 nM T84133 CA2R5W 74538674 IC50 < 100 nM T84133 C9JE6M 75815419 IC50 = 409 nM T84133 CSPU01 76210621 IC50 = 4.1 nM T84133 C16KIR 76283147 IC50 < 100 nM T84133 C8HPY6 76283633 IC50 = 200 nM T84133 C6ZO1T 76309994 IC50 > 1000 nM T84133 CVXP86 76309997 IC50 > 1000 nM T84133 C68NMU 76313712 IC50 > 1000 nM T84133 CGQ3L4 76313713 IC50 > 1000 nM T84133 CG4Y6I 76313715 IC50 = 309 nM T84133 CF91GV 76316930 Ki = 265 nM T84133 COR07S 76317224 IC50 = 849 nM T84133 CL03OP 76317226 IC50 > 1000 nM T84133 C8D5CS 76320933 IC50 > 1000 nM T84133 CKP16F 76320936 IC50 = 72 nM T84133 CQ8K4V 76320937 IC50 = 601 nM T84133 CNF60R 76320938 IC50 = 152 nM T84133 CTN90Q 76324596 IC50 = 16 nM T84133 CM9F4N 76324597 IC50 > 1000 nM T84133 C1WK7Z 76328150 IC50 = 99 nM T84133 C1YUL6 76328154 IC50 = 25 nM T84133 CCTF95 76328155 IC50 > 1000 nM T84133 CH0D1R 76328156 IC50 = 494 nM T84133 C41KHA 76328157 IC50 = 214 nM T84133 C2JPR1 76328158 IC50 = 166 nM T84133 CU2N9I 76328159 IC50 = 305 nM T84133 CFDQ21 76328160 IC50 = 180 nM T84133 C13ALF 76331835 IC50 = 299 nM T84133 CB76NH 76331836 IC50 = 774 nM T84133 CCY1F2 76331837 IC50 > 1000 nM T84133 CAV58P 76331838 IC50 = 89 nM T84133 CVC96N 76331839 IC50 = 208 nM T84133 C8CP3K 76903477 Ki = 0.23 nM T84133 CBTV14 77230235 Ki = 2200 nM T84133 CH90OK 80970089 Ki = 1200 nM T84133 CR95CP 80970101 Ki = 1000 nM T84133 C9E5LR 80970262 Ki = 220 nM T84133 CZ78LM 80970546 Ki = 890 nM T84133 CI43LO 80970589 Ki = 2100 nM T84133 C3NF5J 80970780 Ki = 880 nM T84133 CRE54Q 80970789 Ki = 2800 nM T84133 C3AFV8 80971037 Ki = 3600 nM T84133 CN8A4E 80971045 Ki = 1400 nM T84133 C1QLP8 80971247 Ki = 200 nM T84133 CET3Y9 80971319 Ki = 5300 nM T84133 CA92NJ 80971485 Ki = 1600 nM T84133 CX95WD 80971568 Ki = 130 nM T84133 CAUD50 80971601 Ki = 18 nM T84133 C9USK7 80971716 Ki = 51 nM T84133 C6RJP9 80972029 Ki = 6800 nM T84133 CYV42X 80972233 Ki = 37 nM T84133 CJ8S1R 80972289 Ki = 26 nM T84133 C5K6OY 80972640 Ki = 38 nM T84133 CK03GH 80978295 Ki = 4600 nM T84133 CQU45W 80978577 Ki = 1500 nM T84133 C9L8DC 81177397 Ki = 810 nM T84133 C50CVK 86291015 IC50 = 2.1 nM T84133 CV2GM7 86302601 IC50 = 24.2 nM T84133 C07WDK 86302602 IC50 = 41.5 nM T84133 CF1YH2 86302603 IC50 = 33.2 nM T84133 CM3R1U 86582302 IC50 = 20 nM T84133 C1P6DK 86582454 IC50 = 3 nM T84133 CTSL48 86688163 Ki = 12 nM T84133 C52BXE 86705377 IC50 > 10000 nM T84133 C6RB5X 86766620 Ki = 0.03 nM T84133 CTW8L6 86766622 Ki = 0.44 nM T84133 C9ZB8M 89586284 IC50 = 550 nM T84133 CZ4R0H 89586444 IC50 = 130 nM T84133 CP40LQ 89586661 IC50 = 1000 nM T84133 CZS95W 89586680 IC50 = 2400 nM T84133 CR4AW9 89593396 IC50 = 4.1 nM T84133 C1KY3L 89610300 IC50 = 0.12 nM T84133 CX9RL3 89621955 Ki = 8.5 nM T84133 CKHF70 89633452 Ki = 8.6 nM T84133 CN03MF 89763702 IC50 = 271 nM T84133 CUB2A8 90157072 Ki = 2.1 nM T84133 CF03DW 90168772 IC50 > 20000 nM T84133 CM6J9K 90168778 IC50 > 20000 nM T84133 C2BWK6 90644304 IC50 = 590 nM T84133 CG9H0I 90644305 IC50 = 6800 nM T84133 C17NSX 90644306 IC50 = 9.1 nM T84133 CC3YT0 90644307 IC50 = 8.3 nM T84133 CS3GT1 90644308 IC50 = 9.2 nM T84133 CELX01 90644309 IC50 = 28 nM T84133 CN01QJ 90644310 IC50 = 6.3 nM T84133 CTJ0H5 90644311 IC50 = 220 nM T84133 CF1IX2 90644312 IC50 = 37 nM T84133 CONS07 90644313 IC50 = 97 nM T84133 CW5HG6 90644314 IC50 = 200 nM T84133 CBMX19 90644315 IC50 = 7.3 nM T84133 C4XA2F 90644316 IC50 = 28 nM T84133 CMT94L 90644317 IC50 = 111 nM T84133 CGA67V 90644318 IC50 = 9.5 nM T84133 CCA0B1 90644319 IC50 = 1700 nM T84133 C3MRU1 90645023 IC50 = 15.1 nM T84133 CY9OX3 90645024 IC50 = 0.5 nM T84133 CWVQ98 90645025 IC50 = 5.7 nM T84133 CPZW52 90645026 IC50 = 115 nM T84133 C6GWH1 90645027 IC50 = 39.8 nM T84133 CU64KR 90645028 IC50 = 404 nM T84133 C7T4OL 90645029 IC50 = 105 nM T84133 C0A4ZG 90645030 IC50 = 36.8 nM T84133 C5J4ZG 90645031 IC50 = 51.5 nM T84133 CLQ9X5 90645032 IC50 = 21.5 nM T84133 C2DRU5 90645033 IC50 = 47.3 nM T84133 CO02RJ 90645034 IC50 = 20.7 nM T84133 CA2M6C 90645035 IC50 = 6.7 nM T84133 CX62CZ 90656262 IC50 = 123.2 nM T84133 CE7R3X 90656263 IC50 = 188.2 nM T84133 CPAX85 90656264 IC50 = 11.2 nM T84133 C01DHG 90656265 IC50 = 67.4 nM T84133 C6USP0 90656266 IC50 = 68.5 nM T84133 C3ONJ8 90656267 IC50 = 592.1 nM T84133 CQXK40 90656268 IC50 = 10.4 nM T84133 C5OGT4 90656269 IC50 = 5936.8 nM T84133 CVC4T3 90656270 IC50 = 3217.2 nM T84133 CZ6X5C 90656271 IC50 = 971.2 nM T84133 CNO3S8 90665367 IC50 = 610 nM T84133 C9MDB2 90665368 IC50 = 635 nM T84133 C1GUW7 90665369 IC50 = 3050 nM T84133 CE75WY 90665370 IC50 = 645 nM T84133 CR7ZV2 90665371 IC50 = 4250 nM T84133 C6IP3U 90665372 IC50 = 5150 nM T84133 CYU4G8 90665373 IC50 = 4600 nM T84133 CRJ8D4 90665374 IC50 = 0.4 nM T84133 C7F1IS 90665375 IC50 = 60 nM T84133 CZKD47 90665376 IC50 = 46 nM T84133 C0PWE2 90665377 IC50 = 168 nM T84133 CFB49U 90665378 IC50 = 415 nM T84133 C6NC2P 90665379 IC50 = 400 nM T84133 C2XOF1 90665380 IC50 = 635 nM T84133 C9F5QI 90668357 IC50 = 13900 nM T84133 CQR09V 90668358 IC50 = 7500 nM T84133 CXE08M 90668359 IC50 = 7400 nM T84133 C12BIU 90668360 IC50 = 10900 nM T84133 CG5HV8 90668361 IC50 = 0.24 nM T84133 C2HQ7I 90668362 IC50 = 0.36 nM T84133 C9VRW2 90668363 IC50 = 81.4 nM T84133 CDB74T 90668364 IC50 = 1.78 nM T84133 CTH48K 90668365 IC50 = 95 nM T84133 C07FTL 90668366 IC50 = 199 nM T84133 CX32TC 90668367 IC50 = 1850 nM T84133 C13GCO 90718236 IC50 = 6.3 nM T84133 C1JPD6 91844700 IC50 = 1.5 nM T84133 C60HAJ 91885643 Ki = 4.8 nM T84133 C7F6JY 92135987 IC50 = 27 nM T84133 CYQV05 92471958 IC50 = 510 nM T84133 CPO9J5 116378246 Ki = 680 nM T84133 CO3PG2 116386860 Ki = 1000 nM T84133 C4LER2 117728190 IC50 = 1.2 nM T84133 C1O7RV 117728381 IC50 = 4.4 nM T84133 C9TSE5 117728416 IC50 = 0.6 nM T84133 CH1P0N 117728473 IC50 = 7.4 nM T84133 CA46EP 117728534 IC50 = 3.2 nM T84133 C0G8NY 117728539 IC50 = 21.4 nM T84133 CWZ9R5 117728565 IC50 = 20.4 nM T84133 CIX1E9 117728795 IC50 = 2.2 nM T84133 CSCY01 117949009 IC50 > 10000 nM T84133 CYQ74R 118479645 IC50 = 1700 nM T84133 C0KPH4 118485600 IC50 > 10000 nM T84133 C43GZF 118485601 IC50 > 10000 nM T84133 C8UT1Z 118485623 IC50 > 10000 nM T84133 CC94IQ 118485651 IC50 = 59 nM T84133 CQ9X2T 118525749 IC50 = 35 nM T84133 CA9Z4N 118525753 IC50 = 96 nM T84133 COM19L 118525755 IC50 = 115 nM T84133 CCB0S9 118525772 IC50 = 67 nM T84133 C0SV3H 118525773 IC50 = 19.5 nM T84133 CG4Z8E 118525774 IC50 = 166 nM T84133 CQNY08 118525780 IC50 > 1000 nM T84133 CK3HY2 118525781 IC50 > 300 nM T84133 CGBK61 118525786 IC50 = 953 nM T84133 CYE6W5 118525795 IC50 = 135 nM T84133 C6IK4S 118525796 IC50 = 382 nM T84133 CE3UW6 118525799 IC50 = 172 nM T84133 C8OH0Y 118525801 IC50 = 146 nM T84133 CS23YQ 118525803 IC50 > 280 nM T84133 CP75JF 118525805 IC50 = 63 nM T84133 CCW37N 118525809 IC50 = 280 nM T84133 CR65SL 118525810 IC50 = 161 nM T84133 C5Y6KJ 118525812 IC50 > 1000 nM T84133 CVIU49 118525816 IC50 = 242 nM T84133 C94ZTQ 118525830 IC50 = 54 nM T84133 CM8IQ7 118525835 IC50 = 135 nM T84133 CF34RY 118525847 IC50 > 1000 nM T84133 CJX65U 118525848 IC50 = 280 nM T84133 CQ0LU1 118525854 IC50 = 52 nM T84133 C2PWK5 118534656 IC50 = 47 nM T84133 C5WDF6 118534657 IC50 = 794 nM T84133 C4H2LG 118534683 IC50 = 37 nM T84133 CR40SC 118534699 IC50 = 279 nM T84133 CVYK24 118556943 IC50 > 50000 nM T84133 CX0NV9 118658005 IC50 = 2.6 nM T84133 C01YKC 118658396 IC50 = 13 nM T84133 CSKE85 118707952 IC50 = 20.9 nM T84133 CZY9E8 118707953 IC50 = 115.7 nM T84133 C52ELD 118707954 IC50 = 102.6 nM T84133 C8WQO0 118707955 IC50 = 18.2 nM T84133 CNF3J2 118707956 IC50 = 29.2 nM T84133 CB2C3R 118707957 IC50 = 266.7 nM T84133 CO20GE 118707958 IC50 = 177.2 nM T84133 CZR3G0 118707959 IC50 = 153.1 nM T84133 CBRP26 118707960 IC50 = 8.54 nM T84133 CD67FM 118707961 IC50 = 19.1 nM T84133 C5VPF6 118707962 IC50 = 128.1 nM T84133 CZ31HQ 118707963 IC50 = 71 nM T84133 CJ0G3M 118707964 IC50 = 1.3 nM T84133 C1YX7I 118707965 IC50 = 0.3 nM T84133 C6G7DB 118707966 IC50 = 2.6 nM T84133 C0RCP5 118707967 IC50 = 135.5 nM T84133 CC5X3L 118707968 IC50 = 552.1 nM T84133 CD65SB 118708350 IC50 = 40 nM T84133 COV3E5 118708351 IC50 = 170 nM T84133 CTF9R5 118708352 IC50 = 220 nM T84133 CF7NI4 118708353 IC50 = 1300 nM T84133 CW74UJ 118708354 IC50 = 190 nM T84133 CI1Y9A 118708355 IC50 = 42 nM T84133 C9HR7F 118708356 IC50 = 40 nM T84133 CI18GD 118708357 IC50 = 55 nM T84133 CF68VD 118708358 IC50 = 480 nM T84133 CQ52CE 118708359 IC50 = 900 nM T84133 CMX51I 118708360 IC50 = 1000 nM T84133 C4I9AY 118721431 IC50 = 21000 nM T84133 CIQ2R0 118721671 IC50 = 1000 nM T84133 CY0LR7 118725353 IC50 = 18.4 nM T84133 CBAF10 118725354 IC50 = 4250 nM T84133 C5F3PM 118725355 IC50 = 14 nM T84133 C31ARB 118725356 IC50 = 1550 nM T84133 C5TL8H 118725359 IC50 = 2.86 nM T84133 C7EYI4 118725362 IC50 = 9.8 nM T84133 C5VTG0 118725363 IC50 = 350 nM T84133 C54GSD 118725364 IC50 = 518 nM T84133 C70GAC 118725365 IC50 = 79.3 nM T84133 CP9L2X 118725366 IC50 = 18.6 nM T84133 CEI6R3 118725367 IC50 = 8 nM T84133 CE49ML 118725368 IC50 = 3.73 nM T84133 C1AG7N 118725371 IC50 > 1900 nM T84133 CVDC45 121596889 IC50 = 2.4 nM T84133 C96LCR 122182051 IC50 = 1800 nM T84133 C2WP3Y 122182052 IC50 = 64 nM T84133 CZ2P0D 122182053 IC50 = 330 nM T84133 CXWB12 122185004 IC50 = 3 nM T84133 C8HFW5 122185005 IC50 = 1 nM T84133 CRJE23 122185011 IC50 = 252 nM T84133 C9T3ER 122191265 Ki = 180 nM T84133 CS5UJ1 122192111 Ki = 540 nM T84133 C4QPE7 122192112 Ki = 1300 nM T84133 C5VQJ7 122192113 Ki = 10 nM T84133 C8DIW9 122192114 Ki = 5.1 nM T84133 CMS3N6 122192115 Ki = 590 nM T84133 CS54NV 122192116 Ki = 400 nM T84133 CC3DO7 122192117 Ki = 0.047 nM T84133 CQDZ58 122192118 Ki = 0.055 nM T84133 CS6D4W 122192119 Ki = 0.11 nM T84133 C5XBU8 122192120 Ki = 0.37 nM T84133 CS70BK 122192925 Ki = 87 nM T84133 CI87VG 122192926 Ki = 280 nM T84133 COM57X 122192927 Ki = 123 nM T84133 C6Z1LU 122192928 Ki = 265 nM T84133 C41RCJ 122192929 Ki = 49 nM T84133 CM6ZQ8 122192930 Ki = 61 nM T84133 CV3MK1 122192931 Ki = 64 nM T84133 CJRB26 122192932 Ki = 171 nM T84133 C57BRI 122192933 Ki = 163 nM T84133 CW2O7J 122192934 Ki = 45 nM T84133 C5D4VJ 122192935 Ki > 1000 nM T84133 CEI01K 122192936 Ki = 39 nM T84133 CP3AS6 122192937 Ki = 15 nM T84133 C6ZHK9 122192938 Ki = 13 nM T84133 CIH0P5 122192939 Ki = 7.7 nM T84133 C20PAT 122192940 Ki = 30 nM T84133 CQD1I9 122192941 Ki = 6.3 nM T84133 CVGX87 122192953 Ki = 1 nM T84133 C0DNH8 122192954 Ki = 1.8 nM T84133 CAIJ87 122192955 Ki = 0.025 nM T84133 CN98GL 122193004 Ki = 1124 nM T84133 C1PKY7 122193005 Ki = 109 nM T84133 CS6M9C 122193679 IC50 > 100000 nM T84133 CJKO62 122193703 IC50 = 0.71 nM T84133 C9W1JO 122193704 IC50 = 0.68 nM T84133 C2MNX0 122193705 IC50 = 1.8 nM T84133 C5EHB7 122193706 IC50 = 0.32 nM T84133 C5WI6U 122193707 IC50 = 0.65 nM T84133 COT0R6 122193708 IC50 = 0.27 nM T84133 CJF36H 122193709 IC50 = 0.24 nM T84133 C0J6MS 122193710 IC50 = 0.33 nM T84133 C0XLR7 122193711 IC50 = 0.52 nM T84133 CC9I0U 122193712 IC50 = 3.07 nM T84133 CX30HD 122193713 IC50 = 0.26 nM T84133 CU5O4D 122193714 IC50 > 76 nM T84133 C07INS 122193715 IC50 = 33.5 nM T84133 C6IJH8 122193928 IC50 = 1.16 nM T84133 CNT17O 122193929 IC50 = 1.12 nM T84133 C6Q5UO 122193930 IC50 = 0.36 nM T84133 C1SWM0 122193931 IC50 = 0.47 nM T84133 C9JSX0 122193932 IC50 = 0.3 nM T84133 C6GI3B 122193933 IC50 = 0.37 nM T84133 C9PTW4 122193934 IC50 = 4.98 nM T84133 C5FKM8 122193935 IC50 = 0.76 nM T84133 C4IH7Q 122194381 IC50 = 0.23 nM T84133 CV07GU 122196327 IC50 = 2435.5 nM T84133 CT53EP 122196328 IC50 = 2740.1 nM T84133 C1MO9A 122196329 IC50 = 364.2 nM T84133 CU4N9V 122196331 IC50 = 350.9 nM T84133 CC6SY1 122196335 IC50 = 120.1 nM T84133 CUFV13 122196338 IC50 = 226.6 nM T84133 C3W6MK 122196339 IC50 = 193.6 nM T84133 C31DAM 122196340 IC50 = 1.12 nM T84133 C8K9XA 122196341 IC50 = 1.62 nM T84133 CK2A0O 122196342 IC50 = 1.11 nM T84133 C3CKT2 122196343 IC50 = 2.71 nM T84133 CPD5U0 122196344 IC50 = 1.23 nM T84133 CDWR01 122196345 IC50 = 1.41 nM T84133 CPNO72 122196346 IC50 = 5.02 nM T84133 CBHJ25 122196347 IC50 = 1.85 nM T84133 CFR30U 122196348 IC50 = 6.46 nM T84133 CE9N4M 122196392 IC50 = 1.9 nM T84133 CNA5E2 122196393 IC50 = 18.62 nM T84133 CC46NG 122196394 IC50 = 1.22 nM T84133 CCV89J 122196396 IC50 = 21.2 nM T84133 C2ZV9X 122196397 IC50 = 21.69 nM T84133 C9OG6C 122196398 IC50 = 136.6 nM T84133 CP27SM 122196399 IC50 = 926.4 nM T84133 CBN5D2 122196400 IC50 = 0.21 nM T84133 C2FMR4 122196401 IC50 = 0.33 nM T84133 CR19NH 122196402 IC50 = 0.3 nM T84133 C9I0FA 122196403 IC50 = 0.54 nM T84133 C5P8EK 122196404 IC50 = 1.73 nM T84133 C9AEK1 122196405 IC50 = 0.73 nM T84133 C8WYE5 122196406 IC50 = 11.96 nM T84133 C0M3DA 122196407 IC50 > 10000 nM T84133 C5WBC8 122196408 IC50 = 2984.5 nM T84133 CM3D6N 122196409 IC50 = 28.9 nM T84133 C2RMU9 122196410 IC50 = 41.5 nM T84133 C10LCF 122196411 IC50 = 37 nM T84133 C48VJC 122196412 IC50 = 3.3 nM T84133 CVX7U9 127029185 IC50 > 20000 nM T84133 C4UR7D 127038167 IC50 = 2.95 nM T84133 C4H2TJ 127038168 IC50 = 3.3 nM T84133 CL9JT8 127038169 IC50 = 0.12 nM T84133 CN9BH4 127038170 IC50 = 0.048 nM T84133 CC0L8Y 127038242 Ki = 8.3 nM T84133 CO2CI9 127038507 IC50 = 3.18 nM T84133 CRF5C6 127038508 IC50 = 1.57 nM T84133 CJPX60 127038509 IC50 = 0.11 nM T84133 C7X2VQ 127038510 IC50 = 26.3 nM T84133 C26EAG 127038511 IC50 = 0.41 nM T84133 CTM9E4 127038512 IC50 = 0.33 nM T84133 C6AQ2U 127038513 IC50 = 0.99 nM T84133 CJ1Z4H 127038575 Ki = 1.4 nM T84133 C6HZ8P 127038725 IC50 = 10.3 nM T84133 CV1FM0 127038868 IC50 = 0.87 nM T84133 CADU23 127038869 IC50 = 0.037 nM T84133 C50MRW 127040517 IC50 = 0.46 nM T84133 CAG7Y1 127040518 IC50 = 20.4 nM T84133 CLY63Q 127040519 IC50 = 1.69 nM T84133 C0RT1M 127040594 Ki = 3.1 nM T84133 C95LEY 127041240 IC50 = 110 nM T84133 C8NLE7 127041841 Ki = 0.006 nM T84133 C7VM1D 127041864 Ki = 1.1 nM T84133 CM7Y0H 127041887 Ki = 0.01 nM T84133 CMP85X 127041888 Ki = 0.02 nM T84133 COM5Q1 127042152 Ki = 0.02 nM T84133 C0Q6TF 127042166 Ki = 3.1 nM T84133 CNWS83 127042167 Ki = 19.1 nM T84133 CK7X3P 127042168 Ki = 4.1 nM T84133 CRL5T7 127042169 Ki = 0.4 nM T84133 CC78KF 127042170 Ki = 1.1 nM T84133 CB74PN 127042524 Ki = 15.5 nM T84133 C42NGM 127042525 Ki = 1.7 nM T84133 C9G8FY 127042526 Ki = 0.01 nM T84133 CW38DL 127042532 IC50 = 16 nM T84133 CH9PI1 127042533 IC50 = 120 nM T84133 C8GS0B 127042534 IC50 = 490 nM T84133 CC3W0Z 127042551 Ki = 20.3 nM T84133 C1QGB8 127042552 Ki = 3.6 nM T84133 C4D1OU 127042553 Ki = 54 nM T84133 CVX07H 127042560 Ki = 58 nM T84133 CXK9V3 127049326 IC50 = 2800 nM T84133 CG26VL 127049327 IC50 = 25 nM T84133 CPIX38 127049328 IC50 = 760 nM T84133 C2LGT3 129051755 IC50 = 458 nM T84133 C62CSI 129051756 IC50 = 69 nM T84133 C5RFV2 129051760 IC50 = 84 nM T84133 CH20AQ 129051764 IC50 = 40 nM T84133 CDJ2V1 129051781 IC50 = 198 nM T84133 CUE8J7 129051785 IC50 = 268 nM T84133 C7AD3Z 129051788 IC50 = 28 nM T84133 CACJ46 132489333 IC50 = 153 nM T84133 C9GNP7 132502926 IC50 = 38 nM T84133 CTH6R5 132538329 IC50 = 2 nM T84133 C2P1IU 134129996 IC50 > 100000 nM T84133 CLE03O 134130328 IC50 > 100000 nM T84133 CSN6J0 134130563 IC50 > 100000 nM T84133 C0A1CZ 134131162 IC50 > 100000 nM T84133 C5FTY2 135400457 Ki = 990000 nM T84133 CTR37Z 135408753 Ki = 910000 nM T84133 CB8YM4 135408756 Ki = 450000 nM T84133 CHDC83 135566745 IC50 > 10000 nM T84133 C9IJK1 135566935 IC50 = 6900 nM T84133 CMWA73 136042357 IC50 = 1720 nM T84133 CRP24A 136087045 IC50 = 33300 nM T84133 C7SUX4 136087050 IC50 = 3700 nM T84133 C8UF7G 136087052 IC50 > 50000 nM T84133 CGI17Y 136147441 IC50 < 500 nM T84133 C21FVA 136180322 IC50 = 2000 nM T84133 CQW7T0 136197286 IC50 > 10000 nM T84133 C8TQ7A 136217455 IC50 > 50000 nM T84133 CN8PK6 136927883 IC50 = 8.5 nM T84133 C08KZR 137007094 IC50 = 10800 nM T84133 CQK3V2 137007095 IC50 = 6620 nM T84133 CLE62X 137179301 IC50 = 117 nM T84133 C8FD1X 137243493 IC50 = 3800 nM T84133 CUM3T5 137243503 IC50 > 30000 nM T84133 C9IK5Q 137243508 IC50 = 280 nM T84133 C1JUS2 137243509 IC50 = 100 nM T84133 CI1J9K 137289913 IC50 = 3.3 nM T84133 C74KSG 137332065 IC50 = 1.7 nM T84133 C2N9VT 137348687 IC50 = 7400 nM T84133 CE1MA9 137631455 IC50 = 62 nM T84133 C0YMI5 137631826 IC50 > 10000 nM T84133 C5TDQ8 137632065 IC50 = 61 nM T84133 CQFK31 137633676 IC50 = 243 nM T84133 CGC75I 137633691 IC50 = 68 nM T84133 CAM92S 137634864 IC50 = 391 nM T84133 CIMX51 137636423 IC50 = 75 nM T84133 CAGV95 137636529 IC50 = 327 nM T84133 CX23JH 137637969 IC50 = 60 nM T84133 C1WAT7 137640957 IC50 = 130 nM T84133 CXWU26 137641682 IC50 = 107 nM T84133 C90CHG 137642556 IC50 = 168 nM T84133 C2XW5T 137643774 IC50 = 103 nM T84133 CQC5R0 137644374 IC50 = 116 nM T84133 C1Y7TO 137644422 IC50 = 447 nM T84133 C7MAO1 137645978 IC50 = 113 nM T84133 C24PNB 137650825 IC50 = 336 nM T84133 C2HS7D 137651999 IC50 = 56 nM T84133 C5XH7C 137653888 IC50 = 529 nM T84133 C6C7XH 137655649 IC50 = 452 nM T84133 C7LPA8 137655726 IC50 = 119 nM T84133 CP7Q5D 137656637 IC50 = 76 nM T84133 C7OH1C 137658687 IC50 = 518 nM T84133 CRD93N 137659470 IC50 = 168 nM T84133 CKEY52 137660104 IC50 = 258 nM T84133 C6KYD7 137700754 IC50 = 7310 nM T84133 CM3UF7 137700779 IC50 = 0.44 nM T84133 CPTE92 138319693 IC50 = 46 nM T84133 C2QLX3 138393292 IC50 = 920 nM T84133 CF6B8H 138857395 IC50 = 294 nM T84133 C72GWA 138857396 IC50 = 2.9 nM T84133 C7AHV4 138857397 IC50 = 28 nM T84133 CMW20N 141737696 IC50 > 4000 nM T84133 C8HEG7 141737705 IC50 > 3000 nM T84133 CC64PE 145949747 IC50 = 884 nM T84133 CU9YW0 145950008 IC50 = 381 nM T84133 C0F5PO 145950382 IC50 > 1000 nM T84133 C7Z5JP 145952479 IC50 = 280 nM T84133 CNIV78 145952823 IC50 = 770 nM T84133 C70YLA 145953136 IC50 = 76 nM T84133 C0C6FG 145954733 IC50 = 107 nM T84133 CQN9P3 145954872 IC50 = 163 nM T84133 C2KN1T 145955431 IC50 > 5000 nM T84133 C36IDE 145957514 IC50 > 1000 nM T84133 CW0JY3 145957704 IC50 > 1000 nM T84133 CH7VB3 145957961 IC50 = 145 nM T84133 CMTR43 145958975 IC50 = 268 nM T84133 CYZR45 145959927 IC50 = 315 nM T84133 C37PRT 145967337 IC50 < 100 nM T84133 CF25ZG 145967398 IC50 = 100 nM T84133 CAR1K5 145972948 IC50 = 581 nM T84133 CC7HN2 145974174 IC50 > 100000 nM T84133 CD5P0M 145974821 IC50 > 280 nM T84133 CK1BR0 145978345 IC50 > 100000 nM T84133 CHJ79V 145997874 IC50 > 10000 nM T84133 CY1R9G 147132320 IC50 = 403 nM T84133 C2AHD9 148588374 IC50 = 0.87 nM T84133 CD38ZO 155513157 IC50 = 44 nM T84133 C83XTD 155514176 IC50 = 5.2 nM T84133 C48WQL 155514804 IC50 = 441 nM T84133 C14BPA 155515110 IC50 = 2083 nM T84133 CQAY86 155517940 IC50 = 0.3 nM T84133 C49UIO 155519155 IC50 = 20 nM T84133 CE2MO6 155519440 IC50 = 47 nM T84133 CZM1V6 155520000 IC50 = 138 nM T84133 CF4B7U 155520076 IC50 = 75 nM T84133 CT7K4A 155520403 IC50 = 69 nM T84133 CI6AT8 155520893 IC50 = 44 nM T84133 CUA1X6 155521116 IC50 = 287 nM T84133 CL8CU6 155521936 IC50 > 200000 nM T84133 CWS0T8 155522940 IC50 = 510 nM T84133 CPZ9C5 155523000 IC50 = 1219 nM T84133 CPIE52 155524256 IC50 = 1476 nM T84133 C4J8EY 155524365 IC50 = 0.061 nM T84133 CGY0B7 155526339 IC50 = 292 nM T84133 CX7D8K 155526808 IC50 > 10000 nM T84133 CMPE29 155527485 IC50 = 8.4 nM T84133 C7ERC3 155527562 IC50 = 1 nM T84133 C4PE7I 155528020 IC50 = 78 nM T84133 C47UVA 155528950 IC50 = 105 nM T84133 CVG71O 155529178 IC50 = 105 nM T84133 CQPC31 155530033 IC50 = 110 nM T84133 C74GVU 155530078 IC50 = 279 nM T84133 CZAP29 155530397 IC50 = 416 nM T84133 CT85RG 155530589 IC50 > 200000 nM T84133 CUS48O 155530649 IC50 = 23 nM T84133 C73WIM 155530814 IC50 = 74 nM T84133 C7SI1U 155531139 IC50 = 320 nM T84133 CICH53 155532871 IC50 = 135 nM T84133 C6POE9 155533544 IC50 = 52 nM T84133 C3ZE6S 155535535 IC50 = 12 nM T84133 C8J0FO 155535672 IC50 = 23 nM T84133 CRA93Z 155539143 IC50 = 182 nM T84133 C84NIR 155540213 IC50 = 13.8 nM T84133 C6KEO7 155542008 IC50 = 88 nM T84133 C5QCM6 155545348 IC50 = 4.7 nM T84133 CAK63Q 155545457 IC50 = 0.76 nM T84133 CAD3C9 155545902 IC50 = 123 nM T84133 C7PQ5B 155546577 IC50 = 200 nM T84133 CAD6U2 155546988 IC50 = 2.1 nM T84133 CO3W9J 155549412 IC50 = 23 nM T84133 CXK67C 155551574 IC50 = 440 nM T84133 CZV45E 155554965 IC50 = 275 nM T84133 C2OYG0 155555420 IC50 = 10 nM T84133 CP18OF 155555969 IC50 > 1000 nM T84133 CJE59L 155558096 IC50 = 120 nM T84133 C2DA1W 155561694 IC50 > 500000 nM T84133 CC8I1S 155566153 IC50 = 1920 nM T84133 C95JGC 155566500 IC50 = 62 nM T84133 CT2SY1 155568004 IC50 = 7.6 nM T84133 CQ2R0W 155568588 IC50 > 500000 nM T84133 CYAZ51 66678448 Ki = 0.95 nM T84133 CF8Z7Y 69932178 IC50 = 0.06 nM T84133 D06NIT 135564899 IC50 > 1000 nM T84133 D09RKU 46239428 Ki = 5 nM T84133 D0V4WB 149790 IC50 > 16000 nM T84133 D0VB2W 21501 Ki = 560000 nM T65019 D00MDP 466151 IC50 = 0.3 nM T65019 D0Q8CS 60937 IC50 = 30500 nM T65019 D0VM2L 68740 IC50 = 12600 nM T65019 D05VZE 119031 IC50 = 1.82 nM T65019 D0A4RF 657061 IC50 = 22.91 nM T65019 D0MW3H 9824350 IC50 = 23 nM T65019 D0U2BH 65064 IC50 = 6800 nM T65019 D0G1LL 74221072 IC50 = 50000 nM T65019 D0N6ZA 74221131 IC50 > 100000 nM T65019 D0UM5R 74221070 IC50 = 15000 nM T65019 D01DVX 9847838 IC50 = 499 nM T65019 D03BOZ 3342298 IC50 = 1.1 nM T65019 D0E5GY 9904965 IC50 = 1.9 nM T65019 D0N8NK 11641563 IC50 = 2220 nM T65019 D0P8YC 5362422 IC50 = 2.9 nM T65019 D0T9HG 132519 IC50 = 0.41 nM T65019 C4U7SY 401129 IC50 = 12500 nM T65019 C4D7TS 448002 IC50 = 13 nM T65019 CC54LQ 450256 IC50 > 100000 nM T65019 CG1I8P 467296 IC50 = 15600 nM T65019 CTPW02 467297 IC50 = 3700 nM T65019 CS4O7K 685005 IC50 > 500000 nM T65019 CP1Q6R 703233 IC50 = 55000 nM T65019 C9IFC6 1348435 IC50 = 21000 nM T65019 CN9C8D 2140735 IC50 = 310000 nM T65019 CN6E3U 2366268 IC50 = 7500 nM T65019 CY3TD6 3348132 Ki = 105 nM T65019 C3EI6T 4085085 IC50 = 51000 nM T65019 CBN96T 4358655 IC50 > 100000 nM T65019 CC5O4E 4369384 IC50 = 6500 nM T65019 CZS0G5 5276565 IC50 > 100000 nM T65019 C3JN0F 5277465 IC50 = 33500 nM T65019 CRJK67 5277481 IC50 > 100000 nM T65019 CYF7S5 5277490 IC50 > 100000 nM T65019 CP7BG0 6852146 IC50 = 2200 nM T65019 CN5L2B 6852147 IC50 = 79 nM T65019 CP2XK7 6882342 IC50 = 150000 nM T65019 C76RCQ 9801569 IC50 = 963 nM T65019 CIXD67 9802768 IC50 = 8 nM T65019 CQ46XD 9804842 IC50 = 1700 nM T65019 CTK6J8 9808181 IC50 = 66900 nM T65019 C9RQM7 9808674 IC50 = 7.4 nM T65019 C6KJ9W 9822461 IC50 = 47 nM T65019 C6IX7G 9822926 IC50 = 5.6 nM T65019 CE9AL3 9847113 IC50 = 10.6 nM T65019 C4IEK0 9850035 IC50 = 108 nM T65019 CI8Z0R 9866250 IC50 = 7.4 nM T65019 CJS23I 9868333 Ki > 5290 nM T65019 CLQ29X 9869597 IC50 = 1710 nM T65019 CHU9I8 9871883 IC50 = 4.6 nM T65019 C0ZT7A 9883002 Ki = 37 nM T65019 C3ZG6O 9887870 IC50 = 240 nM T65019 CD79UJ 9890632 IC50 > 100000 nM T65019 CH69LT 9892815 IC50 = 13 nM T65019 CSIB97 9896504 IC50 > 100000 nM T65019 C4YGT6 9928325 IC50 = 56 nM T65019 C03GVA 9932290 Ki = 240 nM T65019 CDXR37 9933197 IC50 = 64 nM T65019 C65ION 9935032 IC50 = 500 nM T65019 CG38KL 9936728 Ki = 140 nM T65019 CQY54S 9952396 IC50 = 88 nM T65019 C9X0YR 9954867 IC50 > 10000 nM T65019 C3Q2UJ 9956686 IC50 = 200 nM T65019 CI5TW9 9956699 IC50 = 20100 nM T65019 CC4WG3 9957228 Ki > 300000 nM T65019 CN76XI 9957653 IC50 = 7 nM T65019 C9DRB7 9966028 IC50 = 2900 nM T65019 CUA65C 9982414 IC50 = 150 nM T65019 CR7T3J 10009978 Ki > 2000 nM T65019 CW2MK1 10043732 Ki = 210 nM T65019 C7O8HD 10044261 IC50 = 2.5 nM T65019 C7CT4E 10045150 IC50 = 1.9 nM T65019 CCF5Z4 10047585 IC50 = 2.08 nM T65019 CB9S7N 10101618 IC50 = 19 ug.mL-1 T65019 C0G7IY 10114318 Ki = 200 nM T65019 CVK61T 10116047 IC50 = 11 nM T65019 C78JHL 10116107 Ki = 390 nM T65019 C7A8MI 10120093 IC50 = 3.7 nM T65019 C7KR3Y 10136680 Ki = 150 nM T65019 CNU93J 10136924 Ki = 440 nM T65019 C1CDF2 10136925 Ki = 330 nM T65019 CJ9EX4 10138303 Ki = 250 nM T65019 CO6PS3 10162900 Ki = 180 nM T65019 CR5H6E 10163627 Ki > 5290 nM T65019 CCX3T6 10183064 Ki = 3070 nM T65019 CK0P3F 10186536 Ki > 5290 nM T65019 CE1LI3 10204303 Ki = 180 nM T65019 CQFP69 10206106 Ki = 340 nM T65019 C4K1MJ 10208262 Ki > 5290 nM T65019 CV5X8A 10224181 IC50 > 30000 nM T65019 CGKU70 10224396 Ki = 240 nM T65019 C2MES9 10271604 Ki > 100000 nM T65019 CGP97S 10274748 Ki = 100 nM T65019 C3IG0K 10280852 IC50 = 4.1 nM T65019 CDU36Y 10296475 Ki = 590 nM T65019 C48IRP 10296785 Ki = 50 nM T65019 CY08WJ 10322755 Ki = 163 nM T65019 C7UZA4 10340758 IC50 = 8.5 nM T65019 C6WZ4F 10367355 IC50 = 34 nM T65019 CFKA79 10395015 Ki = 2000 nM T65019 C5WV1N 10439082 Ki > 2000 nM T65019 C8M9FE 10462640 Ki = 160000 nM T65019 CNQZ36 10483139 Ki > 10000 nM T65019 C9C5EL 10521197 IC50 = 2.3 nM T65019 C21VZS 10573362 IC50 = 17.6 nM T65019 C3R2SO 10580533 Ki = 105 nM T65019 C6FWC1 10808125 IC50 = 13 nM T65019 C2A0IX 10833840 IC50 = 105 nM T65019 C9WPH7 11016072 Ki = 740 nM T65019 CBE68H 11016073 Ki = 330 nM T65019 CR4V2D 11101785 Ki = 380 nM T65019 CD1Q0L 11157488 IC50 = 20000 nM T65019 CEL1F0 11248884 IC50 = 5600 nM T65019 CO7T3M 11261246 IC50 = 7.7 nM T65019 CP17ID 11284983 IC50 = 15000 nM T65019 C1IW7N 11292680 IC50 = 9.8 nM T65019 C8C5AV 11294179 Ki > 10000 nM T65019 CLH50U 11318841 IC50 = 15800 nM T65019 CJ5SU9 11328354 Ki > 300000 nM T65019 C0XR3B 11330861 IC50 = 50118.72 nM T65019 CQH57S 11342435 IC50 = 5000 nM T65019 CU04HF 11419551 IC50 = 13900 nM T65019 COS67B 11456566 IC50 = 30000 nM T65019 C96DRO 11466734 IC50 = 5450 nM T65019 C7QF0G 11467517 IC50 = 11200 nM T65019 CWS35C 11510523 IC50 = 20700 nM T65019 C5VUM2 11517085 Ki = 140 nM T65019 CQ9E6J 11519157 IC50 = 4735 nM T65019 C5MO0U 11526826 IC50 = 1641 nM T65019 C9Y6LH 11533683 IC50 = 19700 nM T65019 CCW1B8 11569185 IC50 = 3121 nM T65019 CW5A4S 11569716 IC50 = 1305 nM T65019 CHV2G1 11575995 Ki > 10000000 nM T65019 CL9K7T 11583525 IC50 = 1950 nM T65019 CTQ87G 11599024 IC50 = 13000 nM T65019 C8IWM1 11605689 IC50 = 553 nM T65019 C0VCJ8 11613810 IC50 = 220 nM T65019 CCBS59 11634234 IC50 = 3642 nM T65019 CNY92D 11640694 Ki > 40000 nM T65019 C1U3EX 11656290 IC50 > 10000 nM T65019 C28WNK 11682752 Ki = 900 nM T65019 CRF7V9 11691964 IC50 = 915 nM T65019 C3U6ZR 11697504 Ki = 11000 nM T65019 C2BJ3X 11716217 Ki = 31910 nM T65019 CCD93H 11730086 Ki = 110 nM T65019 CO8QT0 11753905 Ki = 2800 nM T65019 C4XR5G 11963536 IC50 = 24000 nM T65019 C02BWA 11967143 Ki > 2000 nM T65019 CB80OT 12000718 IC50 > 20000 nM T65019 C43PJZ 12000720 IC50 > 20000 nM T65019 C0K8ZX 12404978 IC50 > 500000 nM T65019 CQTX49 13738810 IC50 > 100000 nM T65019 C8TH1O 14177156 IC50 > 500000 nM T65019 C3N1KV 15629940 IC50 > 100000 nM T65019 CB3A4Z 15941413 Ki = 215 nM T65019 CA40FE 15941550 Ki = 90 nM T65019 CM3D1L 15941553 Ki = 680 nM T65019 CQ0ZL7 15941677 Ki = 145 nM T65019 C6F9WV 15941679 Ki = 360 nM T65019 C7C1HI 15941680 Ki = 240 nM T65019 C6R1LD 15985818 IC50 = 582 nM T65019 CL7KX3 16040152 IC50 = 0.57 ug.mL-1 T65019 CTZ3R1 16040153 IC50 = 3.2 ug.mL-1 T65019 CS46XU 16126723 IC50 = 14 nM T65019 C91EXN 16655061 IC50 = 14800 nM T65019 CQS0F5 16719301 IC50 > 10000 nM T65019 C75XDI 16730519 IC50 > 5000 nM T65019 C50AEZ 18616892 IC50 > 10000 nM T65019 CIEH93 19382975 IC50 = 69000 nM T65019 CK8MP3 20620240 Ki > 10000 nM T65019 CPC4G6 20620273 Ki > 10000 nM T65019 C2E3CY 20620614 Ki > 10000 nM T65019 CC7BF2 20636126 IC50 = 616.6 nM T65019 C6A1QE 20636128 IC50 = 645.65 nM T65019 C4JPZ3 20636129 IC50 = 9332.54 nM T65019 CAU28R 20636149 IC50 = 8709.64 nM T65019 CXS53V 20636183 IC50 = 36.31 nM T65019 C18RXS 20735191 IC50 = 9.5 nM T65019 C4I1OM 20735209 IC50 = 10000 nM T65019 CIC4S9 22004232 IC50 = 71 nM T65019 CZT05X 22484417 Ki > 10000 nM T65019 CZT64B 22484431 Ki > 10000 nM T65019 CAM10T 22485252 IC50 = 24 nM T65019 CBJS34 22485260 IC50 = 3.63 nM T65019 C9MU7N 22485263 IC50 > 10000 nM T65019 CEGJ03 22485276 IC50 = 3486 nM T65019 C7VB8G 22485289 IC50 = 0.73 nM T65019 CNB02I 22485291 IC50 = 10.5 nM T65019 CAY3N6 22485292 IC50 = 159 nM T65019 C94OCJ 22485302 IC50 = 6.8 nM T65019 C3YL5X 22485311 IC50 = 53.9 nM T65019 CWA03L 22485327 IC50 = 3.1 nM T65019 C6JRW5 22485340 IC50 = 13.3 nM T65019 C5JZF1 22485344 IC50 = 47 nM T65019 CI7MY5 22485346 IC50 = 20 nM T65019 CI1YL7 22485347 IC50 = 4 nM T65019 C25OBD 22485356 IC50 = 4.5 nM T65019 C7I0EW 22485367 IC50 = 1.71 nM T65019 CL64TJ 22485368 IC50 = 100.5 nM T65019 CT4GF9 22485381 IC50 > 10000 nM T65019 C27NDB 22485386 IC50 = 160 nM T65019 CTJ9I3 22485392 IC50 = 25.8 nM T65019 C3MG9P 22485396 IC50 = 83 nM T65019 CZY10U 22485408 IC50 = 58.6 nM T65019 C89AGT 22485413 IC50 = 14.9 nM T65019 C8GHU9 22485432 IC50 = 49.4 nM T65019 C9BT5F 22626996 IC50 = 784 nM T65019 C2Q4XK 22707806 IC50 = 9 nM T65019 CIYA45 22985930 IC50 = 53.3 nM T65019 CX32YK 23513795 IC50 = 257 nM T65019 C6IZ1S 23513821 IC50 = 2080 nM T65019 CPNM93 23513825 IC50 = 489 nM T65019 CML90Q 23513831 IC50 = 889 nM T65019 C4R2AJ 23625454 IC50 = 4891 nM T65019 C4R2DA 23645953 Ki > 300000 nM T65019 CWN3I4 23645959 Ki > 300000 nM T65019 CL24JR 23655078 IC50 = 3290 nM T65019 CBI81H 23672150 IC50 = 15 ug.mL-1 T65019 C7KF1N 23729138 IC50 = 2000 nM T65019 CG3J2L 24768528 IC50 = 2370 nM T65019 C5M3YW 24799779 Ki = 2400000 nM T65019 CE29HI 24860424 IC50 = 4320 nM T65019 CT10JE 24860425 IC50 = 3619 nM T65019 CRC98J 24860426 IC50 = 1000 nM T65019 C8MKR0 24860427 IC50 = 7047 nM T65019 CNR3U7 24866945 IC50 = 20000 nM T65019 C4UEM5 24871537 Ki > 50000 nM T65019 CP2L5B 24871655 Ki > 50000 nM T65019 C4SP3O 24936157 IC50 = 3.9 nM T65019 CAQ9Z1 25022681 Ki > 5290 nM T65019 CU6M9K 25060725 IC50 = 3100 nM T65019 CF7X2P 25060975 IC50 = 10500 nM T65019 CVR52U 25066764 IC50 = 1100 nM T65019 CD2KA4 25102047 IC50 = 94 nM T65019 CRW96X 25102048 IC50 = 95 nM T65019 CQ3O9P 25102050 IC50 = 41 nM T65019 CSHA26 25102051 IC50 = 81 nM T65019 C7ADO2 25102197 IC50 = 25 nM T65019 CA5DJ4 25138228 Ki = 4072000 nM T65019 C1TNQ3 25141117 Ki = 1900 nM T65019 CR35QP 25144971 IC50 > 10000 nM T65019 C0Y5BC 25145683 IC50 > 2500 nM T65019 CB7V8Y 25147773 IC50 = 0.32 nM T65019 C3KF1V 25178145 IC50 = 2.1 nM T65019 C8PMK7 25178356 IC50 > 100000 nM T65019 CG5Y2R 25178357 IC50 = 306 nM T65019 C4PZY6 25180866 IC50 = 353 nM T65019 CEP9Q2 25180867 IC50 = 3.9 nM T65019 C9HZG2 25181078 IC50 = 33900 nM T65019 CMYP34 25181079 IC50 = 8950 nM T65019 C7U1YC 25181080 IC50 = 89.8 nM T65019 C85HLG 25181081 IC50 = 260 nM T65019 CHR2P1 25183768 Ki > 25000 nM T65019 C6AR8O 42623563 IC50 > 100000 nM T65019 CX0VP7 42623564 IC50 = 52000 nM T65019 C0H3RD 42627769 IC50 = 6820 nM T65019 CPO1Z3 44123600 IC50 = 91 nM T65019 C25ELB 44143088 IC50 = 72443.6 nM T65019 CL0M7R 44143089 IC50 = 426579.52 nM T65019 C9QDC0 44143091 IC50 = 134896.29 nM T65019 CT80ED 44219901 IC50 = 3400 nM T65019 C94JVY 44219902 IC50 = 2800 nM T65019 C7J6GH 44219903 IC50 = 590 nM T65019 C9J7WL 44219904 IC50 = 11000 nM T65019 CRQ71E 44219905 IC50 = 6500 nM T65019 C4Z0ID 44219906 IC50 = 2400 nM T65019 CRNA25 44220092 IC50 > 1000 nM T65019 C9T5ZF 44220093 IC50 = 14000 nM T65019 CV38TE 44222825 IC50 = 5500 nM T65019 CJI73R 44222826 IC50 = 320 nM T65019 CGQ30N 44222827 IC50 = 1000 nM T65019 CCI64J 44224245 IC50 = 2250 nM T65019 CLRT69 44247751 IC50 = 33 nM T65019 CG7X5F 44272675 IC50 = 19.3 nM T65019 CEHR24 44272853 IC50 = 72 nM T65019 CJU31O 44321285 Ki = 73 nM T65019 C41VFA 44321286 Ki = 40 nM T65019 C5S2ZU 44321484 Ki = 545 nM T65019 CLQ23M 44321485 Ki = 192 nM T65019 CHF76Q 44321540 Ki = 45 nM T65019 CVOL49 44321593 Ki = 63 nM T65019 CB97GK 44321601 Ki = 90 nM T65019 CT0O7Y 44321602 Ki = 1282 nM T65019 CU62BP 44321746 Ki = 41 nM T65019 CQU2K9 44321782 Ki = 217 nM T65019 CV8T3N 44321783 Ki = 60 nM T65019 CIBO50 44321801 Ki = 22 nM T65019 C4E8GU 44321802 Ki = 125 nM T65019 CYDN18 44321803 Ki = 53 nM T65019 C7Z4DQ 44321887 Ki = 32 nM T65019 CFJ20T 44321932 Ki = 41 nM T65019 C9O0VB 44321965 Ki = 2960 nM T65019 C2E3RF 44321966 Ki = 271 nM T65019 CW9S1N 44321967 Ki = 1350 nM T65019 C1FI3O 44321975 Ki = 26 nM T65019 CLB8J6 44321976 Ki = 270 nM T65019 CR0KN1 44322209 Ki = 2030 nM T65019 C5LE1P 44322210 Ki = 92 nM T65019 CQ7AW8 44322211 Ki = 550 nM T65019 CJY2O7 44322214 Ki = 660 nM T65019 CR9GI0 44322215 Ki = 580 nM T65019 CMLA39 44329018 IC50 = 10 nM T65019 C1IE0S 44330147 IC50 > 100000 nM T65019 CE3MT4 44341611 Ki = 30100 nM T65019 CJTZ45 44341652 Ki = 30000 nM T65019 CTQ6P4 44344631 IC50 = 66900 nM T65019 CBH9I5 44344658 IC50 = 930 nM T65019 CGQ92A 44364037 IC50 = 62 nM T65019 C36YLM 44364111 IC50 = 835 nM T65019 CN4T7Q 44364119 IC50 = 521 nM T65019 CH4TE7 44364121 IC50 = 39 nM T65019 CPE91Y 44364122 IC50 = 52 nM T65019 CG2X0C 44364224 IC50 = 1102 nM T65019 C1F8XN 44364249 IC50 = 68 nM T65019 CWM47H 44364250 IC50 = 867 nM T65019 C0W5TL 44364251 IC50 = 20820 nM T65019 C3TPO7 44364266 IC50 = 4613 nM T65019 CJ2B8F 44364280 IC50 = 3108 nM T65019 CV0T6G 44383797 Ki = 9000 nM T65019 C9NIT7 44383842 Ki = 35000 nM T65019 C13LRY 44383990 Ki = 11000 nM T65019 CDQV80 44384020 Ki = 29000 nM T65019 CA2L3U 44384021 Ki = 15000 nM T65019 CT1MN8 44384090 Ki = 180000 nM T65019 CILQ34 44384272 Ki = 9500 nM T65019 CIJ61R 44384273 Ki = 14000 nM T65019 CL59ZH 44384393 Ki = 33000 nM T65019 C0RXF4 44384804 Ki = 1400 nM T65019 CE5RJ0 44385333 Ki = 20000 nM T65019 C5R4EW 44389591 IC50 > 300 nM T65019 C3EZ0W 44391336 IC50 = 50 nM T65019 C1E5JC 44391341 IC50 = 3 nM T65019 CT5Y1X 44391344 IC50 = 620 nM T65019 CP0QS3 44391345 IC50 = 27 nM T65019 CR0Y3D 44391350 IC50 = 16 nM T65019 CMTB94 44391351 IC50 = 70 nM T65019 CC7QW9 44391352 IC50 = 220 nM T65019 C0FC5U 44391354 IC50 = 11 nM T65019 CMS1Z6 44391356 IC50 = 18 nM T65019 CA3NH7 44391357 IC50 = 650 nM T65019 CTK65L 44391360 IC50 = 230 nM T65019 C0S4YB 44391365 IC50 = 120 nM T65019 CN4GJ0 44391366 IC50 = 9300 nM T65019 CKL09S 44391376 IC50 = 510 nM T65019 CVTB31 44391377 IC50 > 30000 nM T65019 C3BPI8 44391397 IC50 = 23 nM T65019 CW90KP 44391398 IC50 = 1400 nM T65019 C1N8KB 44391410 IC50 = 340 nM T65019 CB0HI5 44391419 IC50 = 23 nM T65019 C5XSH0 44391424 IC50 = 8700 nM T65019 CFH41S 44391425 IC50 = 18 nM T65019 C49DCW 44391434 IC50 = 60 nM T65019 CZ89IE 44391435 IC50 = 200 nM T65019 CP0AU9 44391440 IC50 = 260 nM T65019 C9BMR7 44391444 IC50 = 19 nM T65019 CR4U6B 44391445 IC50 = 75 nM T65019 CH59GY 44391449 IC50 = 150 nM T65019 CU7N6G 44391450 IC50 = 150 nM T65019 CD5TX3 44391460 IC50 = 6700 nM T65019 CCK39J 44391461 IC50 = 22 nM T65019 C3V1PB 44391476 IC50 = 36 nM T65019 C37DHM 44391486 IC50 = 220 nM T65019 CZB81D 44395506 IC50 = 83 nM T65019 CAU5R4 44397021 IC50 = 6600 nM T65019 CSO92L 44397377 IC50 = 1.5 nM T65019 CZ45GV 44397680 IC50 = 10900 nM T65019 C91POV 44402021 IC50 = 1490 nM T65019 CYCJ78 44402280 IC50 = 116 nM T65019 CY6WL5 44404502 IC50 = 12302.69 nM T65019 CWGQ46 44404503 IC50 = 15000 nM T65019 CLXM58 44404504 IC50 = 30000 nM T65019 C30DKN 44404553 IC50 = 4 nM T65019 CIC60V 44406452 IC50 = 3000 nM T65019 CVM7Y3 44413975 IC50 = 725 nM T65019 C4X0GA 44413977 IC50 = 488 nM T65019 CH01EO 44413978 IC50 = 891 nM T65019 CQ8HK9 44413979 IC50 = 4850 nM T65019 CBT0P2 44413982 IC50 = 583 nM T65019 CIJ39D 44413983 IC50 = 97 nM T65019 C9BA0V 44413987 IC50 = 1515 nM T65019 CE3WP0 44413991 IC50 = 5910 nM T65019 CDUI73 44413992 IC50 = 12 nM T65019 CH2X6W 44413997 IC50 = 1380 nM T65019 CHN85S 44414002 IC50 = 1900 nM T65019 C2OJ4B 44414029 IC50 = 2740 nM T65019 CT5PC9 44422672 IC50 = 11 nM T65019 CS9D5U 44422720 IC50 = 11 nM T65019 CNWM05 44422723 IC50 = 130 nM T65019 C58LAY 44422724 IC50 = 32 nM T65019 CDQU41 44422736 IC50 = 180 nM T65019 CVUB56 44422737 IC50 = 75 nM T65019 CB8G2W 44422743 IC50 = 26 nM T65019 CFX42T 44422744 IC50 = 6000 nM T65019 C9EL7F 44422749 IC50 = 40000 nM T65019 CO24JF 44423677 IC50 = 9500 nM T65019 C45WZX 44426073 IC50 = 1.6 ug.mL-1 T65019 CWU7G8 44434565 IC50 = 2660 nM T65019 CF9HU5 44434566 IC50 = 53100 nM T65019 CV3M6F 44434578 IC50 = 2490 nM T65019 CB9P0C 44442303 IC50 = 3440 nM T65019 C7HO0Y 44442304 IC50 = 7440 nM T65019 CAR3S2 44442305 IC50 = 3410 nM T65019 CZK0A9 44442306 IC50 = 4160 nM T65019 C71MCV 44442307 IC50 = 5640 nM T65019 CN70HO 44442308 IC50 = 1460 nM T65019 CVE5P0 44442309 IC50 = 5650 nM T65019 C3PT7N 44442310 IC50 = 1860 nM T65019 CGS18B 44442311 IC50 = 3020 nM T65019 CCFV76 44442313 IC50 = 5640 nM T65019 C4HYM6 44442314 IC50 = 1250 nM T65019 CZ2PE6 44442315 IC50 = 1650 nM T65019 C3I7RG 44442317 IC50 = 1020 nM T65019 CD9Y4Q 44445920 IC50 = 60.26 nM T65019 CL67QM 44445921 IC50 = 15.85 nM T65019 C6IS7V 44445922 IC50 = 18.2 nM T65019 CBL68C 44445923 IC50 = 120.23 nM T65019 C5Z4RH 44445924 IC50 = 512.86 nM T65019 CU9O6F 44445925 IC50 = 22.91 nM T65019 CWI9S1 44445926 IC50 = 50.12 nM T65019 CA6CX0 44445927 IC50 = 70.79 nM T65019 CQC1S9 44445928 IC50 = 19.05 nM T65019 C5GU9H 44445929 IC50 = 151.36 nM T65019 CX09NS 44445930 IC50 = 6760.83 nM T65019 C3XD8C 44445931 IC50 = 218.78 nM T65019 C6CPY9 44445932 IC50 = 199.53 nM T65019 CG0Z7I 44478924 IC50 = 4000 nM T65019 CFO27Y 44478926 IC50 = 200 nM T65019 CBZJ29 44478927 IC50 = 710 nM T65019 CRJ24K 44479197 IC50 = 360 nM T65019 CGOH82 44479198 IC50 = 8100 nM T65019 CLV56M 44479199 IC50 = 740 nM T65019 CY92OQ 44479458 IC50 = 120000 nM T65019 CH1QG9 44479459 IC50 = 1300 nM T65019 CB1NT7 44479460 IC50 = 940 nM T65019 C0JQ9L 44479699 IC50 = 860 nM T65019 C0DN1Q 44479700 IC50 = 77000 nM T65019 CTG24W 44479702 IC50 = 18000 nM T65019 CGZ49M 44479703 IC50 = 2100 nM T65019 CAK94X 44563337 IC50 = 1690 nM T65019 CSH4K3 44563364 IC50 > 10000 nM T65019 CAF95R 44563365 IC50 = 1000 nM T65019 CO4FQ1 44563366 IC50 > 10000 nM T65019 C6WA3X 44563401 IC50 > 10000 nM T65019 CX5L7N 44563402 IC50 = 2600 nM T65019 CJ8V4U 44563403 IC50 = 190 nM T65019 CN2BM4 44563404 IC50 = 3100 nM T65019 C3KCV6 44563405 IC50 = 3700 nM T65019 CI0R5M 44563465 IC50 = 1500 nM T65019 C5IQ9Z 44563466 IC50 = 1100 nM T65019 C6ZEW9 44563467 IC50 = 9700 nM T65019 CZ2EL1 44563468 IC50 = 5100 nM T65019 CDV6R7 44563469 IC50 = 730 nM T65019 CJ2BU5 44563487 IC50 = 10000 nM T65019 C1UXP6 44563490 IC50 = 105 nM T65019 CZ0W1A 44563491 IC50 = 3784 nM T65019 C4BD0N 44563493 IC50 = 1237 nM T65019 CNP6M7 44563494 IC50 = 2800 nM T65019 CWD32S 44580184 IC50 = 24000 nM T65019 CQ4ZR1 44580422 IC50 = 930 nM T65019 CK68GT 44580539 Ki = 67.6 nM T65019 CXIY57 44580801 Ki > 10000000 nM T65019 C0OA8Y 44580802 Ki > 10000000 nM T65019 CNC4D7 44581071 Ki > 10000000 nM T65019 CDF48U 44581111 Ki > 10000000 nM T65019 CTW7F2 44601281 IC50 = 41 nM T65019 C19LWR 44634267 IC50 = 23 nM T65019 CACH13 45269631 IC50 = 530 nM T65019 C36HRP 45377138 IC50 > 22000 nM T65019 C6B7ZY 45377564 IC50 > 500000 nM T65019 C5HAR6 45377565 IC50 > 22000 nM T65019 CKR0Q8 45377703 IC50 = 11000 nM T65019 C3SQL2 45378250 IC50 = 300 nM T65019 CQE49A 45378251 IC50 = 0.9 nM T65019 CO4AC6 45378252 IC50 = 210 nM T65019 C42FPG 45378253 IC50 = 4.3 nM T65019 CI82BN 45378254 IC50 = 29 nM T65019 C6MY2W 45380188 IC50 = 240 nM T65019 C9P0DG 45380189 IC50 = 16 nM T65019 CRY0E8 45380190 IC50 = 34 nM T65019 C0MPH3 45380191 IC50 = 1800 nM T65019 CMPE63 45482676 IC50 = 10000 nM T65019 CSX5I9 46175170 IC50 = 3.4 nM T65019 C56WVI 46184724 Ki > 30000 nM T65019 CDQ1K4 46224842 IC50 = 2.8 ug.mL-1 T65019 CH0Z1E 46844314 Ki = 1196 nM T65019 C20BTY 46856241 Ki = 1100 nM T65019 C5L8GF 46871738 IC50 > 10000 nM T65019 CR1KF7 46871739 IC50 = 5000 nM T65019 C8Q6YR 46871740 IC50 > 10000 nM T65019 C58YSM 46871741 IC50 > 10000 nM T65019 C4VEZ3 46882679 IC50 = 19 nM T65019 CR3QW7 46891107 IC50 > 10000 nM T65019 C5MK3A 46891108 IC50 > 10000 nM T65019 CQ5E1H 46891109 IC50 > 10000 nM T65019 C91LGI 46891170 IC50 = 2860 nM T65019 CZPM12 46891172 IC50 > 10000 nM T65019 C2V6MW 46891173 IC50 = 8220 nM T65019 C8S7QX 46891209 IC50 > 10000 nM T65019 C5Y0MN 46891255 IC50 > 10000 nM T65019 CJ16SE 46891256 IC50 > 10000 nM T65019 CNXU57 46891313 IC50 > 10000 nM T65019 CVK0E5 46891356 IC50 > 10000 nM T65019 C89RPO 46891357 IC50 > 10000 nM T65019 CVB6K4 46891358 IC50 > 10000 nM T65019 C0S9WB 46919610 Ki = 120 nM T65019 CE3H7I 46938726 IC50 = 1.33 nM T65019 C9T0HR 46938727 IC50 = 24.9 nM T65019 C0YR7M 46938728 IC50 = 7.1 nM T65019 C2TE8J 47162079 IC50 > 500000 nM T65019 CUD7O0 50941549 IC50 > 10000 nM T65019 CX8N4D 50990920 IC50 = 430 nM T65019 CXF4V3 50990921 IC50 > 8900 nM T65019 CAS94N 51346773 Ki = 480 nM T65019 CP65WT 51346774 Ki = 11000 nM T65019 C5OIA2 51346775 Ki = 32000 nM T65019 CU2SX3 51355576 Ki > 10000 nM T65019 CQM4E7 52936345 IC50 = 6.4 ug.mL-1 T65019 C1Y5UN 52951473 IC50 = 2200 nM T65019 CXYJ67 52951474 IC50 = 1400 nM T65019 C8J9EM 52951589 IC50 = 610 nM T65019 CEAS70 52951591 IC50 = 1100 nM T65019 C4DG1F 52951593 IC50 = 240 nM T65019 C6XJ3V 52951596 IC50 = 4900 nM T65019 C9U3AF 52951710 IC50 = 280 nM T65019 C4M1CA 52951712 IC50 = 4300 nM T65019 C76LDY 52951967 IC50 = 1.3 nM T65019 CYKS94 52951968 IC50 = 1.2 nM T65019 CE0FP3 52951969 IC50 = 100 nM T65019 CL69OM 52951970 IC50 = 100 nM T65019 CMPB74 52951971 IC50 = 17 nM T65019 CZ1TN8 52951972 IC50 = 8 nM T65019 CK08OB 52952074 IC50 = 25 nM T65019 C46AYR 52952075 IC50 = 450 nM T65019 CR32ZW 52952076 IC50 = 300 nM T65019 CJ9O3S 52952077 IC50 = 2100 nM T65019 C3N9TF 52952078 IC50 = 2500 nM T65019 C5S1IG 52952079 IC50 > 10000 nM T65019 CKV9R0 52952178 IC50 = 2900 nM T65019 CV0R6Y 52952179 IC50 = 6100 nM T65019 CE4Q7F 52952273 IC50 > 10000 nM T65019 CMA69V 52952274 IC50 = 6000 nM T65019 C7KB5W 52952275 IC50 = 5400 nM T65019 CRO0X4 52952276 IC50 = 1100 nM T65019 CSJ05E 52952277 IC50 = 1400 nM T65019 C29UJB 52952388 IC50 = 420 nM T65019 C3H5ID 52952389 IC50 = 270 nM T65019 CSX69R 52952390 IC50 = 2300 nM T65019 CB36KP 52952492 IC50 = 900 nM T65019 C67OEU 52952493 IC50 = 2100 nM T65019 CV1I0A 52952597 IC50 = 140 nM T65019 CGI87K 52952598 IC50 = 98 nM T65019 CXWI18 52952599 IC50 > 10000 nM T65019 C46VHP 52952600 IC50 = 2100 nM T65019 CH3G6R 52952601 IC50 > 10000 nM T65019 CC0Y3M 52952602 IC50 > 10000 nM T65019 CLA96C 53232689 Ki > 10000 nM T65019 C3BGW0 53233015 Ki > 40000 nM T65019 CMQZ70 53242178 IC50 > 23000 nM T65019 CRI92N 53311230 IC50 > 10000 nM T65019 C74CKF 53318123 Ki = 790 nM T65019 CB09MA 53318910 IC50 = 7.6 nM T65019 C47DIU 53318911 IC50 = 160 nM T65019 CC6DR2 53318912 IC50 = 4200 nM T65019 C7V1NC 53320225 IC50 = 4600 nM T65019 CVH2B7 53320226 IC50 > 18000 nM T65019 CO8QK2 53320227 IC50 > 3600 nM T65019 CNS3F2 53321542 IC50 = 3600 nM T65019 C1N2BX 53322876 IC50 = 390 nM T65019 CSYW40 53322877 IC50 > 8000 nM T65019 CGUC59 53322878 IC50 = 2600 nM T65019 C3QHA6 53322879 IC50 > 3700 nM T65019 CI3WL5 53323418 Ki = 20000 nM T65019 C1VNZ9 53324198 IC50 = 180 nM T65019 C0H7FQ 53324260 IC50 = 29000 nM T65019 CU7YG9 53325497 IC50 = 900 nM T65019 C4G1HK 53325498 IC50 = 18000 nM T65019 CO5L1I 53325499 IC50 = 17000 nM T65019 CZA03W 53326760 IC50 = 360 nM T65019 CM53CG 53326761 IC50 = 40000 nM T65019 CWR6T4 53326860 IC50 = 56 nM T65019 CPY02U 53327890 IC50 = 2100 nM T65019 CPGE80 53327891 IC50 = 1700 nM T65019 CLJ4G2 53328858 IC50 = 700 nM T65019 C4G3QL 53328859 IC50 = 1600 nM T65019 CX1TW0 53328860 IC50 = 112 nM T65019 C0ZX5G 53329215 IC50 = 6600 nM T65019 CSU52A 53329216 IC50 = 23000 nM T65019 CNB63X 53361475 IC50 = 9330 nM T65019 C6Y2EV 53374826 IC50 > 100000 nM T65019 CX3DU4 53378973 Ki = 12000 nM T65019 CTD1H9 53378974 Ki = 19000 nM T65019 C1IFJ8 53957122 IC50 > 500000 nM T65019 CSUW40 54352406 IC50 = 135 nM T65019 C3M8GZ 54580051 IC50 > 100000 nM T65019 CL0WM9 54580052 IC50 > 10000 nM T65019 CK26XF 54580053 IC50 > 10000 nM T65019 CS1LM9 54580054 IC50 = 226 nM T65019 C3LF0P 54580544 Ki > 10000 nM T65019 C6R3MZ 54580973 Ki > 50000 nM T65019 C8PE1G 54581030 IC50 = 2900 nM T65019 CVO09J 54581546 Ki > 10000 nM T65019 CWKA42 54582019 Ki > 50000 nM T65019 CVK72M 54582073 IC50 = 3100 nM T65019 CBK18O 54582074 IC50 > 10000 nM T65019 CP2F1B 54582075 IC50 > 10000 nM T65019 CZNU23 54582076 IC50 > 10000 nM T65019 C0U5HZ 54582077 IC50 > 7500 nM T65019 CSTG96 54582078 IC50 = 1400 nM T65019 C8SG9Y 54582079 IC50 > 10000 nM T65019 CZI6S3 54582080 IC50 > 7200 nM T65019 CD09BZ 54582543 Ki > 10000 nM T65019 CH6Q2Z 54583016 IC50 > 10000 nM T65019 C3V9LQ 54583017 IC50 = 1200 nM T65019 CT80KQ 54583018 IC50 > 770 nM T65019 CPT4L5 54583019 IC50 > 10000 nM T65019 CK52YD 54583511 Ki > 10000 nM T65019 CBEV27 54584024 IC50 > 10000 nM T65019 CM87DP 54584025 IC50 = 2900 nM T65019 C28GKQ 54585927 IC50 > 10000 nM T65019 CAZ76E 54586892 IC50 > 10000 nM T65019 CM0OQ3 54586893 IC50 > 10000 nM T65019 CK1NS7 54586894 IC50 > 10000 nM T65019 CMC4Y1 54586895 IC50 > 10000 nM T65019 C2MKX5 54586896 IC50 = 8000 nM T65019 CU91QP 54586897 IC50 > 10000 nM T65019 CI08RQ 54586898 IC50 > 10000 nM T65019 C6PRI4 54586899 IC50 > 10000 nM T65019 CG37UX 54587429 Ki > 10000 nM T65019 CL9SC3 54587769 Ki = 16400 nM T65019 C13FSJ 54669762 Ki = 210 nM T65019 CHS01Z 54669766 Ki = 28900 nM T65019 C7E9SG 54757202 Ki = 260 nM T65019 CKJ9S1 56835167 IC50 = 83 nM T65019 C21CLZ 56835168 IC50 = 3900 nM T65019 C0L2TS 56835169 IC50 = 2200 nM T65019 CKEV19 56850269 IC50 > 500000 nM T65019 C13DBR 56850270 IC50 > 500000 nM T65019 C05CTJ 56850271 IC50 = 51000 nM T65019 CX8QD5 56850272 IC50 = 225000 nM T65019 C1I9RE 56850407 IC50 > 500000 nM T65019 CVJ90W 56850408 IC50 = 15000 nM T65019 CPI5G0 56850409 IC50 = 41000 nM T65019 CHE2I1 57345500 Ki > 50000 nM T65019 C63TFM 57345501 Ki > 50000 nM T65019 C8KT2F 57345502 Ki > 50000 nM T65019 C0KPD8 57384084 IC50 = 160 nM T65019 CV67JB 57384091 IC50 = 3800 nM T65019 CN2H9K 57391204 IC50 > 10000 nM T65019 CR8MW2 57391205 IC50 > 10000 nM T65019 CNQ9B2 57392969 IC50 > 100000 nM T65019 CTYP14 57392972 IC50 > 10000 nM T65019 C5VB0U 57392973 IC50 > 10000 nM T65019 CMQL31 57392974 IC50 > 10000 nM T65019 C39OHF 57392975 IC50 > 10000 nM T65019 CDCW73 57394678 IC50 > 500000 nM T65019 CNOH63 57394711 IC50 > 10000 nM T65019 CD50CO 57399918 IC50 > 10000 nM T65019 CK68EY 57403424 IC50 > 10000 nM T65019 C0G2VY 57403564 IC50 = 5 nM T65019 CWH7V8 57561293 IC50 = 239 nM T65019 CY1N3J 57792153 IC50 = 1067 nM T65019 CCKD80 58307579 Ki = 62 nM T65019 C8ITK7 59794408 IC50 = 9501 nM T65019 CAT67H 59910477 IC50 = 1389 nM T65019 CH76IU 70684364 Ki = 190 nM T65019 CZ63AG 70684365 Ki = 280 nM T65019 C0GKT8 70685026 IC50 = 420 nM T65019 CTUN76 70688632 Ki = 580 nM T65019 C3LCG0 70688633 Ki = 140 nM T65019 C1A0VU 70692840 Ki = 5080 nM T65019 C6P3XM 70693710 Ki > 50000 nM T65019 CL7JF9 71304794 IC50 = 2200 nM T65019 CSY30R 71304795 IC50 = 250 nM T65019 CNPG78 71304796 IC50 = 1830 nM T65019 CMW3O0 71451330 Ki = 30000 nM T65019 CDZ3P2 71453147 Ki = 5100 nM T65019 C9QS6E 71456659 Ki = 105 nM T65019 CH5J4A 71602247 IC50 = 1600 nM T65019 CH53IU 71602248 IC50 = 4800 nM T65019 C97EWQ 71602249 IC50 = 4600 nM T65019 CNX9B1 71652215 IC50 = 82 nM T65019 C7RZN9 71652216 IC50 = 310 nM T65019 C0NTU7 71652382 IC50 = 24 nM T65019 CA5XS1 71652383 IC50 = 3700 nM T65019 C7DMX5 71680709 Ki = 11 nM T65019 CFPM82 71680710 Ki = 21 nM T65019 C9ZOM7 71680866 Ki = 6.6 nM T65019 CQ68LT 71680868 Ki = 85000 nM T65019 CV3X1T 71682766 Ki = 410 nM T65019 C5EAO8 71682767 Ki = 68 nM T65019 C80EYX 71682913 Ki = 3000 nM T65019 CIBD03 71682914 Ki = 1200 nM T65019 C41BYG 71682915 Ki = 18 nM T65019 C93XEI 71682916 Ki = 10 nM T65019 CQ29PJ 71682917 Ki > 200000 nM T65019 CFWN65 71683062 Ki > 25000 nM T65019 C3E2VT 71814508 IC50 = 671 nM T65019 CR2L4T 71814509 IC50 = 62 nM T65019 CF21LN 71814684 IC50 = 116 nM T65019 C4YM2D 71814685 IC50 = 915 nM T65019 CZW1P6 71814686 IC50 = 1080 nM T65019 C5SI6C 71814687 IC50 = 7731 nM T65019 CDXZ25 71814688 IC50 = 764 nM T65019 CIZ7K1 71814857 IC50 = 450 nM T65019 C4W9TJ 71814858 IC50 = 1282 nM T65019 CJH9K3 71814859 IC50 = 6897 nM T65019 CCMN52 71814860 IC50 = 4090 nM T65019 CZ9BC5 71814861 IC50 = 350 nM T65019 CU28BE 71815035 IC50 = 1858 nM T65019 C7HN2J 71815036 IC50 = 53584 nM T65019 CLWC38 72193198 IC50 = 100 nM T65019 CX4G0R 72204928 IC50 > 100000 nM T65019 CG9C6U 72204929 IC50 = 3900 nM T65019 C5A6XZ 72204930 IC50 = 26000 nM T65019 C0XZK4 72204931 IC50 > 100000 nM T65019 CM8Y7X 72204932 IC50 > 100000 nM T65019 C6RY4X 72204933 IC50 > 100000 nM T65019 C4N5AB 72204934 IC50 > 100000 nM T65019 C3H2FZ 72205111 IC50 > 100000 nM T65019 CQ0VX7 72205112 IC50 > 100000 nM T65019 CQ7TI1 72205113 IC50 = 43000 nM T65019 CPAW52 72205114 IC50 = 76000 nM T65019 C2LD3J 72205115 IC50 = 49500 nM T65019 CE4J8F 72711063 Ki = 1900 nM T65019 CW2RF1 72711064 Ki = 2100 nM T65019 CC5T1Q 72711065 Ki = 2500 nM T65019 C7YFC8 72711513 IC50 = 21400 nM T65019 CTM4P2 72713638 IC50 = 630 nM T65019 C0N2JX 72713639 IC50 = 590 nM T65019 CF4K8Y 72713862 IC50 = 7200 nM T65019 C3R6JO 72713863 IC50 = 72000 nM T65019 CW9D3V 72713864 IC50 = 1600 nM T65019 CQ6FH3 72713865 IC50 = 940 nM T65019 C4FYB0 72713866 IC50 = 2900 nM T65019 CH6SI1 72713867 IC50 = 1700 nM T65019 CS21QM 72713868 IC50 = 120000 nM T65019 CB56AP 72714081 IC50 = 890 nM T65019 C1CK0E 72714082 IC50 = 113000 nM T65019 CP5Q8W 72714083 IC50 = 123000 nM T65019 CRUH64 72714085 IC50 = 170000 nM T65019 COQZ24 72714091 Ki = 2400 nM T65019 CC0ZX4 72714092 Ki = 2700 nM T65019 CW8I1S 72714093 Ki = 2800 nM T65019 C3Q9LV 72714094 Ki = 3000 nM T65019 CZFY06 72714322 IC50 = 104000 nM T65019 CDY70J 72714323 IC50 = 68000 nM T65019 CD56BA 72714324 IC50 = 19500 nM T65019 CE51LQ 72714333 Ki = 17000 nM T65019 CK6D5F 72714334 Ki = 27000 nM T65019 C9FL7V 72714339 Ki = 2600 nM T65019 C38IDL 73345835 Ki = 7 nM T65019 CCV78D 73346037 IC50 > 99999 nM T65019 CK0TR7 73349097 IC50 = 98907 nM T65019 C57LGA 73349098 IC50 = 33882 nM T65019 C8ROG3 73350414 Ki = 6.2 nM T65019 CF7AB2 73350415 Ki = 70 nM T65019 C2PFM4 73351930 Ki = 310 nM T65019 CA2X8C 73352170 IC50 > 100000 nM T65019 CNW2C8 73353628 IC50 > 10000 nM T65019 CYV0L6 73353629 IC50 > 10000 nM T65019 CI09CY 73354906 Ki = 6 nM T65019 C1HLC9 73355128 IC50 > 10000 nM T65019 C06BPT 73355130 IC50 = 2817 nM T65019 C4SXT6 73356696 IC50 > 10000 nM T65019 CA5T7P 73603957 IC50 = 8000 nM T65019 C8VN1R 74221194 IC50 = 3900 nM T65019 C5LB0U 78426619 IC50 > 100000 nM T65019 CET6N8 78426757 IC50 > 100000 nM T65019 CUE7G4 86287514 IC50 > 50000 nM T65019 CGQ8F3 86287515 IC50 = 8700 nM T65019 CJ37XE 86287516 IC50 = 37000 nM T65019 COV8I9 86291010 IC50 = 1085 nM T65019 CO2FL5 90137145 IC50 = 3400 nM T65019 CRT54C 101910871 IC50 = 86000 nM T65019 C1J3CK 117094707 IC50 = 100000 nM T65019 C5ZS4E 118722686 IC50 = 3500 nM T65019 CIZB24 118722687 IC50 = 18000 nM T65019 C5C0ZX 118722688 IC50 = 8600 nM T65019 CLCW15 122181996 IC50 > 100000 nM T65019 CT7D4F 122181997 IC50 > 100000 nM T65019 CZO32N 122181998 IC50 > 100000 nM T65019 C40DWG 122181999 IC50 > 100000 nM T65019 CJFS09 122190237 IC50 = 5500 nM T65019 CT03QA 127026888 IC50 = 50000 nM T65019 C89QOM 127043503 IC50 = 6311 nM T65019 C9E5YJ 127043505 IC50 = 1614 nM T65019 CW1Q3D 127043506 IC50 = 5424 nM T65019 C1C7WB 127044036 IC50 = 6875 nM T65019 CPF6U7 127044139 IC50 = 7783 nM T65019 CT9B0Q 127044462 IC50 = 4639 nM T65019 CL3X1A 127044649 IC50 = 8805 nM T65019 C8RZ7T 127044651 IC50 = 1000 nM T65019 C3I4PT 127044652 IC50 = 807 nM T65019 CDX86T 127044818 IC50 = 2407 nM T65019 C56OJV 127044819 IC50 = 427 nM T65019 CYA92R 130282633 IC50 = 6500 nM T65019 CO3QE2 130282636 IC50 = 4400 nM T65019 C4MB7N 132285189 Ki = 120 nM T65019 CTN42D 132941363 IC50 = 78000 nM T65019 CT3G2U 134133460 IC50 = 23 nM T65019 C8VLY0 134144890 IC50 = 850 nM T65019 C93ZLI 134145328 IC50 = 900 nM T65019 CHV2U1 135438561 IC50 > 10000 nM T65019 C4FVJ1 135487604 IC50 > 100000 nM T65019 C1MOD4 135567320 IC50 > 10000 nM T65019 CA5JR6 136054481 IC50 > 10000 nM T65019 CV47JN 136054485 IC50 = 8900 nM T65019 CZ48WO 136054487 IC50 > 10000 nM T65019 C8FGT0 136054495 IC50 = 3700 nM T65019 CG70BZ 136054516 IC50 = 5.4 nM T65019 CSM57W 136054520 IC50 = 550 nM T65019 CJG54U 136219136 IC50 > 30000 nM T65019 C3CAV5 136219141 IC50 = 24000 nM T65019 CPB07Z 136241630 IC50 = 4300 nM T65019 CIEW62 136380958 IC50 = 140 nM T65019 C9HS7J 137287436 IC50 = 3.8 nM T65019 C4UMY5 137636781 IC50 > 5000 nM T65019 CR8H9Z 137644167 IC50 > 5000 nM T65019 CB8M6U 137646865 IC50 > 5000 nM T65019 CK4LE6 137647628 IC50 > 10000 nM T65019 CS80YI 137652598 IC50 = 1600 nM T65019 CZB75K 137657128 IC50 > 10000 nM T65019 CC3I9B 137660260 IC50 > 10000 nM T65019 C4H0EM 137661370 IC50 > 5000 nM T65019 CZ8H6N 137661550 IC50 = 7600 nM T65019 C37HMX 137701229 Ki = 53 nM T65019 C1Q2BP 145949247 IC50 > 5000 nM T65019 C6TD4M 145949288 IC50 > 5000 nM T65019 CN9RD6 145949408 IC50 > 5000 nM T65019 C5FWA2 145949488 IC50 > 5000 nM T65019 CZS1N7 145949693 IC50 > 5000 nM T65019 C6IPV3 145949783 IC50 = 435800 nM T65019 CYG32L 145950058 IC50 > 5000 nM T65019 C72LGN 145950074 IC50 > 500000 nM T65019 CU53BP 145950331 IC50 > 5000 nM T65019 CY8C4A 145950332 IC50 > 5000 nM T65019 CAJ25P 145951291 IC50 > 5000 nM T65019 C3EF7N 145952515 IC50 > 5000 nM T65019 CW1GS2 145952760 IC50 > 5000 nM T65019 CFN1R7 145952843 IC50 > 5000 nM T65019 CM6T2O 145953417 IC50 > 5000 nM T65019 C6FYK8 145953609 IC50 > 5000 nM T65019 CV80WQ 145954107 IC50 > 5000 nM T65019 C16VNH 145954604 IC50 > 5000 nM T65019 CQF50V 145954863 IC50 > 5000 nM T65019 C2HAG8 145955226 IC50 = 309300 nM T65019 C8QW9G 145955776 IC50 > 5000 nM T65019 CH0ZO5 145955778 IC50 > 5000 nM T65019 CFDZ62 145955866 IC50 > 5000 nM T65019 CVZ5U7 145955868 IC50 > 5000 nM T65019 C8TPR1 145956198 IC50 > 5000 nM T65019 COR96H 145956298 IC50 = 301100 nM T65019 CR8U7Y 145956318 IC50 > 5000 nM T65019 C7R3FE 145956426 IC50 = 76300 nM T65019 C4S8LU 145956764 IC50 > 5000 nM T65019 CUS0Y9 145957234 IC50 > 5000 nM T65019 CUO69Q 145957392 IC50 > 5000 nM T65019 CX94UK 145957493 IC50 > 5000 nM T65019 C6MHN7 145957508 IC50 > 5000 nM T65019 CQ15DP 145957734 IC50 = 111350 nM T65019 C5K7PV 145958060 IC50 > 5000 nM T65019 CBE02W 145958354 IC50 > 5000 nM T65019 CQL4O0 145959327 IC50 > 5000 nM T65019 CG03OE 145959777 IC50 = 109000 nM T65019 CIQ9J2 145960035 IC50 = 87100 nM T65019 CUAT97 145960347 IC50 > 5000 nM T65019 CZ76WA 145962290 IC50 > 5000 nM T65019 C27MTZ 145962695 IC50 > 5000 nM T65019 CRY63E 145963538 IC50 > 5000 nM T65019 CVCL61 145963739 IC50 > 5000 nM T65019 CFE1A5 145971595 Ki = 119 nM T65019 CWY5X0 145971805 IC50 = 4000 nM T65019 C1FPG2 145972660 IC50 > 5000 nM T65019 CJF73O 145973630 IC50 > 5000 nM T65019 CX7M9L 145976456 IC50 > 5000 nM T65019 C1KPL5 145976497 IC50 = 40000 nM T65019 CPD1B0 145977213 IC50 > 5000 nM T65019 C9Z5DX 145978402 IC50 > 5000 nM T65019 CZ25LW 155512044 IC50 = 57000 nM T65019 C98HMU 155515777 IC50 = 80 nM T65019 CRY3D4 155541376 IC50 = 14 nM T65019 CH40UO 155562232 IC50 = 7 nM T65019 CP9YX2 155567218 IC50 = 26000 nM T65019 C8D5VK 155567855 IC50 = 34000 nM T65019 CLT4Y6 10138589 Ki = 290 nM T65019 D01UNE 44580457 Ki = 160 nM T65019 D03AMR 9849669 Ki = 1200 nM T65019 D04GOO 10111838 IC50 > 100000 nM T65019 D04PAW 16216218 IC50 = 70000 nM T65019 D04VPH 45376872 IC50 = 8300 nM T65019 D05THD 44478925 IC50 = 8300 nM T65019 D06EHW 11625778 IC50 = 772 nM T65019 D06HSC 136117931 IC50 = 80000 nM T65019 D07DRT 46175162 Ki = 4 nM T65019 D07GEL 10344307 Ki = 94 nM T65019 D07MJD 44479701 IC50 = 5400 nM T65019 D09USO 5277466 IC50 = 40000 nM T65019 D09ZOA 25049753 IC50 = 70 nM T65019 D0A0FY 44479457 IC50 = 25000 nM T65019 D0A4TC 446504 IC50 = 7.5 nM T65019 D0B3UN 44580458 Ki = 140 nM T65019 D0G3YZ 11391583 IC50 = 36600 nM T65019 D0H6CK 10160968 Ki > 5290 nM T65019 D0L4EO 11609208 IC50 = 30600 nM T65019 D0L6ND 10089677 IC50 = 0.2 ug.mL-1 T65019 D0NP8A 10370504 IC50 = 1900 nM T65019 D0NV9C 22004198 IC50 = 360 nM T65019 D0P2TS 9818682 IC50 > 10000 nM T65019 D0Q4TA 10044321 IC50 = 2300 nM T65019 D0S9OL 10155934 IC50 = 1300 nM T65019 D0W2UK 6914621 Ki = 15872 nM T65019 D0XK7G 10445302 IC50 = 210 nM T65019 D0Y5IQ 44255320 IC50 = 5000 nM T39919 D00BCP 2727 IC50 = 133000 nM T39919 D00BLL 9849808 IC50 = 133000 nM T39919 D00DKK 5282379 IC50 = 133000 nM T39919 D00FGO 460612 IC50 = 133000 nM T39919 D00IBN 54676228 IC50 = 133000 nM T39919 D00JAU 3749 IC50 = 83200 nM T39919 D00KVO 2082 IC50 = 133000 nM T39919 D00MIN 657298 IC50 = 133000 nM T39919 D00NKB 5546 IC50 = 133000 nM T39919 D00USF 5533 IC50 = 133000 nM T39919 D00WAM 3647 IC50 = 133000 nM T39919 D00WUF 5486971 IC50 = 133000 nM T39919 D00XUN 23894 IC50 = 133000 nM T39919 D00YZA 5453 IC50 = 133000 nM T39919 D01AJY 2284 IC50 = 133000 nM T39919 D01AZG 5073 IC50 = 133000 nM T39919 D01DBQ 452548 IC50 = 34900 nM T39919 D01GBY 124087 IC50 = 133000 nM T39919 D01KKQ 135400182 IC50 = 133000 nM T39919 D01MDT 5487 IC50 = 133000 nM T39919 D01MUR 68844 IC50 = 133000 nM T39919 D01OXI 2578 IC50 = 133000 nM T39919 D01STB 5362129 IC50 = 133000 nM T39919 D01UTL 2995 IC50 = 133000 nM T39919 D01UXC 2249 IC50 = 133000 nM T39919 D01XNB 4594 IC50 = 133000 nM T39919 D01XYJ 35370 IC50 = 133000 nM T39919 D01ZII 2726 IC50 = 133000 nM T39919 D01ZSO 4235 IC50 = 133000 nM T39919 D02DGU 444795 IC50 = 133000 nM T39919 D02DPA 2756 IC50 = 133000 nM T39919 D02FEM 5284447 IC50 = 133000 nM T39919 D02HED 4748 IC50 = 133000 nM T39919 D02LCR 5467 IC50 = 133000 nM T39919 D02NTO 5510 IC50 = 133000 nM T39919 D02STN 132971 IC50 = 133000 nM T39919 D02TLO 3690 IC50 = 133000 nM T39919 D02YIZ 12560 IC50 = 133000 nM T39919 D02ZTJ 5339 IC50 = 1500 nM T39919 D03CQE 5379 IC50 = 133000 nM T39919 D03DDR 3034034 IC50 = 133000 nM T39919 D03ELL 2159 IC50 = 133000 nM T39919 D03HJK 447043 IC50 = 133000 nM T39919 D03JSJ 446596 IC50 = 133000 nM T39919 D03KOZ 1549120 IC50 = 6500 nM T39919 D03KQF 4011 IC50 = 133000 nM T39919 D03KZM 216237 IC50 = 133000 nM T39919 D03NHW 4583 IC50 = 133000 nM T39919 D03QWT 73303 IC50 = 133000 nM T39919 D03RTS 2662 IC50 = 133000 nM T39919 D03TVW 54120 IC50 = 133000 nM T39919 D03TYI 9433 IC50 = 131000 nM T39919 D03VPC 2754 IC50 = 16600 nM T39919 D03XOC 656583 IC50 = 133000 nM T39919 D03YLZ 27200 IC50 = 133000 nM T39919 D04AAW 60613 IC50 = 133000 nM T39919 D04ASH 657180 IC50 = 133000 nM T39919 D04EGX 54746 IC50 = 133000 nM T39919 D04FBR 5281078 IC50 = 83000 nM T39919 D04ITO 6436173 IC50 = 30200 nM T39919 D04JCN 47811 IC50 = 133000 nM T39919 D04JEE 4946 IC50 = 133000 nM T39919 D04JPJ 3950 IC50 = 133000 nM T39919 D04KYY 135401907 IC50 = 133000 nM T39919 D04MSM 2554 IC50 = 133000 nM T39919 D04NXQ 51081 IC50 = 133000 nM T39919 D04OSE 4485 IC50 = 16600 nM T39919 D04RGA 5282415 IC50 = 7100 nM T39919 D04VMT 5253 IC50 = 133000 nM T39919 D04WFD 4543 IC50 = 133000 nM T39919 D04XGT 31593 IC50 = 133000 nM T39919 D04YMH 151166 IC50 = 133000 nM T39919 D04ZTY 444020 IC50 = 133000 nM T39919 D05AFX 4450 IC50 = 133000 nM T39919 D05ARP 135398740 IC50 = 133000 nM T39919 D05DVP 5717 IC50 = 12100 nM T39919 D05EAM 4735 IC50 = 133000 nM T39919 D05FTJ 4044 IC50 = 133000 nM T39919 D05GJW 20279 IC50 = 133000 nM T39919 D05HPI 16134395 IC50 = 133000 nM T39919 D05HSC 6000 IC50 = 9600 nM T39919 D05LEO 3385 IC50 = 133000 nM T39919 D05LKP 5215 IC50 = 133000 nM T39919 D05LYX 3488 IC50 = 10500 nM T39919 D05MFA 135398741 IC50 = 133000 nM T39919 D05MQK 110635 IC50 = 133000 nM T39919 D05OFX 219078 IC50 = 133000 nM T39919 D05QDC 5284513 IC50 = 49000 nM T39919 D05UVD 33624 IC50 = 133000 nM T39919 D05VIL 5284594 IC50 = 133000 nM T39919 D05VIX 3463 IC50 = 133000 nM T39919 D05VLS 5090 IC50 = 133000 nM T39919 D05ZGQ 5281070 IC50 = 133000 nM T39919 D05ZIK 4205 IC50 = 133000 nM T39919 D06ABF 3957 IC50 = 133000 nM T39919 D06BEP 2712 IC50 = 133000 nM T39919 D06CTE 57469 IC50 = 133000 nM T39919 D06FDR 135398739 IC50 = 133000 nM T39919 D06GAM 3357 IC50 = 133000 nM T39919 D06GDY 43815 IC50 = 133000 nM T39919 D06HBQ 91610 IC50 = 6300 nM T39919 D06JPB 5280793 IC50 = 133000 nM T39919 D06NXY 5991 IC50 = 133000 nM T39919 D06OIV 5505 IC50 = 133000 nM T39919 D06OMK 445643 IC50 = 133000 nM T39919 D06OVY 5362065 IC50 = 133000 nM T39919 D06PSS 5311309 IC50 = 133000 nM T39919 D06TNL 3278 IC50 = 133000 nM T39919 D06UDG 60846 IC50 = 133000 nM T39919 D06WTZ 53232 IC50 = 133000 nM T39919 D06XAE 1712095 IC50 = 24500 nM T39919 D06XMU 6013 IC50 = 133000 nM T39919 D06YYD 9578005 IC50 = 133000 nM T39919 D06ZII 969472 IC50 = 133000 nM T39919 D06ZUK 3696 IC50 = 133000 nM T39919 D07ABV 468595 IC50 = 133000 nM T39919 D07BCT 36294 IC50 = 133000 nM T39919 D07CWD 3657 IC50 = 133000 nM T39919 D07DJQ 10219 IC50 = 133000 nM T39919 D07GRH 2749 IC50 = 133000 nM T39919 D07HGR 5362119 IC50 = 133000 nM T39919 D07HVY 64139 IC50 = 133000 nM T39919 D07IEF 2391 IC50 = 133000 nM T39919 D07IPB 454216 IC50 = 36800 nM T39919 D07JGT 4421 IC50 = 57500 nM T39919 D07JVL 3016 IC50 = 133000 nM T39919 D07KSG 2733526 IC50 = 133000 nM T39919 D07QCE 2265 IC50 = 133000 nM T39919 D07SUG 2478 IC50 = 133000 nM T39919 D07TQV 60825 IC50 = 133000 nM T39919 D07UBG 130881 IC50 = 28500 nM T39919 D07UYO 441401 IC50 = 133000 nM T39919 D07VDZ 5284627 IC50 = 133000 nM T39919 D07VLY 31703 IC50 = 19000 nM T39919 D07WEP 3019 IC50 = 133000 nM T39919 D07XGR 3339 IC50 = 133000 nM T39919 D07XSN 6253 IC50 = 133000 nM T39919 D08EBN 41684 IC50 = 133000 nM T39919 D08HVR 6047 IC50 = 133000 nM T39919 D08IWD 57363 IC50 = 51000 nM T39919 D08JIV 2162 IC50 = 133000 nM T39919 D08PIQ 6741 IC50 = 40970 nM T39919 D08QIP 4887 IC50 = 2700 nM T39919 D08QMX 5757 IC50 = 133000 nM T39919 D08ROP 3899 IC50 = 133000 nM T39919 D08USJ 4456 IC50 = 133000 nM T39919 D08VRO 3822 IC50 = 133000 nM T39919 D08VXL 5353788 IC50 = 133000 nM T39919 D08VYV 4168 IC50 = 133000 nM T39919 D08ZEB 2733 IC50 = 133000 nM T39919 D09CZA 5282226 IC50 = 74000 nM T39919 D09DHY 6167 IC50 = 133000 nM T39919 D09DWL 5719 IC50 = 133000 nM T39919 D09EGZ 2719 IC50 = 103900 nM T39919 D09HNR 3002190 IC50 = 7100 nM T39919 D09HVL 16129704 IC50 = 133000 nM T39919 D09IOI 2170 IC50 = 133000 nM T39919 D09IPV 28417 IC50 = 133000 nM T39919 D09JUG 60490 IC50 = 133000 nM T39919 D09LNI 3365 IC50 = 133000 nM T39919 D09LWS 150311 IC50 = 133000 nM T39919 D09MGR 123619 IC50 = 53000 nM T39919 D09NIA 2732 IC50 = 133000 nM T39919 D09QEI 4740 IC50 = 133000 nM T39919 D09TBD 5344 IC50 = 133000 nM T39919 D09WEJ 2446 IC50 = 133000 nM T39919 D09XQF 3767 IC50 = 133000 nM T39919 D09XZB 123631 IC50 = 4600 nM T39919 D0A0OO 65016 IC50 = 133000 nM T39919 D0A2ZX 4173 IC50 = 133000 nM T39919 D0A5SE 134018 IC50 = 1900 nM T39919 D0A9YA 6918296 IC50 = 133000 nM T39919 D0AA2D 2378 IC50 = 133000 nM T39919 D0AD5C 41774 IC50 = 133000 nM T39919 D0AN7B 896 IC50 = 133000 nM T39919 D0AO5H 5578 IC50 = 133000 nM T39919 D0AP9T 53025 IC50 = 133000 nM T39919 D0AV3G 3151 IC50 = 133000 nM T39919 D0AZ3C 5291 IC50 = 133000 nM T39919 D0B1IP 5282375 IC50 = 133000 nM T39919 D0B2GI 3476 IC50 = 64000 nM T39919 D0B2UZ 4917 IC50 = 133000 nM T39919 D0B3HD 2519 IC50 = 133000 nM T39919 D0B5MP 135398513 IC50 = 133000 nM T39919 D0B6TW 135403647 IC50 = 133000 nM T39919 D0B7EB 36462 IC50 = 133000 nM T39919 D0B7NG 2725 IC50 = 133000 nM T39919 D0B8UJ 3011155 IC50 = 133000 nM T39919 D0BA9U 13109 IC50 = 133000 nM T39919 D0BM5G 5381 IC50 = 133000 nM T39919 D0C3YQ 23662354 IC50 = 133000 nM T39919 D0C4RB 36314 IC50 = 133000 nM T39919 D0C6NM 5311221 IC50 = 133000 nM T39919 D0C8EU 5394 IC50 = 133000 nM T39919 D0CL9S 159269 IC50 = 133000 nM T39919 D0CT9C 2907 IC50 = 133000 nM T39919 D0CW1P 9782 IC50 = 133000 nM T39919 D0D0BE 28061 IC50 = 133000 nM T39919 D0D0ZD 441314 IC50 = 133000 nM T39919 D0D1AL 3559 IC50 = 133000 nM T39919 D0D1SG 5755 IC50 = 133000 nM T39919 D0D2VS 60198 IC50 = 133000 nM T39919 D0D4JO 6917864 IC50 = 133000 nM T39919 D0D5GD 3373 IC50 = 133000 nM T39919 D0D5GG 4723 IC50 = 133000 nM T39919 D0D7KC 5488548 IC50 = 133000 nM T39919 D0D7LA 4091 IC50 = 133000 nM T39919 D0D8XY 5311010 IC50 = 133000 nM T39919 D0DJ1B 156391 IC50 = 133000 nM T39919 D0E0SW 53708 IC50 = 133000 nM T39919 D0E1SW 1986 IC50 = 133000 nM T39919 D0E1XL 5284583 IC50 = 133000 nM T39919 D0E6OC 5282230 IC50 = 1000 nM T39919 D0E6XR 3062316 IC50 = 27300 nM T39919 D0E6YQ 1935 IC50 = 23700 nM T39919 D0E7PQ 5311 IC50 = 133000 nM T39919 D0EG1I 9926791 IC50 = 133000 nM T39919 D0EJ6O 2763 IC50 = 133000 nM T39919 D0ES1Q 6918289 IC50 = 44000 nM T39919 D0F2PO 4828 IC50 = 133000 nM T39919 D0F6EO 33613 IC50 = 133000 nM T39919 D0F7CS 6758 IC50 = 133000 nM T39919 D0F8RA 2153 IC50 = 133000 nM T39919 D0F9GE 3108 IC50 = 8300 nM T39919 D0FM2P 82153 IC50 = 133000 nM T39919 D0G3DL 135398735 IC50 = 41900 nM T39919 D0G4OD 54686904 IC50 = 133000 nM T39919 D0G5AG 104762 IC50 = 133000 nM T39919 D0G5UB 2161 IC50 = 2200 nM T39919 D0G7FJ 54677470 IC50 = 133000 nM T39919 D0G8NN 119570 IC50 = 133000 nM T39919 D0G9IU 135403821 IC50 = 35900 nM T39919 D0G9YH 2179 IC50 = 7430 nM T39919 D0GU4K 135413536 IC50 = 133000 nM T39919 D0GY5Z 2244 IC50 = 133000 nM T39919 D0H0KB 5070 IC50 = 133000 nM T39919 D0H0ND 54454 IC50 = 133000 nM T39919 D0H3HM 60795 IC50 = 133000 nM T39919 D0H3WI 37542 IC50 = 133000 nM T39919 D0H6QU 6005 IC50 = 133000 nM T39919 D0H8FH 3702 IC50 = 133000 nM T39919 D0I0EG 44093 IC50 = 133000 nM T39919 D0I2MK 4171 IC50 = 133000 nM T39919 D0I4DQ 5280723 IC50 = 2300 nM T39919 D0I6IB 54677971 IC50 = 133000 nM T39919 D0I7SZ 54892 IC50 = 133000 nM T39919 D0IT2G 5743 IC50 = 133000 nM T39919 D0IT2X 2581 IC50 = 3000 nM T39919 D0J1MI 4030 IC50 = 15500 nM T39919 D0J1VY 5281081 IC50 = 6800 nM T39919 D0J2KV 4932 IC50 = 133000 nM T39919 D0J2MJ 26758 IC50 = 133000 nM T39919 D0J4JM 5770 IC50 = 133000 nM T39919 D0J5DC 2796 IC50 = 133000 nM T39919 D0JC9N 60164 IC50 = 133000 nM T39919 D0JO7Y 104741 IC50 = 133000 nM T39919 D0JV4Q 3002820 IC50 = 133000 nM T39919 D0JY3V 107751 IC50 = 133000 nM T39919 D0K0OZ 5702160 IC50 = 133000 nM T39919 D0K0VO 5639 IC50 = 133000 nM T39919 D0K3MC 3947 IC50 = 133000 nM T39919 D0K3QS 6442177 IC50 = 95000 nM T39919 D0K5CB 2083 IC50 = 133000 nM T39919 D0K6GZ 60464 IC50 = 133000 nM T39919 D0K7HU 6918155 IC50 = 133000 nM T39919 D0K7WK 4595 IC50 = 133000 nM T39919 D0K8KX 5280343 IC50 = 20800 nM T39919 D0KG3R 9875401 IC50 = 133000 nM T39919 D0KR2J 135398508 IC50 = 133000 nM T39919 D0L3DK 6918537 IC50 = 133000 nM T39919 D0L5RW 65015 IC50 = 133000 nM T39919 D0L5WM 2157 IC50 = 133000 nM T39919 D0L6DA 119607 IC50 = 133000 nM T39919 D0L7FM 4911 IC50 = 133000 nM T39919 D0L9ZR 4891 IC50 = 133000 nM T39919 D0M2MR 3475 IC50 = 133000 nM T39919 D0M3QP 441207 IC50 = 133000 nM T39919 D0M4YC 3114 IC50 = 133000 nM T39919 D0M5JI 9560989 IC50 = 133000 nM T39919 D0M5OC 5484727 IC50 = 133000 nM T39919 D0M6DO 2145 IC50 = 133000 nM T39919 D0M8RC 5403 IC50 = 133000 nM T39919 D0M8VE 71360 IC50 = 133000 nM T39919 D0M9BW 68911 IC50 = 133000 nM T39919 D0M9DC 4614 IC50 = 12000 nM T39919 D0MA9N 2955 IC50 = 133000 nM T39919 D0ML1F 60871 IC50 = 133000 nM T39919 D0N0RU 82146 IC50 = 133000 nM T39919 D0N0TZ 60606 IC50 = 133000 nM T39919 D0N1FS 26248 IC50 = 6400 nM T39919 D0N3VR 71616 IC50 = 133000 nM T39919 D0N4OW 644077 IC50 = 133000 nM T39919 D0N5HJ 5462501 IC50 = 133000 nM T39919 D0N5YA 65981 IC50 = 53900 nM T39919 D0N6RF 65999 IC50 = 36000 nM T39919 D0NG7O 60857 IC50 = 133000 nM T39919 D0NJ3V 4680 IC50 = 23130 nM T39919 D0NR6S 3002977 IC50 = 133000 nM T39919 D0NS6H 3152 IC50 = 72900 nM T39919 D0NW3X 71329 IC50 = 133000 nM T39919 D0O1WX 2764 IC50 = 133000 nM T39919 D0O2EM 4463 IC50 = 133000 nM T39919 D0O2SR 47528 IC50 = 133000 nM T39919 D0O3OS 104850 Ki = 4000 nM T39919 D0O4SE 5479 IC50 = 133000 nM T39919 D0O5FY 441130 IC50 = 133000 nM T39919 D0O5WP 148124 IC50 = 133000 nM T39919 D0OB1J 39186 IC50 = 133000 nM T39919 D0OT0O 44561 IC50 = 133000 nM T39919 D0P1UX 5656 IC50 = 133000 nM T39919 D0P7JZ 34359 IC50 = 133000 nM T39919 D0P9RF 5401 IC50 = 36800 nM T39919 D0PQ3G 3440 IC50 = 133000 nM T39919 D0PW7C 51039 IC50 = 133000 nM T39919 D0Q2PE 4539 IC50 = 133000 nM T39919 D0Q2XF 5311027 IC50 = 133000 nM T39919 D0Q3YO 1547484 IC50 = 133000 nM T39919 D0Q4SD 443872 IC50 = 133000 nM T39919 D0Q4XQ 3291 IC50 = 133000 nM T39919 D0Q4YK 4843 IC50 = 133000 nM T39919 D0Q5NX 216326 IC50 = 133000 nM T39919 D0Q5UQ 214348 IC50 = 36500 nM T39919 D0Q6NZ 5281034 IC50 = 133000 nM T39919 D0Q8ZX 2337 IC50 = 133000 nM T39919 D0QL3P 34312 IC50 = 133000 nM T39919 D0R0BX 6604200 IC50 = 20900 nM T39919 D0R0FE 2520 IC50 = 133000 nM T39919 D0R1RS 3715 IC50 = 5800 nM T39919 D0R1WR 4919 IC50 = 133000 nM T39919 D0R2KJ 18381 IC50 = 133000 nM T39919 D0R3FP 6398764 IC50 = 133000 nM T39919 D0R3QY 5665 IC50 = 133000 nM T39919 D0R5RR 119182 IC50 = 133000 nM T39919 D0R7HO 2471 IC50 = 133000 nM T39919 D0R8ER 3229 IC50 = 133000 nM T39919 D0R9OH 5329 IC50 = 133000 nM T39919 D0R9VR 9651 IC50 = 133000 nM T39919 D0S1NZ 5310993 IC50 = 133000 nM T39919 D0S3WH 68827 IC50 = 133000 nM T39919 D0S4BR 1349907 IC50 = 133000 nM T39919 D0S5CU 4499 IC50 = 16500 nM T39919 D0S5UH 2794 IC50 = 44500 nM T39919 D0S5WG 3366 IC50 = 133000 nM T39919 D0S9MC 2789 IC50 = 133000 nM T39919 D0S9SD 60877 IC50 = 133000 nM T39919 D0SH3I 387447 IC50 = 133000 nM T39919 D0SV8E 126941 IC50 = 133000 nM T39919 D0T0KA 4474 IC50 = 88000 nM T39919 D0T1LK 4908 IC50 = 133000 nM T39919 D0T2PL 5280453 IC50 = 133000 nM T39919 D0T2XU 4927 IC50 = 133000 nM T39919 D0T5WK 4506 IC50 = 133000 nM T39919 D0T7US 5281037 IC50 = 133000 nM T39919 D0T8GD 89594 IC50 = 133000 nM T39919 D0T8VY 71771 IC50 = 133000 nM T39919 D0T9DT 2140 IC50 = 133000 nM T39919 D0T9TJ 3034010 IC50 = 133000 nM T39919 D0TR5X 3386 IC50 = 133000 nM T39919 D0U0KW 208902 IC50 = 133000 nM T39919 D0U1OM 60726 IC50 = 133000 nM T39919 D0U2JP 4369359 IC50 = 133000 nM T39919 D0U4CE 104865 IC50 = 22000 nM T39919 D0U4UQ 3639 IC50 = 133000 nM T39919 D0U5GB 92727 IC50 = 47000 nM T39919 D0U5QK 1983 IC50 = 133000 nM T39919 D0U5RT 4909 IC50 = 133000 nM T39919 D0U5SI 4913 IC50 = 133000 nM T39919 D0U8UV 10660 IC50 = 133000 nM T39919 D0UF6M 9568512 IC50 = 133000 nM T39919 D0UL2L 54690031 IC50 = 133000 nM T39919 D0UM7O 3821 IC50 = 133000 nM T39919 D0V4QS 135398745 IC50 = 133000 nM T39919 D0V7CF 5362440 IC50 = 133000 nM T39919 D0V8QT 2708 IC50 = 133000 nM T39919 D0V9BD 2375 IC50 = 133000 nM T39919 D0VM2L 68740 IC50 = 133000 nM T39919 D0VT8P 3324 IC50 = 133000 nM T39919 D0W0BF 2187 IC50 = 133000 nM T39919 D0W9LX 2585 IC50 = 133000 nM T39919 D0WI3T 441243 IC50 = 59000 nM T39919 D0WN0U 3333 IC50 = 133000 nM T39919 D0WS1X 6915944 IC50 = 11600 nM T39919 D0WV3U 4893 IC50 = 12500 nM T39919 D0X0RI 4178 IC50 = 133000 nM T39919 D0X3FX 5284596 IC50 = 133000 nM T39919 D0X4RN 3676 IC50 = 133000 nM T39919 D0X5SD 3117 IC50 = 133000 nM T39919 D0X5XU 451668 IC50 = 133000 nM T39919 D0X6GN 444025 IC50 = 133000 nM T39919 D0X6IU 5959 IC50 = 133000 nM T39919 D0X7DE 4449 IC50 = 71000 nM T39919 D0X7KZ 6918182 IC50 = 133000 nM T39919 D0X7XG 3000226 IC50 = 133000 nM T39919 D0X9RG 5361092 IC50 = 133000 nM T39919 D0X9ZC 47965 IC50 = 133000 nM T39919 D0XF8W 1046 IC50 = 133000 nM T39919 D0Y0SW 3397 IC50 = 133000 nM T39919 D0Y2CJ 4201 IC50 = 133000 nM T39919 D0Y3MO 37768 IC50 = 133000 nM T39919 D0Y5DO 2771 IC50 = 133000 nM T39919 D0Y5UG 2160 IC50 = 133000 nM T39919 D0Y7EM 3332 IC50 = 8200 nM T39919 D0Y7IU 5281004 IC50 = 37000 nM T39919 D0Y7PG 4659569 IC50 = 16700 nM T39919 D0Y7ZU 135398738 IC50 = 133000 nM T39919 D0Y9LL 42884 IC50 = 133000 nM T39919 D0YV1Q 6032 IC50 = 133000 nM T39919 D0Z1RV 135398737 IC50 = 133000 nM T39919 D0Z1ZM 84029 IC50 = 133000 nM T39919 D0Z3DY 2333 IC50 = 17000 nM T39919 D0Z4EI 55245 IC50 = 133000 nM T39919 D0Z4SB 3478 IC50 = 133000 nM T39919 D0Z4UN 6509979 IC50 = 133000 nM T39919 D0Z4ZT 68873 IC50 = 37900 nM T39919 D0Z5BC 5634 IC50 = 63900 nM T39919 D0Z5IU 1548887 IC50 = 133000 nM T39919 D0Z6UC 5358 IC50 = 133000 nM T39919 D0Z7KE 3784 IC50 = 133000 nM T39919 D0Z8EX 18283 IC50 = 133000 nM T39919 D0Z9QR 24066 IC50 = 133000 nM T39919 D0ZB7K 5735 IC50 = 133000 nM T39919 D0ZS8P 2801 IC50 = 133000 nM T39919 D0ZU9R 392622 IC50 = 34000 nM T39919 D00TIG 6917964 IC50 = 133000 nM T39919 D08YWK 6436 IC50 = 133000 nM T39919 D09YDM 24360 IC50 = 7400 nM T39919 D0E3TC 44259 IC50 = 37900 nM T39919 D0G7UX 5284373 IC50 = 133000 nM T39919 D0Q9CY 9915743 IC50 = 23000 nM T39919 D0SD9V 53276 IC50 = 133000 nM T39919 D0TO2R 30751 IC50 = 133000 nM T39919 D0VG0D 11977753 IC50 = 133000 nM T39919 D0Y1FO 472335 IC50 = 5100 nM T39919 D01PIL 54477 IC50 = 133000 nM T39919 D01VAB 2119 IC50 = 133000 nM T39919 D02LHR 33625 IC50 = 133000 nM T39919 D03JPH 54677972 IC50 = 133000 nM T39919 D04BQR 4342 IC50 = 133000 nM T39919 D05RUM 15387 IC50 = 133000 nM T39919 D06ABW 2788 IC50 = 133000 nM T39919 D07XPE 8249 IC50 = 133000 nM T39919 D08SOF 5405 IC50 = 133000 nM T39919 D0C0JT 4495 IC50 = 133000 nM T39919 D0G9ZW 54676478 IC50 = 133000 nM T39919 D0J9GD 64715 IC50 = 133000 nM T39919 D0O2IE 4754 IC50 = 133000 nM T39919 D0OS6O 60149 IC50 = 133000 nM T39919 D0P1JI 312145 IC50 = 63200 nM T39919 D0S6QR 214350 IC50 = 133000 nM T39919 D0T1RG 216235 IC50 = 28400 nM T39919 D0Y2HR 2247 IC50 = 133000 nM T39919 D0Y4FL 6915744 IC50 = 133000 nM T39919 D0Y8UB 82148 IC50 = 133000 nM T39919 C85KQB 2202 IC50 = 133000 nM T39919 CI74WY 2450 IC50 = 133000 nM T39919 CPJ0C2 2747 IC50 = 133000 nM T39919 C36WOC 2800 IC50 = 133000 nM T39919 C7CT6M 2804 IC50 = 133000 nM T39919 CJ0B9F 3158 IC50 = 133000 nM T39919 C0H8GR 3191 IC50 = 133000 nM T39919 CEXU05 3383 IC50 = 133000 nM T39919 COSX53 3519 IC50 = 133000 nM T39919 CO2Y3R 3698 IC50 = 133000 nM T39919 C4ZJT8 3730 IC50 = 133000 nM T39919 CY4WG9 3793 IC50 = 133000 nM T39919 C9LCD8 3823 IC50 = 69000 nM T39919 C2KJI7 3883 IC50 = 133000 nM T39919 C12UDR 4411 IC50 = 133000 nM T39919 C8VXJ6 4888 IC50 = 9800 nM T39919 C93BJO 5039 IC50 = 133000 nM T39919 C5N0SU 5334 IC50 = 133000 nM T39919 C48GPY 5475 IC50 = 133000 nM T39919 C1EYR7 5497 IC50 = 133000 nM T39919 C2U1WA 6216 IC50 = 133000 nM T39919 C59UQE 6279 IC50 = 22500 nM T39919 CC09DB 9703 IC50 = 133000 nM T39919 CO1I7C 11080 IC50 = 133000 nM T39919 CMU2P6 11683 IC50 = 133000 nM T39919 C2J7BV 12947 IC50 = 133000 nM T39919 CVJ2X3 14051 IC50 = 133000 nM T39919 C6RG5E 21233 IC50 = 133000 nM T39919 CJ3OL7 25590 IC50 = 133000 nM T39919 CK21BO 27350 IC50 = 133000 nM T39919 C4VU9Z 31098 IC50 = 133000 nM T39919 CUJ6W7 35455 IC50 = 133000 nM T39919 CZA2C6 39764 IC50 = 133000 nM T39919 CFX82C 47320 IC50 = 133000 nM T39919 C6E5CD 48229 IC50 = 133000 nM T39919 CE8LA7 49659 IC50 = 133000 nM T39919 CU86VK 54459 IC50 = 133000 nM T39919 C7ZUJ4 54840 IC50 = 133000 nM T39919 CC10UB 56801 IC50 = 133000 nM T39919 CQSF39 57004 IC50 = 133000 nM T39919 CH8GS0 60749 IC50 = 133000 nM T39919 CYQ4S7 60822 IC50 = 88500 nM T39919 CHZJ65 60834 IC50 = 133000 nM T39919 C2GKD5 62884 IC50 = 133000 nM T39919 CY8ES4 62935 IC50 = 133000 nM T39919 CA9S6G 62978 IC50 = 8000 nM T39919 C7SO5H 63021 IC50 = 133000 nM T39919 CP8F7B 64143 IC50 = 97000 nM T39919 CD9TC8 64737 IC50 = 133000 nM T39919 C7WUM6 65335 IC50 = 133000 nM T39919 COZ10X 65348 IC50 = 133000 nM T39919 CS7L6J 65957 IC50 = 133000 nM T39919 C7AV1G 68553 IC50 = 133000 nM T39919 C73LEV 71399 IC50 = 133000 nM T39919 C6A4VW 71651 IC50 = 133000 nM T39919 C2F1OT 77997 IC50 = 133000 nM T39919 C1W8YJ 78000 IC50 = 133000 nM T39919 C6NLX4 84003 IC50 = 2700 nM T39919 CVP7G8 101526 IC50 = 133000 nM T39919 C90TYQ 130313 IC50 = 133000 nM T39919 CAR7Y4 146571 IC50 = 133000 nM T39919 C3WVZ6 154068 IC50 = 133000 nM T39919 CI7BE6 219025 IC50 = 133000 nM T39919 CA6ID2 241903 IC50 = 35100 nM T39919 CV80FO 249332 IC50 = 133000 nM T39919 C0VN3D 288216 IC50 = 133000 nM T39919 CLD6J9 441074 IC50 = 45800 nM T39919 CY7HM4 441313 IC50 = 133000 nM T39919 CDU0B1 441351 IC50 = 133000 nM T39919 CVX0K8 443866 IC50 = 133000 nM T39919 C40YBS 444036 IC50 = 133000 nM T39919 C35HJB 656684 IC50 = 133000 nM T39919 CGIY90 688272 IC50 = 133000 nM T39919 CBM17N 3000706 IC50 = 133000 nM T39919 C4BR7C 3005572 IC50 = 133000 nM T39919 CWQI02 3033817 IC50 = 133000 nM T39919 CH86TV 3033968 IC50 = 133000 nM T39919 C2XP0H 3052775 IC50 = 133000 nM T39919 CONV41 4022878 IC50 = 133000 nM T39919 C4SL8Q 5281025 IC50 = 133000 nM T39919 C9QDT1 5281067 IC50 = 133000 nM T39919 CNI9X4 5281888 IC50 = 6000 nM T39919 C4X7RJ 5282408 IC50 = 133000 nM T39919 C10CPM 5282455 IC50 = 26800 nM T39919 CBLX43 5282481 IC50 = 133000 nM T39919 CB4P2S 5289394 IC50 = 133000 nM T39919 CG53MU 5353627 IC50 = 133000 nM T39919 CUA96S 5388961 IC50 = 133000 nM T39919 C5DV8U 5702270 IC50 = 68200 nM T39919 C4GST2 6321416 IC50 = 28000 nM T39919 CC9WJ2 6433334 IC50 = 133000 nM T39919 CQR03B 6526396 IC50 = 133000 nM T39919 C0P8LZ 6602611 IC50 = 133000 nM T39919 CPK20Z 6917733 IC50 = 133000 nM T39919 C9FQ0W 6918092 IC50 = 133000 nM T39919 C9P2HT 9556529 IC50 = 133000 nM T39919 CEO67P 9588170 IC50 = 73200 nM T39919 C5W7MS 9833407 IC50 = 133000 nM T39919 CJL94H 9839243 IC50 = 133000 nM T39919 C7QK8R 9847786 IC50 = 133000 nM T39919 CIWP56 9886273 IC50 = 46000 nM T39919 C5NH4J 9912089 IC50 = 133000 nM T39919 C45JHO 9933004 IC50 = 133000 nM T39919 CIV15Q 10113978 IC50 = 8100 nM T39919 CZ1XW6 10483360 IC50 = 13500 nM T39919 C8BL9W 10695961 IC50 = 24000 nM T39919 CV2E4Z 11476710 IC50 = 34100 nM T39919 CVG4M1 11679357 IC50 = 133000 nM T39919 CZ6PB5 12001375 IC50 = 133000 nM T39919 CCLY36 12004215 IC50 = 133000 nM T39919 C9N5YG 14720269 IC50 = 133000 nM T39919 CGL5Q2 16051965 IC50 = 35600 nM T39919 CA3JL7 16052011 IC50 = 133000 nM T39919 C7WI4H 16204922 IC50 = 133000 nM T39919 CLHO84 16759173 IC50 = 133000 nM T39919 C71VGO 16760285 IC50 = 133000 nM T39919 CUZE40 18004026 IC50 = 133000 nM T39919 C28AYI 18530292 IC50 = 8080 nM T39919 C0REQ9 20055509 IC50 = 133000 nM T39919 CQ31BP 23623618 IC50 = 133000 nM T39919 CFE9R6 23666879 IC50 = 133000 nM T39919 CH59NC 23667631 IC50 = 133000 nM T39919 CWB0H2 23674512 IC50 = 133000 nM T39919 CFLN18 23675322 IC50 = 54200 nM T39919 CD01LT 23685176 IC50 = 133000 nM T39919 C9YI0H 23716436 IC50 = 1900 nM T39919 C3N4GQ 25078429 IC50 = 133000 nM T39919 CW7ZK4 44181971 IC50 = 133000 nM T39919 C4OT7Z 44403122 Ki = 7000 nM T39919 CUA6N3 46783232 IC50 = 133000 nM T39919 C9SCG4 49800073 IC50 = 133000 nM T39919 CRV3P5 54685920 IC50 = 133000 nM T39919 CGK7Y9 54685925 IC50 = 133000 nM T39919 CQ6C4E 56972143 IC50 = 2700 nM T39919 CM5T1V 57393422 IC50 = 133000 nM T39919 CTO71V 72734347 IC50 = 133000 nM T39919 CRZ62F 73355036 IC50 = 133000 nM T39919 C41TDB 135413523 IC50 = 26800 nM T39919 CDN1S3 135413539 IC50 = 133000 nM T39919 CG8C4T 135415564 IC50 = 15900 nM T39919 C27TMO 137648451 IC50 = 7500 nM T39919 CHPC06 137654606 IC50 = 133000 nM T39919 C67IKZ 145948937 IC50 = 133000 nM T39919 C9RLJ3 3661 IC50 = 133000 nM T39919 D01BJB 15032 IC50 = 133000 nM T39919 D01OIK 155774 IC50 = 133000 nM T39919 D03IRR 2206 IC50 = 133000 nM T39919 D04LBT 14957 IC50 = 133000 nM T39919 D07GXY 4850 IC50 = 133000 nM T39919 D08CNS 3748 IC50 = 133000 nM T39919 D09XCX 5694 IC50 = 44900 nM T39919 D0F4QX 5601 IC50 = 133000 nM T39919 D0F5LH 4634 IC50 = 133000 nM T39919 D0J6JT 1355 IC50 = 133000 nM T39919 D0L9PX 5943 IC50 = 133000 nM T39919 D0T5RO 16129706 IC50 = 133000 nM T39231 D01SHZ 9931954 IC50 = 144 nM T39231 D04AIT 5280445 IC50 = 2398.83 nM T39231 D0J9HW 23725625 IC50 = 1230 nM T39231 D00BMF 24958200 IC50 = 2344.23 nM T39231 D0F5TD 135565981 IC50 = 50 nM T39231 C3S7DE 1686 IC50 = 313 nM T39231 CH62DB 1853 IC50 = 112.2 nM T39231 CM82AL 51459 IC50 > 10000 nM T39231 CXG7Y0 76959 IC50 > 100000 nM T39231 CO7Z4L 77793 IC50 = 71 nM T39231 CS74HZ 145726 IC50 = 230 nM T39231 CNVB16 146013 IC50 > 10000 nM T39231 CW9I1J 146492 IC50 > 10000 nM T39231 C4FEY6 147157 IC50 > 10000 nM T39231 CW78JD 151515 IC50 = 233 nM T39231 C0F1IA 229015 IC50 = 310 nM T39231 C7ER4A 229016 IC50 = 794.33 nM T39231 CJ2UB5 236501 IC50 > 100000 nM T39231 C3PS2M 249526 IC50 > 10000 nM T39231 CY65EM 261391 IC50 = 275.42 nM T39231 C2O7DN 265714 IC50 = 360 nM T39231 C8AX6O 466268 IC50 = 5000 nM T39231 CYC75Z 622510 IC50 = 66 nM T39231 CH8FK7 1091861 IC50 = 15848.93 nM T39231 CA6OJ3 1241435 IC50 = 66.07 nM T39231 C40IBK 1506320 IC50 = 398.11 nM T39231 C6EZY0 1511413 IC50 = 251.19 nM T39231 C89WXS 2802462 IC50 = 6 nM T39231 C1HJR0 2817216 IC50 > 10000 nM T39231 CZ07RY 2817491 IC50 = 7 nM T39231 CTO30U 2825267 IC50 > 10000 nM T39231 C48HET 2825269 IC50 = 272 nM T39231 C1NOK3 2946601 IC50 = 1800 nM T39231 CZ8H1N 2959509 IC50 = 1000 nM T39231 CLJ6X7 3163516 IC50 = 630.96 nM T39231 CR26SK 4163640 IC50 = 1100 nM T39231 CT9V6M 4826644 IC50 = 620 nM T39231 C8ZW6Y 5272796 IC50 = 851.14 nM T39231 C4C8BV 5320693 IC50 = 560 nM T39231 CB86MY 5391140 IC50 = 280 nM T39231 C7CIL3 6490174 IC50 > 100000 nM T39231 C4P2UQ 8607850 IC50 > 100000 nM T39231 CAV3P4 9899130 IC50 = 199.53 nM T39231 CI0QP9 11960529 IC50 = 10740 nM T39231 C4Y5DW 12402280 IC50 = 90 nM T39231 CZ0KO4 14668434 IC50 = 31 nM T39231 CO9U6A 14735886 IC50 = 162 nM T39231 C5ZW8I 15989803 IC50 = 1258.93 nM T39231 CCBV16 16013151 IC50 = 1761 nM T39231 CG5A7W 16013152 IC50 = 2550 nM T39231 CPG4V1 16013160 IC50 = 559 nM T39231 CJ2XS5 16031314 IC50 = 395 nM T39231 C9LT3B 16031344 IC50 = 299 nM T39231 C80PHC 16193211 IC50 = 125.89 nM T39231 C4T7EK 16516470 IC50 = 1010 nM T39231 CZ6M5I 22431503 IC50 = 125.89 nM T39231 CO81DU 22432629 IC50 = 31.62 nM T39231 CP9H4Y 22432631 IC50 = 50.12 nM T39231 C0DW5F 22582935 IC50 = 28 nM T39231 CA3TO2 22582936 IC50 = 32 nM T39231 C1Y2MX 24772013 IC50 = 2000 nM T39231 CL8Q0K 24772834 IC50 = 3500 nM T39231 C0IOR9 25015515 IC50 = 3090.3 nM T39231 CMXA39 28825277 IC50 > 100000 nM T39231 CSO1Z6 28825295 IC50 > 100000 nM T39231 C8BKV6 44381234 IC50 = 407.38 nM T39231 CNI3Y5 44483163 IC50 = 131 nM T39231 CEI70H 45116983 IC50 = 144.54 nM T39231 C92MLH 46261432 IC50 = 19.95 nM T39231 C46BCE 46742374 IC50 = 114 nM T39231 C2XI7M 46742375 IC50 = 146 nM T39231 CWF40I 56587957 IC50 = 343 nM T39231 C6O1UZ 58829329 IC50 = 150 nM T39231 CN8AS7 67072266 IC50 > 100000 nM T39231 CD3HT9 67960134 IC50 = 46 nM T39231 C2JKD9 69004309 IC50 > 100000 nM T39231 C7QLY3 71464718 IC50 = 200 nM T39231 C24XZF 71576800 IC50 = 860 nM T39231 CED5V6 71622125 IC50 = 691.83 nM T39231 CI0GU8 71660496 IC50 = 2 nM T39231 CAO96N 71680699 IC50 > 20000 nM T39231 CI98LH 71680701 IC50 = 1300 nM T39231 C40RSX 71680702 IC50 > 20000 nM T39231 CHOZ71 71680703 IC50 = 4300 nM T39231 CL20JN 71680704 IC50 = 1500 nM T39231 CBH64M 71680705 IC50 = 400 nM T39231 C91BGF 71680860 IC50 = 1220 nM T39231 COP6V9 71680863 IC50 = 18 nM T39231 CBS20R 71681023 IC50 = 16 nM T39231 C1KT7H 71681028 IC50 = 10 nM T39231 CH1FS9 71681175 IC50 = 4 nM T39231 CZ1H8S 71681176 IC50 = 4 nM T39231 CCAK12 71681177 IC50 = 3 nM T39231 CHO50K 71681178 IC50 = 11 nM T39231 CJO9X1 71681179 IC50 = 1 nM T39231 CJ34PZ 71681180 IC50 = 4 nM T39231 C2RGP3 71681329 IC50 = 3 nM T39231 CI5E8F 71681330 IC50 = 1 nM T39231 C32RCL 71681331 IC50 = 143 nM T39231 CVJ86T 71681485 IC50 = 4 nM T39231 CY12QO 71681487 IC50 = 4 nM T39231 CH4V6D 71681649 IC50 = 5 nM T39231 CC0UX4 71683057 IC50 > 20000 nM T39231 CGU79X 71683058 IC50 > 20000 nM T39231 CX0M7D 71683059 IC50 > 20000 nM T39231 CFM05A 71683060 IC50 = 1600 nM T39231 C1MP6Q 71683061 IC50 = 540 nM T39231 C7KNH4 71736275 IC50 = 364 nM T39231 CL2H7E 71736276 IC50 = 16 nM T39231 C82YZD 71736278 IC50 = 12 nM T39231 CZS9B1 71736279 IC50 = 12 nM T39231 C2B5MQ 71736447 IC50 = 17 nM T39231 CF5M7C 71736755 IC50 = 13 nM T39231 CMJY69 71737385 IC50 = 17 nM T39231 CO96XF 71819164 IC50 = 262 nM T39231 CMC2J4 72193935 IC50 = 49 nM T39231 CL73DQ 72549316 IC50 = 7.943 nM T39231 CX9BU6 72549541 IC50 = 6.31 nM T39231 C06VKU 72549782 IC50 = 316.23 nM T39231 C46DHU 72724967 IC50 = 9 nM T39231 C8SL4X 72724968 IC50 = 148 nM T39231 CL3J2U 73056614 IC50 = 24 nM T39231 C8DX4G 73293052 IC50 = 14 nM T39231 CK67DZ 73293053 IC50 = 12 nM T39231 CE4PM3 73293055 IC50 = 7 nM T39231 CVTK56 73295340 IC50 = 31 nM T39231 CTWE30 73347820 IC50 = 64000 nM T39231 CNIH86 73351951 IC50 = 1250 nM T39231 CK9X5R 73356483 IC50 = 24 nM T39231 CU3D9N 73388373 IC50 = 2.512 nM T39231 C1OUQ4 73441895 IC50 = 19.95 nM T39231 CZY9U8 73441896 IC50 = 15.85 nM T39231 CR5E3W 73441897 IC50 = 10 nM T39231 CKF92G 73442057 IC50 = 25.12 nM T39231 CC51JH 73442058 IC50 = 3.981 nM T39231 C10MTI 73442172 IC50 = 15.85 nM T39231 CZKO04 73442173 IC50 = 25.12 nM T39231 CKGD48 73442233 IC50 = 7.943 nM T39231 CRO8S1 73442292 IC50 = 15.85 nM T39231 C6QO3Z 73442409 IC50 = 199.53 nM T39231 C1UQI4 73442411 IC50 = 125.89 nM T39231 CSP08U 73442462 IC50 = 398.11 nM T39231 CE8H9P 73442464 IC50 = 50.12 nM T39231 CS9H2V 73442467 IC50 = 19.95 nM T39231 C67FWO 73442584 IC50 = 100 nM T39231 CTUM58 73442643 IC50 = 7.943 nM T39231 CH18VD 73442700 IC50 = 10 nM T39231 C7YZ6G 73442705 IC50 = 63.1 nM T39231 CH3AT1 76280996 IC50 = 6.1 nM T39231 CZ7OL0 76284556 IC50 = 59 nM T39231 C8IT9R 76684090 IC50 = 133.3 nM T39231 CRE2U3 77050682 IC50 > 10000 nM T39231 C9VP6T 86276157 IC50 = 12 nM T39231 C3XO5D 89649815 IC50 = 562.34 nM T39231 C83KNV 89661926 IC50 = 1122.02 nM T39231 CL5RS1 90082725 IC50 = 25.12 nM T39231 C2EFL0 91810427 IC50 = 136 nM T39231 CF8W2B 91928421 IC50 = 19000 nM T39231 C2XR5Q 92045137 IC50 = 9 nM T39231 CV0NZ7 105539834 IC50 = 550 nM T39231 CYQ1E2 117999828 IC50 = 35 nM T39231 COD65L 117999906 IC50 = 18 nM T39231 CLZ1U3 118498201 IC50 = 0.18 nM T39231 CT78JM 118498266 IC50 = 0.2 nM T39231 C1VB9L 118507411 IC50 = 0.24 nM T39231 CI70KV 118717515 IC50 = 181 nM T39231 CRK45H 122177906 IC50 = 245.47 nM T39231 C8GS6E 122177907 IC50 = 331.13 nM T39231 C9SXK6 122177908 IC50 = 700 nM T39231 CH3RJ2 122177909 IC50 = 346.74 nM T39231 CL4A3P 122177910 IC50 = 570 nM T39231 C0ZKD7 122177911 IC50 = 4600 nM T39231 CP1QU7 122177912 IC50 = 2454.71 nM T39231 CVCS41 122177963 IC50 = 370 nM T39231 CDX95C 122177964 IC50 = 290 nM T39231 CYWJ91 122177965 IC50 = 290 nM T39231 CWO65I 122205439 IC50 = 483 nM T39231 C5QD0E 122205440 IC50 = 104 nM T39231 C02SDC 122423373 IC50 = 3200 nM T39231 CF2NO9 127037410 IC50 = 10964.78 nM T39231 CV06MU 131801402 IC50 = 28.84 nM T39231 CD1R6Q 135400456 IC50 = 1406 nM T39231 C9PI7O 135402338 IC50 = 1100 nM T39231 C0HQF2 135404247 IC50 = 140 nM T39231 C95RAN 135405744 IC50 = 528 nM T39231 C6FY0X 135416131 IC50 = 786 nM T39231 C6DBN7 135417258 IC50 = 346 nM T39231 CCY9H6 135417291 IC50 = 53 nM T39231 C1KBX6 135417551 IC50 = 135 nM T39231 C1PE8H 135417609 IC50 = 35 nM T39231 C47LAF 135418940 IC50 = 10 nM T39231 CIS9K5 135421564 IC50 = 224 nM T39231 CM5Q1Z 135430309 IC50 = 67 nM T39231 C4MW7F 135443732 IC50 = 299 nM T39231 CH14EB 135443955 IC50 = 5 nM T39231 C8XI3K 135448518 IC50 = 430 nM T39231 CZ9GA7 135449434 IC50 > 100000 nM T39231 CA0R7X 135452109 IC50 = 346 nM T39231 C9H1VA 135456692 IC50 = 1284 nM T39231 C8J2PC 135456762 IC50 = 48 nM T39231 CHY9C3 135479130 IC50 = 781 nM T39231 CJO81C 135513650 IC50 = 156 nM T39231 C7G6BQ 135513721 IC50 = 73 nM T39231 CU3FW2 135566794 IC50 = 8 nM T39231 C8QDG3 135566882 IC50 = 0.1 nM T39231 CVD04P 135566883 IC50 = 63 nM T39231 CNVM21 135566884 IC50 = 0.1 nM T39231 C4BFY3 135566969 IC50 = 35 nM T39231 C59OUK 135566970 IC50 = 50 nM T39231 C7K5WL 135566971 IC50 = 2423 nM T39231 CN74FK 135566972 IC50 = 153 nM T39231 CRY12I 135566973 IC50 = 22 nM T39231 CU2I7X 135567125 IC50 = 9.12 nM T39231 C37PTU 135567126 IC50 = 5.1 nM T39231 CT1DZ8 135644892 IC50 = 39.4 nM T39231 C38XBR 135652704 IC50 = 20.5 nM T39231 C1G4CE 135741330 IC50 = 93 nM T39231 CAT50N 135741861 IC50 = 485 nM T39231 C4ZGO7 135741892 IC50 = 110 nM T39231 CIL7K3 135742498 IC50 = 322 nM T39231 CS83CJ 135905416 IC50 = 100 nM T39231 C12CPN 136165102 IC50 = 1090 nM T39231 C54NVS 136175126 IC50 = 0.81 nM T39231 CVH7R6 136175127 IC50 = 8.5 nM T39231 CS5PH8 136175128 IC50 = 0.4 nM T39231 CY94ZB 136215772 IC50 = 36 nM T39231 C7JEG1 136215773 IC50 = 44 nM T39231 CF7O2U 136215774 IC50 = 73 nM T39231 CFP0V5 136215897 IC50 = 32 nM T39231 C18GVR 136224209 IC50 = 0.2 nM T39231 C80BWX 136224210 IC50 = 0.2 nM T39231 CBQ6R1 136224211 IC50 = 0.2 nM T39231 C0HS5P 136224212 IC50 = 400 nM T39231 CB19RP 136227775 IC50 = 155 nM T39231 CM4PB2 136236970 IC50 = 12.5 nM T39231 C50JYC 136236972 IC50 = 14 nM T39231 C1WG3C 136236974 IC50 = 17 nM T39231 CF1H5N 136236975 IC50 = 23 nM T39231 CU17IT 136236976 IC50 = 11 nM T39231 C71FDZ 136236977 IC50 = 10 nM T39231 CCL4D6 136236978 IC50 = 24 nM T39231 C9WHB4 136236979 IC50 = 3.3 nM T39231 C68GON 136236980 IC50 = 12 nM T39231 C18MSY 136236981 IC50 = 10 nM T39231 CF01JX 136236982 IC50 = 7 nM T39231 CYF2I1 136236983 IC50 = 1000 nM T39231 C3ZW8J 136236994 IC50 = 1.6 nM T39231 CN0J1C 136236995 IC50 = 35 nM T39231 CHJ8I2 136236997 IC50 = 1.2 nM T39231 C0LB6W 136236998 IC50 = 0.8 nM T39231 CVB4D7 136237000 IC50 = 26 nM T39231 CSB3Y1 136237004 IC50 = 1.5 nM T39231 C4H8ZN 136237010 IC50 = 15 nM T39231 CCL4V0 136240108 IC50 = 0.2 nM T39231 CHM35F 136240109 IC50 = 0.1 nM T39231 C8E0AF 136241425 IC50 = 800 nM T39231 CW17FT 136241426 IC50 = 27 nM T39231 C5NI6F 136241427 IC50 > 46000 nM T39231 CRWN30 136241639 IC50 = 0.2 nM T39231 C2KO4C 136241640 IC50 = 31 nM T39231 C52DUR 136241641 IC50 = 16 nM T39231 CFA4R8 136241642 IC50 = 1 nM T39231 CR07BF 136244504 IC50 = 5000 nM T39231 CHSN59 136245073 IC50 = 907 nM T39231 C7VX4R 136245086 IC50 = 21 nM T39231 CM5JC2 136245087 IC50 > 46000 nM T39231 CCIV06 136245088 IC50 > 46000 nM T39231 C3NX2H 136249376 IC50 = 0.2 nM T39231 C3RIV5 136249377 IC50 = 0.3 nM T39231 CE2I0N 136249378 IC50 = 0.2 nM T39231 CNOA16 136249379 IC50 = 1750 nM T39231 C5REV1 136249380 IC50 = 860 nM T39231 C3IQ7P 136249381 IC50 > 46000 nM T39231 C2P5LK 136253145 IC50 = 50 nM T39231 CHD0B7 136264278 IC50 = 2 nM T39231 C5DAO8 136264279 IC50 = 210 nM T39231 CCE28N 136264280 IC50 = 400 nM T39231 C2YO7J 136264281 IC50 = 640 nM T39231 C0D8MZ 136264443 IC50 = 46 nM T39231 C7HMR2 136264453 IC50 = 37 nM T39231 CUPY84 136268378 IC50 = 65.4 nM T39231 CF3X4M 136372378 IC50 = 101 nM T39231 CUB67C 136404917 IC50 > 100000 nM T39231 CWH02F 136491252 IC50 = 47 nM T39231 CF80AR 136491263 IC50 = 111 nM T39231 C6T9OI 136947736 IC50 = 2.2 nM T39231 C91WJF 136947741 IC50 = 1.3 nM T39231 CFS5Z4 136947743 IC50 = 31 nM T39231 CVM4S9 136947751 IC50 = 35 nM T39231 C9UGV5 137169064 IC50 = 19.4 nM T39231 CMN5H6 137169065 IC50 = 21.3 nM T39231 CF8LC7 137632525 IC50 = 977.24 nM T39231 C8K3CX 137634198 IC50 = 31.62 nM T39231 CS7ZQ8 137637696 IC50 = 33.88 nM T39231 C7V2RQ 137640411 IC50 = 7943.28 nM T39231 CJE2O1 137642565 IC50 = 2691.53 nM T39231 C46GFQ 137643877 IC50 = 6000 nM T39231 CM21PL 137646367 IC50 = 575.44 nM T39231 CIF2B4 137646395 IC50 = 10000 nM T39231 C34NWB 137649146 IC50 = 158.49 nM T39231 CG0P8H 137650831 IC50 = 9332.54 nM T39231 CD0E9C 137653685 IC50 > 10000 nM T39231 C5ZX2H 137653831 IC50 = 7943.28 nM T39231 CX2HY9 137656402 IC50 > 10000 nM T39231 C4UTR7 137656957 IC50 = 4786.3 nM T39231 C72FHM 137660379 IC50 = 9772.37 nM T39231 C74JDS 137660681 IC50 = 1.995 nM T39231 C4R7VI 137701512 IC50 = 14.3 nM T39231 CWLV03 138594154 IC50 = 7.9 nM T39231 CDW5N1 138594164 IC50 = 4.9 nM T39231 CSK82I 138594166 IC50 = 4.8 nM T39231 CD1M0Y 138594171 IC50 = 12.8 nM T39231 C9QYJ3 138594172 IC50 = 11.1 nM T39231 C1XSH7 138594194 IC50 = 36.1 nM T39231 C4JO9N 138594198 IC50 = 3.7 nM T39231 C7I1CT 138594235 IC50 = 13.6 nM T39231 CVI5N9 138594242 IC50 = 7.5 nM T39231 CS8U3T 138594273 IC50 = 9.2 nM T39231 CYR32Z 138594277 IC50 = 3.8 nM T39231 CNSV30 138594278 IC50 = 6.1 nM T39231 C1C2AS 138594290 IC50 = 12 nM T39231 C34OCY 138594292 IC50 = 5.5 nM T39231 CUA1E8 138594320 IC50 = 3.5 nM T39231 CGE6Q5 138594327 IC50 = 11.1 nM T39231 C0RST4 138594360 IC50 = 33.7 nM T39231 C4K7MW 138594363 IC50 = 4.4 nM T39231 CNW2O9 138594369 IC50 = 6.4 nM T39231 C3F7MV 138594378 IC50 = 7.5 nM T39231 C6YU8S 138594385 IC50 = 16 nM T39231 C48AGS 138594414 IC50 = 28.5 nM T39231 CA49EZ 138594436 IC50 = 43.4 nM T39231 CL6EV4 138594465 IC50 = 4.2 nM T39231 CJL05F 138594467 IC50 = 9.9 nM T39231 CX4SL6 138594472 IC50 = 4.4 nM T39231 C3E5IU 138594491 IC50 = 14.1 nM T39231 C13EVQ 138594498 IC50 = 31.5 nM T39231 C4L9XQ 138594506 IC50 = 49.3 nM T39231 CKF1W3 138594528 IC50 = 11.1 nM T39231 C98NUR 138594556 IC50 = 4.4 nM T39231 CDZ43N 138594558 IC50 = 7.9 nM T39231 CLD3J5 138594570 IC50 = 7.7 nM T39231 CWVO67 138594578 IC50 = 18.2 nM T39231 C6QD2W 138594607 IC50 = 10.2 nM T39231 CP6Y5L 138594610 IC50 = 4.5 nM T39231 CSQJ12 138594627 IC50 = 5.3 nM T39231 CEOJ61 138594628 IC50 = 5.8 nM T39231 CU4O9K 138594631 IC50 = 5.3 nM T39231 C0A4FG 138594645 IC50 = 11 nM T39231 CN3U9X 138594667 IC50 = 9 nM T39231 CQK29G 138594732 IC50 = 8.4 nM T39231 CCU4I1 138594747 IC50 = 6.4 nM T39231 C1KWY7 138594763 IC50 = 5.8 nM T39231 C9HR2J 138594785 IC50 = 30.2 nM T39231 CP4NF9 138594790 IC50 = 27.6 nM T39231 CF74SW 138594809 IC50 = 16.8 nM T39231 CF7ZR5 138594952 IC50 = 10 nM T39231 CW5E6D 138594964 IC50 = 16.7 nM T39231 CURM89 138594969 IC50 = 16.6 nM T39231 C72QVS 138595093 IC50 = 118 nM T39231 C8I9CD 142613964 IC50 = 5.4 nM T39231 C5SG1U 145957836 IC50 = 1000 nM T39231 CPR0N4 145962722 IC50 > 100000 nM T39231 C6HOA3 145972257 IC50 = 5700 nM T39231 CA65UC 145974539 IC50 = 3000 nM T39231 C20TJH 145987470 IC50 = 11000 nM T39231 COB76P 145989667 IC50 = 131 nM T39231 CPY72O 153951026 IC50 = 15 nM T39231 CWV08R 155511996 IC50 = 1350 nM T39231 CZ78CA 155513337 IC50 = 14300 nM T39231 CRX36I 155515281 IC50 = 4.3 nM T39231 CC9J2N 155516254 IC50 = 6.3 nM T39231 C6EJ7I 155518170 IC50 = 7779 nM T39231 CIC9H8 155518184 IC50 = 14.9 nM T39231 C1DL6E 155518640 IC50 = 220 nM T39231 CGKW04 155520067 IC50 > 20000 nM T39231 CHV6T4 155521523 IC50 = 2.5 nM T39231 CUM52X 155522687 IC50 = 3.4 nM T39231 CEP6Y5 155528458 IC50 = 79.6 nM T39231 C91IPT 155529963 IC50 = 8.9 nM T39231 CA9XP1 155531429 IC50 = 28.5 nM T39231 CL2PO4 155532179 IC50 = 10.3 nM T39231 C09PYD 155532212 IC50 = 67.6 nM T39231 C4JPD1 155532717 IC50 = 21.3 nM T39231 CZL4U1 155534087 IC50 = 16.2 nM T39231 CV2MX1 155535415 IC50 = 35 nM T39231 CY8RJ7 155537249 IC50 = 131 nM T39231 CWM48X 155538013 IC50 = 19.4 nM T39231 CU65VW 155540828 IC50 = 514 nM T39231 CZN0O1 155541146 IC50 = 5919 nM T39231 CYWG48 155541643 IC50 > 1000 nM T39231 C9INM1 155543325 IC50 = 9.2 nM T39231 CG0J7F 155545779 IC50 = 6.3 nM T39231 CO0E8F 155549220 IC50 = 6.2 nM T39231 CD5C9R 155550189 IC50 > 20000 nM T39231 C4P3QD 155553178 IC50 = 19 nM T39231 CIYH06 155556919 IC50 = 6168 nM T39231 CXAJ25 155557028 IC50 = 53.5 nM T39231 CWH8D0 155561438 IC50 = 7.8 nM T39231 C46UYI 155562058 IC50 = 6008 nM T39231 COH6X1 155564702 IC50 = 6.8 nM T39231 D00RIX 5280443 IC50 = 3162.28 nM T39231 D00TUB 135471356 IC50 = 83 nM T39231 D02CHG 248021 IC50 = 588.84 nM T39231 D03BQJ 688829 IC50 = 47 nM T39231 D04GFX 736736 IC50 > 10000 nM T39231 D04WDX 4858 IC50 = 1348.96 nM T39231 D06NKJ 135439437 IC50 = 475 nM T39231 D07BPT 135457978 IC50 = 32 nM T39231 D0B2WX 135407310 IC50 = 37 nM T39231 D0C5XB 261395 IC50 = 208.93 nM T39231 D0E5EW 135531482 IC50 = 42 nM T39231 D0G5VD 135492389 IC50 = 58 nM T39231 D0GA0Y 135463623 IC50 = 35 nM T39231 D0O6WW 135528341 IC50 = 195 nM T39231 D0OF1I 135417274 IC50 = 873 nM T39231 D0P3CX 689013 IC50 > 10000 nM T39231 D0S0RK 10680 IC50 = 323.59 nM T39231 D0Y1MH 135471354 IC50 = 52 nM T39231 D0YJ3Q 5322065 IC50 = 630 nM T34287 CQ2B5Z 44313403 IC50 = 140000 nM T34287 CH7W9F 44313519 IC50 = 39000 nM T34287 CFEN62 44313520 IC50 = 40000 nM T34287 CQWZ67 44313524 IC50 = 34000 nM T34287 CD2O9V 44313525 IC50 > 200000 nM T34287 CHGO46 44313559 IC50 > 200000 nM T34287 C7GEA5 44313560 IC50 > 200000 nM T34287 CXN3V4 44313599 IC50 = 50000 nM T34287 CLIX86 44313609 IC50 = 14000 nM T34287 CXG87J 44313676 IC50 = 34000 nM T34287 CCP04F 44313751 IC50 > 200000 nM T34287 C0CD4S 44313774 IC50 > 200000 nM T34287 C74CAN 44313775 IC50 = 93000 nM T34287 CYQU68 44313793 IC50 = 21000 nM T34287 CL81DH 44313818 IC50 = 50000 nM T34287 C2BL4S 44313832 IC50 = 15000 nM T34287 C0C7MZ 44313842 IC50 = 6000 nM T34287 CMJ68T 44313861 IC50 > 200000 nM T34287 CCUH40 44313876 IC50 > 200000 nM T34287 C75VKP 44313877 IC50 > 200000 nM T34287 CIVW97 44313898 IC50 > 500000 nM T34287 CYRQ36 44314130 IC50 = 30000 nM T76396 C8SGZ7 9799609 IC50 > 20000 nM T76396 C2H4ZK 9806118 IC50 = 12000 nM T76396 C2TN7S 9807068 IC50 > 50000 nM T76396 C71XRT 9821510 IC50 = 40000 nM T76396 CEL3C9 9824630 IC50 > 50000 nM T76396 CXE1Y8 9842436 IC50 > 20000 nM T76396 CISP20 9844227 IC50 = 11000 nM T76396 CNE6P0 9845017 IC50 = 11000 nM T76396 C7VSU2 9845018 IC50 = 3400 nM T76396 CXH80T 9845019 IC50 = 15000 nM T76396 CNIS42 9846821 IC50 = 24 nM T76396 CML5U3 9848397 IC50 = 15000 nM T76396 CXZ6Q7 9866918 IC50 > 20000 nM T76396 C0QV1K 9871743 IC50 = 12000 nM T76396 C4NJS0 9885760 IC50 = 41000 nM T76396 CRW8C1 9907452 IC50 = 46000 nM T76396 CA8KC0 9912881 IC50 > 50000 nM T76396 CW1KP6 9914569 IC50 = 4600 nM T76396 CF85LV 9915185 IC50 = 6500 nM T76396 CH2KA7 9930818 IC50 = 48000 nM T76396 CY7W8H 9931146 IC50 = 42000 nM T76396 CI8P9X 9952087 IC50 = 46000 nM T76396 CNRX39 9956928 IC50 = 1100 nM T76396 CT3O4V 10138186 IC50 = 4800 nM T76396 CNET60 10206356 IC50 = 1100 nM T76396 C5BJ0E 10238214 IC50 = 3900 nM T76396 COJI94 10862667 IC50 > 50000 nM T76396 C3SM0F 10894628 IC50 = 7400 nM T76396 C4QZ2E 10895064 IC50 = 11000 nM T76396 C5L2FR 10896860 IC50 = 3600 nM T76396 C3T9CI 10916025 IC50 = 16000 nM T76396 C3SQA5 10918896 IC50 = 2700 nM T76396 CYJ0H9 10938254 IC50 > 50000 nM T76396 CG34TZ 10949393 IC50 > 50000 nM T76396 CR8NL2 10950878 IC50 > 50000 nM T76396 C7MJ3I 10960344 IC50 = 11000 nM T76396 CL3A7F 10961614 IC50 = 41000 nM T76396 CS1CI9 10982914 IC50 = 28000 nM T76396 CIS36R 10993420 IC50 > 50000 nM T76396 CJI01L 11004204 IC50 = 1500 nM T76396 C2BX4N 11025461 IC50 = 24000 nM T76396 CPXY41 11037188 IC50 = 19000 nM T76396 CKZP84 11048052 IC50 = 19000 nM T76396 CR9K5V 11069519 IC50 = 6500 nM T76396 CN6QM7 11080796 IC50 ~ 5100 nM T76396 CV73YG 11091386 IC50 = 880 nM T76396 CBY94W 11091976 IC50 = 20000 nM T76396 CY0F2S 11101410 IC50 = 31000 nM T76396 C9COS1 11101729 IC50 = 2800 nM T76396 CRL01V 11111808 IC50 = 14000 nM T76396 CUT1Q0 11728765 IC50 > 50000 nM T76396 C30TBM 11732162 IC50 > 50000 nM T76396 CA4I7V 11824866 IC50 = 36000 nM T76396 C80JFP 17965976 IC50 = 100 nM T76396 C74LVI 44274781 IC50 = 10 nM T76396 C34TGF 44274782 IC50 = 5600 nM T76396 C4XQY2 44274783 IC50 = 1200 nM T76396 C2PNA5 44274804 IC50 = 210 nM T76396 C2U0NZ 44274806 IC50 = 240 nM T76396 CA9MJ4 44274825 IC50 = 1800 nM T76396 CM12CG 44286282 IC50 = 650 nM T76396 C5W8QG 44286298 IC50 = 2800 nM T76396 C4O9EB 44286300 IC50 = 4200 nM T76396 CGOQ58 44286304 IC50 = 2600 nM T76396 CI67NQ 44286315 IC50 = 2100 nM T76396 C2U6PY 44286332 IC50 = 3900 nM T76396 C9QSC5 44286345 IC50 = 2400 nM T76396 C9BH3L 44286376 IC50 = 1200 nM T76396 C5Y8HE 44286420 IC50 = 510 nM T76396 C08IJY 44286579 IC50 = 1600 nM T76396 CT1QP4 44286646 IC50 > 10 nM T76396 CWSA69 44286656 IC50 > 10 nM T76396 C5NG4A 44286723 IC50 = 1100 nM T76396 C4E1KL 44286730 IC50 = 5500 nM T76396 CFO4S0 44286731 IC50 > 10 nM T76396 CCD43U 44286732 IC50 = 42 nM T76396 CQH1L4 44286733 IC50 = 1400 nM T76396 CAH5P4 44286737 IC50 > 10 nM T76396 CENW21 44286755 IC50 = 830 nM T76396 C2I9BP 44286765 IC50 = 1700 nM T76396 C7XLA6 44286767 IC50 > 10 nM T76396 C05LZF 44286768 IC50 = 2100 nM T76396 CYS6L1 44286776 IC50 = 103 nM T76396 C8QG1O 44286780 IC50 = 1800 nM T76396 CKH50S 44286801 IC50 = 990 nM T76396 CT46KR 44286802 IC50 = 8620 nM T76396 CW64TF 44286942 IC50 > 10 nM T76396 CLPC20 44286957 IC50 = 960 nM T76396 C0S4NX 44286958 IC50 > 10 nM T76396 C42IDV 44286959 IC50 = 8600 nM T76396 CNO31Q 44459100 IC50 = 18 nM T76396 CI9ZK4 44459321 IC50 = 40 nM T76396 CN02QA 44459344 IC50 = 740 nM T76396 COA1V2 44459504 IC50 = 430 nM T76396 CEJ0K9 44459509 IC50 = 4100 nM T76396 CL8G5A 44459510 IC50 = 870 nM T76396 CAD74Y 44459594 IC50 = 2400 nM T76396 CG4LH7 44459775 IC50 = 3.1 nM T76396 C39TIB 44459799 IC50 = 360 nM T76396 C6RBS7 44459800 IC50 = 83000 nM T76396 C97BTH 44459819 IC50 = 9.5 nM T76396 CF2XW7 44459847 IC50 = 16 nM T76396 C4KA0M 44459853 IC50 = 92 nM T76396 C7V4FJ 44459924 IC50 > 10000 nM T93788 D00WDY 53477157 EC50 = 14 nM T93788 D01HTO 25025505 EC50 = 87 nM T93788 D0O9XN 11691484 EC50 = 46 nM T93788 D0S4II 24996872 EC50 = 3.4 nM T93788 D0Q3ES 11705608 EC50 = 2.7 nM T93788 C1JLP6 1267327 EC50 = 310 nM T93788 C12OPB 3710394 EC50 = 1000 nM T93788 CT6HM1 3766553 IC50 = 84 nM T93788 CL19MX 3800660 EC50 = 3000 nM T93788 CW7I0V 4400062 EC50 = 200 nM T93788 CBM61L 4993934 EC50 = 1900 nM T93788 C09VLS 10003301 EC50 = 2500 nM T93788 C0VR7W 10049468 IC50 = 50 nM T93788 C14WGV 10094886 EC50 = 1700 nM T93788 C43IKO 11190983 EC50 = 15 nM T93788 CPN90M 11224944 EC50 = 3.5 nM T93788 CA50RX 11271133 EC50 = 14 nM T93788 C7T4LO 11271424 EC50 = 4.2 nM T93788 CM7CW0 11283457 EC50 = 116 nM T93788 CCO2Y6 11397354 EC50 = 0.7 nM T93788 CL4J5R 11465648 EC50 = 7.4 nM T93788 CR5I6K 11503692 EC50 = 9.7 nM T93788 C5GVB6 11641004 EC50 = 31 nM T93788 CS3RW4 11663249 EC50 = 44 nM T93788 C2QWX4 11677830 EC50 = 71 nM T93788 CB4XD1 11691227 EC50 = 1320 nM T93788 C2T8FN 11751802 EC50 = 250 nM T93788 CO36JD 16036825 EC50 = 7.3 nM T93788 CA7P1J 16733804 EC50 = 200 nM T93788 CO8BD9 21897416 EC50 > 10000 nM T93788 COMA70 21897603 EC50 = 2400 nM T93788 C6ARZ3 21897616 EC50 = 435 nM T93788 CDM28O 21897675 EC50 = 8.1 nM T93788 C93QDC 21897744 EC50 = 50.12 nM T93788 CGH9P2 21897819 EC50 > 10000 nM T93788 CACM74 21897825 EC50 = 316.23 nM T93788 C2OVZ5 21897897 EC50 = 5.6 nM T93788 CR0VF4 23649212 EC50 = 131 nM T93788 CBZF78 23653563 EC50 = 50.12 nM T93788 CR9J5G 24822706 EC50 = 22 nM T93788 CE0UN4 24862850 EC50 = 400 nM T93788 C4YU8M 24896777 EC50 = 251.19 nM T93788 C0IXZ8 24896778 EC50 = 10 nM T93788 C06AXF 24897005 EC50 = 19.95 nM T93788 CZJ7U6 24897242 EC50 = 125.89 nM T93788 CXGZ83 24897245 EC50 > 10000 nM T93788 CLNB23 24897458 EC50 = 316.23 nM T93788 CJ9F7N 24897459 EC50 = 251.19 nM T93788 CR04JD 24897884 EC50 > 10000 nM T93788 CML3Z6 24897885 EC50 = 794.33 nM T93788 CLS39J 24898315 EC50 = 1995.26 nM T93788 CHRG37 24899742 EC50 = 12.59 nM T93788 C68CJU 24899747 EC50 = 1584.89 nM T93788 CFD7Y9 24899748 EC50 = 1258.93 nM T93788 CT9OL3 24899996 EC50 = 398.11 nM T93788 C89JDC 24900242 EC50 > 10000 nM T93788 CXF35U 24900244 EC50 = 31.62 nM T93788 C7I8XM 24958871 EC50 = 25 nM T93788 C04VLG 24958872 EC50 = 338 nM T93788 C3QYJ8 24961071 EC50 = 514 nM T93788 C8ZYQ0 24961798 EC50 = 6 nM T93788 CKT12U 24961799 EC50 = 6 nM T93788 CHI91S 24961800 EC50 = 1 nM T93788 CCK8G4 25012362 EC50 = 8 nM T93788 CU72GZ 25012522 EC50 = 98 nM T93788 C0EI7T 25012524 EC50 = 2 nM T93788 C85YLN 25012528 EC50 = 201 nM T93788 CO7AD3 25024141 EC50 = 103 nM T93788 CN75ZE 25052772 EC50 = 19 nM T93788 CP7NC9 25052969 IC50 = 500 nM T93788 C06OMU 25052970 EC50 = 1200 nM T93788 CVF60B 25053040 EC50 = 400 nM T93788 COHV79 25053041 EC50 = 260 nM T93788 C6TQH7 25053042 EC50 = 10 nM T93788 CB9EU8 25053043 EC50 = 430 nM T93788 CN9O5M 25053044 EC50 = 25 nM T93788 C16MFX 25053111 EC50 = 160 nM T93788 C49GZF 25053112 EC50 = 5.1 nM T93788 C85TLK 25053113 EC50 = 1.5 nM T93788 C7E1UM 25053114 EC50 = 660 nM T93788 C9C1PY 25053115 EC50 = 24 nM T93788 C5E0RZ 25053184 EC50 = 17 nM T93788 C0NSW2 25053185 EC50 = 4.7 nM T93788 C8JVE4 25053186 EC50 = 7.8 nM T93788 CN1KA0 25053187 EC50 = 17.1 nM T93788 CY6G1Q 25053188 EC50 = 110 nM T93788 CESK31 25053253 EC50 = 3.4 nM T93788 CM3OE2 25053254 EC50 = 7 nM T93788 CX73WG 25053255 EC50 = 7.9 nM T93788 CZNB62 25138357 EC50 = 133 nM T93788 CMT76B 25138367 EC50 = 63 nM T93788 CS2K9L 25204037 EC50 = 23 nM T93788 C0V6PX 25204038 EC50 = 16 nM T93788 CCO6Y1 25204174 EC50 = 183 nM T93788 C2GC5X 25204242 EC50 = 1700 nM T93788 CG5DU7 25204244 EC50 = 1091 nM T93788 C50QKG 25204645 EC50 = 57 nM T93788 C8GQY7 25204648 EC50 = 724 nM T93788 C9X8DN 25204713 EC50 = 130 nM T93788 C4FIJ0 25260830 EC50 = 17 nM T93788 CYOT98 42646474 EC50 = 95 nM T93788 CO9R2B 44177589 EC50 = 39.81 nM T93788 CMD02U 44177592 EC50 = 794.33 nM T93788 C82IAU 44177593 EC50 > 10000 nM T93788 C8WM0Z 44467183 EC50 = 2 nM T93788 C5ETU8 44467185 EC50 = 4 nM T93788 CYU89I 46208490 Ki = 20 nM T93788 CGI81S 46865202 EC50 = 90 nM T93788 CK42WB 46865203 EC50 = 300 nM T93788 C91WPT 46884780 EC50 > 10000 nM T93788 C4I0MC 46884781 EC50 > 10000 nM T93788 CDTI38 46884819 EC50 > 10000 nM T93788 CZ1QG5 46884820 EC50 = 1900 nM T93788 CND62Y 46884821 EC50 = 2600 nM T93788 CMIP79 46884822 EC50 = 1300 nM T93788 CEGR15 46884857 EC50 = 300 nM T93788 CF2SO1 46884858 EC50 = 100 nM T93788 CJ45TU 46884859 EC50 = 300 nM T93788 CU5KI2 46884902 EC50 = 200 nM T93788 CQDL72 46884903 EC50 = 2000 nM T93788 CB0L3Y 46884904 EC50 = 1800 nM T93788 CS4RO2 46884935 EC50 = 1200 nM T93788 CS1U6Z 46884936 EC50 = 1000 nM T93788 CTY74I 46884937 EC50 = 1000 nM T93788 CNDH97 46884938 EC50 = 1600 nM T93788 C3MZY2 46884986 EC50 = 800 nM T93788 CF8T7O 46884987 EC50 = 2800 nM T93788 C2CIG9 46884988 EC50 > 10000 nM T93788 C1V4KW 46884989 EC50 = 2100 nM T93788 CE71WG 46885048 EC50 = 2000 nM T93788 CVIS54 46885049 EC50 > 10000 nM T93788 CK9TR7 46885050 EC50 = 900 nM T93788 C5JNL7 46885051 EC50 = 2100 nM T93788 C0YZ8U 46885169 EC50 = 1200 nM T93788 COPL82 46885170 EC50 = 700 nM T93788 CIH1K7 46885171 EC50 = 130 nM T93788 C2H5OS 46897575 EC50 = 7.7 nM T93788 CF7UP1 46897577 EC50 = 11 nM T93788 CIF0Y7 46939910 EC50 = 15 nM T93788 C9L4ZU 49855246 EC50 = 1 nM T93788 CC27AL 51029601 EC50 = 65 nM T93788 CWJ36V 51029603 EC50 = 621 nM T93788 CSW80J 51029782 EC50 = 1925 nM T93788 CW19DN 51029876 IC50 = 17 nM T93788 CXJ30Q 51029877 EC50 = 466 nM T93788 CBR8Z2 51029964 EC50 = 45 nM T93788 CPYT82 51029965 EC50 = 3 nM T93788 CY0B7Q 51030053 EC50 = 21 nM T93788 CM0UF3 51030054 EC50 = 5 nM T93788 CW08DZ 51030056 EC50 = 63 nM T93788 C5LO4C 51030336 EC50 = 112 nM T93788 CVY9U0 51030529 EC50 = 54 nM T93788 C07HID 51030707 EC50 = 630.96 nM T93788 CM9PY8 51030710 IC50 = 12 nM T93788 CP6NI2 51030711 EC50 = 7.943 nM T93788 CTI6N7 51030811 EC50 = 75 nM T93788 CZLP32 51030896 EC50 = 21 nM T93788 C1P9UY 51030897 EC50 = 5 nM T93788 CW06HL 51030898 EC50 = 10 nM T93788 C9D8FG 51030899 EC50 = 15.85 nM T93788 CS4X5Z 51030900 EC50 = 15.85 nM T93788 C4QW2B 51030901 EC50 = 2 nM T93788 C70OGS 51030984 EC50 = 20 nM T93788 CX28ZP 51030985 EC50 = 47 nM T93788 C9W8OF 51030987 EC50 = 14 nM T93788 C35XAI 51354342 EC50 = 740 nM T93788 CBG8N3 51354343 EC50 = 2067 nM T93788 C2RCZ0 53235503 EC50 = 3 nM T93788 C6OJF7 53317209 EC50 = 267 nM T93788 CR06WM 53317210 EC50 = 340 nM T93788 C2O9SZ 53317211 EC50 = 868 nM T93788 CT2D0R 53318456 EC50 = 884 nM T93788 CQ8GY0 53318501 EC50 = 808 nM T93788 CV8P3R 53318502 EC50 = 32 nM T93788 C0S9BL 53319831 EC50 = 1380 nM T93788 C0I8YS 53321124 EC50 = 120 nM T93788 CO1HB3 53322450 EC50 = 78 nM T93788 C85UDG 53322927 EC50 = 5980 nM T93788 CO98ZY 53323811 EC50 = 75 nM T93788 CIBE50 53325083 EC50 = 409 nM T93788 CUJ28D 53326341 EC50 = 13 nM T93788 C49ZMH 53390936 EC50 = 13 nM T93788 CHN72W 53469852 EC50 = 4 nM T93788 CP4AU5 53477048 EC50 = 13 nM T93788 CFT8B9 53477049 EC50 = 12 nM T93788 C5I8FB 53477155 EC50 = 16 nM T93788 CXE8V4 53477156 EC50 = 18 nM T93788 CO4S6E 53491642 EC50 = 8.6 nM T93788 C8XHK5 53491715 EC50 = 25.9 nM T93788 C3BFK2 53491780 EC50 = 65.1 nM T93788 C5HV3A 53491781 EC50 = 18.5 nM T93788 C8K0CB 53491782 EC50 = 31.1 nM T93788 C4OC7H 53492264 EC50 = 4.8 nM T93788 C16SZL 53492331 EC50 = 1.2 nM T93788 CGE8C9 53492397 EC50 = 62.6 nM T93788 CCE83O 53492463 EC50 = 54.8 nM T93788 CDQ2M4 53492467 EC50 = 16.1 nM T93788 CQK96E 53492528 EC50 = 8.5 nM T93788 CUJ76Z 53492593 EC50 = 262 nM T93788 C08XHA 53492594 EC50 = 5.9 nM T93788 CQUT71 53630395 EC50 = 11.6 nM T93788 C9K5GR 53630396 EC50 = 265 nM T93788 C1J8XI 53630398 EC50 = 6.3 nM T93788 C9M4QV 53630415 EC50 = 3.8 nM T93788 CEA18U 53630423 EC50 = 33.4 nM T93788 CRS4L7 53630450 EC50 = 14.6 nM T93788 C7EQT9 54580684 EC50 = 2580 nM T93788 CQWV19 54580747 EC50 = 5 nM T93788 C17ICO 54580903 EC50 = 526 nM T93788 CTJA61 54580904 EC50 = 48 nM T93788 C20FZY 54581118 EC50 = 3.4 nM T93788 C3IP1A 54581957 EC50 = 1400 nM T93788 CA37UQ 54581959 EC50 = 103 nM T93788 CDW8U1 54581961 EC50 = 62 nM T93788 C8CTD7 54581962 EC50 = 9 nM T93788 C7APK5 54582694 EC50 = 1150 nM T93788 CZ71VB 54582892 EC50 = 0.2 nM T93788 CZ6KG9 54583401 EC50 = 1239 nM T93788 CQ70UX 54583648 EC50 = 860 nM T93788 CCN3K0 54583892 EC50 = 600 nM T93788 C7GMD0 54583893 EC50 = 39 nM T93788 CL24JP 54583894 EC50 = 57 nM T93788 CG78OW 54583895 EC50 = 30 nM T93788 CSCE48 54583896 EC50 = 20 nM T93788 CY05QH 54584353 Ki = 20 nM T93788 CM1JT0 54584624 EC50 > 20000 nM T93788 CWBJ19 54584625 EC50 = 82 nM T93788 CL8MW9 54584841 EC50 = 76 nM T93788 CIVJ34 54585040 EC50 = 3.4 nM T93788 CR2OQ6 54585806 EC50 = 1900 nM T93788 CDK61R 54585807 EC50 = 11 nM T93788 CS2J3H 54585808 EC50 = 18 nM T93788 C3H6IN 54585809 EC50 = 13 nM T93788 CY4FD8 54586012 EC50 = 42 nM T93788 C64MJP 54586548 EC50 = 558 nM T93788 CEL6P0 54586563 EC50 = 130 nM T93788 CUZF70 54586564 EC50 = 918 nM T93788 C5CGF7 54586777 EC50 = 116 nM T93788 CK5ZC4 54586778 EC50 = 2 nM T93788 C6KS2N 54586779 EC50 = 19 nM T93788 C67NFK 54586780 EC50 = 19 nM T93788 C4ACJ8 54586781 EC50 = 2 nM T93788 CPO85I 54586882 EC50 = 7.5 nM T93788 C03XYL 54586987 EC50 = 7.3 nM T93788 CK3D9N 54587592 EC50 = 62 nM T93788 C39VDT 54587812 EC50 = 831 nM T93788 CZ5IY9 54587813 EC50 = 0.3 nM T93788 C1WZ4V 54589149 EC50 = 60 nM T93788 CO3C4B 54589151 EC50 = 62 nM T93788 C49WCU 54589190 EC50 = 544 nM T93788 CIYV57 54589191 EC50 = 1003 nM T93788 CO7F6Q 54589229 EC50 = 521 nM T93788 C73SNB 54589230 EC50 = 14 nM T93788 C2SNJ3 54589231 EC50 = 78 nM T93788 C8L1JO 54589232 EC50 = 51 nM T93788 C54UCK 54589269 EC50 = 16 nM T93788 C2SP3B 54589270 EC50 = 101 nM T93788 COJI15 54596144 EC50 = 13.7 nM T93788 C7QB1F 56591900 EC50 = 129 nM T93788 CKN41C 56592326 EC50 = 53 nM T93788 C2YXS6 56592327 EC50 = 41 nM T93788 CB2I9X 56592328 EC50 = 42 nM T93788 CF46NB 56592329 EC50 = 79 nM T93788 CMZ0G6 56592412 EC50 > 1000 nM T93788 CM0IL4 56592414 EC50 > 1000 nM T93788 CM1DB2 56592599 EC50 > 1000 nM T93788 C9ZF6B 56643412 EC50 = 74 nM T93788 C0MQ2W 56832511 EC50 = 24 nM T93788 CKC63L 56943106 EC50 = 23.4 nM T93788 C21XMN 56961034 EC50 = 353 nM T93788 C91JWV 56963355 EC50 = 27 nM T93788 CB5V4R 56963356 EC50 = 28.2 nM T93788 C3EL1T 57390603 EC50 = 260 nM T93788 C1C5TR 57390604 EC50 = 2330 nM T93788 CMF49J 57392378 EC50 = 235 nM T93788 CXL42B 57392379 EC50 = 60 nM T93788 CC75BU 57392380 EC50 = 60 nM T93788 C5E9UK 57392504 EC50 = 47 nM T93788 CZKU95 57393406 EC50 = 1410 nM T93788 COHW15 57394106 EC50 = 1000 nM T93788 C2A4UT 57394950 EC50 = 120 nM T93788 CBDV65 57397673 EC50 = 92 nM T93788 CWX87F 57397674 EC50 = 490 nM T93788 CU6O0S 57397675 EC50 = 210 nM T93788 CL0XS2 57397676 EC50 = 132 nM T93788 C8DJ9M 57399342 EC50 = 34 nM T93788 C89CRJ 57399343 EC50 > 5000 nM T93788 C4GXR6 57399344 EC50 = 25 nM T93788 C7HKF8 57399345 EC50 > 5000 nM T93788 CH6KB4 57401105 EC50 = 475 nM T93788 CI1SJ3 57401106 EC50 = 250 nM T93788 C6QIP7 57401198 EC50 = 1100 nM T93788 CBZ4C3 57402128 EC50 = 5.4 nM T93788 CD68KC 57402865 EC50 = 50 nM T93788 C7AGB4 57403665 EC50 = 115 nM T93788 C08QUG 57404926 EC50 = 3423 nM T93788 CYO3V8 57405092 EC50 = 14 nM T93788 CS5P8Y 57415237 EC50 = 100 nM T93788 C1TDX7 57468373 EC50 = 104 nM T93788 C7D5BO 57468382 EC50 = 117 nM T93788 CGI92M 57468398 EC50 = 31 nM T93788 CD7SN3 57468401 EC50 > 10000 nM T93788 C7T2OX 57468409 EC50 = 9 nM T93788 CFA0K6 57468427 EC50 = 5 nM T93788 CYX6F2 57468435 EC50 = 32 nM T93788 C12DVB 57468459 EC50 = 11 nM T93788 C7VF2J 57550042 EC50 = 18 nM T93788 CI63JT 57550050 EC50 = 870 nM T93788 CN4AZ7 57550070 EC50 = 41 nM T93788 C3ANB4 57550087 EC50 = 37 nM T93788 CGAF21 57550101 EC50 = 12 nM T93788 CT4XG6 58016984 EC50 = 79.43 nM T93788 C8Z2EV 58016989 EC50 = 50.12 nM T93788 CSX9K6 58016997 EC50 > 10000 nM T93788 C91ITW 58016999 EC50 = 630.96 nM T93788 CN4B6V 58017000 EC50 = 158.49 nM T93788 CS0B5T 58017005 EC50 = 316.23 nM T93788 CH1IX9 58017008 EC50 = 1995.26 nM T93788 CR3NF9 58017011 EC50 = 79.43 nM T93788 CE15RN 58017018 EC50 = 125.89 nM T93788 CPJD17 58017023 EC50 = 501.19 nM T93788 CSQ59A 58017025 EC50 = 100 nM T93788 CS7JH1 58017027 EC50 = 501.19 nM T93788 CTIP85 58017028 EC50 = 125.89 nM T93788 CX61OG 58017032 EC50 = 79.43 nM T93788 CZ2QA6 58017033 EC50 = 25.12 nM T93788 CU63JN 58017035 EC50 = 251.19 nM T93788 C9W8VD 58017036 EC50 = 79.43 nM T93788 C32MKS 58017038 EC50 = 158.49 nM T93788 CZE6U9 58017039 EC50 = 251.19 nM T93788 C84HGI 58017045 EC50 = 63.1 nM T93788 CZHW78 58017047 EC50 = 1000 nM T93788 CF86HB 58017059 EC50 = 398.11 nM T93788 C2LP9G 58074082 EC50 = 16 nM T93788 CKCV24 58114293 EC50 = 43.6 nM T93788 CO95HL 58116587 EC50 = 87 nM T93788 CDY74O 58116595 EC50 = 8800 nM T93788 C6L8YG 58190314 EC50 = 6 nM T93788 CH64EP 58190317 EC50 = 19.95 nM T93788 C7AY1J 58190324 EC50 = 12 nM T93788 C10KEY 58190329 EC50 = 63.1 nM T93788 CI63UA 58190330 EC50 = 20 nM T93788 CAGF43 58190343 EC50 = 64 nM T93788 C2L8TG 58190347 EC50 = 54 nM T93788 C3A4KQ 58190389 EC50 = 39 nM T93788 C5K1EG 58190395 EC50 = 2217 nM T93788 CA4G8T 58190401 EC50 = 234 nM T93788 C3PA2V 58190405 EC50 = 41 nM T93788 CON8B6 58190423 EC50 = 54 nM T93788 CB0V9M 59234074 EC50 = 353 nM T93788 CC1L3O 60152410 EC50 = 31 nM T93788 C5NW9S 60155096 EC50 = 1084 nM T93788 C0Z1NG 60155097 EC50 = 485 nM T93788 C84NFQ 60155098 EC50 > 30000 nM T93788 CHN8K5 60155099 EC50 = 186 nM T93788 C4YBX8 60155100 EC50 = 737 nM T93788 CQ34SH 60155182 EC50 > 7500 nM T93788 CU69NX 60155183 EC50 = 161 nM T93788 C7RYQ5 60155184 EC50 = 893 nM T93788 CI28PS 60155273 EC50 = 156 nM T93788 CXP75O 60155274 EC50 = 29 nM T93788 C9LGW7 60155364 EC50 = 79 nM T93788 C5F3JO 60155365 EC50 = 39 nM T93788 C4VJ1C 60155366 EC50 = 16 nM T93788 C18HZU 60155367 EC50 > 1937 nM T93788 CXA1Q4 60155457 EC50 = 63 nM T93788 CM3OX4 60155458 EC50 > 30000000 nM T93788 CG03LC 60155459 EC50 = 154 nM T93788 C6XG4H 60155460 EC50 = 184 nM T93788 C4TH9X 60155461 EC50 = 100 nM T93788 CL41YN 60155543 EC50 = 25 nM T93788 CX0PT7 62706030 EC50 = 51 nM T93788 CPR29D 62706192 EC50 = 210 nM T93788 CBR1J6 62706193 EC50 = 145 nM T93788 C6JZS7 62706349 EC50 = 270 nM T93788 C9QXO1 62706352 EC50 = 736 nM T93788 CN2XQ4 62706354 EC50 = 511 nM T93788 C13TEN 62706355 EC50 = 268 nM T93788 CLJ6A2 62706513 EC50 = 86 nM T93788 C2C4SU 62706514 EC50 = 770 nM T93788 C3P1WQ 62706516 EC50 = 550 nM T93788 CIB14P 62706517 EC50 = 1029 nM T93788 C53CKU 62706518 EC50 = 46 nM T93788 C8ALV4 62706691 EC50 = 272 nM T93788 CK6DX5 62706692 EC50 = 734 nM T93788 C9WVI6 62707006 EC50 = 58 nM T93788 CQ3R2L 66554587 EC50 = 505 nM T93788 C7KXP6 66554590 EC50 = 707 nM T93788 CJB58T 66554759 EC50 = 1030 nM T93788 CN62FS 66554760 EC50 = 38 nM T93788 C0S7TI 66554933 EC50 = 63 nM T93788 C80TYS 66556121 EC50 = 16 nM T93788 CL6E7G 66556122 EC50 = 57 nM T93788 C2TLX9 66556297 EC50 = 6.4 nM T93788 CKC76E 66556631 EC50 = 134 nM T93788 C4L7EO 66556985 EC50 = 42 nM T93788 C14BKV 66561292 EC50 = 33 nM T93788 CC6RH8 66574514 EC50 = 13.8 nM T93788 C7YQS4 66826123 EC50 = 100000000 nM T93788 CAS64Z 66963482 EC50 > 300 nM T93788 C0VD5C 66963512 EC50 = 20 nM T93788 CLB8H7 66963587 EC50 = 20 nM T93788 CFA02S 66963820 EC50 = 190 nM T93788 C41YUC 66963944 EC50 = 560 nM T93788 CBHA32 66963969 EC50 = 190 nM T93788 CCT84Y 66963996 EC50 = 4 nM T93788 CY8FU4 66964035 EC50 = 880 nM T93788 CM8X6G 66964040 EC50 = 3 nM T93788 CE10UM 66964044 EC50 = 170 nM T93788 CWA7I2 66964068 EC50 = 180 nM T93788 C6AU3Y 66964159 EC50 = 73 nM T93788 CI12ZB 66964172 EC50 = 243 nM T93788 CYB30V 66964174 EC50 = 1200 nM T93788 CXB50V 66964195 EC50 = 164 nM T93788 CB9U5D 66964295 EC50 = 10 nM T93788 CJQ0R1 66964459 EC50 = 86 nM T93788 CBP0V7 66964466 EC50 = 40 nM T93788 CE9DN2 66964510 EC50 = 11 nM T93788 CDO06R 66964555 EC50 = 1 nM T93788 CI4D3Q 66964595 EC50 > 10000 nM T93788 CM6QF7 66964599 EC50 = 40 nM T93788 CT2S3O 66964600 EC50 = 140 nM T93788 CH3KD5 66964621 EC50 = 290 nM T93788 CUI2X7 66964622 EC50 = 16 nM T93788 CR4O5S 66964658 EC50 = 340 nM T93788 CA6VM4 66964662 EC50 = 110 nM T93788 CG3WV5 66964682 EC50 = 1300 nM T93788 CWS5M3 66964756 EC50 = 130 nM T93788 CF35RW 66964802 EC50 = 62 nM T93788 CUA2J7 66964831 EC50 = 53 nM T93788 C1LY4J 66964852 EC50 = 63 nM T93788 CJ01UH 67449544 EC50 = 9.6 nM T93788 C73NJP 67449861 EC50 = 13 nM T93788 CGDH12 67449879 EC50 = 47 nM T93788 CQ4AN2 67450521 EC50 = 651 nM T93788 CO9M8S 67450901 EC50 = 427 nM T93788 C8OEN6 67450949 EC50 = 11 nM T93788 CFXC10 67451300 EC50 = 776 nM T93788 C20IRD 67606673 EC50 = 19.3 nM T93788 CG5E0I 67607375 EC50 = 15 nM T93788 CX45AB 67633261 EC50 = 2.78 nM T93788 CKHT83 67950429 EC50 = 5.32 nM T93788 CAT15Y 68021765 EC50 = 37 nM T93788 CHO94B 68021862 EC50 = 70 nM T93788 CXM35D 68021864 EC50 = 31 nM T93788 CUL1T2 68021959 EC50 = 21 nM T93788 C61YKH 68021978 EC50 = 52 nM T93788 CT1L6E 68022035 EC50 = 13 nM T93788 C7V0LF 68022196 EC50 = 63 nM T93788 C7AS8M 68022224 EC50 = 42 nM T93788 COG3A9 68022271 EC50 = 97 nM T93788 C95FCX 68036465 EC50 = 6 nM T93788 CI1DR8 68036798 EC50 = 49 nM T93788 C8L7PV 68036809 EC50 = 10 nM T93788 C2WJ4D 68036822 EC50 = 188 nM T93788 CZS1M5 68036918 EC50 = 26 nM T93788 C27XCG 68036931 EC50 = 10 nM T93788 CDM27X 68036951 EC50 = 19 nM T93788 CSE08J 68039954 EC50 = 4 nM T93788 C5WC9G 68040003 EC50 = 16 nM T93788 CCZ6Y5 68040038 EC50 = 7 nM T93788 CK21EZ 68040046 EC50 = 25 nM T93788 C0VHJ6 68211518 EC50 = 67 nM T93788 CVR1U4 68211526 EC50 = 82 nM T93788 C96SFV 68211777 EC50 = 5 nM T93788 COC2V7 68211779 EC50 = 78 nM T93788 CQ5X0V 68211781 EC50 = 122 nM T93788 COT43B 68211784 EC50 = 34 nM T93788 CIP2R1 68211791 EC50 = 2 nM T93788 C8SQA4 68211912 EC50 = 28 nM T93788 CY7NQ6 68211918 EC50 = 70 nM T93788 CF3VW9 68229751 EC50 = 52 nM T93788 CQPU67 68230018 EC50 = 36.8 nM T93788 CDPS39 68230201 EC50 = 8.3 nM T93788 CVA87O 68230212 EC50 = 3 nM T93788 CYV6B4 68230358 EC50 = 5.3 nM T93788 CA2YH5 68240224 EC50 = 70 nM T93788 C1TQ9C 68240419 EC50 = 7 nM T93788 CO8Z1E 68240486 EC50 = 51 nM T93788 CG3B4U 68299301 EC50 = 39 nM T93788 CU0A1F 68299305 EC50 = 240 nM T93788 CTQ78Y 68299308 EC50 = 1200 nM T93788 C14NSX 68385332 EC50 = 21 nM T93788 CN12IT 70680969 EC50 = 538 nM T93788 C0VEM7 70680970 EC50 = 441 nM T93788 CBE03K 70682125 EC50 = 254 nM T93788 C8D6ZB 70683088 EC50 > 30000 nM T93788 CKM4C2 70683089 EC50 = 1890 nM T93788 C7BPF4 70683090 EC50 = 29 nM T93788 CRTD40 70683091 EC50 = 29 nM T93788 CD0I2O 70684960 EC50 = 236 nM T93788 CKN95T 70685174 EC50 = 131 nM T93788 CUQ92A 70685175 EC50 = 172 nM T93788 CD7RB3 70687121 EC50 = 44 nM T93788 CY0N4S 70687331 EC50 = 122 nM T93788 C84GET 70687332 EC50 = 18 nM T93788 C6LN3I 70688972 EC50 = 78 nM T93788 CL68HK 70689385 EC50 = 1345 nM T93788 CBY8T6 70689386 EC50 = 53 nM T93788 CTJL92 70689387 EC50 = 485 nM T93788 CJY73E 70691486 EC50 = 456 nM T93788 CV8QT4 70691487 EC50 = 7 nM T93788 CJS34X 70692694 EC50 = 2610 nM T93788 CM4P5Z 70693582 EC50 = 489 nM T93788 CA9R2G 70693583 EC50 = 535 nM T93788 C35ASU 70693584 EC50 = 76 nM T93788 C8JUY5 70693585 EC50 = 396 nM T93788 CX0E3Y 70693586 EC50 = 12 nM T93788 C5T6JA 70695705 EC50 = 140 nM T93788 CG1XU6 70796891 EC50 = 17 nM T93788 C83TQO 70810684 EC50 = 200 nM T93788 CKP4O8 70855957 EC50 = 3.3 nM T93788 CLKU89 70856302 EC50 = 2 nM T93788 C2OH1E 71081343 EC50 = 142 nM T93788 CCXB25 71081352 EC50 = 56 nM T93788 C6DW7Q 71081378 EC50 > 1000 nM T93788 CTWH36 71081448 EC50 = 68 nM T93788 C2BND6 71081449 EC50 = 98 nM T93788 CY9IP1 71081450 EC50 = 46 nM T93788 CWC86N 71081517 EC50 = 369 nM T93788 C1XHA8 71116039 EC50 = 2.1 nM T93788 C4YJI5 71116044 EC50 = 1.1 nM T93788 C2M4CU 71116111 EC50 = 4.8 nM T93788 CWFL92 71116113 EC50 = 7.1 nM T93788 CI09HU 71128813 EC50 = 1.7 nM T93788 CDP0X1 71128816 EC50 = 3.1 nM T93788 CX15DJ 71134925 EC50 = 35 nM T93788 C4ZEN1 71135255 EC50 = 1.5 nM T93788 C6B2XM 71135993 EC50 = 47 nM T93788 C5AUY8 71136686 EC50 = 1.7 nM T93788 CY3N9S 71140721 EC50 = 2.5 nM T93788 CSEU81 71208589 EC50 = 2 nM T93788 CTQJ18 71208637 EC50 = 3 nM T93788 C2PSM5 71208866 EC50 = 3 nM T93788 CYK27V 71287378 EC50 = 386 nM T93788 CT51PO 71287404 EC50 = 103 nM T93788 C9OC0D 71450290 EC50 = 158.49 nM T93788 CZQE65 71452110 EC50 = 21 nM T93788 CRF56L 71453941 EC50 = 30 nM T93788 CLIA38 71455380 EC50 = 630.96 nM T93788 CF8EI7 71455832 EC50 = 2 nM T93788 C52GYP 71457626 EC50 = 228 nM T93788 C94UFY 71459020 EC50 > 10000 nM T93788 C1AS4O 71459320 EC50 = 93 nM T93788 CP32HG 71459321 EC50 = 398.11 nM T93788 CXZ79V 71461092 EC50 = 501.19 nM T93788 C7RH2E 71462834 EC50 = 800 nM T93788 C2AY8E 71462835 EC50 = 100 nM T93788 CKOZ97 71471638 EC50 = 82 nM T93788 CV78KN 71471711 EC50 = 3 nM T93788 CYT2N9 71471779 EC50 = 26 nM T93788 CAQ08G 71471851 EC50 = 781 nM T93788 C9JV4A 71474021 EC50 = 2.3 nM T93788 CW4UL3 71474456 EC50 = 8.7 nM T93788 CDO0M1 71491707 EC50 = 25 nM T93788 C3MK2J 71491755 EC50 = 67 nM T93788 CDR72Y 71519025 EC50 > 10000 nM T93788 C7CW1F 71519026 EC50 = 240 nM T93788 CJ29OT 71519027 EC50 = 462 nM T93788 C5LV7I 71519189 EC50 = 260 nM T93788 C9F2HA 71519190 EC50 = 864 nM T93788 CIRC04 71519192 EC50 = 83 nM T93788 C5L7YM 71519193 EC50 = 498 nM T93788 CZ0O9G 71524800 EC50 > 10000 nM T93788 C4E0UB 71524801 EC50 > 10000 nM T93788 C1GOB4 71524802 EC50 > 10000 nM T93788 CPC67E 71524845 EC50 > 10000 nM T93788 CX0HP2 71524846 EC50 > 10000 nM T93788 C62LOK 71524848 EC50 > 10000 nM T93788 CO2PS5 71524849 EC50 > 10000 nM T93788 CM2A0F 71531541 EC50 = 14 nM T93788 C34LHD 71545377 EC50 = 559 nM T93788 C3WM2U 71545378 Ki = 1970 nM T93788 C3KF1D 71545379 Ki = 586 nM T93788 C6HC8D 71545380 EC50 = 130 nM T93788 CGR96T 71545381 EC50 = 40 nM T93788 CK2R7U 71545535 EC50 = 88 nM T93788 CV15FW 71545536 EC50 = 145 nM T93788 C6JDU1 71545537 EC50 = 155 nM T93788 C09LAW 71545538 EC50 = 75 nM T93788 C3SB6R 71545698 EC50 = 40 nM T93788 CD9PH4 71545699 EC50 = 121 nM T93788 C87LNP 71545700 Ki = 131 nM T93788 CSP17W 71546032 Ki > 8148 nM T93788 C6C9MQ 71546033 Ki > 8148 nM T93788 C20IJM 71546034 EC50 = 164 nM T93788 CVQO13 71546035 EC50 = 49 nM T93788 CP9I5A 71546036 EC50 = 16 nM T93788 CMGZ54 71546198 Ki > 7318 nM T93788 CY7D8H 71546199 Ki = 814 nM T93788 C75OBG 71546200 EC50 = 691 nM T93788 CMX3O9 71546201 EC50 = 1028 nM T93788 C5GEA2 71546202 EC50 = 144 nM T93788 C5PS7U 71546701 EC50 = 274 nM T93788 C2GTU1 71546853 Ki = 133 nM T93788 C5E2DN 71546854 EC50 = 202 nM T93788 CVU95B 71546855 Ki = 94 nM T93788 C0K7MN 71546856 EC50 = 39 nM T93788 CUC38V 71546857 EC50 = 17 nM T93788 CZQ7I0 71547006 Ki = 18 nM T93788 CYG0K4 71547007 Ki = 15 nM T93788 CIL7K6 71547008 Ki = 7 nM T93788 CATD09 71547153 EC50 = 1049 nM T93788 CFO9U7 71562723 EC50 = 11.5 nM T93788 C4NYA9 71562724 EC50 = 1.5 nM T93788 C8SX0I 71562725 EC50 > 10000 nM T93788 CPDO92 71562726 EC50 = 6.7 nM T93788 C4IMF0 71562845 EC50 = 4.9 nM T93788 C0QF2W 71562846 EC50 = 1.4 nM T93788 CB2F3M 71573174 EC50 = 0.8 nM T93788 CFD8Y0 71617876 EC50 > 1000 nM T93788 CLV15A 71654936 EC50 = 8400 nM T93788 C7ZT6C 71654937 EC50 = 660 nM T93788 C73QOD 71654938 EC50 = 810 nM T93788 CSO8Q5 71654939 EC50 = 270 nM T93788 C6LB8Q 71654940 EC50 = 380 nM T93788 C0SL8O 71655012 EC50 = 960 nM T93788 C0CEI6 71655013 EC50 = 1600 nM T93788 CP5U6A 71655014 EC50 = 380 nM T93788 C1F7DV 71655015 EC50 = 440 nM T93788 C5U2SI 71655016 EC50 = 1710 nM T93788 CS5C9G 71655017 EC50 = 2120 nM T93788 CN1O2A 71655092 EC50 = 2060 nM T93788 C9F8JQ 71655093 EC50 = 13 nM T93788 CJ2C0H 71655094 EC50 = 130 nM T93788 CATY06 71655095 EC50 = 4000 nM T93788 CV3E0U 71655096 EC50 = 2740 nM T93788 C2KQM7 71655097 EC50 = 31 nM T93788 CRM32P 71655175 EC50 = 350 nM T93788 CNP0B9 71655176 EC50 = 2950 nM T93788 C3YWF0 71655177 EC50 = 610 nM T93788 C9FNO1 71655178 EC50 = 50 nM T93788 C40DNC 71655179 EC50 = 16 nM T93788 C7WPG4 71655180 EC50 = 160 nM T93788 CAKV27 71655250 EC50 = 450 nM T93788 C31RYO 71655251 EC50 = 91 nM T93788 C6MP4D 71655252 EC50 = 68 nM T93788 C73IXR 71655253 EC50 = 89 nM T93788 C38LKC 71655254 EC50 = 300 nM T93788 CUB71C 71655255 EC50 = 1060 nM T93788 C4LP8D 71655315 EC50 = 20 nM T93788 CC2E1S 71713968 EC50 = 45 nM T93788 CD19YH 71716097 Ki = 33 nM T93788 CV17DK 71716738 EC50 = 47 nM T93788 C8O5AK 71717057 EC50 > 10000 nM T93788 CO2B1U 71717058 EC50 > 10000 nM T93788 CC3L9V 71717059 EC50 = 1000 nM T93788 CM68ZB 71717312 Ki = 125 nM T93788 CUV09L 71717324 EC50 = 300 nM T93788 C57MSH 71717334 EC50 = 181 nM T93788 CHDN36 71717681 EC50 > 10000 nM T93788 CT02GM 71718289 EC50 = 1000 nM T93788 CH8J2D 71718290 EC50 > 10000 nM T93788 CGBW84 71718892 EC50 > 10000 nM T93788 CL28YO 71719746 Ki = 948 nM T93788 CZ7BL8 71720095 EC50 > 10000 nM T93788 CW4M7K 71720096 EC50 = 1000 nM T93788 CPMS07 71720493 EC50 = 38 nM T93788 C9F0ZD 71720494 EC50 = 15 nM T93788 C4OL0Q 71720750 EC50 > 10000 nM T93788 C68DRE 71720751 EC50 > 10000 nM T93788 C30NBJ 71722055 EC50 = 11 nM T93788 CP2EY7 72188621 EC50 = 20 nM T93788 CF9I2U 72945517 EC50 = 19 nM T93788 CZQL46 72945518 EC50 = 15 nM T93788 CH1DA7 72945519 EC50 = 121 nM T93788 CM7EQ0 72945706 EC50 = 23 nM T93788 CH3KN2 72945707 EC50 = 11 nM T93788 C4B3SM 72945708 EC50 = 13 nM T93788 CYE12L 72945709 EC50 = 69 nM T93788 C23YTU 72945710 EC50 = 299 nM T93788 CG28EU 72945711 EC50 = 19 nM T93788 CGV82Z 72945895 EC50 = 224 nM T93788 C64CUT 72945896 EC50 = 382 nM T93788 CT93UL 72945897 EC50 = 238 nM T93788 CF39JH 72945898 EC50 > 30000 nM T93788 CNEP39 72945899 EC50 = 11 nM T93788 CQD6X0 72945900 EC50 = 9 nM T93788 CK5F2R 72946091 EC50 = 33 nM T93788 COEL45 72946092 EC50 = 16 nM T93788 CQ0I8V 72946093 EC50 = 357 nM T93788 CZMF40 72946094 EC50 = 493 nM T93788 CGK87R 73348101 EC50 = 630.96 nM T93788 CNM19T 73348866 EC50 = 7 nM T93788 CEF4B6 73350444 IC50 = 1 nM T93788 C5ON3C 73351961 EC50 = 11 nM T93788 CA95TW 73353419 EC50 = 6 nM T93788 CG7R3F 73353420 IC50 = 8 nM T93788 CB9YC7 73354930 EC50 = 79 nM T93788 CS90NU 73354931 IC50 = 3 nM T93788 C46PFQ 73357217 EC50 = 50.12 nM T93788 CK9T1Y 76309728 EC50 = 18 nM T93788 C2FUH7 76309729 EC50 = 131 nM T93788 CJ2M6A 76309730 EC50 = 61 nM T93788 CHK8N4 76309731 EC50 = 37 nM T93788 C8GA1B 76309732 EC50 = 32 nM T93788 C7FA4M 76309733 EC50 = 44 nM T93788 CP98VM 76310374 EC50 = 190 nM T93788 CRF25S 76310375 EC50 = 80 nM T93788 CIC5H2 76310376 EC50 = 100 nM T93788 CLW2K8 76310377 EC50 = 590 nM T93788 CP2C1O 76310397 EC50 = 120 nM T93788 CG35AY 76310438 EC50 = 2600 nM T93788 CZMC38 76310439 EC50 = 8.4 nM T93788 CEUA45 76310440 EC50 = 25 nM T93788 CPN8X0 76310441 EC50 = 21 nM T93788 C9FHP1 76310464 EC50 = 520 nM T93788 CLM1B6 76313416 EC50 = 15 nM T93788 CBQN52 76314040 EC50 = 70 nM T93788 CBA5Y4 76314041 EC50 = 310 nM T93788 C2RBC6 76314042 EC50 = 30 nM T93788 C0BO3U 76314043 EC50 = 100 nM T93788 CSR01W 76314044 EC50 = 50 nM T93788 C71KTD 76314045 EC50 = 290 nM T93788 CC0T9X 76314046 EC50 = 550 nM T93788 CQZ42U 76314047 EC50 = 540 nM T93788 CEX20O 76314048 EC50 = 90 nM T93788 C5GX3R 76314049 EC50 = 100 nM T93788 C1Y7ST 76314096 EC50 = 770 nM T93788 C3WX7M 76314115 EC50 = 3.9 nM T93788 C6O9DC 76316923 EC50 = 30 nM T93788 CWY57O 76316924 EC50 = 30 nM T93788 CEKG37 76316925 EC50 = 330 nM T93788 CF2P0G 76316926 EC50 > 5000 nM T93788 CH4C1Q 76316927 EC50 = 112 nM T93788 CL1CQ3 76316928 EC50 = 2120 nM T93788 C7RMQ3 76316929 EC50 > 30000 nM T93788 C8HM5Q 76317599 EC50 = 140 nM T93788 CZE2C1 76317600 EC50 = 40 nM T93788 C6RSN9 76317666 EC50 = 4800 nM T93788 CMYI68 76317689 EC50 = 44 nM T93788 CF9YM4 76317690 EC50 = 490 nM T93788 CZAG95 76320654 EC50 = 24 nM T93788 C70EDY 76320655 EC50 = 15 nM T93788 CFP85B 76320656 EC50 = 166 nM T93788 CFH1N6 76320657 EC50 = 50 nM T93788 C92DQF 76320658 EC50 = 34 nM T93788 CG28EB 76320659 EC50 = 18 nM T93788 CSAO79 76321321 EC50 = 80 nM T93788 C1GY3S 76321322 EC50 = 50 nM T93788 C8JI2C 76321323 EC50 = 80 nM T93788 CH01KT 76321324 EC50 = 4300 nM T93788 CF3JM5 76321325 EC50 = 180 nM T93788 CX7LQ3 76321373 EC50 = 2400 nM T93788 CZM0K5 76324299 EC50 = 112 nM T93788 CN60XY 76324300 EC50 = 42 nM T93788 C9AG5H 76324301 EC50 = 54 nM T93788 CS6MC7 76324302 EC50 = 38 nM T93788 C0QNR4 76324928 EC50 = 110 nM T93788 CH8MK5 76324929 EC50 = 80 nM T93788 CWAX90 76324930 EC50 = 1500 nM T93788 C3JZU2 76324931 EC50 = 50 nM T93788 C6C5OD 76324932 EC50 = 270 nM T93788 CD0P3F 76324933 EC50 = 90 nM T93788 CA3O5D 76324934 EC50 = 70 nM T93788 C0K9BQ 76324949 EC50 > 30000 nM T93788 CAH91F 76324976 EC50 = 120 nM T93788 C3P5HT 76324977 EC50 = 25 nM T93788 C43DST 76324996 EC50 = 1700 nM T93788 C26MHI 76327867 EC50 = 24 nM T93788 CP3VI7 76327868 EC50 = 38 nM T93788 CRC1N8 76328493 EC50 = 180 nM T93788 CBM47D 76328494 EC50 = 60 nM T93788 CQC2W3 76328495 EC50 = 60 nM T93788 CA7T2L 76328496 EC50 = 30 nM T93788 CM83BG 76328497 EC50 = 80 nM T93788 CLT09R 76328549 EC50 = 530 nM T93788 CN82FC 76328564 EC50 = 6.8 nM T93788 CA8JB0 76331519 EC50 = 25 nM T93788 CM4QH5 76331520 EC50 = 7 nM T93788 CT0RW4 76331521 EC50 = 86 nM T93788 CQFZ48 76332169 EC50 = 130 nM T93788 C8BZ5R 76332170 EC50 = 100 nM T93788 CV76UF 76332171 EC50 = 320 nM T93788 C40DUR 76332172 EC50 = 90 nM T93788 CWBF71 76332173 EC50 = 770 nM T93788 CH23MG 76332174 EC50 = 860 nM T93788 C0H6SK 76332225 EC50 = 68 nM T93788 C0XJO8 76335131 EC50 = 18 nM T93788 CF6S7P 76335814 EC50 = 100 nM T93788 C3BNF9 76335815 EC50 = 60 nM T93788 C28FTZ 76335830 EC50 = 270 nM T93788 CRZ07L 76335866 EC50 = 1400 nM T93788 CLE6X0 76335867 EC50 = 2500 nM T93788 CT4XY9 76335868 EC50 = 160 nM T93788 C1KL8Q 76683707 EC50 = 55 nM T93788 CA6XJ7 76683708 EC50 = 14 nM T93788 C9Z1TP 76683709 EC50 = 9 nM T93788 CQX8U3 76683715 EC50 = 31 nM T93788 CQH2D6 76683814 EC50 = 78 nM T93788 C0EK4U 76683914 EC50 = 48 nM T93788 C1EBJ5 76683917 EC50 = 8 nM T93788 CDGL78 76684031 EC50 = 52 nM T93788 C10CNR 76684033 EC50 = 29 nM T93788 CWQF87 76684133 EC50 = 63 nM T93788 CL9JB3 86566993 EC50 = 716 nM T93788 CLO4Z6 86709924 EC50 = 7.91 nM T93788 CUW93G 86717800 EC50 = 4.5 nM T93788 C2FP3R 87217189 EC50 = 58 nM T93788 CER7N3 88567661 EC50 = 17 nM T93788 C83JRE 89583782 EC50 = 1.8 nM T93788 C1ZPE2 89583933 EC50 = 9.4 nM T93788 CU74LB 89584002 EC50 = 0.2 nM T93788 CBQ8J0 89584012 EC50 = 0.8 nM T93788 CR0P6K 89584034 EC50 = 0.2 nM T93788 C4NZW1 89584050 EC50 = 1.5 nM T93788 CZOJ21 89584118 EC50 = 0.7 nM T93788 CG29VI 90115611 EC50 = 4.2 nM T93788 C75OYT 90116115 EC50 = 3.2 nM T93788 C0A7DJ 90148901 EC50 = 4.5 nM T93788 CPE2L1 90656488 EC50 = 9000 nM T93788 C7CPS9 90656489 EC50 = 1100 nM T93788 CO03AL 90656490 EC50 > 10000 nM T93788 CC48DN 90656491 EC50 > 10000 nM T93788 CYF04H 90656492 EC50 > 10000 nM T93788 C2I8LO 90656529 EC50 = 541 nM T93788 C1X2PV 90665949 EC50 = 25.12 nM T93788 CKY18S 90665950 EC50 = 158.49 nM T93788 C31ZSK 90666908 EC50 = 100 nM T93788 CXKO79 90666909 EC50 = 630.96 nM T93788 C1JB5U 90666910 EC50 = 15.85 nM T93788 C9W6EJ 90666911 EC50 = 199.53 nM T93788 CE5J4N 90666912 EC50 = 199.53 nM T93788 CI02ZU 90666913 EC50 = 199.53 nM T93788 CTP5L0 90666914 EC50 = 501.19 nM T93788 C5DJT8 90666915 EC50 = 1258.93 nM T93788 CL54KY 90666916 EC50 = 1584.89 nM T93788 C80DYO 91824767 EC50 = 5 nM T93788 C21PRZ 102361261 EC50 = 54 nM T93788 C8ZM9J 117678530 EC50 = 0.4 nM T93788 C5CL8X 117684497 EC50 = 2.2 nM T93788 C2QPR5 118709765 EC50 = 173 nM T93788 CGQ8K4 118709767 EC50 = 1200 nM T93788 CXG4W7 118709768 EC50 = 140 nM T93788 CT5Y4F 118711210 EC50 = 132 nM T93788 CFND64 118711211 EC50 = 21 nM T93788 C1K7AS 118711212 EC50 = 13.6 nM T93788 C9VIB0 118711213 EC50 = 6.53 nM T93788 CHJQ06 118711214 EC50 = 92.9 nM T93788 CD9CK6 118711215 EC50 = 19.9 nM T93788 CRZY56 118711216 EC50 = 65.5 nM T93788 CON5I0 118711217 EC50 = 196 nM T93788 C29OWT 118711218 EC50 = 186 nM T93788 CVK7D2 118711219 EC50 = 9.2 nM T93788 C9U2WG 118711775 EC50 = 9.86 nM T93788 COP9C4 118711776 EC50 = 22 nM T93788 C0J2QH 118711777 EC50 = 326 nM T93788 CA21CR 118711778 EC50 = 14.3 nM T93788 CQS5M1 118711779 EC50 = 29.3 nM T93788 CTL50A 118711780 EC50 = 6.8 nM T93788 C65LOQ 118711781 EC50 = 4.83 nM T93788 CSL1I4 118711782 EC50 = 24.9 nM T93788 C09AEX 118711783 EC50 = 13.2 nM T93788 C27LYA 118711784 EC50 = 8.51 nM T93788 CDJ1I4 118711785 EC50 = 69.9 nM T93788 C8R6MZ 118711787 EC50 = 151 nM T93788 C2EH6Z 118711788 EC50 = 37 nM T93788 C65TWF 118711789 EC50 = 76.3 nM T93788 C02WJT 118711790 EC50 = 17.4 nM T93788 CHC73U 118711791 EC50 = 24.7 nM T93788 C7IF1L 118711792 EC50 = 72.8 nM T93788 CB67JI 118711793 EC50 = 761 nM T93788 C2QRV5 118711794 EC50 = 21.2 nM T93788 CM4R6H 118711795 EC50 = 14 nM T93788 CDO2R1 118711796 EC50 = 43.4 nM T93788 C9OZK0 118711797 EC50 = 4.7 nM T93788 C0RM8O 118711798 EC50 = 6.12 nM T93788 CJ3U7V 118715130 EC50 > 10000 nM T93788 CFES75 118715131 EC50 > 10000 nM T93788 C46OKY 118715132 EC50 > 10000 nM T93788 CG6C2I 118715133 EC50 > 10000 nM T93788 C9IPD5 118715134 EC50 > 10000 nM T93788 CV7I4Q 118715135 EC50 > 10000 nM T93788 CS6CW7 118720403 EC50 > 10 nM T93788 CQ6ND5 118720404 EC50 = 23 nM T93788 C96JBI 118720405 EC50 = 0.5 nM T93788 CJQ58U 118720406 EC50 = 38 nM T93788 C4Y0OG 118720407 EC50 = 2 nM T93788 CF7NW4 118720408 EC50 = 3 nM T93788 C6BP7I 118720409 EC50 = 8 nM T93788 CBT12E 118720410 EC50 = 74 nM T93788 CYC0Q6 118720411 EC50 = 101 nM T93788 C08BWN 118720412 EC50 = 3 nM T93788 CP95WQ 118720413 EC50 = 125 nM T93788 CEZK35 118720414 EC50 = 7 nM T93788 CP9JI8 118720415 EC50 = 20 nM T93788 CUNM53 118720416 EC50 = 11 nM T93788 CKX32F 118720417 EC50 = 25 nM T93788 CMX50B 118720418 EC50 = 34 nM T93788 C9BEO3 118720419 EC50 = 3 nM T93788 C0N4CQ 118720420 EC50 = 214 nM T93788 CM8F5R 118720421 EC50 = 73 nM T93788 CP2C9I 118720422 EC50 = 298 nM T93788 CG0VK4 118720423 EC50 = 2 nM T93788 C5CI4Z 118720424 EC50 = 436 nM T93788 CW50AC 118720425 EC50 = 21 nM T93788 C57HWX 118720426 EC50 = 15 nM T93788 C8XDH9 118720427 EC50 = 530 nM T93788 COB3W5 118720428 EC50 = 2 nM T93788 CVXN53 118720429 EC50 = 35 nM T93788 CP4SV0 118720430 EC50 = 20 nM T93788 CF87IO 118720431 EC50 = 2 nM T93788 CY6HT5 118720432 EC50 = 6 nM T93788 CPC71H 118722570 EC50 = 21 nM T93788 CTL19H 118722571 EC50 = 55 nM T93788 C2JGB3 118722572 EC50 = 10 nM T93788 CKD42B 118722573 EC50 = 133 nM T93788 C6PMQ1 118722574 EC50 = 150 nM T93788 C3ZL5Y 118722575 EC50 = 15 nM T93788 CR3UB2 118722576 EC50 = 7 nM T93788 CX1W8N 118722577 EC50 = 27 nM T93788 C49DXR 118722578 EC50 = 4 nM T93788 CW5GK1 118722579 EC50 = 58 nM T93788 C50GXM 118722580 EC50 = 158 nM T93788 CEI62G 118722581 EC50 = 4 nM T93788 C9UG3Z 118722582 EC50 = 8 nM T93788 C5XH4V 118722583 EC50 = 91 nM T93788 C6Q3RV 118722584 EC50 = 1102 nM T93788 CCWD82 118722585 EC50 = 4 nM T93788 CZ0DG2 118722586 EC50 = 18 nM T93788 CI3R9V 118722587 EC50 = 6 nM T93788 C6Z4FK 122184143 EC50 = 38.4 nM T93788 CP80EY 122184144 EC50 = 107 nM T93788 C4MZF8 122184145 EC50 = 48.8 nM T93788 CR9O1L 122184146 EC50 = 291 nM T93788 CZS80P 122184147 EC50 = 14 nM T93788 CHY08E 122184148 EC50 = 9.1 nM T93788 C07AXY 122184149 EC50 = 10.7 nM T93788 CQT12A 122184150 EC50 = 30.3 nM T93788 CP42FU 122184151 EC50 > 100000 nM T93788 CIB30N 122191630 EC50 = 3.3 nM T93788 CYI12O 122191631 EC50 = 2.4 nM T93788 CW1NI3 122191632 EC50 = 1.7 nM T93788 C5GRC3 122191633 EC50 = 0.8 nM T93788 CCTM93 122194337 EC50 = 17 nM T93788 C9MBL0 122194338 EC50 = 44 nM T93788 C7C4WK 122194339 EC50 = 65 nM T93788 CXAK04 122194420 EC50 = 5 nM T93788 CXV30P 122194421 EC50 = 268 nM T93788 C0DFN8 127048479 EC50 = 177 nM T93788 CIC9S6 127048480 EC50 = 266 nM T93788 CQL9H0 127048481 EC50 = 197 nM T93788 CRY0I8 127048482 EC50 = 27 nM T93788 CW09RY 127048491 EC50 = 46 nM T93788 C97SDN 127048492 EC50 = 10 nM T93788 CHT2M6 127048493 EC50 = 14 nM T93788 CQIB34 127048494 EC50 = 92 nM T93788 C2V1CS 127048495 EC50 = 11 nM T93788 CP7Y0X 127048787 EC50 = 20 nM T93788 C0XV9A 127048820 EC50 = 23 nM T93788 CP6C2G 127048821 EC50 = 30 nM T93788 CX7K0M 127048822 EC50 = 220 nM T93788 CK1R4X 127050518 EC50 = 10 nM T93788 C0EN7J 127050519 EC50 = 4 nM T93788 C04MCY 127050520 EC50 = 15 nM T93788 C5DA9S 132486941 EC50 = 65 nM T93788 CY4FW5 134131905 EC50 = 1.3 nM T93788 CMY0V5 134132485 EC50 = 1900 nM T93788 C1T4DP 134134925 EC50 > 2000 nM T93788 C6R3US 134135618 EC50 = 1.6 nM T93788 CVE5Z8 134136399 EC50 = 0.6 nM T93788 CTZ0Y6 134136992 EC50 = 44.2 nM T93788 CRL94F 134137238 EC50 > 2000 nM T93788 C6UXF4 134138752 EC50 = 6.2 nM T93788 CY2HZ6 134139363 EC50 > 2000 nM T93788 C1JF9T 134139552 EC50 > 2000 nM T93788 CY9RM8 134142930 EC50 = 1.5 nM T93788 CFG3B4 134146906 EC50 > 2000 nM T93788 C9KWZ2 134147816 EC50 = 3.5 nM T93788 CZSA25 134147992 EC50 = 1.5 nM T93788 C8ALS5 134150100 EC50 > 2000 nM T93788 C0G5PV 134151859 EC50 = 950 nM T93788 C5U4GE 134152907 EC50 = 205 nM T93788 C4XS1N 134156472 EC50 > 2000 nM T93788 C3MU5V 134156958 EC50 = 1.4 nM T93788 CIRH31 137631474 EC50 = 61 nM T93788 CF8W4G 137631845 EC50 = 4.9 nM T93788 CCM7B3 137632132 EC50 = 5.6 nM T93788 C2B8YF 137632493 EC50 = 98 nM T93788 CINX05 137632674 EC50 = 48.2 nM T93788 C8J9AS 137632950 EC50 = 9 nM T93788 CF9QR4 137632997 EC50 = 171 nM T93788 CW9R5V 137633747 EC50 = 10 nM T93788 C3BCO0 137633771 EC50 = 252 nM T93788 C6PU4J 137634756 EC50 = 793 nM T93788 CV5E4H 137634873 EC50 = 3.1 nM T93788 CT72HP 137635337 EC50 = 310 nM T93788 CY10HA 137637825 EC50 = 5.6 nM T93788 C50UHW 137637873 EC50 = 27 nM T93788 CNI5D0 137637925 EC50 = 199 nM T93788 C9P7HM 137637929 EC50 = 18 nM T93788 CJX6U4 137638009 EC50 = 155 nM T93788 C78HPO 137638017 EC50 = 73 nM T93788 CGA3P4 137638546 EC50 > 10000 nM T93788 CWYG89 137639896 EC50 = 60 nM T93788 CM3VF9 137639995 EC50 = 92 nM T93788 CEYK56 137641046 EC50 = 39 nM T93788 C7K9VU 137642901 EC50 = 586 nM T93788 CYOZ07 137642936 EC50 = 64 nM T93788 CHA47F 137643188 EC50 = 19 nM T93788 CQ5DI1 137643239 EC50 = 67 nM T93788 C7AJG1 137643726 EC50 = 77 nM T93788 C7SH2E 137643838 EC50 = 315 nM T93788 C4EMC3 137643882 EC50 = 321 nM T93788 CH1P4Y 137643950 EC50 > 1000 nM T93788 CUGP54 137645678 EC50 = 391 nM T93788 CV4H9N 137645720 EC50 = 110 nM T93788 CB8CX4 137647821 EC50 = 82 nM T93788 CY7OR0 137648824 EC50 = 105 nM T93788 CEYZ80 137648888 EC50 = 201 nM T93788 C7BXJ2 137649810 EC50 = 1.8 nM T93788 CJVM79 137650572 EC50 = 53 nM T93788 C4F9GB 137651939 EC50 = 83 nM T93788 CHQI31 137651954 EC50 = 512 nM T93788 C3QD8P 137651958 EC50 = 2 nM T93788 C0E5FI 137653591 EC50 = 77.7 nM T93788 CPR76C 137655251 EC50 = 7 nM T93788 C97RZV 137655380 EC50 = 319 nM T93788 C1W9SE 137656527 EC50 = 53 nM T93788 CU9KZ4 137656911 EC50 = 15 nM T93788 CMF10H 137656947 EC50 = 78 nM T93788 CL9VW3 137657254 EC50 = 156 nM T93788 CNE31G 137659062 EC50 = 18 nM T93788 CS6G8H 137659500 EC50 = 1.2 nM T93788 CTK8D1 137660158 EC50 = 67 nM T93788 CI7Q4L 137660484 EC50 = 57 nM T93788 C1BXZ4 137660724 EC50 = 83 nM T93788 C7L5MD 137661403 EC50 = 13 nM T93788 C30NUT 137661559 EC50 = 33 nM T93788 CW1VR8 139436992 EC50 = 12 nM T93788 C9MX3E 139437014 EC50 = 4920 nM T93788 CB5Q2E 139437017 EC50 = 57 nM T93788 CO7T8R 139437037 EC50 = 458 nM T93788 CLO92I 139437040 EC50 = 82 nM T93788 C6BW7F 139437096 EC50 = 324 nM T93788 C0KI5D 140251500 EC50 = 31 nM T93788 CAE54O 140251501 EC50 = 13 nM T93788 CQA4W0 140251511 EC50 = 23 nM T93788 C2K4QW 140251527 EC50 = 40 nM T93788 CA5CF8 140251528 EC50 = 18 nM T93788 CU2ND3 140251533 EC50 = 34 nM T93788 C2VA1I 140253894 EC50 = 101 nM T93788 C8Z2XA 140253895 EC50 = 128 nM T93788 CT6D1A 140253898 EC50 = 17 nM T93788 CNQ53I 140254089 EC50 = 235 nM T93788 C8T6NF 140254101 EC50 = 169 nM T93788 CING28 144479903 EC50 = 334 nM T93788 C2OX1H 145949313 EC50 = 5.1 nM T93788 C0M3YQ 145949889 EC50 = 97 nM T93788 CYOH06 145951687 EC50 = 212 nM T93788 CQX3I6 145955539 EC50 = 13 nM T93788 CWIC73 145957126 EC50 = 10 nM T93788 CKW4D7 145959739 EC50 = 3.5 nM T93788 CJD7L6 145962089 EC50 = 6 nM T93788 CJF21C 145963524 EC50 = 8 nM T93788 CPL94Z 145964295 EC50 = 21 nM T93788 C1YM2B 145964891 EC50 = 82 nM T93788 C85JQK 145964999 EC50 = 211 nM T93788 CH6R3O 145965514 EC50 = 182 nM T93788 C4ZM3X 145966434 EC50 = 100 nM T93788 C6SX5I 145966749 EC50 = 7 nM T93788 CZ1IP0 145967361 EC50 = 18 nM T93788 C4ZTN9 145967591 EC50 = 225 nM T93788 CT0WU8 145967680 EC50 = 830 nM T93788 CZKG72 145968038 EC50 = 1.995 nM T93788 CTI20V 145968103 EC50 = 2388 nM T93788 CF61IA 145968330 EC50 = 123 nM T93788 C7UK3H 145968709 EC50 = 49 nM T93788 CJ0KF3 145968993 EC50 = 2590 nM T93788 CIB03W 145969583 EC50 = 154 nM T93788 CSUM19 145969910 EC50 = 5.012 nM T93788 CB23AP 145970094 EC50 = 511 nM T93788 CFO6S8 145970276 EC50 = 19 nM T93788 CC5I3B 145970536 EC50 = 157 nM T93788 CU3PZ7 145970589 EC50 = 348 nM T93788 C8VGL2 145971166 EC50 = 183 nM T93788 C5HW3K 145971825 EC50 = 88 nM T93788 C1RCP7 145972319 EC50 = 10 nM T93788 CA31ZR 145973091 EC50 = 14 nM T93788 CCT96L 145973632 EC50 = 2.6 nM T93788 C0VY7G 145974170 EC50 = 95 nM T93788 C3KXP2 145975486 EC50 = 5 nM T93788 CPD46L 145975897 EC50 = 240 nM T93788 CQ2H6F 145976125 EC50 = 4 nM T93788 CS15QM 145976269 EC50 = 29 nM T93788 C3A5RU 145976366 EC50 = 27 nM T93788 CR42QN 145977018 EC50 = 4 nM T93788 C1CF9N 145978481 EC50 = 209 nM T93788 CFXA96 145978767 EC50 = 78 nM T93788 CV21OC 145978800 EC50 = 780 nM T93788 C8WE1P 145982637 EC50 = 8.1 nM T93788 C3ILT5 145983137 EC50 = 36 nM T93788 CPS7J2 145983474 EC50 = 44 nM T93788 CAR8P2 145983613 EC50 = 1000 nM T93788 CV06WH 145983959 EC50 > 10000 nM T93788 CS3V1K 145983970 EC50 = 3200 nM T93788 C2FZP3 145984093 EC50 = 2.2 nM T93788 CT8R0W 145984643 EC50 = 126 nM T93788 CHX51B 145985013 EC50 = 179 nM T93788 CN9B7H 145985036 EC50 = 2100 nM T93788 CQW14Z 145985107 EC50 = 345 nM T93788 CG97IV 145986139 EC50 = 49 nM T93788 C4L2EY 145986191 EC50 = 147 nM T93788 C7J6XS 145986357 EC50 = 25.12 nM T93788 C7GK3H 145990715 EC50 > 100000 nM T93788 CEA10I 145993111 EC50 = 321 nM T93788 CA8HW6 145993236 EC50 = 360 nM T93788 CM25YZ 155511104 EC50 = 4.21 nM T93788 C4HCA5 155513850 EC50 = 3.12 nM T93788 CV68IT 155514874 EC50 = 64 nM T93788 CCT2U1 155514929 EC50 = 29 nM T93788 CCA49B 155515010 EC50 = 44 nM T93788 C1XLC0 155515632 EC50 = 98 nM T93788 CVM52W 155516183 EC50 = 2457 nM T93788 CIT8G6 155517437 EC50 = 139 nM T93788 CM2F9X 155517636 EC50 = 8.78 nM T93788 C2XQY5 155521067 EC50 = 7 nM T93788 CK02AF 155522754 EC50 = 85 nM T93788 CCP59K 155523981 EC50 = 13.98 nM T93788 C03QFB 155524213 EC50 = 86 nM T93788 C24HCO 155525761 EC50 = 12.34 nM T93788 C5E1PD 155525764 EC50 = 31 nM T93788 CIP62K 155525822 EC50 = 7.12 nM T93788 C62FVA 155527157 EC50 = 25 nM T93788 CGP1Y7 155528031 EC50 = 15 nM T93788 C5OQV0 155528272 EC50 = 12.31 nM T93788 CQA30H 155528891 EC50 = 12.43 nM T93788 CDOI91 155530128 EC50 = 59 nM T93788 C70MHT 155530371 EC50 = 13.56 nM T93788 C2FO7T 155531204 EC50 = 261 nM T93788 CQ1OH3 155531494 EC50 = 5 nM T93788 CPH54I 155532104 EC50 = 301 nM T93788 CQ1F0P 155532657 EC50 = 89 nM T93788 CH6XR0 155532730 EC50 = 42 nM T93788 CYKT59 155534233 EC50 = 13 nM T93788 CU48LF 155536150 EC50 = 11.12 nM T93788 CCH57L 155537620 EC50 = 3.67 nM T93788 CYP63K 155537900 EC50 > 1000 nM T93788 C3PWV4 155538381 EC50 = 69 nM T93788 CEVC80 155538763 EC50 = 27 nM T93788 CF72OA 155539620 EC50 = 27 nM T93788 C7IMF1 155541499 EC50 > 1000 nM T93788 CS40NT 155542312 EC50 = 8.17 nM T93788 CGP4Z6 155544367 IC50 = 4620 nM T93788 CH25ZD 155549064 EC50 = 6 nM T93788 C16QAN 155550456 EC50 = 720 nM T93788 CQ14SC 155551991 EC50 = 33 nM T93788 CWP6G5 155553659 EC50 = 16 nM T93788 C2CD7U 155564944 EC50 = 426 nM T93788 CX7G8Q 155565475 EC50 = 3.59 nM T93788 CRV9Y2 155566096 EC50 = 430 nM T93788 CSK6A1 155566114 EC50 = 5 nM T93788 CAP48C 155567012 EC50 = 45 nM T93788 CX4O7N 155568284 EC50 = 10.43 nM T93788 CMC2A9 155568311 EC50 = 19 nM T93788 CSZ7N9 155569398 EC50 = 39 nM T93788 D00GTC 5332859 EC50 = 2500 nM T93788 D01GPC 53235534 EC50 = 4 nM T93788 D01VZL 11462546 EC50 = 1900 nM T93788 D06QYM 51346816 EC50 = 80 nM T93788 D07MBC 5283454 EC50 = 2200 nM T93788 D08HOK 11282871 EC50 = 1.1 nM T93788 D09ROS 54582152 EC50 = 0.6 nM T93788 D0I2EL 53630394 EC50 = 0.9 nM T93788 D0R5QF 24939268 EC50 = 0.65 nM T93788 D0VA7C 54580880 EC50 = 3600 nM T93788 D0X3NW 53630410 EC50 = 0.5 nM T50688 D07XHO 4413 IC50 = 12000 nM T50688 D09ZIO 448812 IC50 = 570 nM T50688 D0BN9X 60947 IC50 = 0.37 nM T50688 D0GY5Z 2244 IC50 = 5000 nM T50688 D01TJY 53340771 IC50 > 10 nM T50688 D09ZXO 176873 IC50 = 590 nM T50688 D0Q5LF 9961766 IC50 > 100000 nM T50688 D00VAJ 178080 IC50 = 2.38 nM T50688 D01QQM 3038484 IC50 = 1.4 nM T50688 D02VIP 9955461 Ki = 3300 nM T50688 D03GCN 9885190 IC50 = 25 nM T50688 D03QHI 9933077 IC50 = 0.4 nM T50688 D05JXR 9805266 IC50 = 72 nM T50688 D06LGC 9906649 IC50 = 50 nM T50688 D07EXV 60957 IC50 = 2 nM T50688 D08CQL 164393 Ki = 2 nM T50688 D08LIG 153986 IC50 > 3 nM T50688 D0B9SR 9868426 Ki = 3800 nM T50688 D0C7JH 6918252 IC50 = 29 nM T50688 D0D7GE 9824171 IC50 = 0.49 nM T50688 D0H1PN 9955286 IC50 = 4.7 nM T50688 D0I7EU 9827266 Ki = 1.6 nM T50688 D0K0NP 9812185 IC50 = 12 nM T50688 D0LK9N 66000 IC50 = 80 nM T50688 D0LT1S 9823503 Ki = 30000 nM T50688 D0M6YE 44343680 Ki = 175 nM T50688 D0N0BI 5491394 IC50 = 1.14 nM T50688 D0P8JX 177831 IC50 = 32 nM T50688 D0S3RB 216230 IC50 = 0.06 nM T50688 D0SV7D 80274 IC50 = 28 nM T50688 D0U4ZY 10031011 IC50 = 6 nM T50688 D0U6BB 44343739 IC50 = 94 nM T50688 D0W4OL 132814 IC50 = 88 nM T50688 D0Y0AP 173614 IC50 = 7.943 nM T50688 D0Z0XQ 44343754 IC50 = 30 nM T50688 D0Z9LD 9804438 IC50 = 1600 nM T50688 C7CL3Y 107775 IC50 = 7900 nM T50688 CE19HD 132605 IC50 = 1700 nM T50688 C0XC5J 164450 IC50 = 120 nM T50688 C81ZQR 164519 IC50 = 30 nM T50688 CFQU71 177231 IC50 = 0.25 nM T50688 C5HE6N 446808 IC50 = 12500 nM T50688 CE5LI6 448813 IC50 = 19 nM T50688 C7M9QB 756604 IC50 = 9600 nM T50688 C2E9ZX 3080994 IC50 = 31 nM T50688 CJ2PE8 3081210 Ki = 4200 nM T50688 CY7WS4 9799158 IC50 = 1000 nM T50688 CU7VY5 9800226 IC50 = 8500 nM T50688 C2ST5A 9801767 IC50 = 6 nM T50688 CS40VO 9802158 IC50 = 5500 nM T50688 C86OSU 9802663 IC50 > 10000 nM T50688 CH19JX 9804758 IC50 > 10000 nM T50688 C3OYQ7 9805923 IC50 = 0.068 nM T50688 CNM8S0 9806690 IC50 = 40000 nM T50688 CBJ9Q5 9807152 IC50 = 2.3 nM T50688 C68UYS 9808123 IC50 = 380 nM T50688 CH05GX 9809459 Ki < 1 nM T50688 C8Z1BK 9818983 IC50 = 8300 nM T50688 C5UOC7 9819970 IC50 = 200 nM T50688 CJ75TL 9821561 IC50 = 115 nM T50688 C19PBH 9821600 IC50 = 3.9 nM T50688 CO2Z6V 9822136 Ki = 28000 nM T50688 C4TA8N 9823909 Ki = 4 nM T50688 C4LTP2 9825687 IC50 = 23.8 nM T50688 CO73TV 9825696 IC50 = 25.3 nM T50688 C3B7WM 9825804 IC50 = 0.1 nM T50688 CLR39O 9826223 IC50 = 10 nM T50688 CFZP14 9826756 IC50 = 0.25 nM T50688 C6DLN9 9827351 IC50 = 6.1 nM T50688 CQ25XG 9827352 IC50 = 0.0058 nM T50688 C7I0XB 9827873 IC50 = 22 nM T50688 CB8GP1 9828375 IC50 = 0.31 nM T50688 CJ9HV0 9828819 IC50 = 0.16 nM T50688 C1OP9I 9828979 IC50 = 9800 nM T50688 CR8OB5 9829206 Ki = 2.3 nM T50688 CA1XU5 9842047 IC50 = 2 nM T50688 CTDP48 9843636 IC50 = 688 nM T50688 C7L0QF 9844010 IC50 = 125.89 nM T50688 C1SJR6 9844061 IC50 = 138 nM T50688 C31UCL 9844289 Ki = 30000 nM T50688 C25SWU 9844694 IC50 = 113 nM T50688 C0L7UV 9845476 IC50 = 22000 nM T50688 CPK21J 9845731 IC50 = 42 nM T50688 CZ0AS2 9846634 IC50 = 965 nM T50688 CY63LZ 9846660 IC50 = 533 nM T50688 CG0H4P 9847624 IC50 > 10000 nM T50688 C13KPA 9848051 Ki < 10000 nM T50688 CAR4I2 9849008 IC50 > 10000 nM T50688 C12AFP 9849392 IC50 = 35 nM T50688 C13OZW 9850433 IC50 = 0.78 nM T50688 CTM7V0 9851337 IC50 = 257 nM T50688 C2XD7P 9851886 IC50 > 100000 nM T50688 CCUK35 9853139 IC50 = 5 nM T50688 CR38MP 9853559 IC50 = 34700 nM T50688 CEAF74 9858710 IC50 = 32466 nM T50688 C6E3OL 9863046 Ki = 0.0465 nM T50688 C7SME4 9863277 IC50 = 110 nM T50688 CR0D9E 9864936 IC50 = 36 nM T50688 C0G1XS 9865309 IC50 = 439 nM T50688 CS4T0P 9865840 IC50 = 153 nM T50688 CZC31S 9867414 IC50 = 46 nM T50688 CR7T6A 9868824 IC50 = 105 nM T50688 CP4U2K 9869048 IC50 > 10000 nM T50688 CPKL80 9869692 IC50 > 100000 nM T50688 C2ZAK6 9870468 IC50 > 400000 nM T50688 CHC56Q 9870640 IC50 = 0.3 nM T50688 C9KN3Q 9872164 IC50 = 0.21 nM T50688 C31WAF 9872696 IC50 = 240 nM T50688 C48OAX 9872930 IC50 = 6 nM T50688 C3JA4P 9884008 IC50 = 270 nM T50688 C5EJN9 9884317 IC50 > 20000 nM T50688 C1RP4J 9884941 IC50 = 20 nM T50688 CV4T6H 9885053 IC50 > 20000 nM T50688 CJ5Z0U 9885197 IC50 = 43 nM T50688 C13WGE 9886306 IC50 > 10000 nM T50688 C1EQN3 9888685 IC50 = 104 nM T50688 C6ODX3 9888704 IC50 = 23000 nM T50688 C7B3KI 9893323 IC50 = 8 nM T50688 C49EQN 9893755 IC50 = 11 nM T50688 C6PNG8 9894403 IC50 = 3200 nM T50688 C1ZWO4 9904909 IC50 = 13 nM T50688 CNX29T 9907082 IC50 = 9 nM T50688 CMU27A 9907178 IC50 = 76 nM T50688 C2DTH6 9907685 IC50 = 1.9 nM T50688 CC6PJ4 9908437 Ki > 10000 nM T50688 CVK15W 9908440 IC50 = 15 nM T50688 C43TPN 9910543 IC50 > 10000 nM T50688 C25HTY 9910653 IC50 = 10000 nM T50688 CE34GC 9910784 IC50 = 2.7 nM T50688 CR9C5Z 9911060 Ki > 50000 nM T50688 CD7I4Y 9911639 Ki = 9000 nM T50688 CV97OQ 9912737 Ki = 0.17 nM T50688 CBZ20D 9913337 IC50 = 0.0013 nM T50688 CR13IL 9914166 IC50 > 1000 nM T50688 COT86Q 9915619 IC50 = 21 nM T50688 C69XAB 9916695 IC50 = 1300 nM T50688 CF4J2Z 9923982 IC50 > 20000 nM T50688 CUBV32 9924032 IC50 > 20000 nM T50688 CCPD70 9927009 IC50 = 1.1 nM T50688 C40MDV 9927904 IC50 = 39 nM T50688 CTNI30 9929455 IC50 = 196 nM T50688 CJPZ87 9930471 IC50 = 4360 nM T50688 CR5N6D 9931153 IC50 = 18 nM T50688 CODI28 9932234 IC50 = 0.016 nM T50688 CC42WD 9932423 IC50 = 1800 nM T50688 CT6S7L 9933202 IC50 = 6000 nM T50688 CMJ76L 9936566 IC50 = 27000 nM T50688 CP8IO3 9941178 IC50 = 10100 nM T50688 C3G5RK 9941719 IC50 = 4100 nM T50688 CUC31Q 9950075 IC50 > 50000 nM T50688 CN2Y5D 9950151 IC50 = 33 nM T50688 CLA39Q 9950422 IC50 = 600 nM T50688 C1UK7T 9953715 Ki = 36000 nM T50688 CDQ17J 9953718 IC50 = 10 nM T50688 CYG4S2 9954358 IC50 > 10000 nM T50688 C9CKS6 9956141 IC50 = 263 nM T50688 C4XK2S 9956830 IC50 = 170 nM T50688 CDU79H 9957105 IC50 = 0.59 nM T50688 CH1Y7E 9957565 IC50 = 80 nM T50688 CGP18L 9957723 IC50 = 43 nM T50688 C3VWH1 9957860 IC50 = 21.88 nM T50688 CWUC80 9958350 Ki = 128 nM T50688 C2EX4U 9972378 IC50 = 24000 nM T50688 C3PYH6 9975679 IC50 = 10000 nM T50688 C2QOL4 9978473 IC50 = 580 nM T50688 C9M2JU 9978549 IC50 = 213 nM T50688 CUIF89 9979634 IC50 = 150 nM T50688 CIXB62 9979842 IC50 > 3000 nM T50688 C9PL2H 9980010 IC50 = 740 nM T50688 C26PYH 9980810 IC50 = 59000 nM T50688 CW2ZR6 9982004 IC50 = 15 nM T50688 CXN45H 9983052 IC50 = 14000 nM T50688 CS9QB2 9983098 Ki = 3 nM T50688 CYA0W2 9983143 IC50 = 95.1 nM T50688 CPE58N 9984136 IC50 > 3000 nM T50688 CV2D0B 9984142 IC50 = 44 nM T50688 CS9VD0 9984206 IC50 = 8 nM T50688 C81DKG 9993820 IC50 = 35000 nM T50688 CN3EO0 9994930 IC50 = 5800 nM T50688 CLB29G 9996802 IC50 = 20 nM T50688 CY94QV 9999236 IC50 = 74 nM T50688 CI1HJ3 10002632 IC50 = 108 nM T50688 C6CWQ8 10003119 IC50 = 2004 nM T50688 CEJ78G 10004109 IC50 = 880 nM T50688 CV0G6H 10004443 IC50 = 18 nM T50688 C24MDH 10022569 IC50 = 3800 nM T50688 C7UZI3 10024672 IC50 = 8000 nM T50688 CBT02G 10026044 IC50 = 6610 nM T50688 CEC9V5 10026930 IC50 = 61 nM T50688 CEJ31C 10027119 IC50 = 484 nM T50688 CGT4D2 10027594 IC50 = 10882 nM T50688 CZ47BK 10027732 IC50 = 1170 nM T50688 C5CZ8A 10028351 IC50 > 10000 nM T50688 C06INP 10029120 IC50 = 37 nM T50688 CY0T9L 10030149 IC50 = 278 nM T50688 C0SU3C 10031320 IC50 = 290 nM T50688 CE2CK1 10032445 IC50 > 100000 nM T50688 CR2F8U 10043404 IC50 = 48 nM T50688 CKYE52 10044478 IC50 = 320 nM T50688 CW9O1B 10045567 IC50 = 10000 nM T50688 CPM36N 10045699 IC50 = 302 nM T50688 C6ZM5H 10047912 IC50 = 35 nM T50688 CGA89W 10049569 IC50 > 10000 nM T50688 C27XYG 10050154 IC50 = 70000 nM T50688 C86AUR 10050355 IC50 = 1100 nM T50688 CD6SV4 10050710 IC50 = 2400 nM T50688 CLS1F7 10051002 IC50 = 65.4 nM T50688 COH3U6 10052945 IC50 = 57.6 nM T50688 C89RLI 10067208 IC50 = 79 nM T50688 C40FMW 10069462 IC50 = 330 nM T50688 C2R7TW 10069591 IC50 = 780 nM T50688 CM5PL6 10069800 IC50 = 47 nM T50688 C3WZR0 10069974 IC50 = 1200 nM T50688 C7UNJ1 10071004 IC50 = 0.061 nM T50688 C25GLI 10072571 IC50 = 100 nM T50688 CFSU38 10073745 IC50 = 2 nM T50688 CK0G2T 10073952 IC50 = 350 nM T50688 CH0Y4Z 10074600 IC50 = 1470 nM T50688 C7C6FP 10074635 Ki = 1.5 nM T50688 C4AW6G 10075410 IC50 = 7 nM T50688 C6B7OI 10087503 IC50 = 18000 nM T50688 CT4O8V 10092389 IC50 = 36000 nM T50688 CO8J9N 10093461 IC50 = 158 nM T50688 C67KRY 10094447 IC50 = 54 nM T50688 CV83XM 10095387 IC50 = 240 nM T50688 CF65YE 10095540 IC50 = 5200 nM T50688 C82XUE 10095734 IC50 = 0.5 nM T50688 CLN76R 10096459 IC50 = 4050 nM T50688 CDEA39 10096654 IC50 = 4030 nM T50688 C6JLQ8 10097012 IC50 > 1000 nM T50688 C1EO7I 10098015 IC50 = 30 nM T50688 CS2A6F 10098382 IC50 = 24.4 nM T50688 C1X6MY 10099012 Ki = 110 nM T50688 CA05EG 10101088 Ki = 45 nM T50688 CESP84 10113832 IC50 > 30000 nM T50688 CWT3Y7 10136986 IC50 = 950 nM T50688 COFK25 10160125 IC50 = 20 nM T50688 CNBL36 10160126 IC50 = 34000 nM T50688 C1O0GR 10162362 IC50 = 12607 nM T50688 CX7A1Z 10164947 IC50 = 747 nM T50688 CDL31V 10165701 IC50 = 419 nM T50688 CV0G1X 10181237 IC50 = 1020 nM T50688 CO8D9C 10196873 IC50 > 10000 nM T50688 CPT2Q5 10224943 IC50 = 1400 nM T50688 C53NHL 10228662 IC50 = 8130 nM T50688 CIZ09S 10230114 IC50 = 3 nM T50688 C0M7FC 10248023 IC50 = 40 nM T50688 CJG6U3 10251891 IC50 = 23 nM T50688 CH9AD2 10252306 IC50 > 1000000 nM T50688 CM9UQ8 10252576 IC50 = 80.3 nM T50688 C7T4BQ 10252696 IC50 = 6200 nM T50688 COT17X 10254067 IC50 = 65000 nM T50688 CK8S7O 10254771 IC50 > 100000 nM T50688 CQS29V 10254830 IC50 = 45000 nM T50688 C0J5CR 10254942 IC50 = 29 nM T50688 CZ2R6D 10255598 IC50 = 3500 nM T50688 CHX06T 10255701 IC50 = 260 nM T50688 C59BFD 10256182 IC50 = 10 nM T50688 C9JOB1 10274638 IC50 = 16000 nM T50688 CD04QE 10279663 IC50 = 474 nM T50688 C7E8PX 10281105 IC50 = 0.44 nM T50688 CIF59V 10281222 IC50 = 0.18 nM T50688 C9CST0 10281487 IC50 = 18 nM T50688 CJE72C 10295656 IC50 = 35774 nM T50688 CR2YI9 10297636 IC50 = 81.9 nM T50688 CF2A5U 10317079 IC50 = 74 nM T50688 CX80NC 10318813 IC50 = 364 nM T50688 CK5LC9 10319753 IC50 = 1500 nM T50688 CB80UA 10320733 IC50 = 1900 nM T50688 C20SHE 10322151 IC50 = 3000 nM T50688 CECM40 10322684 IC50 = 18 nM T50688 CH5F6W 10322871 IC50 > 10000 nM T50688 CUZ8V6 10323749 IC50 = 4500 nM T50688 CXMC15 10325138 IC50 = 1000000 nM T50688 C7PN3T 10326558 IC50 = 4120 nM T50688 C0WZS7 10326940 IC50 = 20 nM T50688 CMP36Y 10327110 IC50 = 1.5 nM T50688 C4I2TF 10335848 IC50 = 904 nM T50688 CSO64L 10335906 IC50 = 30000 nM T50688 C14ZPK 10336754 IC50 = 2800 nM T50688 COL4X9 10340606 IC50 = 95000 nM T50688 C84KLV 10340994 IC50 = 2400 nM T50688 CYXW23 10343956 IC50 = 260 nM T50688 CR5VI0 10344187 IC50 = 1000 nM T50688 C75OLX 10344202 IC50 = 110 nM T50688 CD1C7I 10345263 IC50 = 224 nM T50688 CF18LZ 10345912 IC50 = 384 nM T50688 CJ19HI 10346506 IC50 = 36.31 nM T50688 C62KDF 10347784 Ki = 0.1 nM T50688 C1ZC2P 10348465 IC50 = 1600 nM T50688 CZPQ03 10348588 Ki = 8750 nM T50688 CM5C9S 10348589 Ki = 20 nM T50688 C39XZM 10359266 IC50 = 256 nM T50688 C2JU5Z 10359401 IC50 = 133 nM T50688 C52YXA 10363350 IC50 = 321 nM T50688 CI3AF9 10367229 IC50 = 6195 nM T50688 CQ04DG 10367832 IC50 = 36.2 nM T50688 C98AHY 10368152 IC50 = 43 nM T50688 CY1R0K 10368440 IC50 = 4362 nM T50688 C1O9DY 10369377 IC50 = 400 nM T50688 CVOY03 10369856 IC50 = 61000 nM T50688 C9THO5 10371227 IC50 = 20 nM T50688 CS24DZ 10381857 IC50 = 760 nM T50688 CK8U5J 10384651 IC50 = 64 nM T50688 CQ4H3K 10386147 IC50 = 772 nM T50688 C28BIN 10386305 IC50 = 5 nM T50688 CY51PK 10388633 IC50 = 38000 nM T50688 CZ8L0B 10389185 IC50 = 313 nM T50688 CU7V6R 10390852 IC50 = 23000 nM T50688 C7OEB8 10391124 IC50 = 0.041 nM T50688 C31WGJ 10391128 IC50 = 340 nM T50688 CC0L8M 10392074 IC50 = 4230 nM T50688 C4J3XW 10394724 Ki = 24.5 nM T50688 CL9SM7 10404377 IC50 = 100 nM T50688 C3LZ7E 10405336 IC50 = 491 nM T50688 CBL9Y6 10407528 IC50 = 290 nM T50688 C74LKV 10409937 IC50 = 1000 nM T50688 CEP9G0 10410948 IC50 = 559 nM T50688 CWH42Z 10411419 IC50 = 1000 nM T50688 CO0FY6 10411523 IC50 > 10000 nM T50688 C7B3MO 10412184 IC50 > 10000 nM T50688 CR0F1T 10412890 IC50 = 37.6 nM T50688 C7NQW0 10413380 IC50 = 4260 nM T50688 CAHU62 10413821 IC50 = 17500 nM T50688 CZ30YD 10414275 IC50 = 23.99 nM T50688 CFP6E5 10414330 IC50 = 1 nM T50688 CZ12CP 10415384 IC50 = 480 nM T50688 C2F0NO 10422987 IC50 > 100000 nM T50688 C71VHN 10426654 IC50 = 2600 nM T50688 C5VN6I 10427709 IC50 = 280 nM T50688 C4KL7O 10433389 IC50 = 600 nM T50688 CUHY62 10433896 IC50 = 27 nM T50688 C69WHT 10434168 IC50 = 500 nM T50688 C2PZQ3 10434644 IC50 = 50000 nM T50688 CTGO27 10434789 IC50 = 22000 nM T50688 CRP82B 10435346 IC50 > 10000 nM T50688 C9F2QA 10436174 IC50 = 252 nM T50688 CD8MU7 10436196 IC50 = 11200 nM T50688 C1ME0S 10436235 IC50 = 39.4 nM T50688 CT60XI 10437052 IC50 = 12000 nM T50688 C04HQK 10437073 IC50 = 32.7 nM T50688 C9KNC8 10437414 IC50 = 25000 nM T50688 CSM7T9 10437869 IC50 = 50 nM T50688 C37TNI 10439316 Ki = 143 nM T50688 C6X8SU 10449316 IC50 = 150 nM T50688 CN83LC 10449423 IC50 = 115 nM T50688 C0IA8K 10455265 IC50 = 2600 nM T50688 C6AWI9 10456038 IC50 = 7600 nM T50688 C1XTA5 10456473 IC50 > 10000 nM T50688 C6G9YM 10457584 IC50 = 187 nM T50688 C9ZN4U 10457840 IC50 = 2515 nM T50688 CX69EL 10458074 Ki = 26 nM T50688 CBR94V 10458089 IC50 = 19000 nM T50688 C6P0ZM 10458809 IC50 > 50000 nM T50688 CGW9B0 10459259 IC50 = 15600 nM T50688 CQV26D 10459311 IC50 = 2 nM T50688 C1OPH5 10459371 IC50 = 10 nM T50688 CZ7LH3 10461739 Ki = 175 nM T50688 CM2L0R 10472801 IC50 = 1240 nM T50688 C3RJ9D 10473093 IC50 = 5700 nM T50688 C0H5CG 10473844 IC50 = 500 nM T50688 CJB80U 10475325 Ki = 3.2 nM T50688 CQ0PO9 10476004 IC50 = 63 nM T50688 C7J5NX 10478278 IC50 = 12000 nM T50688 C2S0VX 10478439 IC50 = 800 nM T50688 C04EHN 10478966 IC50 = 50000 nM T50688 CZ8G3U 10479133 IC50 = 140 nM T50688 C5FX7L 10479186 IC50 = 636 nM T50688 C0NVB7 10479802 IC50 = 405 nM T50688 C0KN6P 10479916 IC50 = 4940 nM T50688 CM48CA 10480140 IC50 = 4500 nM T50688 CUT7N4 10480781 IC50 = 75900 nM T50688 C9S2RZ 10480903 IC50 = 2 nM T50688 C6IAB4 10482388 IC50 = 559 nM T50688 C9OM3L 10482416 IC50 = 13.5 nM T50688 C45MRF 10483616 IC50 > 100000 nM T50688 CH8Z5U 10484706 Ki = 125 nM T50688 CZSU97 10495925 IC50 < 100000 nM T50688 CX9CY0 10497921 IC50 = 9000 nM T50688 C57YIO 10498183 IC50 = 27 nM T50688 CIDX93 10498794 IC50 = 0.42 nM T50688 C32ENG 10498863 IC50 = 1.6 nM T50688 C7MEW6 10500045 Ki = 1200 nM T50688 C9NI6T 10500892 IC50 = 170 nM T50688 CO57MY 10501597 IC50 = 1400 nM T50688 CM0ZW9 10503055 IC50 = 250 nM T50688 CE5N7J 10504150 IC50 = 14 nM T50688 C1U8TQ 10504200 IC50 > 1000 nM T50688 C5UMV6 10504763 IC50 = 37 nM T50688 C0U6NB 10504802 IC50 = 170 nM T50688 CF24JN 10505627 IC50 = 9000 nM T50688 CWLQ37 10506080 IC50 = 7 nM T50688 CR26WA 10506313 IC50 = 390 nM T50688 CS9N1R 10506318 IC50 = 900 nM T50688 CT1FK6 10506679 IC50 = 57 nM T50688 C3W8VJ 10507104 IC50 = 39 nM T50688 CZ70VF 10507218 IC50 = 2000 nM T50688 CC58KL 10507483 IC50 = 6500 nM T50688 CXS79H 10507484 IC50 = 11000 nM T50688 CKT5B3 10521604 IC50 = 850 nM T50688 CPI81M 10521872 IC50 = 0.12 nM T50688 C3ZK9B 10521873 IC50 = 5 nM T50688 CHF70E 10523877 Ki = 1750 nM T50688 C2HV8Y 10524492 IC50 = 0.13 nM T50688 C17VLR 10525508 IC50 = 78 nM T50688 C2KW1M 10525856 IC50 = 0.81 nM T50688 CW37AZ 10526036 IC50 > 1000 nM T50688 C4VN0A 10526120 IC50 = 21 nM T50688 C7DQU0 10526203 Ki > 50000 nM T50688 CEU48D 10526463 IC50 = 180 nM T50688 CA7Q1M 10526820 IC50 = 340 nM T50688 COY51D 10527580 IC50 = 0.14 nM T50688 CD6T3L 10527653 IC50 > 1000 nM T50688 C43BPT 10527958 IC50 = 12 nM T50688 C0D6XG 10528000 IC50 = 6000 nM T50688 C4P5VR 10528032 IC50 = 4200 nM T50688 C16HLY 10528334 IC50 = 6000 nM T50688 CGE0P3 10528399 Ki = 540 nM T50688 C2AX9H 10528472 IC50 = 32 nM T50688 CV06QK 10528788 IC50 = 300 nM T50688 C0T5IM 10529317 IC50 = 6300 nM T50688 CM4Z9C 10529546 IC50 = 1000 nM T50688 CC9GJ8 10529586 IC50 = 24 nM T50688 C0G5VX 10529678 IC50 = 95 nM T50688 CUY9Q0 10529865 IC50 > 10000 nM T50688 C3FG5K 10530186 IC50 = 9 nM T50688 CQ8JT1 10530357 IC50 = 4.3 nM T50688 C61HVA 10530613 IC50 = 260 nM T50688 CG1H4C 10531830 IC50 = 27.3 nM T50688 C2L1PJ 10531967 IC50 = 1600 nM T50688 CF0CS2 10541651 IC50 = 18000 nM T50688 CU95VC 10544052 IC50 = 16000 nM T50688 CPC51L 10544691 IC50 = 46000 nM T50688 C1WA0R 10545460 IC50 = 9900 nM T50688 CD1Y5N 10546320 IC50 = 440 nM T50688 CBS2F4 10548981 IC50 > 1000 nM T50688 CWA51X 10549838 IC50 = 3 nM T50688 CY4QG2 10549931 IC50 = 0.92 nM T50688 C3ST9M 10549992 IC50 = 130 nM T50688 C1SJN7 10551324 IC50 = 96 nM T50688 C8Y3PH 10551831 IC50 = 125 nM T50688 CBJ70D 10551898 IC50 = 15 nM T50688 CEO2N5 10552647 IC50 = 930 nM T50688 CR6TH2 10553451 IC50 = 2630 nM T50688 C7BLP8 10553605 IC50 = 180 nM T50688 C1OP8Z 10554323 IC50 = 45 nM T50688 CZD20R 10555279 IC50 = 3100 nM T50688 CAFZ87 10555310 IC50 = 260 nM T50688 C1S5KM 10555762 IC50 = 31.3 nM T50688 CPX62H 10567014 IC50 = 630 nM T50688 C02LOP 10569012 IC50 = 260 nM T50688 CTKA09 10569078 IC50 = 1200 nM T50688 C45UKM 10569143 IC50 = 12000 nM T50688 C63AQL 10569459 IC50 = 4100 nM T50688 C7PIF3 10569520 IC50 = 7400 nM T50688 C5K6LD 10570053 IC50 = 190 nM T50688 CR0WY1 10570641 IC50 = 12000 nM T50688 C6ST5A 10570949 IC50 = 500 nM T50688 CU01OT 10572765 Ki = 290 nM T50688 CI4CM8 10573992 IC50 = 170 nM T50688 C95HGK 10574096 IC50 = 130 nM T50688 CAWF40 10574237 Ki > 100000 nM T50688 CDZR27 10574289 IC50 = 360 nM T50688 CMN41A 10574669 IC50 = 7.2 nM T50688 CC9M4O 10574710 IC50 = 0.2 nM T50688 C1K8IY 10574717 IC50 = 85 nM T50688 COA4T1 10574792 IC50 = 8.1 nM T50688 C75XGA 10574888 IC50 = 2500 nM T50688 C73VFG 10574923 IC50 = 20 nM T50688 C01GQV 10575330 IC50 = 36 nM T50688 C47OMC 10575410 IC50 = 5000 nM T50688 C5P1NG 10575581 IC50 = 73 nM T50688 CI35XW 10576070 Ki = 80 nM T50688 C6NM7V 10576167 IC50 = 69 nM T50688 CXZP31 10576168 IC50 = 67 nM T50688 CB67ER 10576733 IC50 = 13000 nM T50688 CV3QL4 10577095 IC50 = 1.8 nM T50688 CX1K0N 10577150 IC50 = 21 nM T50688 CKP4H6 10577279 IC50 = 1.5 nM T50688 CJ3T2Q 10577940 IC50 = 12 nM T50688 CU75WP 10578810 IC50 = 81 nM T50688 CZ9VX1 10579340 IC50 = 21.3 nM T50688 C0U1CG 10582643 IC50 > 10000 nM T50688 CWG26D 10591778 IC50 = 44000 nM T50688 CQ5LE9 10592825 IC50 = 10000 nM T50688 CF15AC 10593246 IC50 = 77000 nM T50688 CLA3Q4 10595524 IC50 = 160 nM T50688 CS15AP 10596310 IC50 = 16000 nM T50688 CZ9ES6 10596311 IC50 = 25300 nM T50688 CDK10F 10597871 IC50 = 40 nM T50688 CKS6B5 10598109 IC50 = 60 nM T50688 C8TQ3C 10598184 IC50 = 42 nM T50688 CDM3L1 10598267 IC50 = 2200 nM T50688 CC4AS1 10598742 IC50 = 0.13 nM T50688 CM38KV 10598938 IC50 = 1030 nM T50688 C9SM8R 10599499 IC50 = 230 nM T50688 C4I2EJ 10599577 IC50 = 88 nM T50688 CE7DI4 10600322 IC50 = 47 nM T50688 CNO98S 10600933 IC50 = 0.34 nM T50688 CJ16VT 10601205 IC50 = 0.52 nM T50688 C6WK7Z 10601297 IC50 = 3 nM T50688 CC52PM 10601502 IC50 = 1.8 nM T50688 CI09PZ 10601521 IC50 = 32 nM T50688 CSZ1C6 10601709 IC50 = 3.6 nM T50688 CA04QH 10601955 IC50 = 0.85 nM T50688 CLA7F4 10602103 IC50 = 11 nM T50688 CA0NM6 10602590 IC50 = 26 nM T50688 C39IPX 10603319 IC50 = 12 nM T50688 C07MCW 10603422 IC50 = 470 nM T50688 CAW3U8 10603619 IC50 = 11 nM T50688 C0EU7G 10603811 IC50 = 34.7 nM T50688 CPVM74 10604005 IC50 = 2 nM T50688 CDXB14 10606654 IC50 > 1000 nM T50688 CJ49TW 10615755 IC50 = 1100 nM T50688 CY86JI 10617432 IC50 > 100000 nM T50688 CNB89K 10620252 IC50 > 10000 nM T50688 C1V9UK 10620480 IC50 = 0.26 nM T50688 C7N8UQ 10621705 IC50 > 1000 nM T50688 CRFI52 10622095 IC50 = 0.1 nM T50688 CB7X1D 10622197 IC50 = 500 nM T50688 CUME64 10622650 IC50 = 0.21 nM T50688 CT9U1I 10622651 IC50 = 2810 nM T50688 CZ1D7P 10622934 IC50 = 0.22 nM T50688 CIL20A 10623555 IC50 = 31 nM T50688 C35QBJ 10623736 IC50 = 350 nM T50688 C1VC0O 10624584 IC50 = 3.8 nM T50688 C5FGS8 10624764 Ki = 800 nM T50688 CLR06I 10626114 IC50 = 57 nM T50688 CMQA47 10626357 IC50 = 5.1 nM T50688 C08FHO 10627561 IC50 = 3410 nM T50688 CUBJ20 10628601 IC50 = 67 nM T50688 CA03HK 10639257 IC50 = 55000 nM T50688 C0CFP3 10639900 IC50 = 5000 nM T50688 CBZ8U6 10641657 IC50 = 4200 nM T50688 CF8CK1 10644680 IC50 = 0.58 nM T50688 CLV5I7 10645125 IC50 = 300 nM T50688 C1TKQ4 10645607 IC50 = 8000 nM T50688 CMB93Z 10645847 Ki > 50000 nM T50688 CS5PN3 10647720 IC50 > 1000 nM T50688 CM54PX 10647971 IC50 > 1000 nM T50688 C0EFS9 10648519 IC50 = 85000 nM T50688 C5ABX8 10648597 Ki = 26 nM T50688 CX98VN 10648960 IC50 = 1500 nM T50688 CY38BT 10649923 IC50 = 6500 nM T50688 CHV18W 10650104 IC50 = 74 nM T50688 C91EXP 10650216 IC50 = 5.4 nM T50688 CI3E1K 10650223 IC50 = 44 nM T50688 CIW40L 10650245 IC50 = 5.8 nM T50688 CW5KO9 10650595 IC50 = 41000 nM T50688 C4QO9H 10651012 IC50 = 130 nM T50688 CXQ5B4 10663504 IC50 = 23000 nM T50688 CI0K7L 10665207 IC50 = 26700 nM T50688 CD82QM 10666108 IC50 = 27000 nM T50688 C5OQJ8 10666236 IC50 = 1800 nM T50688 C8SH0G 10667601 IC50 = 4000 nM T50688 CP18RM 10669069 IC50 = 460 nM T50688 C6V4RM 10669472 IC50 = 2100 nM T50688 C0F7QU 10669861 IC50 = 10000 nM T50688 C3TJ1R 10669871 IC50 = 0.15 nM T50688 CUIE47 10670418 IC50 = 20 nM T50688 CU13QF 10670421 IC50 = 100 nM T50688 C8QTJ0 10670464 IC50 = 78 nM T50688 C7UA2O 10671221 IC50 = 230 nM T50688 CPMD78 10671690 IC50 = 41 nM T50688 CK87TJ 10672605 IC50 > 10000 nM T50688 C8O5EP 10672609 IC50 = 61 nM T50688 CMB4O8 10673127 IC50 > 10000 nM T50688 CVX5L8 10673284 IC50 = 5000 nM T50688 C5C4KF 10673305 IC50 = 34 nM T50688 C4OU1Z 10673351 IC50 = 67 nM T50688 C1K4VA 10673587 IC50 = 290 nM T50688 C9AO8W 10673593 IC50 = 15 nM T50688 CNZ52W 10674738 IC50 = 4400 nM T50688 CN07MA 10675175 IC50 = 47.3 nM T50688 C5CO8D 10675509 IC50 = 64 nM T50688 CY10JG 10678157 IC50 > 1000 nM T50688 CMV21P 10678163 IC50 > 1000 nM T50688 C6R4MV 10678165 IC50 > 10000 nM T50688 CO35RT 10686097 IC50 = 28000 nM T50688 CF73WA 10687020 IC50 = 60 nM T50688 CG68IP 10688817 IC50 = 310 nM T50688 CL61KC 10689869 IC50 = 140 nM T50688 CDVJ25 10690277 IC50 = 410 nM T50688 CNW32D 10690754 IC50 = 1800 nM T50688 C6U0EH 10691302 IC50 > 10000 nM T50688 CM4I0K 10692763 Ki = 52000 nM T50688 CBJ5U8 10693286 IC50 = 1.7 nM T50688 CX6R5Z 10693378 IC50 = 1 nM T50688 CIP7S4 10693570 IC50 = 2.6 nM T50688 C7F6CR 10693833 Ki = 2.5 nM T50688 CTV09E 10695326 Ki = 19 nM T50688 C6G5SF 10696089 IC50 = 50 nM T50688 COE2C0 10696268 Ki = 2 nM T50688 CT08OR 10696562 IC50 = 570 nM T50688 CLYC49 10697230 IC50 = 10 nM T50688 CX26BU 10697338 IC50 > 10000 nM T50688 C3SF8N 10697605 IC50 = 32000 nM T50688 CFG8O6 10698251 IC50 = 400 nM T50688 CYV8S2 10698274 IC50 = 66 nM T50688 CHL29X 10698729 IC50 = 10 nM T50688 C98TZX 10699307 IC50 = 1370 nM T50688 CWP46I 10710664 IC50 = 36600 nM T50688 CBH0X7 10710665 IC50 = 38200 nM T50688 CRP1Q5 10711631 IC50 = 18000 nM T50688 C57MHS 10711633 IC50 = 11000 nM T50688 CK6OM7 10711689 IC50 = 91 nM T50688 CXE5V7 10712480 IC50 = 43700 nM T50688 CU90KW 10714203 Ki = 560 nM T50688 CIMF59 10715577 Ki > 50000 nM T50688 C4D2UE 10716904 IC50 = 138 nM T50688 C3CG9M 10717156 IC50 = 40 nM T50688 C9JRQ6 10717165 IC50 = 180 nM T50688 C30YKM 10718276 IC50 = 34000 nM T50688 CPZ2J1 10718421 IC50 = 110 nM T50688 CI3F1Z 10719036 IC50 = 0.18 nM T50688 CJ9WY6 10719690 Ki = 14900 nM T50688 C9T4FM 10720025 IC50 = 18 nM T50688 CB2JR1 10720397 IC50 = 180 nM T50688 CY40LK 10720760 IC50 = 850 nM T50688 C4LY7B 10720773 IC50 = 0.66 nM T50688 CWM1H4 10721018 IC50 = 4 nM T50688 CYM68T 10721510 IC50 = 57 nM T50688 CRD6A2 10734460 IC50 = 19000 nM T50688 C4DL1X 10735250 IC50 = 1100 nM T50688 CD8QH7 10736235 IC50 = 7500 nM T50688 C7ISZ3 10737628 Ki = 1500 nM T50688 CMCP54 10737883 IC50 = 40 nM T50688 CO9EB6 10739023 IC50 = 50 nM T50688 C3JG8M 10739084 IC50 = 0.16 nM T50688 CFEW14 10740150 IC50 = 50000 nM T50688 CY40JW 10741088 IC50 = 21 nM T50688 C0WB5V 10741543 IC50 = 5000 nM T50688 C32HFP 10741551 IC50 = 65 nM T50688 CTF43Q 10741717 IC50 = 3 nM T50688 CW1V6I 10741784 IC50 = 180 nM T50688 C5F6IQ 10742630 IC50 = 210 nM T50688 CQ43HK 10743381 IC50 = 2 nM T50688 CA5BC6 10743635 IC50 = 10000 nM T50688 C3EY2G 10744029 IC50 = 32 nM T50688 CQN7C5 10744439 IC50 = 5.3 nM T50688 CWTH73 10744841 IC50 = 36 nM T50688 C72AXW 10744879 IC50 = 3100 nM T50688 CPW19S 10744934 IC50 = 7800 nM T50688 C0XJY2 10745059 IC50 = 13 nM T50688 CS7YL2 10745179 IC50 = 190 nM T50688 C5N0JC 10745304 IC50 = 5000 nM T50688 CE0DW6 10745412 IC50 = 3.8 nM T50688 C2YL0X 10745414 IC50 = 2.7 nM T50688 CDHZ35 10745638 IC50 = 770 nM T50688 CPQ9N3 10746038 IC50 = 65 nM T50688 CTZG52 10746372 IC50 = 74 nM T50688 CI6W7O 10747110 IC50 = 22 nM T50688 C5GA7Z 10747212 IC50 = 11 nM T50688 CJ6EY5 10760011 IC50 = 48000 nM T50688 C2J5DF 10760306 IC50 = 14000 nM T50688 C2UVP6 10760519 IC50 = 0.073 nM T50688 CWA45B 10762449 IC50 = 14000 nM T50688 CU79QS 10764595 IC50 = 2.5 nM T50688 CD5BH1 10765679 IC50 = 0.75 nM T50688 C0BW1Q 10765828 IC50 = 90 nM T50688 C36RIG 10765872 IC50 = 50000 nM T50688 CC47BU 10765873 IC50 = 1000 nM T50688 C65WOR 10766035 IC50 = 1000 nM T50688 C0Q8ET 10766137 IC50 = 20 nM T50688 CC06BN 10766594 IC50 = 31 nM T50688 C4XFU2 10767331 IC50 = 3000 nM T50688 CUB46C 10767352 IC50 = 600 nM T50688 CRK0M2 10767647 IC50 = 2 nM T50688 CL1XE6 10767757 IC50 = 10 nM T50688 CO15MH 10769104 IC50 = 5000 nM T50688 CH35PG 10780340 IC50 > 100000 nM T50688 CD38LF 10780686 IC50 = 48000 nM T50688 CG1B9U 10781733 IC50 = 2300 nM T50688 CDZM40 10781802 IC50 = 60 nM T50688 CL9M4R 10783789 IC50 = 6000 nM T50688 CJBT94 10784172 IC50 = 5 nM T50688 C7QDL1 10786753 IC50 = 0.13 nM T50688 CJE7P8 10788151 IC50 = 330 nM T50688 C0Z5PU 10788266 IC50 = 21000 nM T50688 CBJK78 10788353 IC50 = 630 nM T50688 CR2Y3H 10788405 Ki = 8 nM T50688 CYC0D7 10788947 IC50 = 1 nM T50688 CU6M5W 10788997 IC50 = 250000 nM T50688 C5B6MC 10789118 IC50 = 13 nM T50688 C25HXT 10789240 IC50 = 0.24 nM T50688 CRLY08 10790058 IC50 > 1000 nM T50688 CL07VH 10790223 IC50 = 250 nM T50688 CL48DH 10790594 IC50 = 0.65 nM T50688 CIMC29 10790917 IC50 = 55 nM T50688 CRME39 10791865 IC50 > 10000 nM T50688 CD60VX 10791985 IC50 = 7 nM T50688 CGI2S3 10792202 IC50 = 83 nM T50688 C0IFV7 10792261 IC50 = 13 nM T50688 CKU3Z4 10792272 IC50 = 570 nM T50688 C90EQR 10793103 IC50 = 4000 nM T50688 C9L4KF 10793351 IC50 = 790 nM T50688 CG47UL 10793849 IC50 = 72 nM T50688 C5YSV2 10794013 IC50 = 5.6 nM T50688 CQE3T7 10794762 IC50 = 96 nM T50688 C56FMJ 10807406 IC50 = 340 nM T50688 C9Z1JU 10807527 IC50 = 54 nM T50688 CE80DB 10807712 IC50 = 290 nM T50688 CG70RV 10808878 IC50 = 3 nM T50688 CRJ80X 10808969 IC50 = 6000 nM T50688 CR2SG6 10809369 IC50 = 250 nM T50688 CKW54J 10810465 IC50 = 65 nM T50688 CANY49 10810509 IC50 = 594 nM T50688 CS87IC 10810880 IC50 = 6300 nM T50688 CG5Y0D 10811208 IC50 = 163 nM T50688 C5GU3F 10811614 IC50 = 10000 nM T50688 C0GAW3 10811724 IC50 = 46 nM T50688 C1EI3C 10811745 IC50 = 590 nM T50688 C2E5AI 10813353 IC50 = 18 nM T50688 C6AV1O 10813355 IC50 = 0.89 nM T50688 C0BO1X 10813883 Ki = 750 nM T50688 C86QIK 10814015 IC50 = 68 nM T50688 CQSR19 10814133 IC50 = 1600 nM T50688 CKHJ63 10814581 IC50 = 55 nM T50688 CXQD50 10814626 IC50 = 35 nM T50688 CL35GT 10815092 IC50 = 160 nM T50688 CZA18Q 10815853 IC50 = 36 nM T50688 CNG0H1 10816131 IC50 > 100000 nM T50688 C8X6GV 10816353 IC50 = 8.6 nM T50688 CVL1Q5 10816922 IC50 = 22.3 nM T50688 CXY5H4 10817117 IC50 = 8 nM T50688 CL5M9B 10817315 IC50 = 363 nM T50688 CC79QZ 10829524 IC50 = 64000 nM T50688 C7NLW3 10830476 IC50 = 870 nM T50688 CI7HF0 10830837 IC50 = 47000 nM T50688 C9LZ8N 10830937 IC50 = 30 nM T50688 C7QS2L 10831902 IC50 = 5800 nM T50688 CA8X9M 10831903 IC50 = 4000 nM T50688 CGRC85 10832778 IC50 = 600 nM T50688 CAWT74 10833338 IC50 = 210 nM T50688 CYBU67 10837146 IC50 = 360 nM T50688 CCW4P0 10838744 IC50 = 30000 nM T50688 CVX39A 10838945 IC50 = 0.21 nM T50688 C65XRV 10839051 IC50 = 0.37 nM T50688 C7I6UV 10839864 IC50 = 3.8 nM T50688 CSK2Z4 10839940 IC50 = 5 nM T50688 C06QAI 10839976 IC50 > 100000 nM T50688 CKN51D 10840512 IC50 = 11 nM T50688 CTJ61U 10840969 IC50 = 36000 nM T50688 CY9DP7 10841676 IC50 = 21 nM T50688 C7EB4Y 10844291 IC50 > 1000 nM T50688 C9XK7J 10844292 IC50 = 1000 nM T50688 C1OFW6 10850199 IC50 = 48000 nM T50688 CMU8D1 10853893 IC50 > 100000 nM T50688 CIV0X1 10961560 IC50 = 2900 nM T50688 C08BCF 10993678 IC50 = 7300 nM T50688 CDK7W9 10994476 IC50 > 10000 nM T50688 CTW0P5 11102917 IC50 > 10000 nM T50688 C79OJR 11133736 IC50 = 580 nM T50688 C1S0PM 11169785 Ki = 206 nM T50688 CBO8Q0 11181082 Ki = 6840 nM T50688 CXEH75 11187899 IC50 = 733 nM T50688 CQF31D 11190947 Ki = 973 nM T50688 C2JZ6C 11192964 Ki = 7300 nM T50688 CJU1K7 11200734 IC50 > 10000 nM T50688 C5SH1R 11227896 Ki = 3660 nM T50688 CN74QM 11234552 IC50 = 660 nM T50688 CQG0I1 11234588 IC50 = 350 nM T50688 C4HFS8 11234619 IC50 = 17 nM T50688 C8A5RL 11237915 Ki = 3940 nM T50688 C83HIU 11246220 IC50 = 1610 nM T50688 CR2JN6 11246637 IC50 = 329 nM T50688 CPQ2H7 11246987 IC50 = 841 nM T50688 C5JXU9 11257283 IC50 = 5183 nM T50688 CDN62X 11269177 IC50 = 4 nM T50688 CY1LH0 11281059 IC50 = 68 nM T50688 C98HYU 11284340 IC50 = 1 nM T50688 CSH76U 11284767 IC50 = 24630 nM T50688 CWN52M 11292505 IC50 = 730 nM T50688 CVW45L 11292510 IC50 = 5 nM T50688 CA7EI1 11304190 IC50 = 212 nM T50688 CVQ9A3 11304592 IC50 = 3600 nM T50688 C7HTY1 11307791 IC50 = 2 nM T50688 C51AZT 11315587 IC50 = 6490 nM T50688 C82ZFG 11337742 IC50 = 5700 nM T50688 C7VDO8 11372991 IC50 = 21 nM T50688 CZJ15G 11374651 IC50 = 90 nM T50688 CZ5E4X 11374986 IC50 = 20 nM T50688 CTS8G9 11384491 IC50 = 222 nM T50688 CV1NT6 11386324 IC50 = 120 nM T50688 C45EBU 11394236 IC50 = 12500 nM T50688 C4KU1F 11395891 IC50 = 700 nM T50688 CZO3H7 11399588 IC50 = 9000 nM T50688 CL8AO4 11406569 IC50 = 751 nM T50688 CS4PY1 11406925 IC50 = 4100 nM T50688 CNP04F 11410732 IC50 = 16 nM T50688 CVI7S8 11441000 IC50 = 410 nM T50688 CE6FI4 11452378 IC50 = 1020 nM T50688 C9L2OX 11452690 IC50 > 10000 nM T50688 CEWT48 11452816 Ki = 4.2 nM T50688 CJCF34 11486406 IC50 = 3400 nM T50688 CDIR54 11486773 IC50 > 10000 nM T50688 CZ8I5T 11489856 IC50 = 5 nM T50688 C50FQZ 11489885 IC50 = 1640 nM T50688 C5NEM0 11546965 IC50 = 168 nM T50688 CFZ2O9 11613998 IC50 > 50000 nM T50688 CGU84F 11721315 IC50 > 50000 nM T50688 C2ONX6 11721442 IC50 = 8000 nM T50688 CLHR18 11723405 IC50 > 10000 nM T50688 CO7K6Z 11740268 IC50 = 105 nM T50688 CF9IT7 11740665 IC50 = 3 nM T50688 CUW59R 11741589 IC50 = 14000 nM T50688 CY35MP 11742524 IC50 = 26000 nM T50688 C01BWL 11742781 IC50 = 35 nM T50688 C7GV2M 11743323 IC50 = 29 nM T50688 C9CX0F 11743586 IC50 = 101 nM T50688 CE5H7K 11744415 IC50 = 11200 nM T50688 CIO0X8 11744424 IC50 = 300 nM T50688 CS1Q9P 11744536 IC50 > 10000 nM T50688 CZ9GM1 11749950 IC50 = 112 nM T50688 CR7NP5 11751578 IC50 = 25 nM T50688 C2KZ5U 11752405 IC50 = 5 nM T50688 CBS24R 11754911 IC50 = 3 nM T50688 CV63YK 11755157 IC50 = 29 nM T50688 CMY21B 11756777 IC50 = 65 nM T50688 CPXI40 11757187 IC50 > 3000 nM T50688 C3DCM0 11757316 IC50 = 1000000 nM T50688 CEN37T 11757623 IC50 = 220 nM T50688 C8MFU9 11772736 IC50 = 7400 nM T50688 CB5MA7 11791726 IC50 = 9800 nM T50688 C8S1AR 11791783 IC50 = 760 nM T50688 C4H6KF 11791858 IC50 = 39000 nM T50688 C39KJR 11792525 IC50 = 3.5 nM T50688 C98GJL 11792811 IC50 = 48 nM T50688 C7PY0U 11793130 IC50 = 4000 nM T50688 CV51NX 11796444 IC50 = 1350 nM T50688 CPKC53 11797034 IC50 = 47 nM T50688 CA1FD8 11797035 IC50 = 27 nM T50688 C9KVR6 11797667 IC50 = 200 nM T50688 C5GTQ0 11798113 IC50 = 200 nM T50688 CFL9C4 11799328 IC50 = 3000 nM T50688 CHIN14 11799438 IC50 = 51 nM T50688 CT4D1K 11799915 IC50 > 100000 nM T50688 C4U1TD 11800065 IC50 = 78000 nM T50688 CZ06CB 11800170 IC50 = 600 nM T50688 C2BC6I 11800172 IC50 = 11 nM T50688 C4Z5HL 11800506 IC50 = 23 nM T50688 CW73UB 11800522 IC50 = 14 nM T50688 CD0GH5 11800573 IC50 > 100000 nM T50688 COT19X 11800615 IC50 = 410 nM T50688 CYC1X9 11800819 IC50 = 8100 nM T50688 C30JTG 11801283 IC50 = 5.7 nM T50688 CBF42H 11802695 IC50 = 22 nM T50688 C7EKZ0 11975699 Ki = 7.1 nM T50688 C1E9BA 12096120 IC50 = 660 nM T50688 CNA3W7 14563588 IC50 = 20000 nM T50688 CB2TD1 14796453 IC50 = 2300 nM T50688 C04GKV 15030977 IC50 = 27000 nM T50688 CV0AL8 15088298 IC50 > 200000 nM T50688 C3U8TD 15088299 IC50 = 138000 nM T50688 CDP35E 15088300 Ki = 14500 nM T50688 CKGL39 15088301 IC50 = 113000 nM T50688 C6BDE1 15088302 IC50 > 200000 nM T50688 CMK62Y 15088303 IC50 > 200000 nM T50688 C7ZOQ1 15088304 IC50 > 200000 nM T50688 C2DSH8 15088306 IC50 > 200000 nM T50688 CBL38Q 15088307 IC50 > 200000 nM T50688 CC34KU 15088308 IC50 > 200000 nM T50688 CR9ZP3 15088309 IC50 > 200000 nM T50688 CR5N7E 15088310 IC50 = 97000 nM T50688 CI69AO 15088312 IC50 > 200000 nM T50688 CNIV75 15088313 Ki < 10000 nM T50688 C6JVF0 15088314 IC50 = 102000 nM T50688 C17RXP 15088315 Ki = 4200 nM T50688 CV2UN6 15088316 IC50 > 200000 nM T50688 CGS1Y3 15088321 Ki = 3000 nM T50688 CW54MQ 15088322 Ki = 720 nM T50688 CCR3J9 15088323 Ki = 720 nM T50688 COR10Z 15088329 IC50 = 370 nM T50688 C9O8TU 15223439 IC50 = 122 nM T50688 CI7C9X 15223440 IC50 = 50 nM T50688 CP9S4I 15233759 IC50 = 170 nM T50688 CSF4Y8 15295775 IC50 = 5000 nM T50688 C69FBX 15297021 IC50 = 4.2 nM T50688 CVD8Z5 15337543 IC50 = 0.09 nM T50688 CAJ1P8 15337548 IC50 = 0.13 nM T50688 C9ZL2Y 15380364 IC50 = 125 nM T50688 C9N0XP 15428414 IC50 = 8 nM T50688 CR2MA3 15432278 IC50 = 1090 nM T50688 CMZN94 15483869 IC50 = 40 nM T50688 C7DT2P 15483870 IC50 = 24 nM T50688 C0WJ7R 15483871 IC50 = 7 nM T50688 CMES74 15486068 Ki = 30000 nM T50688 C1V8GD 15488825 Ki = 1.5 nM T50688 C2YG3M 15491369 Ki = 2300 nM T50688 COEP73 15491370 Ki = 20000 nM T50688 CZ2R8G 15491452 IC50 = 1300 nM T50688 CN0LX5 15491453 IC50 = 780 nM T50688 C3VOW7 15491454 IC50 = 460 nM T50688 CZX58V 15516067 Ki > 50000 nM T50688 CZBP40 15545291 IC50 = 11 nM T50688 CJGB65 15545292 IC50 = 72 nM T50688 C6WGZ9 15545293 IC50 = 610 nM T50688 CU60GO 15545294 IC50 = 71 nM T50688 CS81PK 15545295 IC50 = 26 nM T50688 C3OPX2 15547267 IC50 = 210 nM T50688 CZ48KQ 15838053 IC50 = 10 nM T50688 CDVB07 15850631 IC50 = 45 nM T50688 CG9FV3 15850632 IC50 = 2800 nM T50688 CKPV73 15850737 IC50 = 55 nM T50688 CM79QV 15850743 IC50 = 110 nM T50688 CM8G3S 15859412 IC50 > 10000 nM T50688 CW8LN2 15859413 IC50 = 2450 nM T50688 CT1DI8 15859414 IC50 = 2800 nM T50688 C95OGC 15859418 IC50 = 80 nM T50688 CEC41O 15859419 IC50 = 925 nM T50688 CFJ08N 15859420 IC50 = 235 nM T50688 CUQ9A2 15859421 IC50 = 55 nM T50688 C56IZT 15859422 IC50 = 9 nM T50688 CE6FO4 15859423 IC50 > 10000 nM T50688 C1VMK9 15859424 IC50 = 1000 nM T50688 C2B8GR 15887956 IC50 = 3 nM T50688 CKPY93 15887958 IC50 = 9 nM T50688 C8QO3Z 15887960 IC50 = 600 nM T50688 C8QIB4 15888084 Ki > 30000 nM T50688 CUY2F9 15931145 Ki = 1900 nM T50688 C7A0NY 15931147 IC50 > 200000 nM T50688 C9LSV8 16211712 Ki > 1000000 nM T50688 CTGC60 16678135 IC50 = 2300 nM T50688 CU8YQ3 16756502 IC50 = 7.7 nM T50688 C0KW3V 16756505 IC50 > 50000 nM T50688 C04JOX 16756621 IC50 = 50000 nM T50688 C4CU7T 16756622 IC50 > 50000 nM T50688 CFH96E 16756623 IC50 > 50000 nM T50688 CB15RX 16756849 IC50 = 12000 nM T50688 CM18ZN 16756955 IC50 > 50000 nM T50688 CL38IU 16756956 IC50 = 11000 nM T50688 CW5P8L 16756957 IC50 > 50000 nM T50688 CRWZ62 17788068 IC50 = 2700 nM T50688 C2DN9B 18394355 Ki > 50000 nM T50688 CAOR56 18660413 IC50 = 25000 nM T50688 C2HD8G 18967498 IC50 = 31000 nM T50688 C3T0QV 19034178 IC50 = 330000 nM T50688 C0O6XT 19076730 IC50 = 4810 nM T50688 C9G7ZK 19697937 IC50 = 0.098 nM T50688 C8SCL4 19757280 IC50 = 4880 nM T50688 CHV3L9 19757296 IC50 = 5880 nM T50688 CJ4L3C 19757333 IC50 = 4720 nM T50688 CW4IN3 19757343 IC50 = 2870 nM T50688 CY19FN 19962234 IC50 = 46 nM T50688 CXLO94 20587795 IC50 = 255 nM T50688 C7FR8G 20639626 IC50 = 28 nM T50688 CW64DV 20666951 IC50 = 21900 nM T50688 C85SOV 20666970 IC50 = 54 nM T50688 C61WDP 20666971 IC50 = 128 nM T50688 CX52NV 20666990 IC50 = 148 nM T50688 CVJ8N2 20667011 IC50 = 253 nM T50688 CMV17G 20667012 IC50 = 172 nM T50688 CQ8ME6 20667015 IC50 = 22 nM T50688 CR2X4L 20694723 IC50 = 4.2 nM T50688 CE57KZ 20694724 IC50 = 0.057 nM T50688 C6VZA8 20709789 IC50 > 10000 nM T50688 CEI27V 21053920 IC50 > 10000 nM T50688 C3TR2D 21191396 IC50 = 285 nM T50688 CE5Z3R 21191398 IC50 = 57 nM T50688 CGI19E 21191399 IC50 = 14.3 nM T50688 CN1Q0M 21191405 IC50 = 1000 nM T50688 C3GK7N 21191409 IC50 = 93 nM T50688 CQJ5Z3 21191417 IC50 = 3190 nM T50688 CU4FN2 21191441 IC50 = 4710 nM T50688 CM96YE 21191461 IC50 = 12.5 nM T50688 C7XYV3 21191470 IC50 = 6 nM T50688 C6X9US 21465966 IC50 = 80 nM T50688 CA10BL 21465982 IC50 = 31 nM T50688 CUJS70 21699778 IC50 > 10000 nM T50688 C2N6QA 21927945 IC50 = 9298 nM T50688 CT6N9S 22094645 IC50 = 1.2 nM T50688 CMS31G 22098946 IC50 = 1830 nM T50688 CE5G2I 22098949 IC50 = 2170 nM T50688 C2U1YQ 22098952 IC50 = 8270 nM T50688 CEU65M 22098953 IC50 = 670 nM T50688 CO4JK1 22098959 IC50 = 817 nM T50688 CN1Q2O 22098975 IC50 = 97 nM T50688 C94AUL 22098977 IC50 = 14.1 nM T50688 C7T2YX 22402471 IC50 = 2300000 nM T50688 CP2DW6 22451718 Ki = 1.9 nM T50688 CAD90V 22451721 Ki = 1.5 nM T50688 CG6FE5 22451739 Ki = 2 nM T50688 CJRA54 22451788 Ki = 22500 nM T50688 CP47JN 22451902 Ki = 4.7 nM T50688 CXVB03 22594242 IC50 = 110 nM T50688 CDJH42 22594251 IC50 = 1495 nM T50688 CPF73W 22594331 IC50 > 100000 nM T50688 CHR03I 22594351 IC50 = 1700 nM T50688 CFL7X5 22594355 IC50 = 552 nM T50688 CHVR74 22611774 IC50 = 200 nM T50688 CVM5Q1 22611776 IC50 > 100 nM T50688 C5LH4U 22611792 IC50 = 3 nM T50688 C2WR9E 22611889 IC50 > 100 nM T50688 C4V7BI 22645287 IC50 = 10 nM T50688 CB43DX 22866013 IC50 = 1.1 nM T50688 CFG40R 22975644 IC50 = 15000 nM T50688 C0MNQ9 23286727 IC50 = 47 nM T50688 CR6T1J 23297694 Ki = 1 nM T50688 CXZD95 23297711 Ki = 2 nM T50688 CWKA89 23297715 Ki = 1.7 nM T50688 CG7YV4 23297719 Ki = 1.5 nM T50688 CMG08E 23297721 Ki = 2 nM T50688 C7ETA1 23297736 Ki = 2 nM T50688 C0Y4GH 23297800 Ki = 650 nM T50688 CK21RA 23377844 IC50 = 210 nM T50688 CQ6M4A 23377846 IC50 = 9 nM T50688 C4OH9D 23377874 IC50 = 90 nM T50688 CMET78 23435760 IC50 = 3500 nM T50688 CKF08G 23435786 IC50 = 15000 nM T50688 CYND24 23729562 IC50 = 165 nM T50688 C96PUZ 23729563 IC50 = 30 nM T50688 CZ17YE 23731146 IC50 = 560 nM T50688 CHXT18 23731243 IC50 = 2000 nM T50688 CEA9Z8 23731244 IC50 = 12 nM T50688 CNK5O6 23731245 IC50 = 620 nM T50688 C6W9OS 23731246 IC50 = 15 nM T50688 CK7OW6 24779699 Ki = 47 nM T50688 C9L0QD 24864721 IC50 > 10000 nM T50688 CY6WR2 24872066 IC50 = 40200 nM T50688 CUM4E3 24872070 IC50 = 71700 nM T50688 CG09DH 24872646 IC50 = 77700 nM T50688 CRS65Q 24873110 IC50 = 87200 nM T50688 C0HZ7E 24873345 IC50 = 105000 nM T50688 CIS68P 25032865 IC50 > 10000 nM T50688 C07BZQ 25107507 IC50 = 2440 nM T50688 CK3FM6 25107508 IC50 = 12080 nM T50688 CN3I9J 25107569 IC50 = 15200 nM T50688 CB6H7T 25107570 IC50 = 1450 nM T50688 CC40FO 25107571 IC50 = 2000 nM T50688 C1QC4Y 25107572 IC50 = 1200 nM T50688 CKJ04T 25107573 IC50 > 100000 nM T50688 CN8Y0B 25107634 IC50 = 1780 nM T50688 C84XCZ 25107635 IC50 = 39000 nM T50688 CCY26A 25107636 IC50 > 100000 nM T50688 CO03GM 25107637 IC50 = 36500 nM T50688 CNR43C 25107638 IC50 = 2850 nM T50688 CDAC04 25107705 IC50 = 1690 nM T50688 CYS45L 25107706 IC50 = 28400 nM T50688 CYS98D 25107707 IC50 > 100000 nM T50688 CRV78W 25107708 IC50 = 54000 nM T50688 CF85WU 25107709 IC50 = 29300 nM T50688 C23YAU 25107770 IC50 = 11300 nM T50688 CQZ70E 25107771 IC50 = 9110 nM T50688 CEK7G5 25107772 IC50 = 14000 nM T50688 C3V7JU 25107773 IC50 = 2800 nM T50688 CM37RS 42607047 IC50 = 6100 nM T50688 C7K4HE 42607050 IC50 = 13000 nM T50688 CU12VE 44265226 IC50 = 0.89 nM T50688 C2POH5 44265246 IC50 = 4.76 nM T50688 CGXU38 44265249 IC50 = 0.55 nM T50688 C2E7AU 44265252 IC50 = 1 nM T50688 CD42GT 44265261 IC50 = 0.12 nM T50688 CW7O2R 44265293 IC50 = 0.57 nM T50688 CD0H6O 44268215 IC50 = 28900 nM T50688 CJ61GR 44268230 IC50 = 238 nM T50688 CRM0K3 44268269 IC50 = 25 nM T50688 C8TF4A 44268270 IC50 = 11900 nM T50688 CXP9A4 44268271 IC50 = 25 nM T50688 CVFP98 44268272 IC50 = 4 nM T50688 C5EM9S 44268276 IC50 = 252 nM T50688 CC7DE0 44268284 IC50 = 25 nM T50688 C5BM8E 44268287 IC50 > 50000 nM T50688 CJ6Z2H 44268288 IC50 > 50000 nM T50688 C2IVR7 44268289 IC50 = 17 nM T50688 CA4YL6 44268290 IC50 = 1200 nM T50688 C1LVS0 44268294 IC50 = 106 nM T50688 CP5X7D 44268296 IC50 = 225 nM T50688 CEZ7N8 44268297 IC50 = 47 nM T50688 C73WBY 44268298 IC50 = 1800 nM T50688 CS2ZJ9 44268312 IC50 = 17 nM T50688 CLJ7Y2 44268313 IC50 = 90 nM T50688 CCAR38 44268323 IC50 = 87 nM T50688 C6WRH9 44268328 IC50 = 1500 nM T50688 CH37FJ 44268364 IC50 = 4200 nM T50688 CK5IS7 44268370 IC50 = 136 nM T50688 CTD26Z 44268372 IC50 = 254 nM T50688 CRE92V 44268373 IC50 = 873 nM T50688 CC5LU4 44268375 IC50 = 320 nM T50688 CH75WX 44268376 IC50 = 447 nM T50688 CKY45X 44274285 IC50 = 3 nM T50688 CT6BV5 44279130 IC50 > 25000 nM T50688 CJY68U 44279133 IC50 = 40 nM T50688 CUB27L 44279166 IC50 = 130 nM T50688 CZ0FM9 44279167 IC50 = 3000 nM T50688 CWY2K6 44279184 IC50 > 25000 nM T50688 C7ES8I 44279259 IC50 = 70 nM T50688 C7B6NR 44279334 IC50 = 30 nM T50688 CT9RZ4 44279442 IC50 = 40 nM T50688 C42DBS 44279484 IC50 = 20 nM T50688 CC8PD2 44279492 IC50 = 6700 nM T50688 C54NRA 44279715 IC50 = 950 nM T50688 C1UJ3V 44279716 IC50 > 25000 nM T50688 CG0DB7 44279740 IC50 = 30 nM T50688 CSX2U6 44279775 IC50 = 8400 nM T50688 C2D3ML 44280044 IC50 = 250 nM T50688 C9XS5E 44281584 IC50 = 229.09 nM T50688 C31-JUL 44281660 IC50 = 270 nM T50688 C9GC6L 44281698 IC50 = 120 nM T50688 C90AZN 44281715 IC50 = 158.49 nM T50688 C7LP6X 44281716 IC50 = 640 nM T50688 CZ03QI 44281717 IC50 = 4500 nM T50688 C1MIW6 44282009 IC50 = 75.86 nM T50688 CX2PV9 44282032 IC50 = 130 nM T50688 C48KBZ 44283063 IC50 = 9.6 nM T50688 CF7C8I 44283067 IC50 = 15.6 nM T50688 C2FV0E 44283118 IC50 = 25000 nM T50688 CK0RD4 44283161 IC50 = 38 nM T50688 CXE01A 44283190 IC50 = 15.1 nM T50688 C12RPS 44283197 IC50 = 233 nM T50688 C4VW3I 44283198 IC50 = 181 nM T50688 C9ZQW4 44283202 IC50 = 11 nM T50688 C6KLR5 44283203 IC50 = 7 nM T50688 CMV19L 44283204 IC50 = 45 nM T50688 CNI3F9 44283232 IC50 = 80 nM T50688 C74CWT 44283235 IC50 = 0.71 nM T50688 CN45TM 44283254 IC50 = 69 nM T50688 CVS5P4 44283263 IC50 = 641 nM T50688 CX2PH8 44283275 IC50 = 121 nM T50688 CH29QO 44283299 IC50 = 152 nM T50688 C7FCI9 44283300 IC50 = 9.1 nM T50688 C2M4JN 44283364 IC50 = 528 nM T50688 C5R6PO 44283380 IC50 = 125 nM T50688 C09EHM 44283639 IC50 = 661 nM T50688 C20PIF 44285420 IC50 = 1000 nM T50688 C6MH2U 44285421 IC50 = 15848.93 nM T50688 CA3TB7 44285426 IC50 = 39810.72 nM T50688 CNQ7E3 44285443 IC50 = 2511.89 nM T50688 C5EG0I 44285469 IC50 < 10000 nM T50688 CC2WX5 44285470 IC50 = 25.12 nM T50688 CAD27K 44285483 IC50 = 1584.89 nM T50688 CWD58N 44285484 IC50 = 1995.26 nM T50688 CF3W1R 44285487 IC50 = 199.53 nM T50688 C4CYX6 44285495 IC50 = 1000 nM T50688 C46ICR 44285506 IC50 = 1258.93 nM T50688 CAE80Z 44285637 IC50 = 250 nM T50688 CH53NW 44285682 IC50 = 3981.07 nM T50688 C8ABI1 44287422 IC50 = 20000 nM T50688 CYAQ68 44287423 IC50 = 29900 nM T50688 C3X2LJ 44287428 IC50 = 50000 nM T50688 CQ3AF6 44287550 IC50 = 24000 nM T50688 C5PCQ0 44287569 IC50 = 8 nM T50688 C29LXN 44287570 IC50 = 28 nM T50688 CQL21H 44287634 IC50 = 20000 nM T50688 C7YE0G 44287879 IC50 = 2700 nM T50688 CTQV91 44290954 IC50 = 1220 nM T50688 CE3K5Y 44290956 IC50 > 100000 nM T50688 CNFY65 44291131 IC50 = 5000 nM T50688 CY98UX 44291379 IC50 = 120 nM T50688 CE3FQ7 44291381 IC50 = 510 nM T50688 C7XC0O 44291383 IC50 = 560 nM T50688 C6D0JM 44291385 IC50 = 1070 nM T50688 CK26HJ 44291464 IC50 > 100000 nM T50688 CKO25V 44291466 IC50 = 2 nM T50688 CM7H6A 44291467 IC50 > 100000 nM T50688 C9ZF8D 44291479 IC50 = 5 nM T50688 C7FIO4 44291481 IC50 = 20 nM T50688 C39PZH 44291483 IC50 = 40 nM T50688 C6O9CT 44291485 IC50 = 20 nM T50688 CUZ73G 44291499 IC50 = 2000 nM T50688 CAP83N 44291732 IC50 = 270 nM T50688 C0Q8WF 44291756 IC50 = 110 nM T50688 C6PHG5 44291757 IC50 = 78000 nM T50688 CQ2XC4 44291759 IC50 = 770 nM T50688 C5SM4O 44294710 IC50 = 96 nM T50688 C1CO9H 44294758 IC50 = 120 nM T50688 C6Y9PG 44294759 IC50 = 70 nM T50688 CO0JI2 44294760 IC50 = 3000 nM T50688 C37PMJ 44295006 IC50 = 200 nM T50688 CJ4PE2 44295049 IC50 = 25000 nM T50688 CR7QI4 44295086 IC50 > 20000 nM T50688 CVE2D8 44295087 IC50 = 1600 nM T50688 CHB3R8 44295112 IC50 = 470 nM T50688 C8N3TI 44295122 IC50 = 3 nM T50688 CZA76L 44295135 IC50 > 20000 nM T50688 CYF93D 44295211 IC50 > 25000 nM T50688 C8N3ZC 44295212 IC50 = 2000 nM T50688 C89PDG 44295213 IC50 = 3000 nM T50688 CTN25K 44295235 IC50 = 220 nM T50688 CD91SB 44296029 Ki = 11000 nM T50688 CESC21 44296030 Ki = 1100 nM T50688 C0NBT5 44296032 Ki = 8200 nM T50688 C0EIC6 44296106 Ki = 160000 nM T50688 CDX37F 44296107 Ki = 8500 nM T50688 CXM37J 44296126 Ki = 14000 nM T50688 CBY2N4 44296179 Ki = 5000 nM T50688 C1BDP7 44296242 Ki = 41500 nM T50688 C0R6QX 44296243 Ki = 32000 nM T50688 CYA4E9 44296248 Ki = 8000 nM T50688 CAFV23 44296408 IC50 > 3000 nM T50688 C74ZEK 44296431 IC50 > 3000 nM T50688 CFN8Q6 44296449 Ki = 3650 nM T50688 C1YD3S 44296450 Ki > 50000 nM T50688 CYSG84 44296458 IC50 > 3000 nM T50688 C4FI2N 44296514 IC50 > 3000 nM T50688 C9U3QW 44296519 IC50 > 3000 nM T50688 CQHJ16 44296532 IC50 > 3000 nM T50688 CX0Q1T 44296543 Ki = 40500 nM T50688 C2TE9R 44296548 IC50 > 3000 nM T50688 C5GY7H 44296579 IC50 > 3000 nM T50688 CYZT93 44296580 IC50 > 3000 nM T50688 C7S1JY 44296604 IC50 > 3000 nM T50688 CP89DV 44296642 IC50 > 3000 nM T50688 C1KYA3 44296682 IC50 = 10000 nM T50688 CH0JP8 44296684 IC50 = 180 nM T50688 CC0TN6 44296689 IC50 = 10000 nM T50688 CUEC26 44296697 IC50 = 350 nM T50688 C2NU5B 44296726 IC50 = 550 nM T50688 CZ17IX 44296740 IC50 > 3000 nM T50688 C3A7PY 44296742 IC50 = 10000 nM T50688 CAH14O 44296744 IC50 = 850 nM T50688 CZG93V 44296762 IC50 > 10000 nM T50688 CJRK46 44296797 IC50 > 10000 nM T50688 CY26ES 44296824 IC50 > 3000 nM T50688 CCEF03 44296851 IC50 > 3000 nM T50688 C27UPR 44296852 IC50 > 3000 nM T50688 C0FK5Q 44296857 IC50 > 3000 nM T50688 CR9U6E 44296858 IC50 > 3000 nM T50688 CS2E4W 44296864 IC50 > 10000 nM T50688 CS62KL 44296866 IC50 = 5000 nM T50688 C0KY3B 44296868 IC50 > 10000 nM T50688 C27HKT 44296892 IC50 = 200 nM T50688 CVAF21 44296901 IC50 > 3000 nM T50688 C5O8IC 44296903 IC50 > 3000 nM T50688 C4ZG0D 44297806 IC50 = 1100 nM T50688 CC4LU8 44297807 IC50 = 1600 nM T50688 C6F1CD 44297814 IC50 = 10000 nM T50688 CGZ82H 44297845 IC50 = 300000 nM T50688 C0KX7H 44297846 IC50 = 530 nM T50688 CY35IN 44297847 IC50 = 2000 nM T50688 CX2PK9 44300973 IC50 = 7000 nM T50688 CA78QS 44300974 IC50 > 10000 nM T50688 CPJU95 44300981 IC50 > 10000 nM T50688 C9YT1L 44300986 IC50 = 65 nM T50688 CWP15R 44301007 IC50 = 19 nM T50688 CL84GY 44301008 IC50 = 28 nM T50688 CSCA61 44301010 IC50 > 10000 nM T50688 CX3Y4B 44301021 IC50 = 27 nM T50688 CPW8S2 44301026 IC50 = 9 nM T50688 CP1F5U 44301032 IC50 = 57 nM T50688 COX26S 44301040 IC50 = 15 nM T50688 C9OU5P 44301044 IC50 = 12 nM T50688 CO6HW2 44301065 Ki = 2.3 nM T50688 CWP52F 44301068 IC50 = 9000 nM T50688 CLCO73 44301083 IC50 > 10000 nM T50688 C6DZ3F 44301106 IC50 = 11 nM T50688 CC4LO8 44301244 IC50 = 3000 nM T50688 CIJ28H 44301270 IC50 = 13 nM T50688 C4W3LK 44301283 IC50 = 51 nM T50688 C7VC5T 44301286 IC50 > 10000 nM T50688 CBT2O3 44301295 IC50 = 15 nM T50688 CI39XL 44301310 IC50 > 10000 nM T50688 CZ14EM 44301350 IC50 > 10000 nM T50688 C3MSY1 44301352 IC50 = 8 nM T50688 C5OA0I 44301363 IC50 = 81 nM T50688 C0G3LI 44301379 IC50 = 8 nM T50688 CWBC76 44301520 Ki = 2.1 nM T50688 C9QIP0 44303539 IC50 = 500 nM T50688 CC3H4P 44303550 IC50 = 105 nM T50688 C39FGB 44303551 IC50 = 1350 nM T50688 CA3X5V 44303563 IC50 = 40 nM T50688 C4AO7I 44303592 IC50 = 17 nM T50688 CPX4L1 44303611 IC50 = 65 nM T50688 CRJP53 44303836 IC50 = 17 nM T50688 CTBK03 44303837 IC50 = 35 nM T50688 CO5KC2 44304468 IC50 = 20000 nM T50688 CR30VX 44304469 IC50 = 6 nM T50688 CC9H7K 44304480 IC50 = 3.5 nM T50688 CJ68BM 44304481 IC50 = 0.5 nM T50688 CYKT90 44304483 IC50 = 4.7 nM T50688 CA09ZS 44304485 IC50 = 210 nM T50688 C5TY8F 44304495 IC50 = 434 nM T50688 CK7YC1 44304496 IC50 = 12 nM T50688 C4E1TI 44304497 IC50 = 18 nM T50688 CEY8V5 44304498 IC50 = 1.4 nM T50688 CT5KO2 44304499 IC50 = 500 nM T50688 CPD08J 44304500 IC50 = 25 nM T50688 CE42YV 44304526 IC50 = 35 nM T50688 CB3A9F 44304531 IC50 = 6 nM T50688 CBZ12F 44304532 IC50 = 11.4 nM T50688 C3FJ5K 44304541 IC50 = 80 nM T50688 CEX49N 44304547 IC50 = 75000 nM T50688 CSNM29 44304548 IC50 = 14 nM T50688 C5KQ1N 44304549 IC50 = 4850 nM T50688 C1IYO2 44304571 IC50 = 5.7 nM T50688 CZG56O 44304572 IC50 = 260 nM T50688 CR25CI 44304573 IC50 = 4600 nM T50688 C8KS3L 44304576 IC50 = 75 nM T50688 C1K4WA 44304587 IC50 = 20 nM T50688 C12GLJ 44304588 IC50 = 7.5 nM T50688 C0WA7Z 44304604 IC50 = 110 nM T50688 C47YWJ 44304607 IC50 = 31 nM T50688 CFPV93 44304608 IC50 = 5.6 nM T50688 CE1N6V 44304609 IC50 = 43 nM T50688 C21SEM 44304613 IC50 = 5.3 nM T50688 CFC0P2 44304619 IC50 = 12 nM T50688 C2G4XE 44304624 IC50 = 6.6 nM T50688 CM78IK 44304645 IC50 = 33 nM T50688 CR9Z7P 44304646 IC50 = 100 nM T50688 CF82AW 44304647 IC50 = 2.9 nM T50688 CGRU80 44304650 IC50 = 2.6 nM T50688 CY2R9X 44304655 IC50 = 70 nM T50688 CC5B3K 44304656 IC50 = 150 nM T50688 CFTN27 44304659 IC50 = 4780 nM T50688 CL5K9N 44304660 IC50 = 4 nM T50688 C3E5VJ 44304661 IC50 = 22 nM T50688 CAVK91 44304674 IC50 = 38 nM T50688 CTY01P 44304675 IC50 = 6.8 nM T50688 CWCM82 44304679 IC50 = 4 nM T50688 CKR7Y0 44304718 IC50 = 1.6 nM T50688 CS30ZM 44304723 IC50 = 3 nM T50688 CLI42H 44304724 IC50 = 35 nM T50688 C8A3KN 44304725 IC50 = 310 nM T50688 CX1E3B 44304726 IC50 = 9.5 nM T50688 CKN1E4 44304733 IC50 = 590 nM T50688 CE87NH 44304744 IC50 = 19 nM T50688 C7FOJ3 44304745 IC50 = 132 nM T50688 C1VY6U 44304785 IC50 = 4.5 nM T50688 CPS9C0 44304808 IC50 = 5.4 nM T50688 C1NFJ0 44304842 IC50 = 4 nM T50688 CMZC63 44304843 IC50 = 2.8 nM T50688 CK68QA 44304844 IC50 = 2.7 nM T50688 CRN6V1 44304845 IC50 = 7 nM T50688 C5YNE8 44304874 IC50 = 1 nM T50688 CEA9H3 44304875 IC50 = 29 nM T50688 CMTQ46 44304901 IC50 = 8 nM T50688 C2H8DU 44304902 IC50 = 28 nM T50688 C0CMR7 44304903 IC50 = 1060 nM T50688 CX69MO 44304904 IC50 = 22 nM T50688 CVDR16 44304905 IC50 = 3.6 nM T50688 C8RYE9 44304952 IC50 = 17 nM T50688 CG2N3X 44304953 IC50 = 500 nM T50688 CME60P 44304954 IC50 = 231 nM T50688 CS12DA 44305003 IC50 = 2.5 nM T50688 CM67BS 44305004 IC50 = 12 nM T50688 CH0F7S 44305008 IC50 = 103 nM T50688 CF9ZI0 44305062 IC50 = 4185 nM T50688 CG6P3Y 44305143 IC50 = 4 nM T50688 CI3OA0 44305239 IC50 = 1700 nM T50688 CIF0U5 44305476 IC50 = 49 nM T50688 CWF31T 44305508 IC50 = 140 nM T50688 C5Y3IP 44305645 IC50 = 2700 nM T50688 CP5O4B 44305658 IC50 = 3300 nM T50688 CQOS32 44305694 IC50 = 31 nM T50688 C1A5QE 44305716 IC50 = 44 nM T50688 CA82VR 44305726 IC50 = 210 nM T50688 CB21HD 44305872 IC50 = 35000 nM T50688 CJ9C1D 44306030 IC50 = 7000 nM T50688 CM9ZV1 44306543 IC50 = 707945.78 nM T50688 CX40ZQ 44306545 IC50 = 30199.52 nM T50688 CO8LM1 44306547 IC50 = 741310.24 nM T50688 C5QM2G 44306568 IC50 = 100 nM T50688 CUY0W7 44306569 IC50 = 200 nM T50688 CL59SB 44306616 IC50 = 758577.58 nM T50688 C6K3TO 44306710 IC50 = 7585.78 nM T50688 CP09ST 44306715 IC50 = 52480.75 nM T50688 CCH6E0 44306731 IC50 = 100 nM T50688 CE78JY 44306747 IC50 = 100000 nM T50688 CD6C2J 44306765 IC50 = 200 nM T50688 C9F5ZP 44306766 IC50 = 2000 nM T50688 CCU8M2 44306772 IC50 = 630.96 nM T50688 CC9N4L 44306786 IC50 = 302 nM T50688 C0BXH2 44306842 IC50 = 363.08 nM T50688 CL3AD9 44306932 IC50 = 128.82 nM T50688 C19BET 44306947 IC50 = 199526.23 nM T50688 CLM91S 44307016 IC50 = 1905.46 nM T50688 C7L5JI 44307035 IC50 = 9120.11 nM T50688 CAD8H2 44307043 IC50 = 6456.54 nM T50688 CHLY12 44307056 IC50 = 5011.87 nM T50688 C8WD1N 44307070 IC50 = 5248.07 nM T50688 C3YZB0 44307099 IC50 = 91201.08 nM T50688 CBZ6D8 44307217 IC50 = 3467.37 nM T50688 CIX09R 44307237 IC50 = 2511.89 nM T50688 CN36PV 44307238 IC50 = 239.88 nM T50688 C0DGS2 44307241 IC50 = 794.33 nM T50688 CJ7BQ2 44307259 IC50 = 109647.82 nM T50688 C8A5MJ 44307296 IC50 = 758577.58 nM T50688 C80FZA 44307297 IC50 = 33113.11 nM T50688 CI59NO 44307365 IC50 = 4073.8 nM T50688 C6B5JQ 44315195 IC50 = 2.7 nM T50688 CK2B7R 44315447 IC50 = 2.6 nM T50688 CMZJ69 44315702 IC50 = 23.7 nM T50688 CJN6H3 44315779 IC50 = 2 nM T50688 C8LQ3E 44315780 IC50 = 20 nM T50688 C5XE1O 44315792 IC50 = 20 nM T50688 CPT6R4 44315793 IC50 = 20 nM T50688 C2TE0B 44316045 IC50 = 6 nM T50688 C7P1CL 44316059 IC50 = 7 nM T50688 CDVZ48 44316106 IC50 = 2 nM T50688 C9B8CD 44316156 IC50 = 5 nM T50688 CUBM67 44316184 IC50 = 3 nM T50688 CA0P1Z 44316450 IC50 = 52 nM T50688 CAI6P7 44316522 IC50 = 4.8 nM T50688 C8DRY2 44316532 IC50 = 4 nM T50688 CYTL98 44316560 IC50 = 200 nM T50688 C6QU9I 44316563 IC50 > 50000 nM T50688 C4U2XO 44316579 IC50 = 224 nM T50688 C13IEA 44317739 IC50 = 8 nM T50688 C5UTI9 44318089 IC50 = 16 nM T50688 C9XH0Y 44318100 IC50 = 32 nM T50688 CZ5R4V 44318107 IC50 = 129 nM T50688 C97YTO 44318110 IC50 = 53 nM T50688 COB28I 44318124 IC50 = 47 nM T50688 CA65ZG 44318139 IC50 = 78 nM T50688 CMO5P7 44318169 IC50 = 630 nM T50688 CR3D0I 44319347 IC50 = 41 nM T50688 CT73SX 44319352 IC50 = 260 nM T50688 CAP0X7 44319363 IC50 = 56 nM T50688 C20MFD 44319365 IC50 = 1700 nM T50688 CJUP56 44319437 IC50 = 680 nM T50688 CV9CP5 44319448 IC50 = 100 nM T50688 C58SYJ 44319608 IC50 = 1800 nM T50688 CFN08C 44319632 IC50 = 220 nM T50688 CS67MW 44320027 IC50 > 1000 nM T50688 C91SAN 44320056 IC50 > 1000 nM T50688 CC4UG8 44320077 IC50 > 1000 nM T50688 CAVD13 44320155 IC50 > 1000 nM T50688 C95KAZ 44320173 IC50 = 88 nM T50688 CSV1C2 44320174 IC50 > 1000 nM T50688 C7GXI5 44320211 IC50 = 540 nM T50688 CWS24X 44320274 IC50 > 1000 nM T50688 C1W8ID 44320282 IC50 = 30 nM T50688 C6F7OI 44320305 IC50 = 340 nM T50688 CN08CV 44320306 IC50 > 1000 nM T50688 CVX0F7 44320364 IC50 = 720 nM T50688 C3SXG5 44320893 IC50 = 18 nM T50688 C5FAY7 44321219 IC50 > 1000 nM T50688 CC25UD 44321220 IC50 > 1000 nM T50688 C8X5IP 44321235 IC50 > 100 nM T50688 CME9U8 44321274 IC50 = 6 nM T50688 C82THY 44321295 IC50 = 8.7 nM T50688 CN41VK 44321296 IC50 = 1.4 nM T50688 CA5ZE4 44321313 IC50 = 62 nM T50688 CSX9Z2 44321328 IC50 = 9.8 nM T50688 CM8P0R 44321368 IC50 = 100 nM T50688 C5PBW9 44321507 IC50 > 100 nM T50688 C26IPS 44321551 IC50 > 100 nM T50688 C5ZAL0 44321567 IC50 = 730 nM T50688 C7UOZ5 44321682 IC50 > 100 nM T50688 C4BTK5 44321683 IC50 = 42 nM T50688 CFSI83 44321913 IC50 = 440 nM T50688 CIX50Z 44321934 IC50 = 2.7 nM T50688 C82IOL 44322337 IC50 = 0.6 nM T50688 C7PYO4 44322627 IC50 = 0.12 nM T50688 C5AG3Y 44322644 IC50 = 0.51 nM T50688 CKY2F1 44329896 Ki > 25000 nM T50688 CKXQ61 44329897 Ki > 25000 nM T50688 C79CIF 44329957 IC50 > 10000 nM T50688 C91OLV 44329959 IC50 > 10000 nM T50688 CUQ2M9 44330009 IC50 = 7100 nM T50688 CUK74V 44330015 Ki = 2100 nM T50688 C38PGY 44330039 Ki > 25000 nM T50688 CF9SY3 44330086 Ki > 25000 nM T50688 CAT6Y2 44330200 Ki > 25000 nM T50688 CSIG14 44333548 IC50 > 10000 nM T50688 C2E3VH 44333550 IC50 = 1700 nM T50688 C23DVQ 44333621 IC50 > 10000 nM T50688 C4X3KB 44333751 IC50 = 860 nM T50688 CY84IA 44333752 IC50 > 10000 nM T50688 CLE04Q 44333753 IC50 = 5200 nM T50688 CE8G2W 44336187 IC50 = 68200 nM T50688 C67WVQ 44336210 IC50 > 200000 nM T50688 CUG16W 44336218 Ki = 780 nM T50688 C3V7ZN 44336250 IC50 > 200000 nM T50688 C9KXF4 44336279 IC50 = 52000 nM T50688 C7D6EU 44336336 Ki = 5300 nM T50688 CHDR52 44336478 IC50 > 10000 nM T50688 CB5QP3 44336511 IC50 > 10000 nM T50688 C2R8GS 44336762 IC50 > 10000 nM T50688 CW9RO6 44336769 IC50 = 90 nM T50688 C52LJU 44336770 IC50 > 8000 nM T50688 CDLE79 44337733 Ki = 47000 nM T50688 CN0K7Q 44337734 Ki = 30000 nM T50688 CY5R8E 44337742 Ki = 29000 nM T50688 CAQZ60 44337758 Ki = 2750 nM T50688 CA47BJ 44337773 Ki = 28000 nM T50688 C4LEU0 44340569 IC50 = 667 nM T50688 CTRQ17 44341096 IC50 = 198000 nM T50688 CX46NY 44343237 IC50 > 25000 nM T50688 CPW4H8 44343633 IC50 = 59 nM T50688 C0R2ZS 44343700 IC50 = 20 nM T50688 CO8P3W 44343737 IC50 = 3.5 nM T50688 CG83NM 44343750 IC50 = 50 nM T50688 C6IC2T 44343773 IC50 = 160 nM T50688 C95EFU 44343896 IC50 > 90 nM T50688 CELV48 44350342 IC50 > 1000000 nM T50688 CP4R1A 44350344 IC50 = 1400 nM T50688 CDE56C 44350392 IC50 = 34000 nM T50688 CEP6G1 44350415 IC50 > 100000 nM T50688 C7J9NH 44350447 IC50 = 7300 nM T50688 CH6UX8 44350448 IC50 = 11000 nM T50688 C4C2PF 44350449 IC50 = 5600 nM T50688 CP4TD3 44350450 IC50 > 100000 nM T50688 C2V8FY 44350717 IC50 = 330 nM T50688 CMLD50 44350731 IC50 = 1200 nM T50688 CEFL68 44351621 IC50 > 200000 nM T50688 CCQ08X 44351628 Ki = 4 nM T50688 CH1O6S 44351664 Ki = 1900 nM T50688 C61BOQ 44351682 Ki = 106 nM T50688 C6SN9U 44351704 Ki = 271 nM T50688 CM5X6P 44351788 IC50 = 76600 nM T50688 C8XB4U 44351866 Ki = 3130 nM T50688 C1QGR5 44351885 IC50 = 17700 nM T50688 C9FUW5 44352004 IC50 = 70000 nM T50688 CEQ93X 44353584 IC50 = 2400 nM T50688 CCAZ98 44359505 IC50 = 1100 nM T50688 CTI3C9 44359535 IC50 = 5200 nM T50688 CK04UD 44359546 IC50 = 39000 nM T50688 CB42IU 44359616 IC50 = 6400 nM T50688 CA1DP5 44359630 IC50 = 2500 nM T50688 CZ68AH 44359656 IC50 = 3700 nM T50688 CIPX97 44359766 IC50 > 100000 nM T50688 CNLV75 44359767 IC50 > 100000 nM T50688 CV8JY9 44362649 IC50 = 1300 nM T50688 C68QVP 44362650 IC50 = 15000 nM T50688 CPT04Y 44362651 IC50 = 45000 nM T50688 C35BCT 44362902 IC50 = 14000 nM T50688 C3TSZ6 44362908 IC50 = 170 nM T50688 CTO32M 44362922 IC50 = 510 nM T50688 C80OTL 44362923 IC50 = 170 nM T50688 CI2UG4 44362951 IC50 > 300000 nM T50688 CY07RK 44363126 Ki = 8 nM T50688 CN9M2P 44363186 Ki = 90 nM T50688 CIY64N 44364493 IC50 = 110 nM T50688 CSRM97 44364562 IC50 = 140 nM T50688 C6EUK9 44364573 IC50 = 229.09 nM T50688 CXO4Y9 44364601 IC50 = 4466.84 nM T50688 C1LIW7 44364621 IC50 = 63 nM T50688 C6IFM5 44364673 IC50 = 6.1 nM T50688 C92MKD 44364694 IC50 = 210 nM T50688 CI7BH0 44364738 IC50 = 1500 nM T50688 CHK71U 44365992 IC50 = 17.9 nM T50688 C3E1ID 44366016 IC50 = 0.37 nM T50688 CT7DQ8 44366048 IC50 = 48 nM T50688 C2QNL7 44366077 IC50 = 0.36 nM T50688 CU0WI3 44366139 IC50 = 66.8 nM T50688 CD8RZ0 44366167 IC50 = 0.24 nM T50688 C1WHZ3 44366226 IC50 = 13.5 nM T50688 C3AM0D 44366227 IC50 = 0.1 nM T50688 CZH23I 44366235 IC50 = 0.1 nM T50688 CT58MH 44366375 IC50 = 0.5 nM T50688 CNZQ89 44366409 IC50 = 157 nM T50688 C1J2CW 44366410 IC50 > 10000 nM T50688 CN2L3U 44367917 Ki = 500 nM T50688 CVGB31 44368140 Ki = 2 nM T50688 CO1SR9 44368152 Ki > 50000 nM T50688 CB0TF6 44368570 IC50 = 776 nM T50688 C47OWF 44368757 IC50 > 10000 nM T50688 CAS01N 44372658 IC50 = 21000 nM T50688 CGIP26 44372909 IC50 = 10400 nM T50688 CYD6H2 44372941 IC50 = 30000 nM T50688 C4NU0I 44372954 IC50 = 81000 nM T50688 C6B5FO 44372955 IC50 = 31000 nM T50688 CFO34W 44372962 IC50 = 100000 nM T50688 COYQ79 44372977 IC50 = 30000 nM T50688 CHS2V0 44373024 IC50 > 30000 nM T50688 C8WQ3F 44373152 IC50 = 8900 nM T50688 CKR0X7 44373170 IC50 = 87000 nM T50688 C6X9UK 44373176 IC50 = 24000 nM T50688 CAIJ06 44373182 IC50 > 30000 nM T50688 C09MLI 44373256 IC50 = 30000 nM T50688 C89GTD 44373300 IC50 > 100000 nM T50688 CU12HA 44373303 IC50 = 19000 nM T50688 C68DAQ 44373341 IC50 = 45000 nM T50688 CQE4R3 44373603 IC50 = 30000 nM T50688 C4V3KU 44373605 IC50 = 30000 nM T50688 CJC35L 44376533 IC50 = 0.54 nM T50688 CXON13 44376539 IC50 = 0.36 nM T50688 C4D2SH 44376550 IC50 = 1 nM T50688 C68SYL 44376551 IC50 = 0.36 nM T50688 CJA9Q6 44376578 IC50 = 7.6 nM T50688 CA3UC1 44376579 IC50 = 1.7 nM T50688 CHV7T9 44376681 IC50 = 2.2 nM T50688 CA5FS3 44376772 IC50 = 48000 nM T50688 CC0WL9 44376773 IC50 = 0.37 nM T50688 CHZ0Q1 44376790 IC50 = 7.9 nM T50688 C8O7TA 44378089 Ki = 110 nM T50688 C7HTK1 44378106 Ki = 2650 nM T50688 C5XJ1T 44378195 Ki = 2.1 nM T50688 C7L5ZE 44378218 Ki = 26 nM T50688 C8MJ9S 44378222 Ki = 65 nM T50688 CJE6O9 44378223 Ki = 25300 nM T50688 CWK48R 44378224 Ki = 820 nM T50688 C4PIV6 44378302 Ki > 10000 nM T50688 C2X4KT 44378303 Ki = 82 nM T50688 CAE13J 44378307 Ki = 27 nM T50688 CQ3EA4 44378320 Ki = 9.5 nM T50688 CPAQ56 44378327 Ki = 15100 nM T50688 CM5YQ1 44378331 Ki = 2.5 nM T50688 CD6C9K 44378336 Ki = 7040 nM T50688 C7CTJ8 44378360 Ki > 100000 nM T50688 C4K6LW 44378361 Ki = 280 nM T50688 CTZO38 44378378 Ki = 1250 nM T50688 C89JAB 44378400 Ki = 430 nM T50688 C7O9AP 44378401 Ki = 20 nM T50688 C3C8VJ 44378494 Ki = 188 nM T50688 C4SKJ9 44378558 Ki = 2.1 nM T50688 CL9UT4 44378583 Ki = 135 nM T50688 C42USR 44378584 Ki = 77 nM T50688 CN9Z4W 44378585 Ki = 610 nM T50688 CR51ID 44378699 IC50 = 16 nM T50688 CAO29R 44378701 IC50 = 150 nM T50688 CWP41H 44378720 IC50 = 3 nM T50688 C2U6ZA 44378747 IC50 = 14 nM T50688 CT9H2B 44378748 IC50 = 3 nM T50688 CNS75M 44378858 IC50 = 20 nM T50688 CENU52 44378961 IC50 = 2 nM T50688 C3UQT1 44378995 IC50 = 38 nM T50688 CHC7N5 44379066 IC50 = 430 nM T50688 CSA20X 44381676 IC50 = 109.65 nM T50688 CZTW31 44381688 IC50 = 39.81 nM T50688 C6R8KC 44381737 IC50 = 85.11 nM T50688 CY1U0D 44381774 IC50 = 114.82 nM T50688 CL9FU3 44381783 IC50 = 40.74 nM T50688 CMB53C 44381797 IC50 = 38.02 nM T50688 CQ9UO5 44381825 IC50 = 151.36 nM T50688 CQ06HD 44381864 IC50 = 125.89 nM T50688 C42PBL 44381878 IC50 = 331.13 nM T50688 CKE79T 44381879 IC50 = 190.55 nM T50688 CS9V1U 44381881 IC50 = 380 nM T50688 CS51QV 44381885 IC50 = 18197.01 nM T50688 CLGQ87 44381898 IC50 = 29000 nM T50688 C84FJL 44381902 IC50 = 134.9 nM T50688 CJ5MH7 44381905 IC50 = 40.74 nM T50688 CDV3U9 44381908 IC50 = 130 nM T50688 CN5EU2 44381918 IC50 = 34 nM T50688 C4TCZ8 44381942 IC50 = 230000 nM T50688 C48UAI 44381947 IC50 = 75.86 nM T50688 C8B3LU 44381948 IC50 = 42.66 nM T50688 C45BHN 44381953 IC50 = 9200 nM T50688 C9ZOW8 44381959 IC50 = 40.74 nM T50688 CQ08VO 44381964 IC50 = 1659.59 nM T50688 CP3D6M 44381975 IC50 = 33113.11 nM T50688 C5ERH4 44381977 IC50 = 44.67 nM T50688 C6ECI7 44381991 IC50 = 37.15 nM T50688 C1NXQ2 44381992 IC50 = 2800 nM T50688 C6K4IV 44382000 IC50 = 186.21 nM T50688 CNQY28 44382002 IC50 = 707.95 nM T50688 C5O1SY 44382014 IC50 = 30.9 nM T50688 CN21FS 44382015 IC50 = 38.02 nM T50688 C9D6RZ 44382030 IC50 = 79.43 nM T50688 C8RYM7 44382051 IC50 = 501.19 nM T50688 COZA49 44382083 IC50 = 40.74 nM T50688 CSW25H 44382135 IC50 = 79.43 nM T50688 CW80ED 44382136 IC50 = 79.43 nM T50688 CZB83R 44382356 IC50 = 4900 nM T50688 C3L4XR 44382357 IC50 = 270 nM T50688 C1GOE5 44382394 IC50 = 23 nM T50688 CE18UX 44382445 IC50 = 13 nM T50688 CE7L0H 44382481 IC50 = 331131.12 nM T50688 C3W0TK 44382482 IC50 > 30000 nM T50688 CWDC18 44383692 IC50 > 100000 nM T50688 CAY53C 44383697 IC50 = 3600 nM T50688 CB2KW6 44383745 IC50 = 12000 nM T50688 C3Q0GH 44383752 IC50 = 800 nM T50688 CBH12Q 44383755 IC50 = 53000 nM T50688 CY70ZS 44383803 IC50 = 2600 nM T50688 CRJ1M9 44383805 IC50 = 23000 nM T50688 CCR0M8 44383848 IC50 = 17000 nM T50688 C1E0CL 44384154 IC50 = 850 nM T50688 C28CSF 44384225 IC50 = 3500 nM T50688 CG0I7U 44384233 IC50 = 170 nM T50688 CZOH46 44384400 IC50 = 55000 nM T50688 C3VKC9 44384418 IC50 = 47000 nM T50688 CWY40J 44384448 IC50 = 3600 nM T50688 CWX1O8 44384452 IC50 = 1500 nM T50688 CR51GC 44384509 IC50 = 13000 nM T50688 C2PXN3 44384519 IC50 > 100000 nM T50688 C1SKZ8 44384644 IC50 = 690 nM T50688 CBV4X3 44384707 IC50 = 1900 nM T50688 C1U0OM 44384812 IC50 = 360 nM T50688 CD95EQ 44384863 IC50 > 100000 nM T50688 CE1LV5 44385010 IC50 = 9 nM T50688 CM27CY 44385012 IC50 = 11 nM T50688 CRO89U 44385014 IC50 = 16 nM T50688 CACQ93 44385048 IC50 = 13 nM T50688 CZIJ16 44385402 IC50 = 12000 nM T50688 CVYB52 44393453 IC50 = 170 nM T50688 CAD12L 44393517 IC50 = 25 nM T50688 CS2I9D 44394317 IC50 = 13 nM T50688 CL9GN5 44394834 IC50 = 79.3 nM T50688 CIS4X5 44394933 IC50 = 15719 nM T50688 CA30XW 44394981 IC50 = 56.4 nM T50688 C4X2PI 44395065 IC50 = 2850 nM T50688 C0IN2J 44395933 IC50 = 1100 nM T50688 CL1AJ8 44395975 IC50 = 2900 nM T50688 CK4YH8 44396023 IC50 = 870 nM T50688 C3DN8C 44396062 IC50 = 4700 nM T50688 CC62KR 44400343 Ki = 5190 nM T50688 C8OA0D 44400345 Ki = 59050 nM T50688 CK5ZW7 44400347 Ki = 3940 nM T50688 CE18LD 44407524 IC50 = 423 nM T50688 CZ4O2D 44407529 IC50 = 22 nM T50688 CV36MS 44407555 IC50 = 91 nM T50688 C9XIY5 44407556 IC50 = 64 nM T50688 C1E7HF 44407560 IC50 = 17 nM T50688 CW8MQ7 44407577 IC50 = 126 nM T50688 C03KFP 44407668 IC50 = 216 nM T50688 C7CP1X 44407779 IC50 = 1217 nM T50688 C5LF3K 44412296 IC50 = 16.2 nM T50688 C87QUH 44455076 IC50 > 10000 nM T50688 C7A1WN 44458461 IC50 = 1.2 nM T50688 CX0A3S 44458463 IC50 = 1.5 nM T50688 C6L5HF 44458472 IC50 = 102 nM T50688 CB30EA 44458473 IC50 = 0.86 nM T50688 CV9OB8 44458488 IC50 = 0.55 nM T50688 C5Y4DU 44458504 IC50 = 260 nM T50688 CMR2F1 44459058 IC50 = 9700 nM T50688 C13NVH 44459345 IC50 > 100000 nM T50688 CDKG38 44459361 IC50 = 160 nM T50688 C9G5ZA 44459507 IC50 = 240 nM T50688 C70KPC 44459508 IC50 = 270 nM T50688 C9X7AN 44459610 IC50 = 332 nM T50688 C3UHE0 44459630 IC50 = 8 nM T50688 C4YO1S 44459631 IC50 = 160 nM T50688 C8V9BY 44459642 IC50 = 250 nM T50688 CM03VR 44459643 IC50 = 100000 nM T50688 CKR0S7 44459645 IC50 = 100000 nM T50688 CQRA01 44459646 IC50 = 2400 nM T50688 C2T4XF 44459647 IC50 = 3450 nM T50688 C9MTP5 44459648 IC50 = 50000 nM T50688 CQU0Y3 44459649 IC50 = 250 nM T50688 CG5T2Y 44459650 IC50 = 319 nM T50688 CX4JZ1 44459666 IC50 = 2 nM T50688 C9WBE0 44459668 IC50 = 30000 nM T50688 CGLX83 44459727 IC50 = 9700 nM T50688 COKC08 44459728 IC50 = 5000 nM T50688 C6O8ZD 44459743 IC50 = 4 nM T50688 CMU71G 44459764 IC50 = 2 nM T50688 C4HV0D 44459765 IC50 = 830 nM T50688 C0V8SK 44459766 IC50 = 60 nM T50688 CWR7Q1 44459770 IC50 = 1 nM T50688 CAXJ53 44459773 IC50 = 7 nM T50688 CVS29Q 44459774 IC50 = 616 nM T50688 CU95CL 44459843 IC50 = 23 nM T50688 CFJC10 44459851 IC50 = 43 nM T50688 CGJ3Y7 44459852 IC50 = 210 nM T50688 C56CVI 44459873 IC50 = 1160 nM T50688 C9CAP7 44459874 IC50 = 260 nM T50688 C8XH7Y 44461765 Ki = 2.5 nM T50688 C5DA7R 44461812 Ki = 1.3 nM T50688 CH2XK6 44461891 Ki = 1.5 nM T50688 C8N6XQ 44462164 IC50 = 11 nM T50688 C1HQL7 44462165 IC50 = 28 nM T50688 C9PWK3 44462196 IC50 = 32 nM T50688 C87CFQ 44462263 IC50 = 1060 nM T50688 CY4L8W 44549109 IC50 = 61 nM T50688 C4FW5Y 44549223 IC50 = 38 nM T50688 C7IXB3 44550126 IC50 = 21.3 nM T50688 CW9N7S 44550127 IC50 = 101 nM T50688 CK4UM8 44550445 IC50 = 154 nM T50688 C3QU6T 44550446 IC50 = 36 nM T50688 CS0Z3D 44550447 IC50 = 70 nM T50688 CH9M4W 44550573 IC50 = 106 nM T50688 C5V7GK 44550574 IC50 = 121 nM T50688 CB7R0U 44550575 IC50 = 27 nM T50688 CN3T7E 44550576 IC50 = 7.3 nM T50688 CO8EM6 44550577 IC50 = 140.6 nM T50688 C4XF2A 44550689 IC50 = 355 nM T50688 C4T6XP 44550690 IC50 = 38 nM T50688 CUWQ62 44550691 IC50 = 71 nM T50688 C69RIT 44550947 IC50 = 28 nM T50688 C4U9VF 44591153 IC50 > 10000 nM T50688 CER2H0 44591154 IC50 > 10000 nM T50688 C7TX9N 44591155 IC50 > 10000 nM T50688 C5VBY3 44820665 IC50 = 95 nM T50688 CKV5P7 45264021 IC50 = 32 nM T50688 C9RHC0 45483715 IC50 = 429 nM T50688 C4E8LZ 45483796 IC50 = 25 nM T50688 CU58DV 45483797 IC50 = 51 nM T50688 C18VUC 45483798 IC50 = 20 nM T50688 C89ZFA 46224777 IC50 = 34400 nM T50688 C5X1NZ 46224858 IC50 = 121000 nM T50688 CDG6B1 46224859 IC50 = 159000 nM T50688 CKM2X1 46224860 IC50 = 14800 nM T50688 CL39GY 46224861 IC50 = 76700 nM T50688 C56PVC 46226894 IC50 > 50000 nM T50688 CVXH79 46226896 IC50 = 2300 nM T50688 CBKZ57 46226897 IC50 = 8900 nM T50688 C30JXH 46226899 IC50 = 15000 nM T50688 C2WHK1 46226900 IC50 = 9700 nM T50688 C5H9YT 46226901 IC50 = 16500 nM T50688 CV8W7P 46226902 IC50 = 7700 nM T50688 C83EWD 46226903 IC50 = 5200 nM T50688 CRVU54 46226904 IC50 = 18000 nM T50688 CE85AX 46226905 IC50 = 11800 nM T50688 C0Y1TB 46232105 IC50 = 0.56 nM T50688 CP7U9T 50907449 IC50 > 10000 nM T50688 C6XNM0 53380822 IC50 > 100000 nM T50688 C1KFQ0 53380823 IC50 > 100000 nM T50688 C7JWD0 53380936 IC50 > 100000 nM T50688 C97KGD 53380937 IC50 > 100000 nM T50688 CKV6Q2 53380938 IC50 > 100000 nM T50688 C47WIH 53380939 IC50 > 100000 nM T50688 CY3RO0 53380940 IC50 > 10000 nM T50688 C3R8PW 53380941 IC50 > 100000 nM T50688 C2G6VQ 54580191 IC50 = 0.94 nM T50688 C1D8YQ 54581193 IC50 = 0.98 nM T50688 C0YTW6 54583189 IC50 = 0.4 nM T50688 CY08RT 54586079 IC50 = 0.023 nM T50688 CY7EQ4 56658817 IC50 = 6 nM T50688 C7I1EZ 56660024 IC50 = 350 nM T50688 C6OI5V 56660094 IC50 > 100000 nM T50688 CKFI81 56660095 IC50 > 100000 nM T50688 C0RFN9 56661197 IC50 = 230 nM T50688 CRT92P 56663492 IC50 = 37 nM T50688 CJR9F6 56666913 IC50 = 6.8 nM T50688 CHO1R7 56666917 IC50 = 6.5 nM T50688 CKR2H3 56666921 IC50 = 6.5 nM T50688 CETB80 56669198 IC50 = 1.7 nM T50688 CIH3K9 56670363 IC50 = 5.5 nM T50688 CF96ZL 56672656 IC50 = 18 nM T50688 CV68RB 56676028 IC50 = 11.6 nM T50688 CTXA08 56676029 IC50 = 1.3 nM T50688 CV3B1N 56676031 IC50 = 3260 nM T50688 CR3Q0L 56677204 IC50 = 270 nM T50688 C5EPH9 56677206 IC50 = 1200 nM T50688 CDP40K 56679353 IC50 = 1.8 nM T50688 CT7U8L 56683905 IC50 > 100000 nM T50688 C3CDB4 56683906 IC50 > 100000 nM T50688 CRCK01 56949775 IC50 = 22.7 nM T50688 C64ETP 56949776 EC50 = 40.8 nM T50688 CI2Z8J 56949777 IC50 = 62.5 nM T50688 C6A8YO 56949924 IC50 = 136 nM T50688 CPBN64 56949925 IC50 = 1154 nM T50688 C54RZY 56949926 IC50 = 1322 nM T50688 CM90UN 57390370 IC50 = 1.2 nM T50688 CB57DW 57391171 IC50 = 1500 nM T50688 CWJ4I7 57391565 IC50 = 3400 nM T50688 C7APO2 57392934 IC50 = 1100 nM T50688 CZ2A0S 57392935 IC50 > 100000 nM T50688 CX16KB 57393324 IC50 = 45000 nM T50688 CR72PQ 57393920 IC50 = 4.4 nM T50688 C6EWL9 57394677 IC50 = 49000 nM T50688 C8T2ZJ 57395044 IC50 > 100000 nM T50688 C9F4OL 57398232 IC50 = 2000 nM T50688 C5OAB7 57398233 IC50 > 100000 nM T50688 CY39KP 57398234 IC50 > 100000 nM T50688 CODX48 57399879 IC50 = 2200 nM T50688 C93VSX 57399880 IC50 = 33000 nM T50688 C5WOZ3 57399881 IC50 = 31000 nM T50688 C9ZL5X 57400230 IC50 = 31000 nM T50688 CPZR79 57400272 IC50 = 60000 nM T50688 CJGQ60 57400873 IC50 = 6.3 nM T50688 CS2ZY1 57401658 IC50 = 1800 nM T50688 CG90KP 57403382 IC50 = 34000 nM T50688 C3CKA6 57403383 IC50 = 80000 nM T50688 C4OB6Z 57403384 IC50 = 2500 nM T50688 CKI4S8 57403776 IC50 = 2500 nM T50688 CR71ZG 59665343 IC50 > 10000 nM T50688 C31IUF 69863577 IC50 > 10000 nM T50688 CM2AD4 70696326 IC50 > 10000 nM T50688 CAF23V 71452640 IC50 > 200000 nM T50688 C23GSR 71459889 IC50 = 28000 nM T50688 C8EM7Y 71550913 IC50 > 10000 nM T50688 CU95LC 71574160 IC50 > 10000 nM T50688 COJ8Y4 71574161 IC50 > 10000 nM T50688 C8V4UB 71574356 IC50 > 10000 nM T50688 C9J7NH 71652207 IC50 = 42600 nM T50688 CLH52G 71654374 IC50 > 200000 nM T50688 C8GDV7 71654376 IC50 > 200000 nM T50688 CY29LR 71654530 IC50 > 200000 nM T50688 C3K6PT 71654532 IC50 > 200000 nM T50688 C3X7FP 71654534 IC50 = 1210 nM T50688 CCGP56 71654535 IC50 = 665 nM T50688 CZG3Y9 71654536 IC50 = 17600 nM T50688 C5D2OL 71698598 IC50 > 300000 nM T50688 CGYN76 71698686 IC50 > 300000 nM T50688 CD0Z5K 71698687 IC50 > 300000 nM T50688 C0DUT2 71698688 IC50 > 300000 nM T50688 C60JTA 71698689 IC50 > 300000 nM T50688 C35ZJV 71698690 IC50 > 300000 nM T50688 C9XSB5 71698770 IC50 = 78400 nM T50688 CRN95M 71698771 IC50 > 300000 nM T50688 C0LW4G 71698774 IC50 > 300000 nM T50688 CH26JR 71698775 IC50 = 16800 nM T50688 C0WR9F 71699124 IC50 = 14000 nM T50688 CZKL39 71699125 IC50 = 96000 nM T50688 C27TZK 71699126 IC50 = 55000 nM T50688 CD12FS 71699127 IC50 = 35000 nM T50688 CFN7Q4 71699199 IC50 = 12000 nM T50688 C7RTF0 71699200 IC50 = 4700 nM T50688 C8JE0W 71699201 IC50 = 2200 nM T50688 CRAG19 71699203 IC50 > 300000 nM T50688 CYAH23 71699286 IC50 > 300000 nM T50688 CM8E7F 71699287 IC50 = 25800 nM T50688 C9Y3DN 71699288 IC50 = 12800 nM T50688 C8B7QE 72949858 IC50 > 5000 nM T50688 CZ2P8U 73345565 IC50 = 30 nM T50688 CQAE56 73345568 IC50 = 220 nM T50688 CU1VZ5 73345570 IC50 = 60 nM T50688 CPT7S8 73345576 IC50 = 248 nM T50688 C0BJ1F 73345752 IC50 = 850 nM T50688 C9UD8K 73346937 Ki = 42000 nM T50688 CKG2D8 73346996 IC50 = 7970 nM T50688 C1Z4HB 73346997 IC50 > 200000 nM T50688 COP75R 73347022 IC50 = 1790 nM T50688 C5E4ZO 73347079 Ki = 13.7 nM T50688 CZ6Y9R 73347081 IC50 = 10 nM T50688 CZ35TD 73347085 IC50 = 352 nM T50688 CGM9F7 73347087 IC50 = 70 nM T50688 C89ENA 73347090 IC50 = 1 nM T50688 CN1A2D 73347092 IC50 = 400 nM T50688 C7IC1G 73347403 IC50 > 300000 nM T50688 CHLG51 73348500 IC50 = 150 nM T50688 CD1RB5 73348588 Ki = 4.8 nM T50688 CO9L2V 73348591 IC50 = 20 nM T50688 C43LWV 73348592 IC50 = 20 nM T50688 CM37AE 73348593 IC50 = 10 nM T50688 CT1RG5 73348594 IC50 = 40 nM T50688 CF1UL2 73348680 IC50 = 6000 nM T50688 C7Y3ZB 73348933 IC50 > 300000 nM T50688 CO15PX 73350083 IC50 = 200000 nM T50688 CU0GS5 73350084 IC50 = 385000 nM T50688 CH4VE1 73350172 Ki = 24.3 nM T50688 CQL5F8 73350174 Ki = 35 nM T50688 CQ5D7B 73350175 IC50 = 20 nM T50688 CJEH13 73350177 IC50 = 10 nM T50688 C20AJB 73350179 IC50 = 4 nM T50688 C19PJE 73350181 IC50 = 17 nM T50688 CRHV46 73351571 Ki = 58 nM T50688 C2F3YZ 73351673 IC50 = 210 nM T50688 CJA25I 73351674 IC50 = 150 nM T50688 C6NCQ1 73351675 IC50 = 50 nM T50688 C46ULG 73351676 IC50 = 150 nM T50688 C8B6NV 73351677 IC50 = 31 nM T50688 CIYV49 73351678 IC50 = 6 nM T50688 CY76LM 73353036 IC50 = 40500 nM T50688 CA6GB7 73353037 IC50 = 55300 nM T50688 CKW5X4 73353038 IC50 > 200000 nM T50688 CM94NF 73353043 IC50 = 32200 nM T50688 CR5HL8 73353062 Ki = 3300 nM T50688 CUE1A8 73353139 Ki = 8.5 nM T50688 C20FGN 73353141 IC50 = 40 nM T50688 CP6AJ3 73353143 IC50 = 30 nM T50688 CUPR57 73353147 IC50 = 30 nM T50688 C83RAM 73353150 IC50 = 29 nM T50688 CX47JD 73353160 IC50 = 120 nM T50688 C3QZ4W 73354557 IC50 = 82000 nM T50688 CUP3W4 73354558 IC50 = 9600 nM T50688 C6OX7Q 73354659 Ki = 58 nM T50688 CV3OI9 73354660 Ki = 9.3 nM T50688 CRY2K3 73354661 Ki = 26 nM T50688 CAJ27W 73354663 IC50 = 70 nM T50688 CT4A5S 73354664 IC50 = 90 nM T50688 C6XTP9 73354667 IC50 = 16 nM T50688 CZ1BL4 73354668 IC50 = 20 nM T50688 CC19KU 73356070 Ki = 75000 nM T50688 C1LZI2 73356125 IC50 = 11400 nM T50688 C8GVU2 73356136 IC50 = 26 nM T50688 C4EJK0 73356213 IC50 = 20 nM T50688 CH8G5C 73356216 IC50 = 120 nM T50688 CPG36Q 73356217 IC50 = 15 nM T50688 CD1S3N 73356221 IC50 = 50 nM T50688 CI07FE 90645591 IC50 = 947000 nM T50688 C8N6OE 90654504 IC50 > 10000 nM T50688 CRY16L 91930237 IC50 = 13 nM T50688 C3I5NZ 118709463 IC50 = 1.5 nM T50688 CY1IS6 118718872 IC50 = 10 nM T50688 CHD10T 118753906 IC50 = 220 nM T50688 CE7PC8 118753907 IC50 = 7900 nM T50688 CJX84K 122192536 IC50 = 320 nM T50688 CC57KE 122192704 IC50 = 79 nM T50688 C6PBW7 122192706 IC50 = 0.22 nM T50688 CGI3N9 122192708 IC50 = 0.96 nM T50688 CMU5L2 134132719 IC50 = 7600 nM T50688 CFO64Z 134132799 IC50 = 18800 nM T50688 C7FPL9 134135111 IC50 = 200 nM T50688 C3D0AC 134135726 IC50 = 7900 nM T50688 C4MU0L 134136847 IC50 = 6380 nM T50688 C1WMQ0 134137198 IC50 = 5400 nM T50688 CR2BO9 134137328 IC50 > 100000 nM T50688 CP5S6D 134137433 IC50 = 1330 nM T50688 CCN09H 134137713 IC50 > 100000 nM T50688 CSW65H 134138739 IC50 = 80 nM T50688 C7K5IZ 134139108 IC50 = 4010 nM T50688 CAP65B 134140093 IC50 > 100000 nM T50688 CB6SA2 134143022 IC50 = 370 nM T50688 CXNR60 134143874 IC50 = 520 nM T50688 C0UL6E 134146896 IC50 = 3290 nM T50688 CCGZ12 134147635 IC50 = 280 nM T50688 C5EL6I 134148127 IC50 = 24600 nM T50688 CZY3O5 134151321 IC50 = 2100 nM T50688 C4LV7R 134152693 IC50 = 1080 nM T50688 CIC9T4 134153084 IC50 = 3400 nM T50688 C3H8BS 134153267 IC50 = 1650 nM T50688 CMN95S 134153892 IC50 = 12700 nM T50688 C46ICN 134157552 IC50 = 12800 nM T50688 CJL87N 135949396 IC50 = 323 nM T50688 CSCN42 135983770 IC50 = 167 nM T50688 CR8K5L 135983772 IC50 = 6300 nM T50688 C1WEK2 136048740 IC50 = 20 nM T50688 CW4IZ6 136056116 IC50 = 400 nM T50688 CBVF84 136094924 IC50 = 3.8 nM T50688 C61NCW 136094926 IC50 = 150 nM T50688 CT1QN2 136224837 IC50 = 15300 nM T50688 CN8BW0 136224847 IC50 = 16000 nM T50688 C7KE9J 136224848 IC50 = 870 nM T50688 C7R1TS 136224849 IC50 = 890 nM T50688 CG24CQ 136224854 IC50 = 260 nM T50688 C4IE0Q 137028367 IC50 = 2.2 nM T50688 CL4K9J 137175047 IC50 = 55 nM T50688 CDQ5J6 137175053 IC50 = 1.8 nM T50688 CVAK07 137175055 IC50 = 1.53 nM T50688 C9C4AK 137175068 IC50 = 1.57 nM T50688 CACK48 137659180 IC50 = 2.3 nM T50688 C17RZG 155515221 IC50 = 5804 nM T50688 CHT1J6 155515540 IC50 > 1000 nM T50688 CQ5C4M 155516533 IC50 > 1000 nM T50688 CZY8F6 155520344 IC50 = 5028 nM T50688 C2GJ5V 155527654 IC50 > 10000 nM T50688 CPIL79 155528977 IC50 > 10000 nM T50688 CJZU81 155532583 IC50 > 10000 nM T50688 CJ7O2X 155534687 IC50 > 1000 nM T50688 CWF98D 155552156 IC50 > 1000 nM T50688 C80PGY 155563043 IC50 > 10000 nM T50688 CEF3T8 155563936 IC50 > 1000 nM T50688 C2M7AJ 15677293 IC50 = 30000 nM T50688 C5FR9J 44385169 IC50 = 43000 nM T50688 CXT94Y 44403730 IC50 = 14 nM T50688 D01XUU 9958398 IC50 = 8 nM T50688 D04BHL 177230 IC50 = 60 nM T50688 D04XTP 44322318 IC50 = 0.027 nM T50688 D05AGK 11743533 IC50 = 17 nM T50688 D06LHH 9805998 IC50 = 13 nM T50688 D06LKH 123811 IC50 = 120 nM T50688 D06LUT 44379110 IC50 = 3440 nM T50688 D07WDB 104802 IC50 = 76 nM T50688 D08RLR 9862322 IC50 = 67 nM T50688 D0A0KS 9851104 IC50 = 12000 nM T50688 D0B4JU 15409414 IC50 = 195 nM T50688 D0C8LA 9913833 IC50 = 9 nM T50688 D0H3UO 9984308 IC50 = 26 nM T50688 D0LV6B 130667 IC50 = 1700 nM T50688 D0M7KS 52942958 Ki = 110 nM T50688 D0O5OM 10742947 IC50 = 25000 nM T50688 D0R3CY 9952958 IC50 = 1200 nM T50688 D0S8DT 10324223 IC50 = 15 nM T50688 D0W5ZK 177364 IC50 = 12 nM T73482 D00OVU 24965990 Ki = 0.3981 nM T73482 D02RXG 6918287 Ki = 250 nM T73482 D06CKX 25195495 Ki = 0.3 nM T73482 D08SCL 46190695 IC50 = 1986 nM T73482 D0A7ZK 56944144 Ki = 2.512 nM T73482 D0FK6O 67116280 Ki = 1277 nM T73482 D0NN5A 25128145 Ki = 0.631 nM T73482 D06BTF 23727689 IC50 = 13 nM T73482 C91DAE 185394 Ki = 1300 nM T73482 CKN27R 645882 Ki > 15848.93 nM T73482 CW90GD 647720 Ki > 15848.93 nM T73482 CMQ23R 833756 Ki = 36 nM T73482 C5NO3B 855282 Ki > 15848.93 nM T73482 C1Q7FH 1034375 Ki = 1200 nM T73482 CCN92H 1207917 Ki = 6700 nM T73482 CEX5I0 1301005 IC50 = 21 nM T73482 CK8ZP2 1725151 IC50 > 10000 nM T73482 C7L9OX 1784975 IC50 > 10000 nM T73482 CZ0AJ2 2273636 IC50 > 10000 nM T73482 CDC1E3 2796191 Ki = 216 nM T73482 CC79VB 2860019 Ki = 6300 nM T73482 C4JH3Z 2870209 Ki = 30700 nM T73482 CV53JP 3119056 IC50 > 10000 nM T73482 CF8RB9 3119749 Ki = 2700 nM T73482 CG01OM 3213606 Ki > 15848.93 nM T73482 C4X9CJ 3213619 Ki > 15848.93 nM T73482 C4XGO6 3213626 Ki > 15848.93 nM T73482 C8WE7J 3213637 Ki > 15848.93 nM T73482 CL6KP4 3213649 Ki = 2511.89 nM T73482 C89CAQ 3213663 Ki > 15848.93 nM T73482 C7XRC5 3213671 Ki = 630.96 nM T73482 CA9E7M 3213679 Ki > 15848.93 nM T73482 CL7PN8 3213689 Ki = 1258.93 nM T73482 CFPR85 3213696 Ki = 794.33 nM T73482 CLX9G8 3213712 Ki > 15848.93 nM T73482 C9L6CG 3213744 Ki = 2511.89 nM T73482 CU8F4X 3213776 Ki = 2511.89 nM T73482 CJ93NE 3213793 Ki > 15848.93 nM T73482 CHS5V2 3213803 Ki > 15848.93 nM T73482 C4O1NG 3213835 Ki = 1995.26 nM T73482 C0IW7Z 3213904 Ki > 15848.93 nM T73482 C3XD5Z 3213915 Ki > 15848.93 nM T73482 CM2S1K 3213928 Ki = 794.33 nM T73482 C32UAN 3213941 Ki > 15848.93 nM T73482 C5R4LA 3213958 Ki > 15848.93 nM T73482 CYM81H 3213966 Ki = 1995.26 nM T73482 C8XAM0 3213992 Ki = 1000 nM T73482 CS0VF3 3214024 Ki = 3162.28 nM T73482 C2J1TB 3634416 Ki = 12000 nM T73482 C3O5WZ 5165198 Ki > 15848.93 nM T73482 C04ZBY 5218889 Ki = 800 nM T73482 CT23BD 6418917 Ki = 1100 nM T73482 CX1BS0 6859582 Ki = 7600 nM T73482 CTYZ64 9798764 Ki = 28 nM T73482 C7SN9C 9936247 IC50 = 5300 nM T73482 CR3LK5 9978819 Ki = 1995.26 nM T73482 C2ELV0 9978820 Ki = 1000 nM T73482 CK0F1B 10024157 Ki < 10000 nM T73482 C25NXP 10024223 Ki = 1000 nM T73482 CR4VC2 10044549 Ki = 2511.89 nM T73482 C8TZF9 10046197 Ki = 63.1 nM T73482 CO41BA 10046198 Ki > 5011.87 nM T73482 CER65W 10048862 Ki = 6.31 nM T73482 CC0V9S 10069829 Ki = 251.19 nM T73482 C8SHP4 10112247 IC50 > 10000 nM T73482 C7UL5G 10113123 Ki = 8 nM T73482 C8MS0F 10139334 IC50 = 18 nM T73482 C41SAC 10144095 IC50 = 52 nM T73482 C5CZ0J 10201185 Ki = 5.012 nM T73482 CV0Y8N 10204153 Ki = 1.1 nM T73482 CVN2Q8 10208109 IC50 = 17 nM T73482 C46ROY 10250023 Ki = 100 nM T73482 CTHA73 10278102 IC50 = 119 nM T73482 C69ZAN 10316124 Ki = 125.89 nM T73482 CYB3G4 10316232 Ki = 2511.89 nM T73482 CQNX31 10316508 Ki = 79.43 nM T73482 CWU80C 10337554 Ki = 398.11 nM T73482 CJSX37 10386388 Ki = 501.19 nM T73482 CZS4R9 10387337 Ki = 39.81 nM T73482 C8OF7V 10407090 Ki = 63.1 nM T73482 CA3E0X 10409682 IC50 > 10000 nM T73482 C4E9ZR 10433189 Ki = 501.19 nM T73482 C3LJ1G 10453273 Ki = 19.95 nM T73482 C5FBU7 10473775 Ki < 10000 nM T73482 CZ1J7A 10475401 IC50 > 10000 nM T73482 CX7M8O 10864072 IC50 = 127 nM T73482 C7OM4V 10864264 IC50 = 552 nM T73482 CBM0E3 10864538 IC50 = 19 nM T73482 CUPD25 10874416 IC50 = 9475 nM T73482 CV83MQ 10884498 IC50 = 5731 nM T73482 C8ZEK0 10906648 IC50 = 8425 nM T73482 CKV5W9 10918096 IC50 = 1460 nM T73482 C2VF5E 10918199 IC50 = 37 nM T73482 CVI01B 10929426 IC50 = 1906 nM T73482 C0MWO4 10939830 IC50 = 44 nM T73482 CVG1W4 10939855 IC50 = 1113 nM T73482 CKNF23 10951393 IC50 = 49 nM T73482 C4ZTW3 10951496 IC50 = 8 nM T73482 C8E5LJ 10962350 IC50 = 129 nM T73482 CE68HD 10983971 IC50 = 200 nM T73482 CADV49 10983972 IC50 = 2008 nM T73482 CRNI02 10994188 IC50 = 4274 nM T73482 CR9S3I 10994415 IC50 = 4771 nM T73482 C9KAL2 11016474 IC50 > 10000 nM T73482 C5W8OD 11016554 IC50 = 118 nM T73482 CC0IG1 11038242 IC50 = 1182 nM T73482 C4DX9L 11049263 IC50 = 1138 nM T73482 C3NL0R 11071336 IC50 = 45 nM T73482 CZF1P3 11071351 IC50 = 10000 nM T73482 C47DCI 11081493 IC50 = 268 nM T73482 C8RK9Q 11081686 IC50 = 3138 nM T73482 CF9D3V 11102681 IC50 > 10000 nM T73482 C5G1WK 11123332 IC50 = 4464 nM T73482 CGA21K 11146397 IC50 = 21 nM T73482 C16TCJ 11180190 Ki = 4.15 nM T73482 CM26ZQ 11734173 IC50 = 75 nM T73482 C6KE0W 11744563 Ki = 79.43 nM T73482 CZ0TU8 11812976 IC50 = 690 nM T73482 CM6A3U 11960895 Ki = 3 nM T73482 CHV29L 11960929 Ki = 8 nM T73482 CQD14I 12047522 IC50 > 10000 nM T73482 C5SR3I 12997499 IC50 > 10000 nM T73482 CXGJ06 15949515 Ki = 27 nM T73482 CDXM06 15949516 Ki = 86 nM T73482 CBF2K7 15949607 Ki = 40 nM T73482 C1EIU3 15949609 Ki = 130 nM T73482 CA3C9D 15949610 Ki = 28 nM T73482 C9V6OR 15949701 Ki = 500 nM T73482 C75IUA 15949702 Ki = 2300 nM T73482 CM61GE 15949703 Ki = 69 nM T73482 CJ4X8D 15993497 IC50 > 10000 nM T73482 C52SLH 16002587 Ki > 6309.57 nM T73482 C81AUJ 16046844 Ki = 79.43 nM T73482 C0BLR7 16048438 Ki = 954.99 nM T73482 C9RM2Y 16752731 IC50 = 6 nM T73482 CKH6B4 18592212 Ki = 7.943 nM T73482 CK7L1A 18592214 Ki > 2511.89 nM T73482 CT6ON8 18592216 Ki = 1995.26 nM T73482 CJBK87 20911062 IC50 = 3455 nM T73482 CQE54R 22599910 IC50 > 10000 nM T73482 CW7F3D 22599915 IC50 > 10000 nM T73482 CKL08P 22599923 IC50 > 10000 nM T73482 CIO42U 24737677 IC50 = 10 nM T73482 CBC56J 24748750 IC50 = 26 nM T73482 CH6TN9 24759955 IC50 = 17 nM T73482 CY3X7G 24760024 IC50 = 12 nM T73482 C4R8OV 24760087 IC50 = 29 nM T73482 C9B2DL 24760747 IC50 = 119 nM T73482 C43PRK 24760748 IC50 = 166 nM T73482 CB3TQ1 24808511 IC50 = 27 nM T73482 C1H3AN 24808514 Ki = 1.8 nM T73482 CK5LN1 24853522 IC50 = 7 nM T73482 COB2P9 24882716 Ki = 1.2 nM T73482 CB9SA1 24896566 Ki = 462 nM T73482 CZ9EQ2 24959177 IC50 = 40 nM T73482 C9MI0U 24959178 IC50 = 16 nM T73482 CJR42H 24959549 IC50 = 18 nM T73482 CY58BS 24959912 IC50 = 45 nM T73482 C50TAB 24960290 IC50 = 1066 nM T73482 C5UF2L 24960654 IC50 = 313 nM T73482 CTE96G 24961018 IC50 = 717 nM T73482 CUI6E1 24961746 IC50 = 20 nM T73482 C35DNF 24961747 IC50 = 32 nM T73482 C67KNQ 24962111 IC50 = 203 nM T73482 C57LWU 24962112 IC50 = 3902 nM T73482 CG43WT 24962115 IC50 = 459 nM T73482 CK9H5Y 24962833 IC50 = 431 nM T73482 CL6N8O 24962835 IC50 = 312 nM T73482 C95RZN 24964358 Ki = 1700 nM T73482 C9IUP7 24964576 Ki = 0.8 nM T73482 C38UID 24964578 Ki = 0.5 nM T73482 CYEP21 24964937 Ki = 0.3 nM T73482 C5I9DX 24965290 Ki = 0.2 nM T73482 C5SFH2 24965291 Ki = 0.3 nM T73482 CGP45R 24965643 Ki = 0.78 nM T73482 CSI6H9 24965645 Ki = 1.8 nM T73482 CFS95W 24968277 Ki = 0.7 nM T73482 CPQD14 24992490 IC50 = 3098 nM T73482 CTI38U 25060119 Ki = 94.5 nM T73482 CTX03U 25060120 Ki = 7250 nM T73482 C8XKP2 25060382 Ki = 3350 nM T73482 CXE52R 25060383 Ki = 1105 nM T73482 CD6CA4 25060384 Ki = 2975 nM T73482 C6L1VC 25060653 Ki = 236 nM T73482 C8DO2L 25060654 Ki = 273 nM T73482 CN7V6R 25060655 Ki = 833 nM T73482 C0K6WX 25060657 Ki = 1087 nM T73482 C5U9ZY 25060899 Ki = 1073 nM T73482 CDBQ73 25060900 Ki = 5150 nM T73482 C56RMG 25060902 Ki = 747 nM T73482 CMOS06 25063585 IC50 = 108 nM T73482 CF5AB2 25063587 IC50 = 358 nM T73482 CJY0H7 25063628 IC50 = 993 nM T73482 C7ZP8R 25063664 IC50 = 180 nM T73482 C9KY3W 25063665 IC50 = 1031 nM T73482 C39RAF 25063701 IC50 = 669 nM T73482 C15XCU 25127493 Ki = 1 nM T73482 CY5X1A 25204740 IC50 = 13 nM T73482 C03XSU 25225718 Ki = 720 nM T73482 CF5MV8 25809483 IC50 > 10000 nM T73482 C07DOP 26719840 IC50 = 31 nM T73482 CW2U6O 30560665 IC50 = 9191 nM T73482 CYL39Q 40924317 Ki = 6.31 nM T73482 C7IKX4 42604859 Ki = 900 nM T73482 CT13OI 44219762 Ki = 2 nM T73482 CI4BE6 44270595 EC50 > 1000000 nM T73482 CW30VO 44270596 EC50 > 1000000 nM T73482 C26BKD 44270597 EC50 > 1000000 nM T73482 C39TRO 44270625 EC50 > 1000000 nM T73482 C5PO4S 44270635 EC50 > 1000000 nM T73482 C87IBU 44270666 EC50 > 1000000 nM T73482 CMB6A1 44270673 EC50 > 1000000 nM T73482 C1OM8C 44270674 EC50 > 1000000 nM T73482 CZW96I 44270676 EC50 > 1000000 nM T73482 CQ56DO 44270709 EC50 > 1000000 nM T73482 C6GJW8 44359225 IC50 = 3600 nM T73482 CUPE16 44359281 IC50 = 3670 nM T73482 C68CJQ 44359282 IC50 = 1130 nM T73482 C9H4QW 44359283 IC50 > 10000 nM T73482 C5FKZ8 44359335 IC50 > 10000 nM T73482 CQP59C 44359365 IC50 = 5900 nM T73482 CIO8P6 44359366 IC50 > 10000 nM T73482 CE4FG6 44359367 IC50 = 3850 nM T73482 C7SO5Y 44359405 IC50 > 10000 nM T73482 CCG51L 44359415 IC50 = 5500 nM T73482 CX4C8G 44359451 IC50 > 10000 nM T73482 CSY89K 44359452 IC50 > 10000 nM T73482 CA31JT 44359467 IC50 > 10000 nM T73482 C9YK1T 44359482 IC50 > 10000 nM T73482 CFJI51 44359494 IC50 > 10000 nM T73482 COVU19 44359603 IC50 > 10000 nM T73482 CUQ13D 44359613 IC50 = 2300 nM T73482 CN73FK 44359637 IC50 = 7000 nM T73482 CR9E8A 44359650 IC50 > 10000 nM T73482 CN3HL7 44376980 Ki = 66069.34 nM T73482 C9QD1O 44376981 EC50 = 1380 nM T73482 CD62VI 44393273 Ki < 10000 nM T73482 C47MUJ 44393285 Ki < 5011.87 nM T73482 CT3U9Z 44393313 Ki = 125.89 nM T73482 C5QNK7 44393337 Ki < 10000 nM T73482 CIWP10 44393338 Ki < 10000 nM T73482 C81EBC 44393370 Ki = 501.19 nM T73482 C4X2QA 44393375 Ki < 10000 nM T73482 CH0UI9 44405008 EC50 = 5.7 nM T73482 CM1IS8 44454577 Ki = 10 nM T73482 CA39CP 44454599 Ki = 1400 nM T73482 C1BD8E 44454602 Ki = 2500 nM T73482 CR35JH 44454877 Ki = 15 nM T73482 C9OD7E 44454878 Ki = 2 nM T73482 CLRZ97 44454915 Ki = 0.7 nM T73482 CZG78N 44454916 Ki = 120 nM T73482 CYIO02 44454917 Ki = 3 nM T73482 CSLE81 44454943 Ki = 39 nM T73482 CWPB72 44454946 Ki = 9 nM T73482 C2RO9B 44454947 Ki = 49 nM T73482 C3I1LF 44463491 Ki = 1.995 nM T73482 CJY9N1 44555825 IC50 = 170 nM T73482 C92PMB 44555872 IC50 = 74 nM T73482 C2JT5F 44555974 IC50 = 85 nM T73482 C9UH1P 44555976 IC50 = 1677 nM T73482 C7P2VN 44555978 IC50 = 30 nM T73482 CJU9R7 44556023 IC50 = 94 nM T73482 C38KGZ 44556024 IC50 = 91 nM T73482 C3A8UM 44563904 IC50 = 19 nM T73482 C3IA9R 44563928 IC50 = 5 nM T73482 CCRY94 44563929 IC50 = 49 nM T73482 C5ASO0 44564034 IC50 = 3600 nM T73482 CR0T4G 44564035 IC50 = 731 nM T73482 CQ6Y4K 44564036 IC50 = 1565 nM T73482 CFA0L2 44564038 IC50 = 5300 nM T73482 C7R9DP 44574230 Ki = 9800 nM T73482 CZQ2N6 44574255 Ki = 930 nM T73482 C7IYO9 44574256 Ki = 63 nM T73482 C67JEM 44574257 Ki = 51 nM T73482 CUZK61 44580808 IC50 > 10000 nM T73482 C2R8YC 44580809 IC50 > 10000 nM T73482 C0LDE2 44580810 IC50 > 10000 nM T73482 CHIG04 44580825 IC50 = 2486 nM T73482 C6HQ2K 44580862 IC50 > 10000 nM T73482 CLP6W7 44580863 IC50 > 10000 nM T73482 C0BJI8 44580864 IC50 > 10000 nM T73482 CLKU70 44580865 IC50 = 886 nM T73482 C5INH4 44580886 IC50 = 4875 nM T73482 C2HT8N 44580887 IC50 = 1107 nM T73482 CUM2B9 44580888 IC50 = 888 nM T73482 C3FSE5 44580889 IC50 > 10000 nM T73482 CJ3HV2 44580912 IC50 = 1373 nM T73482 CEB05Y 44580913 IC50 = 2527 nM T73482 CC8D7N 44580914 IC50 = 1709 nM T73482 CY0A2T 44580945 IC50 = 17 nM T73482 CR8EL1 44580946 IC50 = 5 nM T73482 C2O6MI 44580947 IC50 = 12 nM T73482 CA36HG 44580948 IC50 = 6 nM T73482 CE4UV6 44580968 IC50 = 8 nM T73482 CVMS64 44580969 IC50 = 8 nM T73482 CNUF76 44581140 IC50 > 10000 nM T73482 CHZO78 44581141 IC50 > 10000 nM T73482 COUS06 44581168 IC50 > 10000 nM T73482 CNK67Y 44581169 IC50 > 10000 nM T73482 CZ03FY 44581170 IC50 > 10000 nM T73482 C41ZJE 44581171 IC50 > 10000 nM T73482 C97LXJ 44581172 IC50 > 10000 nM T73482 C6L7IF 44588748 Ki = 751 nM T73482 CDP50A 44588857 Ki = 1245 nM T73482 C1SYK4 44633765 Ki = 1584 nM T73482 CRM6C5 45259003 Ki = 10.5 nM T73482 C1QS3Y 45259004 Ki = 0.5 nM T73482 CH97EI 45375925 IC50 = 1950 nM T73482 CMRT28 45555989 IC50 = 6300 nM T73482 CB4O9P 46190694 Ki = 2700 nM T73482 C3KB9Q 46191662 IC50 = 3000 nM T73482 CRM02K 46191726 IC50 = 10000 nM T73482 CBGP17 46191727 IC50 = 10000 nM T73482 CJK6P2 46195690 Ki = 1000 nM T73482 CSJ27E 46204871 Ki = 2.2 nM T73482 CI34NU 46205522 Ki = 720 nM T73482 C2U1KF 46211807 Ki = 760 nM T73482 C0LQ6S 46211878 Ki = 900 nM T73482 C51BQE 46211883 Ki = 415 nM T73482 C48TNW 46211956 Ki = 2700 nM T73482 C21ICG 46212134 Ki = 965 nM T73482 C8R3SM 46212185 Ki = 910 nM T73482 CFV4Q2 46212296 Ki = 0.41 nM T73482 CHD1J4 46212539 Ki = 1030 nM T73482 CO7N9S 46212746 Ki = 4756 nM T73482 CT6F9H 46868664 Ki = 0.39 nM T73482 CNJR98 46868665 Ki = 6.2 nM T73482 CRK9B5 46868791 Ki = 4.1 nM T73482 C1KRZ6 46868793 Ki = 54 nM T73482 C7DH6F 46880346 IC50 = 10000 nM T73482 CP4C1B 46880347 IC50 = 63 nM T73482 C9Y3QE 46880348 IC50 = 1424 nM T73482 CMPE07 46880349 IC50 = 161 nM T73482 CJBC31 46880388 IC50 = 1919 nM T73482 CZ3C8T 46880389 IC50 = 402 nM T73482 C8ECV5 46880449 IC50 = 128 nM T73482 C29IMV 46880450 IC50 = 10000 nM T73482 C6JK5G 46880451 IC50 = 769 nM T73482 CFX08U 46883808 Ki = 1 nM T73482 C9C0FR 46883864 Ki = 12 nM T73482 CFL51W 46883865 Ki = 870 nM T73482 CR56NI 46883908 Ki = 0.4 nM T73482 CH5M1P 49793266 Ki = 8500 nM T73482 C51JSQ 49797987 Ki = 0.6 nM T73482 CS19WL 49797988 Ki = 0.9 nM T73482 CS9WK7 49798002 Ki = 10 nM T73482 C39KIH 49798003 Ki = 2 nM T73482 CR0C5N 49798004 Ki = 160 nM T73482 CNV6E4 49798005 Ki = 345 nM T73482 C3F0HR 49798028 Ki = 0.6 nM T73482 C72ADP 49798029 Ki = 7.6 nM T73482 C1X8TR 49798030 Ki = 0.4 nM T73482 C2BS3P 49805788 IC50 = 155 nM T73482 C0DKB7 50799599 Ki = 88 nM T73482 CS1O7E 52918933 Ki = 441 nM T73482 C51EGW 52942033 Ki > 15848.93 nM T73482 C65JKN 52944312 Ki > 15848.93 nM T73482 CFC12V 52944709 Ki > 15848.93 nM T73482 C9X3BC 52946457 Ki > 15848.93 nM T73482 CY9JU2 52948927 Ki > 15848.93 nM T73482 CJ4S2D 53242191 Ki = 288.4 nM T73482 CCZL67 53242213 Ki = 4 nM T73482 C8TC5B 53259112 Ki = 549.54 nM T73482 C68ERM 53259279 Ki = 1548.82 nM T73482 CK5CM6 53259467 Ki = 1424 nM T73482 C6U4FE 53259634 Ki = 58.88 nM T73482 CXKZ15 53259635 Ki = 18.62 nM T73482 C1HT7I 53259636 Ki = 275.42 nM T73482 C5E6TF 54576281 Ki = 4363 nM T73482 CI64JB 54579367 IC50 = 3784 nM T73482 CUG05N 54579583 IC50 = 2379 nM T73482 CAG6V1 54579585 IC50 > 10000 nM T73482 CLT6O5 54588789 IC50 = 998 nM T73482 C0OIE7 54751924 IC50 = 3000 nM T73482 C96GZT 54765113 IC50 = 6 nM T73482 CA0YR4 56659966 Ki = 10 nM T73482 CC6M4B 56663428 Ki = 501.19 nM T73482 CK76VA 56663429 Ki = 50.12 nM T73482 CU84LF 56670285 Ki = 125.89 nM T73482 C37HIB 56673796 Ki = 2511.89 nM T73482 C3CO2F 56673797 Ki = 6.31 nM T73482 CPT8J3 56673798 Ki = 1 nM T73482 CPE3R9 56680444 Ki = 398.11 nM T73482 C5TY1F 56680445 Ki = 7.943 nM T73482 CG6D7M 56680446 Ki = 39.81 nM T73482 CC0QF6 56683774 Ki = 0.1585 nM T73482 C35PTG 56683775 Ki = 0.1259 nM T73482 CW80YF 56943752 Ki = 30 nM T73482 CP5UD4 56944043 Ki = 2 nM T73482 C6F3VI 56944044 Ki = 137 nM T73482 CU87RH 56944045 Ki = 39 nM T73482 C67OXC 56944143 Ki = 3 nM T73482 C0BKG3 56944244 Ki = 32 nM T73482 C6GDX1 56944245 Ki = 39 nM T73482 CNY8F7 56944337 Ki = 121 nM T73482 C09WRF 56944429 Ki = 7 nM T73482 CAP79V 56944521 Ki = 43 nM T73482 C3SY9G 56944522 Ki = 9 nM T73482 CJ5T0W 56944620 Ki = 1 nM T73482 CX41CZ 56968452 Ki = 489.78 nM T73482 C6RH9Z 56970209 Ki = 812.83 nM T73482 CZQ5T1 56970417 Ki = 1621 nM T73482 C7I0LP 56970421 Ki = 21 nM T73482 C15GZB 56970625 Ki = 1445.44 nM T73482 CB4F3T 56970626 Ki = 371.54 nM T73482 CF7M3A 56970628 Ki = 660.69 nM T73482 CRV8S0 56970857 Ki = 1412.54 nM T73482 CDIO92 56970858 Ki = 512.86 nM T73482 CK9SF5 57388373 Ki > 2000 nM T73482 C56ORS 57388650 Ki = 106 nM T73482 CYQ43V 57388812 IC50 = 56.1 nM T73482 C1DF3J 57389725 IC50 = 3.22 nM T73482 CF08CS 57389801 IC50 = 5.54 nM T73482 CKDI91 57389883 IC50 = 119 nM T73482 C4FC6Z 57390049 IC50 = 9.06 nM T73482 C2LTP8 57390051 IC50 = 908 nM T73482 CB4CA1 57391006 IC50 = 1600 nM T73482 CAPD05 57392800 IC50 = 2300 nM T73482 C5WV2G 57396272 IC50 = 1600 nM T73482 C8DY2G 57398059 IC50 = 2600 nM T73482 C0K1PV 57403243 IC50 > 10000 nM T73482 C40IOT 57403244 IC50 = 1500 nM T73482 C9NHI3 58394291 IC50 = 10000 nM T73482 CXA3T8 58488153 Ki = 1 nM T73482 CI7U5V 60168601 IC50 = 5.4 nM T73482 CE9IM4 66733985 IC50 = 547 nM T73482 C8XNW4 67153780 IC50 = 53 nM T73482 CXQ94P 67153782 IC50 = 1426 nM T73482 C5FN3I 67209228 Ki = 778 nM T73482 C4PGT2 67209346 Ki = 29 nM T73482 CX2F3S 67209359 Ki = 274 nM T73482 CC2IT1 67209405 Ki = 20 nM T73482 CSQ3W1 67209426 Ki = 2667 nM T73482 CB7W0G 67209575 Ki = 970 nM T73482 C69PEQ 67209610 Ki = 800 nM T73482 C0C4JF 67209817 Ki = 63 nM T73482 CU5C8L 67251476 Ki = 1479.11 nM T73482 CC6X2O 67252378 Ki = 9.12 nM T73482 C4KC6Q 67281908 Ki = 3 nM T73482 CZ4L7E 67282493 Ki = 12 nM T73482 C3Q6ZA 67282848 Ki = 14 nM T73482 C4R1IH 67283149 Ki = 6 nM T73482 C0S7IR 67289227 Ki = 776.25 nM T73482 C15EQH 67380581 Ki = 3600 nM T73482 CH6EW0 67473922 Ki = 224 nM T73482 C1I7OW 67473934 Ki = 1016 nM T73482 CK18IT 67473935 Ki = 391 nM T73482 C2VD6Q 67473936 Ki = 1581 nM T73482 C42FLR 67473937 Ki = 138 nM T73482 CK1Q3V 67473938 Ki = 124 nM T73482 C2D4VM 67980311 Ki = 106 nM T73482 C0U9GM 67980666 Ki = 1068 nM T73482 CEVG41 68058790 Ki = 938 nM T73482 CDQ31I 68058793 Ki = 73 nM T73482 CTL92R 68083077 Ki = 81 nM T73482 CW8FR2 69080080 IC50 = 1950 nM T73482 CUIC59 69080156 IC50 = 25 nM T73482 CCB80U 69080186 IC50 = 107 nM T73482 CV4NO2 69080188 IC50 = 121 nM T73482 CN5H2Z 69080268 IC50 = 22 nM T73482 C58BVC 69080890 IC50 = 264 nM T73482 CE4I3Q 69080992 IC50 = 216 nM T73482 CJ7VG2 69081444 IC50 = 141 nM T73482 C49PMK 69081570 IC50 = 9 nM T73482 CNJ7K2 69081619 IC50 = 191 nM T73482 C4IW9J 69081640 IC50 = 65 nM T73482 CU4Z7I 69081642 IC50 = 40 nM T73482 CY0K1B 69081717 IC50 = 284 nM T73482 CD8RY3 69081742 IC50 = 19 nM T73482 CI3M2O 69081821 IC50 = 142 nM T73482 CSX60D 69081873 IC50 = 65 nM T73482 C30PMS 69081899 IC50 = 1407 nM T73482 CJI32G 69081964 IC50 = 16 nM T73482 CIN3O2 69082001 IC50 = 619 nM T73482 C3RDA0 69082236 IC50 = 75 nM T73482 C0QY5T 69082267 IC50 = 3486 nM T73482 CUW42P 69082306 IC50 = 77 nM T73482 C72OGM 69082473 IC50 = 4385 nM T73482 CJ93CT 69082475 IC50 = 32 nM T73482 C8L6DC 69082510 IC50 = 45 nM T73482 C6QB2K 69082516 IC50 = 3 nM T73482 CHS32F 69082545 IC50 = 3380 nM T73482 C95XAQ 69082595 IC50 = 899 nM T73482 CNK12W 69082599 IC50 = 2680 nM T73482 CW6MR8 69082645 IC50 = 44 nM T73482 C61XNT 69082665 IC50 = 4883 nM T73482 CD5HB2 69082678 IC50 = 177 nM T73482 CV94BF 69082681 IC50 = 154 nM T73482 CLX8D3 69082742 IC50 = 225 nM T73482 CJ45VT 69082766 IC50 = 412 nM T73482 CB70SA 69082817 IC50 = 136 nM T73482 COE39Z 69082854 IC50 = 927 nM T73482 C96STB 69082926 IC50 = 54 nM T73482 C6PR7O 69083435 IC50 = 193 nM T73482 CQ1IK8 69083745 IC50 = 1249 nM T73482 CPLG25 69083777 IC50 = 2 nM T73482 CJ6A5F 69084016 IC50 = 299 nM T73482 CKH1J6 69084057 IC50 = 1270 nM T73482 C3WL1H 69084118 IC50 = 4 nM T73482 C4E9VH 69084152 IC50 = 675 nM T73482 CT2NK9 69084345 IC50 = 44 nM T73482 CQPA54 69084621 IC50 = 1800 nM T73482 C2P3LC 69085010 IC50 = 724 nM T73482 C4NU5T 69085032 IC50 = 330 nM T73482 C4SXT9 69085047 IC50 = 14 nM T73482 C8T0RS 69085151 IC50 = 5 nM T73482 C4RU6S 69085189 IC50 = 14 nM T73482 CA4U1J 69085230 IC50 = 169 nM T73482 C9WX0M 69085295 IC50 = 1086 nM T73482 C4LM9J 69085642 IC50 = 531 nM T73482 CV76IC 69085689 IC50 = 550 nM T73482 C19PIM 69085726 IC50 = 34 nM T73482 C0Z1PN 69915149 Ki = 200 nM T73482 CP0N1Y 69915187 Ki = 52 nM T73482 C4I6UA 69915196 Ki = 4 nM T73482 C81MDP 69932186 Ki = 33 nM T73482 CA47RE 70169296 IC50 = 4364 nM T73482 CHS9N3 70681618 IC50 < 1 nM T73482 CB2QP1 70681619 IC50 = 8 nM T73482 C4NVY5 70681620 IC50 = 14 nM T73482 CUS92R 70683739 IC50 = 5 nM T73482 CM41XZ 70683740 IC50 = 6 nM T73482 CAU6W8 70683741 IC50 = 0.8 nM T73482 CDL7J3 70683742 IC50 = 145 nM T73482 C86KLO 70683743 IC50 > 2000 nM T73482 C4BOP2 70683744 IC50 = 390 nM T73482 C8PTI4 70685886 IC50 = 15 nM T73482 CWJ49Q 70685887 IC50 = 7 nM T73482 C5X8YM 70685888 IC50 = 6 nM T73482 C9O3RU 70685889 IC50 = 40 nM T73482 CFB9I0 70685890 IC50 = 1 nM T73482 CR7O0Q 70685891 IC50 = 121 nM T73482 C8YIC1 70685892 IC50 = 7 nM T73482 C6B1TJ 70687123 IC50 = 280 nM T73482 C80BKR 70687129 IC50 = 2500 nM T73482 C8G0AY 70688011 IC50 = 9 nM T73482 CTM9C1 70688012 IC50 = 2 nM T73482 C1IZ0S 70690040 IC50 = 4 nM T73482 CGA5E6 70690041 IC50 = 2 nM T73482 CCQR15 70690042 IC50 = 0.8 nM T73482 C3BRE9 70692193 IC50 = 3 nM T73482 CVT4S0 70692194 IC50 = 146 nM T73482 C0VL4I 70692195 IC50 = 27 nM T73482 C36FDI 70694255 IC50 = 2 nM T73482 CG4N1Z 70694256 IC50 = 12 nM T73482 CA58UO 70694257 IC50 = 6 nM T73482 C7UW0O 70696349 IC50 = 13 nM T73482 C0J2OK 70696350 IC50 = 10 nM T73482 CIPR26 70696351 IC50 = 2 nM T73482 CB3VS5 70816735 Ki > 4000 nM T73482 CWHM94 70816905 Ki = 175 nM T73482 C4RMS1 70817021 Ki = 2287 nM T73482 C94LXI 70817051 Ki = 783 nM T73482 CSCO94 70817059 Ki = 357 nM T73482 C7DO1N 70817239 Ki = 3 nM T73482 C6L7FH 70817382 Ki = 8 nM T73482 CTQ7C0 70818984 Ki = 660 nM T73482 CY03PE 70856594 Ki = 109 nM T73482 C7Q8ST 71522361 Ki = 1.1 nM T73482 C34TKD 71526207 Ki = 569 nM T73482 C2RO5Y 71526208 IC50 = 8400 nM T73482 CZ7JD6 71527494 Ki = 0.3 nM T73482 CE9SK3 71543409 Ki = 829 nM T73482 CR01NT 71555054 Ki = 4100 nM T73482 CTS09B 71579478 IC50 = 344 nM T73482 C12KAY 71579479 IC50 = 90 nM T73482 CJN41M 71580771 IC50 = 10000 nM T73482 C3QZ7D 71580772 IC50 = 10000 nM T73482 CV8N1K 71580773 IC50 = 10000 nM T73482 C4C9IF 71580858 IC50 = 10000 nM T73482 CX6G8Z 71580859 IC50 = 10000 nM T73482 CW7K4I 71580860 IC50 = 4171 nM T73482 CDC7T6 71580861 IC50 = 150 nM T73482 CQ2KC8 71580862 IC50 = 283 nM T73482 CL26RK 71580946 IC50 = 134 nM T73482 C9FIW3 71580947 IC50 = 3980 nM T73482 CAS05K 71580948 IC50 = 537 nM T73482 C0ND2T 71580949 IC50 = 10000 nM T73482 C5WL4U 71580950 IC50 = 492 nM T73482 C1NL7J 71624633 Ki = 900 nM T73482 CWAY56 71716523 IC50 = 1645 nM T73482 C1NP2M 72543760 IC50 = 1.25 nM T73482 CHU29Z 72699430 IC50 = 10.6 nM T73482 C1HMV0 72699854 IC50 = 1.07 nM T73482 CBF7O2 72699855 IC50 = 1.82 nM T73482 CKL84I 72699856 IC50 = 1.84 nM T73482 C1RY5X 72699949 IC50 = 1.26 nM T73482 C3I2OZ 72699950 IC50 = 0.82 nM T73482 CC70PO 72699951 IC50 = 3.06 nM T73482 C6HEI3 72700096 IC50 = 3.58 nM T73482 CH04OF 72700180 IC50 = 1.81 nM T73482 C5BKV3 72700181 IC50 = 2.01 nM T73482 CYJ2T4 72700265 IC50 = 1.58 nM T73482 CO7BI8 72700266 IC50 = 1.4 nM T73482 CL1U4W 72700267 IC50 = 2.45 nM T73482 CJN5K0 72700268 IC50 = 6.15 nM T73482 CZ8K4T 72700362 IC50 = 9.45 nM T73482 C7BY8D 72700363 IC50 = 1.93 nM T73482 CHCM80 72700366 IC50 = 14.7 nM T73482 CZDM79 72700457 IC50 = 4.39 nM T73482 CTLC87 72700458 IC50 = 1.9 nM T73482 CSWL87 72700459 IC50 = 86.6 nM T73482 CPV92B 72700460 IC50 = 1.1 nM T73482 C5JT0D 72700462 IC50 = 1.26 nM T73482 CWZ0T6 72700543 IC50 = 0.767 nM T73482 CP8G5V 72700544 IC50 = 4.39 nM T73482 COSK78 72700626 IC50 = 1.62 nM T73482 C68GDU 72700698 IC50 = 3.24 nM T73482 CMP5F9 72703893 IC50 < 10000 nM T73482 C7ZAH6 72703894 IC50 < 10000 nM T73482 CW3NX0 72704097 Ki = 20.42 nM T73482 CEY4I0 72704098 Ki = 1318.26 nM T73482 COTU10 72704099 Ki = 707.95 nM T73482 CGV76N 72704100 Ki = 758.58 nM T73482 CBE48L 72707143 Ki = 19.95 nM T73482 CO0U6I 72720554 Ki = 15.85 nM T73482 CVO7T2 72720555 Ki = 1 nM T73482 CD8Z5T 72720556 Ki = 39.81 nM T73482 CXG47B 72720982 Ki = 1.259 nM T73482 CBW93F 72721081 Ki = 63.1 nM T73482 CHN0B5 72721178 Ki = 316.23 nM T73482 C4OD7F 72721280 Ki = 25.12 nM T73482 C41JEL 72721380 Ki = 6.31 nM T73482 C50CDB 72721381 Ki = 63.1 nM T73482 CG8PX4 72721795 Ki = 50.12 nM T73482 CLD36Y 72721986 Ki = 25.12 nM T73482 C3JBG7 72721987 Ki = 1.995 nM T73482 C82DJS 72722084 Ki = 0.3981 nM T73482 CYC8U4 72722088 Ki = 12.59 nM T73482 C46UAR 72722089 Ki = 2.512 nM T73482 C6Q3OM 72725148 Ki = 1900 nM T73482 C3R1AC 72725149 Ki = 65000 nM T73482 C8DAZ2 73346054 IC50 = 5 nM T73482 C2C7BU 73347449 IC50 = 16 nM T73482 CO7CY6 73347581 IC50 = 10 nM T73482 CB8F6U 73348981 IC50 = 72 nM T73482 C8KLQ1 73350080 EC50 = 1340 nM T73482 CGZ7E4 73352057 IC50 = 378 nM T73482 CA9H1U 73353033 EC50 > 1000000 nM T73482 CJ4N5L 73353523 IC50 = 30 nM T73482 CB63NL 73356120 EC50 > 1000000 nM T73482 CIC73L 73356574 IC50 = 17 nM T73482 CH7S6O 73356708 Ki = 1400 nM T73482 C15PYW 73673014 Ki = 56 nM T73482 C34LXD 74221626 Ki = 757 nM T73482 C6M7RX 74221720 Ki = 572 nM T73482 CN53AG 74221903 Ki = 2517 nM T73482 CAIZ14 74221990 Ki = 1662 nM T73482 C7SZG6 74222158 Ki = 114 nM T73482 C6J9LF 74222159 Ki = 3568 nM T73482 C5J9EI 74222241 Ki = 1170 nM T73482 CZA0I9 74222326 Ki = 519 nM T73482 C07NHS 74222327 Ki = 1155 nM T73482 CGI5K2 74222402 Ki = 594 nM T73482 CZO3V4 74222406 Ki = 1611 nM T73482 CL15XT 74222492 Ki = 790 nM T73482 CA1N8P 74222754 Ki = 5765 nM T73482 CP9U0C 74222941 Ki = 1128 nM T73482 CX5L0W 76072813 Ki = 287 nM T73482 CF5Z2M 76310080 Ki = 3550 nM T73482 C28XZD 76310131 EC50 = 1130 nM T73482 CE5A0O 76310198 EC50 = 1040 nM T73482 CFS27O 76310208 EC50 = 526 nM T73482 CJO7X0 76310209 EC50 = 535 nM T73482 CE92OC 76310210 EC50 = 1560 nM T73482 CG3RK5 76310211 EC50 = 3070 nM T73482 CLY90X 76310431 IC50 > 10000 nM T73482 C6W4YC 76310456 IC50 = 1150 nM T73482 CT20QS 76313798 EC50 = 5700 nM T73482 C9V7HM 76313820 EC50 = 144 nM T73482 C07WGU 76313901 EC50 = 1360 nM T73482 C5ZE9C 76317346 EC50 = 1910 nM T73482 CEVZ91 76317683 IC50 = 17 nM T73482 C6CFQ9 76321148 EC50 = 2480 nM T73482 CP8M6Z 76321165 EC50 = 739 nM T73482 CM5HF7 76321386 IC50 = 2649 nM T73482 C9DZN3 76324691 EC50 = 1900 nM T73482 C1XSG9 76324989 IC50 = 32 nM T73482 CB3K9C 76328274 EC50 = 1370 nM T73482 CR6W3T 76328275 EC50 = 143 nM T73482 C6I7AK 76328558 IC50 = 14 nM T73482 C3O9LC 76331924 EC50 = 78.9 nM T73482 CRUK21 76331925 EC50 = 212 nM T73482 CVR8O9 76331964 EC50 = 865 nM T73482 CC9AR4 76332010 EC50 = 493 nM T73482 C54AVH 76332217 IC50 = 1590 nM T73482 C48LQC 76332218 IC50 = 2423 nM T73482 CNK25I 76332219 IC50 = 9704 nM T73482 C0ZN3F 76332238 IC50 = 537 nM T73482 CA1Z7X 76335540 EC50 = 1200 nM T73482 CV8NM6 76335605 EC50 = 3230 nM T73482 CVK6J7 76335606 EC50 = 422 nM T73482 CS2Y8O 76335607 EC50 = 3070 nM T73482 C2RVH7 76335608 EC50 = 3060 nM T73482 CRQ65T 76335879 IC50 > 10000 nM T73482 C0N3ZY 76534175 Ki = 391 nM T73482 CJG45W 76900605 Ki = 310 nM T73482 CXS7B6 77107594 Ki = 1.3 nM T73482 CVK3R4 78324905 Ki = 140 nM T73482 CZ8FN7 86267288 IC50 = 397 nM T73482 CEQ2V4 86269345 IC50 = 82 nM T73482 C9WI2E 86271116 Ki = 8 nM T73482 C9PVK1 86276237 IC50 = 18 nM T73482 CF4QX9 86278359 Ki = 800 nM T73482 C0PUY4 86291876 Ki = 64 nM T73482 CK6WQ1 86291877 Ki = 59 nM T73482 CHB7U8 86291879 IC50 = 828 nM T73482 CR32FQ 86292273 Ki = 120 nM T73482 CU0NT8 86298249 Ki = 130 nM T73482 CH4XK1 86302551 Ki = 0.5 nM T73482 CL7C5E 86302552 Ki = 0.9 nM T73482 C47MVU 86695644 IC50 = 14 nM T73482 CK9I5Y 89789751 IC50 = 3 nM T73482 C39TXO 89789760 IC50 = 2 nM T73482 C9I6NQ 89789762 IC50 = 264 nM T73482 C8S7BC 89789778 IC50 = 81 nM T73482 C0M7SQ 89789795 IC50 = 86 nM T73482 CERC67 89789843 IC50 = 20 nM T73482 CY9O3G 90405964 Ki = 12 nM T73482 C2WGJ3 90654337 Ki = 75 nM T73482 C8YE0S 90654338 Ki = 0.56 nM T73482 CZIE39 90654339 Ki = 470 nM T73482 C6TGU4 90654340 Ki = 17 nM T73482 CK38IX 90654341 Ki = 135 nM T73482 CL7KM1 90654342 Ki = 27 nM T73482 CFQS07 90654343 IC50 = 83 nM T73482 C8APK1 90654344 Ki = 26 nM T73482 C71YVR 90654345 Ki = 24 nM T73482 C2E5MT 90654346 Ki = 866 nM T73482 CPKH23 90654347 Ki = 211 nM T73482 CN7CX5 90654348 Ki = 18 nM T73482 CF0T9O 90654349 Ki = 76 nM T73482 C37MYP 90654350 Ki = 339 nM T73482 CJT36M 90654351 Ki = 108 nM T73482 CJ0Z5H 90656176 Ki = 0.7 nM T73482 CCW7S2 90656177 Ki = 0.3 nM T73482 C3EN1D 90656178 Ki = 2 nM T73482 CRK0W5 90656179 Ki = 4.5 nM T73482 CDN8Y4 90656180 Ki = 1.8 nM T73482 CJUS40 90656181 Ki = 1.8 nM T73482 CPSI06 90656182 Ki = 0.4 nM T73482 C8ZFG3 91801202 Ki = 1.585 nM T73482 C0DFT8 91809243 Ki = 166 nM T73482 CP0CE9 91810287 Ki = 140 nM T73482 CXO4N6 117668910 Ki = 430 nM T73482 C4HZ0N 117857721 IC50 = 3840 nM T73482 CJA8G5 117859490 IC50 > 10000 nM T73482 C1O2AH 117859572 IC50 = 21 nM T73482 C0CPN6 117859931 IC50 = 330 nM T73482 CZ20RX 118020300 IC50 = 10.1 nM T73482 C2Z1IN 118020504 IC50 = 61.5 nM T73482 CNI86H 118020539 IC50 = 245 nM T73482 CNKV57 118167452 Ki = 324 nM T73482 CSA7U9 118175269 Ki = 834 nM T73482 C72NVT 118175279 Ki = 6.3 nM T73482 CDAS04 118180165 Ki = 12 nM T73482 CK90HX 118435993 Ki = 1887 nM T73482 CF52MN 118715605 Ki = 2400 nM T73482 C4VR8L 118715606 IC50 > 10000 nM T73482 CG8MX4 118715607 IC50 > 10000 nM T73482 C1WKZ9 118715608 IC50 > 10000 nM T73482 CW4Z5M 118715609 IC50 = 4650 nM T73482 CN36LS 118715610 IC50 = 15000 nM T73482 C51JPK 118715611 IC50 = 10000 nM T73482 C1J2CY 118715612 Ki = 1500 nM T73482 CN14EP 118715613 Ki = 930 nM T73482 CNWA97 118716929 Ki > 10000 nM T73482 C3NW1S 118716930 Ki > 10000 nM T73482 CI3TK2 118716931 Ki = 4161 nM T73482 C5WRI1 118716932 Ki = 7.2 nM T73482 C5OQ4Y 118716933 Ki = 2994 nM T73482 C36PCB 118716934 Ki = 7535 nM T73482 CCT4Y0 118716935 Ki = 10000 nM T73482 CWJ69M 118716936 Ki = 6841 nM T73482 C9YEL0 118716937 Ki > 10000 nM T73482 CG5R1B 118716938 Ki = 5538 nM T73482 CHK4C7 118716939 Ki > 10000 nM T73482 CG75OB 118716940 Ki = 747 nM T73482 CG52QK 118716941 Ki = 772 nM T73482 C0QS6Y 118716942 Ki = 206 nM T73482 C10SEV 118716943 Ki = 1425 nM T73482 CAF89K 118716944 Ki = 291 nM T73482 C60JTD 118716945 Ki = 832 nM T73482 C2U1BX 118716946 Ki = 505 nM T73482 C83SPX 118716947 Ki = 106 nM T73482 C5ELB1 118716948 Ki = 103 nM T73482 C37UXI 118726303 Ki = 5.5 nM T73482 CFN4Y7 118726304 Ki = 106 nM T73482 C1Z7TR 118726305 Ki = 9 nM T73482 CX51TS 118726306 Ki = 13 nM T73482 CLQ34R 118726309 Ki = 470 nM T73482 CZ3OB5 118726310 Ki = 1100 nM T73482 C9WN2G 118726311 Ki = 510 nM T73482 CHM76O 118726312 Ki = 19000 nM T73482 C5S4RU 118726313 Ki = 1360 nM T73482 CS09EU 118726314 Ki = 1200 nM T73482 CN2KE3 118731950 IC50 = 3960 nM T73482 CF4QD0 118731951 IC50 = 7030 nM T73482 CYNB60 118731952 IC50 = 1980 nM T73482 C0VU1B 118731953 IC50 = 5780 nM T73482 CH8T0S 118731954 IC50 = 2400 nM T73482 C7KX2R 118731955 IC50 = 8720 nM T73482 CWA05F 118731956 IC50 = 3620 nM T73482 CC3PT6 118731957 IC50 = 467 nM T73482 CXEO47 118731958 IC50 = 1200 nM T73482 CTY98B 118736949 Ki = 12 nM T73482 C19HQW 118736950 Ki = 37 nM T73482 CRJ9L8 118736951 Ki = 14000 nM T73482 C82NQB 118736952 Ki = 57 nM T73482 CVO72M 118736953 Ki = 49 nM T73482 CWH08B 118736954 Ki = 470 nM T73482 CLAR49 118736955 Ki = 39 nM T73482 C3G6VD 118736956 Ki = 350 nM T73482 CCK3A9 118736957 Ki = 1400 nM T73482 CYBN01 118736958 Ki = 360 nM T73482 CLNY63 118736959 IC50 = 10000 nM T73482 CNU4D7 118736960 IC50 = 7100 nM T73482 CKFZ15 118736961 IC50 = 3300 nM T73482 COPD90 118736962 IC50 > 10000 nM T73482 CJ3VD1 118736963 IC50 > 10000 nM T73482 CMRB20 121231398 Ki = 393 nM T73482 CYHP86 122179999 Ki > 2000 nM T73482 CI3Q9N 122180000 Ki > 2000 nM T73482 CND0S5 122180001 Ki = 171 nM T73482 C0T3SD 122180002 Ki = 2491 nM T73482 C6CG5E 122180317 Ki = 6850 nM T73482 CQR14H 122180318 Ki = 5300 nM T73482 CE36GC 122180319 Ki > 10000 nM T73482 CVL0Q7 122180320 Ki > 10000 nM T73482 CW8H2J 122180321 Ki > 10000 nM T73482 CS1JC7 122180322 Ki = 1398 nM T73482 C6FVZ0 122180323 Ki = 925 nM T73482 CX9JG0 122180324 Ki = 267 nM T73482 CQU2H9 122180325 Ki = 765 nM T73482 CA5CP8 122180326 Ki = 1320 nM T73482 C6CAZ0 122180327 Ki > 10000 nM T73482 CRVB56 122180328 Ki > 10000 nM T73482 CAL3T2 122180329 Ki = 623 nM T73482 C3OJS0 122180330 Ki = 471 nM T73482 C4YIX5 122180331 Ki = 1800 nM T73482 C2DZ3Y 122180332 Ki = 3300 nM T73482 C0W3JG 122180333 Ki > 10000 nM T73482 C6EF1H 122180334 Ki = 557 nM T73482 C8SD7F 122180335 Ki = 257 nM T73482 C2WV9G 122180336 Ki = 1640 nM T73482 CJ1AP3 122180337 Ki = 2280 nM T73482 CBN0J2 122180338 Ki = 1960 nM T73482 CEA80S 122180339 Ki = 5780 nM T73482 CTG4B2 122180340 Ki = 3650 nM T73482 C6Y0JD 122180341 Ki = 680 nM T73482 CTCN25 122180342 Ki = 3090 nM T73482 C35BFD 122180343 Ki = 346 nM T73482 C80QZN 122180344 Ki = 5750 nM T73482 C6YIR4 122180345 Ki = 4630 nM T73482 CO1AK6 122184039 Ki = 0.06 nM T73482 C5XOD3 122184040 Ki = 23 nM T73482 CAYV10 122184041 IC50 = 259 nM T73482 CUWG52 122184042 Ki = 19 nM T73482 CTL34Z 122184043 Ki = 10 nM T73482 CVRO25 122184044 Ki = 12 nM T73482 C3WUY1 122184045 Ki = 4 nM T73482 C9HF4M 122191823 EC50 = 5227 nM T73482 CBI0X1 122191829 EC50 = 9248 nM T73482 CQ8FE7 122192247 EC50 = 6134 nM T73482 C5YRQ9 122192248 EC50 = 5720 nM T73482 CMX26J 122192250 EC50 = 2750 nM T73482 C4TX5S 122195752 Ki = 7 nM T73482 CD57NR 127027859 Ki = 34 nM T73482 CM91FC 127037650 IC50 = 16 nM T73482 CBT18A 127037651 IC50 = 45 nM T73482 CLD41N 127037996 IC50 = 2.7 nM T73482 C8INE9 127038060 IC50 = 16 nM T73482 CC3T8J 127038061 IC50 = 23 nM T73482 CJ03FI 127038062 IC50 = 3.5 nM T73482 CACI97 127038343 IC50 = 60 nM T73482 C4P7YM 127038416 IC50 = 33 nM T73482 C54FRL 127038812 IC50 = 64 nM T73482 CV6QR8 127038813 IC50 = 3.4 nM T73482 CRE04H 127038817 IC50 = 13 nM T73482 C71SOB 127038818 IC50 = 22 nM T73482 CRY01S 127038819 IC50 = 111 nM T73482 CSHM50 127038820 IC50 = 9.1 nM T73482 CNG1V0 127038821 IC50 = 11 nM T73482 CW47SG 127038822 IC50 = 8.3 nM T73482 CV8Z7T 127039127 IC50 = 3.8 nM T73482 CVOW03 127039128 IC50 = 26 nM T73482 C5IX1B 127039129 IC50 = 33 nM T73482 C1YUH6 127039134 IC50 = 11 nM T73482 C1NZ6H 127039135 IC50 = 17 nM T73482 CIBD78 127040414 IC50 = 28 nM T73482 COM28D 127040734 IC50 = 131 nM T73482 C37QEO 127040735 IC50 = 28 nM T73482 C6DEH8 127040736 IC50 = 108 nM T73482 CAX2I9 127040737 IC50 = 8.5 nM T73482 CTW7A2 127041999 Ki = 398.11 nM T73482 C07JPS 127042658 IC50 = 35 nM T73482 CX46KS 129093666 Ki = 1.96 nM T73482 CMZL51 129093667 Ki = 12.5 nM T73482 CP4TZ9 129093668 Ki = 6.21 nM T73482 CQ3I9T 129093669 Ki = 7.3 nM T73482 C5ZB7M 129093671 Ki = 13.9 nM T73482 C7M4SR 129093672 Ki = 12.1 nM T73482 C10DMA 129093673 Ki = 4.16 nM T73482 C4ABF5 129093675 Ki = 5.94 nM T73482 C4SU9L 129093829 Ki = 12 nM T73482 C40IXC 129093915 Ki = 2.1 nM T73482 C37OWP 129093916 Ki = 5.13 nM T73482 C9WTZ8 129093917 Ki = 3.47 nM T73482 CSB23A 129093918 Ki = 2.27 nM T73482 C3BI6O 129093944 Ki = 2.98 nM T73482 C8OD1A 129093945 Ki = 5.85 nM T73482 C1NF8H 129093946 Ki = 1.7 nM T73482 CDH9X8 129093947 Ki = 2.05 nM T73482 CV37XJ 129093951 Ki = 1.93 nM T73482 CRA76C 129093952 Ki = 7.6 nM T73482 CET1F7 129093953 Ki = 4.05 nM T73482 C2LWQ1 129093954 Ki = 2.07 nM T73482 CJB3M8 129093969 Ki = 6.19 nM T73482 CKL03Y 129093972 Ki = 12.6 nM T73482 CHB4I5 129093973 Ki = 1.81 nM T73482 C59FVA 129093974 Ki = 5.05 nM T73482 CSFT64 132537576 Ki = 1.36 nM T73482 CU58RD 135314438 Ki = 2.06 nM T73482 C9RA0Q 135314513 Ki = 22.5 nM T73482 CPZ89B 135314564 Ki = 8.14 nM T73482 C75NWT 136227358 IC50 > 30000 nM T73482 C9WUL6 137632260 Ki = 14 nM T73482 C24MIN 137632538 IC50 > 10000 nM T73482 C61SQF 137633141 Ki = 2.44 nM T73482 C3UBF8 137634720 IC50 = 489 nM T73482 CH4KC1 137635768 Ki = 42.3 nM T73482 C0BRG6 137636340 IC50 = 113 nM T73482 C0G8TB 137637342 IC50 = 3239 nM T73482 C4W3YF 137637374 Ki = 8.99 nM T73482 C7FUO1 137638475 Ki = 31.6 nM T73482 C04EGF 137638805 IC50 = 293 nM T73482 CYB93R 137638895 IC50 = 5020 nM T73482 CZ91SV 137638898 IC50 > 10000 nM T73482 CQ5J0X 137639504 Ki = 320 nM T73482 CT90FM 137640166 IC50 > 10000 nM T73482 C79OCZ 137641214 Ki = 7.25 nM T73482 CIPJ41 137641369 IC50 = 1963 nM T73482 C5OXI1 137642484 IC50 = 759 nM T73482 CX3MK7 137642825 IC50 = 1895 nM T73482 CNM4F9 137643075 Ki = 541 nM T73482 C2DIV4 137644135 IC50 = 1910 nM T73482 C6M0BL 137644509 IC50 = 216 nM T73482 C9ABK7 137644534 IC50 = 327 nM T73482 C6KM9A 137645155 Ki = 6.37 nM T73482 C2MRK0 137645329 Ki = 18.9 nM T73482 C9GP2E 137645716 Ki = 10 nM T73482 CC6KI7 137646689 IC50 = 3918 nM T73482 CF98UE 137647371 IC50 = 502 nM T73482 C2BQ4U 137648163 IC50 = 1010 nM T73482 C4VD0P 137649196 IC50 > 10000 nM T73482 CLZ2N8 137649834 IC50 = 226 nM T73482 C1TW0K 137650367 Ki = 12 nM T73482 C7X0SU 137651169 Ki = 849 nM T73482 CR5F0I 137652411 IC50 = 303 nM T73482 C36YGM 137653736 Ki = 389 nM T73482 CPE53S 137654752 Ki = 1.92 nM T73482 C08XSJ 137655492 IC50 > 10000 nM T73482 C1MJG9 137655850 IC50 = 1636 nM T73482 C7R3IU 137656102 Ki = 14 nM T73482 CQ0UG7 137657078 IC50 = 2973 nM T73482 C7VFU4 137657849 IC50 = 736 nM T73482 CF7Q6D 137658206 IC50 = 908 nM T73482 C63RQO 137658775 IC50 = 517 nM T73482 C89FIO 137659457 IC50 = 1776 nM T73482 CNH3U0 137660075 IC50 > 10000 nM T73482 C38LZW 137660448 Ki = 11.2 nM T73482 CQ0J2X 137660887 IC50 = 401 nM T73482 CUMN86 137662108 Ki = 66 nM T73482 CNX2Q5 137662177 Ki = 12.9 nM T73482 CZ4S3O 144671360 IC50 = 89 nM T73482 CF0Z8D 145714283 Ki = 15.85 nM T73482 CS9B7W 145971593 Ki = 1.97 nM T73482 C27YQH 145975735 Ki = 187 nM T73482 C7CO2P 145977763 Ki = 17.8 nM T73482 C6VWK3 145979924 Ki = 4800 nM T73482 CGRU50 145989367 Ki = 5400 nM T73482 C3M1WQ 145994245 Ki = 3100 nM T73482 CQD73L 155515631 Ki = 502 nM T73482 C2B1ZG 155517489 Ki > 10 nM T73482 CH3MT0 155519961 Ki > 10 nM T73482 C9D3AS 155520434 Ki = 5.89 nM T73482 CF1N4P 155524300 Ki = 461 nM T73482 CWL04C 155524427 Ki = 4.34 nM T73482 CB3JY5 155525887 Ki = 5.51 nM T73482 C5EM4D 155532688 Ki = 9.35 nM T73482 C4VQ8A 155543013 Ki > 10 nM T73482 CP7I4W 155543165 Ki > 10 nM T73482 CFMK42 155543728 Ki = 101 nM T73482 CIY9N3 155554119 Ki > 10 nM T73482 CQ30PW 155557825 Ki = 20.9 nM T73482 CRDS43 155566853 Ki = 842 nM T73482 CM93SV 155567436 Ki = 7.45 nM T73482 CQ1RW5 155568320 Ki > 10000 nM T73482 D01SUL 9869934 Ki = 5.012 nM T73482 D02MDC 9981404 Ki = 900 nM T73482 D08MXD 73349109 Ki = 1.1 nM T73482 D0J3PJ 4331799 Ki = 22 nM T73482 D0KP3K 10065953 Ki = 8.7 nM T73482 D0R4BT 10046856 Ki = 100 nM T73482 D0U0TS 10408514 IC50 > 10000 nM T73482 D0UZ4J 6604926 Ki = 14 nM T36483 D0VA0I 10077130 IC50 = 1.1 nM T36483 D0PU8T 10459564 IC50 = 31.62 nM T36483 D08ELM 9832212 IC50 = 5 nM T36483 CO6X0U 128205 IC50 = 9000 nM T36483 C98PBF 752812 IC50 = 10000 nM T36483 CX79RF 807100 IC50 = 1120 nM T36483 C0DXY9 877874 IC50 = 1680 nM T36483 C1HPL9 1047175 IC50 = 900 nM T36483 C4U2DR 1047178 IC50 = 2866 nM T36483 C82PVQ 1047179 IC50 = 98 nM T36483 CWTG42 1048267 IC50 = 199.53 nM T36483 C48FJQ 1361448 IC50 = 3120 nM T36483 CYN6E5 2858257 IC50 = 33 nM T36483 CCIE45 2858875 IC50 = 65 nM T36483 C1QC2W 3109060 IC50 = 316.23 nM T36483 CLBW26 3378161 IC50 = 1410 nM T36483 CXU4P3 3751851 IC50 = 359 nM T36483 CZS63L 4259181 IC50 = 56 nM T36483 C8LYU1 4314709 IC50 = 964 nM T36483 CD4YR5 7006478 EC50 > 800000 nM T36483 C2ST5A 9801767 IC50 = 700 nM T36483 CO28KU 9805672 IC50 = 1000 nM T36483 CB6E8G 9808447 EC50 = 760 nM T36483 CSV54F 9809471 EC50 = 1000 nM T36483 C8UDN9 9810474 IC50 = 1600 nM T36483 CVDI10 9810475 IC50 = 6700 nM T36483 CK1NW8 9810477 EC50 = 2900 nM T36483 C3B7WM 9825804 IC50 = 20 nM T36483 CZWL57 9831601 IC50 = 30000 nM T36483 C2HY1Z 9831828 IC50 = 5000 nM T36483 C6CRK1 9831948 IC50 = 5600 nM T36483 CAW29Z 9844209 IC50 = 22 nM T36483 C69RDJ 9847494 IC50 = 150 nM T36483 CBKT76 9851501 EC50 = 1200 nM T36483 C75JUE 9853816 IC50 = 270 nM T36483 CSB56V 9855084 EC50 = 8000 nM T36483 CN48IZ 9865055 IC50 = 27 nM T36483 CR80DB 9869359 IC50 = 21.5 nM T36483 CGET90 9875040 EC50 = 21000 nM T36483 CWI9F8 9875337 EC50 = 1100 nM T36483 CW18TC 9886874 IC50 = 15 nM T36483 CC85QB 9889179 IC50 = 10 nM T36483 CRK15D 9890926 Ki = 11 nM T36483 CXWF97 9895920 EC50 = 460 nM T36483 CV8GN6 9896668 IC50 > 100000 nM T36483 CO93LE 9897054 IC50 = 25 nM T36483 C8H1QX 9908345 IC50 = 22 nM T36483 CG36KH 9919038 IC50 = 570 nM T36483 CC75WO 9931987 IC50 = 10 nM T36483 CT67FC 9934461 IC50 = 23 nM T36483 C7NWE2 9937578 EC50 = 3900 nM T36483 CL28YV 9951647 IC50 = 6.3 nM T36483 CJH61W 9960837 EC50 = 1000 nM T36483 CB7PQ1 9961058 EC50 = 510 nM T36483 CC3BO7 9962227 EC50 = 1000 nM T36483 CBI45Z 9982475 EC50 = 185000 nM T36483 CK0OF1 9986700 EC50 = 800000 nM T36483 CYH1Z5 9986822 EC50 = 400 nM T36483 CXIF90 9987318 EC50 = 600000 nM T36483 CAHV37 10000177 IC50 = 52 nM T36483 CEOA76 10010285 EC50 = 200 nM T36483 C6RMX0 10032001 EC50 = 109300 nM T36483 CWZ42G 10032227 EC50 = 700 nM T36483 C0UD8L 10054163 EC50 = 15000 nM T36483 C2UJ7B 10054787 EC50 = 730000 nM T36483 CJ9P1Z 10078162 EC50 = 19000 nM T36483 C60PZS 10078455 EC50 > 1200000 nM T36483 C03XAC 10079418 EC50 = 10 nM T36483 C82XUE 10095734 IC50 = 20 nM T36483 CU25DY 10099272 EC50 > 800000 nM T36483 C19QPS 10101423 EC50 = 270 nM T36483 C8K9OD 10120960 IC50 = 1200 nM T36483 C1TB4S 10161572 IC50 = 350 nM T36483 CO5NT2 10162707 IC50 = 830 nM T36483 CN0ZW5 10164471 IC50 = 4440 nM T36483 C7XNK5 10184176 IC50 = 1100 nM T36483 CT96NH 10204371 IC50 = 6600 nM T36483 CG52LT 10206026 IC50 = 430 nM T36483 CB32WA 10227544 IC50 = 2100 nM T36483 CBSL17 10246587 Ki = 12 nM T36483 CNG2M1 10257805 EC50 = 200000 nM T36483 CUO92S 10259068 EC50 = 500 nM T36483 C19IWT 10260648 EC50 > 800000 nM T36483 CMX30H 10276545 IC50 = 130 nM T36483 CLE90J 10278388 IC50 = 3700 nM T36483 CT69SW 10279248 IC50 = 3200 nM T36483 C28CZY 10300275 IC50 = 120 nM T36483 CME8H2 10325208 EC50 = 70000 nM T36483 CD7B9J 10328351 IC50 = 3100 nM T36483 CF9Q3K 10345602 Ki = 1900 nM T36483 CKZ0T7 10348644 EC50 = 1200 nM T36483 CSU8H4 10350578 EC50 = 500 nM T36483 CCGH96 10350886 IC50 = 7.5 nM T36483 CL9EB4 10351173 EC50 = 3300 nM T36483 C4AZW0 10371218 EC50 = 1300 nM T36483 C8EPN7 10390481 Ki = 6600 nM T36483 CB65WG 10394462 EC50 > 800000 nM T36483 COZ92M 10415062 EC50 > 800000 nM T36483 CM3ZX0 10416585 EC50 = 415000 nM T36483 C4QX8B 10416597 EC50 = 235000 nM T36483 CI5AZ6 10416607 EC50 = 800000 nM T36483 CO8U9A 10416608 EC50 > 800000 nM T36483 C0C3ZK 10416646 EC50 = 200 nM T36483 CGDA78 10416780 EC50 = 350000 nM T36483 C1Q6JH 10417097 EC50 = 140 nM T36483 C6KA0H 10418424 EC50 = 24500 nM T36483 CHAN91 10439025 EC50 > 800000 nM T36483 C21MID 10439062 EC50 = 500000 nM T36483 C8M7SV 10441247 EC50 > 800000 nM T36483 CXZJ53 10461499 EC50 = 11700 nM T36483 C02WYD 10461589 EC50 = 28000 nM T36483 CTY5H0 10462502 EC50 = 400000 nM T36483 CO02ET 10484360 EC50 = 21400 nM T36483 CE0PF1 10484500 EC50 > 800000 nM T36483 C4VN0A 10526120 IC50 = 80 nM T36483 CMVI23 10557086 IC50 = 24 nM T36483 CRFI52 10622095 IC50 = 90 nM T36483 C2FLV0 10628873 IC50 = 29 nM T36483 CTF43Q 10741717 IC50 = 80 nM T36483 CI96NX 10747898 EC50 = 1800 nM T36483 CF9Y3J 10771636 IC50 = 19 nM T36483 C4SQ5G 10818136 EC50 = 720 nM T36483 CIR3E1 10819322 IC50 = 300 nM T36483 CQ6G0B 10925413 IC50 = 1500 nM T36483 CD25QZ 11502485 IC50 = 25 nM T36483 C5ZWX6 11502697 IC50 = 1000 nM T36483 CNOC42 11503433 IC50 = 46 nM T36483 CQE03H 11508687 IC50 = 850 nM T36483 CRT82D 11509594 IC50 = 325 nM T36483 CA7D8B 11515660 IC50 = 1500 nM T36483 C43BGM 11516923 IC50 = 900 nM T36483 CVT96B 11537143 IC50 = 300 nM T36483 C2BM8L 11544606 IC50 = 150 nM T36483 CR6UX2 11544845 IC50 = 210 nM T36483 C4M3HK 11553497 IC50 = 11 nM T36483 CQZI28 11559190 IC50 = 1250 nM T36483 C8RZJ4 11567556 IC50 = 14 nM T36483 C38CUB 11576348 IC50 = 100 nM T36483 C9PG8E 11582568 IC50 = 26 nM T36483 C1TE7Q 11583548 IC50 = 25 nM T36483 C9QN7H 11603083 IC50 = 143 nM T36483 CO2P9S 11610042 IC50 = 250 nM T36483 C5B9MN 11611061 IC50 = 13 nM T36483 CN5C2X 11611425 IC50 = 204 nM T36483 CN9VJ8 11618945 IC50 = 29 nM T36483 C3H2TL 11624004 IC50 > 5000 nM T36483 C23DJQ 11639231 IC50 = 550 nM T36483 CAT1C0 11645276 IC50 = 4000 nM T36483 CO37QK 11647382 IC50 = 19 nM T36483 C4CY7V 11652756 IC50 = 1100 nM T36483 CI6QM8 11661666 IC50 = 28 nM T36483 CD5SX3 11674764 IC50 = 725 nM T36483 C6UGL9 11682882 IC50 = 467 nM T36483 CO92VG 11684648 IC50 = 50 nM T36483 CS7FH4 11688420 IC50 = 2100 nM T36483 CV4OW8 11690507 IC50 = 19 nM T36483 C6VQH5 11691128 IC50 = 44 nM T36483 C4AYW2 11697104 IC50 = 35 nM T36483 CD2M6O 11702885 IC50 = 325 nM T36483 CPJG59 11703925 IC50 = 3500 nM T36483 CIYF09 11712191 IC50 > 300 nM T36483 C8G1ZT 11718309 IC50 = 3681 nM T36483 CV9Q1B 11758525 EC50 = 800 nM T36483 C9K6JA 11764645 EC50 > 800000 nM T36483 C4JG1W 11803290 IC50 = 25 nM T36483 CZ74PR 11803426 EC50 = 3700 nM T36483 CLDX73 11803455 IC50 = 193000 nM T36483 CDXL23 11818750 EC50 = 2000 nM T36483 C90MCQ 12018757 IC50 = 2990 nM T36483 CG6Q4B 12018758 IC50 = 910 nM T36483 CP15ZG 12018759 IC50 = 990 nM T36483 CT7Z2V 12018762 IC50 = 140 nM T36483 C2B8GR 15887956 IC50 = 4000 nM T36483 CKPY93 15887958 IC50 = 65000 nM T36483 C8QO3Z 15887960 IC50 = 40000 nM T36483 CKVM71 16046150 IC50 = 18 nM T36483 CG2NT3 16100342 IC50 = 41 nM T36483 CCG1W9 16100343 IC50 = 845 nM T36483 CY5FP4 16100350 IC50 = 37 nM T36483 CRF9T3 16100351 IC50 = 53 nM T36483 CRNU53 16100352 IC50 = 28 nM T36483 CQD1R6 16100353 IC50 = 481 nM T36483 CM07ZP 17187522 IC50 = 770 nM T36483 CPW18A 17187534 IC50 = 1100 nM T36483 CPFW98 17187609 IC50 = 970 nM T36483 CZWL06 17222599 IC50 = 199.53 nM T36483 C3Y2KE 17222608 IC50 = 1800 nM T36483 CHVR74 22611774 IC50 = 28000 nM T36483 CVM5Q1 22611776 IC50 > 10000 nM T36483 C5LH4U 22611792 IC50 = 2000 nM T36483 C2WR9E 22611889 IC50 > 10000 nM T36483 C4V7BI 22645287 IC50 = 8000 nM T36483 C7EQ5O 23628249 IC50 = 7.6 nM T36483 C5EG4O 23630913 IC50 = 22 nM T36483 CN1EW7 23630914 IC50 = 200 nM T36483 CE86TG 23630915 IC50 = 80 nM T36483 C1PKN9 23631103 IC50 = 17 nM T36483 C69YXL 23631104 IC50 = 26 nM T36483 CD7WU0 23631105 IC50 = 25 nM T36483 CSC80P 23631106 IC50 = 26 nM T36483 C4C5JA 23631184 IC50 = 19 nM T36483 CS89QV 23631185 IC50 = 13 nM T36483 C26ENM 23631186 IC50 = 21 nM T36483 CSKH79 23631187 IC50 = 11 nM T36483 C83UCD 23631188 IC50 = 8 nM T36483 CO5CD4 23631275 IC50 = 33.5 nM T36483 CNGH14 23631277 IC50 = 762 nM T36483 CM93CL 23631278 IC50 = 550 nM T36483 CI8HF9 23631279 IC50 = 37.5 nM T36483 C2F6CI 23631374 IC50 = 15.5 nM T36483 CZR10M 23631375 IC50 = 1101 nM T36483 CHN4X8 23631376 IC50 = 18.5 nM T36483 CEP5C7 23631377 IC50 = 101 nM T36483 CD4MH1 23631464 IC50 = 25 nM T36483 C6RH3X 23631554 IC50 = 224 nM T36483 CXUF30 23631639 IC50 = 153 nM T36483 C4L9ZI 23631640 IC50 = 295 nM T36483 CEI32D 23631809 IC50 = 600 nM T36483 CH9AO6 23631810 IC50 = 113 nM T36483 CH25IR 23631811 IC50 = 8 nM T36483 C59OSL 23631812 IC50 = 15 nM T36483 C9GVK3 23631813 IC50 = 16.5 nM T36483 CNB2Z0 23631900 IC50 = 600 nM T36483 CP23YQ 24830436 Ki = 17 nM T36483 CC65LO 24830595 Ki = 6.1 nM T36483 CO8MA9 24878827 Ki = 13 nM T36483 C6IX1G 24878828 Ki = 20 nM T36483 C0N4AJ 24878829 Ki = 30 nM T36483 C6W9PK 24878871 Ki = 6.4 nM T36483 CC2E7B 24878872 Ki = 6.5 nM T36483 CQ4VO9 24878873 Ki = 6.2 nM T36483 C1DJS3 24878874 Ki = 4.4 nM T36483 C45EUD 24878875 Ki = 4.8 nM T36483 CB6P4R 24878927 Ki = 11 nM T36483 CV7SN0 24878928 Ki = 10 nM T36483 CDX49C 24878929 Ki = 44 nM T36483 CBCR43 24878930 Ki = 4.1 nM T36483 CJB97D 24878981 Ki = 89 nM T36483 C6Y5DM 24878982 Ki = 3.7 nM T36483 CCV09N 24878983 Ki = 5.9 nM T36483 CAF0C7 24878984 Ki = 11 nM T36483 CC4A6K 24879035 Ki = 367 nM T36483 CMH5P1 24879036 Ki = 1.8 nM T36483 CBE9L3 24879037 Ki = 11 nM T36483 C1MXQ6 24879038 Ki = 5.9 nM T36483 CFU61L 24879079 Ki = 11 nM T36483 C9RND0 44264660 Ki = 14000 nM T36483 CQ2R6H 44280522 IC50 = 7600 nM T36483 CE9G2Z 44280585 EC50 = 760 nM T36483 CK18FO 44280607 EC50 = 28000 nM T36483 CBKV73 44280608 EC50 = 1700 nM T36483 CN95GQ 44280649 IC50 = 4000 nM T36483 CQ95NM 44280650 IC50 = 1400 nM T36483 CFZX80 44280651 EC50 = 5000 nM T36483 CK34GX 44280660 IC50 = 3000 nM T36483 CY8WM5 44280667 EC50 = 5800 nM T36483 CCF1H9 44280683 EC50 = 8000 nM T36483 C0PFB8 44280685 EC50 = 1300 nM T36483 CYV23Q 44280703 IC50 = 7000 nM T36483 CZBU08 44280731 IC50 = 10000 nM T36483 C47GQL 44280767 EC50 = 1000 nM T36483 CE9LF7 44280768 EC50 = 3100 nM T36483 CHP49J 44280804 EC50 = 2000 nM T36483 CU0K5H 44280805 IC50 = 25000 nM T36483 C78GZV 44280822 EC50 = 4200 nM T36483 CK8W4F 44280835 IC50 = 27000 nM T36483 CFW53T 44280876 IC50 = 10000 nM T36483 C4SZK0 44280877 EC50 = 2100 nM T36483 C9T8SX 44280878 IC50 = 46000 nM T36483 CXAT87 44280898 IC50 = 10000 nM T36483 CCS25K 44280899 IC50 = 4400 nM T36483 C9C0HI 44280905 IC50 = 2600 nM T36483 C2JD9S 44280935 EC50 = 2400 nM T36483 CG7X6F 44280936 EC50 = 7900 nM T36483 C84DSX 44280949 EC50 = 1200 nM T36483 CC6HB0 44280954 IC50 = 16000 nM T36483 CS5FV7 44280955 EC50 = 4900 nM T36483 CJMQ02 44281047 EC50 = 14000 nM T36483 C18ZQK 44281069 IC50 = 13000 nM T36483 C0GKP4 44281070 IC50 = 2300 nM T36483 C3QA2W 44281079 IC50 = 2400 nM T36483 CT27UM 44281080 IC50 = 2900 nM T36483 CDH74W 44281081 IC50 = 2000 nM T36483 C6J3CG 44281172 EC50 = 10500 nM T36483 CM29OK 44281173 IC50 = 9000 nM T36483 C7C4ZT 44281174 IC50 = 18000 nM T36483 CV2Q5K 44281237 EC50 = 2600 nM T36483 C2EU9P 44281263 IC50 = 5000 nM T36483 C50SCD 44281264 IC50 = 56000 nM T36483 CW94SR 44281289 EC50 = 9700 nM T36483 C5P7QN 44289942 IC50 > 100000 nM T36483 CF4J5T 44289951 IC50 > 100000 nM T36483 CQ32XB 44289954 IC50 = 8000 nM T36483 CPI04Z 44290058 IC50 = 5400 nM T36483 C51LBS 44290059 IC50 = 6200 nM T36483 C0LT9V 44290102 IC50 = 2700 nM T36483 CYDK89 44290104 IC50 = 10000 nM T36483 CLPO09 44290110 IC50 = 60000 nM T36483 C8LZ7F 44290166 IC50 = 4100 nM T36483 CHI87Y 44290181 IC50 = 5000 nM T36483 C2R4LT 44290206 IC50 = 24000 nM T36483 CYS73M 44290207 IC50 = 24000 nM T36483 CRP2J4 44290231 IC50 = 5700 nM T36483 CGT83M 44290234 IC50 = 8200 nM T36483 C7TF4J 44290251 IC50 = 94000 nM T36483 CWM53Q 44290276 IC50 = 53000 nM T36483 C2PY9U 44290300 IC50 = 2700 nM T36483 C74XUM 44305776 IC50 = 300 nM T36483 CGF8T4 44305882 IC50 = 1250 nM T36483 CEA1W6 44305896 IC50 = 870 nM T36483 C8D0JY 44305897 IC50 = 524 nM T36483 C9OL6V 44305939 IC50 = 4500 nM T36483 CH1ZU6 44305942 IC50 = 1750 nM T36483 CN0BF5 44305944 IC50 = 3200 nM T36483 CY7D3U 44305948 IC50 = 100 nM T36483 CZL50Q 44305953 IC50 = 4900 nM T36483 C2IQS3 44305954 IC50 = 100 nM T36483 C0EM9F 44305955 IC50 = 9600 nM T36483 CB90FJ 44306065 IC50 = 1230 nM T36483 CNR6Y4 44306066 IC50 = 2625 nM T36483 C7AC4M 44306076 IC50 = 6875 nM T36483 CUG1B0 44306336 IC50 = 600 nM T36483 CGX38W 44306402 IC50 = 310 nM T36483 CRIA53 44306403 IC50 = 230 nM T36483 C5QFP0 44306404 IC50 = 1000 nM T36483 C4IXK0 44306499 IC50 = 1300 nM T36483 CO70XF 44306500 IC50 = 140 nM T36483 CT2JH0 44306501 IC50 = 70 nM T36483 CDV41R 44306540 IC50 = 640 nM T36483 C2FYC6 44306599 IC50 = 100 nM T36483 C9QYF1 44306611 IC50 = 400 nM T36483 CFEN89 44306612 IC50 = 36500 nM T36483 C9C6OD 44306657 IC50 = 4800 nM T36483 CT7L9J 44306658 IC50 = 3500 nM T36483 CAVY39 44306659 IC50 = 400 nM T36483 C0QVF7 44306660 IC50 = 900 nM T36483 CW6R7A 44306696 IC50 = 2000 nM T36483 C1G9RQ 44306697 IC50 = 240 nM T36483 CY9QL2 44306698 IC50 = 200 nM T36483 CM90EW 44306708 IC50 = 1300 nM T36483 C8VJ7B 44306732 IC50 = 500 nM T36483 CR9J2L 44306761 IC50 = 440 nM T36483 CT58LC 44306762 IC50 = 100 nM T36483 CJL6R7 44306894 IC50 = 900 nM T36483 C20CMS 44306903 IC50 = 2300 nM T36483 CRV4M7 44309450 IC50 = 2000 nM T36483 CE85SQ 44309461 IC50 = 230 nM T36483 CB20GZ 44309471 IC50 = 70 nM T36483 C9RP0K 44309472 IC50 = 500 nM T36483 CQJD59 44309477 IC50 = 120 nM T36483 C81MZX 44309730 IC50 = 480 nM T36483 CU4TG6 44309750 IC50 = 160 nM T36483 CID42J 44309751 IC50 = 330 nM T36483 C7Y1QM 44309776 IC50 = 430 nM T36483 C9SBO3 44309777 IC50 = 310 nM T36483 CF98YJ 44309838 IC50 = 22000 nM T36483 CJU6I8 44309958 IC50 = 35 nM T36483 CLFB39 44309959 IC50 = 70 nM T36483 C7MVQ9 44310191 IC50 = 90 nM T36483 CW2Z1T 44310308 IC50 = 60 nM T36483 C1ZCH0 44310323 IC50 = 130 nM T36483 CJN6H3 44315779 IC50 > 10000 nM T36483 C8LQ3E 44315780 IC50 = 20000 nM T36483 C5XE1O 44315792 IC50 = 5000 nM T36483 CPT6R4 44315793 IC50 = 7000 nM T36483 C2TE0B 44316045 IC50 = 2000 nM T36483 C7P1CL 44316059 IC50 = 7000 nM T36483 CDVZ48 44316106 IC50 = 4000 nM T36483 C9B8CD 44316156 IC50 = 800 nM T36483 CUBM67 44316184 IC50 = 1000 nM T36483 CAI6P7 44316522 IC50 = 300 nM T36483 C8DRY2 44316532 IC50 = 3000 nM T36483 CYTL98 44316560 IC50 = 11000 nM T36483 C6QU9I 44316563 IC50 > 50000 nM T36483 C2D5ZR 44324193 IC50 = 700 nM T36483 CIJF13 44328197 IC50 = 9000 nM T36483 CKC07Y 44328340 IC50 = 3100 nM T36483 C7M8TH 44328342 IC50 = 13000 nM T36483 C1SG3Y 44328381 IC50 = 3400 nM T36483 C5HI4J 44328383 IC50 = 9700 nM T36483 CL2FU7 44328523 IC50 = 300 nM T36483 CNS8K1 44328562 IC50 = 6000 nM T36483 C3B6RN 44328579 IC50 = 1324 nM T36483 CV5XZ1 44328647 IC50 = 734 nM T36483 C8I3EG 44328728 IC50 = 1500 nM T36483 CWI9D5 44338787 IC50 = 500 nM T36483 CM05QN 44338791 IC50 = 90 nM T36483 C5A6JX 44338864 IC50 = 360 nM T36483 C89OIS 44338865 IC50 = 5000 nM T36483 CQ6I8E 44338875 IC50 = 500 nM T36483 C73QCH 44338882 IC50 = 600 nM T36483 CLUN47 44338885 IC50 = 1600 nM T36483 CHY5J0 44338886 IC50 = 3300 nM T36483 CVA3B2 44338887 IC50 > 10000 nM T36483 CCLA27 44338895 IC50 = 2000 nM T36483 C3V2YS 44338903 IC50 > 10000 nM T36483 CZ69BK 44338917 IC50 = 1000 nM T36483 C20HJG 44338928 IC50 > 10000 nM T36483 C91WXN 44338929 IC50 = 130 nM T36483 CI1Q0K 44338944 IC50 = 70 nM T36483 CM8C9F 44338946 IC50 = 400 nM T36483 CMKH71 44339001 IC50 = 2210 nM T36483 C9ZK0U 44339002 IC50 = 290 nM T36483 CY5V7Z 44339029 IC50 = 120 nM T36483 C2AE6H 44339030 IC50 = 6420 nM T36483 CWRP93 44339048 IC50 > 10000 nM T36483 CIE4V2 44339055 IC50 = 3220 nM T36483 CD3O4Z 44339056 IC50 = 5000 nM T36483 CUP92F 44339060 IC50 = 12000 nM T36483 CO45AF 44339061 IC50 > 40000 nM T36483 CG4R7X 44339070 IC50 = 500 nM T36483 CSY5W6 44339157 IC50 = 1310 nM T36483 C3BM0F 44339173 IC50 = 130 nM T36483 C0W4UH 44354022 EC50 = 31000 nM T36483 CZ3P4T 44354052 EC50 = 800000 nM T36483 C4AFJ8 44354055 EC50 = 10 nM T36483 CB3Y0N 44354062 EC50 > 800000 nM T36483 C2IA5K 44354106 EC50 = 120 nM T36483 CX1B6H 44354107 EC50 = 40000 nM T36483 CC1H6G 44354108 EC50 = 130 nM T36483 C4C8FX 44354285 EC50 = 150 nM T36483 C2MVY1 44354323 EC50 = 30 nM T36483 C84VLR 44354387 EC50 = 600000 nM T36483 C4BY2H 44354460 EC50 = 260000 nM T36483 CL94CB 44403839 IC50 = 400 nM T36483 CGN3M7 44408615 IC50 = 730 nM T36483 CV14NJ 44408616 IC50 = 150 nM T36483 C48NRV 44408709 IC50 = 700 nM T36483 CV2FB8 44408711 IC50 = 390 nM T36483 CL8ET4 44408851 IC50 = 60 nM T36483 CGZ5L1 44408873 IC50 = 15 nM T36483 CPHR30 44408874 IC50 = 155 nM T36483 CJ1WK6 44409029 IC50 = 500 nM T36483 C10MZB 44409033 IC50 = 300 nM T36483 CWLA42 44409034 IC50 = 28 nM T36483 C5BN2E 44409039 IC50 = 2151 nM T36483 CFGH09 44409050 IC50 = 800 nM T36483 C8WJN0 44409057 IC50 = 25 nM T36483 C85SAC 44409062 IC50 = 500 nM T36483 C2ME6W 44409074 IC50 = 50 nM T36483 C7IBZ8 44409076 IC50 = 300 nM T36483 CO85YX 44409077 IC50 = 219 nM T36483 C3I2XK 44409082 IC50 = 125 nM T36483 CQ9ZP8 44409083 IC50 = 1250 nM T36483 C0AM4W 44409228 IC50 = 275 nM T36483 CCL1W8 44409232 IC50 = 30 nM T36483 CFI18T 44409248 IC50 = 50 nM T36483 CPM0H5 44409253 IC50 = 100 nM T36483 C49FKT 44409259 IC50 = 68 nM T36483 CK82DA 44409265 IC50 = 1000 nM T36483 C3E8ZK 44409278 IC50 = 290 nM T36483 C14SBI 44409289 IC50 = 800 nM T36483 C9V7SR 44416466 IC50 = 426 nM T36483 CGU2I4 44416487 IC50 = 7000 nM T36483 CT5AF6 44416541 IC50 = 1500 nM T36483 CAC6W5 44416542 IC50 = 200 nM T36483 CXO31W 44416562 IC50 = 150 nM T36483 CVQ20M 44416563 IC50 = 3500 nM T36483 CJB97L 44416567 IC50 = 623 nM T36483 CVD1L4 44416588 IC50 = 2000 nM T36483 CIEH73 44416634 IC50 = 7000 nM T36483 C16OSE 44416654 IC50 = 217 nM T36483 CB6K0L 44416672 IC50 = 8000 nM T36483 CIK31H 44416690 IC50 = 150 nM T36483 C2WUH0 44416691 IC50 = 62 nM T36483 C0DPY7 44416717 IC50 = 3750 nM T36483 CBD0K2 44416724 IC50 = 5000 nM T36483 CO40PE 44416740 IC50 = 74 nM T36483 CN3IR6 44418837 IC50 = 80 nM T36483 C73PLG 44418838 IC50 = 28 nM T36483 CIR8G5 44418839 IC50 = 72 nM T36483 CEV27S 44418840 IC50 = 829 nM T36483 C8G3KX 44418842 IC50 = 38.5 nM T36483 CD51EF 44418844 IC50 = 147 nM T36483 CH43LA 44418846 IC50 = 70 nM T36483 C3VI2T 44418847 IC50 = 1374 nM T36483 CF0KU1 44418848 IC50 = 97 nM T36483 C8H0DE 44418849 IC50 = 16.5 nM T36483 CBZ93Y 44418850 IC50 = 15 nM T36483 C9DOX5 44418854 IC50 = 28 nM T36483 COX93N 44418855 IC50 = 12 nM T36483 C5NRG9 44418858 IC50 = 11 nM T36483 CEH4F5 44428104 Ki = 4.3 nM T36483 CR2ZA7 44432691 IC50 = 3600 nM T36483 CPY1T2 44432692 IC50 = 350 nM T36483 CG8V5A 44432693 IC50 = 43 nM T36483 CR6PH9 44432704 IC50 = 130 nM T36483 CPCF39 44432705 IC50 = 285 nM T36483 CW51XH 44432706 IC50 = 263 nM T36483 CRT4L1 44432707 IC50 = 115 nM T36483 CPOM02 44432708 IC50 = 29 nM T36483 CG0Q7L 44432710 IC50 = 3300 nM T36483 CQK89F 44432711 IC50 = 12 nM T36483 C7KMN5 44432712 IC50 = 16 nM T36483 C1RVW9 44432713 IC50 = 36 nM T36483 CV5Z8K 44432714 IC50 = 11 nM T36483 C6VPH0 44432715 IC50 = 47 nM T36483 C70NXO 44432716 IC50 = 1320 nM T36483 CO9IN1 44432717 IC50 = 145 nM T36483 C9FB6J 44432718 IC50 = 22 nM T36483 COP92K 44432719 IC50 = 2144 nM T36483 C2N4DU 44432720 IC50 = 207 nM T36483 C42LFE 44432721 IC50 = 88 nM T36483 C6LU8S 44432756 IC50 = 440 nM T36483 CL1ON3 44432763 IC50 = 65 nM T36483 CG35DW 44432767 IC50 = 31.5 nM T36483 CFD86M 44432770 IC50 = 137.5 nM T36483 CQU32G 44432771 IC50 = 225 nM T36483 CMDL57 44432772 IC50 = 46.5 nM T36483 C5EK6H 44432773 IC50 = 10 nM T36483 C8E9BN 44432774 IC50 = 120 nM T36483 CPR7M9 44432775 IC50 = 29 nM T36483 CDV3F2 44432778 IC50 = 328 nM T36483 C8T3YF 44432779 IC50 = 13 nM T36483 C20FMS 44432783 IC50 = 15.5 nM T36483 CZS35O 44432786 IC50 = 330 nM T36483 C7PE6B 44432790 IC50 = 10 nM T36483 CC1V7G 44432791 IC50 = 20.5 nM T36483 CWHP50 44432795 IC50 = 63.5 nM T36483 CU36DS 44432798 IC50 = 14.5 nM T36483 C7XSD8 44432803 IC50 = 7 nM T36483 C2M6BU 44432806 IC50 = 85.5 nM T36483 CXZ5V1 44432814 IC50 = 7.5 nM T36483 C5QCT4 44432817 IC50 = 14.5 nM T36483 C8Y1ER 44432831 IC50 = 12000 nM T36483 C6MW3X 44432833 IC50 = 580 nM T36483 CL3E7S 44432836 IC50 = 90 nM T36483 CO0NA4 44432839 IC50 = 9170 nM T36483 C1RU9S 44432840 IC50 = 3139 nM T36483 C4N9BO 44432842 IC50 = 225 nM T36483 C4GPB7 44432843 IC50 = 12.5 nM T36483 C0PO8C 44584151 IC50 = 20000 nM T36483 C3ZGS2 44826171 EC50 = 1900 nM T36483 CE5Q1R 44826172 EC50 = 1900 nM T36483 CDXT67 49766539 IC50 = 520 nM T36483 C4AZ6G 49766546 IC50 = 2200 nM T36483 C1ER8F 50910530 IC50 = 3000 nM T36483 C3U5JP 50910534 IC50 = 520 nM T36483 CX5K9E 50910535 IC50 = 710 nM T36483 C29DEG 50910547 IC50 = 1290 nM T36483 CPYE39 50910548 IC50 = 3160 nM T36483 CE03PW 50910549 IC50 = 2640 nM T36483 C8N0ID 51003683 IC50 = 340 nM T36483 C0JNG8 52940892 Ki = 144 nM T36483 C35CDM 52940897 Ki = 337 nM T36483 C3FX0H 52942074 Ki = 240 nM T36483 CA42IG 52942093 Ki = 42 nM T36483 C9SET2 52946929 Ki = 250 nM T36483 CBC61R 52946957 Ki = 49 nM T36483 C3H4PS 52947767 Ki = 12 nM T36483 C8AQ3X 52948306 Ki = 75 nM T36483 C5EO4F 52949425 Ki = 61 nM T36483 CBJ6D3 52949514 Ki = 15 nM T36483 CVBF92 53245432 IC50 = 600 nM T36483 CH05IO 53245434 IC50 = 480 nM T36483 CUG2I9 53245435 IC50 = 390 nM T36483 C9AD3Q 53245451 IC50 = 380 nM T36483 C4G2IS 53245483 IC50 = 2280 nM T36483 CNJL95 56668146 IC50 > 100000 nM T36483 C7C6XG 56671606 IC50 = 3900 nM T36483 CQN67G 56949066 IC50 = 970 nM T36483 C8JZM0 57404483 IC50 = 8.1 nM T36483 CL08XW 57404484 IC50 = 4.6 nM T36483 C72MWG 57404504 IC50 = 6.4 nM T36483 C6I9BF 57892463 IC50 = 31.62 nM T36483 CN9C2H 58187662 Ki = 35 nM T36483 C5UYB6 58939091 Ki = 14 nM T36483 C82PJI 59016133 Ki = 8 nM T36483 C4D0OU 59016136 Ki = 20 nM T36483 CNK7S5 59016155 Ki = 19.5 nM T36483 CX7GJ3 59110442 IC50 = 28 nM T36483 CQ70WI 59110450 IC50 = 22 nM T36483 CTE5W4 59110452 IC50 = 13 nM T36483 CNFW51 59110475 IC50 = 25 nM T36483 C1WUI8 59110479 IC50 = 33 nM T36483 CW5IM9 59110483 IC50 = 27 nM T36483 C2UTJ9 60003490 IC50 = 24 nM T36483 C8R2GE 70681077 IC50 = 8.8 nM T36483 CNV1K4 70683199 IC50 = 20 nM T36483 CH1QU9 70683205 IC50 = 8.6 nM T36483 CH1YU2 70683207 IC50 = 64 nM T36483 CRNG89 70685279 IC50 = 20 nM T36483 CP0K5B 70685280 IC50 = 35 nM T36483 CDHT12 70685282 IC50 = 49 nM T36483 CP67OG 70687423 IC50 = 225 nM T36483 CS7AR2 70687424 IC50 = 21 nM T36483 CE30ZT 70687425 IC50 = 513 nM T36483 CL78ZH 70687427 IC50 = 18 nM T36483 CIH25U 70693686 IC50 = 45 nM T36483 CN16RX 70695800 IC50 = 451 nM T36483 CTX46Q 71770951 IC50 > 30000 nM T36483 CK6EG1 72547305 IC50 = 1100 nM T36483 C1DEP5 72547306 IC50 = 220 nM T36483 CP6WG0 72547307 IC50 = 1.3 nM T36483 CU7L1V 72547308 IC50 = 210 nM T36483 CER7U3 72547551 IC50 = 7.2 nM T36483 CJLV20 72547552 IC50 = 26 nM T36483 CM5K7P 72547553 IC50 = 6 nM T36483 C5K1HR 72547554 IC50 = 50 nM T36483 CR89KZ 72547555 IC50 = 43 nM T36483 CEX78Z 72547556 IC50 = 2.7 nM T36483 CK87FB 73347045 EC50 = 110000 nM T36483 CJ9AL1 76285459 Ki = 5 nM T36483 C34FDW 76309941 IC50 = 2100 nM T36483 CY1TQ8 76309942 IC50 = 2000 nM T36483 C2XWP7 76310287 Ki = 239 nM T36483 C5MU6P 76310288 Ki = 12 nM T36483 CH4PG5 76310289 Ki = 24 nM T36483 C1R3JF 76310290 Ki = 25 nM T36483 CVL9M1 76313663 IC50 = 120 nM T36483 CQ4HY7 76313664 IC50 = 67 nM T36483 COMF86 76317165 IC50 = 280 nM T36483 CJO03F 76317166 IC50 = 360 nM T36483 C4OQ6V 76317512 Ki = 31 nM T36483 C3JBO9 76317513 Ki = 384 nM T36483 CQ54MK 76317514 Ki = 12.5 nM T36483 CU76WL 76324547 IC50 = 230 nM T36483 CH0DZ8 76324857 Ki = 13.5 nM T36483 CY4GX2 76328106 IC50 = 53 nM T36483 CV3BH9 76328107 IC50 = 33 nM T36483 COU9Q7 76328415 Ki = 14.5 nM T36483 C3SHJ4 76331783 IC50 = 7800 nM T36483 CCY2S9 76331784 IC50 = 230 nM T36483 C5HI1X 76332095 Ki = 98 nM T36483 CRW4D8 76332096 Ki = 32 nM T36483 C3U5BQ 76332097 Ki = 15 nM T36483 C3AFJ4 76335370 IC50 = 470 nM T36483 CN5AD3 76335371 IC50 = 980 nM T36483 CS43RT 76335372 IC50 = 67 nM T36483 CH01JU 76335711 Ki = 140 nM T36483 CU24GV 76335712 Ki = 180 nM T36483 C6Q7CA 76335713 Ki = 12.9 nM T36483 CIV74S 86302495 Ki = 5.1 nM T36483 CJ64EC 86302515 Ki = 8.9 nM T36483 C96WJL 90644636 Ki = 21 nM T36483 CIZK39 90644637 Ki = 15.5 nM T36483 C2Y9BG 90644638 Ki = 267 nM T36483 CK65RM 90644639 Ki = 26.5 nM T36483 COJ1Z8 90644640 Ki = 28 nM T36483 CB2F7G 90644641 Ki = 43 nM T36483 CRS60E 90644642 Ki = 25 nM T36483 CEWU84 90644643 Ki = 232 nM T36483 CN5YF3 90644644 Ki = 31.5 nM T36483 CML79P 90644645 Ki = 392 nM T36483 C1LHG8 90663288 IC50 = 23 nM T36483 CIZL42 90663289 IC50 = 270 nM T36483 C7RCD2 90663290 IC50 = 20 nM T36483 CR0G1L 90663291 IC50 = 46 nM T36483 CHZ9C1 90663292 IC50 = 40 nM T36483 CD9O6M 90663293 IC50 = 21.9 nM T36483 CP3BC7 90663294 IC50 = 250 nM T36483 CR7TN4 90663295 IC50 = 17 nM T36483 C0B1OR 90663296 IC50 = 870 nM T36483 CR40WY 90663297 IC50 = 32000 nM T36483 CUT54F 90663298 IC50 = 41 nM T36483 C2RVY5 90663299 IC50 = 500 nM T36483 C3S7PT 90663300 IC50 = 370 nM T36483 C37WFI 90663301 IC50 = 470 nM T36483 C3Z2BI 90663302 IC50 = 85000 nM T36483 CE5K8S 90663303 IC50 = 1000 nM T36483 CMB35Q 90663304 IC50 = 110 nM T36483 C2AIV3 90663305 IC50 = 64000 nM T36483 C8MBP2 90663306 IC50 = 34 nM T36483 CNP70T 90663307 IC50 = 99 nM T36483 CJB2G3 90663308 IC50 = 7600 nM T36483 CW5G6D 90663309 IC50 = 1180 nM T36483 CZW03D 90663310 IC50 = 320 nM T36483 CP37FV 90663311 IC50 = 28 nM T36483 CBRO21 90663312 IC50 = 200 nM T36483 C4UHS1 90663313 IC50 = 4 nM T36483 CUF1J9 90663314 IC50 = 16.6 nM T36483 C4V7TC 90663315 IC50 = 6.6 nM T36483 C43MOB 90663316 IC50 = 25 nM T36483 CSHL28 90663317 IC50 = 340 nM T36483 CV65ED 90663318 IC50 = 9 nM T36483 CEG37C 90663319 IC50 = 19 nM T36483 CR7Y3D 90663320 IC50 = 28 nM T36483 C0PHI2 90663321 IC50 = 130 nM T36483 CH7N5Y 90663322 IC50 = 500 nM T36483 C6X8QP 90663323 IC50 > 100000 nM T36483 C6T1GU 90663324 IC50 = 3440 nM T36483 CT15QB 90663325 IC50 = 42 nM T36483 CE2N9R 90663326 IC50 = 93 nM T36483 C8H3EK 90663327 IC50 = 39 nM T36483 CE7L2P 90663328 IC50 = 7.5 nM T36483 CI13QM 90663329 IC50 = 950 nM T36483 C1O8PU 90663330 IC50 = 40000 nM T36483 CMEZ14 90663331 IC50 = 680 nM T36483 CI8EF5 90663332 IC50 = 4670 nM T36483 C4W1ZL 90663333 IC50 = 3930 nM T36483 C4CN1K 90663334 IC50 = 110 nM T36483 C4S7IR 90663335 IC50 = 61 nM T36483 C2TI1O 90663336 IC50 = 630 nM T36483 CYXO35 90663337 IC50 = 21700 nM T36483 CEH10F 90663338 IC50 = 880 nM T36483 CMXW50 90663339 IC50 = 2320 nM T36483 CQO2T5 90663340 IC50 = 310 nM T36483 CL0MR2 90663341 IC50 = 350 nM T36483 CC9E6Y 90663342 IC50 = 9900 nM T36483 CE28ZM 90663343 IC50 = 1630 nM T36483 C0K6HW 90663344 IC50 = 260 nM T36483 CM6CH8 90663345 IC50 = 170 nM T36483 C8AD0J 90663346 IC50 = 24 nM T36483 CB1R3C 90663347 EC50 = 67000 nM T36483 CVZ0Q7 90663348 IC50 = 246 nM T36483 C9U6PF 90663350 IC50 = 340 nM T36483 CP8AT5 90663351 IC50 = 7550 nM T36483 CTV12X 90663352 IC50 = 1120 nM T36483 C2Y3KZ 90663353 IC50 = 4710 nM T36483 C5QR4T 90663354 IC50 = 560 nM T36483 C7XQS8 90663355 IC50 = 24 nM T36483 C1IEB4 90663356 IC50 = 2730 nM T36483 CH0I1E 90663358 IC50 = 66700 nM T36483 C8T4KN 90663359 EC50 = 270 nM T36483 CJ2PY5 90663360 IC50 = 220 nM T36483 COS70P 90663563 IC50 = 1190 nM T36483 C50FEG 90663732 IC50 = 19 nM T36483 CE5V6U 117072551 IC50 = 1700 nM T36483 CNS91H 117909194 IC50 = 28.7 nM T36483 CR07ZG 117909666 IC50 = 4.22 nM T36483 C6N8SM 117909768 IC50 = 3.08 nM T36483 C4OVE8 118714099 IC50 > 10000 nM T36483 CC4LA1 118953461 IC50 > 30000 nM T36483 C13EIL 118967091 IC50 > 30000 nM T36483 C5OKW0 118967130 IC50 > 30000 nM T36483 CE3CN6 118971057 IC50 > 30000 nM T36483 CT4RP7 118971061 IC50 > 30000 nM T36483 CD7AN0 118971371 IC50 > 30000 nM T36483 CQD4P5 121469330 IC50 = 0.99 nM T36483 C5Y7VT 125407509 IC50 > 30000 nM T36483 CW03MF 126961335 IC50 > 50000 nM T36483 CDR2I3 127049415 IC50 = 100 nM T36483 C2UJ0N 127050656 IC50 = 60 nM T36483 C2V5EI 127050657 IC50 = 10 nM T36483 CYBO14 127050658 IC50 = 50 nM T36483 CK7U9R 127050672 IC50 = 130 nM T36483 CF6M7Y 127050673 IC50 = 30 nM T36483 CE80LC 127050934 IC50 = 30 nM T36483 C2ENH5 127050971 IC50 = 40 nM T36483 C31MDQ 127051545 IC50 = 60 nM T36483 C9YT7Q 127051546 IC50 = 70 nM T36483 CD2LB1 127051547 IC50 = 80 nM T36483 CUO21P 134137936 IC50 > 10000 nM T36483 CP12TG 136209460 IC50 ~ 90000 nM T36483 CU67ND 137631870 IC50 = 9500 nM T36483 CK38CP 137632009 IC50 = 3000 nM T36483 C7XYM6 137632193 IC50 = 12000 nM T36483 C6KND9 137632824 IC50 > 100000 nM T36483 C21SWT 137632975 IC50 = 8700 nM T36483 C61BPT 137633371 IC50 = 32000 nM T36483 CE3WA8 137634922 IC50 > 100000 nM T36483 CPY6H8 137635753 IC50 > 100000 nM T36483 C3TI7G 137637794 IC50 = 14000 nM T36483 CGF2X7 137638549 IC50 = 19000 nM T36483 CZ0T3W 137638930 IC50 > 100000 nM T36483 C50LQS 137639606 IC50 = 20000 nM T36483 C5R9AQ 137641036 IC50 > 100000 nM T36483 CA60IO 137641321 IC50 > 100000 nM T36483 CCUE34 137642658 IC50 > 100000 nM T36483 C4WEG7 137643571 IC50 > 100000 nM T36483 C1F4YR 137644873 IC50 = 55000 nM T36483 CSP79Y 137645208 IC50 = 1500 nM T36483 C2VK3O 137645447 IC50 > 100000 nM T36483 CH6JZ5 137647264 IC50 = 23000 nM T36483 CTS03I 137648050 IC50 > 100000 nM T36483 CO6ZT4 137649563 IC50 = 7000 nM T36483 C14CLO 137649807 IC50 > 100000 nM T36483 CY7VL5 137651100 IC50 > 100000 nM T36483 CYU8K1 137651696 IC50 > 100000 nM T36483 C8V7XZ 137652024 IC50 = 87000 nM T36483 CDA2K4 137652763 IC50 > 100000 nM T36483 CCZY19 137653180 IC50 = 8100 nM T36483 C5YMI9 137653221 IC50 > 100000 nM T36483 CR6TX5 137653750 IC50 = 14000 nM T36483 C8B4DQ 137654003 IC50 > 100000 nM T36483 C91MIW 137654212 IC50 = 21000 nM T36483 C2E9JM 137654568 IC50 = 29000 nM T36483 CF4S7T 137654736 IC50 > 100000 nM T36483 CM2HE5 137655130 IC50 = 10000 nM T36483 CG07RC 137656188 IC50 > 100000 nM T36483 C8AZ7S 137657212 IC50 > 100000 nM T36483 CZP1K2 137657357 IC50 > 100000 nM T36483 CCX5T7 137658131 IC50 > 100000 nM T36483 C10QES 137658217 IC50 > 100000 nM T36483 CP1QS4 137659611 IC50 = 9100 nM T36483 CIW4T5 137660576 IC50 > 100000 nM T36483 C0YHD2 137661486 IC50 = 650 nM T36483 CCU4J5 137661676 IC50 = 17000 nM T36483 CB3HI7 145967675 IC50 > 10000 nM T36483 CF4V1J 145968568 IC50 = 19.95 nM T36483 CW70RF 145970191 IC50 = 290 nM T36483 CTEJ01 145971090 IC50 = 100000 nM T36483 CKVH05 154688304 IC50 = 398.11 nM T36483 COY7A6 154688307 IC50 = 370 nM T36483 CPX6Q0 155512671 IC50 = 40 nM T36483 CNY3Z8 155519325 IC50 = 398.11 nM T36483 C5CJF2 155526775 IC50 = 10 nM T36483 CQN9L7 155536026 IC50 = 30 nM T36483 CFDM94 155549751 IC50 = 140 nM T36483 CN4WT6 155564785 IC50 = 130 nM T36483 CHY4T0 44306337 IC50 = 150 nM T36483 C2DVJ6 44306349 IC50 = 6100 nM T36483 D00KRL 10132921 IC50 > 10000 nM T36483 D0BV3B 16214871 Ki = 19 nM T36483 D0I2VE 9853822 IC50 = 440 nM T36483 D0QK2E 9804049 Ki = 2.7 nM T12797 D02OZK 11404337 EC50 = 600 nM T12797 D03TTE 135513044 Ki = 1470 nM T12797 D0B1UL 136002683 Ki = 460 nM T12797 D0CR9A 136183441 Ki = 930 nM T12797 D0L8WH 11228183 Ki > 20000 nM T12797 CVD64E 36941 Ki > 100000 nM T12797 CB6E4Y 720528 IC50 = 2100 nM T12797 C2I9CA 779754 IC50 = 300 nM T12797 CBO6D7 1074953 IC50 = 450 nM T12797 C87OXF 1180669 IC50 > 50000 nM T12797 C4Y5CT 1180675 IC50 > 50000 nM T12797 COW3Q9 1180676 IC50 = 600 nM T12797 CGAM30 1582605 Ki = 6140 nM T12797 C07WVL 1654287 IC50 = 4100 nM T12797 CW2UC7 1664226 IC50 = 2400 nM T12797 CJ5FD3 1673604 IC50 = 2600 nM T12797 CN96HL 2268888 IC50 > 10000 nM T12797 C4LM7K 16654625 IC50 > 50000 nM T12797 CMO71D 16654638 IC50 = 8700 nM T12797 C3S2BO 16654639 IC50 = 11100 nM T12797 C8AYR4 16654640 IC50 = 1000 nM T12797 CG8IE3 16654650 IC50 > 10000 nM T12797 CVWX79 16654652 IC50 = 400 nM T12797 C8INE7 16654653 IC50 = 600 nM T12797 CLT31W 16654654 IC50 = 1100 nM T12797 C3K7AN 16654655 IC50 = 690 nM T12797 CR93CM 16654656 IC50 = 1700 nM T12797 CY3D6Z 16654661 IC50 = 2100 nM T12797 CL3BH9 16654662 IC50 = 1300 nM T12797 C6NH0G 16654665 IC50 > 10000 nM T12797 CTZS48 16654669 IC50 = 620 nM T12797 CKX1T5 16654670 IC50 = 6200 nM T12797 CH4C1D 16654672 IC50 = 8300 nM T12797 CC76JQ 16654674 IC50 = 10500 nM T12797 C8EIO1 16654677 IC50 = 1200 nM T12797 CD6YT8 16654679 IC50 = 2000 nM T12797 CX1JA7 16654730 IC50 = 10800 nM T12797 CY5UW9 16654772 IC50 = 3900 nM T12797 CXO2S9 44191694 IC50 = 550 nM T12797 CHT92S 44191696 IC50 = 1300 nM T12797 C83UCJ 44191750 IC50 = 670 nM T12797 CMS39X 44191815 IC50 = 5000 nM T12797 C0J3RT 44192144 IC50 = 400 nM T12797 C97RQU 44192145 IC50 = 2000 nM T12797 C57VCY 44224066 IC50 = 730 nM T12797 CH2E4R 44609307 Ki = 2340 nM T12797 CG2NH7 46236925 IC50 = 590 nM T12797 C78NZA 46236926 IC50 = 770 nM T12797 CUB3N9 52943093 IC50 = 29000 nM T12797 C8C7FS 71451698 EC50 = 25500 nM T12797 CJA8N4 71455243 EC50 = 8200 nM T12797 COH24E 71455246 EC50 = 17800 nM T12797 CVC5F8 71455247 EC50 = 21500 nM T12797 CUG8N7 71462421 EC50 = 24000 nM T12797 CP3Y2O 71548702 Ki = 1110 nM T12797 CS02CG 71549001 Ki = 3180 nM T12797 C37AJW 71549412 Ki = 17260 nM T12797 C3C7QO 86765310 Ki = 3360 nM T12797 C5W2EA 118734957 Ki > 660 nM T12797 C76SBJ 122622651 Ki = 3700 nM T12797 CR19KU 122622656 Ki = 900 nM T12797 CFR02M 122622711 Ki = 170 nM T12797 CY2J6L 122622713 Ki = 1700 nM T12797 C0AYP2 122622799 Ki = 3000 nM T12797 CE4MG7 122622800 Ki = 1600 nM T12797 C0KP5W 122622803 Ki = 810 nM T12797 CIH4M1 122622824 Ki = 3800 nM T12797 CBFO10 122622827 Ki = 760 nM T12797 C6JOM4 122622922 Ki = 3400 nM T12797 CY9OL2 122623097 Ki = 570 nM T12797 C59MST 122623143 Ki = 150 nM T12797 C9YU0H 122623413 Ki = 1000 nM T12797 CJ5P7N 122623425 Ki = 4600 nM T12797 C1R4UJ 122633925 Ki = 1100 nM T12797 C26QUL 122633937 Ki = 14800 nM T12797 CB4J7Z 134130355 Ki < 0.1 nM T12797 CC9OV6 134131166 Ki = 32 nM T12797 C9MFV2 136002682 Ki = 870 nM T12797 C6FY0E 136002684 Ki = 470 nM T12797 C9RD0X 136032611 Ki = 470 nM T12797 CC09EN 136183442 Ki = 9330 nM T12797 CYJD84 136183443 Ki = 3530 nM T12797 CF8HV7 136183446 IC50 = 122 nM T12797 CCVP03 145994390 Ki = 100 nM T12797 C1R8MS 155522698 Ki = 390 nM T12797 C5L4DX 155523696 Ki = 250 nM T12797 CQN1B8 155524663 Ki > 70000 nM T12797 CB89NA 155528220 Ki > 70000 nM T12797 CU9CX1 155529604 Ki = 280 nM T12797 CUS28M 155542793 Ki = 84 nM T12797 CVBF96 155545115 Ki = 10600 nM T12797 CL4HF7 155547093 Ki = 100 nM T12797 C4KGR1 155556368 Ki = 62000 nM T12797 D05RDP 992586 Ki = 5330 nM T12797 D0V7PX 454878 IC50 > 10000 nM T60897 D05EAM 4735 IC50 = 300 nM T60897 CPQ3D4 1202786 IC50 = 188000 nM T60897 C9C0OM 2714312 IC50 = 31400 nM T60897 C85XHT 7509342 IC50 = 69400 nM T60897 CYOS08 8119828 IC50 = 104000 nM T60897 C3NIY8 16456878 IC50 = 188000 nM T60897 CBXR07 45840460 IC50 = 149800 nM T60897 CEL91T 56923561 IC50 = 109200 nM T60897 C2IT1Z 91383855 IC50 = 277 nM T60897 CU3RP8 124141953 IC50 = 52 nM T71266 D01NEC 51042438 IC50 = 1.3 nM T71266 D01ZAQ 25227436 IC50 = 8 nM T71266 D02NNV 3038525 IC50 > 5000 nM T71266 D02ZQS 16095342 IC50 = 1510 nM T71266 D09IYM 24905401 IC50 = 50 nM T71266 D0E3TC 44259 IC50 = 5 nM T71266 D0I4TH 24788740 IC50 = 8 nM T71266 D0MS3Z 16725726 IC50 = 9 nM T71266 D0W3RW 24964624 IC50 = 65 nM T71266 D03BNU 59604787 IC50 > 10000 nM T71266 D0T3ME 156422 IC50 > 30000 nM T71266 CWN6P7 5702541 IC50 = 662 nM T71266 CG17TN 6914611 IC50 = 35 nM T71266 C7E2QK 6914613 IC50 = 354 nM T71266 CIAL53 9819282 IC50 > 50000 nM T71266 C41QWA 9857146 IC50 > 10000 nM T71266 CI0AW6 9871034 IC50 = 27000 nM T71266 CS5KX9 9938299 IC50 > 10000 nM T71266 CJX43Z 10055074 IC50 = 7400 nM T71266 C7TA9J 10113568 IC50 = 17378.01 nM T71266 CEV18B 10128689 IC50 > 50000 nM T71266 C7PK4U 10152003 IC50 > 50000 nM T71266 C4FUG5 10152760 IC50 > 50000 nM T71266 CMO32F 10152761 IC50 = 21870 nM T71266 CMR17F 10174144 IC50 > 50000 nM T71266 CLP79V 10196532 IC50 = 3200 nM T71266 CI8MW4 10216627 IC50 = 73 nM T71266 C0O8FI 10217663 IC50 = 33100 nM T71266 CY6MJ3 10218178 IC50 > 50000 nM T71266 C8V6RI 10240275 IC50 = 7200 nM T71266 CD3W6Y 10289038 IC50 > 50000 nM T71266 C2LP9A 10289671 IC50 = 2400 nM T71266 C4MOF8 10312133 IC50 = 1613 nM T71266 CAK9U4 10415819 IC50 = 1228 nM T71266 C2ON6C 11246455 IC50 = 179 nM T71266 C49NET 11256399 IC50 = 380 nM T71266 C6C3JX 11281930 IC50 > 10000 nM T71266 CBOP58 11293798 Ki = 4890 nM T71266 C5ACQ0 11348837 IC50 = 3000 nM T71266 C26BZX 11362471 Ki > 10000 nM T71266 CWXB93 11397177 Ki > 10000 nM T71266 CVG3L6 11502369 IC50 = 990 nM T71266 CK2WT3 11510023 IC50 = 1500 nM T71266 CL2I5O 11517293 IC50 = 19000 nM T71266 C05MTD 11522988 IC50 = 4700 nM T71266 C8IHX9 11538014 IC50 = 5400 nM T71266 CTG83F 11539329 Ki > 9500 nM T71266 CBIY48 11544625 IC50 = 5000 nM T71266 C2QDA9 11559783 IC50 = 2900 nM T71266 CACS26 11561968 Ki > 2000 nM T71266 C9THO1 11567357 IC50 = 610 nM T71266 CW4Z9E 11575743 IC50 = 280 nM T71266 CMIL86 11590363 Ki > 9500 nM T71266 C4Z1YB 11610430 IC50 = 1100 nM T71266 C9T6SC 11640926 Ki > 9500 nM T71266 C7XEV0 11664023 IC50 = 2474 nM T71266 CJB19K 11667833 IC50 = 18000 nM T71266 C0V7SU 11675388 IC50 = 57 nM T71266 CU0E8O 11690457 Ki > 10000 nM T71266 CDF53M 11718648 IC50 = 2600 nM T71266 C9A6KM 11857236 IC50 = 3 nM T71266 C39VTW 11959283 IC50 = 70 nM T71266 C36HDX 11959286 IC50 = 30 nM T71266 CO0A4K 11959314 IC50 = 1 nM T71266 C12CRJ 11959377 IC50 = 22 nM T71266 C1WDQ0 11959682 IC50 = 49 nM T71266 CMW89V 11959683 IC50 = 17 nM T71266 C7N6CQ 15604547 IC50 = 76 nM T71266 CFPW41 16007116 Ki > 9500 nM T71266 CZK8V6 16043304 IC50 = 2.6 nM T71266 C9TU1O 16046126 IC50 > 1000 nM T71266 C7Z4LV 16095343 IC50 = 1290 nM T71266 C54YXC 16121514 IC50 = 72.44 nM T71266 CJXU82 21103111 IC50 > 50000 nM T71266 CF9YE6 21103119 IC50 > 50000 nM T71266 C5AR9M 21103197 IC50 > 50000 nM T71266 CN1O7X 23647016 IC50 > 50000 nM T71266 CJ3EO0 23647017 IC50 = 3973 nM T71266 CH14KD 23647018 IC50 > 50000 nM T71266 CQ5Z0J 23647019 IC50 > 50000 nM T71266 C2JTA3 23647573 IC50 = 39 nM T71266 C7YG1N 24759534 IC50 > 100000 nM T71266 CW3JR8 24783593 IC50 = 10 nM T71266 C05MQY 24783594 IC50 = 23 nM T71266 C93TIM 24786152 IC50 = 5 nM T71266 CSY9Z6 24788164 IC50 = 10 nM T71266 CFR62V 24788432 IC50 = 5 nM T71266 C2JNI3 24788623 IC50 = 13 nM T71266 CMR7F1 24788739 IC50 = 5 nM T71266 CY1ZS7 24803305 IC50 = 2 nM T71266 C2ANO6 24804134 IC50 = 3 nM T71266 CSH8A5 24804780 IC50 = 3 nM T71266 CUTH13 24805273 IC50 = 20 nM T71266 CA9F3Y 25023714 IC50 = 398 nM T71266 C8Z4PI 25023715 IC50 = 1410 nM T71266 CV96QX 25023716 IC50 = 1290 nM T71266 C5INV4 25023717 IC50 = 1549 nM T71266 CPOH02 25023718 IC50 = 3020 nM T71266 C6F7RD 25023719 IC50 = 2290 nM T71266 C1JEU6 25023729 IC50 = 69 nM T71266 CR8JP7 25023735 IC50 = 9 nM T71266 C4W7LY 25023736 IC50 = 16 nM T71266 COV3Q4 25061501 IC50 = 12 nM T71266 C8NR9H 25170562 IC50 = 5 nM T71266 CS9LC3 25170563 IC50 = 12 nM T71266 CN8YZ4 25170991 IC50 = 26 nM T71266 CSY93F 25190765 IC50 > 1000000 nM T71266 C0BCX6 25190766 IC50 = 1610 nM T71266 C19TVC 25190767 IC50 = 774 nM T71266 CK9V3Y 25190768 IC50 = 56.6 nM T71266 CD7S6Q 25190770 IC50 = 3750 nM T71266 C3HU6A 25190771 IC50 = 2.38 nM T71266 CHN5O0 25190977 IC50 = 2 nM T71266 COWB90 25221040 IC50 = 6 nM T71266 CC25TV 25222706 IC50 = 3 nM T71266 C1IG7E 25243798 IC50 > 10000 nM T71266 CH65JV 25243799 IC50 > 10000 nM T71266 CBQO98 42602095 IC50 = 30 nM T71266 CJ61SE 42602096 IC50 = 15 nM T71266 CI42XG 42602097 IC50 = 24 nM T71266 CD2AH4 42602175 IC50 = 22 nM T71266 CSWA85 42602176 IC50 = 40 nM T71266 C1LUN4 42602178 IC50 = 7 nM T71266 C8O3EA 42602260 IC50 = 15 nM T71266 C93NKL 42602264 IC50 = 4 nM T71266 C5OHU9 44414317 IC50 = 5200 nM T71266 CBO18Y 44414320 IC50 = 660 nM T71266 CWD30R 44414422 IC50 = 240 nM T71266 C25ZRP 44414445 IC50 > 25000 nM T71266 CW4HT5 44414446 IC50 > 25000 nM T71266 CCH43E 44414447 IC50 = 11 nM T71266 C4FI1S 44414467 IC50 > 25000 nM T71266 C2CE5X 44414470 IC50 = 27 nM T71266 CI2G5K 44414471 IC50 = 1300 nM T71266 C93QFH 44414472 IC50 = 7000 nM T71266 CTDY95 44414507 IC50 = 1000 nM T71266 CY58PE 44414508 IC50 > 25000 nM T71266 C91ZIP 44414529 IC50 = 2800 nM T71266 CI26HQ 44414530 IC50 = 820 nM T71266 CIMY48 44414553 IC50 = 2400 nM T71266 C3JHE6 44414577 IC50 > 25000 nM T71266 C0E4CL 44414579 IC50 = 4.8 nM T71266 C1FU3D 44414608 IC50 > 25000 nM T71266 C6R9AN 44414634 IC50 = 2300 nM T71266 CQB9Z0 44414635 IC50 > 25000 nM T71266 CYX64I 44414652 IC50 = 2100 nM T71266 CC21KN 44414653 IC50 = 7400 nM T71266 CQ93OC 44414655 IC50 > 25000 nM T71266 COP8A3 44449880 IC50 = 1900 nM T71266 CDEJ84 44450004 IC50 = 11280 nM T71266 C8OG1V 44517709 IC50 = 4000 nM T71266 C0DJS1 44591843 IC50 = 2 nM T71266 CX52YW 44591844 IC50 = 1 nM T71266 C1LS6V 44591845 IC50 = 3 nM T71266 CSZ5R9 44592438 IC50 = 40 nM T71266 CTS95L 44592502 IC50 = 2 nM T71266 CSKZ16 44592503 IC50 = 2 nM T71266 COY57J 44592504 IC50 = 2 nM T71266 C3CDV8 44592505 IC50 = 2 nM T71266 CAZE46 46175126 IC50 = 270 nM T71266 CQ5SD4 46190876 IC50 = 10 nM T71266 CY3HW5 46224684 IC50 = 1100 nM T71266 CB5H9C 46225574 IC50 = 15 nM T71266 C8M1DT 46225589 IC50 = 1 nM T71266 C60XUQ 46226079 IC50 = 1 nM T71266 C5PCH8 46226080 IC50 = 2 nM T71266 C6UD1Y 46226095 IC50 = 19 nM T71266 C7IF4T 46226096 IC50 = 10 nM T71266 CUDZ46 46226135 IC50 = 500 nM T71266 C0P4CT 46226136 IC50 = 2 nM T71266 CPH49S 46226137 IC50 = 1 nM T71266 CM5X8B 46226156 IC50 = 1 nM T71266 CLS29B 46872626 IC50 > 10000 nM T71266 C3HG7B 46882134 IC50 = 900 nM T71266 CTSE94 46882135 IC50 = 4600 nM T71266 CSY9H1 46882136 IC50 = 27000 nM T71266 CO16JL 46882137 IC50 = 12 nM T71266 CJEM76 46882138 IC50 = 42 nM T71266 CRZ91X 46882835 IC50 = 360000 nM T71266 CS0V9G 46882836 IC50 = 28000 nM T71266 CU8WX3 46882837 IC50 = 900000 nM T71266 C2O8RZ 46886323 IC50 > 1000 nM T71266 C70BLN 46886550 IC50 = 65 nM T71266 CCV96R 46886665 IC50 = 43 nM T71266 CC1Y0M 52941299 IC50 = 5769 nM T71266 CDT94U 52941495 IC50 = 2056 nM T71266 C9UF6K 52941555 IC50 = 485 nM T71266 CYM80Q 52942489 IC50 = 13916 nM T71266 CS09YT 52942516 IC50 = 6073 nM T71266 CQ08WT 52942668 IC50 = 1122 nM T71266 CHW04J 52943916 IC50 = 754 nM T71266 CY8BV4 52944892 IC50 = 746 nM T71266 CEM95A 52946401 IC50 = 6079 nM T71266 CKE3C7 52946402 IC50 = 1464 nM T71266 C3Q4CU 52947490 IC50 = 8410 nM T71266 CR9E1Z 52947590 IC50 = 25110 nM T71266 CE81HA 52950003 IC50 = 363 nM T71266 C3TU8R 52950063 IC50 = 666 nM T71266 C7MC5G 52950205 IC50 = 2718 nM T71266 C8NA4L 53384644 IC50 > 30000 nM T71266 CPC5D2 56603995 IC50 = 40 nM T71266 CS7U9L 56965952 IC50 = 170 nM T71266 CQP7E0 57750290 IC50 = 18 nM T71266 CNBO65 57750312 IC50 = 30 nM T71266 C2F9DS 57750315 IC50 = 105 nM T71266 CZ08KN 57750321 IC50 = 36 nM T71266 CUY8T6 57750329 IC50 = 582 nM T71266 CK4W1L 57750342 IC50 = 10 nM T71266 CM5X9L 57750343 IC50 = 523 nM T71266 CBY5E4 57750369 IC50 = 15 nM T71266 CSI9Y4 57750382 IC50 = 270 nM T71266 C6GH7X 57750391 IC50 = 150 nM T71266 CL7CW0 57750402 IC50 = 100 nM T71266 CA4G5W 57750407 IC50 = 6 nM T71266 CM7XL6 57750408 IC50 = 16 nM T71266 CY4Z8R 57750418 IC50 = 176 nM T71266 C87LKR 58191080 IC50 = 3 nM T71266 CZPF92 58191081 IC50 = 2 nM T71266 CZA32V 58344912 IC50 = 22000 nM T71266 CPVF85 58344916 IC50 = 24000 nM T71266 CD3LX9 58344922 IC50 = 700 nM T71266 CS8ZY7 58344924 IC50 = 390 nM T71266 C89NVR 58344941 IC50 = 170 nM T71266 CYK74H 58344983 IC50 = 370 nM T71266 CRJ47B 58345005 IC50 = 71000 nM T71266 CIOV02 58345019 IC50 > 100000 nM T71266 CY62SG 58345029 IC50 = 660 nM T71266 CM5HE1 58345070 IC50 > 10000 nM T71266 CO18NP 58345151 IC50 = 390 nM T71266 CV61YJ 58345169 IC50 > 100000 nM T71266 CW6SC9 58345215 IC50 > 100000 nM T71266 CFLZ87 58345232 IC50 = 2500 nM T71266 CYBT41 58345302 IC50 = 660 nM T71266 C4PE7X 58345314 IC50 = 400 nM T71266 C8X3WB 58458198 IC50 = 4160 nM T71266 C20XPF 58458267 IC50 > 2000 nM T71266 CP85TJ 58458278 IC50 = 1 nM T71266 CT79LH 58458379 IC50 = 83 nM T71266 CXJ63M 59603829 IC50 > 100000 nM T71266 CQEU96 59603842 IC50 = 330 nM T71266 CPVD45 59670809 IC50 = 21 nM T71266 C32WHR 59670989 IC50 = 12 nM T71266 CDWQ04 59671004 IC50 = 28 nM T71266 C43HZT 59671085 IC50 = 73 nM T71266 C0BRA5 59671144 IC50 = 45 nM T71266 CEYW16 59671148 IC50 = 4 nM T71266 C50NWX 59671151 IC50 = 2 nM T71266 CZH4W5 59671179 IC50 = 7 nM T71266 C8FY0G 59671180 IC50 = 7 nM T71266 C1MR8Q 60097495 IC50 > 2500 nM T71266 CC3MB4 60155179 IC50 > 100000 nM T71266 C9QB8G 60155270 IC50 = 2600 nM T71266 CM6NF2 60155627 IC50 > 10000 nM T71266 C62SQG 60155628 IC50 = 86 nM T71266 COS39T 60155629 IC50 = 430 nM T71266 CV63UL 67240318 IC50 > 10000 nM T71266 CP8OI2 67304551 IC50 > 10000 nM T71266 CY76UR 67305743 IC50 = 8.1 nM T71266 C3UKG8 67312397 IC50 = 5.4 nM T71266 CM6TZ3 67312506 IC50 = 26 nM T71266 C5DGR9 69036886 IC50 = 10000 nM T71266 CS8UF1 70675988 IC50 = 5 nM T71266 C2W5BX 70675991 IC50 = 798 nM T71266 CUJA60 70676312 IC50 = 4 nM T71266 CRBW21 70676316 IC50 = 27 nM T71266 CGX49K 70676464 IC50 = 3 nM T71266 C5D1LV 70687790 IC50 = 9120.11 nM T71266 CKT60L 71455860 Ki > 9000 nM T71266 CQV96E 71583048 IC50 = 4260 nM T71266 CSPR52 71583049 IC50 = 8065 nM T71266 CNT5F3 71583050 IC50 = 756 nM T71266 CH7I0W 71583051 IC50 = 2893 nM T71266 CJ2T9E 76332983 IC50 > 10000 nM T71266 C1HW4B 89735655 IC50 = 2400 nM T71266 C8GZ2B 135449326 Ki = 1800 nM T71266 CC73PA 138911338 IC50 = 1.7 nM T71266 CSU93V 155077019 IC50 = 0.12 nM T71266 C2MD1Q 155513187 IC50 > 10000 nM T71266 CL5DR0 155525783 IC50 = 0.1 nM T71266 CHS21A 155553831 IC50 = 65 nM T71266 CG95WV 155563831 IC50 = 4 nM T71266 CEIW13 155566807 IC50 = 700 nM T71266 D00ERW 44444843 Ki = 7157 nM T71266 D00HVA 11624601 Ki > 9500 nM T71266 D05APZ 135398501 IC50 > 2119 nM T71266 D05JRA 25190769 IC50 = 14.6 nM T71266 D09FFE 449241 IC50 = 200 nM T71266 D0I1FJ 11393719 IC50 = 646 nM T71266 D0J3LR 11634725 Ki > 4000 nM T71266 D0L2WP 46225540 IC50 = 1 nM T71266 D0OX1T 10172943 IC50 = 51 nM T71266 D0Q3NG 11715520 Ki > 9500 nM T71266 D0S7IE 11658882 Ki > 9500 nM T99948 D0OK1S 117941742 IC50 = 146 nM T99948 D0WQ9X 117951478 IC50 = 18 nM T99948 C1RCQ7 117941376 IC50 = 110 nM T99948 C7BVK6 117941458 IC50 = 1010 nM T99948 C6AL2M 117941533 IC50 = 6 nM T99948 C03JDG 117941658 IC50 = 6 nM T99948 CG3T5I 117941713 IC50 = 6 nM T99948 CL56TV 117941821 IC50 = 6 nM T99948 CYH13Z 117941887 IC50 = 80 nM T99948 CD0QR5 118434635 IC50 = 1.4 nM T99948 C4N1MD 121452782 IC50 = 6 nM T99948 C7P6CO 131839624 IC50 = 2.25 nM T99948 C2X0IF 145992098 IC50 = 5.2 nM T99948 D02BZV 91663303 IC50 = 6 nM T66538 D09BVL 4552 IC50 = 5888.44 nM T66538 D0S6QR 214350 EC50 = 352 nM T66538 CY1Z5T 232768 IC50 = 15135.61 nM T66538 CZU3E2 459332 IC50 = 13489.63 nM T66538 CEH76V 483833 IC50 = 18620.87 nM T66538 C7VH5Q 483836 IC50 = 17378.01 nM T66538 C7X9HU 740278 IC50 = 11748.98 nM T66538 CD5ZH7 830720 IC50 = 30199.52 nM T66538 C1UWX0 837857 IC50 = 26915.35 nM T66538 CFZ4U5 839448 IC50 = 11220.18 nM T66538 C3E4FV 868972 IC50 = 12302.69 nM T66538 C10NVJ 1124061 IC50 = 30902.95 nM T66538 CDOR89 1234642 IC50 = 12589.25 nM T66538 CU2FW1 2798242 IC50 = 3090.3 nM T66538 CLS15O 2798243 IC50 = 3467.37 nM T66538 CXW6L7 2946791 IC50 = 691.83 nM T66538 CTD1P7 2953683 IC50 = 3090.3 nM T66538 CU4P0Z 3011444 IC50 = 30902.95 nM T66538 CB0NG4 3011445 IC50 = 15135.61 nM T66538 C2MTJ0 3011446 IC50 = 11748.98 nM T66538 C0D3AK 3491594 IC50 = 19498.45 nM T66538 CL82TS 3605484 IC50 = 2511.89 nM T66538 C7Q9TV 4050379 IC50 = 251.19 nM T66538 CND86W 5073804 IC50 = 9332.54 nM T66538 CPW4Y1 9815734 EC50 = 8120 nM T66538 CJGX96 9881289 EC50 = 5070 nM T66538 CLHQ23 9990728 IC50 = 17782.79 nM T66538 C0T8UE 10035337 EC50 = 5130 nM T66538 CAQW79 10038562 EC50 = 4430 nM T66538 C6BEY4 10064074 IC50 = 3.236 nM T66538 C0GQF7 10083014 EC50 = 3340 nM T66538 C2CGW9 10243969 IC50 = 144.54 nM T66538 CQ8G6K 10263172 EC50 = 3860 nM T66538 C05UVN 10263770 EC50 = 15100 nM T66538 CJY45S 10331385 IC50 = 112201.85 nM T66538 CI1P3F 10354434 EC50 = 6750 nM T66538 C9N3KR 10356396 IC50 = 2630.27 nM T66538 CDFW74 10398337 EC50 = 6940 nM T66538 CX1SL4 10444440 IC50 = 13803.84 nM T66538 CUO6A4 10469103 EC50 = 17000 nM T66538 CS0OM5 10515414 IC50 = 154881.66 nM T66538 CF5I6P 10634209 IC50 = 93325.43 nM T66538 C9HG2C 10660593 IC50 = 24547.09 nM T66538 CG8W9V 10709096 IC50 = 37153.52 nM T66538 CI4P9O 10729882 IC50 = 93325.43 nM T66538 CN9KY8 10778936 IC50 = 28183.83 nM T66538 CU0BP4 10800545 IC50 = 104712.85 nM T66538 C5JQ8A 10849039 IC50 = 18620.87 nM T66538 CL8IW0 10849172 IC50 = 54954.09 nM T66538 C56UXE 10903109 IC50 = 79432.82 nM T66538 CX7S5A 10967695 IC50 = 2454.71 nM T66538 C0DS8B 10968747 IC50 = 8709.64 nM T66538 C5YA6S 10969679 IC50 = 5888.44 nM T66538 C8GK5I 11000844 IC50 = 6918.31 nM T66538 C2G6LX 11042812 IC50 = 1548.82 nM T66538 C7TDS2 11065065 IC50 = 3019.95 nM T66538 C6U8KG 11108600 IC50 = 10964.78 nM T66538 COF9D1 11109578 IC50 = 2137.96 nM T66538 CA38LS 11254734 IC50 = 190.55 nM T66538 CZ7K3W 11335564 IC50 = 7762.47 nM T66538 CL01DC 11392406 IC50 = 645.65 nM T66538 CCV2U0 11437030 IC50 = 27.54 nM T66538 C1GZ8U 11471747 IC50 = 446.68 nM T66538 C7O3AF 11472034 IC50 = 371.54 nM T66538 C3BI1D 11536112 IC50 = 10232.93 nM T66538 CRP35C 11651603 IC50 = 13489.63 nM T66538 C59YUQ 11779066 IC50 = 27.54 nM T66538 CJ58MG 11782023 IC50 = 3311.31 nM T66538 COM63L 11818496 IC50 = 177.83 nM T66538 CFJ3I2 11820396 EC50 = 5860 nM T66538 C1MZQ9 11823359 IC50 = 54954.09 nM T66538 CR72ZX 15717694 IC50 = 1445.44 nM T66538 CM7J9B 16099761 IC50 = 4073.8 nM T66538 CX2MQ8 16099762 IC50 = 5248.07 nM T66538 CKS0L7 16099763 IC50 = 30199.52 nM T66538 CTHR97 16099764 IC50 = 11748.98 nM T66538 CD3Q8R 16099767 IC50 = 11220.18 nM T66538 C7LAE8 18103922 IC50 = 15848.93 nM T66538 C7CZD5 24285062 IC50 = 134.9 nM T66538 C7EI0Y 24285063 IC50 = 8128.31 nM T66538 C8PTB6 44570449 IC50 = 281.84 nM T66538 CK2G5D 136029155 EC50 = 13400 nM T08123 D0R0MW 5329102 IC50 = 28 nM T08123 D08ZPO 448043 IC50 = 244 nM T08123 D0E3TC 44259 IC50 = 1 nM T08123 D0H2HZ 60194098 IC50 = 3981.07 nM T08123 D0HY9S 73386890 IC50 = 48 nM T08123 CY13DC 360689 IC50 = 5760 nM T08123 CCX69G 580694 IC50 = 100 nM T08123 CD5NJ1 953496 IC50 = 520 nM T08123 C6XYA1 953540 IC50 = 4460 nM T08123 CCN24W 1563747 IC50 = 2000 nM T08123 C3GZ8M 2358577 IC50 = 10000 nM T08123 CA6F4S 2360386 IC50 = 10000 nM T08123 CR09XN 2410620 IC50 = 194 nM T08123 C38OMQ 2727431 IC50 = 173 nM T08123 C85TOM 2727432 IC50 = 50 nM T08123 CI6H0F 2727439 IC50 = 1555 nM T08123 C3T2PD 2820108 Ki = 234 nM T08123 CRH5G3 5723593 Ki = 740 nM T08123 C85LJF 6463365 IC50 = 15.85 nM T08123 C02UYV 6918633 Ki = 5464 nM T08123 C0FV5J 7190424 IC50 = 215 nM T08123 C6XW2C 7190426 IC50 = 187 nM T08123 CPD45M 8272290 IC50 = 12000 nM T08123 CQ53PX 9567224 IC50 = 4100 nM T08123 CC90FJ 9869737 IC50 = 4600 nM T08123 C0BDP2 10313195 Ki = 2702 nM T08123 CSHT79 11056377 Ki = 240 nM T08123 C14SYJ 11088637 Ki = 2793 nM T08123 CFH5T7 11099263 Ki = 137 nM T08123 CQ29JI 11120348 Ki = 156 nM T08123 CID08M 16798824 IC50 = 200 nM T08123 CI5ST3 17982588 IC50 = 204 nM T08123 C5QWZ2 18561027 IC50 = 167 nM T08123 C5JWI9 21184460 Ki = 94 nM T08123 CR85BP 21184514 Ki = 863 nM T08123 C0ZGI1 21184532 Ki = 993 nM T08123 C8PBY4 21184553 Ki = 5583 nM T08123 CW1Q9P 21184562 Ki = 454 nM T08123 C19NOL 22500220 IC50 = 1500 nM T08123 C7YG1N 24759534 IC50 = 14 nM T08123 C7A5ET 24772735 Ki = 13 nM T08123 CJR3M7 25014542 IC50 = 15 nM T08123 CNQ9G5 25218180 IC50 = 46 nM T08123 C29RMK 36982503 IC50 = 12.59 nM T08123 CBY14D 39378356 IC50 = 48 nM T08123 CMI4D7 43668876 IC50 = 103 nM T08123 C8IHL7 44252884 IC50 = 1.3 nM T08123 C4X5CN 44444551 IC50 = 781 nM T08123 C7W5DZ 45790300 Ki = 2193 nM T08123 CB4JL5 45909952 IC50 > 10000 nM T08123 CVJU38 46233842 IC50 = 46 nM T08123 CQ9A7L 46234188 IC50 = 5 nM T08123 C0AF2X 46234666 IC50 = 2970 nM T08123 CPEO49 46843906 IC50 = 3.5 nM T08123 CGTM17 46898099 IC50 = 67 nM T08123 CM73EY 46912329 IC50 = 4900 nM T08123 C2B6VG 46912330 IC50 = 390 nM T08123 CXC70W 46912331 Ki = 182 nM T08123 C9MN1J 46912430 IC50 = 880 nM T08123 CQWY38 46912641 IC50 = 440 nM T08123 CZ3G6S 46913411 IC50 = 110 nM T08123 CV7T6O 47051749 IC50 = 343 nM T08123 CZ4MI0 49678035 IC50 = 351 nM T08123 C53SWY 49830719 IC50 = 22265 nM T08123 CYM4B1 49873378 IC50 > 1000 nM T08123 CAQ8F7 51356954 IC50 = 63.1 nM T08123 C5HP1Z 51356955 IC50 = 25.12 nM T08123 CJK6W0 51357233 IC50 = 19.95 nM T08123 CCP4R8 51357236 IC50 > 25118.86 nM T08123 CQ8O4Y 51357512 IC50 = 39.81 nM T08123 C90CUV 51357515 IC50 = 94 nM T08123 CIPU75 51357517 IC50 = 2511.89 nM T08123 CF1H2I 52109436 IC50 = 633 nM T08123 CCT8U0 54673065 IC50 = 770 nM T08123 C1ZF5H 54754832 Ki = 11 nM T08123 CK1Z7L 54755067 Ki = 7 nM T08123 CY9KA8 54755181 Ki = 13 nM T08123 CSY80Z 54755789 Ki = 9 nM T08123 CGAC06 56786904 IC50 = 1900 nM T08123 CCGZ21 56940771 Ki = 27 nM T08123 CDIS83 56940772 Ki = 4.2 nM T08123 CF5T4L 56941359 IC50 = 170 nM T08123 CJ7O0S 56941360 IC50 = 410 nM T08123 CZO64R 56941655 Ki = 2.4 nM T08123 CI92PK 56942076 Ki = 147 nM T08123 C6IQ2P 56943105 Ki = 0.3 nM T08123 CGA0P9 57334382 Ki = 776 nM T08123 C5TJ4U 57334383 Ki = 928 nM T08123 C5WX2V 57334384 Ki = 561 nM T08123 CQP86G 57334387 Ki = 341 nM T08123 CTF0M7 57334388 Ki = 64 nM T08123 CA95WC 57334531 Ki = 198 nM T08123 CQ0C7W 57334533 Ki = 53 nM T08123 CCE18Y 57334534 Ki = 293 nM T08123 CF46ZH 57334685 Ki = 4226 nM T08123 C0YD1F 57334686 Ki = 186 nM T08123 CO5I8C 57334687 Ki = 367 nM T08123 C2X1OV 57334689 Ki = 700 nM T08123 CZJM56 57334838 Ki = 286 nM T08123 CB0V4Q 57334992 Ki = 355 nM T08123 CN1C0Y 57334993 Ki = 348 nM T08123 CQVG63 57335145 Ki = 1598 nM T08123 C2YX3K 57335445 Ki = 2535 nM T08123 CVQO80 57335590 Ki = 2219 nM T08123 C9TB0Q 57336018 Ki = 143 nM T08123 CZ81QY 57336022 Ki = 1650 nM T08123 C1IX2E 57336023 Ki = 225 nM T08123 C4I0QW 58494270 Ki = 54 nM T08123 C2W0OD 58539094 Ki = 1 nM T08123 C5UTG9 58539095 Ki = 6 nM T08123 C7G2XB 58539106 Ki = 4 nM T08123 C60QVD 58539109 Ki = 2 nM T08123 C6CDB7 58539140 Ki = 1 nM T08123 CB3TQ8 58539146 Ki = 58 nM T08123 C8NG0L 58539237 Ki = 12 nM T08123 C19LBX 58539246 Ki = 3 nM T08123 C7WRQ5 58539268 Ki = 7 nM T08123 C97ZGJ 58539301 Ki = 3 nM T08123 CXJ63M 59603829 IC50 < 10 nM T08123 CQEU96 59603842 IC50 = 3.1 nM T08123 C9PUK6 59618824 Ki = 44 nM T08123 CPC0J1 59618832 IC50 = 530 nM T08123 C4NP7V 59618853 IC50 = 410 nM T08123 CPG7N9 59618867 IC50 = 830 nM T08123 CPKJ27 59618871 IC50 = 97 nM T08123 C30PWU 59618913 IC50 = 1600 nM T08123 CULS42 59618916 IC50 = 130 nM T08123 CQW85Z 59618941 IC50 = 390 nM T08123 C3NDI8 59618946 IC50 = 2400 nM T08123 CK08DV 59618947 IC50 = 68 nM T08123 C8OH4T 59618953 IC50 = 170 nM T08123 CZ6I4N 59618971 IC50 = 150 nM T08123 C0FJE7 59618977 IC50 = 3000 nM T08123 C1E5YI 59619022 IC50 = 86 nM T08123 C2IV1R 59619059 IC50 = 4700 nM T08123 CJXN91 59619097 IC50 = 300 nM T08123 C4EHP8 59619113 IC50 = 1900 nM T08123 CHMP08 59619145 IC50 = 250 nM T08123 CFW1M3 60196513 Ki = 301 nM T08123 C5FJU9 60197123 Ki = 160 nM T08123 C0PYI9 60197124 Ki = 97 nM T08123 CG0OM3 60197218 Ki = 189 nM T08123 C9MC6A 60197321 Ki = 133 nM T08123 CPG4K0 60197831 Ki = 2242 nM T08123 CSZ6I5 66556035 IC50 = 251.19 nM T08123 CWU8E6 66556279 IC50 <= 500 nM T08123 C7MD5X 66556536 IC50 = 1258.93 nM T08123 CD3WZ0 66827038 IC50 = 4 nM T08123 CUGS26 66828963 Ki = 44 nM T08123 C3AQY8 66829086 IC50 = 15 nM T08123 CSOR32 66829097 IC50 = 3 nM T08123 CN3WO7 66994399 IC50 = 6186 nM T08123 C4P2VS 67106997 IC50 = 7.943 nM T08123 CGD1O0 67107000 IC50 = 12.59 nM T08123 CC18RT 67107081 IC50 = 15.85 nM T08123 CH91GR 67107177 IC50 = 12.59 nM T08123 C9SV4B 67107224 IC50 = 19.95 nM T08123 CUF6E1 67107237 IC50 = 7.943 nM T08123 CJQ52M 67107333 IC50 = 10 nM T08123 CL7KA9 67107360 IC50 = 15.85 nM T08123 CIV97A 67107407 IC50 = 39.81 nM T08123 CMD36P 67108013 IC50 = 10 nM T08123 CV63UL 67240318 IC50 > 10000 nM T08123 CA4VO9 67814206 Ki = 5 nM T08123 CZ8U0Y 67817055 Ki = 9 nM T08123 C49CYH 67818467 Ki = 6 nM T08123 C2HYA3 67818622 Ki = 2 nM T08123 C59DOP 67988921 Ki = 6 nM T08123 C30CWB 68069662 Ki = 7.8 nM T08123 C6XF7V 68069685 IC50 = 11 nM T08123 CI9SU3 68069764 Ki = 4600 nM T08123 C2LFT7 68107702 IC50 = 39.81 nM T08123 C3KQW0 68107965 IC50 = 8.9 nM T08123 CP2Q3S 68108534 IC50 = 7.943 nM T08123 C6VMC2 68108924 IC50 = 63.1 nM T08123 C6QJH5 68239103 IC50 = 1231 nM T08123 CP61LD 68295403 Ki = 295 nM T08123 CQ1D0B 68778984 IC50 = 130 nM T08123 C5DGR9 69036886 IC50 = 167 nM T08123 C3C6EI 69048008 Ki = 557 nM T08123 CHF59A 69048861 Ki = 92 nM T08123 C7E1HF 69081779 IC50 = 140 nM T08123 CUG5E9 69081998 Ki = 2 nM T08123 CM38XA 69083959 IC50 = 99 nM T08123 CR05LF 69085771 Ki = 6 nM T08123 CQ86JW 69091994 Ki = 21 nM T08123 C72ZVX 69092378 Ki = 11 nM T08123 C5Y3OZ 69092949 Ki = 1 nM T08123 C4WG1A 69093006 Ki = 3 nM T08123 C0NA7R 69093113 Ki = 4 nM T08123 CN3A5C 69093123 Ki = 3 nM T08123 C8EF1H 69093313 Ki = 41 nM T08123 CER1B9 69093374 Ki = 0.7 nM T08123 C2U6AZ 69093445 IC50 = 36 nM T08123 C6Z9GS 69093717 Ki = 3 nM T08123 CJ91XV 69281457 Ki = 9 nM T08123 CK2PS4 69281523 Ki = 2 nM T08123 CNK07L 69281529 Ki = 6 nM T08123 CXKU75 69281543 Ki = 4 nM T08123 CV3XD9 69281569 Ki = 2 nM T08123 CN82OH 69281678 Ki = 8 nM T08123 CC9NG8 69281703 Ki = 2 nM T08123 CD07CR 69281708 Ki = 2 nM T08123 C3GTU1 69762142 IC50 > 10000 nM T08123 C9K3LU 69936228 IC50 = 251.19 nM T08123 CAVH70 69936275 IC50 = 125.89 nM T08123 CB3NM4 69936458 IC50 = 10 nM T08123 CR25CZ 69936757 IC50 = 199.53 nM T08123 CD0ME9 69936791 IC50 = 1258.93 nM T08123 CRO43B 69937003 IC50 = 7.943 nM T08123 CBO21X 69937058 IC50 = 50.12 nM T08123 C6Q7NH 70096101 Ki = 5 nM T08123 CJ96RN 70099013 Ki = 6 nM T08123 CC5Y7E 71060772 IC50 = 412 nM T08123 C48ZLN 71060894 IC50 = 10 nM T08123 C81ZNG 71060941 IC50 = 66 nM T08123 C10CHQ 71060955 IC50 = 15 nM T08123 CP4QU7 71060982 IC50 = 378 nM T08123 CGMJ84 71060999 IC50 = 17 nM T08123 CK35TB 71061025 IC50 = 5 nM T08123 C2UR3H 71061036 IC50 = 1 nM T08123 C94IAV 71061083 IC50 = 23 nM T08123 CT2N7Y 71061182 IC50 = 55 nM T08123 CI3LN8 71061196 IC50 = 12 nM T08123 CH0E6M 71061284 EC50 = 242 nM T08123 CY9E5Z 71061321 IC50 = 59 nM T08123 CTF14U 71061353 IC50 = 142 nM T08123 C8YF0R 71061365 IC50 = 17 nM T08123 CE31SP 71061394 IC50 = 49 nM T08123 CAOC46 71061450 IC50 = 145 nM T08123 CSZ1O5 71061479 IC50 = 56 nM T08123 CIZ49M 71061494 IC50 = 121 nM T08123 CWO0S3 71061505 IC50 = 7 nM T08123 C57NEV 71061537 IC50 = 9 nM T08123 CJ73DM 71154928 IC50 = 1.2 nM T08123 C0T8HO 71450027 Ki = 1 nM T08123 CJK05F 71451846 Ki = 2 nM T08123 CL0M4V 71451847 Ki = 1 nM T08123 CKW32R 71451848 Ki = 2 nM T08123 CH27NO 71451849 Ki = 3 nM T08123 C0DJ8P 71451850 Ki = 4 nM T08123 CVNI90 71453547 Ki = 10 nM T08123 CX4LE5 71453548 Ki = 6 nM T08123 CAN57Z 71455263 Ki = 20 nM T08123 C5R3PF 71455393 Ki = 7 nM T08123 CPY5K3 71457046 Ki = 33 nM T08123 C1X6YV 71457047 Ki = 20 nM T08123 CTA0O7 71457164 Ki = 1 nM T08123 CML7F1 71458913 Ki = 11 nM T08123 C56AHL 71460830 Ki = 8 nM T08123 CYR35K 71460831 Ki = 9 nM T08123 CR6O7Q 71462440 Ki = 7 nM T08123 C2BUG4 71519483 IC50 = 965 nM T08123 CBN10O 71531214 IC50 = 466 nM T08123 CDM85H 71531360 IC50 = 205 nM T08123 CBXY59 71548179 Ki = 0.5 nM T08123 CAO1X2 71553438 IC50 = 6 nM T08123 C7ZQI4 71553439 IC50 = 5 nM T08123 C4EG2A 71578245 IC50 = 23 nM T08123 CWNO83 71578246 IC50 = 47 nM T08123 C3HK8A 71578314 IC50 = 7270 nM T08123 CIH0S5 71578315 IC50 = 39 nM T08123 C5EQN0 71578667 IC50 = 1313 nM T08123 CDLM98 71578668 IC50 = 2168 nM T08123 C17PUR 71578669 IC50 = 76 nM T08123 CUJ0E2 71578670 IC50 = 13 nM T08123 CD1TB6 71578671 IC50 = 18 nM T08123 C2ARC8 71578672 IC50 = 1727 nM T08123 CU49PG 71578673 IC50 = 2112 nM T08123 CR86ZT 71578754 IC50 = 134 nM T08123 C52VUT 71578755 IC50 = 164 nM T08123 C8YW5N 71578756 IC50 = 211 nM T08123 C8UL0Q 71578757 IC50 = 253 nM T08123 C8F5ED 71578758 IC50 = 3305 nM T08123 C7WGE9 71578759 IC50 = 265 nM T08123 CE2OV5 71578843 IC50 = 179 nM T08123 C0MD7S 71578844 IC50 = 309 nM T08123 CB1M4Z 71578845 IC50 = 511 nM T08123 CZLQ18 71578846 IC50 = 2020 nM T08123 CH93UE 71578847 IC50 = 22128 nM T08123 C0R5BV 71578848 IC50 = 19542 nM T08123 C95CTL 71578849 IC50 = 2026 nM T08123 CM92KY 71578927 IC50 = 2470 nM T08123 CHV29Y 71578928 IC50 = 8 nM T08123 CZYD04 71578929 IC50 = 77 nM T08123 C1U9BV 71578930 IC50 = 26 nM T08123 CYS49J 71578931 IC50 = 75 nM T08123 C0QMZ1 71578932 IC50 = 67 nM T08123 C8IB6O 71578933 IC50 = 117 nM T08123 C87JUI 71579008 IC50 = 33 nM T08123 CAB95H 71579009 IC50 = 141 nM T08123 CZ0I3G 71579010 IC50 = 48 nM T08123 C8QZI2 71579011 IC50 = 581 nM T08123 CHGE58 71579086 IC50 = 3117 nM T08123 CR6GF2 71579087 IC50 = 162 nM T08123 CTW3D7 71579088 IC50 = 798 nM T08123 CD92LR 71579089 IC50 = 2068 nM T08123 C3NVQ1 71579090 IC50 > 4000 nM T08123 C20NET 71579091 IC50 > 100000 nM T08123 CA27BQ 71579092 IC50 > 100000 nM T08123 CEKJ06 71579169 IC50 > 100000 nM T08123 C9OJM2 71579170 IC50 = 4570 nM T08123 CGDW70 71579171 IC50 = 18000 nM T08123 C2T6XH 71579172 IC50 = 1230 nM T08123 CZW4T9 71579173 IC50 = 2270 nM T08123 C40ESW 71579260 IC50 = 9 nM T08123 C27CXJ 71579261 IC50 = 14 nM T08123 CW16ZS 71579330 IC50 = 16 nM T08123 CS7A4H 71579331 IC50 = 12 nM T08123 C1DSG0 71579332 IC50 = 28 nM T08123 CNTV53 71579333 IC50 = 48 nM T08123 C8YMF0 71579334 IC50 = 109 nM T08123 CS59YL 71579335 IC50 = 10 nM T08123 CGZ73I 71579413 IC50 = 14 nM T08123 C0YD6V 71579414 IC50 = 27 nM T08123 CBZ5H8 71579415 EC50 = 1599 nM T08123 CQ0KM2 71579416 IC50 = 281 nM T08123 CYA1G3 71579417 IC50 = 450 nM T08123 C5O6GN 71579418 IC50 = 498 nM T08123 CMO25Q 71579419 IC50 = 1177 nM T08123 CV65KO 71618473 EC50 = 62 nM T08123 C3OS8U 71714087 IC50 = 11 nM T08123 C92AZQ 71714088 IC50 = 14 nM T08123 CN1Y9I 71714230 IC50 = 7 nM T08123 CM6NE9 71714231 IC50 = 9 nM T08123 CG28AP 71714232 IC50 = 3 nM T08123 C91CRY 71714233 IC50 = 8 nM T08123 C67HDT 71714234 IC50 < 3 nM T08123 CRS05F 71714235 IC50 < 3 nM T08123 CVC19T 71714373 IC50 = 4 nM T08123 CD5C8J 71714374 IC50 = 4 nM T08123 C51ISR 71714375 IC50 = 31 nM T08123 C5HJK2 71714376 IC50 = 7 nM T08123 C70SJV 71714377 IC50 < 3 nM T08123 CK7T2U 71714378 IC50 = 150 nM T08123 CRA97Q 71716389 IC50 = 2512 nM T08123 CD6TF5 71717133 IC50 = 2020 nM T08123 CVN80C 71717134 EC50 = 435 nM T08123 C0YFP8 71718226 IC50 = 35 nM T08123 CM5SW1 71718384 IC50 = 55 nM T08123 CFSN02 71718965 IC50 = 88597 nM T08123 C8HMA7 71719424 IC50 = 168 nM T08123 CKNB62 71720020 IC50 = 9 nM T08123 C2BCG9 71720168 IC50 = 71 nM T08123 C27MEF 71720656 EC50 = 290 nM T08123 C8ON1P 71720813 EC50 = 731 nM T08123 C2JUF3 71720814 IC50 = 1747 nM T08123 CXH7N3 71736610 Ki = 1.2 nM T08123 C3UE2O 71736769 Ki = 3.1 nM T08123 C2OGC1 71736927 Ki = 4.1 nM T08123 CNU94W 71737255 Ki = 151 nM T08123 CIJ6V1 72191820 Ki = 0.7 nM T08123 CT9UK8 72201342 Ki = 3 nM T08123 C6T2UJ 72201343 Ki = 3 nM T08123 COGM19 72201489 Ki = 0.9 nM T08123 C6M1YO 72706006 IC50 = 20 nM T08123 CXP2V3 72706157 IC50 = 69 nM T08123 CYGI30 72706399 IC50 = 8 nM T08123 CA3E7M 72706402 IC50 = 20 nM T08123 C7A4BC 72706513 IC50 = 28 nM T08123 CCX6R1 72706517 IC50 = 9 nM T08123 C0XM9Z 72706586 IC50 = 8 nM T08123 C95GZV 72706839 IC50 = 26 nM T08123 CX48SV 72706841 IC50 = 5 nM T08123 C68GYC 72706904 IC50 = 122 nM T08123 CWN2A7 72706906 IC50 = 6 nM T08123 CLOE10 72706962 IC50 = 16 nM T08123 CCQ5I1 72707018 IC50 = 95 nM T08123 C3V8ZX 72707020 IC50 = 79 nM T08123 CX75YR 73352604 IC50 = 398.11 nM T08123 CHY9T6 76310861 Ki = 6 nM T08123 C4A0CF 76328935 Ki = 2 nM T08123 CAB9W0 76336221 IC50 = 53 nM T08123 C4Q5IN 76514427 Ki = 1640 nM T08123 C9WH0O 77068229 IC50 = 387 nM T08123 C8BAS5 77105954 IC50 = 710 nM T08123 C20QLI 77105957 IC50 = 390 nM T08123 CEOC93 77105960 IC50 = 540 nM T08123 C52TFP 77106161 IC50 = 280 nM T08123 C5RI9B 77106162 IC50 = 600 nM T08123 C12MFU 77106364 IC50 = 910 nM T08123 C4B3OS 77106759 IC50 = 160 nM T08123 C5NYW0 77106960 IC50 = 1300 nM T08123 CLB1A4 78319901 IC50 = 0.76 nM T08123 C0ED6J 78319902 IC50 = 2 nM T08123 CS9U2F 78321156 IC50 = 3.8 nM T08123 CUTK65 78321839 IC50 = 7.2 nM T08123 C9NL4K 78322146 IC50 = 41 nM T08123 CEF9C7 78323982 IC50 = 10 nM T08123 C6W5QH 78323983 IC50 = 2.2 nM T08123 CL06IB 85472082 IC50 = 15 nM T08123 C56VDQ 85472857 IC50 = 12 nM T08123 CY2PF9 85472971 IC50 = 98 nM T08123 CU6B5D 86275848 Ki = 0.06 nM T08123 CYD43G 86287677 IC50 = 108 nM T08123 CM2A5T 86287678 IC50 = 27 nM T08123 C4HZ0K 86287740 IC50 = 50 nM T08123 CN2H3I 86287744 Ki = 0.5 nM T08123 C0NT3J 86287745 IC50 = 85 nM T08123 CQ1OI2 86287807 Ki = 3 nM T08123 C7M1KT 86287812 Ki = 31 nM T08123 CNJO04 86287875 Ki = 4 nM T08123 CG9XP0 86287876 Ki = 6 nM T08123 CZ31RV 86295257 Ki = 3.5 nM T08123 C1HW4B 89735655 IC50 = 62 nM T08123 CKYX09 89887060 Ki = 46 nM T08123 C57VTG 89887105 Ki = 372 nM T08123 C67WIJ 89889447 Ki = 39 nM T08123 COLS74 89889448 IC50 = 31 nM T08123 CKB38T 89914324 IC50 = 20 nM T08123 CIA65G 89914405 IC50 = 42 nM T08123 C2J8EP 89914567 IC50 = 18 nM T08123 CJ8D0S 89914904 IC50 = 18 nM T08123 CEO2Z8 89915076 IC50 = 37 nM T08123 CZ75OC 89915123 IC50 = 5 nM T08123 CW8Z6M 90398640 IC50 = 134 nM T08123 CPN72Q 90400634 IC50 = 6.4 nM T08123 C0T1HM 90400705 IC50 = 4.4 nM T08123 CEU52A 90400735 IC50 = 2.6 nM T08123 CK1U9Q 90400782 IC50 = 0.8 nM T08123 CU83QB 90400825 IC50 = 13 nM T08123 CMR3Z2 90400868 IC50 = 83 nM T08123 CMXV30 90400979 IC50 = 0.7 nM T08123 CX59BA 90401078 IC50 < 0.6 nM T08123 CNT0B7 90401093 IC50 = 18 nM T08123 C7LN1D 91623338 IC50 = 204 nM T08123 CEPI85 102532139 IC50 = 30 nM T08123 C9JC0V 117653476 Ki = 23 nM T08123 C1TF9K 118368174 IC50 = 33 nM T08123 CJA6T0 118711382 IC50 = 496 nM T08123 CN26EQ 118711383 IC50 = 242 nM T08123 CKTW37 118711384 IC50 = 349 nM T08123 CN8R0C 118711385 IC50 = 880 nM T08123 C02PGS 118711386 IC50 = 66 nM T08123 CIZ89U 118711387 IC50 = 2290 nM T08123 C9YVC5 118711388 IC50 = 2489 nM T08123 CYZP82 118711389 IC50 = 12600 nM T08123 CP4I3E 118711390 IC50 = 32000 nM T08123 C2S3NT 118711391 IC50 = 4330 nM T08123 COJ9R7 118711392 IC50 = 91 nM T08123 CV8FB5 118711393 IC50 = 95 nM T08123 C3Q6ZG 118711394 IC50 = 2760 nM T08123 C38MFC 118711395 IC50 = 1260 nM T08123 CNX90H 118711396 IC50 = 1070 nM T08123 C2GXW0 118711397 IC50 = 2110 nM T08123 CYI4C5 118711398 IC50 = 2070 nM T08123 CBIA81 118711399 IC50 = 78 nM T08123 C4KEP1 118711400 IC50 = 373 nM T08123 C4EVI2 118711401 IC50 = 1350 nM T08123 C41FJN 118711402 IC50 = 12635 nM T08123 CJH46F 118711403 IC50 = 236 nM T08123 CUM9T7 118711404 IC50 = 549 nM T08123 C1V9IW 118711405 IC50 = 6202 nM T08123 CB5O6N 118711406 IC50 = 9124 nM T08123 CG40AO 118711407 IC50 = 1211 nM T08123 C06EWA 118711408 IC50 = 763 nM T08123 CE0W9G 118711409 IC50 = 21858 nM T08123 CNL54X 118711410 IC50 = 32000 nM T08123 CDTB86 118711411 IC50 = 32000 nM T08123 CJ03UP 118711412 IC50 = 1461 nM T08123 CW7VI0 118711413 IC50 = 400 nM T08123 CUV48F 118711414 IC50 = 488 nM T08123 CNV50B 118711415 IC50 = 525 nM T08123 CST6F7 118711416 IC50 = 5850 nM T08123 CZEO41 118711417 IC50 = 1145 nM T08123 CKUG73 118711418 IC50 = 115 nM T08123 C74FZL 118711419 IC50 = 110 nM T08123 CB47ZY 118714386 IC50 = 261 nM T08123 CP27FW 118714387 IC50 = 163 nM T08123 CN3X5T 118714393 IC50 = 31 nM T08123 C97GTN 118714394 IC50 > 10000 nM T08123 CQOY61 118714395 IC50 = 46 nM T08123 CS1F8A 118725474 IC50 = 115 nM T08123 CB8IJ7 118725475 IC50 = 5223 nM T08123 CIT2O4 118725476 IC50 = 393 nM T08123 CC8EJ6 118725477 IC50 = 117 nM T08123 CIQ5T2 118725478 IC50 = 80 nM T08123 CV8B3E 118725479 IC50 = 686 nM T08123 CT03NG 118725480 IC50 = 2243 nM T08123 CHJ78I 118725505 IC50 = 1199 nM T08123 CGJ75M 118725506 IC50 = 8 nM T08123 C5CY0G 118725507 IC50 = 111 nM T08123 CTR71E 118725508 IC50 = 2331 nM T08123 CZ7LM6 118725509 IC50 = 139 nM T08123 C54JEF 118725510 IC50 = 222 nM T08123 CR9ML7 118725554 IC50 = 99 nM T08123 CAD9B8 118731632 IC50 = 72 nM T08123 CBM50V 118731633 IC50 = 51.2 nM T08123 CJSX41 118731634 IC50 > 1000 nM T08123 CF8IT2 118731635 IC50 = 654 nM T08123 CE31VZ 118731636 IC50 > 1000 nM T08123 CPD5M4 118731637 IC50 > 1000 nM T08123 CSQ8D3 118731638 IC50 > 1000 nM T08123 C0HG6I 118731639 IC50 > 1000 nM T08123 C1QNH2 118731640 IC50 > 1000 nM T08123 CC4V7Z 118731641 IC50 > 1000 nM T08123 C84HRP 118731642 IC50 > 1000 nM T08123 CR0UN5 118731643 IC50 > 1000 nM T08123 C4WEK7 118731644 IC50 > 1000 nM T08123 CA04ZD 118731645 IC50 > 1000 nM T08123 CNEC23 118731646 IC50 > 1000 nM T08123 CNG07R 118731647 IC50 > 1000 nM T08123 C9J5VH 118731648 IC50 > 1000 nM T08123 C2YQK9 118731649 IC50 > 1000 nM T08123 CIU1F4 118731650 IC50 > 1000 nM T08123 C9ROB3 118731651 IC50 > 1000 nM T08123 CLOF30 118731652 IC50 > 1000 nM T08123 CM7RP3 118731653 IC50 > 1000 nM T08123 C0KM7P 118731654 IC50 > 1000 nM T08123 C2Y7MH 118733361 IC50 = 130 nM T08123 C39LIM 126691326 IC50 = 4.13 nM T08123 CYU38M 127046607 Ki = 305 nM T08123 CIA9X7 127047484 Ki = 159 nM T08123 COI8G1 127047659 Ki = 28 nM T08123 CO1SP2 127047756 Ki = 5610 nM T08123 C7BRS1 127048109 Ki = 30 nM T08123 CO8Z2N 129900111 IC50 = 714 nM T08123 CK8R5Y 134145931 IC50 = 130 nM T08123 CIP61L 134153498 IC50 = 754 nM T08123 C54FXD 134957362 IC50 > 10000 nM T08123 CA9ME4 135325094 IC50 = 5.55 nM T08123 CVSO41 135325140 IC50 = 6.39 nM T08123 CVN7D3 135399193 IC50 = 3830 nM T08123 CBV30L 135402333 IC50 = 3110 nM T08123 CMA49H 135406018 IC50 = 2170 nM T08123 C6NWV2 135438718 IC50 = 15400 nM T08123 CY06RE 135439090 IC50 = 110 nM T08123 CVQ6I5 135442567 IC50 = 2980 nM T08123 C0O2VG 135443554 Ki = 3450 nM T08123 CLIC03 135468562 IC50 = 13200 nM T08123 C1KLP4 135478724 IC50 = 3690 nM T08123 C2PRQ9 135481207 IC50 = 5400 nM T08123 C05WVF 135491980 IC50 = 20 nM T08123 CNU3X6 135541201 IC50 = 7270 nM T08123 C6DE1S 135543409 IC50 = 1700 nM T08123 C1DW2N 135553979 IC50 = 1340 nM T08123 CTM91E 135600848 IC50 = 2340 nM T08123 CRE6X9 135982538 Ki = 550 nM T08123 C3ZC0S 136035743 IC50 = 53 nM T08123 C9RT5K 136386182 IC50 = 280 nM T08123 C1ZNX7 136386185 IC50 = 1020 nM T08123 C2E4SY 136577433 IC50 = 1200 nM T08123 CK9V1P 137199823 IC50 = 10 nM T08123 CA1B4T 137631885 Ki = 136 nM T08123 CZ2WJ1 137632774 IC50 = 205 nM T08123 CT2BI3 137633878 IC50 = 9100 nM T08123 CJK0Y9 137635622 IC50 = 728 nM T08123 CE3TS9 137636366 IC50 = 2200 nM T08123 CS9H7X 137636896 IC50 = 102 nM T08123 C7XTV2 137637903 IC50 = 57000 nM T08123 C1D0ZQ 137639268 IC50 = 44 nM T08123 CKW84R 137641709 IC50 = 1995.26 nM T08123 COH0Z7 137642181 IC50 = 2900 nM T08123 CT76GD 137642252 IC50 = 15848.93 nM T08123 CLF8W2 137643090 IC50 = 64 nM T08123 C0PDY6 137643960 Ki = 23 nM T08123 CQTK16 137646685 IC50 = 256 nM T08123 C2WIN1 137647763 IC50 = 28 nM T08123 CO0G8M 137649243 IC50 > 25118.86 nM T08123 CH3CM6 137650444 Ki = 783 nM T08123 CTAP14 137651126 Ki = 95 nM T08123 CUY89G 137651440 IC50 = 210 nM T08123 CQY7I9 137651563 IC50 > 25118.86 nM T08123 CG6BX0 137653375 IC50 = 11000 nM T08123 C9XAD7 137653470 IC50 = 12000 nM T08123 C7EPY6 137654369 IC50 = 13000 nM T08123 C8VPB4 137654430 IC50 = 44 nM T08123 C1L0DX 137655129 Ki = 225 nM T08123 C12RCY 137657070 IC50 = 3600 nM T08123 CU3LS5 137657223 IC50 = 6700 nM T08123 C71WCI 137658381 IC50 = 6.6 nM T08123 CY1C7A 137658612 IC50 = 13000 nM T08123 CN2W4L 137659738 IC50 = 5800 nM T08123 CM9BJ8 137659810 IC50 = 93 nM T08123 C46OEV 137660994 IC50 = 170 nM T08123 CZ9BN4 138320062 IC50 = 0.001 nM T08123 C7HO6Z 138550167 IC50 = 2.6 nM T08123 C19EZB 138550184 IC50 = 20.2 nM T08123 CLXQ83 138550248 IC50 = 1 nM T08123 C3HO8V 138550388 IC50 = 4.4 nM T08123 CRS3P0 138550552 IC50 = 0.9 nM T08123 C3Z6KF 141301379 IC50 = 20 nM T08123 CQ9M7D 142423799 IC50 = 1530 nM T08123 CQJ1X6 142423813 IC50 = 0.94 nM T08123 CF8KR7 142423880 IC50 = 8.7 nM T08123 C3RWS0 145964556 IC50 = 130 nM T08123 CBKU04 145965102 IC50 = 5350 nM T08123 CV9GM5 145966574 IC50 = 6980 nM T08123 CE41QV 145971783 IC50 = 7490 nM T08123 C1S4OD 145972297 IC50 = 760 nM T08123 CK8P5F 145974450 IC50 = 550 nM T08123 CU3V0W 145975422 IC50 = 1500 nM T08123 CIYM29 145975752 IC50 = 5930 nM T08123 C85WPK 145976833 IC50 = 120 nM T08123 C5M4RL 145977765 IC50 = 490 nM T08123 COG17U 146405943 IC50 = 280 nM T08123 C9YT1C 146405944 IC50 = 160 nM T08123 CC84BD 146405947 IC50 = 370 nM T08123 CT1Q0U 146405949 IC50 = 370 nM T08123 CDX63Y 146405954 IC50 = 330 nM T08123 C4V1QD 146405955 IC50 = 370 nM T08123 CMEB27 146405958 IC50 = 980 nM T08123 CRO92Y 146405959 IC50 = 170 nM T08123 CDFY63 146405961 IC50 = 1120 nM T08123 CE8SG3 146405966 IC50 = 260 nM T08123 CNC6Y1 153407886 IC50 = 3.31 nM T08123 C2J7UI 154031581 IC50 = 3.21 nM T08123 CR2GM1 155511660 IC50 = 12.59 nM T08123 C0TSM8 155511739 IC50 = 19.95 nM T08123 C2MD1Q 155513187 IC50 > 10000 nM T08123 CNY51A 155514319 IC50 = 25.12 nM T08123 CU6QY4 155515764 IC50 > 10000 nM T08123 CN4IB6 155516354 IC50 = 19.95 nM T08123 C8G4EJ 155516586 IC50 = 39.81 nM T08123 CI8RQ9 155516974 IC50 = 2 nM T08123 C6H0FR 155517433 IC50 = 3.31 nM T08123 CSJY76 155517776 IC50 = 25.12 nM T08123 CVH0P8 155519454 IC50 = 19.95 nM T08123 CH60UK 155521075 IC50 = 12.59 nM T08123 CG20IT 155522201 IC50 > 10000 nM T08123 C9TSH7 155522966 IC50 = 31.62 nM T08123 CZY05O 155524160 IC50 = 25.7 nM T08123 CZW45D 155525803 IC50 = 39.81 nM T08123 CE9KC4 155529925 IC50 > 10000 nM T08123 C8P4QZ 155530738 IC50 = 12.59 nM T08123 CR70GX 155532115 IC50 = 25.12 nM T08123 C2CG1A 155537016 IC50 > 10000 nM T08123 CH3I8Z 155539469 IC50 = 10 nM T08123 CB0OK8 155540491 IC50 = 19.95 nM T08123 CL3MR0 155542649 IC50 = 50.12 nM T08123 CI84SJ 155543889 IC50 > 10000 nM T08123 CO1CN9 155547476 IC50 = 25.12 nM T08123 CV4B5R 155548069 IC50 = 15.85 nM T08123 CC1LI7 155550279 IC50 = 39.81 nM T08123 C93CKT 155553547 IC50 = 63.1 nM T08123 CX8GR9 155553934 IC50 = 15.85 nM T08123 CJ1BF3 155557829 IC50 = 1 nM T08123 C8HWI4 155558510 IC50 = 7.943 nM T08123 C4M9WK 155558971 IC50 = 9.73 nM T08123 CBO2R8 155561624 IC50 = 19.95 nM T08123 CM6L9J 155562224 IC50 = 12.59 nM T08123 CYQI51 155562763 Ki = 3900 nM T08123 C4BWO7 155566862 IC50 = 19.95 nM T08123 CS12BT 155569011 IC50 = 13 nM T08123 CP17HA 155569379 IC50 = 63.1 nM T08123 D01OXV 76328936 Ki = 2 nM T08123 D01XYD 16760524 IC50 = 22 nM T08123 D07ADX 54764565 IC50 = 11 nM T08123 D0B6KT 72706837 IC50 = 278 nM T08123 D0J5FK 58539171 Ki = 1 nM T08123 D0R2WK 16038120 IC50 = 6.1 nM T08123 D0U3NI 53246941 IC50 = 16 nM T08123 D0WK9R 72706840 IC50 = 3 nM T08123 D0YQ8V 46236221 IC50 = 35 nM T56588 D0I0DL 3689 IC50 = 75900 nM T56588 C63KYD 66637 EC50 = 10000 nM T56588 CD48TY 694463 IC50 = 426000 nM T56588 CD5RW2 1279398 IC50 = 1400 nM T56588 C5Z6NT 3113150 IC50 = 2700 nM T56588 CXF09D 4231127 EC50 = 2800 nM T56588 CN85UI 4235339 IC50 = 2700 nM T56588 CI28HT 22432385 EC50 = 6700 nM T56588 CA72VD 44322229 IC50 = 14000 nM T56588 CIC1G6 46861929 IC50 = 3900 nM T56588 C39CGI 56653056 IC50 = 50000 nM T56588 C4KWB0 56654447 EC50 = 29000 nM T56588 C7XPS1 66727815 IC50 = 2400 nM T56588 D06XGK 105074 EC50 = 78000 nM T56588 D09HXX 4787937 IC50 > 10000 nM T04123 CU5ND3 57514697 IC50 > 200000 nM T04123 C0IJ2X 118737463 IC50 > 50000 nM T04123 C12OHP 122187565 IC50 > 50000 nM T04123 CXHR32 122187566 IC50 > 50000 nM T04123 C59OUG 122187567 IC50 > 50000 nM T76285 C0NJ2B 645025 IC50 = 350 nM T76285 CRM9S6 674647 IC50 = 1150 nM T76285 CN06WE 685663 IC50 = 630 nM T76285 C5UAR2 910374 IC50 = 3220 nM T76285 C83UKT 1223927 IC50 = 5980 nM T76285 CAX45S 3332652 IC50 = 1810 nM T76285 CW7YG3 3724041 IC50 = 3420 nM T76285 C9KGH4 13224102 IC50 = 3150 nM T76285 CG19LI 23342610 IC50 = 1260 nM T76285 C7I0CN 32937631 IC50 = 2772 nM T76285 CRZ62F 73355036 IC50 = 1270 nM T76285 C5M9IT 101891745 Ki = 68100 nM T76285 C8HPR3 127045881 IC50 = 369 nM T76285 CZ58ER 127045883 IC50 = 856 nM T76285 CM1QX6 132584225 IC50 = 2250 nM T76285 CDF79W 145950387 IC50 > 100000 nM T76285 C9VIW7 145951405 IC50 = 1140 nM T76285 CI0DE8 145952129 IC50 > 100000 nM T76285 C8WY3S 145952263 IC50 > 100000 nM T76285 CCE24P 145953494 IC50 > 100000 nM T76285 CHSD24 145955401 IC50 > 100000 nM T76285 CVM5E8 145957948 IC50 > 100000 nM T76285 CVC6A1 145958826 IC50 > 100000 nM T76285 C8LWV3 145958854 IC50 = 390 nM T76285 CYG9B0 145958960 IC50 = 360 nM T76285 C6YJ4N 145961405 IC50 > 100000 nM T76285 CJ0IQ6 145962930 IC50 > 100000 nM T76285 CHN5E3 145974297 IC50 = 2420 nM T76285 CWKM51 145979441 IC50 = 230 nM T76285 CDQ0T6 145981705 IC50 = 410 nM T76285 CE8N3X 145987231 IC50 = 12400 nM T76285 C87AJL 145988932 IC50 = 1260 nM T76285 CVWI49 145990949 IC50 = 2260 nM T76285 CTQ21M 145991361 IC50 = 1220 nM T76285 CPI0F4 145992202 IC50 = 320 nM T76285 CFW27N 145992560 IC50 = 510 nM T76285 CI4C2R 145992946 IC50 = 2370 nM T76285 C4QID1 145993905 IC50 = 1530 nM T76285 C5JWS2 155512949 IC50 = 6602 nM T76285 C83ARF 155516516 IC50 = 3424 nM T76285 CD0Q7G 155516795 IC50 = 1810 nM T76285 CZ1I3O 155522133 IC50 = 255 nM T76285 CUH9K1 155527208 IC50 = 1624 nM T76285 C4HMC0 155530954 IC50 = 1079 nM T76285 CVX03O 155532639 IC50 = 1790 nM T76285 C0SBV5 155532733 IC50 = 1203 nM T76285 C64ULP 155536432 IC50 = 710 nM T76285 C1J0QI 155537162 IC50 = 1550 nM T76285 CE29XR 155538214 IC50 = 5426 nM T76285 CT98MF 155538277 IC50 = 807 nM T76285 CV3YF4 155540276 IC50 = 1525 nM T76285 CYH39A 155541761 IC50 = 2578 nM T76285 C10HXE 155543015 IC50 = 2409 nM T76285 CB8J0V 155549452 IC50 = 1014 nM T76285 CB2PX0 155549933 IC50 = 230 nM T76285 CI17FY 155556622 IC50 = 13520 nM T76285 CP6TE8 155557159 IC50 = 1510 nM T76285 C3RFG8 155559027 IC50 = 490 nM T76285 C1B4XC 155560220 IC50 = 1354 nM T76285 CV3X5K 155560593 IC50 = 3963 nM T76285 CGZ6L8 155561305 IC50 = 2675 nM T76285 CMNZ48 155561927 IC50 = 2892 nM T76285 C25AMC 155563065 IC50 = 214 nM T76285 CE1JW7 155564260 IC50 = 20510 nM T76285 C9XDT6 155566859 IC50 = 254 nM T76285 C75NHE 155567060 IC50 = 1724 nM T76285 C2UO0Y 155568526 IC50 = 1240 nM T76285 CTJK02 155568923 IC50 = 47010 nM T76285 CVTY16 155569460 IC50 = 2267 nM T60366 D0L4FS 5280961 IC50 = 26000 nM T60366 D0U3EP 445154 IC50 = 19000 nM T60366 CVIJ45 10520980 IC50 = 7400 nM T60366 CXVZ64 10542828 IC50 = 5200 nM T60366 CG1QD8 10689330 IC50 = 3900 nM T60366 CL79EJ 44418841 IC50 = 1.95 ug.mL-1 T60366 C15SEA 44418843 IC50 = 7.83 ug.mL-1 T60366 CM5X6O 44559035 IC50 > 30000 nM T60366 CXD56M 44559036 IC50 = 2200 nM T60366 CYP32C 44559037 IC50 = 2100 nM T60366 C4N6IJ 44559077 IC50 = 1100 nM T60366 CQZ5A3 44559078 IC50 = 2300 nM T60366 D04FIN 629965 IC50 = 3400 nM T60366 D04ZDD 44559034 IC50 = 2600 nM T60366 D0F3QP 5889042 IC50 = 4700 nM T60366 D0N4YR 10712965 IC50 = 3600 nM T16993 D0AF6O 71731823 IC50 = 3.3 nM T16993 D0OB0F 5328940 IC50 = 490 nM T16993 D06KTJ 53252276 IC50 = 51 nM T16993 D0E3TC 44259 IC50 = 1.8 nM T16993 D0T3ME 156422 IC50 = 17000 nM T16993 CB7WK3 5938113 IC50 = 42700 nM T16993 C5HW8Y 9949798 IC50 = 480 nM T16993 CACS26 11561968 Ki > 2000 nM T16993 CU0E8O 11690457 Ki > 2000 nM T16993 C3VRO9 44557921 IC50 > 10000 nM T16993 CLS29B 46872626 IC50 > 10000 nM T16993 CEQN27 52936621 Ki > 1000 nM T16993 C8NA4L 53384644 IC50 > 30000 nM T16993 C9UD0Y 56599956 IC50 = 25 nM T16993 C1MR8Q 60097495 IC50 > 1000 nM T16993 CV63UL 67240318 IC50 > 10000 nM T16993 CBE1V7 69284028 IC50 = 2.6 nM T16993 CPG3A5 86302574 IC50 > 30000 nM T16993 CE4GW0 123328993 IC50 = 210 nM T16993 C28QUP 137652864 IC50 = 5911 nM T16993 C38KLH 138393287 IC50 = 0.49 nM T16993 C2MD1Q 155513187 IC50 > 10000 nM T16993 C1RD6I 155520028 IC50 = 4.7 nM T16993 CWB35U 155523839 IC50 > 4000 nM T16993 CID82K 155524475 IC50 = 14 nM T16993 C4ZUI1 155524823 IC50 = 410 nM T16993 CLO7U1 155525161 IC50 > 4000 nM T16993 CNX69I 155525990 IC50 = 2.7 nM T16993 CMC65B 155527759 IC50 > 4000 nM T16993 C47UCR 155534288 IC50 = 57 nM T16993 C78MZC 155536330 IC50 = 2 nM T16993 CJ5FA1 155537070 IC50 > 1300 nM T16993 CO6CG8 155541167 IC50 = 510 nM T16993 CDG12I 155546428 IC50 = 440 nM T16993 CBO07E 155554038 IC50 = 460 nM T16993 CU8L9S 155554641 IC50 = 440 nM T16993 C3CSG4 155554781 IC50 = 10 nM T16993 CJQ65O 155560050 IC50 = 31 nM T16993 CP9HG1 155563860 IC50 > 4000 nM T16993 D09PTP 57325421 IC50 = 85 nM T16993 D0K5UF 72710568 IC50 = 2 nM T73475 D00MDP 466151 IC50 = 54 nM T73475 D05VZE 119031 IC50 = 4.1 nM T73475 D0MW3H 9824350 IC50 = 18.5 nM T73475 D0N4IV 10718956 IC50 > 1000 nM T73475 D0U2BH 65064 IC50 = 21500 nM T73475 D00UCC 9827497 IC50 = 11000 nM T73475 D01DVX 9847838 IC50 = 466 nM T73475 D03BOZ 3342298 IC50 = 210 nM T73475 D05VNG 9908389 IC50 = 11 nM T73475 D0P8YC 5362422 IC50 = 2.4 nM T73475 D0T9HG 132519 IC50 = 33 nM T73475 D0Y1XT 128564 IC50 = 30 nM T73475 CNA81R 1836 IC50 > 50000 nM T73475 CY78XM 4218 Ki = 30 nM T73475 CFY8Q2 4230 IC50 = 232 nM T73475 CDJS43 154136 IC50 = 460 nM T73475 C50IPY 154137 IC50 = 366 nM T73475 C7ROG5 177347 IC50 > 10000 nM T73475 C4U7SY 401129 IC50 = 72000 nM T73475 CV60YH 445010 IC50 = 3393 nM T73475 CK9M3P 445018 IC50 > 10000 nM T73475 C4D7TS 448002 Ki = 13000 nM T73475 CG1I8P 467296 IC50 > 100000 nM T73475 CTPW02 467297 IC50 > 100000 nM T73475 C9I8WB 478379 Ki = 3 nM T73475 CP0JM7 2109230 Ki = 10000 nM T73475 CN6E3U 2366268 IC50 > 10000 nM T73475 CY3TD6 3348132 Ki > 2000 nM T73475 CQ4VL5 5287415 IC50 = 3900 nM T73475 CJ3QI1 5288814 IC50 > 10000 nM T73475 C5IDT0 5289314 Ki = 850 nM T73475 CQEF36 6539670 IC50 = 180 nM T73475 CP7BG0 6852146 EC50 = 4 nM T73475 CN5L2B 6852147 IC50 = 460 nM T73475 C7Y1BX 9543420 IC50 = 886 nM T73475 CIXD67 9802768 IC50 > 10000 nM T73475 CQ46XD 9804842 IC50 = 20000 nM T73475 C6KJ9W 9822461 IC50 = 1700 nM T73475 C1MPW9 9823182 IC50 > 50000 nM T73475 C8IMT2 9847787 IC50 = 2.2 nM T73475 C7VXJ5 9848025 IC50 = 2.2 nM T73475 C4IEK0 9850035 IC50 = 9000 nM T73475 C8GE7U 9862764 IC50 > 50000 nM T73475 CJS23I 9868333 Ki = 25 nM T73475 CG17NZ 9869811 IC50 > 10000 nM T73475 C38BVX 9870100 IC50 > 1000 nM T73475 CHU9I8 9871883 IC50 = 7000 nM T73475 C0ZT7A 9883002 Ki = 96000 nM T73475 CZBK85 9886177 IC50 > 50000 nM T73475 C4PB5Z 9887544 IC50 = 3 nM T73475 C3ZG6O 9887870 IC50 = 7200 nM T73475 CD1U5P 9889190 IC50 > 10000 nM T73475 C27HMG 9889517 IC50 = 0.78 nM T73475 CH69LT 9892815 Ki = 7000 nM T73475 CSIB97 9896504 IC50 > 30000 nM T73475 C2R5CX 9905493 IC50 = 895 nM T73475 CN6WJ1 9909994 IC50 = 440 nM T73475 CM2F7R 9910302 IC50 = 1.2 nM T73475 CK5OV9 9930210 IC50 = 39 nM T73475 CDXR37 9933197 IC50 > 10000 nM T73475 C65ION 9935032 IC50 > 10000 nM T73475 CG38KL 9936728 Ki = 1.5 nM T73475 C16HTN 9948666 Ki = 3400 nM T73475 CN76XI 9957653 IC50 = 925 nM T73475 CVG0O2 9959014 IC50 > 1000 nM T73475 CFQ15E 9976696 IC50 = 45 nM T73475 C0HL2X 9976697 IC50 = 30 nM T73475 C09LSY 9979489 Ki > 6368 nM T73475 CO09PN 9983251 IC50 = 931 nM T73475 CJGR30 9983604 IC50 = 2590 nM T73475 CB2J3S 9999667 IC50 = 2000 nM T73475 C6U3CK 10006134 IC50 = 905 nM T73475 CR7T3J 10009978 Ki = 177 nM T73475 CJ6H8O 10019658 IC50 = 2027 nM T73475 C6WHU4 10023722 IC50 = 18 nM T73475 CJR59P 10031295 Ki > 6368 nM T73475 CLXN48 10047373 IC50 = 16500 nM T73475 CAN59F 10047708 IC50 = 1.6 nM T73475 CLZ87W 10051236 Ki = 635 nM T73475 CJK0R1 10074190 IC50 = 3307 nM T73475 C8AEK4 10093420 IC50 = 0.3 nM T73475 CA6X2Z 10095338 IC50 = 1.1 nM T73475 CMY3X2 10098158 IC50 = 3.1 nM T73475 C2XV5J 10098250 IC50 = 1020 nM T73475 C3V2HW 10099112 IC50 = 15000 nM T73475 C7A8MI 10120093 IC50 > 10000 nM T73475 CYU19P 10127901 Ki > 6370 nM T73475 CH0UW2 10129190 Ki > 6370 nM T73475 CUG62E 10155007 IC50 > 40000 nM T73475 CLQ89T 10155008 IC50 > 40000 nM T73475 CR5H6E 10163627 Ki = 5858 nM T73475 CZO5V4 10164317 IC50 = 20 nM T73475 CGB27E 10174981 Ki > 6370 nM T73475 CL47AR 10175070 Ki > 6370 nM T73475 C4ULO6 10175077 Ki > 6370 nM T73475 C84ZQD 10175219 Ki > 6370 nM T73475 CIT0H4 10175323 Ki > 6370 nM T73475 C95IGP 10175331 Ki > 6370 nM T73475 CT7U0M 10175426 Ki > 6370 nM T73475 CK0P3F 10186536 Ki = 4075 nM T73475 C51RPY 10195069 Ki > 6370 nM T73475 CCHX74 10195307 Ki > 6370 nM T73475 C94KHT 10195527 Ki > 6370 nM T73475 CDG35O 10196192 Ki > 6370 nM T73475 C4K1MJ 10208262 Ki = 3502 nM T73475 CG8FA4 10218128 Ki > 6370 nM T73475 C7Y2US 10218353 Ki > 6370 nM T73475 CV5X8A 10224181 IC50 > 30000 nM T73475 C7T0WH 10229644 IC50 = 8570 nM T73475 CO8M7Q 10239526 Ki > 6370 nM T73475 CEO4X5 10239762 Ki > 6370 nM T73475 CU7TQ3 10239803 Ki > 6370 nM T73475 CBM0Y4 10252411 Ki < 100 nM T73475 C2V4MP 10253549 IC50 = 3245 nM T73475 CB6SE4 10256227 IC50 = 40 nM T73475 C0CE3N 10269452 IC50 = 4800 nM T73475 C0QS9V 10269453 IC50 = 590 nM T73475 CR7JN6 10279317 Ki = 79 nM T73475 C3IG0K 10280852 IC50 > 10000 nM T73475 CR48SA 10289842 Ki > 6370 nM T73475 CO60CU 10290029 Ki > 6370 nM T73475 CE1KM9 10311498 Ki > 6370 nM T73475 CJ15OB 10311501 Ki > 6370 nM T73475 C5F0EV 10311947 Ki > 6370 nM T73475 C7G6QW 10312268 Ki > 6370 nM T73475 CQ5IT9 10312372 Ki > 6370 nM T73475 CIDW49 10319098 Ki > 6368 nM T73475 CG23FV 10320328 IC50 = 5400 nM T73475 CJWH74 10321975 Ki > 6368 nM T73475 CQH5D4 10324032 IC50 = 5.9 nM T73475 C94ANQ 10347529 IC50 = 845 nM T73475 C9FU5G 10362663 IC50 = 909 nM T73475 CH89GT 10365752 IC50 = 3.6 nM T73475 CI0T8K 10366352 Ki > 6368 nM T73475 C6WZ4F 10367355 IC50 = 2424 nM T73475 CFKA79 10395015 Ki = 834 nM T73475 CS32HR 10435935 IC50 = 1.5 nM T73475 C5WV1N 10439082 Ki = 1336 nM T73475 CA7DM9 10474389 IC50 = 500 nM T73475 CNQZ36 10483139 Ki > 10000 nM T73475 C9XC8Y 10493383 IC50 = 2100 nM T73475 C6KD0A 10498747 IC50 = 23 nM T73475 C36OMW 10502172 IC50 = 1400 nM T73475 C5V8HJ 10502382 IC50 < 24 nM T73475 CSN17G 10502708 IC50 = 4200 nM T73475 CBNM82 10503128 IC50 = 105 nM T73475 C9LJR5 10503737 IC50 = 54 nM T73475 C2C7TE 10504472 IC50 = 450 nM T73475 C6D7JF 10506147 IC50 = 36000 nM T73475 CBT12Q 10522080 IC50 = 1082 nM T73475 CC2F5Y 10522311 IC50 = 821 nM T73475 CZ36JW 10523383 IC50 = 16000 nM T73475 CQEH42 10524134 IC50 = 263 nM T73475 CYU87N 10524260 IC50 = 612 nM T73475 COT07L 10525329 IC50 = 14000 nM T73475 C61GSD 10525562 IC50 = 642 nM T73475 C14XUW 10526101 IC50 = 1522 nM T73475 CJK6G1 10526509 IC50 = 420 nM T73475 CWLD37 10526788 IC50 = 7100 nM T73475 CHS9Q5 10527785 IC50 > 10000 nM T73475 CJ0D7G 10528505 IC50 = 1018 nM T73475 CO2R0P 10544323 IC50 = 10000 nM T73475 C4PK0U 10549114 IC50 = 30 nM T73475 C4TA1K 10549256 IC50 = 60 nM T73475 CHCI01 10549577 IC50 = 620 nM T73475 C2HJ1U 10549764 IC50 = 1695 nM T73475 CRHP20 10550304 IC50 = 2173 nM T73475 C7WQ5Z 10550399 IC50 = 140 nM T73475 CNQ75F 10551139 IC50 = 6086 nM T73475 CCH0K3 10551483 IC50 = 908 nM T73475 C5UD0A 10551910 IC50 = 100000 nM T73475 CNE73L 10552476 IC50 = 3290 nM T73475 CI8XG0 10554869 IC50 = 6800 nM T73475 CT7O9M 10569678 IC50 = 4500 nM T73475 C8RWE4 10569743 IC50 = 31000 nM T73475 CE14GM 10570702 IC50 = 7200 nM T73475 CS9Y3Q 10573446 IC50 = 520 nM T73475 C61IUN 10574937 IC50 = 183 nM T73475 C9L5OM 10579282 IC50 = 123 nM T73475 CIUO27 10593253 IC50 = 2546 nM T73475 CUTS47 10594564 IC50 = 7000 nM T73475 CN4Y6H 10594565 IC50 = 19000 nM T73475 CYNC76 10596158 IC50 = 11000 nM T73475 C0R8ND 10599533 IC50 = 710 nM T73475 CQCW86 10599579 IC50 = 785 nM T73475 CW18QK 10599594 IC50 = 27 nM T73475 CR1JI4 10600645 IC50 = 3400 nM T73475 C6RH4O 10601640 IC50 = 1200 nM T73475 CG32FM 10613145 IC50 = 1200 nM T73475 CZD9B3 10617580 IC50 = 1102 nM T73475 CL02BO 10618584 IC50 = 4500 nM T73475 C0JGS3 10621776 IC50 > 10000 nM T73475 CL5QN9 10622296 IC50 = 710 nM T73475 CL62YC 10622822 IC50 = 354 nM T73475 CZJB31 10622970 IC50 = 2694 nM T73475 C98KGO 10625860 IC50 = 1134 nM T73475 CL43CO 10627365 IC50 = 716 nM T73475 C7KGM3 10642071 IC50 = 1058 nM T73475 CWRY91 10642128 IC50 = 537 nM T73475 CI2QB9 10642965 IC50 = 381 nM T73475 C2O1XM 10647817 IC50 = 1100 nM T73475 C5RWF4 10648802 IC50 = 1283 nM T73475 C27QHB 10663143 IC50 = 2390 nM T73475 CGSX70 10664302 IC50 = 1860 nM T73475 C97KZU 10665624 IC50 = 4800 nM T73475 CF0E6H 10668745 IC50 = 7900 nM T73475 C8HK0C 10669534 IC50 = 1460 nM T73475 CAI72H 10670246 IC50 = 4900 nM T73475 CY6QC1 10670819 IC50 = 2690 nM T73475 CPG5O2 10671155 IC50 = 416 nM T73475 C09LJR 10671827 IC50 = 401 nM T73475 CXTP56 10688727 IC50 = 82 nM T73475 C0OJ9C 10689683 IC50 = 2200 nM T73475 CSA80H 10692194 IC50 = 8700 nM T73475 CS5CL7 10692307 IC50 = 39 nM T73475 CR5KF8 10692994 IC50 = 100000 nM T73475 CDI12G 10693559 IC50 = 17 nM T73475 CB70DA 10693592 IC50 = 9800 nM T73475 CVML68 10693881 IC50 = 8500 nM T73475 CW6CF7 10696226 IC50 = 2700 nM T73475 C6MWX8 10696713 IC50 = 22050 nM T73475 C4IWF2 10714988 IC50 = 7400 nM T73475 CO9KV7 10715115 IC50 = 89 nM T73475 CE1D6G 10716217 IC50 < 100 nM T73475 C0ZX6T 10717308 IC50 = 3100 nM T73475 C7OSW8 10718200 IC50 = 610 nM T73475 CI64YZ 10718883 IC50 = 824 nM T73475 C35MRE 10719092 IC50 = 785 nM T73475 C51DZG 10737732 IC50 = 7500 nM T73475 C1LS5U 10738104 IC50 = 240 nM T73475 CL74TG 10738165 IC50 = 53 nM T73475 C76ANK 10739335 IC50 = 483 nM T73475 C0T2VK 10740460 IC50 = 787 nM T73475 CKJD45 10741133 IC50 = 78000 nM T73475 CL64BU 10741592 IC50 = 16 nM T73475 C4MQ8L 10742072 IC50 = 840 nM T73475 CHW23E 10742387 IC50 = 79 nM T73475 CCH94Q 10743507 IC50 = 1890 nM T73475 C9ILP3 10745718 IC50 = 15000 nM T73475 CE09PI 10757715 IC50 = 4300 nM T73475 C68THN 10763851 IC50 = 922 nM T73475 CAG53Y 10764489 IC50 = 509 nM T73475 C0ZJB9 10764600 IC50 = 27680 nM T73475 CJE76M 10764871 IC50 = 7400 nM T73475 CQ0KM4 10765140 IC50 = 790 nM T73475 C7Q2EM 10767236 IC50 = 3000 nM T73475 CLAP90 10785969 IC50 > 1000 nM T73475 C2FA7J 10787997 IC50 = 3500 nM T73475 C16XQR 10788211 IC50 = 1400 nM T73475 C0DFB9 10788617 IC50 = 170 nM T73475 CNAE08 10788733 IC50 = 2100 nM T73475 CKV2O8 10789493 IC50 = 483 nM T73475 CM74LH 10789594 IC50 > 1000 nM T73475 C45UGJ 10789671 IC50 = 850 nM T73475 C9NZ4W 10789711 IC50 = 502 nM T73475 CWCD73 10805054 IC50 = 12300 nM T73475 CN8I3Z 10808172 IC50 > 9994 nM T73475 CT1AI4 10810573 IC50 = 2700 nM T73475 CV3ZA5 10812444 IC50 = 4350 nM T73475 CZB7L2 10812929 IC50 < 100 nM T73475 C4TF0K 10813874 IC50 = 490 nM T73475 CCIL63 10813879 IC50 = 680 nM T73475 CS7BY4 10816934 IC50 = 8600 nM T73475 CX2E1C 10829071 IC50 = 313 nM T73475 C3AI5Z 10831752 IC50 = 22000 nM T73475 CLK9P7 10832592 IC50 = 12848 nM T73475 CF50HD 10832925 IC50 = 77000 nM T73475 C5OG4U 10833497 IC50 = 5600 nM T73475 C48PYQ 10836923 IC50 = 497 nM T73475 CH8OV4 10837276 IC50 = 110 nM T73475 CF40VH 10837557 IC50 = 1700 nM T73475 CY4J9A 10838149 IC50 = 2400 nM T73475 C3UCL2 10854279 IC50 = 1500 nM T73475 CAU0I3 10885834 IC50 = 3950 nM T73475 CXHA75 10928874 IC50 = 9870 nM T73475 CG2DK0 11016448 IC50 = 1740 nM T73475 CODQ51 11016616 IC50 = 3660 nM T73475 C9RU4I 11059620 IC50 = 5650 nM T73475 C1N5PT 11070986 IC50 = 4370 nM T73475 C18EIZ 11071831 IC50 = 2650 nM T73475 CY1SR9 11113744 IC50 > 10000 nM T73475 C2YBQ7 11134935 IC50 = 8510 nM T73475 C43ONW 11202395 Ki > 636 nM T73475 CO7T3M 11261246 IC50 > 10000 nM T73475 CP17ID 11284983 IC50 = 866 nM T73475 C1IW7N 11292680 IC50 > 1000 nM T73475 C8C5AV 11294179 Ki > 10000 nM T73475 CLH50U 11318841 IC50 = 458 nM T73475 C0XR3B 11330861 IC50 = 1640 nM T73475 CQH57S 11342435 IC50 = 1100 nM T73475 C9ABX8 11397130 Ki > 6368 nM T73475 COS67B 11456566 IC50 = 3010 nM T73475 CJ46KN 11508259 Ki = 9000 nM T73475 C5VUM2 11517085 Ki > 50000 nM T73475 CHV2G1 11575995 Ki > 10000000 nM T73475 CNY92D 11640694 Ki > 60000 nM T73475 CK9F4P 11673778 IC50 > 50000 nM T73475 C28WNK 11682752 Ki = 295000 nM T73475 C3U6ZR 11697504 Ki > 50000 nM T73475 C7CED0 11733417 IC50 > 10000 nM T73475 CO8QT0 11753905 Ki = 6 nM T73475 CKM6P2 11795228 IC50 = 15740 nM T73475 CCSD72 11795621 IC50 = 41 nM T73475 C47OIA 11797154 IC50 = 920 nM T73475 CJ4VL3 11797382 IC50 > 1000 nM T73475 CCD4W2 11797992 IC50 = 2093 nM T73475 CHQR96 11798386 IC50 = 1032 nM T73475 CQ9HE2 11811551 IC50 = 4240 nM T73475 CLW3F1 11812791 IC50 > 10000 nM T73475 C02BWA 11967143 Ki > 2000 nM T73475 CB80OT 12000718 IC50 > 20000 nM T73475 C43PJZ 12000720 IC50 > 20000 nM T73475 C1AJO7 13968141 IC50 > 300000 nM T73475 CA2H8V 14303060 IC50 = 4100 nM T73475 CGH19T 15296844 IC50 > 300000 nM T73475 CB3A4Z 15941413 Ki = 48500 nM T73475 CA40FE 15941550 Ki = 31000 nM T73475 CM3D1L 15941553 Ki = 39000 nM T73475 CQ0ZL7 15941677 Ki = 18000 nM T73475 C6R1LD 15985818 IC50 = 961 nM T73475 CQS0F5 16719301 IC50 > 10000 nM T73475 C75XDI 16730519 IC50 = 1700 nM T73475 C2W1VA 16739287 Ki > 6000 nM T73475 C3S2TQ 17754305 IC50 > 40000 nM T73475 CSY0N8 18394511 IC50 > 300000 nM T73475 CK8MP3 20620240 Ki = 8600 nM T73475 CPC4G6 20620273 Ki > 10000 nM T73475 CPK09X 20651316 IC50 = 23 nM T73475 CG1BD4 20689551 IC50 > 10000 nM T73475 CAS84B 22004289 Ki = 237 nM T73475 C1MCG7 22004293 Ki = 605 nM T73475 C36WFA 22096205 IC50 > 100000 nM T73475 CZT64B 22484431 Ki > 10000 nM T73475 CD3U8A 23627203 Ki > 2500 nM T73475 C3TWS6 24178109 Ki = 1600 nM T73475 C5M3YW 24799779 Ki = 110000 nM T73475 CFL04M 24881245 IC50 > 300000 nM T73475 CLIC14 24881246 IC50 > 300000 nM T73475 C4FI5C 24901479 IC50 = 71000 nM T73475 CAQ9Z1 25022681 Ki > 6368 nM T73475 CA86UE 25049752 Ki = 823 nM T73475 C82NLV 25049754 Ki = 3000 nM T73475 C6QFV4 25049756 Ki = 4000 nM T73475 CU6M9K 25060725 IC50 = 20000 nM T73475 CF7X2P 25060975 IC50 = 32000 nM T73475 CVR52U 25066764 IC50 > 22 nM T73475 CA5DJ4 25138228 Ki = 128000 nM T73475 CX6D9J 25138245 Ki > 3000 nM T73475 C7A6JQ 25138250 Ki = 33000 nM T73475 C6N7EQ 25138258 Ki = 1336 nM T73475 C7AD1J 25138259 Ki = 311 nM T73475 CJ9TQ2 25138260 Ki = 1527 nM T73475 CUT8I7 25138261 Ki = 2992 nM T73475 CBD9X6 25138262 Ki = 3311 nM T73475 C8LX1S 25138263 Ki = 1145 nM T73475 C3OV1L 25138264 Ki > 6368 nM T73475 C92WVM 25138265 Ki = 811 nM T73475 CMCS41 25138266 Ki > 6368 nM T73475 C1FJV5 25138267 Ki > 6368 nM T73475 C9N6WT 25138268 Ki > 6368 nM T73475 CF4QI1 25138269 Ki > 6368 nM T73475 C6P5UL 25138270 Ki > 6368 nM T73475 CQE0L7 25138271 Ki = 2647 nM T73475 C59XWU 25138272 Ki = 726 nM T73475 C1TNQ3 25141117 IC50 = 475 nM T73475 CR35QP 25144971 IC50 > 10000 nM T73475 C0Y5BC 25145683 IC50 > 2500 nM T73475 CHR2P1 25183768 Ki > 25000 nM T73475 C6AR8O 42623563 IC50 > 100000 nM T73475 CX0VP7 42623564 IC50 > 100000 nM T73475 CPO1Z3 44123600 IC50 = 3025 nM T73475 CCI64J 44224245 IC50 = 7830 nM T73475 CAR34Y 44263877 IC50 > 10000 nM T73475 CEV08N 44263913 IC50 = 737 nM T73475 C5ZI0X 44263926 IC50 = 88 nM T73475 CO3C1E 44263994 IC50 = 2780 nM T73475 C9XJ7U 44264020 IC50 = 10000 nM T73475 C6L0MJ 44264021 IC50 = 369 nM T73475 CJ1WE7 44264036 IC50 = 776 nM T73475 C50QFR 44264375 IC50 = 3460 nM T73475 C6YT3K 44280285 Ki = 1420 nM T73475 C8XUJ3 44280321 Ki = 3225 nM T73475 CC2O3U 44280323 Ki = 78 nM T73475 CM2TZ4 44280335 Ki = 114 nM T73475 CIE09F 44280336 Ki = 5 nM T73475 CA1V6Y 44280345 Ki = 18 nM T73475 CI9L2E 44280411 Ki > 620 nM T73475 C96NMF 44287796 IC50 = 70 nM T73475 CQ5IG7 44287805 IC50 = 33 nM T73475 CHOV34 44287806 IC50 = 50 nM T73475 CYAG29 44287899 IC50 = 2 nM T73475 CX5QB3 44287917 IC50 = 10 nM T73475 CCM31I 44288043 IC50 = 10 nM T73475 C1YT7H 44288071 IC50 = 10 nM T73475 CF2DZ9 44288091 IC50 = 3.1 nM T73475 CMY2N4 44288092 IC50 = 1 nM T73475 CCS20R 44288093 IC50 = 1 nM T73475 C2Y0PK 44302023 IC50 > 10000 nM T73475 C5S3UO 44302024 IC50 > 10000 nM T73475 C8ERW6 44302042 IC50 = 8540 nM T73475 CWB83G 44302076 IC50 = 5150 nM T73475 CY1J9U 44302096 IC50 = 9128 nM T73475 CW94ZQ 44302164 IC50 > 10000 nM T73475 CQ54PZ 44302166 IC50 = 500 nM T73475 C9U3XT 44302167 IC50 = 5000 nM T73475 C5X1WY 44302183 IC50 > 10000 nM T73475 C7G3BN 44302200 IC50 = 24061 nM T73475 C70QWV 44302327 IC50 = 40000 nM T73475 CZP20C 44302339 IC50 = 7069 nM T73475 CO73BW 44302357 IC50 > 10000 nM T73475 CNL4E2 44302361 IC50 = 20 nM T73475 CCW65Y 44302378 IC50 = 2000 nM T73475 CYG80V 44302385 IC50 = 10000 nM T73475 C7ZBR4 44302396 IC50 = 1000 nM T73475 C8S5WT 44302397 IC50 = 2000 nM T73475 CPC25G 44302409 IC50 = 7960 nM T73475 C4QL0I 44302411 IC50 = 3000 nM T73475 C4NDA2 44302416 IC50 = 20498 nM T73475 C24ZWF 44302429 IC50 > 10000 nM T73475 CYL71W 44302432 IC50 = 2000 nM T73475 C5H6OV 44302627 IC50 = 15147 nM T73475 C6QR7C 44302634 IC50 > 10000 nM T73475 CG8KJ0 44302661 IC50 = 5470 nM T73475 CX1M3Q 44302666 IC50 = 6340 nM T73475 C36CQP 44302952 IC50 = 4450 nM T73475 CLH14M 44305978 IC50 = 5.7 nM T73475 CZ49UN 44305988 IC50 = 2.6 nM T73475 C6I8JA 44306058 IC50 = 25 nM T73475 CB5EY3 44306200 IC50 = 4.2 nM T73475 C0YOH1 44306202 IC50 = 2.5 nM T73475 CMA39E 44306203 IC50 = 1.6 nM T73475 CL58OS 44306208 IC50 = 900 nM T73475 CAY2S4 44306209 IC50 = 110 nM T73475 C27NJX 44306277 IC50 = 180 nM T73475 C6O1AN 44306279 IC50 = 2.8 nM T73475 C89IQW 44318090 IC50 = 3640 nM T73475 CLQ23M 44321485 Ki = 210 nM T73475 CT0O7Y 44321602 Ki = 4 nM T73475 CV8T3N 44321783 Ki = 370 nM T73475 C4E8GU 44321802 Ki = 2100 nM T73475 C7Z4DQ 44321887 Ki = 117 nM T73475 CFJ20T 44321932 Ki = 605 nM T73475 CW9S1N 44321967 Ki = 1800 nM T73475 CI5X0G 44339523 IC50 = 4.2 nM T73475 CB9K8T 44339536 IC50 = 3.3 nM T73475 C2R3XN 44339554 IC50 = 13 nM T73475 C2CRY1 44339556 IC50 = 8.6 nM T73475 CTBU53 44339564 IC50 = 29 nM T73475 C58OSK 44339567 IC50 = 4.2 nM T73475 CX2KJ3 44339574 IC50 = 68 nM T73475 CEK3G0 44339588 IC50 = 5.7 nM T73475 C7ZR6H 44339589 IC50 = 220 nM T73475 C0WP9C 44339590 IC50 = 8 nM T73475 C5C2LI 44339654 IC50 = 4.3 nM T73475 C2SZB1 44342614 IC50 = 20 nM T73475 CQ60YD 44360219 IC50 = 330 nM T73475 CT4C6P 44360260 IC50 = 17651 nM T73475 CY5I3O 44360286 IC50 = 637 nM T73475 C40OCB 44360287 IC50 = 38 nM T73475 C3IW9L 44360784 IC50 = 18 nM T73475 CGQ92A 44364037 IC50 = 12040 nM T73475 CN4T7Q 44364119 IC50 = 21420 nM T73475 CH4TE7 44364121 IC50 = 7136 nM T73475 CPE91Y 44364122 IC50 = 10471.29 nM T73475 C1F8XN 44364249 IC50 = 3162.28 nM T73475 CWM47H 44364250 IC50 = 10690 nM T73475 C3TPO7 44364266 IC50 = 21380 nM T73475 C90CYD 44367175 IC50 = 5235 nM T73475 C2DV0R 44367276 IC50 = 294 nM T73475 C5BAW2 44367284 IC50 = 1792 nM T73475 C2YG5E 44367285 IC50 = 6724 nM T73475 CUDF82 44367309 IC50 = 2083 nM T73475 C3EV2A 44384940 IC50 > 50000 nM T73475 C0XE8K 44384941 IC50 > 50000 nM T73475 C3IJO9 44384994 IC50 > 50000 nM T73475 CWGQ46 44404503 IC50 = 534 nM T73475 CLXM58 44404504 IC50 = 1260 nM T73475 C1K3QM 44406655 IC50 = 200 nM T73475 C6YG5S 44406678 IC50 > 1000 nM T73475 CT5PC9 44422672 IC50 = 150 nM T73475 CS9D5U 44422720 IC50 = 450 nM T73475 CNWM05 44422723 IC50 = 2000 nM T73475 C58LAY 44422724 IC50 = 1400 nM T73475 CDQU41 44422736 IC50 = 20000 nM T73475 CVUB56 44422737 IC50 = 2900 nM T73475 CB8G2W 44422743 IC50 = 1100 nM T73475 CFX42T 44422744 IC50 = 50000 nM T73475 C9EL7F 44422749 IC50 = 130000 nM T73475 CJN1K9 44439853 Ki > 6370 nM T73475 CV58YW 44441018 Ki > 6368 nM T73475 CV85PN 44441019 Ki > 6368 nM T73475 C5O2WK 44441020 Ki > 6368 nM T73475 CU67WS 44441021 Ki > 6368 nM T73475 CXZ53B 44441022 Ki > 6368 nM T73475 C8S7UT 44441023 Ki > 6368 nM T73475 CT4PZ9 44441024 Ki > 6368 nM T73475 CU9GE6 44441025 Ki > 6368 nM T73475 CB2IT4 44441026 Ki > 6368 nM T73475 CN4X2F 44441027 Ki > 6368 nM T73475 CPF45Y 44441028 Ki > 6368 nM T73475 CAM23N 44441029 Ki > 6368 nM T73475 C23BPG 44441030 Ki = 5371 nM T73475 C5YMT6 44441031 Ki > 6368 nM T73475 C9A6GJ 44441032 Ki > 6368 nM T73475 CYSU19 44441033 Ki > 6368 nM T73475 C7T6EI 44445816 IC50 = 1819.7 nM T73475 CG9JS8 44445817 IC50 = 7585.78 nM T73475 CBX8S1 44445818 IC50 = 2570.4 nM T73475 CCYD65 44445819 IC50 = 1584.89 nM T73475 C3XG5N 44445820 IC50 = 2290.87 nM T73475 C58PEZ 44445821 IC50 = 9120.11 nM T73475 CRS83Q 44445822 IC50 = 309.03 nM T73475 CPO4U0 44445823 IC50 = 7413.1 nM T73475 CEQ8O0 44445824 IC50 = 851.14 nM T73475 CEOB52 44445825 IC50 = 446.68 nM T73475 CKEG37 44445826 IC50 = 2570.4 nM T73475 CHO12U 44445827 IC50 = 1000 nM T73475 C85EBJ 44445828 IC50 = 10964.78 nM T73475 CIJ70S 44445829 IC50 = 1202.26 nM T73475 COYD74 44445830 IC50 = 10964.78 nM T73475 CJ2BU5 44563487 IC50 = 6150 nM T73475 CHQG04 44576676 Ki = 10000 nM T73475 CR65DO 44576708 Ki = 1800 nM T73475 C9CB2Z 44576709 Ki = 602 nM T73475 C2QFY7 44576710 Ki = 625 nM T73475 C0BQV5 44576711 Ki = 5500 nM T73475 CU2IP7 44576753 Ki = 6600 nM T73475 C2QE3W 44576754 Ki = 6000 nM T73475 C8QHV1 44576806 Ki = 8600 nM T73475 C93LDF 44576807 Ki = 289 nM T73475 C9T2KO 44576808 Ki = 4800 nM T73475 C4RL6Y 44576809 Ki = 3000 nM T73475 CJ41MB 44576851 Ki = 7000 nM T73475 C9PUW2 44576877 Ki = 5000 nM T73475 C1F8WD 44576903 Ki = 3100 nM T73475 CTA01K 44576904 Ki = 2200 nM T73475 CK68GT 44580539 Ki = 75 nM T73475 CXIY57 44580801 Ki = 4617000 nM T73475 C0OA8Y 44580802 Ki > 10000000 nM T73475 CNC4D7 44581071 Ki = 1500000 nM T73475 CDF48U 44581111 Ki > 10000000 nM T73475 C56WVI 46184724 Ki = 6000 nM T73475 CL2U4Z 46829322 Ki = 1500 nM T73475 CH0Z1E 46844314 Ki > 40000 nM T73475 C20BTY 46856241 Ki = 3769 nM T73475 C5L8GF 46871738 IC50 > 10000 nM T73475 C0S9WB 46919610 Ki = 47000 nM T73475 C2S7PK 46942365 Ki = 2000 nM T73475 C7XW1Q 50907084 Ki = 344 nM T73475 C8RL5Q 50907292 Ki = 4000 nM T73475 CAS94N 51346773 Ki = 11000 nM T73475 CP65WT 51346774 Ki = 26000 nM T73475 C5OIA2 51346775 Ki = 35000 nM T73475 CU2SX3 51355576 Ki > 10000 nM T73475 CLA96C 53232689 Ki = 970 nM T73475 C3BGW0 53233015 Ki = 18100 nM T73475 CWH47R 53319228 Ki = 984 nM T73475 CI3WL5 53323418 Ki = 120000 nM T73475 C6Y2EV 53374826 IC50 > 100000 nM T73475 C3LF0P 54580544 Ki > 10000 nM T73475 CVO09J 54581546 Ki = 3000 nM T73475 CD09BZ 54582543 IC50 > 10000 nM T73475 CK52YD 54583511 Ki = 6000 nM T73475 CG37UX 54587429 Ki = 7100 nM T73475 CL9SC3 54587769 Ki = 13500 nM T73475 CHS01Z 54669766 Ki = 160000 nM T73475 C7E9SG 54757202 Ki = 116000 nM T73475 C62FZC 56835063 IC50 = 57700 nM T73475 C0L2TS 56835169 IC50 = 39000 nM T73475 CQU16V 57339411 Ki = 10700 nM T73475 C6LM3B 57339412 Ki = 7000 nM T73475 CWH7V8 57561293 IC50 > 40000 nM T73475 CY1N3J 57792153 IC50 = 1242 nM T73475 CCKD80 58307579 Ki > 25000 nM T73475 CMW3O0 71451330 Ki > 200 nM T73475 C9QS6E 71456659 Ki > 2000 nM T73475 C1U0FV 71601333 IC50 = 1150 nM T73475 C6KEH0 71680708 Ki > 25000 nM T73475 C7DMX5 71680709 Ki > 25000 nM T73475 CFPM82 71680710 Ki > 12000 nM T73475 C9ZOM7 71680866 Ki = 4000 nM T73475 CQ68LT 71680868 Ki > 100000 nM T73475 CFH2V0 71681183 Ki = 4100 nM T73475 CV3X1T 71682766 Ki > 20000 nM T73475 C5EAO8 71682767 Ki > 100000 nM T73475 C80EYX 71682913 Ki > 50000 nM T73475 C41BYG 71682915 Ki > 20000 nM T73475 C93XEI 71682916 Ki = 36000 nM T73475 CQ29PJ 71682917 Ki > 200000 nM T73475 CFWN65 71683062 Ki = 5700 nM T73475 C50SID 71817098 Ki = 18500 nM T73475 C38IDL 73345835 Ki = 11 nM T73475 CW01EA 73349535 IC50 > 100000 nM T73475 C8ROG3 73350414 Ki = 91 nM T73475 CF7AB2 73350415 Ki = 50 nM T73475 C2PFM4 73351930 Ki = 230 nM T73475 CI09CY 73354906 Ki = 12 nM T73475 C6H5TU 73354941 Ki = 6000 nM T73475 CGQ8F3 86287515 IC50 = 100000 nM T73475 CJ37XE 86287516 IC50 = 100000 nM T73475 COV8I9 86291010 IC50 = 1008 nM T73475 CRT54C 101910871 IC50 = 100000 nM T73475 CYA92R 130282633 IC50 = 180 nM T73475 CO3QE2 130282636 IC50 = 210 nM T73475 CTN42D 132941363 IC50 = 100000 nM T73475 C83FAY 134130294 Ki = 3760 nM T73475 CHV2U1 135438561 IC50 > 10000 nM T73475 CA5JR6 136054481 IC50 > 10000 nM T73475 CV47JN 136054485 IC50 > 10000 nM T73475 CZ48WO 136054487 IC50 > 10000 nM T73475 C8FGT0 136054495 IC50 > 10000 nM T73475 CG70BZ 136054516 IC50 = 30 nM T73475 CSM57W 136054520 IC50 = 2000 nM T73475 CXNG40 136118011 Ki = 1000 nM T73475 C1IOH9 136118012 Ki > 6368 nM T73475 CIEW62 136380958 IC50 = 1000 nM T73475 C9HS7J 137287436 IC50 = 7.3 nM T73475 C0I6RH 137632487 IC50 = 1102 nM T73475 CZ8H6N 137661550 IC50 = 100000 nM T73475 CZ25LW 155512044 IC50 = 100000 nM T73475 D02EFQ 10549609 IC50 = 11000 nM T73475 D03AMR 9849669 Ki = 660 nM T73475 D04GOO 10111838 IC50 > 100000 nM T73475 D04PAW 16216218 IC50 = 44000 nM T73475 D04VPH 45376872 IC50 > 22000 nM T73475 D06EHW 11625778 IC50 > 5000 nM T73475 D06HSC 136117931 IC50 = 15000 nM T73475 D07DRT 46175162 Ki = 3000 nM T73475 D07GEL 10344307 Ki = 0.8 nM T73475 D07SPC 24857837 Ki = 2800 nM T73475 D08ELY 9838786 IC50 = 1100 nM T73475 D09GIL 66160 IC50 > 50000 nM T73475 D09ZOA 25049753 Ki = 5000 nM T73475 D0A4TC 446504 IC50 = 106 nM T73475 D0B0UI 44428664 IC50 = 100000 nM T73475 D0B3UN 44580458 Ki = 626 nM T73475 D0BI8T 44288042 IC50 = 0.23 nM T73475 D0G3YZ 11391583 IC50 > 98000 nM T73475 D0H6CK 10160968 Ki = 18 nM T73475 D0K4TI 49292 IC50 > 50000 nM T73475 D0N6CD 10565532 IC50 = 290 nM T73475 D0N8YA 159596 IC50 > 100000 nM T73475 D0Q4TA 10044321 IC50 > 50000 nM T73475 D0Q9LC 44385624 IC50 > 50000 nM T73475 D0R2BO 194777 IC50 = 8.3 nM T73475 D0W2UK 6914621 Ki = 259 nM T73475 D0XK7G 10445302 Ki = 4000 nM T73475 D0Y5IQ 44255320 IC50 = 5000 nM T73475 D0Y7NV 2220392 IC50 > 50000 nM T03896 D09ZZW 503536 IC50 = 1500 nM T03896 C6IQV0 482174 IC50 = 5700 nM T03896 CY61LO 487910 IC50 = 1700 nM T03896 C6K5JV 487911 IC50 = 16000 nM T03896 C3J5VH 487912 IC50 = 1000 nM T03896 CZNK70 487918 IC50 = 330 nM T03896 CDN3F2 487919 IC50 = 1630 nM T03896 CT76XW 487920 IC50 = 2100 nM T03896 CVA82G 487921 IC50 = 460 nM T03896 CBR46W 487922 IC50 = 1400 nM T03896 CAJ64Q 490750 IC50 < 1000 nM T03896 CMO49H 491114 IC50 = 4300 nM T03896 COB17R 492544 IC50 > 50000 nM T03896 C68MZE 492548 IC50 > 100000 nM T03896 C4JO9E 492549 IC50 = 3280 nM T03896 C1JEY2 492550 IC50 = 300 nM T03896 CRML27 492552 IC50 = 380 nM T03896 C84QRW 493418 IC50 = 5700 nM T03896 CY1WF7 497453 IC50 = 3000 nM T03896 C43PXV 503499 IC50 = 2400 nM T03896 C2BSI5 503516 IC50 = 14000 nM T03896 CFRT87 503517 IC50 = 5400 nM T03896 C3JB0U 503520 IC50 = 13000 nM T03896 CA72XJ 503521 IC50 = 5200 nM T03896 CF14KO 503522 IC50 = 7400 nM T03896 CH18YP 503523 IC50 = 4600 nM T03896 CG6T1D 503524 IC50 = 4100 nM T03896 CLY7T8 503525 IC50 = 750 nM T03896 C37MIA 503526 IC50 = 1000 nM T03896 C8U2AD 503527 IC50 = 12000 nM T03896 CO6R4G 503528 IC50 = 2000 nM T03896 CHA5F8 503529 IC50 > 50000 nM T03896 C41DVG 503530 IC50 = 21000 nM T03896 C5XRJ6 503531 IC50 = 1200 nM T03896 CI1V6W 503532 IC50 > 50000 nM T03896 C84DXH 503533 IC50 = 1400 nM T03896 C7R3CM 503534 IC50 = 2000 nM T03896 CCMU16 503535 IC50 = 3000 nM T03896 C1E4IO 504181 IC50 = 2700 nM T03896 CEJ6U1 504182 IC50 = 1800 nM T03896 CZDS90 504183 IC50 = 1600 nM T03896 C04ONL 504184 IC50 = 2200 nM T03896 C65XPH 504185 IC50 = 11000 nM T03896 CRZN68 504186 IC50 = 42000 nM T03896 CK8CA2 504187 IC50 > 60000 nM T03896 C01MYV 504188 IC50 = 5800 nM T03896 C4C5WD 504189 IC50 = 4300 nM T03896 CIB52E 504190 IC50 = 230 nM T03896 CQ6L1G 504191 IC50 = 12000 nM T03896 C4CW5A 504192 IC50 > 60000 nM T03896 C09ACU 504193 IC50 > 60000 nM T03896 C7T0AD 504194 IC50 = 1300 nM T03896 C7VZY1 504195 IC50 > 60000 nM T03896 CU4EK0 504196 IC50 = 3600 nM T03896 COUS53 504197 IC50 = 5300 nM T03896 CTE3B4 504198 IC50 = 7700 nM T03896 CT81MP 504676 IC50 = 3500 nM T03896 C9FI5K 504680 IC50 = 10600 nM T03896 C8IFN4 504681 IC50 = 31000 nM T03896 CV6OY3 506523 IC50 = 1400 nM T03896 CQX7S4 506524 IC50 = 390 nM T03896 CXD73I 506525 IC50 = 1800 nM T03896 C6ANI5 506528 IC50 = 9000 nM T03896 CRU30I 507613 IC50 = 900 nM T03896 CI8SQ4 511361 IC50 > 50000 nM T03896 C02LPN 511362 IC50 = 30000 nM T03896 CJIW67 511363 IC50 = 13000 nM T03896 C3KG1M 511364 IC50 = 43000 nM T03896 CU85HK 511365 IC50 = 10700 nM T03896 C20EKN 511366 IC50 = 5900 nM T03896 C3FX8J 511367 IC50 = 31000 nM T03896 C4DEY1 511368 IC50 = 3700 nM T03896 CC2J9M 511369 IC50 = 5600 nM T03896 CIU5M2 511370 IC50 = 11000 nM T03896 C5CG4I 511371 IC50 = 5000 nM T03896 CTO87P 511372 IC50 = 2700 nM T03896 C5BJ6S 511373 IC50 = 26000 nM T03896 CDWB40 511374 IC50 = 15000 nM T03896 CDH29C 511375 IC50 = 31000 nM T03896 C8ZJD7 511376 IC50 = 31000 nM T03896 CJ56OH 513150 IC50 < 10000 nM T03896 C5BN4U 513891 IC50 = 12000 nM T03896 CVI54C 657065 IC50 = 1200 nM T03896 CUC54L 3008068 IC50 = 5000 nM T03896 CJ5NO6 3008069 IC50 = 34000 nM T03896 CQO9Y3 3008070 IC50 > 32000 nM T03896 CXM1K9 3008071 IC50 > 50000 nM T03896 CJ2NY3 3008418 IC50 = 20000 nM T03896 CIJ2T0 3008419 IC50 > 50000 nM T03896 CWD1X0 3008420 IC50 = 14000 nM T03896 C4K2JP 3008421 IC50 > 50000 nM T03896 CAN83S 3008422 IC50 = 13000 nM T03896 CMDQ27 4468931 IC50 = 1800 nM T03896 CK9WY1 5278824 IC50 = 100 nM T03896 C5MEQ4 5278825 IC50 = 110 nM T03896 C1F0AN 5278826 IC50 = 45 nM T03896 CV0O6S 5482516 IC50 = 15600 nM T03896 CEM30Z 5483089 IC50 = 8900 nM T03896 CJL21S 9853197 IC50 = 60 nM T03896 CJW4M9 9917616 IC50 = 11000 nM T03896 C39ZBC 10207572 IC50 = 30000 nM T03896 CGA86Z 10259200 IC50 = 12000 nM T03896 CJ46UK 10439772 IC50 = 420 nM T03896 COM8C5 21148125 IC50 = 16000 nM T03896 C1TW3V 22209806 IC50 > 50000 nM T03896 C8GVX3 22209808 IC50 > 50000 nM T03896 C6AS7E 22209811 IC50 = 3300 nM T03896 CLW13P 22209812 IC50 = 1700 nM T03896 C1TA6Z 22209813 IC50 = 440 nM T03896 CGUC83 22210989 IC50 = 58000 nM T03896 CV97ER 22210996 IC50 = 18000 nM T03896 C2BA1K 22211000 IC50 = 27000 nM T03896 C78AKX 22211010 IC50 > 100000 nM T03896 CL7M9B 22211011 IC50 = 32000 nM T03896 C1L8TE 22211012 IC50 = 18000 nM T03896 C0NYS5 22211016 IC50 = 50000 nM T03896 C67QJW 22211018 IC50 > 100000 nM T03896 CV9S2O 22211019 IC50 = 13000 nM T03896 C4UB6Q 22211020 IC50 = 14000 nM T03896 CBUV46 22211021 IC50 = 62000 nM T03896 CS9B7N 22211022 IC50 > 100000 nM T03896 CK81WO 25078062 IC50 = 3400 nM T03896 CYDW71 44268661 IC50 > 60000 nM T03896 C6S3AT 44268682 IC50 > 60000 nM T03896 CDJ0X4 44308299 IC50 > 100000 nM T03896 CIO1C2 44308345 IC50 > 100000 nM T03896 CX14BI 44308422 IC50 > 100000 nM T03896 CE3PS8 44308752 IC50 = 34000 nM T03896 CK2P5O 44375061 IC50 > 50000 nM T03896 C4CVW1 44375110 IC50 > 50000 nM T03896 C72KUL 44375154 IC50 = 9400 nM T03896 C1SBO9 44375192 IC50 > 50000 nM T03896 C42GUE 44375229 IC50 = 5300 nM T03896 CX76FI 44388198 IC50 = 350 nM T03896 CVW6O4 44399745 IC50 = 79432.82 nM T03896 CDRP83 44399750 IC50 = 50118.72 nM T03896 CW6NY8 44399751 IC50 = 5011.87 nM T03896 CM5W8Q 44399752 IC50 = 6309.57 nM T03896 C34WSP 44399753 IC50 = 10000 nM T03896 CE0T1O 44399754 IC50 = 1995.26 nM T03896 CT86CR 44399784 IC50 = 25118.86 nM T03896 C6GWS9 44399837 IC50 = 31622.78 nM T03896 C4AI1T 44399861 IC50 = 100000 nM T03896 CTX79F 44399866 IC50 = 25118.86 nM T03896 CP4KB7 44399867 IC50 = 794.33 nM T03896 C0WRU5 44399868 IC50 = 15848.93 nM T03896 C8JP2A 44399889 IC50 = 50118.72 nM T03896 CO4H3V 44399938 IC50 = 10000 nM T03896 CYH7F9 44399975 IC50 = 6309.57 nM T03896 CZRF38 44399976 IC50 = 6309.57 nM T03896 CATH48 44399977 IC50 = 6309.57 nM T03896 CL9NS3 44399978 IC50 > 199526.23 nM T03896 C9YO4K 44399979 IC50 > 199526.23 nM T03896 CX8M3O 44400003 IC50 = 39810.72 nM T03896 C4X1OG 44400004 IC50 = 19952.62 nM T03896 C5EV1S 44400005 IC50 = 158489.32 nM T03896 CFRU27 44400006 IC50 = 199526.23 nM T03896 C7FO3T 44400007 IC50 = 251188.64 nM T03896 CA6P2U 44400008 IC50 = 100000 nM T03896 CQP47M 44400009 IC50 = 7943.28 nM T03896 CCRB97 44400010 IC50 = 3981.07 nM T03896 CT40SR 44400033 IC50 = 31622.78 nM T03896 CA96HO 44400076 IC50 > 1000000 nM T03896 CX7O2Z 44400112 IC50 > 199526.23 nM T03896 C6Z5NC 44400113 IC50 > 199526.23 nM T03896 C6PCE5 44400114 IC50 = 31622.78 nM T03896 C95CRD 44400115 IC50 = 19952.62 nM T03896 CW5G3Z 73347065 IC50 > 50000 nM T03896 C6TNQ8 135412361 IC50 = 800 nM T03896 C53AWL 135434400 IC50 = 100 nM T96685 D04VIS 5318517 IC50 > 50000 nM T96685 D0X8ED 2327 IC50 = 5520 nM T96685 CHO1C9 57411333 IC50 = 790 nM T96685 CWDS87 57411452 IC50 = 50 nM T96685 C80DZY 57411679 IC50 = 10 nM T96685 CFK47B 67974063 IC50 = 2000 nM T96685 C2AZ4Y 67974101 IC50 > 400000 nM T96685 C5WEF0 67974104 IC50 = 25 nM T96685 C1TDA4 67974531 Ki = 2900 nM T96685 CKF7Q0 88537798 IC50 = 2000 nM T96685 C3RG6K 118714691 IC50 < 316.23 nM T96685 C1RE2H 127048545 IC50 = 3200 nM T96685 C49ZUL 127048546 IC50 = 790 nM T96685 CMI9A1 127048547 IC50 = 16000 nM T96685 CZ0C2N 127049887 IC50 = 630 nM T96685 C1JKC3 127049888 IC50 = 40 nM T96685 C13CQL 127049889 IC50 = 130 nM T96685 C27EYZ 127050129 IC50 = 16000 nM T96685 CJY3X7 127050185 IC50 = 25 nM T96685 CUR27K 127050186 IC50 = 7.9 nM T96685 C2ZQ3K 127050187 IC50 = 50 nM T96685 CU25TE 127050188 IC50 = 130 nM T96685 CZ5HL0 127051361 IC50 = 100 nM T96685 CO9FC4 127051362 IC50 = 130 nM T96685 C6OQG1 127052625 IC50 > 400000 nM T96685 CGV38D 127052626 IC50 = 100 nM T96685 CID97C 127052627 IC50 = 320 nM T96685 C16QBR 127052916 IC50 = 25 nM T96685 CEN92U 139053061 IC50 = 9800 nM T96685 C30ADT 145720921 IC50 = 34600 nM T96685 C3Z7VP 145720922 IC50 = 31200 nM T96685 C2P8OS 155511240 IC50 > 50000 nM T96685 CC8BF7 155512761 IC50 > 50000 nM T96685 CH5Q6L 155513950 IC50 = 26080 nM T96685 CG5PJ1 155514298 IC50 > 50000 nM T96685 C8VIL0 155514673 IC50 > 50000 nM T96685 CO4UH6 155514972 IC50 > 50000 nM T96685 CL97GC 155519990 IC50 > 50000 nM T96685 CN5UZ3 155522384 IC50 > 50000 nM T96685 C5LD2B 155526242 IC50 > 50000 nM T96685 C83ERS 155527164 IC50 > 50000 nM T96685 CHD3X6 155531906 IC50 = 9360 nM T96685 CV94KJ 155536434 IC50 > 50000 nM T96685 CXRM78 155537131 IC50 = 4800 nM T96685 C4E3TM 155538663 IC50 > 50000 nM T96685 CRS3E7 155546305 IC50 > 50000 nM T96685 C9XI0U 155558113 IC50 > 50000 nM T96685 CV5R2F 155560152 IC50 > 50000 nM T96685 C9WB1Q 155563330 IC50 > 50000 nM T96685 CW4YG8 155565340 IC50 > 50000 nM T96685 C0S5VT 155569173 IC50 > 50000 nM T22976 D03TGJ 5282192 Ki = 10400 nM T22976 D07XSN 6253 IC50 > 1000000 nM T22976 CP25DX 65049 IC50 = 285000 nM T22976 CPJ56E 452395 IC50 = 1300 nM T22976 CUW3B2 491807 IC50 = 27000 nM T22976 C8WS5I 491808 IC50 > 1000000 nM T22976 CYTV93 491811 IC50 = 801000 nM T22976 CA89BP 6476766 IC50 = 6300 nM T22976 CJB97H 6476767 IC50 = 402000 nM T22976 CZ1A0R 10097595 IC50 = 6800 nM T22976 C0PHT1 14606828 IC50 = 320 nM T22976 C3KA2N 16098860 IC50 = 45000 nM T22976 CH5P6G 16098865 IC50 = 5200 nM T22976 CH04XP 16098866 IC50 = 2400 nM T22976 C8MT2I 16098867 IC50 = 23000 nM T22976 CLIM56 16098869 IC50 = 114000 nM T22976 CL3T9X 16098872 IC50 = 1900 nM T22976 CF47QA 16098873 IC50 = 45000 nM T22976 C5GB9K 16098879 IC50 = 1900 nM T22976 CI4T9J 16098880 IC50 = 23000 nM T22976 CAF50V 16098881 IC50 = 1800 nM T22976 CI78AT 16121720 Ki = 290 nM T22976 C4MUA1 22489180 IC50 = 801000 nM T22976 C68QKG 44418800 IC50 = 390 nM T22976 CQY8X5 44437450 IC50 = 120000 nM T22976 C5H7LS 44437451 IC50 = 28000 nM T22976 CD0AN5 44437452 IC50 > 500000 nM T22976 C4YH3T 44437453 IC50 = 120000 nM T22976 C9LD5Y 44437454 IC50 > 1000000 nM T22976 CMB67C 44437455 IC50 = 480000 nM T22976 C5QFP6 44437456 IC50 = 74000 nM T22976 CJO51G 44437457 IC50 = 44000 nM T22976 CE1I4N 44437473 IC50 = 55000 nM T22976 CC0I1J 44437474 IC50 = 61000 nM T22976 C08ZMK 44437475 IC50 = 6400 nM T22976 CNPK62 44437476 IC50 = 3800 nM T22976 C2QO0P 44437477 IC50 = 187000 nM T22976 C9OE0G 44437478 IC50 > 500000 nM T22976 CO0N8X 44437480 IC50 > 1000000 nM T22976 C3BJE2 46197226 IC50 > 500000 nM T22976 C8WR4I 46197456 IC50 = 250 nM T22976 C2Y0QN 46197457 Ki = 12 nM T22976 CPA6D7 46700799 IC50 = 230 nM T22976 CWJY16 46874452 IC50 = 43000 nM T22976 C1PCR5 46884564 IC50 = 46 nM T22976 C4NK8W 46884565 IC50 = 42 nM T22976 C48RWL 46884566 IC50 = 1100 nM T22976 CN9RI6 46884567 IC50 = 4000 nM T22976 CZX1E7 46885197 Ki = 150 nM T22976 C5EPV6 46885249 IC50 = 400 nM T22976 C8DP0M 46885250 IC50 = 150 nM T22976 CQWV32 46885301 IC50 = 300 nM T22976 CG74UX 46885302 IC50 = 150 nM T22976 CUR4G7 46913823 IC50 = 91 ug.mL-1 T22976 CSQL06 54768280 IC50 = 60 ug.mL-1 T22976 CB9DU0 54768281 IC50 > 200 ug.mL-1 T22976 CUN04G 54768283 IC50 > 200 ug.mL-1 T22976 C2P3CT 90663608 IC50 > 1000000 nM T22976 CV0HE2 135499520 IC50 > 500000 nM T22976 C4K1FL 136118006 IC50 > 500000 nM T22976 CQGF80 136118007 IC50 > 500000 nM T22976 CR37CF 136118008 IC50 > 500000 nM T22976 D00KWL 16098859 IC50 = 2500 nM T22976 D02CCD 44418795 IC50 = 500 nM T22976 D07GKK 16098875 IC50 = 9700 nM T22976 D0C7YS 160155 Ki = 20000 nM T22976 D0I6UV 6477686 Ki = 500 nM T22976 D0O7GD 452142 IC50 = 4700 nM T22976 D0W8AD 16098874 IC50 = 4700 nM T32590 D09KTS 24821094 IC50 = 2.89 nM T32590 D0E6XR 3062316 IC50 = 0.3 nM T32590 D0OB0F 5328940 IC50 = 40 nM T32590 D02TUL 118115473 Ki = 131 nM T32590 D08AOZ 86582336 IC50 = 28 nM T32590 D0E3TC 44259 IC50 = 21.6 nM T32590 D0G5XV 135565884 IC50 = 2.95 nM T32590 CK5N6B 23657635 IC50 = 28 nM T32590 CSNC57 25110758 IC50 = 560 nM T32590 C0GOX5 25110759 IC50 = 500 nM T32590 CC2R7S 25110760 IC50 = 310 nM T32590 C36FXD 25138012 IC50 = 2 nM T32590 CP6N4G 25138050 IC50 = 220 nM T32590 CJL25F 25169253 IC50 = 700 nM T32590 CA98KR 44432441 IC50 = 1400 nM T32590 C8ZRE3 53356518 IC50 = 55 nM T32590 CJBL48 56925034 IC50 = 119 nM T32590 CZ3TG1 59375154 IC50 = 172 nM T32590 CV63UL 67240318 IC50 > 10000 nM T32590 C7VJ6A 70647728 IC50 = 180 nM T32590 COU73Y 71226944 IC50 = 45 nM T32590 C40JOZ 71235465 IC50 = 256 nM T32590 C54XWG 72190869 IC50 > 10000 nM T32590 CX75YR 73352604 IC50 = 79.43 nM T32590 C64SIO 92042864 IC50 = 36 nM T32590 C8HYU9 117926195 IC50 > 10000 nM T32590 C37DUM 121293882 IC50 = 26 nM T32590 CXQR89 121294143 IC50 = 2.3 nM T32590 CFKD32 122191637 IC50 = 95 nM T32590 CV89JM 132231876 IC50 = 15 nM T32590 C59HOQ 134277578 IC50 = 0.55 nM T32590 C0PZ5R 134277599 IC50 = 0.67 nM T32590 C7PWJ2 134277617 IC50 = 0.14 nM T32590 CRA2H1 134277633 IC50 = 0.47 nM T32590 CXJ8I0 134277643 IC50 = 0.18 nM T32590 C02RIA 134277647 IC50 = 0.2 nM T32590 CGH42R 134277652 IC50 = 0.25 nM T32590 COA14U 134277654 IC50 = 0.18 nM T32590 CQK0B5 134277685 IC50 = 0.76 nM T32590 C6S8VC 134277696 IC50 = 0.32 nM T32590 C49PIO 134277748 IC50 = 0.39 nM T32590 CD7VK4 134277767 IC50 = 0.59 nM T32590 CZ5E6L 134277773 IC50 = 0.42 nM T32590 C2CFK7 134277780 IC50 = 0.29 nM T32590 C6E7LW 134277790 IC50 = 0.21 nM T32590 C6T7NW 134277796 IC50 = 0.16 nM T32590 CU8ZP5 134277800 IC50 = 0.22 nM T32590 CTR4K6 134277828 IC50 = 0.14 nM T32590 CJ03PU 135566610 IC50 = 55.7 nM T32590 CQ9A5I 135566611 IC50 = 241.4 nM T32590 C42TOW 135566612 IC50 = 77.5 nM T32590 CN48IF 135566613 IC50 = 440.9 nM T32590 C67IYS 135566618 IC50 = 73.8 nM T32590 CP5SD0 136016241 IC50 = 66.5 nM T32590 C3Z4AT 137321159 IC50 > 10000 nM T32590 CZOD53 137633880 IC50 = 132 nM T32590 C7BJY5 137636807 IC50 = 282 nM T32590 CO89DX 137649100 IC50 = 231 nM T32590 CINE03 137652514 IC50 = 464 nM T32590 C28QUP 137652864 IC50 = 883 nM T32590 C4OD9Q 145967187 IC50 = 2.5 nM T32590 CE31VG 145979714 IC50 > 10000 nM T32590 C9BX4U 145988956 IC50 = 2990 nM T32590 C2MD1Q 155513187 IC50 > 10000 nM T32590 C3NA2I 155519537 IC50 = 358 nM T32590 D01RHR 71519693 IC50 = 1.9 nM T32590 D04PEI 11467730 IC50 = 11000 nM T32590 D04TLI 23657507 IC50 = 0.4 nM T32590 D06BJG 71556703 IC50 = 1.4 nM T62820 D00ENY 33032 EC50 = 290 nM T62820 D03FZT 25195461 EC50 = 65 nM T62820 D0B6RA 9834591 EC50 = 23.4 nM T62820 D0T3DG 9886034 Ki = 2.2 nM T62820 D01VZE 67705089 Ki = 7.43 nM T62820 D0D4OW 57338826 Ki = 20.1 nM T62820 D01FUB 25125217 EC50 = 195 nM T62820 D0P4BQ 9857256 Ki > 10000 nM T62820 D0U5CS 213056 EC50 = 5.1 nM T62820 D0ZV0R 16660135 IC50 > 10000 nM T62820 C0MLE4 1217 Ki > 1000000 nM T62820 CL8RX5 1222 Ki = 51000 nM T62820 COM10L 1297 Ki = 20000 nM T62820 CSM0F5 5115 IC50 = 577000 nM T62820 CZBT42 73537 EC50 = 110000 nM T62820 C8NO0Z 77937 EC50 > 1000000 nM T62820 C9H6OS 92136 EC50 = 35000 nM T62820 CUBH61 101122 EC50 > 1000000 nM T62820 CP05EH 136950 EC50 = 3500 nM T62820 CLMU31 165627 EC50 > 1000000 nM T62820 C34YGT 173564 EC50 > 1000000 nM T62820 CUT07K 177491 Ki > 300000 nM T62820 CR68YU 231345 EC50 > 1000000 nM T62820 C37ROZ 439282 Ki = 230 nM T62820 CO9KU6 443586 Ki > 1000000 nM T62820 C0S8TR 521212 EC50 = 3000 nM T62820 C3EP1R 627502 EC50 = 360 nM T62820 CW0CU9 798232 EC50 = 794.33 nM T62820 CB6X3Q 851990 EC50 = 5011.87 nM T62820 CNI89V 1617110 Ki = 205000 nM T62820 C5F8YH 2733519 EC50 > 600000 nM T62820 CZV0P5 3246152 Ki = 2000 nM T62820 C0HCI6 3461070 EC50 = 15848.93 nM T62820 COJV81 4521898 EC50 > 10000 nM T62820 CZ1Q5P 4694355 Ki = 30000 nM T62820 C05WNA 5310956 EC50 = 380 nM T62820 C7J6KQ 6604704 EC50 = 13000 nM T62820 C9INH1 6604707 EC50 > 1000000 nM T62820 CD68LI 6604795 Ki > 1000000 nM T62820 C6QSA9 7157252 EC50 > 300000 nM T62820 CL2OR7 7504549 EC50 = 155 nM T62820 C9PJQ1 9794208 EC50 = 0.16 nM T62820 CL8JI1 9837114 EC50 = 37000 nM T62820 CG3EN9 9885546 Ki = 85 nM T62820 C31YKH 9885608 EC50 = 1500 nM T62820 C9ACB3 9979770 EC50 = 229 nM T62820 CH54PF 9991661 EC50 = 122000 nM T62820 C9HD5C 9999945 EC50 = 3365 nM T62820 C1LK5F 10002415 EC50 = 2013 nM T62820 C0GN6F 10012356 Ki > 1000000 nM T62820 CQJP31 10012681 Ki = 122000 nM T62820 C82AGD 10026879 EC50 = 421 nM T62820 C6T7VH 10050046 EC50 = 1041 nM T62820 CAU7N4 10059959 EC50 > 300000 nM T62820 CYD93S 10070087 EC50 = 939 nM T62820 CYZ69A 10089411 Ki = 2700 nM T62820 CH6LU7 10103891 EC50 > 1000000 nM T62820 C8H3UO 10176324 EC50 > 10 nM T62820 C9XQK6 10198133 EC50 = 3.9 nM T62820 CL4NP9 10198359 EC50 = 10000 nM T62820 CAZ8P0 10198574 EC50 > 300000 nM T62820 CFDX64 10241509 EC50 > 300000 nM T62820 C7DU2G 10249222 EC50 = 72 nM T62820 C3TAF8 10251009 EC50 = 304 nM T62820 CUA94S 10262421 EC50 > 300000 nM T62820 CZ7A5Y 10263168 Ki > 1000000 nM T62820 CI86MW 10318576 EC50 = 380 nM T62820 CX12HM 10330132 Ki = 4800 nM T62820 CR94QY 10343566 EC50 = 878 nM T62820 CMW4B2 10353365 EC50 = 0.089 nM T62820 CZ09YG 10358265 IC50 = 20000 nM T62820 CQ1L0O 10359073 Ki = 18000 nM T62820 C6MTC4 10374869 EC50 > 1000000 nM T62820 C09LUW 10375719 IC50 > 200000 nM T62820 C29WLU 10407808 EC50 = 1823 nM T62820 C1IDG8 10413231 EC50 = 93 nM T62820 C3KHU7 10465017 EC50 > 300000 nM T62820 CK9MN4 10465478 EC50 = 40000 nM T62820 CO9MK3 10489913 EC50 > 300000 nM T62820 C34LSX 10489914 EC50 > 300000 nM T62820 C2TRI8 10492773 IC50 = 180 nM T62820 CU9BA6 10513894 EC50 > 300000 nM T62820 CQGZ24 10513895 EC50 > 300000 nM T62820 CYC9W8 10513896 EC50 > 300000 nM T62820 CG48QI 10515174 IC50 = 1100 nM T62820 CH9VN3 10560963 EC50 = 38000 nM T62820 CP0B8Q 10567792 IC50 = 240 nM T62820 C0P9JO 10587622 IC50 = 850 nM T62820 C20AXL 10607617 IC50 = 6500 nM T62820 CDN69Z 10609381 EC50 > 1000000 nM T62820 C57GCR 10656383 Ki > 1000000 nM T62820 C8FP7I 10681240 EC50 > 300000 nM T62820 C06TDU 10688450 IC50 = 220 nM T62820 CC6T7Z 10704895 EC50 > 300000 nM T62820 CC7JP9 10704896 EC50 > 300000 nM T62820 CD0E3P 10710505 IC50 = 1400 nM T62820 CBQV60 10732318 IC50 = 450 nM T62820 CC2PB0 10752213 EC50 > 300000 nM T62820 C27KWL 10752214 EC50 > 300000 nM T62820 CQTF38 10775369 EC50 = 54000 nM T62820 C6D9IL 10778385 IC50 = 1000 nM T62820 CQE5Y9 10783272 IC50 = 4360 nM T62820 C4Q3RT 10807972 IC50 = 200 nM T62820 CACY46 10826383 IC50 = 1000 nM T62820 C8MOC5 10828532 IC50 = 1800 nM T62820 C9BK1A 10846649 EC50 = 330 nM T62820 CHZ17V 10852666 IC50 = 240 nM T62820 CDO7A1 10979251 Ki = 420 nM T62820 CJ5B8P 11084869 EC50 = 7.5 nM T62820 CYP5U8 11187949 EC50 = 340 nM T62820 CSO7B4 11211597 IC50 = 25 nM T62820 CW74TN 11213605 EC50 = 186 nM T62820 CR7BZ3 11220424 EC50 = 19.8 nM T62820 C7UD6I 11235624 IC50 = 38 nM T62820 CNK6Y5 11269030 IC50 = 52 nM T62820 C7Z0HY 11271167 EC50 = 559 nM T62820 C8LSU6 11275666 EC50 = 21.2 nM T62820 CT4IL9 11281280 IC50 = 41 nM T62820 C3D0LM 11298568 Ki = 983 nM T62820 C9ASF3 11304010 IC50 = 7 nM T62820 CL1VX3 11310142 EC50 = 63.6 nM T62820 CX2T1N 11344646 EC50 = 28.6 nM T62820 C5FJ9P 11442010 IC50 = 15 nM T62820 CA50PD 11481048 Ki > 100000 nM T62820 C8N4QS 11484819 IC50 = 10 nM T62820 C8WX9P 11494153 EC50 = 4550 nM T62820 C97CIJ 11495483 EC50 = 819 nM T62820 C8P1GV 11496256 EC50 = 223 nM T62820 CYA2N5 11496550 EC50 = 442 nM T62820 C6NY5K 11503055 IC50 = 17000 nM T62820 CZF3H8 11510036 EC50 = 770 nM T62820 C9WAF1 11516962 EC50 = 782 nM T62820 CDC6P9 11530877 EC50 = 1532 nM T62820 CI3OW7 11531272 EC50 = 384 nM T62820 CTU14V 11531870 EC50 = 1500 nM T62820 CC4N0E 11537726 EC50 = 1717 nM T62820 CPA6R9 11539379 EC50 = 761 nM T62820 CQ5H1B 11543205 EC50 = 1000000 nM T62820 CB0VJ1 11545979 EC50 = 1060 nM T62820 C5JM0L 11546303 EC50 = 575 nM T62820 CW8H0Q 11559750 IC50 = 4.45 nM T62820 C3XIQ9 11559813 EC50 = 1987 nM T62820 C5TUG1 11575058 EC50 = 677 nM T62820 CHT79E 11583075 EC50 = 122 nM T62820 CGX8F6 11596869 EC50 = 201 nM T62820 CH2S1Q 11598292 EC50 = 276 nM T62820 CW3FH5 11625861 EC50 = 282 nM T62820 CZY8V2 11626305 EC50 = 676 nM T62820 CNC9T1 11626955 EC50 = 6 nM T62820 CG3YQ2 11631795 EC50 = 3273 nM T62820 CD9R3H 11633075 EC50 = 195 nM T62820 CZT84F 11646457 EC50 = 1093 nM T62820 C8YP5I 11648184 EC50 = 1160 nM T62820 C2W7YU 11648510 EC50 = 839 nM T62820 C2HBF6 11654949 EC50 = 892 nM T62820 CGKW60 11655609 EC50 = 188 nM T62820 CY59LG 11656255 EC50 = 1090 nM T62820 C3Y7PG 11656483 EC50 = 225 nM T62820 CVF97L 11663312 EC50 = 165 nM T62820 CFU63A 11663353 EC50 = 600 nM T62820 C5KEH1 11676185 EC50 = 589 nM T62820 C14GIR 11677757 EC50 = 270 nM T62820 CZ07JS 11684927 EC50 = 562 nM T62820 C8HCT2 11690041 EC50 = 5000 nM T62820 C57MBJ 11690196 EC50 = 293.5 nM T62820 CV4RD5 11691077 EC50 = 371 nM T62820 C0NU2Y 11691221 EC50 = 629 nM T62820 CBR6C9 11697718 EC50 = 291 nM T62820 CEV5N0 11699129 EC50 = 515 nM T62820 C72PVA 11710164 EC50 = 3855 nM T62820 C9ZS4H 11743092 EC50 = 3313 nM T62820 CASI54 11768848 EC50 = 10000 nM T62820 C96YUT 11820180 Ki = 23000 nM T62820 C38KRJ 11950553 EC50 = 984 nM T62820 CAQ78H 11950742 EC50 = 6367 nM T62820 C74FOC 11950744 EC50 = 1172 nM T62820 CWQ97C 11950745 EC50 = 2263 nM T62820 C4QLG1 11950746 EC50 = 3591 nM T62820 CCL2D8 11950926 EC50 = 1070 nM T62820 CB6DL5 11950927 EC50 = 559 nM T62820 CH2VY3 11951099 EC50 = 318 nM T62820 C0RP3G 11951270 EC50 = 1356 nM T62820 CY64JV 11951271 EC50 = 3544 nM T62820 CVIC83 11951272 EC50 = 1010 nM T62820 CQH10X 11951447 EC50 = 879 nM T62820 CQK7Y4 11951449 EC50 = 451 nM T62820 CAG3J7 11951806 EC50 = 228 nM T62820 CG1E3F 11951986 EC50 = 755 nM T62820 C57ARC 11951987 EC50 = 652 nM T62820 C20KVE 11951989 EC50 = 1130 nM T62820 C8NOX0 11951991 EC50 = 765 nM T62820 C84IEZ 11952168 EC50 = 598 nM T62820 CQR48X 11952169 EC50 = 779 nM T62820 CD47VA 11952347 EC50 = 788 nM T62820 CSW38G 15420544 EC50 > 10000 nM T62820 CP9Y7Q 15479143 EC50 = 0.56 nM T62820 CZ8PK5 15840277 EC50 > 1000000 nM T62820 CG3Q6X 16739372 EC50 > 1000000 nM T62820 C04GUC 17758443 Ki = 235000 nM T62820 C0Z2XO 17758444 Ki > 300000 nM T62820 CGZF13 17758445 Ki > 300000 nM T62820 C1GSZ4 17758449 Ki > 300000 nM T62820 CZW76I 17758450 Ki > 300000 nM T62820 CT64UF 17758554 Ki > 300000 nM T62820 C3X6WB 17758555 Ki > 300000 nM T62820 C1AD2J 17758556 Ki > 300000 nM T62820 CS5B7A 18138918 IC50 > 30000 nM T62820 CWEO80 18756981 Ki = 447000 nM T62820 CKX67J 18997192 EC50 > 30000 nM T62820 C5WYI2 21309795 IC50 = 312 nM T62820 CHR6P2 21393580 EC50 = 25130 nM T62820 CZ29VM 22368592 EC50 = 7810 nM T62820 C0K9DR 22884216 IC50 = 339000 nM T62820 CUB64E 23521659 EC50 = 140 nM T62820 CVMA40 23521677 EC50 = 200 nM T62820 C6X1VR 23521689 EC50 = 1100 nM T62820 CZ59GV 23521692 EC50 = 620 nM T62820 C9ZV0F 23521693 EC50 = 440 nM T62820 CRD2S7 23521697 EC50 = 36 nM T62820 CCB78W 23521698 EC50 = 180 nM T62820 CF8VY9 23521708 EC50 = 160 nM T62820 CE8Q1M 23521709 EC50 = 360 nM T62820 CK8MX3 23521713 EC50 = 1400 nM T62820 CGUN98 23521714 EC50 = 780 nM T62820 CP2SU0 23521725 EC50 = 4200 nM T62820 C8O4CW 23521727 EC50 = 1600 nM T62820 CLMX41 23521731 EC50 > 30000 nM T62820 CT9JZ3 23521734 EC50 = 2100 nM T62820 CBO38Y 23770349 EC50 = 3897 nM T62820 CDM85B 24809650 EC50 = 260 nM T62820 COM9A1 24809653 EC50 = 1170 nM T62820 C3Z2PD 24809687 EC50 = 2040 nM T62820 CSCW01 24815434 EC50 = 199.53 nM T62820 CBF6J9 24815439 EC50 = 125.89 nM T62820 C0DYP7 24815883 EC50 = 100 nM T62820 CN9AY0 24815976 EC50 = 100 nM T62820 C2A0LT 24849462 EC50 = 79.43 nM T62820 CYC98A 24849789 EC50 = 794.33 nM T62820 CB3T7C 24905650 IC50 > 1000000 nM T62820 C3BFR8 25002587 EC50 = 398 nM T62820 CB9E3V 25002939 EC50 = 390 nM T62820 CJ7KB0 25002941 EC50 = 372 nM T62820 CNK9Y0 25003298 EC50 = 347 nM T62820 CW23YC 25004010 EC50 = 174 nM T62820 CYHF64 25004352 EC50 = 186 nM T62820 CJ25HL 25008615 EC50 = 43 nM T62820 C6QGZ0 25073303 EC50 = 330 nM T62820 C9QYD4 25073615 EC50 = 1355 nM T62820 C01DRP 25173209 EC50 = 590 nM T62820 CY14JP 25173286 EC50 = 15 nM T62820 CW3PJ4 25173287 EC50 = 203 nM T62820 C43DFR 25173365 EC50 = 262 nM T62820 C4I9XA 25173448 EC50 = 117 nM T62820 CJS37O 25173616 EC50 = 7.9 nM T62820 CI0JF4 25173617 EC50 = 236 nM T62820 CRN46Z 25173691 EC50 = 75 nM T62820 CP21EC 25173697 EC50 = 84 nM T62820 C3CVG6 25173773 EC50 = 22.1 nM T62820 C7C5EF 25173776 EC50 = 142 nM T62820 CQYT89 25173778 EC50 = 76 nM T62820 CU3OL2 42610041 EC50 > 3162.28 nM T62820 C5E9CV 42610165 EC50 = 617 nM T62820 CL4R0H 42610166 EC50 = 234.42 nM T62820 CSUC90 42610167 EC50 = 2140 nM T62820 CUS06A 42629118 EC50 = 30 nM T62820 CK79XC 44155315 EC50 = 590 nM T62820 C7TXJ0 44155316 EC50 = 640 nM T62820 C65SXE 44155420 EC50 = 640 nM T62820 CQ3J6G 44155423 EC50 = 1170 nM T62820 CIU0E1 44155534 EC50 = 3820 nM T62820 CP6MG4 44155535 EC50 = 7150 nM T62820 CS6EZ9 44155538 EC50 = 640 nM T62820 CN9S0U 44155540 EC50 = 790 nM T62820 CMP31T 44155642 EC50 = 590 nM T62820 CJ49DN 44155643 EC50 = 4450 nM T62820 CK0N6G 44155644 EC50 = 1760 nM T62820 CV82HP 44155645 EC50 = 250 nM T62820 CA53BU 44155747 EC50 = 760 nM T62820 CKC0G4 44155748 EC50 = 1930 nM T62820 CQFB84 44155754 EC50 = 3300 nM T62820 C1GDO0 44155863 EC50 = 5870 nM T62820 CL94YO 44155986 EC50 = 1220 nM T62820 C5Y9DK 44155989 EC50 = 1350 nM T62820 CROL98 44156621 EC50 = 2700 nM T62820 C0TUD5 44178197 EC50 = 31 nM T62820 CNF72Q 44190035 IC50 > 10000 nM T62820 CMW71K 44285839 IC50 = 34 nM T62820 CL13FV 44302605 IC50 > 300000 nM T62820 C03QML 44302608 IC50 = 36000 nM T62820 C2H6QV 44302609 IC50 = 50000 nM T62820 CP1QS5 44302686 IC50 = 42000 nM T62820 C0V9DN 44302818 IC50 > 300000 nM T62820 CDM1P2 44302819 IC50 = 75000 nM T62820 C1GV9Q 44302837 IC50 > 300000 nM T62820 C1FJU0 44302855 IC50 > 300000 nM T62820 C34AVQ 44302856 IC50 = 37300 nM T62820 CLF56U 44302896 IC50 > 300000 nM T62820 C9Y6QA 44302913 IC50 > 300000 nM T62820 CC7BN3 44302929 IC50 > 300000 nM T62820 CKL1M8 44302930 IC50 = 61000 nM T62820 C9U0NH 44302931 IC50 = 46200 nM T62820 CD5XY2 44302932 IC50 > 300000 nM T62820 CFTA38 44322537 Ki = 1000 nM T62820 C7E8SH 44322745 Ki = 40000 nM T62820 CWV7F0 44322840 Ki = 110 nM T62820 CGL0Z3 44322843 Ki > 1000000 nM T62820 C2SKJ1 44322921 Ki = 330 nM T62820 CGK17I 44335500 EC50 = 2100 nM T62820 CB50YL 44335501 EC50 = 100 nM T62820 CZ08NT 44335514 EC50 = 1600 nM T62820 CKZ18D 44335554 EC50 = 16 nM T62820 CLK90Z 44335555 EC50 = 17 nM T62820 CZJ2H7 44335573 EC50 = 32 nM T62820 CQ1HE8 44335577 EC50 = 27 nM T62820 C7QOB9 44335578 EC50 = 18 nM T62820 CH4G8A 44335613 EC50 = 640 nM T62820 CWP53G 44335614 EC50 = 230 nM T62820 C6V3KJ 44335615 EC50 = 88 nM T62820 C4OXT1 44335626 EC50 = 29 nM T62820 CHO13Z 44335650 EC50 = 2500 nM T62820 CBY2Z8 44335670 EC50 = 310 nM T62820 C9Y6KA 44335710 EC50 > 30000 nM T62820 CHV03D 44338561 EC50 > 1000000 nM T62820 CL47OE 44345358 IC50 = 1600 nM T62820 CSZ48I 44345382 IC50 > 10000 nM T62820 CA57SX 44345536 IC50 > 10000 nM T62820 CGNR10 44345546 IC50 > 10000 nM T62820 CDRU87 44348706 IC50 = 180 nM T62820 CSJE56 44348769 IC50 = 1000 nM T62820 CUD35Q 44348846 IC50 = 190 nM T62820 C1IHR4 44348859 IC50 = 3100 nM T62820 CI06ET 44348911 IC50 = 220 nM T62820 C2O8QK 44348939 IC50 = 430 nM T62820 CM3T1Q 44348993 IC50 = 180 nM T62820 C7P2EA 44361401 Ki = 23 nM T62820 CF0LY9 44361402 Ki > 10000 nM T62820 C92YEO 44390403 EC50 = 596 nM T62820 C3ZR0Q 44392629 EC50 = 558 nM T62820 C5DUF6 44392645 EC50 = 890 nM T62820 CAS07C 44392671 EC50 = 578 nM T62820 CEZV70 44392708 EC50 = 4237 nM T62820 C90LMY 44395191 EC50 = 1418 nM T62820 CS6FD4 44395282 EC50 = 495 nM T62820 C3UGL7 44395299 EC50 = 918 nM T62820 CWZ6X4 44395327 EC50 = 241 nM T62820 C13GYT 44395381 EC50 = 7517 nM T62820 CHN13C 44397878 EC50 = 134 nM T62820 CAK39T 44406220 EC50 > 1000000 nM T62820 CH9J0V 44406221 EC50 > 1000000 nM T62820 CSD19C 44429217 EC50 > 1000000 nM T62820 CNZ16W 44429224 EC50 = 320000 nM T62820 C32RYA 44429225 EC50 > 1000000 nM T62820 CTQ29Z 44452714 IC50 = 3.49 nM T62820 CE8U7D 44452715 IC50 > 10000 nM T62820 CZG3T6 44569826 Ki > 1000000 nM T62820 CJ28TF 44569827 Ki > 1000000 nM T62820 CFZ64A 44569859 Ki > 1000000 nM T62820 CUW74T 44569860 Ki > 1000000 nM T62820 C62SAU 44591647 EC50 = 384 nM T62820 CQT61H 44591682 EC50 > 10000 nM T62820 CMP93S 44591683 EC50 > 10000 nM T62820 CA9XV2 44591684 EC50 = 5 nM T62820 CMV24G 44591685 EC50 > 10000 nM T62820 CHA08V 44591686 EC50 > 10000 nM T62820 C8FDN4 44591712 EC50 = 88 nM T62820 CC80XU 44591713 EC50 = 35 nM T62820 C80IYJ 44591714 EC50 = 280 nM T62820 CO5SY0 44591715 EC50 = 28 nM T62820 C2SEU1 44591744 EC50 = 158 nM T62820 C6F3WG 44591745 EC50 = 41 nM T62820 C2Y9IM 44591746 EC50 = 275 nM T62820 CRWM68 44591747 EC50 = 53 nM T62820 C0FY8H 44591748 EC50 = 26 nM T62820 CV5ZY0 44591770 EC50 = 97 nM T62820 CZ7ES9 44591771 EC50 = 183 nM T62820 C2OK6Y 44591772 EC50 = 32 nM T62820 CE0XV7 44591773 EC50 = 70 nM T62820 CET50O 44591774 EC50 = 4790 nM T62820 C64BTP 44591792 EC50 = 7550 nM T62820 C2ACY5 44591793 EC50 = 4380 nM T62820 CQL3J1 44591794 EC50 = 380 nM T62820 C72UIG 44591795 EC50 = 595 nM T62820 CX3T0N 44591796 EC50 = 3400 nM T62820 CJL2U9 44591797 EC50 = 1800 nM T62820 C20RKX 44591812 EC50 = 3060 nM T62820 CUJ69X 44591813 EC50 = 6360 nM T62820 CFAM64 45082292 Ki = 22387.21 nM T62820 CLBT94 46190877 EC50 = 79.43 nM T62820 CC4P3Q 46215704 EC50 = 160 nM T62820 CQ15ZS 46215708 EC50 = 501 nM T62820 CI0V4Q 46215709 EC50 = 230 nM T62820 C8ONP5 46215876 EC50 = 320 nM T62820 CCG69D 46215878 EC50 = 120 nM T62820 CNGE57 46216056 EC50 = 1660 nM T62820 C68EGY 46225320 EC50 = 316.23 nM T62820 CGH0M1 46225334 EC50 = 125.89 nM T62820 COFU37 46225335 EC50 = 199.53 nM T62820 C9XTG3 46225336 EC50 = 316.23 nM T62820 C96LBQ 46225337 EC50 = 501.19 nM T62820 C2HJY9 46225356 EC50 > 12589.25 nM T62820 CLYI35 46225357 EC50 = 63.1 nM T62820 CUTK50 46225358 EC50 = 125.89 nM T62820 C0UFE6 46225359 EC50 = 125.89 nM T62820 CS41AG 46225371 EC50 = 158.49 nM T62820 CGXJ25 46225372 EC50 = 158.49 nM T62820 CIG9F3 46225373 EC50 = 501.19 nM T62820 C4AYM0 46225374 EC50 = 794.33 nM T62820 CF1BR5 46225375 EC50 = 2511.89 nM T62820 C2REY9 46225383 EC50 = 12589.25 nM T62820 CC4Q8A 46225384 EC50 = 12589.25 nM T62820 CROL08 46225385 EC50 = 251.19 nM T62820 C9SN2I 46225386 EC50 = 50.12 nM T62820 CTI46Y 46225387 EC50 = 1995.26 nM T62820 CQK36B 46225407 EC50 = 125.89 nM T62820 CJU6S2 46225408 EC50 = 199.53 nM T62820 C6MC8Z 46225569 EC50 = 316.23 nM T62820 CS6Y9W 46225581 EC50 = 100 nM T62820 C78DON 46225582 EC50 = 158.49 nM T62820 CC8E3T 46225583 EC50 = 199.53 nM T62820 CML42B 46225584 EC50 = 39.81 nM T62820 C78MOX 46225585 EC50 > 3162.28 nM T62820 CI8C9S 46226929 EC50 = 630.96 nM T62820 CQUC74 46226930 EC50 = 977.24 nM T62820 C5F2MW 46226931 EC50 > 3162.28 nM T62820 CPEX32 46226933 EC50 > 3162.28 nM T62820 CGA3E8 46226934 EC50 = 1096.48 nM T62820 C6H1AE 46226952 EC50 = 851.14 nM T62820 CNXU31 46227786 EC50 = 158.49 nM T62820 C5KR8V 46227787 EC50 = 141.25 nM T62820 C56GKB 46227789 EC50 = 2290.87 nM T62820 CPI15K 46227790 EC50 = 645.65 nM T62820 C6K4BZ 46227792 EC50 = 446.68 nM T62820 CU9P1W 46227795 EC50 = 446.68 nM T62820 CFCB23 46227797 EC50 = 186 nM T62820 C31PAF 46700737 EC50 > 10000 nM T62820 CGS4F2 46836713 EC50 > 10000 nM T62820 CY8XU6 46887116 EC50 > 3000 nM T62820 CFZ75A 46887158 EC50 > 3000 nM T62820 CQ41EL 46887159 EC50 > 30000 nM T62820 CXRI94 46887204 EC50 > 30000 nM T62820 CD67PX 46887230 EC50 > 3000 nM T62820 C45HKB 46887231 EC50 > 3000 nM T62820 C2MF1C 46887232 EC50 > 3000 nM T62820 CWZU14 46887270 EC50 > 30000 nM T62820 CJIM29 46887271 EC50 = 1200 nM T62820 CBAG30 46887272 EC50 = 790 nM T62820 CJHM17 46887273 EC50 = 1300 nM T62820 CSO97X 46887318 EC50 > 30000 nM T62820 CQ2D0E 46887319 EC50 = 3440 nM T62820 CX8VI9 46887320 EC50 = 660 nM T62820 C8TFQ1 46887321 EC50 > 30000 nM T62820 CJ2TX5 46887322 EC50 = 360 nM T62820 CT46QN 46887367 EC50 = 590 nM T62820 CY8FH1 46887368 EC50 > 30000 nM T62820 CH9E7C 46887369 EC50 = 580 nM T62820 CQT58Z 46887370 EC50 = 360 nM T62820 CGZN85 46887371 EC50 = 350 nM T62820 CS80HA 46887372 EC50 = 240 nM T62820 CR0YT6 46887414 EC50 > 30000 nM T62820 C0H4YC 46887415 EC50 = 4110 nM T62820 CTHJ09 46887416 EC50 = 2190 nM T62820 CIBN32 46887417 EC50 = 840 nM T62820 CG03PK 46887418 EC50 = 780 nM T62820 CVIK59 46887459 EC50 > 30000 nM T62820 CF03GW 46887460 EC50 = 1180 nM T62820 CP2TE4 46887461 EC50 > 30000 nM T62820 C93HPN 46887462 EC50 > 30000 nM T62820 CT7CI1 46887463 EC50 > 30000 nM T62820 C7J3KZ 46887490 EC50 > 30000 nM T62820 CY87VO 46887491 EC50 > 30000 nM T62820 CW30ZV 46887492 EC50 > 30000 nM T62820 C4YJ6U 46887493 EC50 = 450 nM T62820 CD54VL 46887494 EC50 > 30000 nM T62820 CT50LF 46917716 EC50 = 199.53 nM T62820 CF6SM9 46917791 EC50 = 251.19 nM T62820 CJM4V9 46927956 EC50 > 50 nM T62820 CV6F9U 49799828 IC50 > 300000 nM T62820 C48MCL 49801368 Ki = 7.079 nM T62820 C5JV9D 49801369 Ki = 7.943 nM T62820 C2IS7M 49801370 Ki = 2.239 nM T62820 C49ZYG 49801371 Ki = 63.1 nM T62820 CHXD02 49822037 EC50 = 116 nM T62820 C8O0MB 49822115 Ki = 7.586 nM T62820 CET89N 49822116 EC50 = 45.7 nM T62820 C9CG2Q 49822195 EC50 = 132 nM T62820 CDC62Z 50992248 EC50 = 13 nM T62820 CN3TR7 51030965 EC50 = 159 nM T62820 CWE2O4 51033723 IC50 > 10000 nM T62820 C0L2SP 51036108 EC50 = 29 nM T62820 CAU6D5 51036701 EC50 = 430 nM T62820 CBI3A0 51036916 EC50 = 332 nM T62820 C3GQ8O 51037131 EC50 = 2200 nM T62820 CE4KP1 51050257 Ki > 10000 nM T62820 CQP6K5 51357936 EC50 = 76 nM T62820 C2DQ9V 51357937 EC50 = 3 nM T62820 C8SD6H 52941386 EC50 > 100000 nM T62820 CP97IL 52941387 EC50 > 100000 nM T62820 CN07TX 52944782 IC50 = 62000 nM T62820 CL4EM5 52947232 EC50 > 100000 nM T62820 C8JM1S 52947499 EC50 > 100000 nM T62820 CP8U6O 52948863 EC50 > 100000 nM T62820 CN1HU8 53235518 EC50 > 10000 nM T62820 CY58NO 53240406 EC50 = 5.6 nM T62820 C1WA5P 53316861 EC50 = 5011.87 nM T62820 CFGH56 53316862 EC50 = 630.96 nM T62820 CFA9L0 53317704 EC50 = 3162.28 nM T62820 COE1L6 53319016 EC50 > 10000 nM T62820 CI8V6B 53320175 EC50 = 501.19 nM T62820 CT2AE4 53320176 EC50 > 50118.72 nM T62820 CK54CE 53320818 EC50 = 398.11 nM T62820 C8XED2 53321493 EC50 = 158.49 nM T62820 CUXT69 53322147 EC50 = 1258.93 nM T62820 C30TGS 53322148 EC50 = 794.33 nM T62820 CD8L0K 53322149 EC50 = 794.33 nM T62820 CW36CH 53322382 EC50 > 10000 nM T62820 CYVT61 53323491 EC50 = 1584.89 nM T62820 CGXD80 53323492 EC50 = 630.96 nM T62820 CWQZ96 53323493 EC50 = 5011.87 nM T62820 CZJ14E 53324151 EC50 = 316.23 nM T62820 CEGK43 53324152 EC50 = 7943.28 nM T62820 CN3LP1 53324803 EC50 = 3981.07 nM T62820 CB27GO 53325450 EC50 = 630.96 nM T62820 CE45SV 53325451 EC50 = 1258.93 nM T62820 C6N0PC 53325452 EC50 = 398.11 nM T62820 CTJ85B 53325603 EC50 = 2511.89 nM T62820 C6I1SJ 53326074 EC50 = 2511.89 nM T62820 CV7Z8X 53326075 EC50 = 794.33 nM T62820 CN56WI 53326709 EC50 = 316.23 nM T62820 CCO07V 53326710 EC50 = 1995.26 nM T62820 CD2N3U 53326711 EC50 > 10000 nM T62820 CIHC67 54582001 IC50 > 30000 nM T62820 CJRG27 54761054 EC50 = 61 nM T62820 CFT41P 54761055 EC50 = 379 nM T62820 CJ8OE4 56587985 IC50 > 10000 nM T62820 CD2X1L 56651050 EC50 = 31 nM T62820 C61WQL 56968082 EC50 = 2.6 nM T62820 CYG7E8 57459475 EC50 = 696 nM T62820 CKD7Y0 57459477 EC50 = 56 nM T62820 CT70FL 57459480 EC50 = 468 nM T62820 C90COW 57459481 EC50 = 386 nM T62820 C9F4NA 57459482 EC50 = 31 nM T62820 C8Z3RY 57459483 EC50 = 299 nM T62820 C8VI3M 57459485 EC50 = 1120 nM T62820 CA2M4E 57459487 EC50 = 61.66 nM T62820 CLWD45 57459488 EC50 = 8.2 nM T62820 CC8E4J 57459494 EC50 = 6 nM T62820 CL2CK9 57459497 EC50 = 10.5 nM T62820 CEK6D7 57459500 EC50 = 116 nM T62820 CNFW08 57459501 EC50 = 24 nM T62820 CX0PZ8 57459504 EC50 = 178 nM T62820 CD2S1O 57459512 EC50 = 944 nM T62820 CH0R4N 57459517 EC50 = 149 nM T62820 CON7Q3 57459524 EC50 = 400 nM T62820 CL5DB3 57459542 EC50 = 519 nM T62820 C5S9BF 57459635 EC50 = 39 nM T62820 CH92AS 57459636 EC50 = 74 nM T62820 CH9X5W 57459640 EC50 = 102 nM T62820 C8YMH1 57459655 EC50 = 1230 nM T62820 CX0M2P 58081135 EC50 = 85 nM T62820 CBN30U 58103861 EC50 = 125 nM T62820 CKT7V5 58103890 EC50 = 150 nM T62820 CF9ID2 58966955 EC50 = 251.19 nM T62820 CCIL93 59234239 EC50 = 102 nM T62820 C4ZR5Q 59391336 EC50 = 361 nM T62820 CFCO74 59497075 EC50 = 251 nM T62820 CQ23OR 59497100 EC50 = 170 nM T62820 CW70SA 59599459 EC50 = 309.5 nM T62820 CF45DO 59599475 EC50 = 1076 nM T62820 C12XMG 59599515 EC50 = 1431 nM T62820 CIB19F 59599538 EC50 = 682 nM T62820 CC8W5L 59599545 EC50 = 87.4 nM T62820 CJIV72 59599552 EC50 = 39.3 nM T62820 C3OAM1 59599555 EC50 = 227 nM T62820 C1MJ8Z 59599565 EC50 = 470 nM T62820 CF3TQ4 59599568 EC50 = 319 nM T62820 CV91KQ 59599576 EC50 = 404.5 nM T62820 C1VAB2 59599577 EC50 = 109.6 nM T62820 CD5T6R 59599580 EC50 = 17.9 nM T62820 CHX74C 59599616 EC50 = 561.5 nM T62820 CYAQ39 60096178 EC50 = 8.37 nM T62820 C38GPO 60096183 EC50 = 26.5 nM T62820 C2NRC3 60096190 EC50 = 18.1 nM T62820 C63MKC 60096194 EC50 = 508 nM T62820 CMUL95 60096201 EC50 = 3.77 nM T62820 CW32CB 60096204 EC50 = 19.1 nM T62820 C8JAU2 60096211 EC50 = 257 nM T62820 C5PSF3 60096224 EC50 = 7.44 nM T62820 CXO4R6 60096228 EC50 = 6.32 nM T62820 C8N4UB 60096231 EC50 = 47.5 nM T62820 C9V3NZ 60096236 EC50 = 17.1 nM T62820 C38CBK 60096246 EC50 = 16 nM T62820 CN3OV8 60096250 EC50 = 6.97 nM T62820 C36ZLG 66612837 EC50 = 8510 nM T62820 CODX64 66784246 Ki = 14.79 nM T62820 C45ADN 66784262 Ki = 8.913 nM T62820 CV24AF 66784529 Ki = 3.02 nM T62820 CD7H3O 66784572 Ki = 3.631 nM T62820 CBP9O0 66784675 Ki = 11.75 nM T62820 CRFC93 66784890 Ki = 61.66 nM T62820 CQEC97 66785010 Ki = 6.761 nM T62820 C95WBM 66785027 Ki = 10.23 nM T62820 C6Q3OW 66785087 Ki = 3.631 nM T62820 CEIB16 66785101 Ki = 18.62 nM T62820 CRL4I1 66785182 Ki = 53.7 nM T62820 CBKT87 66785300 Ki = 3.89 nM T62820 CYK47D 66785393 Ki = 7.413 nM T62820 CR8QA6 66785551 Ki = 1.95 nM T62820 CDB31N 66785780 Ki = 3.162 nM T62820 C0GYH5 66786069 Ki = 5.248 nM T62820 CMD85A 66786131 Ki = 21.88 nM T62820 CB5EH8 66786493 Ki = 2.188 nM T62820 CG74XS 66786816 Ki = 6.457 nM T62820 CQE6Z9 66786902 Ki = 1.514 nM T62820 CJ1RB0 66787355 Ki = 5.012 nM T62820 COA08L 66787433 Ki = 11.75 nM T62820 CXN92C 66788653 EC50 = 55 nM T62820 C4PU9N 67056056 EC50 = 125 nM T62820 C3LDX1 67056141 EC50 = 149 nM T62820 C8YML5 67060140 EC50 = 274 nM T62820 CA2ZJ9 67060162 EC50 = 14 nM T62820 CBX67G 67246999 EC50 > 10000 nM T62820 C06MTQ 67705326 IC50 = 16.3 nM T62820 C7MLP4 67705376 IC50 = 26.1 nM T62820 CB16WU 67707808 IC50 = 18.8 nM T62820 C5K7QG 67974411 EC50 > 10000 nM T62820 CKY17T 68107697 EC50 = 1230 nM T62820 CY4OD9 68107740 EC50 = 57 nM T62820 CY49XO 68107810 EC50 = 15 nM T62820 C4SZ3V 68107813 EC50 = 9.7 nM T62820 C7VM6D 68108294 EC50 = 26 nM T62820 CA27NW 68108429 EC50 = 13.5 nM T62820 CB46KM 68108457 EC50 = 15 nM T62820 CKX84T 68108471 EC50 = 10 nM T62820 CZ7V1I 68108567 EC50 = 26 nM T62820 CFLO79 68108604 EC50 = 57 nM T62820 CZ60TR 68108857 Ki = 1.905 nM T62820 CM30YB 68109272 Ki = 38.9 nM T62820 CUQF38 68109333 Ki = 11.48 nM T62820 CZT19E 68109335 Ki = 6.026 nM T62820 CLC7E5 68109379 Ki = 61.66 nM T62820 CTYB39 68109425 Ki = 22.91 nM T62820 CH51BY 68109580 Ki = 2.042 nM T62820 CW3B2L 68109605 Ki = 10 nM T62820 CF1KB3 68109677 Ki = 6.026 nM T62820 C09TPQ 68109941 Ki = 0.8913 nM T62820 CCT07V 68290289 EC50 > 10000 nM T62820 C03JUE 68290572 EC50 > 10000 nM T62820 C8SO0Q 69092138 EC50 = 38 nM T62820 C2KV0O 69093106 EC50 = 26 nM T62820 CAQ62Y 69093344 IC50 = 7.3 nM T62820 C8IQ4U 69093439 EC50 = 37 nM T62820 CM4RD0 69093509 EC50 = 11 nM T62820 CY85RI 69093542 EC50 = 65 nM T62820 C72AHD 69093928 EC50 = 6.9 nM T62820 C0SDE4 69344751 EC50 = 251.19 nM T62820 CM1IS6 69929497 EC50 = 115 nM T62820 CZT05A 69929646 EC50 = 1286 nM T62820 CKV8E4 69929785 EC50 = 37 nM T62820 C5RI0Z 69930179 EC50 = 36 nM T62820 CG7F5Z 70051296 IC50 = 4990 nM T62820 CBK2Y6 70051926 EC50 = 1.3 nM T62820 CZ6XT7 70052526 EC50 = 7.6 nM T62820 C6PC1G 70209638 Ki = 2.57 nM T62820 C5M4GY 70681519 EC50 = 550 nM T62820 CARF46 70681520 EC50 = 1072 nM T62820 CW4MP8 70683629 EC50 = 3169 nM T62820 CEA04N 70683630 EC50 > 10000 nM T62820 CQL6G8 70683631 EC50 = 100 nM T62820 C85SZD 70685761 EC50 = 1150 nM T62820 C8ERQ5 70685762 EC50 = 363 nM T62820 C6HE1D 70685763 EC50 = 110 nM T62820 COV8Q0 70685764 EC50 = 42 nM T62820 C1X8ZL 70685765 EC50 = 832 nM T62820 CC68DO 70685766 EC50 = 275 nM T62820 CEY5P6 70685767 EC50 = 263 nM T62820 C5DM9I 70685768 EC50 = 230 nM T62820 CJSO08 70685769 EC50 = 64 nM T62820 C9KUT6 70689923 EC50 = 290 nM T62820 CGY70F 70689924 EC50 = 646 nM T62820 CRT73C 70689925 EC50 = 460 nM T62820 C3BOE9 70689926 EC50 = 1479 nM T62820 C6QGI9 70689927 EC50 = 447 nM T62820 C1I3RE 70689928 EC50 = 138 nM T62820 CLR8F3 70689929 EC50 = 100 nM T62820 CPZ9Y1 70689930 EC50 = 100 nM T62820 C9UV8C 70692086 EC50 = 479 nM T62820 CF3M0X 70694131 EC50 = 126 nM T62820 CH4JU9 70694132 EC50 = 933 nM T62820 CRP6A5 70696263 EC50 = 166 nM T62820 CB47XM 70696264 EC50 = 30 nM T62820 CXW7U0 70977933 EC50 = 148 nM T62820 CL52RS 71128783 EC50 = 531 nM T62820 CJIX85 71131322 EC50 = 0.58 nM T62820 C4JV5H 71135411 EC50 = 10.4 nM T62820 CE8L3P 71136640 EC50 = 12.4 nM T62820 CGH26Q 71136653 EC50 = 11.2 nM T62820 CW04KN 71136654 EC50 = 74 nM T62820 CAN01B 71136655 EC50 = 16.5 nM T62820 CHC91O 71137008 EC50 = 44.3 nM T62820 CH0W1O 71137010 EC50 = 13.9 nM T62820 CUB8G1 71137011 EC50 = 6.4 nM T62820 CP07IN 71137012 EC50 = 4.5 nM T62820 C28ZBK 71137034 EC50 = 11.8 nM T62820 C3N8ZO 71450118 EC50 = 501 nM T62820 CKRS61 71451227 EC50 = 330 nM T62820 CT1BS3 71454787 EC50 = 110 nM T62820 C4M0QE 71456562 EC50 = 190 nM T62820 C2R6AX 71457756 EC50 = 20 nM T62820 C0NG5K 71457757 EC50 = 4.1 nM T62820 C2D9WH 71458417 EC50 = 250 nM T62820 CV3I2G 71460259 EC50 = 710 nM T62820 C3L2SU 71461395 EC50 = 7.5 nM T62820 CKB65W 71462632 EC50 = 155 nM T62820 CNXB36 71476419 EC50 = 5.2 nM T62820 CNIW83 71479388 EC50 = 16 nM T62820 C8U0CT 71681823 EC50 = 8.2 nM T62820 CO5P1V 71681824 EC50 = 47.9 nM T62820 C6EIO9 71681825 EC50 = 12.2 nM T62820 CLH9N3 71681826 EC50 = 1170 nM T62820 CXW8R2 72714783 EC50 > 10000 nM T62820 C0HF5W 73347368 IC50 = 17000 nM T62820 CV75AO 76318478 IC50 = 132 nM T62820 CAO8Y5 76318479 IC50 = 100 nM T62820 C7L8CN 76322143 IC50 = 91 nM T62820 CG4M8N 76322144 IC50 = 89 nM T62820 C79TKZ 76332991 IC50 = 89 nM T62820 CY1V4K 76336598 IC50 = 133 nM T62820 C9J2QX 83821056 EC50 > 5000 nM T62820 CBA80Q 86691853 EC50 = 86 nM T62820 C3G4HD 86695984 IC50 = 19.9 nM T62820 CT2AF5 88593167 EC50 = 58 nM T62820 CWF97K 89497505 EC50 = 49 nM T62820 CDX7Q3 89497771 EC50 = 181 nM T62820 CFL05V 89497792 EC50 = 192 nM T62820 C3M8QU 89554892 IC50 = 146 nM T62820 C8BO4X 89735006 EC50 = 57 nM T62820 CL3AW7 89735130 EC50 = 26 nM T62820 C4RZ1G 89735186 EC50 = 70 nM T62820 C0TB9P 89735344 EC50 = 184 nM T62820 CF2UO1 89735510 EC50 = 112 nM T62820 C8FWH7 89735528 EC50 = 103 nM T62820 CC4O3J 89735530 EC50 = 80 nM T62820 C5F6VD 89735654 EC50 = 81 nM T62820 C0S7DT 89735684 EC50 = 313 nM T62820 CWZQ47 90098428 EC50 = 0.65 nM T62820 C53GQO 90668092 EC50 = 158.49 nM T62820 CZ80IY 90668093 EC50 = 125.89 nM T62820 CQ5HN3 90668094 EC50 = 251.19 nM T62820 C0X2RG 90668095 EC50 = 199.53 nM T62820 CEWD61 90668096 EC50 = 398.11 nM T62820 C0HCM5 90668097 EC50 = 158.49 nM T62820 CQ3V9Y 90668098 EC50 = 1995.26 nM T62820 C72VAL 90668099 EC50 = 316.23 nM T62820 CCG30J 90668100 EC50 = 501.19 nM T62820 CNR0U3 90668101 EC50 = 1258.93 nM T62820 C0KD7H 90668102 EC50 = 199.53 nM T62820 CLI30Z 90668103 EC50 = 251.19 nM T62820 CG1RM7 90668104 EC50 = 50118.72 nM T62820 CM2D0H 90668105 EC50 = 501.19 nM T62820 C7CN6Q 117821004 IC50 = 79.43 nM T62820 C4E9MZ 117821189 IC50 > 50118.72 nM T62820 CT7RL6 117821319 IC50 = 6.918 nM T62820 C8U9BX 117824335 IC50 = 8.913 nM T62820 C2XN3Z 117967312 EC50 = 28 nM T62820 C2CT0F 117968349 EC50 = 1.8 nM T62820 C56RJX 117968551 EC50 = 10 nM T62820 CW9RK2 117968589 EC50 = 5.5 nM T62820 CR3N4W 117971665 EC50 = 0.4 nM T62820 CA6NR3 117971683 EC50 = 13 nM T62820 C8UJ2M 117971685 EC50 = 0.5 nM T62820 C05WAR 117971699 EC50 = 6.1 nM T62820 CWN0I9 117972015 EC50 = 11 nM T62820 C9U1VQ 117972041 EC50 = 60 nM T62820 C4PY1O 117972044 EC50 = 17 nM T62820 CR6F0S 117972047 EC50 = 32 nM T62820 C3KJ0X 117972056 EC50 = 0.4 nM T62820 C7NX4A 117972153 EC50 = 16 nM T62820 C3J2TC 117972155 EC50 = 4 nM T62820 CK53MQ 117972250 Ki = 1 nM T62820 CD96PA 117972256 EC50 = 11 nM T62820 C7MP4F 118263352 EC50 = 195 nM T62820 CYZT31 118714734 EC50 = 2951 nM T62820 CVR15F 118714735 EC50 = 10715 nM T62820 CA9ZG2 118714736 EC50 = 871 nM T62820 CO69FH 118714737 EC50 = 3311 nM T62820 CW69AX 118714738 EC50 = 31623 nM T62820 C3UEW2 118714739 EC50 = 661 nM T62820 C1OCW6 118714740 EC50 = 3090 nM T62820 CR08AY 118714741 EC50 = 4677 nM T62820 C7O9PF 118714742 EC50 = 95 nM T62820 CR68DH 118714743 EC50 = 282 nM T62820 C7GXQ1 118714744 EC50 = 55 nM T62820 C6B0HF 118714745 EC50 = 178 nM T62820 CS89QO 118714746 EC50 = 355 nM T62820 CGLM54 118714747 EC50 = 81 nM T62820 C30EPW 118714748 EC50 = 141 nM T62820 COT2Z8 118714749 EC50 = 89 nM T62820 CZ4SW5 118714750 EC50 = 49 nM T62820 CGZ67Y 118714751 EC50 = 48 nM T62820 CVB84O 118714752 EC50 = 46 nM T62820 CN3Q6K 118714753 EC50 = 35 nM T62820 C4XA9K 118714754 EC50 = 98 nM T62820 CO5UN2 118714755 EC50 = 68 nM T62820 CHDR32 118714756 EC50 = 31 nM T62820 CX8W3I 118714757 EC50 = 151 nM T62820 CJ5G3Q 118718091 EC50 = 251000 nM T62820 C8SYH1 121447916 IC50 = 207 nM T62820 CUC13P 122187795 IC50 > 30000 nM T62820 CCP5U2 122195692 EC50 > 10000 nM T62820 CH2AO4 122539788 IC50 = 78 nM T62820 C1V8CY 123289788 EC50 = 1.3 nM T62820 C8RX0A 127038185 EC50 = 12870 nM T62820 CC0GA3 127038550 EC50 = 4624 nM T62820 CE0HT8 127039577 EC50 = 15 nM T62820 CS0G9A 127042771 EC50 = 191 nM T62820 CPZ70S 127052897 EC50 = 29 nM T62820 C38BRY 131801162 EC50 > 10000 nM T62820 CFC05Q 131954513 EC50 > 10000000 nM T62820 CW31CD 134129940 IC50 = 225 nM T62820 CI3PC4 134130002 EC50 = 6.8 nM T62820 C5F2YL 134130007 EC50 = 720 nM T62820 C5VEF0 134130172 EC50 = 1.7 nM T62820 C4VC9I 134130276 EC50 = 20 nM T62820 CUF61M 134130477 EC50 = 180 nM T62820 CKF21A 134130478 EC50 = 230 nM T62820 CHJF62 134130869 EC50 > 15000 nM T62820 CN74PQ 134131242 EC50 = 18 nM T62820 C0GE9K 134131273 EC50 > 3000 nM T62820 C3YM2R 134131309 EC50 = 2700 nM T62820 CNO62D 134131394 EC50 = 13 nM T62820 C28FZN 134131502 EC50 = 29 nM T62820 CL2UY8 134132133 Ki = 76 nM T62820 CP8C5N 134137754 IC50 = 34.5 nM T62820 CQT7H6 134138062 IC50 = 1130 nM T62820 CL7G4D 134139744 IC50 = 149 nM T62820 C5I6FC 134141510 IC50 = 215 nM T62820 CR4DE8 134144056 IC50 = 306 nM T62820 C5JNX4 134144441 IC50 = 280 nM T62820 CO1H6B 134152341 IC50 = 387 nM T62820 CL72ZY 134154496 IC50 = 210 nM T62820 CB8W0T 134155683 IC50 = 66.9 nM T62820 C1SFP5 134156113 EC50 = 17 nM T62820 CIR31F 134157889 EC50 = 22 nM T62820 C3EGM5 137321168 IC50 > 10000 nM T62820 CR5AB3 137634033 Ki = 595 nM T62820 C5TQS6 137635882 Ki = 1520 nM T62820 CBE4N9 137652320 Ki = 8.71 nM T62820 C48WZJ 137652500 Ki = 25.12 nM T62820 CBI4Z5 137656301 Ki = 627 nM T62820 CU2I6G 137659992 EC50 = 42.5 nM T62820 CK1ZQ3 146036859 EC50 = 10 nM T62820 C12SMP 146036860 EC50 = 140 nM T62820 CSO3M7 146036861 EC50 = 70 nM T62820 C6VB4M 146036862 EC50 = 30 nM T62820 C75DOJ 146036869 EC50 = 80 nM T62820 CHRX58 155511507 EC50 = 270 nM T62820 C7PNF3 155513095 EC50 = 50 nM T62820 CE2H9M 155514221 EC50 = 1070 nM T62820 CKYU94 155515810 EC50 = 27 nM T62820 CQN01W 155518472 EC50 = 90 nM T62820 CMTX16 155518831 EC50 = 79 nM T62820 CQ8A2I 155519573 EC50 = 190 nM T62820 C71GAL 155519836 EC50 = 141 nM T62820 CID23O 155519900 EC50 = 18 nM T62820 C5P9JY 155522079 EC50 = 600 nM T62820 CV3XK1 155523303 EC50 = 118 nM T62820 C89LOV 155524603 EC50 = 290 nM T62820 C7QRL8 155525998 EC50 = 29 nM T62820 CIE50K 155527610 EC50 = 180 nM T62820 C54IPT 155531064 EC50 = 23 nM T62820 C84PHE 155531978 EC50 = 33 nM T62820 CU87TZ 155533313 Ki = 112.2 nM T62820 CDTL70 155534303 EC50 = 15 nM T62820 C1OR2A 155535327 EC50 = 730 nM T62820 CNA3K4 155536450 EC50 = 13 nM T62820 C6BHP1 155536501 EC50 = 20 nM T62820 CYXE53 155538270 IC50 > 10000 nM T62820 CMJB23 155539343 EC50 = 210 nM T62820 CMCG93 155539952 IC50 = 45 nM T62820 CGH8T5 155540333 EC50 = 50 nM T62820 C0WE5P 155546950 EC50 = 70 nM T62820 CHK4N9 155548817 Ki = 6.166 nM T62820 CHI78O 155549028 EC50 = 71 nM T62820 CU63FZ 155550797 EC50 = 68 nM T62820 CJSF38 155551721 EC50 = 28 nM T62820 CA63SC 155552204 EC50 = 64 nM T62820 CZO03P 155552571 EC50 = 140 nM T62820 CVO21I 155553087 EC50 = 86 nM T62820 CEK92P 155554782 EC50 = 400 nM T62820 C2YX8U 155559438 EC50 = 620 nM T62820 C1GS6A 155559961 EC50 = 60 nM T62820 C3J6RS 155560108 EC50 = 2240 nM T62820 CZF2C1 155560423 EC50 = 37 nM T62820 C5G2HN 155562956 EC50 = 14 nM T62820 C5GK8N 155565811 EC50 = 70 nM T62820 CBN31S 155565817 EC50 = 18 nM T62820 C7HQ8B 155566352 EC50 = 6 nM T62820 C2KY7F 155566740 EC50 = 17 nM T62820 C6HT0Y 155567522 EC50 = 60 nM T62820 C1DML9 155567633 Ki = 4.169 nM T62820 CK4XC6 44322529 Ki = 75 nM T62820 D00EPM 73755217 IC50 > 30000 nM T62820 D00HKQ 25002940 EC50 = 316 nM T62820 D00NCL 46836562 EC50 > 10000 nM T62820 D01EAQ 11362035 EC50 = 14 nM T62820 D01EVA 6278000 Ki > 100000 nM T62820 D01YEN 1233 Ki = 110000 nM T62820 D02DEF 49765871 EC50 = 4.8 nM T62820 D03IES 44335556 EC50 = 24 nM T62820 D04DKM 104766 EC50 = 2000 nM T62820 D04GWD 59234231 Ki = 26.3 nM T62820 D04JKL 2071 Ki > 1000000 nM T62820 D04MVR 11530404 IC50 > 10000 nM T62820 D05TFE 5218788 Ki > 100000 nM T62820 D06DUE 40539 Ki = 113000 nM T62820 D06PAK 10058694 Ki = 3.9 nM T62820 D06SDD 9837317 EC50 = 0.57 nM T62820 D07GRG 10197984 EC50 = 2.69 nM T62820 D07MHL 9868580 EC50 = 27.54 nM T62820 D08BXD 9825084 EC50 = 270 nM T62820 D08CAB 83887 EC50 > 1000000 nM T62820 D08JKW 46830123 EC50 = 82 nM T62820 D08OCG 10047169 EC50 = 348 nM T62820 D09AQK 4545574 Ki > 300000 nM T62820 D09QUN 58368068 EC50 > 10000 nM T62820 D09RPR 16737207 Ki > 10000 nM T62820 D09UBS 10428048 Ki = 110 nM T62820 D09YEQ 11158623 IC50 = 14 nM T62820 D0D2GL 3972752 Ki = 11000 nM T62820 D0DX6U 23725699 IC50 > 10000 nM T62820 D0EK6P 5310984 Ki = 450 nM T62820 D0I6WA 44595851 Ki = 79.43 nM T62820 D0IO8J 3025961 Ki > 100000 nM T62820 D0J2WN 5311344 IC50 = 8000 nM T62820 D0J8OW 446355 IC50 = 4300 nM T62820 D0L0YF 4236420 EC50 > 1000000 nM T62820 D0N0NJ 15508178 IC50 = 121000 nM T62820 D0N2TP 44190040 IC50 > 10000 nM T62820 D0N9UZ 9819927 IC50 = 2.9 nM T62820 D0O1AK 23327 EC50 > 1000000 nM T62820 D0OH2P 5311040 Ki > 300000 nM T62820 D0OS8Y 15985251 IC50 > 10000 nM T62820 D0OT9B 5960 EC50 > 1000000 nM T62820 D0OV2V 6324634 IC50 = 400 nM T62820 D0P2VP 11708219 EC50 > 1000000 nM T62820 D0P3XO 5311459 Ki = 577000 nM T62820 D0PN6Z 179394 Ki = 129000 nM T62820 D0Q6VH 5311432 Ki > 100000 nM T62820 D0R0IB 56587994 IC50 > 10000 nM T62820 D0S6DK 5311455 EC50 = 48000 nM T62820 D0SL4Q 46190878 EC50 = 125.89 nM T62820 D0T5SU 158397 EC50 > 1000000 nM T62820 D0Y1WV 5310979 Ki = 110 nM T62820 D0YO8B 5311457 Ki = 84000 nM T25317 D00HPK 47641 Ki = 1500 nM T25317 D01AYJ 1549008 Ki > 50000 nM T25317 D01XBA 5035 Ki = 1 nM T25317 D06XMU 6013 Ki > 100000 nM T25317 D07BSQ 5994 Ki > 100000 nM T25317 D07KSG 2733526 Ki = 5 nM T25317 D0CT9Y 1548953 Ki = 1 nM T25317 D0D1AL 3559 Ki = 190 nM T25317 D0D7TB 9417 Ki = 13 nM T25317 D0L5WM 2157 Ki = 25 nM T25317 D0R4OM 5566 Ki = 8 nM T25317 D0Z6ST 2467 Ki = 60 nM T25317 D0I8FV 5567 Ki = 165 nM T25317 D00KVE 9907323 Ki = 1.72 nM T25317 D0K6NS 6536 Ki = 11 nM T25317 C5VS0H 10098 Ki > 100000 nM T25317 CTF7Z4 50266 Ki = 51 nM T25317 C0LQ7N 65638 Ki = 2 nM T25317 CY79XW 72027 Ki = 18 nM T25317 CN26SL 93365 Ki = 30 nM T25317 C3SG4X 185834 Ki = 1 nM T25317 CU2RH4 202478 Ki = 2200 nM T25317 CK0JI9 1548955 Ki = 2 nM T25317 C97VGU 5474589 Ki = 54 nM T25317 CFO08L 6437849 Ki = 34000 nM T25317 C2UV7A 6439331 Ki = 3 nM T25317 C1M9QS 6713949 Ki = 583 nM T25317 CD8H3W 9799239 Ki = 0.6 nM T25317 CJ96KD 9820591 Ki = 1.7 nM T25317 CXYJ93 9841596 Ki = 15 nM T25317 C78DMI 9951886 Ki = 450 nM T25317 CZ0AT6 9954083 Ki = 2 nM T25317 CQ9NP6 11198145 Ki = 5 nM T25317 CDFB43 11743300 Ki = 8500 nM T25317 CL7XE8 13998486 Ki = 39 nM T25317 CD4N5E 15163141 Ki = 1 nM T25317 C10CLM 16061352 Ki > 100000 nM T25317 CZL87E 44303090 Ki = 500 nM T25317 CX7W3K 44398003 Ki = 441 nM T25317 C2MZH9 44398036 Ki = 4 nM T25317 C7C2TW 44398114 Ki = 6 nM T25317 C17XVW 44398137 Ki = 654 nM T25317 C0N2XB 44474938 Ki = 455 nM T25317 CU63SQ 50994498 Ki = 211 nM T25317 CUL3W2 57402462 Ki = 233 nM T25317 CGKR02 71582863 IC50 = 17000 nM T25317 CZ39OQ 71583076 IC50 = 8000 nM T25317 C0RHL6 71583188 IC50 = 15000 nM T25317 CXF49Y 71583302 IC50 = 7000 nM T25317 C02KCO 71583303 IC50 = 27000 nM T25317 CYT02N 71583304 IC50 = 17000 nM T25317 CME46I 71584577 IC50 = 11000 nM T25317 CN37SA 71584578 IC50 = 7000 nM T25317 CO79PJ 73345319 Ki = 9300 nM T25317 D00FUO 4416 Ki = 0.9 nM T25317 D02WJT 7333 Ki = 6700 nM T25317 D03TNT 5753 Ki > 100000 nM T39123 D04GEI 46700761 EC50 = 5.2 nM T39123 D0P9KL 49787129 Ki = 0.036 nM T39123 CP36DZ 8478 Ki = 3600 nM T39123 C37NQO 9919540 EC50 = 3.3 nM T39123 C4SHQ7 10010442 IC50 = 16000 nM T39123 C2QEH4 10301495 Ki = 708 nM T39123 CDR52W 10328205 EC50 = 1.4 nM T39123 C7CJH5 11622248 Ki = 0.089 nM T39123 CZJ6B1 16735508 EC50 = 1.6 nM T39123 CQ6F7E 16735509 EC50 = 3.1 nM T39123 C3F1BN 16735511 EC50 = 3 nM T39123 C39KOX 16735542 EC50 = 0.99 nM T39123 CEPD53 16735543 EC50 = 1.2 nM T39123 CN80DX 16735544 EC50 = 3 nM T39123 C6JWF7 16735567 EC50 > 100 nM T39123 CQ30OG 16735729 EC50 = 1.7 nM T39123 CGR7X8 16735730 EC50 = 0.8 nM T39123 C8YW4E 16735731 EC50 = 2 nM T39123 C20VSA 16735779 EC50 = 1.3 nM T39123 CQ04DO 16735780 EC50 > 100 nM T39123 CR8GT6 16735781 EC50 = 2.7 nM T39123 CN3KA2 16736169 EC50 = 3.3 nM T39123 C4CPV9 16736170 EC50 = 1.7 nM T39123 CGS86D 16736191 EC50 = 3 nM T39123 CQJ8C7 16736192 EC50 = 2.1 nM T39123 CVQ4E2 16736193 EC50 = 1.2 nM T39123 CW3MQ4 16736392 EC50 = 4.7 nM T39123 CVZ82U 16737378 EC50 = 0.99 nM T39123 CURY37 16737730 EC50 = 5 nM T39123 C0PT2L 16738337 EC50 = 1.7 nM T39123 CM15JY 24992020 EC50 = 1.2 nM T39123 CQA87N 24993005 EC50 = 3.3 nM T39123 CJXU79 24993970 EC50 = 1.9 nM T39123 CM0VA1 24994272 EC50 = 1.8 nM T39123 C2BCY3 24994895 EC50 = 4.4 nM T39123 C43WRQ 24995205 EC50 = 2.8 nM T39123 C5FM7Y 24995518 EC50 = 1.2 nM T39123 CQ0AX6 24995519 EC50 = 5.2 nM T39123 C10SWN 24996155 EC50 = 2.3 nM T39123 CMG2H1 24996486 EC50 = 1.6 nM T39123 CT6PL0 24996487 EC50 = 4.9 nM T39123 C70UHN 24996490 EC50 = 0.43 nM T39123 CL1UD5 24996809 EC50 = 1.1 nM T39123 CK17PD 24996810 EC50 = 2.4 nM T39123 C52IBC 25075960 EC50 = 0.56 nM T39123 CL34UW 25075963 EC50 = 0.65 nM T39123 CIO6F0 25075965 EC50 = 1.4 nM T39123 COI6C1 25075973 EC50 = 0.47 nM T39123 CA89SK 25075978 EC50 = 5.2 nM T39123 CH9NM7 25084920 EC50 = 0.073 nM T39123 C36SXI 25084922 EC50 = 2.8 nM T39123 C6S2CB 25138123 IC50 = 0.12 nM T39123 C0APO3 25138124 EC50 = 2.5 nM T39123 C8RYH9 25138125 EC50 = 5.4 nM T39123 CV8O2Q 25138126 IC50 = 32 nM T39123 CPF6T8 25138127 IC50 = 460 nM T39123 CZL08E 25138128 IC50 = 380 nM T39123 CLE2X9 25138129 EC50 = 4.3 nM T39123 CAG05L 25138130 IC50 = 32 nM T39123 CRBW20 25138131 IC50 = 0.24 nM T39123 C0XMG1 25138132 IC50 = 240 nM T39123 CA58FK 44419644 Ki = 82.7 nM T39123 C5LYA4 44419664 Ki = 10000 nM T39123 CEM4B9 44419672 Ki = 9.4 nM T39123 CK9I3C 44419676 Ki = 88.1 nM T39123 C5SU4A 44419677 Ki = 10000 nM T39123 C3NX6G 44425065 EC50 = 3.1 nM T39123 CETO79 46906646 IC50 > 30000 nM T39123 CXWN52 46906647 IC50 = 890 nM T39123 CY4L2G 53318788 IC50 > 30000 nM T39123 CSGI29 57653049 EC50 = 0.75 nM T39123 C32WXO 57653056 EC50 = 2.3 nM T39123 CQ3E0F 71449398 EC50 = 0.24 nM T39123 CVNR92 71449399 Ki = 0.12 nM T39123 CRM3V8 71449427 EC50 = 0.023 nM T39123 C5HTR3 71449428 EC50 = 0.36 nM T39123 C4ZNW1 71449429 EC50 = 0.15 nM T39123 CM5F3O 71451197 EC50 = 0.11 nM T39123 CG85XR 71451222 EC50 = 1.5 nM T39123 CSL41G 71451223 EC50 = 0.33 nM T39123 CSJ9V7 71453041 EC50 = 0.13 nM T39123 CF6TH4 71454755 EC50 = 0.041 nM T39123 CDE4V6 71454783 EC50 = 0.065 nM T39123 CTKG87 71454784 EC50 = 3.9 nM T39123 C8MU2C 71456524 IC50 = 0.61 nM T39123 CDQ5R8 71456525 IC50 = 0.49 nM T39123 C4PGM7 71456556 EC50 = 1.4 nM T39123 CH08JC 71456557 EC50 = 0.32 nM T39123 C2O4EW 71458409 EC50 = 7.2 nM T39123 CJN7H4 71458410 EC50 = 0.27 nM T39123 C6OFU9 71458411 EC50 = 76 nM T39123 C15TJE 71458412 EC50 = 0.29 nM T39123 C53GHV 71460218 EC50 = 0.13 nM T39123 C6UF1I 71460219 EC50 = 0.1 nM T39123 CCD8U3 71460220 EC50 = 0.098 nM T39123 CKUG49 71460251 EC50 = 5.8 nM T39123 C59CNG 71460252 EC50 = 0.029 nM T39123 C7AXG0 71460253 EC50 = 0.34 nM T39123 C8B3OF 71460254 EC50 = 1.4 nM T39123 C8FA9K 71461936 Ki = 0.046 nM T39123 C0IL1S 71461937 IC50 = 0.51 nM T39123 CC8AD0 71461938 EC50 = 0.05 nM T39123 CV7N6I 71461939 EC50 = 0.24 nM T39123 CJV5K8 71461940 EC50 = 0.072 nM T39123 CFX17J 71461962 EC50 = 0.039 nM T39123 C1XEW4 71461963 EC50 = 10 nM T39123 CRPE69 72711369 Ki = 0.045 nM T39123 C9DYJ7 72711370 Ki = 0.062 nM T39123 C19QVF 72711589 Ki = 0.086 nM T39123 C5UPE8 72711802 Ki = 0.12 nM T39123 CYT42N 72711803 Ki = 0.055 nM T39123 C2JD9A 72712017 Ki = 0.29 nM T39123 CN16AD 72712018 Ki = 0.11 nM T39123 CCJ3Q2 72712230 Ki = 0.052 nM T39123 CRJF51 72712231 Ki = 0.51 nM T39123 CV60KA 72712449 Ki = 0.12 nM T39123 CO1E6F 72712450 Ki = 0.2 nM T39123 C47VKG 72712666 Ki = 0.21 nM T39123 C95OKS 72712667 Ki = 0.044 nM T39123 C2E3SM 72712870 Ki = 0.21 nM T39123 COGF32 72712871 Ki = 0.2 nM T39123 CT4H1A 72713068 Ki = 0.12 nM T39123 CBNS46 72713069 Ki = 0.086 nM T39123 CY40CT 72713283 Ki = 0.032 nM T39123 C74TQW 72713284 Ki = 0.065 nM T39123 CG56KH 72713503 Ki = 0.2 nM T39123 CG1Z9Y 72713504 Ki = 0.11 nM T39123 C4VM7N 90324505 EC50 = 0.07 nM T39123 C3S1VA 90324512 EC50 = 120 nM T39123 C2AY1B 90324535 EC50 = 0.07 nM T39123 C6OKG1 90488921 EC50 = 2.5 nM T39123 C8EBD0 118707476 Ki = 0.074 nM T39123 CZ9FT5 118707477 Ki = 0.086 nM T39123 C6AUZ9 118707478 Ki = 0.052 nM T39123 C57NZB 118707479 EC50 = 4.4 nM T39123 CFD65J 118707480 EC50 = 1.5 nM T39123 CN1LZ9 118707481 EC50 = 0.59 nM T39123 C18IBL 118707482 Ki = 0.096 nM T39123 CGVP49 118707483 EC50 = 2.8 nM T39123 CJ4N0R 118707484 Ki = 0.037 nM T39123 CO3MI9 118707485 Ki = 0.036 nM T39123 C1WIM0 118707486 Ki = 0.028 nM T39123 CYV39R 118707487 Ki = 0.2 nM T39123 CPOR71 118707488 EC50 = 1.3 nM T39123 C35SAG 118707489 EC50 = 0.49 nM T39123 CO46GB 118707490 EC50 = 0.63 nM T39123 CJ24EG 118707491 Ki = 0.12 nM T39123 CR7O5H 118707492 Ki = 0.039 nM T39123 CF42GO 118707493 EC50 = 0.8 nM T39123 C91JFU 118707494 Ki = 0.034 nM T39123 CRVI37 118707495 Ki = 0.027 nM T39123 C9T0QG 118707496 Ki = 0.089 nM T39123 CT8S3P 118707497 Ki = 0.038 nM T39123 CD0WC6 118708107 Ki = 0.026 nM T39123 C7TXJ1 118735592 EC50 = 0.6 nM T39123 CV67KT 118735593 EC50 = 0.006 nM T39123 C7GMR6 118735594 EC50 = 0.9 nM T39123 C6B9SG 118735595 EC50 = 0.1 nM T39123 CHW34M 118735596 EC50 = 0.08 nM T39123 C5X7QV 118735679 EC50 = 13.9 nM T39123 C68ZHV 118735680 EC50 = 7.2 nM T39123 C1G0AZ 118735681 EC50 = 182 nM T39123 CFJ68R 118735682 EC50 > 500 nM T39123 CW5Y1F 118735683 EC50 = 2.9 nM T39123 C12CFY 118735684 EC50 = 24.4 nM T39123 CE1LW7 118735685 EC50 = 1.6 nM T39123 CU61JE 118735686 EC50 = 216 nM T39123 C4EDS9 134132372 EC50 = 0.48 nM T39123 CLCJ20 134135834 EC50 = 2.7 nM T39123 CP24SX 134143614 EC50 = 3.6 nM T39123 CP5FD6 134150351 EC50 = 0.49 nM T39123 C2WXP1 134150893 EC50 = 5.8 nM T39123 CV3ZI2 134151953 EC50 = 2 nM T39123 CW95DP 134154824 EC50 = 1.9 nM T39123 CI3OY0 134157013 EC50 = 0.61 nM T39123 CU37XC 134157281 EC50 = 22 nM T39123 C30FKQ 134157735 EC50 = 5.5 nM T39123 CH7OX8 135401501 IC50 = 3.6 nM T39123 CJ6N0V 135410889 IC50 = 10 nM T39123 CGEL62 135410891 IC50 = 25 nM T39123 C8U0TV 135528869 IC50 = 2100 nM T39123 CF0Z2T 135936864 IC50 = 1100 nM T39123 CR71AU 135936875 IC50 = 3.7 nM T39123 COQU30 136016359 IC50 = 24000 nM T39123 CR5X2P 136016360 IC50 = 34 nM T39123 CJR7Q3 136016361 IC50 = 33000 nM T39123 C1Z7SR 136016362 IC50 = 30 nM T39123 CG1HK6 136016372 IC50 = 120 nM T39123 C0PDO9 136016373 IC50 = 490 nM T39123 CQ47XG 136016379 IC50 = 480 nM T39123 CZVA18 136016380 IC50 = 7.4 nM T39123 CT73EU 136016381 IC50 = 9.8 nM T39123 CW5C9G 136016382 IC50 = 19 nM T39123 C7N9GK 136016389 IC50 = 12 nM T39123 C1QX4H 136016390 IC50 = 120 nM T39123 CKE02M 136016391 IC50 = 14 nM T39123 CMO0T8 136016392 IC50 = 45 nM T39123 C2HO5R 136016397 IC50 = 31 nM T39123 C97USJ 136016398 IC50 = 15 nM T39123 CF4B8O 136016399 IC50 = 32 nM T39123 CK8RP5 136016406 IC50 = 32 nM T39123 CTF9P2 136016407 IC50 = 8 nM T39123 CWI8P3 136016412 IC50 = 11 nM T39123 CKGQ75 136016413 IC50 = 1200 nM T39123 C0AQ7F 136016436 IC50 = 1500 nM T39123 C6X2DT 136016437 IC50 = 9900 nM T39123 C27HJQ 136016443 IC50 = 570 nM T39123 C1SLG4 136016444 IC50 = 51 nM T39123 CIAW82 136016471 IC50 = 180 nM T39123 C4X6FN 136016472 IC50 = 4.6 nM T39123 C2A3NT 136016473 IC50 = 10 nM T39123 CB62WX 136016474 IC50 = 10 nM T39123 CZ1M4G 136016475 IC50 = 16 nM T39123 C30HUY 136016476 IC50 = 10 nM T39123 C3E0AK 136016477 IC50 = 18 nM T39123 CBN5P4 136016478 IC50 = 17 nM T39123 C65OCQ 136016479 IC50 = 8 nM T39123 CJNO30 136016480 IC50 = 22 nM T39123 CT3M4D 136016481 IC50 = 9.7 nM T39123 C60IKA 136016482 IC50 = 7.9 nM T39123 C5T4QK 136016483 IC50 = 18 nM T39123 CIF8U7 136016484 IC50 = 14 nM T39123 CAFQ17 136016486 IC50 = 20 nM T39123 CYB5V3 136016487 IC50 = 4.1 nM T39123 CP67NX 136016488 IC50 = 8.4 nM T39123 C6S5WT 136016489 IC50 = 16 nM T39123 CGLB52 136016490 IC50 = 12 nM T39123 C80OZB 136016491 IC50 = 30 nM T39123 C6FPZ0 136016492 IC50 = 15 nM T39123 CL8G2K 136016493 IC50 = 30 nM T39123 CSIC76 136016517 IC50 = 7.3 nM T39123 CX94OU 136016518 IC50 = 15 nM T39123 C7I4EX 136016519 IC50 = 11 nM T39123 C9DES8 136016521 IC50 = 9.7 nM T39123 C6VIE8 136016522 IC50 = 18 nM T39123 CXM7G2 136016523 IC50 = 20 nM T39123 CJEY60 155514052 EC50 = 0.17 nM T39123 CS0K9I 155518633 EC50 = 0.89 nM T39123 C5MIX2 155522287 EC50 = 0.058 nM T39123 CFH80A 155527587 EC50 = 0.13 nM T39123 CKL19Y 155529496 EC50 = 0.62 nM T39123 C0WQA2 155529648 EC50 = 0.028 nM T39123 C9TNM5 155533419 EC50 = 0.27 nM T39123 C3DY9F 155534572 EC50 = 7.7 nM T39123 CXH7J8 155534639 EC50 = 0.23 nM T39123 C7W0RS 155535993 EC50 = 1.4 nM T39123 C05WMX 155536247 EC50 = 0.11 nM T39123 C1Z6WR 155538456 EC50 = 0.6 nM T39123 C3H6MD 155541282 EC50 = 1.5 nM T39123 C2M6UZ 155545453 EC50 = 0.037 nM T39123 C0F5ZQ 155547611 EC50 = 130 nM T39123 CQ6OT8 155547823 EC50 = 0.024 nM T39123 C1F2AE 155548337 EC50 = 0.16 nM T39123 CZ21YV 155549139 EC50 = 0.24 nM T39123 CO8GB1 155550061 EC50 = 0.022 nM T39123 C1J4YQ 155550676 EC50 = 2.1 nM T39123 C7PS9D 155551159 EC50 = 0.068 nM T39123 C3ZJ1N 155554573 EC50 = 0.33 nM T39123 CRQ10Z 155559289 EC50 = 0.13 nM T39123 CA1R6T 155559308 EC50 = 8.2 nM T39123 C06LPU 155565826 EC50 = 0.12 nM T39123 CW5M4U 16735568 EC50 = 1 nM T39123 D01VSI 25240297 Ki = 0.035 nM T39123 D08UWO 53320361 IC50 = 830 nM T39123 D0JE3Z 16735569 EC50 = 0.45 nM T84791 C5Z1QA 96028 IC50 = 10300 nM T84791 C0ZI3J 11298263 IC50 > 100000 nM T84791 CKI97Z 12344252 IC50 = 25100 nM T84791 CKSL53 12507616 IC50 = 2900 nM T84791 COF8W3 13008156 IC50 = 1600 nM T84791 CGW49I 25146686 IC50 = 7100 nM T84791 C84YXH 74763382 IC50 > 30000 nM T84791 C7S6YM 90348686 IC50 = 11000 nM T84791 CAZ6F3 123132902 IC50 = 60 nM T84791 CP60WQ 126599605 IC50 = 15000 nM T84791 CL9DA5 126599606 IC50 = 30000 nM T84791 CIM95P 126599607 IC50 > 100000 nM T84791 CZM3T2 126599609 IC50 = 7000 nM T84791 CBZ9G6 126599610 IC50 > 100000 nM T84791 CD57UE 126599615 IC50 > 100000 nM T84791 C05JCQ 126599616 IC50 > 50000 nM T84791 C27LVH 126599619 IC50 = 24000 nM T84791 CQ4OX7 126599621 IC50 = 6900 nM T84791 CU9IB6 126599623 IC50 = 15300 nM T84791 C50GVU 126599624 IC50 < 500 nM T84791 CE4U8C 126599625 IC50 = 4000 nM T84791 C3NUF1 126599626 IC50 = 7000 nM T84791 CG5JH7 126599627 IC50 = 500 nM T84791 CH8TE6 126599628 IC50 = 20000 nM T84791 CAY4G6 126599629 IC50 = 41000 nM T84791 CEQ96X 126599630 IC50 = 68000 nM T84791 CY86ZU 126599632 IC50 = 16000 nM T84791 CF35OY 126599634 IC50 = 18000 nM T84791 C0X4TK 126609831 IC50 > 100000 nM T84791 CQ9KN4 129892190 IC50 = 5.8 nM T84791 C43MXV 137644429 IC50 = 300 nM T84791 CRD19U 137644814 IC50 > 100000 nM T84791 C97ABQ 137644943 IC50 > 100000 nM T84791 C97MXP 137648465 IC50 > 100000 nM T84791 C2JPC1 137656599 IC50 = 35000 nM T09395 CBZ7P2 2928097 Ki = 49 nM T09395 CERF41 3151315 Ki = 1120 nM T09395 CL4GK5 13686033 IC50 = 6755 nM T09395 CY5SQ3 13755302 IC50 = 0.01 ug.mL-1 T09395 C2WEO7 44332503 IC50 = 0.05 ug.mL-1 T09395 C1XHA3 44332504 IC50 = 0.04 ug.mL-1 T09395 CN2K5O 44332505 IC50 = 0.01 ug.mL-1 T09395 CC47JX 44332506 IC50 = 0.04 ug.mL-1 T09395 CX83UG 118165178 IC50 > 100000 nM T09395 CWX3Z7 118165190 IC50 > 100000 nM T09395 C3S5OA 118165200 IC50 = 105 nM T09395 C95RGM 118165205 IC50 = 23100 nM T09395 C3Y0TE 118165222 IC50 > 100000 nM T09395 CE9Z3K 118165243 IC50 = 163 nM T09395 C2VZW7 118165257 IC50 = 385 nM T09395 CIJN30 118165260 IC50 = 765 nM T09395 CA8YG6 118165270 IC50 > 100000 nM T09395 C84VSY 118165287 IC50 = 123 nM T09395 C6X5HK 118165290 IC50 = 36 nM T09395 CNFT52 118165293 IC50 > 100000 nM T09395 CB59GF 118165313 IC50 = 175 nM T09395 CFIV09 118165354 IC50 = 389 nM T09395 CZ8RQ9 118165413 IC50 = 1011 nM T09395 C3F6XG 118165440 IC50 = 232 nM T09395 CWI08V 118165445 IC50 = 4160 nM T09395 CA9E0U 118165472 IC50 = 1525 nM T09395 CDAC50 118165497 IC50 = 384 nM T09395 CWP90I 118165555 IC50 > 100000 nM T09395 CM6JI8 118165621 IC50 = 945 nM T09395 C8V1IU 118165625 IC50 = 1175 nM T09395 CNPW85 118165709 IC50 = 149 nM T09395 CAZ25P 118165748 IC50 = 2255 nM T09395 C65DLT 118165752 IC50 > 100000 nM T09395 CA9UQ1 118165756 IC50 = 123 nM T09395 CATZ25 118165760 IC50 > 100000 nM T09395 CN4O5K 118165763 IC50 = 84 nM T09395 CR5HV8 121410292 IC50 = 870 nM T09395 CVE96K 121410294 IC50 = 495 nM T09395 CK9G7V 121410328 IC50 = 1800 nM T09395 CQ3KL4 121410329 IC50 = 1430 nM T09395 CBN62U 121410340 IC50 = 1900 nM T09395 CNF06J 121410352 IC50 = 1200 nM T09395 CR70JL 126641909 IC50 = 41 nM T09395 CT7M6Q 126641926 IC50 = 82 nM T09395 CLG67Z 126641948 IC50 = 48 nM T09395 CVAC39 126641974 IC50 = 580 nM T09395 C1ZTB7 126641995 IC50 = 44 nM T09395 CA81IH 126642266 IC50 = 47 nM T09395 CNJL38 126642277 IC50 = 59 nM T09395 CIW02N 126642282 IC50 = 87 nM T09395 CO09EN 155514507 IC50 = 180 nM T09395 CGWL21 155515495 IC50 = 1850 nM T09395 CPZ1J2 155515757 IC50 = 530 nM T09395 CVS35D 155518925 IC50 = 395 nM T09395 CS0ER5 155528109 IC50 = 330 nM T09395 C2WPD6 155530588 IC50 = 21 nM T09395 CYH2Z6 155530878 IC50 = 145 nM T09395 CGKM58 155542422 IC50 = 44 nM T09395 CN9LP5 155551221 IC50 = 27 nM T09395 CGV1M3 155552611 IC50 = 505 nM T09395 CM5VI1 155561970 IC50 = 19500 nM T94879 D05MQK 110635 IC50 = 1.2 nM T94879 D0C9SY 135400189 Ki = 0.7 nM T94879 D0F9GE 3108 IC50 = 574 nM T94879 D0NJ3V 4680 IC50 = 8800 nM T94879 D0Y5JC 9869929 Ki = 5 nM T94879 D0Y9ZE 4197 IC50 = 740 nM T94879 D0Z7ZM 135398744 Ki = 1.6 nM T94879 D03QJL 3671 IC50 = 103000 nM T94879 D05OQG 5318997 IC50 = 5900 nM T94879 D09OCK 135430955 IC50 = 4.2 nM T94879 D0A9IY 135564558 IC50 > 10000 nM T94879 D0L0BX 5318980 IC50 = 2200 nM T94879 D0M9FQ 11465695 IC50 = 0.5012 nM T94879 D0T5PO 5092 IC50 = 720 nM T94879 D05VBJ 71295299 IC50 > 10000 nM T94879 D0WS3T 72706254 IC50 = 260 nM T94879 D00SPK 23665864 IC50 = 3.7 nM T94879 D00YPW 135399235 Ki = 130 nM T94879 D01QUF 9842576 Ki > 100000 nM T94879 D02EMR 151170 IC50 > 10000 nM T94879 D05VLN 55690 IC50 = 58000 nM T94879 D0BK6B 3021729 IC50 > 10000 nM T94879 D0F0CS 5723 IC50 > 10000 nM T94879 D0K2BQ 71356 Ki = 7500 nM T94879 D0N5SC 135536943 IC50 = 1.23 nM T94879 D0W8OH 135529458 IC50 = 80 nM T94879 CVQ0G5 1348 IC50 = 500 nM T94879 C03NGJ 1713 IC50 = 230 nM T94879 CH8J2B 4977 Ki = 600000 nM T94879 CCJ8F0 5353 IC50 = 21000 nM T94879 C3B8VG 5369 IC50 = 1 nM T94879 CAMB41 100554 IC50 = 5500 nM T94879 C9T3FB 105007 IC50 = 1580 nM T94879 CGA17S 127779 Ki = 6500 nM T94879 C1H8NR 155248 IC50 > 50000 nM T94879 CH2P8A 158961 Ki = 600000 nM T94879 CVN23X 158962 Ki = 600000 nM T94879 CL27HC 160179 IC50 = 9300 nM T94879 CYWS98 185848 IC50 > 40000 nM T94879 C78DLE 205964 IC50 = 360 nM T94879 C1B6ZL 662965 IC50 > 50000 nM T94879 C3A4HW 675226 IC50 = 8600 nM T94879 CA56MW 675227 IC50 = 3900 nM T94879 CHAB75 696516 IC50 = 1900 nM T94879 CW2U6N 698956 IC50 = 420 nM T94879 CYBA13 719250 IC50 = 4700 nM T94879 C1HM0K 832282 IC50 = 4300 nM T94879 C9KVI7 832283 IC50 = 22000 nM T94879 CM6Q1D 869895 IC50 = 2400 nM T94879 C6QBR5 874599 IC50 = 540 nM T94879 CR7A3U 930420 IC50 = 1200 nM T94879 CWIA36 987187 IC50 = 5600 nM T94879 CT62PH 987189 IC50 = 3100 nM T94879 CO0Z8N 1002275 IC50 = 1700 nM T94879 CXQ4P8 1183964 IC50 = 860 nM T94879 CZQ09F 1204882 IC50 = 7200 nM T94879 CHP0S3 1204883 IC50 = 570 nM T94879 C0JM2Q 1215407 IC50 = 700 nM T94879 CZ2XI5 1271431 IC50 = 3100 nM T94879 COW58U 1277329 IC50 = 190 nM T94879 C6VF0S 1490272 IC50 = 840 nM T94879 CQ69OY 1490552 IC50 = 1100 nM T94879 CD0G9E 1553819 IC50 = 14000 nM T94879 CYD6E3 1553838 IC50 = 190 nM T94879 CXP17G 1604254 IC50 = 4600 nM T94879 C8JLO0 2243267 IC50 = 370 nM T94879 CTQ23N 2452792 IC50 = 800 nM T94879 CLNU08 2456309 IC50 = 740 nM T94879 CYP23V 2465033 IC50 = 800 nM T94879 CE70KT 2471983 IC50 = 1200 nM T94879 CE4D1W 2789492 IC50 = 5600 nM T94879 CFC30O 2789499 IC50 = 1000 nM T94879 C4LSR7 2886111 IC50 > 10000 nM T94879 C6AT3L 2930929 IC50 = 6300 nM T94879 CD70ZG 3119958 IC50 = 8700 nM T94879 C4MSC9 3120507 IC50 = 3000 nM T94879 CPX4V3 4352680 IC50 = 130620 nM T94879 C5IZS9 4636426 IC50 = 746450 nM T94879 CC3LA4 4672917 IC50 = 8500 nM T94879 C5P0LU 4672918 IC50 = 29300 nM T94879 C3JHM8 4687521 IC50 = 1.2 nM T94879 C0JVX6 4867627 IC50 = 4900 nM T94879 CN0Z3D 4880961 IC50 = 11000 nM T94879 C0C9HP 6610310 IC50 = 19 nM T94879 CAYS61 6918354 IC50 = 4000 nM T94879 CB40PM 6918356 IC50 = 200 nM T94879 CI7K0P 6918667 IC50 = 69800 nM T94879 CP1GO7 6918668 IC50 > 84900 nM T94879 CA05PF 6918674 IC50 = 700 nM T94879 C87WYR 6918795 IC50 > 67300 nM T94879 CRGE51 6918796 IC50 > 101000 nM T94879 CUP4M8 6918797 IC50 > 50700 nM T94879 C0LRO8 6918798 IC50 > 101000 nM T94879 C53ESK 6918799 IC50 > 91000 nM T94879 CU1E0G 6918800 IC50 > 101000 nM T94879 CRU46D 7161211 IC50 = 3250 nM T94879 CQ41MA 8055545 IC50 = 2300 nM T94879 CZF0N3 8055573 IC50 = 2400 nM T94879 CN86QP 8078832 IC50 = 2500 nM T94879 CI15SH 9797222 IC50 = 14000 nM T94879 CNC2F4 9798336 IC50 > 1000000 nM T94879 CFJ62Y 9799389 IC50 > 10000 nM T94879 CZH08Y 9802738 IC50 = 7.2 nM T94879 CDV76T 9803328 Ki = 0.29 nM T94879 CR09LM 9805655 IC50 = 0.3 nM T94879 CB57DJ 9807085 IC50 = 72 nM T94879 CXF0J7 9818343 IC50 = 10 nM T94879 C1CXA5 9818702 IC50 = 5000 nM T94879 CSOX21 9819114 IC50 = 2.8 nM T94879 C1MN3A 9821924 IC50 = 2 nM T94879 C7FY1U 9824408 IC50 = 1.1 nM T94879 C4J2XE 9836643 IC50 > 101000 nM T94879 C4YB1S 9844037 IC50 = 5.3 nM T94879 C5YQB0 9859898 IC50 = 78000 nM T94879 CZGM43 9864862 IC50 = 22000 nM T94879 CEI5P4 9868140 IC50 = 440 nM T94879 C92GMV 9879320 IC50 = 13000 nM T94879 C0Q5VN 9880010 IC50 > 101000 nM T94879 CWD1F6 9880288 IC50 > 101000 nM T94879 C2NK8E 9888568 IC50 = 0.56 nM T94879 C0P8ZH 9892886 Ki = 0.21 nM T94879 CC05QE 9901606 IC50 = 101000 nM T94879 CMBO89 9912467 IC50 = 2000 nM T94879 CBA29H 9922545 IC50 > 101000 nM T94879 CKF4C2 9922691 IC50 = 73200 nM T94879 CY17NM 9922999 IC50 = 8400 nM T94879 C70AMC 9924305 IC50 = 7270 nM T94879 CKI6N2 9924468 IC50 > 88000 nM T94879 C6AZ5F 9924709 IC50 > 101000 nM T94879 C54ICU 9927654 IC50 = 3500 nM T94879 C60BWM 9933503 IC50 = 0.8 nM T94879 CX1UV7 9946954 IC50 = 20160 nM T94879 C7OP5A 9947052 IC50 = 3970 nM T94879 C04HAV 9949594 IC50 = 225 nM T94879 C53AVJ 9951793 IC50 = 2.3 nM T94879 CE8ZD7 9954790 IC50 = 0.93 nM T94879 CH46TF 9954942 Ki = 0.23 nM T94879 C8X7RN 9956576 IC50 = 0.1 nM T94879 C2OYA1 9957043 IC50 = 0.55 nM T94879 CJO0X4 9966737 IC50 = 10940 nM T94879 CFP1Y5 9966830 IC50 > 101000 nM T94879 C9NKY4 9967652 IC50 = 74000 nM T94879 CI6AX1 9968005 IC50 > 101000 nM T94879 C7PCS8 9968050 IC50 = 40350 nM T94879 CFB48Q 9968370 IC50 = 98000 nM T94879 CU73AJ 9968471 IC50 > 101000 nM T94879 C0AP8O 9969020 IC50 = 17880 nM T94879 C9X7PF 9972372 IC50 = 8800 nM T94879 CL6V2I 9973407 IC50 = 770 nM T94879 CCDX84 9973586 IC50 = 0.53 nM T94879 C5AE2I 9973597 IC50 > 200000 nM T94879 CTQ59Y 9975543 IC50 = 3600 nM T94879 CW3S7O 9977675 IC50 > 1000000 nM T94879 C05RPA 9977814 IC50 = 2700 nM T94879 C20XIY 9985391 IC50 = 2200 nM T94879 CHG4K5 9992525 IC50 = 64000 nM T94879 CO87TV 9994528 IC50 = 100 nM T94879 CC86WM 9995163 IC50 = 6800 nM T94879 CB9EY5 9995187 IC50 = 90 nM T94879 CWJ0K5 9995367 IC50 = 210 nM T94879 CZR07N 9995467 IC50 = 930 nM T94879 C3GHJ7 9996490 IC50 = 105 nM T94879 CH70VI 9996675 IC50 = 1100 nM T94879 CE5O4D 9998316 IC50 = 350 nM T94879 CYS20P 10004422 IC50 = 38000 nM T94879 CB41WF 10017397 IC50 = 3000 nM T94879 CKE92N 10017795 IC50 = 3600 nM T94879 CHJ73C 10018556 IC50 = 8700 nM T94879 CI9WK7 10021158 IC50 = 1300 nM T94879 C6MUC5 10024867 IC50 = 2500 nM T94879 C5E4QJ 10030897 Ki = 0.24 nM T94879 C1G5XC 10032458 IC50 = 6500 nM T94879 CE25WO 10039122 IC50 = 4400 nM T94879 CUYW65 10039809 IC50 = 20000 nM T94879 C0SZB8 10039848 IC50 = 36300 nM T94879 CJ1Q7Z 10040540 IC50 = 50 nM T94879 CJ05CZ 10040882 IC50 = 15000 nM T94879 CK5VB0 10041530 IC50 = 14000 nM T94879 C9FD1X 10041853 IC50 = 7500 nM T94879 CT6Y9J 10043209 IC50 > 1000000 nM T94879 CY6FQ4 10053217 IC50 = 3 nM T94879 CD1N4K 10062262 IC50 = 1000 nM T94879 CHCJ86 10065791 IC50 = 810 nM T94879 CC6PO8 10066654 IC50 > 40000 nM T94879 C3MA2L 10067044 IC50 > 1000000 nM T94879 C5FCT6 10070215 IC50 = 0.6 nM T94879 COSV65 10074226 Ki = 0.23 nM T94879 CG39NX 10083598 IC50 = 40000 nM T94879 C5P7AS 10083609 IC50 = 6000 nM T94879 C7YBR0 10083610 IC50 = 33000 nM T94879 CAX67L 10084334 IC50 = 3000 nM T94879 CP6W8T 10086869 IC50 = 18500 nM T94879 CLB5S6 10087203 IC50 = 11000 nM T94879 CNA75V 10087755 IC50 = 1400 nM T94879 CJ16FV 10087963 IC50 > 1000000 nM T94879 CSP05N 10088555 IC50 = 730 nM T94879 CRW6E1 10088941 IC50 > 40000 nM T94879 C09ZNQ 10088960 IC50 = 2.6 nM T94879 C0O6MQ 10089225 IC50 = 2300 nM T94879 C13QUP 10089597 IC50 = 65000 nM T94879 CARY56 10091146 IC50 > 200000 nM T94879 CP8I5O 10093297 IC50 = 9800 nM T94879 CS4QG0 10095269 IC50 = 900 nM T94879 C61QRH 10096810 IC50 = 49000 nM T94879 CN23KJ 10105662 IC50 = 18000 nM T94879 CP3D7N 10108060 IC50 = 6000 nM T94879 C12LED 10109572 IC50 > 101000 nM T94879 CT0A4J 10113055 IC50 = 9 nM T94879 CPWL59 10113972 IC50 = 8 nM T94879 C5GRV3 10117157 IC50 = 56 nM T94879 C2PBD6 10131447 IC50 = 19300 nM T94879 C3AOI5 10138533 IC50 = 134 nM T94879 C8XPO7 10145438 Ki = 0.2 nM T94879 C4F3SH 10151707 IC50 = 1.585 nM T94879 C3H1IG 10161792 IC50 = 750 nM T94879 C89DXP 10181676 IC50 = 6 nM T94879 C5HC2X 10182563 IC50 = 52400 nM T94879 CK3TY8 10187239 IC50 = 2.089 nM T94879 CJZK81 10195399 IC50 = 1.9 nM T94879 C3GN8K 10200432 IC50 > 101000 nM T94879 CK81LJ 10203901 Ki = 4 nM T94879 CEY6F7 10205437 IC50 = 10.96 nM T94879 CLW92Y 10205894 IC50 = 65 nM T94879 CULN70 10206649 Ki = 0.31 nM T94879 C8JR4W 10221093 IC50 = 44000 nM T94879 CFGO46 10221904 IC50 = 60000 nM T94879 C8V6FE 10225063 IC50 = 2 nM T94879 CX35CL 10244508 IC50 = 6200 nM T94879 CGA50J 10244709 IC50 = 230 nM T94879 CT7RC0 10245770 IC50 = 15000 nM T94879 CC80XO 10247363 IC50 = 620 nM T94879 CP4YR0 10248176 IC50 > 1000000 nM T94879 C8G3BJ 10249105 IC50 = 3.5 nM T94879 C7MQZ1 10249183 IC50 > 1000000 nM T94879 C3AFN6 10250999 IC50 = 8300 nM T94879 CRK1U0 10252045 IC50 = 53000 nM T94879 C7GTC0 10264205 IC50 = 3020 nM T94879 C5VQL9 10264224 IC50 = 26000 nM T94879 CP70US 10267904 IC50 = 13800 nM T94879 CQ61CV 10268304 IC50 = 68400 nM T94879 C1QU2B 10268305 IC50 = 9470 nM T94879 C1VL9A 10269511 IC50 = 0.48 nM T94879 CH9C4K 10269859 IC50 = 23600 nM T94879 CR92JY 10270352 IC50 > 101000 nM T94879 C7CHR0 10270536 IC50 = 12600 nM T94879 C1VH6L 10279632 Ki = 8 nM T94879 C1FA4P 10288830 IC50 = 1.6 nM T94879 C3YO7N 10289243 IC50 = 1.288 nM T94879 CISQ36 10291967 IC50 = 63000 nM T94879 CKR74B 10292282 IC50 = 840 nM T94879 CA54BI 10294138 IC50 = 4 nM T94879 CKQ8I4 10313609 IC50 = 860 nM T94879 CUE72P 10314633 IC50 = 16 nM T94879 CJO72N 10315684 IC50 = 14 nM T94879 CIPN48 10316358 IC50 = 22000 nM T94879 C36AGZ 10321525 IC50 = 240 nM T94879 C90QZM 10324834 IC50 = 2.1 nM T94879 CRJW04 10334696 IC50 = 4000 nM T94879 C5K1LH 10336744 IC50 = 480 nM T94879 C6AQ0U 10338401 IC50 > 200000 nM T94879 C4GB5L 10338602 IC50 = 38 nM T94879 C52EPV 10339653 IC50 > 1000000 nM T94879 CMJG73 10342601 IC50 = 1200 nM T94879 CK05FV 10343476 IC50 = 68000 nM T94879 C32IUF 10344870 IC50 = 40000 nM T94879 CHZL20 10345264 IC50 = 1.6 nM T94879 CA18KO 10347662 IC50 = 20000 nM T94879 CC4W3M 10349233 IC50 = 24000 nM T94879 CQD9O7 10355498 IC50 = 6000 nM T94879 C4BL9Q 10358104 IC50 = 20000 nM T94879 CG8V6F 10358836 IC50 = 9000 nM T94879 CEIW08 10359077 IC50 = 175000 nM T94879 CP5S1A 10359273 IC50 = 165 nM T94879 C7QYK3 10359377 IC50 = 2150 nM T94879 CR35FX 10378878 IC50 = 15000 nM T94879 C2H9SE 10380126 IC50 = 4000 nM T94879 C6E5OY 10380621 IC50 = 5900 nM T94879 C5EVH3 10381520 IC50 = 380 nM T94879 C0J7OV 10382041 IC50 = 11000 nM T94879 C9IK3H 10382413 IC50 = 120 nM T94879 C52DNX 10384462 IC50 = 5500 nM T94879 CF6A1Q 10385088 IC50 > 200000 nM T94879 CZ6X9Y 10391444 IC50 = 3100 nM T94879 CQOX84 10393352 IC50 = 3.5 nM T94879 C9-APR-07 10394586 IC50 = 34000 nM T94879 CI8B3P 10401473 IC50 = 1000 nM T94879 C6E0PG 10401818 IC50 = 2000 nM T94879 C7X4EW 10402019 IC50 = 630 nM T94879 C78SRU 10403787 IC50 = 72 nM T94879 CUF0X6 10404302 IC50 > 1000000 nM T94879 C0ADP3 10404378 IC50 = 56000 nM T94879 CV3I5E 10405045 IC50 = 380 nM T94879 CP8ZV5 10408375 IC50 = 140 nM T94879 C4BF5Y 10411270 IC50 = 1.4 nM T94879 CQUE27 10413015 IC50 = 37000 nM T94879 CS7J4V 10414339 IC50 = 16 nM T94879 C0ZLB5 10423102 IC50 = 1000 nM T94879 C5ZQG3 10426854 IC50 = 5500 nM T94879 C5HMX2 10428149 IC50 = 32000 nM T94879 CB2X9W 10429802 IC50 = 110 nM T94879 CAW23H 10434818 IC50 > 1000000 nM T94879 CH76CS 10443650 IC50 = 42000 nM T94879 CBH5V4 10445800 IC50 = 24000 nM T94879 CZ8IC4 10448177 IC50 > 1000000 nM T94879 CYU38H 10448853 IC50 = 1600 nM T94879 C1RZ9E 10449000 IC50 > 1000000 nM T94879 C18EHX 10449737 IC50 = 1300 nM T94879 CU2HN6 10450290 IC50 > 200000 nM T94879 C9IF7Y 10451065 IC50 = 4.8 nM T94879 CY4O0K 10452443 IC50 = 38000 nM T94879 CI1H7F 10452463 IC50 = 0.05 nM T94879 C4LOK1 10454517 IC50 = 3600 nM T94879 CR04LJ 10456913 IC50 = 54000 nM T94879 CASV91 10466228 IC50 = 34000 nM T94879 C6IP3N 10468291 IC50 = 24000 nM T94879 C6PXC2 10471556 IC50 = 31 nM T94879 C2FYT6 10471617 IC50 = 2300 nM T94879 C2DEO3 10472374 IC50 > 200000 nM T94879 CBMI84 10473521 IC50 = 810 nM T94879 CF0I6O 10479155 IC50 = 13000 nM T94879 C5CI3G 10479468 IC50 = 53000 nM T94879 CZ92DR 10481735 IC50 = 9 nM T94879 CE2RJ7 10499713 IC50 = 420 nM T94879 C0N5LU 10504068 IC50 = 0.53 nM T94879 C71AJB 10520277 IC50 = 19 nM T94879 CSZ7L0 10520799 IC50 = 19 nM T94879 CPWU60 10524067 IC50 = 8000 nM T94879 CG1QK8 10542139 IC50 = 6200 nM T94879 C7LG4O 10543051 IC50 = 26000 nM T94879 C7K5PG 10544204 IC50 = 26 nM T94879 C0Z1CT 10546352 IC50 = 63 nM T94879 CCK5F8 10549901 IC50 = 120 nM T94879 CMK39Q 10553487 IC50 = 200 nM T94879 CQW79N 10554042 IC50 = 10000 nM T94879 CTYQ03 10565296 IC50 = 7500 nM T94879 C1DO9H 10573238 IC50 = 275 nM T94879 CI8GS1 10574005 IC50 = 590 nM T94879 CY9P5W 10575733 IC50 = 30000 nM T94879 CFY5J3 10576937 IC50 = 305 nM T94879 CYD4Z2 10592106 IC50 = 140 nM T94879 C4HVR8 10595830 IC50 = 5600 nM T94879 CRKT15 10597744 IC50 = 43 nM T94879 C71YLE 10598277 IC50 = 4 nM T94879 CJ7CU4 10603606 IC50 = 1000 nM T94879 CR9H4Z 10617782 IC50 = 4500 nM T94879 CK3GR5 10624131 IC50 = 20000 nM T94879 C25WRZ 10627119 IC50 = 9000 nM T94879 CC68NQ 10636956 IC50 = 100 nM T94879 CE57IW 10639502 IC50 = 3300 nM T94879 C0U8KD 10642598 IC50 = 10000 nM T94879 CX61NW 10642809 IC50 = 810 nM T94879 CNK65G 10646809 IC50 = 100000 nM T94879 CKNA14 10648008 IC50 = 20000 nM T94879 C32TRJ 10659857 IC50 = 240 nM T94879 C9GJ5K 10660011 IC50 = 13000 nM T94879 C8KWM5 10663015 IC50 = 34 nM T94879 CP13SC 10663562 IC50 = 80 nM T94879 COQ17R 10666144 IC50 = 9200 nM T94879 CBQ24O 10668762 IC50 = 4000 nM T94879 C1R9VY 10669652 IC50 = 110 nM T94879 CB9Y7A 10669693 IC50 = 40000 nM T94879 CWYZ15 10670833 IC50 = 2 nM T94879 C2Y5HF 10675032 IC50 = 800 nM T94879 CW12SY 10690095 IC50 = 510 nM T94879 CV6WT3 10692240 IC50 > 30000 nM T94879 C29YKI 10692613 IC50 = 1200 nM T94879 C0FPL8 10692684 IC50 = 800 nM T94879 CI6ON5 10698519 IC50 = 4000 nM T94879 C2JTX7 10715358 IC50 = 400 nM T94879 C1I8VM 10716045 IC50 = 1500 nM T94879 CDMP96 10717370 IC50 = 30000 nM T94879 CCI8R7 10729204 IC50 > 100000 nM T94879 C2P5VY 10731865 IC50 = 610 nM T94879 CSQG30 10741916 IC50 = 0.55 nM T94879 CTCS25 10753773 IC50 = 100 nM T94879 C3X8UM 10754735 IC50 = 800 nM T94879 C4EG9Z 10759241 IC50 = 19 nM T94879 CEIZ87 10761565 IC50 = 54 nM T94879 CINX82 10763354 IC50 = 20000 nM T94879 COVG15 10764868 IC50 = 120 nM T94879 C51XRM 10776762 IC50 = 2400 nM T94879 CR4O8B 10781567 IC50 = 16000 nM T94879 C7O8WB 10787783 IC50 = 180 nM T94879 CLM42P 10788651 IC50 = 20000 nM T94879 C7U2NT 10808382 IC50 = 140 nM T94879 CEI0J8 10809340 IC50 = 49 nM T94879 CDF43L 10810826 IC50 = 66 nM T94879 CTMX70 10815441 IC50 = 58000 nM T94879 CA9UW6 10816539 IC50 = 200 nM T94879 C5V1AY 10828080 IC50 = 60 nM T94879 C0SEG5 10830345 IC50 = 6000 nM T94879 CI0XH5 10833134 IC50 = 98 nM T94879 CT6VP3 10834312 IC50 = 560 nM T94879 C8HY0A 10835448 IC50 = 11 nM T94879 CZY5K8 10836947 IC50 = 600 nM T94879 CG2O1B 10836974 IC50 = 200 nM T94879 CR50XV 10841036 IC50 = 40000 nM T94879 CJ0TR9 10854527 IC50 = 100 nM T94879 CW3T1L 10863491 Ki = 154 nM T94879 C9TH7M 10863695 Ki = 1.75 nM T94879 CH0B6V 10885231 Ki = 188 nM T94879 CQ8YB7 10897309 Ki = 1.78 nM T94879 C0RTU9 10897531 EC50 = 9.5 nM T94879 CG0LM2 10907083 Ki = 0.4 nM T94879 CB6U4L 10929261 Ki = 0.47 nM T94879 CL1RW3 10929391 Ki = 0.21 nM T94879 C0BS9L 10939795 Ki = 0.71 nM T94879 C4KLI7 10951390 Ki = 1.14 nM T94879 C9UXZ6 10951441 Ki = 1.01 nM T94879 CP59RB 10968191 IC50 = 22300 nM T94879 C3GAM5 10973079 IC50 = 0.03 nM T94879 C96GWI 10983515 IC50 = 0.7 nM T94879 C84LQY 10983963 Ki = 2.59 nM T94879 CJCO78 10992580 Ki = 1.08 nM T94879 CKX30W 10994934 Ki = 0.61 nM T94879 C3EH8D 11006014 Ki = 24.7 nM T94879 CF7RW4 11016445 Ki = 2.64 nM T94879 CX1GO8 11016581 Ki = 2.71 nM T94879 CR7C1N 11017676 EC50 = 12 nM T94879 CO05WV 11024165 IC50 = 3900 nM T94879 CJMS98 11025421 Ki = 1.2 nM T94879 C3QT7I 11028215 Ki = 0.53 nM T94879 C98IUO 11039211 Ki = 0.76 nM T94879 CF6BL1 11049430 Ki = 62.8 nM T94879 C7B4MG 11071221 Ki = 1.71 nM T94879 CIO28H 11092703 Ki = 0.99 nM T94879 CG74CI 11093245 EC50 = 130 nM T94879 CW2AS4 11103879 Ki = 0.29 nM T94879 CRV32I 11114031 Ki = 3.74 nM T94879 C72TWL 11123617 Ki = 246 nM T94879 CX3N0E 11123630 Ki = 0.31 nM T94879 C24VFA 11125005 EC50 = 37 nM T94879 CL3DT7 11145432 Ki = 0.73 nM T94879 CU5C3E 11145600 Ki = 0.61 nM T94879 C3B1QP 11161553 IC50 = 21000 nM T94879 C6OH2Y 11212743 Ki = 0.22 nM T94879 CA8E0W 11212836 Ki = 0.58 nM T94879 C0FSV9 11225074 IC50 = 0.07 nM T94879 C8TD3U 11247946 IC50 = 0.14 nM T94879 C01VJK 11270159 Ki = 23.3 nM T94879 CF7R3Y 11270592 Ki = 1.06 nM T94879 C26HWL 11270869 IC50 = 0.78 nM T94879 C4R1UG 11270952 Ki = 11 nM T94879 CRZ9V8 11293623 Ki = 3.48 nM T94879 CGO29X 11318932 IC50 = 7600 nM T94879 CY9O2K 11351010 Ki = 0.35 nM T94879 CY71CZ 11351116 Ki = 4.53 nM T94879 C1YTA6 11351932 Ki = 118 nM T94879 CREQ98 11373312 IC50 = 95000 nM T94879 C4H9WX 11375723 IC50 = 320 nM T94879 CVT52P 11385644 Ki = 113 nM T94879 CPJ0Z3 11396900 Ki = 601 nM T94879 C4V6DZ 11418838 Ki = 12.5 nM T94879 C45VZC 11438405 IC50 > 16000 nM T94879 CKZ43J 11496164 IC50 = 0.08 nM T94879 CO9WX8 11497051 IC50 = 1.7 nM T94879 CS5P1N 11502459 IC50 = 2.1 nM T94879 C7S4QZ 11539946 IC50 = 1.01 nM T94879 C4ZYH9 11547485 IC50 = 2.5 nM T94879 C50BPN 11554196 IC50 = 0.65 nM T94879 CJ41RB 11560313 IC50 = 0.4 nM T94879 CJ1R6X 11568346 IC50 = 0.007 nM T94879 CL83VR 11574797 IC50 = 0.65 nM T94879 C86YZS 11575452 IC50 = 0.78 nM T94879 C53ARX 11582654 IC50 = 9.52 nM T94879 C1TOQ3 11583812 IC50 = 6.48 nM T94879 CY5JK4 11589901 IC50 = 34 nM T94879 CI6AW2 11590842 IC50 = 0.09 nM T94879 C58OXQ 11596704 IC50 = 3.3 nM T94879 CG5LT6 11605112 IC50 = 3.15 nM T94879 C7JLT3 11611915 IC50 = 0.07 nM T94879 CLU3G9 11639525 IC50 = 10 nM T94879 CO6XA4 11647832 IC50 = 0.72 nM T94879 CRK10B 11669288 IC50 = 67 nM T94879 C0B7RV 11675647 IC50 = 1.5 nM T94879 C1WV4T 11682414 IC50 = 0.5 nM T94879 C5LPU2 11690391 IC50 = 0.76 nM T94879 C5PHZ0 11710213 IC50 = 1300 nM T94879 CT69CO 11718514 IC50 = 2.6 nM T94879 C1RX0I 11720166 IC50 = 0.35 nM T94879 C7BAC0 11724504 IC50 = 4300 nM T94879 CM5T9U 11724564 IC50 = 35000 nM T94879 CNL0G1 11725859 IC50 = 10 nM T94879 C0AKJ4 11742456 IC50 > 100000 nM T94879 CA1E6R 11754694 Ki = 0.53 nM T94879 C26CKE 11754697 IC50 = 300 nM T94879 C6ERQ9 11755313 Ki = 18 nM T94879 CMP35Y 11762536 Ki = 0.15 nM T94879 C57BPZ 11763070 Ki = 1.3 nM T94879 C1K3JX 11764545 IC50 = 37000 nM T94879 CF23VJ 11775013 IC50 = 0.5012 nM T94879 C23DSJ 11782534 IC50 = 9300 nM T94879 C5EFC7 11793221 IC50 = 1000 nM T94879 CGA1F8 11794425 IC50 = 3000 nM T94879 CUM8A9 11795949 IC50 = 4300 nM T94879 C3LO2Q 11799196 IC50 = 3.1 nM T94879 C0GP6R 11812647 Ki = 0.35 nM T94879 C1J9UP 11813138 Ki = 0.52 nM T94879 CMU6W8 11826705 Ki = 1.74 nM T94879 CB4RS5 11826881 Ki = 2.09 nM T94879 C29HOL 11828590 EC50 = 44 nM T94879 CT5C0K 11849942 IC50 = 100 nM T94879 CS42FO 11849943 IC50 = 240 nM T94879 C2FZY3 11850012 IC50 = 470 nM T94879 CRY1U7 11850013 IC50 = 140 nM T94879 CVJ1X4 11850014 IC50 = 50 nM T94879 CAPF41 11850015 IC50 = 180 nM T94879 C4GQ2P 11850016 IC50 = 38 nM T94879 C4YP5D 11850079 IC50 = 40 nM T94879 C8VUW0 11850080 IC50 = 23 nM T94879 CJ6ZX9 11850081 IC50 = 8.3 nM T94879 CQ2JU9 11850082 IC50 = 79 nM T94879 CSI25Y 11850083 IC50 = 95 nM T94879 CW6D5J 11850144 IC50 = 370 nM T94879 CT9LD7 11850145 IC50 = 1500 nM T94879 C14ZXU 11850147 IC50 = 390 nM T94879 CU7X9W 11850294 IC50 = 71 nM T94879 C8ZM2F 11850366 IC50 = 220 nM T94879 CLI6G9 11850367 IC50 = 100 nM T94879 CC59AF 11850439 IC50 = 1400 nM T94879 CUK49V 11988837 Ki = 600 nM T94879 CFIO49 11988967 Ki = 1600 nM T94879 C2D0NG 11989101 Ki = 590 nM T94879 C65ABT 11989102 Ki = 1200 nM T94879 C05CLB 11992443 IC50 = 0.68 nM T94879 C0Z3KV 11992527 IC50 = 0.9 nM T94879 CXW57M 11992528 IC50 = 0.26 nM T94879 CH86SQ 11992529 IC50 = 0.11 nM T94879 CIX0V4 11992531 IC50 = 1.05 nM T94879 C7X4LC 11992631 IC50 = 0.78 nM T94879 C1B4XD 11992634 IC50 = 0.05 nM T94879 CAG1U6 11992635 IC50 = 0.1 nM T94879 CHT82G 11992739 IC50 = 0.09 nM T94879 CR4CA6 11992740 IC50 = 0.14 nM T94879 CIOU94 11992741 IC50 = 0.25 nM T94879 C95DJC 11992742 IC50 = 0.24 nM T94879 C0KM5I 11992827 IC50 = 1.1 nM T94879 CM57ID 11992831 IC50 = 0.07 nM T94879 CPX16N 11993169 IC50 = 0.07 nM T94879 C0Q4KT 11993170 IC50 = 0.04 nM T94879 C3HOV8 11993171 IC50 = 0.05 nM T94879 CZ7YR6 11993243 IC50 = 2.59 nM T94879 C4VY3X 11993244 IC50 = 0.34 nM T94879 CP4J1S 11993342 IC50 = 0.14 nM T94879 C0QZ6W 11993365 IC50 = 0.15 nM T94879 COQ5N2 11993435 IC50 = 0.43 nM T94879 C39KLP 11993437 IC50 = 1.17 nM T94879 CL8TM7 11993463 IC50 = 0.13 nM T94879 C1ZDC4 11993465 IC50 = 0.08 nM T94879 CK63SM 11993560 IC50 = 1.65 nM T94879 CIRM68 11993561 IC50 = 0.07 nM T94879 C6W2LU 11993562 IC50 = 0.13 nM T94879 C6VI5Z 12020635 Ki = 126 nM T94879 C48IYW 12020642 Ki = 24 nM T94879 CJC01W 12020645 Ki > 1000 nM T94879 CJ4H1G 12020670 Ki = 123 nM T94879 C6D0MG 12069381 IC50 = 1.4 nM T94879 C6S8LD 12355883 IC50 = 1500 nM T94879 CX0C7I 12993019 Ki = 543 nM T94879 CNR05L 12993020 Ki = 126 nM T94879 CO3G0B 12993027 Ki = 0.98 nM T94879 C09OJP 12993038 Ki = 2.07 nM T94879 CI18JL 13026433 IC50 = 1610 nM T94879 C51CKG 14583584 IC50 = 45500 nM T94879 C2ZX8H 14756622 IC50 = 1000 nM T94879 CVT43Z 15473392 IC50 = 60 nM T94879 C2RT6A 15500912 IC50 = 1.9 nM T94879 C8E4IH 15524307 IC50 = 11 nM T94879 C12BUL 15524308 IC50 = 19 nM T94879 CAC5H0 15606258 IC50 = 91000 nM T94879 C3BI9R 15951010 IC50 > 2000 nM T94879 CW6MV8 15981426 IC50 = 26 nM T94879 CYE3L9 16038477 IC50 = 2.6 nM T94879 C9OF5R 16038616 IC50 = 3.7 nM T94879 C8FJM7 16038617 IC50 = 4.5 nM T94879 C4T6CP 16038618 IC50 = 1.2 nM T94879 CIR42U 16038756 IC50 = 12 nM T94879 CF3UG1 16066664 IC50 = 0.04 nM T94879 CG1V8D 17799315 IC50 = 2.7 nM T94879 C1PZ8C 18734933 IC50 > 16000 nM T94879 C6OJI9 18796635 IC50 = 8900 nM T94879 C1FJL6 18796640 IC50 > 100000 nM T94879 CRJO82 18796649 IC50 = 4000 nM T94879 CA16YO 18796653 IC50 = 780 nM T94879 CKCM70 18796657 IC50 = 2200 nM T94879 C36LEN 18796668 IC50 = 1300 nM T94879 C0L8NR 18796689 IC50 = 1900 nM T94879 CBF8M6 18796697 IC50 = 1000 nM T94879 C3RH7V 18796719 IC50 = 11000 nM T94879 CC2WD9 18796725 IC50 > 100000 nM T94879 CNSH93 18796735 IC50 = 2000 nM T94879 CHK4Z7 18796752 IC50 = 32000 nM T94879 CNZ3I1 18796756 IC50 = 4600 nM T94879 CC1LP2 18796767 IC50 = 1000 nM T94879 C2FN9A 18796769 IC50 = 26000 nM T94879 CUE4A2 18796773 IC50 = 2000 nM T94879 C02JXD 18796791 IC50 = 1700 nM T94879 CQ8I5K 18796795 IC50 = 3500 nM T94879 CDC76R 20299686 IC50 = 26 nM T94879 CNX2D5 20646826 IC50 = 0.86 nM T94879 C36XCM 20646828 IC50 = 4.4 nM T94879 C1H2WT 20709323 IC50 = 1.8 nM T94879 C58VPG 21212519 IC50 = 2100 nM T94879 CXM8E3 21704212 IC50 = 0.79 nM T94879 CRY9Z1 21704213 IC50 = 0.32 nM T94879 CS09OZ 21704217 IC50 = 0.5 nM T94879 CH53WM 21704221 IC50 = 14 nM T94879 C7RK1W 21920272 IC50 = 5180 nM T94879 CH7N9S 21920275 IC50 = 7000 nM T94879 CV04DH 21920370 IC50 > 101000 nM T94879 C97JPF 22004355 IC50 = 6.7 nM T94879 C7DJ9E 22004357 IC50 = 2.6 nM T94879 CY6QT7 22004369 IC50 = 1.7 nM T94879 C2STP3 22004386 IC50 = 6.8 nM T94879 C7ZH2R 22004388 IC50 = 0.3 nM T94879 COM30K 22004392 IC50 = 0.7 nM T94879 C37JNS 22004412 IC50 = 0.7 nM T94879 C64YFT 22226537 IC50 = 553 nM T94879 C5G6BS 22226562 IC50 = 30 nM T94879 C70JWO 22226563 IC50 = 94 nM T94879 C8TEV5 22601583 IC50 = 0.4 nM T94879 C2FMU0 22601651 IC50 = 1.3 nM T94879 CNGD52 22744443 IC50 = 1.2 nM T94879 CMIO49 23527107 IC50 = 100 nM T94879 CZD94A 23527108 IC50 = 19 nM T94879 CW96SI 23624262 IC50 = 561 nM T94879 CXB78L 23624298 IC50 > 5000 nM T94879 C4S6VD 23654252 IC50 > 50000 nM T94879 CAJ57O 24751843 IC50 = 79000 nM T94879 CR0D6X 24751988 IC50 > 400000 nM T94879 CL79TD 24751991 IC50 = 65000 nM T94879 C51ZNR 24774842 IC50 > 5000 nM T94879 CQ19ZC 24775191 IC50 = 3500 nM T94879 C9WGI4 24802717 IC50 = 919 nM T94879 C4Y3FK 24883368 IC50 = 1.6 nM T94879 C5F6SD 24956185 IC50 = 26 nM T94879 CA9PN0 24957913 IC50 = 17 nM T94879 C6EQG2 24963293 IC50 = 0.2 nM T94879 CJ43BX 24963638 IC50 = 0.18 nM T94879 CLDO78 24963639 IC50 = 0.72 nM T94879 CG1BJ3 24965774 IC50 = 0.21 nM T94879 CDC01R 24965775 IC50 = 0.33 nM T94879 CDF34R 24966125 IC50 = 0.22 nM T94879 CNO40A 24966126 IC50 = 0.3 nM T94879 CY0G1A 24966127 IC50 = 0.23 nM T94879 CS56UN 24966128 IC50 = 1.08 nM T94879 CA25UL 24969619 IC50 = 0.31 nM T94879 C3AFU0 25093775 IC50 = 3.28 nM T94879 C93DZI 25147798 IC50 > 50000 nM T94879 CPC08B 25179287 IC50 > 50000 nM T94879 COB03R 25179478 IC50 = 40000 nM T94879 C1AV7L 30105766 IC50 = 8 nM T94879 C43UKE 42628078 IC50 = 2.4 nM T94879 CICF39 42629702 IC50 = 1850 nM T94879 CM3X9S 42629827 IC50 > 1000 nM T94879 CQN26J 42629945 IC50 = 1240 nM T94879 C6O5FX 42630062 IC50 = 2080 nM T94879 C71ZNR 42630180 IC50 = 1440 nM T94879 C4RHY0 42630191 IC50 > 5000 nM T94879 CT6RS9 42630192 IC50 = 5165 nM T94879 CYZL43 42630317 IC50 = 8780 nM T94879 CH42OZ 42630318 IC50 > 5000 nM T94879 C7X5AH 42630437 IC50 = 2050 nM T94879 CEPY38 43826154 IC50 = 200000 nM T94879 CQU19I 44180409 IC50 = 30300 nM T94879 CW8OB3 44243146 Ki = 10600 nM T94879 C19SIQ 44249786 IC50 = 14.5 nM T94879 C03DAV 44249787 IC50 = 2.3 nM T94879 CJ1GS3 44249944 IC50 = 0.9 nM T94879 CAL8X3 44264943 IC50 = 1 nM T94879 C59QCJ 44274690 IC50 = 3.89 nM T94879 C9KV6Y 44274762 IC50 = 6.457 nM T94879 CXA6Y3 44274773 IC50 = 0.61 nM T94879 CF4H9A 44274775 IC50 = 0.8913 nM T94879 CW7J4K 44274797 IC50 = 1.995 nM T94879 C9VK6M 44274798 IC50 = 5.012 nM T94879 CTP4O5 44274817 IC50 = 2.818 nM T94879 CA6J8T 44274920 IC50 = 3000 nM T94879 CV1ZA7 44280486 IC50 = 3.6 nM T94879 CG8R0W 44280487 IC50 = 4 nM T94879 CS0FX4 44280546 IC50 = 2.7 nM T94879 C05SIA 44280556 IC50 = 12.8 nM T94879 CA9KV4 44280558 IC50 = 8.4 nM T94879 CY74KE 44280614 IC50 = 19.8 nM T94879 C4RO9D 44280635 IC50 = 2.5 nM T94879 CH7W2T 44280722 IC50 = 1.2 nM T94879 CTO54N 44280723 IC50 = 0.7 nM T94879 CXRU70 44280792 IC50 = 13.2 nM T94879 CO7NV0 44280794 IC50 = 164 nM T94879 CG8I6M 44280801 IC50 = 57 nM T94879 CDQ8B2 44280847 IC50 = 1.5 nM T94879 C0N3JE 44280911 IC50 = 2 nM T94879 C3DHJ2 44280985 IC50 = 1.9 nM T94879 CA3GF6 44280994 IC50 = 127 nM T94879 CXB40D 44281036 IC50 = 28.6 nM T94879 CA1HN8 44281061 IC50 = 15.7 nM T94879 C7TKW4 44281095 IC50 = 7.1 nM T94879 CK3W1B 44281096 IC50 = 4 nM T94879 CC81DV 44281265 IC50 = 132 nM T94879 CNO94A 44281273 IC50 > 1000 nM T94879 CO1L0H 44282267 IC50 = 160 nM T94879 C79RGL 44282685 IC50 = 270 nM T94879 CK8Y4F 44286951 IC50 = 160 nM T94879 CNW8B7 44287071 IC50 = 73 nM T94879 CDHP47 44287318 IC50 = 0.6 nM T94879 C2O0JN 44307127 IC50 = 530 nM T94879 C2FW1A 44310350 IC50 = 2900 nM T94879 COP54Y 44318505 IC50 = 1.5 nM T94879 CK0N6P 44318516 IC50 = 0.95 nM T94879 C4AWN5 44318518 IC50 = 1.23 nM T94879 CP30VE 44318806 IC50 = 0.73 nM T94879 CH4T3J 44318846 IC50 = 0.7 nM T94879 CKLM51 44318862 IC50 = 150 nM T94879 CX5SO4 44320719 IC50 = 77 nM T94879 C1SI7O 44320739 IC50 = 551 nM T94879 C3TZ6O 44320740 IC50 = 105 nM T94879 CH18VT 44320762 IC50 = 135 nM T94879 C45ZJD 44320781 IC50 = 130 nM T94879 CF1DO2 44320804 IC50 = 160 nM T94879 CLBV45 44320831 IC50 = 28 nM T94879 C6RS5T 44320847 IC50 = 1360 nM T94879 CVS5D1 44320863 IC50 = 20 nM T94879 C0GM7F 44320900 IC50 = 315 nM T94879 C13WMT 44320988 IC50 = 12 nM T94879 CP78QN 44320989 IC50 = 26 nM T94879 CP34EA 44321012 IC50 = 63 nM T94879 CN8Z1I 44321013 IC50 = 24 nM T94879 CDP87G 44321026 IC50 = 3.5 nM T94879 C9G0OQ 44321064 IC50 = 19 nM T94879 CWMD23 44321111 IC50 = 5.5 nM T94879 CPEB60 44321112 IC50 = 10 nM T94879 CX9L7V 44321135 IC50 = 11 nM T94879 C51CET 44321137 IC50 = 5 nM T94879 CD0QO6 44321152 IC50 = 93 nM T94879 C69MZC 44321154 IC50 = 5420 nM T94879 CUV0W1 44321156 IC50 > 10000 nM T94879 CP71YV 44321172 IC50 = 16 nM T94879 CXNO48 44321173 IC50 > 10000 nM T94879 C7NE6Q 44321175 IC50 > 10000 nM T94879 C81WUS 44321176 IC50 = 1500 nM T94879 C4QO0A 44321178 IC50 > 10000 nM T94879 CZWA59 44321202 IC50 = 60 nM T94879 C4B1WH 44321204 IC50 = 73 nM T94879 CIAN09 44321224 IC50 = 1810 nM T94879 C86ATM 44321229 IC50 = 100 nM T94879 CR54IA 44321231 IC50 > 10000 nM T94879 C4VFQ5 44321253 IC50 = 91 nM T94879 CYVA51 44321254 IC50 > 10000 nM T94879 CUQ3R1 44321255 IC50 = 100 nM T94879 C7BM6I 44321261 IC50 = 59 nM T94879 CZ16IY 44324251 IC50 = 30000 nM T94879 CCX9Z3 44324252 IC50 = 24000 nM T94879 CG6UT1 44324296 IC50 = 20000 nM T94879 C8M4WJ 44324373 IC50 = 22000 nM T94879 CY5HZ7 44324390 IC50 = 9000 nM T94879 C5KYV6 44324391 IC50 = 8000 nM T94879 C5C4QX 44324507 IC50 = 22000 nM T94879 CNK2F8 44331802 IC50 = 270 nM T94879 CGFP09 44336826 IC50 = 0.82 nM T94879 C98VIX 44336827 IC50 = 0.69 nM T94879 C1L6SG 44336834 IC50 = 1.1 nM T94879 CH8RY1 44336844 IC50 = 1.8 nM T94879 C1AC3Z 44336847 IC50 = 0.3 nM T94879 C0NT4K 44336855 IC50 = 0.33 nM T94879 C9WLD8 44336856 IC50 = 2 nM T94879 CUME98 44336924 IC50 = 0.58 nM T94879 CM1BO3 44348247 IC50 = 32000 nM T94879 CY5L6J 44348257 IC50 = 11000 nM T94879 CD5ZW3 44348484 IC50 = 650 nM T94879 C80PGJ 44348564 IC50 = 1500 nM T94879 CY0T1M 44348625 IC50 = 9600 nM T94879 CG98RE 44358477 Ki = 3.32 nM T94879 C3H4MR 44358478 Ki = 2.49 nM T94879 CBD52Z 44358886 Ki = 4.66 nM T94879 C7LN0W 44363056 IC50 = 50 nM T94879 C71YUD 44363183 IC50 = 3000 nM T94879 CF0IB6 44377834 IC50 = 105 nM T94879 CWO45S 44377842 Ki = 145 nM T94879 C27ZVC 44377867 Ki = 132 nM T94879 C7TXQ3 44377869 Ki = 179 nM T94879 CSW1J4 44377881 Ki = 219 nM T94879 C27TDG 44377933 Ki > 100 nM T94879 C8XM3I 44377988 IC50 = 100 nM T94879 C5IOH4 44378004 IC50 = 95 nM T94879 C85XCK 44378015 Ki = 850 nM T94879 C0H7KF 44378030 Ki > 5000 nM T94879 CU29OZ 44378056 Ki = 130 nM T94879 CLV13K 44378110 Ki > 10000 nM T94879 CL3SI5 44378121 Ki = 50.6 nM T94879 CYA76O 44378142 IC50 > 10000 nM T94879 C6IOU8 44378149 Ki = 8.11 nM T94879 CBQ5W3 44378155 IC50 = 67 nM T94879 CR30BD 44378165 Ki = 32.3 nM T94879 CHL5D9 44378187 Ki = 77.5 nM T94879 CV5Y1A 44378199 Ki = 64.2 nM T94879 CT8NH9 44383851 IC50 > 10000 nM T94879 C19CRH 44383901 IC50 = 19700 nM T94879 CR9O3I 44383902 IC50 > 30000 nM T94879 CW47HV 44383906 IC50 = 17700 nM T94879 CL86MY 44383907 IC50 > 10000 nM T94879 CW63HQ 44383912 IC50 > 10000 nM T94879 CF98LG 44384286 IC50 > 10000 nM T94879 CN1WS7 44384345 IC50 = 66700 nM T94879 C01XPL 44384404 IC50 = 22700 nM T94879 CWPR87 44384405 IC50 = 2900 nM T94879 C59SDR 44384406 IC50 = 3900 nM T94879 C7WT4G 44384540 IC50 = 18200 nM T94879 C4RQB0 44384541 IC50 = 21200 nM T94879 CRZ5G8 44384546 IC50 > 100000 nM T94879 C6W4GY 44384713 IC50 = 56100 nM T94879 CKH7M8 44384714 IC50 > 30000 nM T94879 C0ZGU6 44385109 IC50 = 12100 nM T94879 CE80VB 44385244 IC50 = 1700 nM T94879 CH5GU8 44385282 IC50 = 14900 nM T94879 CL50UE 44385283 IC50 = 9700 nM T94879 CSN56E 44386916 IC50 = 3.981 nM T94879 C13HPW 44393651 IC50 > 101000 nM T94879 CJ6GB5 44393709 IC50 = 11600 nM T94879 CQP01D 44393950 IC50 = 18770 nM T94879 CU1CQ8 44394047 IC50 = 80000 nM T94879 CJYC83 44397324 IC50 = 2070 nM T94879 CZUY06 44397327 IC50 = 5620 nM T94879 CB64FY 44397328 IC50 = 1690 nM T94879 CDJ87T 44397345 IC50 = 6190 nM T94879 C5CTF6 44397346 IC50 = 140 nM T94879 C2T7BQ 44397347 IC50 = 680 nM T94879 C39VBJ 44397348 IC50 = 3350 nM T94879 CU3BF4 44397365 IC50 = 1840 nM T94879 CRTY10 44397366 IC50 = 2930 nM T94879 CYFD01 44397379 IC50 = 1510 nM T94879 C4VS1H 44397382 IC50 = 74 nM T94879 C8YCU6 44397384 IC50 = 3190 nM T94879 CQD8Z7 44397386 IC50 = 13 nM T94879 CCL9D6 44397387 IC50 = 620 nM T94879 CSAQ43 44397397 IC50 = 3190 nM T94879 C7MZ8J 44397413 IC50 = 5990 nM T94879 C8KA6R 44397415 IC50 = 920 nM T94879 CR8P4T 44397447 IC50 = 3280 nM T94879 C9TK8I 44397448 IC50 = 5150 nM T94879 CF2AP3 44397474 IC50 = 230 nM T94879 CQT12O 44397490 IC50 = 2720 nM T94879 C6FJV7 44397494 IC50 = 1280 nM T94879 CZ5QV6 44397495 IC50 = 2130 nM T94879 CAP7W0 44397504 IC50 = 1210 nM T94879 CU13ES 44397515 IC50 = 96 nM T94879 CQY79V 44397539 IC50 = 8900 nM T94879 CTAI27 44397548 IC50 = 1470 nM T94879 C98ZCS 44397556 IC50 = 270 nM T94879 CMC12S 44397573 IC50 = 6490 nM T94879 CL15YW 44397574 IC50 = 3810 nM T94879 C6GIS2 44397576 IC50 = 10000 nM T94879 C65PLD 44397577 IC50 = 4520 nM T94879 C8MFC2 44397582 IC50 = 3300 nM T94879 C3PN4D 44397598 IC50 = 790 nM T94879 CE2GZ3 44397599 IC50 = 6680 nM T94879 CY0KB5 44397600 IC50 = 2660 nM T94879 C86IAQ 44397602 IC50 = 1900 nM T94879 CR0D6I 44397603 IC50 = 8760 nM T94879 CD67XW 44397612 IC50 = 6090 nM T94879 C1ISA5 44397619 IC50 = 7820 nM T94879 CG2XI7 44397621 IC50 = 6250 nM T94879 C1HBU8 44397622 IC50 = 3160 nM T94879 CA1FG3 44397627 IC50 = 9070 nM T94879 C1FJH9 44397640 IC50 = 74 nM T94879 CV2Q1K 44397643 IC50 = 17 nM T94879 C69WZC 44397646 IC50 = 130 nM T94879 CC8Z3A 44397647 IC50 = 3680 nM T94879 C1VB8P 44397694 IC50 = 630 nM T94879 CV2M0A 44397708 IC50 = 3500 nM T94879 C8MZF1 44397709 IC50 = 4580 nM T94879 C2OA3Y 44397724 IC50 = 9460 nM T94879 CJIK26 44397727 IC50 = 320 nM T94879 CFP7S8 44397728 IC50 = 350 nM T94879 CERQ57 44397746 IC50 = 2640 nM T94879 C2PJ6R 44397748 IC50 = 10000 nM T94879 CAQD83 44397749 IC50 = 1100 nM T94879 C5GLC2 44397761 IC50 = 40 nM T94879 CUZY95 44397764 IC50 = 8620 nM T94879 CQCN29 44397781 IC50 = 770 nM T94879 C0B2YM 44397782 IC50 = 830 nM T94879 CWL0A9 44397785 IC50 = 3410 nM T94879 CSN79W 44397799 IC50 = 1800 nM T94879 C20BLM 44397801 IC50 = 1830 nM T94879 CJG87Q 44397802 IC50 = 500 nM T94879 CP1CU7 44397810 IC50 = 650 nM T94879 CI7HS1 44397811 IC50 = 6070 nM T94879 C9SQ1V 44397814 IC50 = 1450 nM T94879 CZF29N 44397816 IC50 = 190 nM T94879 CIVF18 44397836 IC50 = 890 nM T94879 CP18FI 44397837 IC50 = 2580 nM T94879 CRMN86 44397859 IC50 = 3200 nM T94879 CC7B3S 44397860 IC50 = 460 nM T94879 C01CAI 44397871 IC50 = 10000 nM T94879 C8Y0WF 44397874 IC50 = 7650 nM T94879 CJ6B1W 44397876 IC50 = 2420 nM T94879 C28ERI 44397877 IC50 = 2490 nM T94879 C6Y9XN 44397888 IC50 = 520 nM T94879 CIOM21 44397889 IC50 = 430 nM T94879 CVQ8C1 44397891 IC50 = 1240 nM T94879 CX3M5J 44397892 IC50 = 270 nM T94879 CYX72U 44397904 IC50 = 3100 nM T94879 C5JS4T 44397906 IC50 = 8910 nM T94879 CVB7K2 44397908 IC50 = 2200 nM T94879 CP8CW5 44397940 IC50 = 9430 nM T94879 CFHR09 44397941 IC50 = 9280 nM T94879 CP62TK 44397956 IC50 = 4990 nM T94879 C6UY9Z 44397957 IC50 = 4250 nM T94879 C23GTH 44397958 IC50 = 8430 nM T94879 CG36QI 44397976 IC50 = 10000 nM T94879 CDK84C 44397977 IC50 = 7560 nM T94879 CB3ZG1 44397979 IC50 = 1030 nM T94879 C4AO1D 44397980 IC50 = 9870 nM T94879 CW65CR 44397987 IC50 = 5470 nM T94879 C1DQW5 44397991 IC50 = 40 nM T94879 CP8F9A 44397992 IC50 = 8580 nM T94879 CM1ZW4 44401687 IC50 = 230 nM T94879 C0YZV7 44401690 IC50 = 33 nM T94879 C7CDY2 44401692 IC50 = 74 nM T94879 CT8R0Q 44401694 IC50 = 81 nM T94879 CDSE04 44401695 IC50 = 90 nM T94879 CB3RC6 44401705 IC50 = 60 nM T94879 CA59PR 44401708 IC50 = 81 nM T94879 CXA4D6 44401724 IC50 = 23 nM T94879 C17ODM 44401727 IC50 = 430 nM T94879 CX0AZ7 44401742 IC50 = 270 nM T94879 C3G2RU 44401767 IC50 = 350 nM T94879 C4BJ3U 44401771 IC50 = 38 nM T94879 C0F9ZD 44401772 IC50 = 2.3 nM T94879 CM45YT 44401790 IC50 = 33 nM T94879 CA1SR3 44401812 IC50 = 29 nM T94879 CN63AH 44401816 IC50 = 30 nM T94879 CVOW53 44401827 IC50 = 32 nM T94879 CVCN36 44401831 IC50 = 920 nM T94879 C59TYU 44401851 IC50 = 200 nM T94879 C78VHO 44401870 IC50 = 13000 nM T94879 CSM4X8 44401879 IC50 = 20 nM T94879 CZU4T7 44401880 IC50 = 3.3 nM T94879 C01BEI 44401886 IC50 = 100 nM T94879 CU4AR1 44401892 IC50 = 5.3 nM T94879 C14LNK 44401904 IC50 = 60 nM T94879 CVPZ92 44401905 IC50 = 28 nM T94879 C0BRH8 44401908 IC50 = 450 nM T94879 CN4T6Z 44401928 IC50 = 145 nM T94879 CV17OM 44401929 IC50 = 14 nM T94879 CK9VN7 44401931 IC50 = 320 nM T94879 C9Q1ET 44401943 IC50 = 40 nM T94879 CB98IX 44401972 IC50 = 130 nM T94879 CD51UN 44401977 IC50 = 100 nM T94879 C19QCE 44401981 IC50 = 48 nM T94879 C04BTX 44401982 IC50 = 15 nM T94879 C7MY1S 44402027 IC50 = 59 nM T94879 C6XA7P 44402060 IC50 = 3100 nM T94879 CTZ52C 44402073 IC50 = 28 nM T94879 C4P8RN 44402077 IC50 = 35 nM T94879 C6S8KA 44402114 IC50 = 40 nM T94879 CDNZ52 44402130 IC50 = 180 nM T94879 CP78NL 44402133 IC50 = 1100 nM T94879 CWVH96 44402149 IC50 = 100 nM T94879 C9BN6H 44402168 IC50 = 6.5 nM T94879 CQM65U 44402195 IC50 = 160 nM T94879 CM90NL 44402196 IC50 = 980 nM T94879 C6IY5O 44402213 IC50 = 39 nM T94879 C4O7QE 44402239 IC50 = 22 nM T94879 C4P0AC 44402278 IC50 = 75 nM T94879 C1GPC2 44402295 IC50 = 7.8 nM T94879 CCZ2E8 44438552 IC50 = 462 nM T94879 CB1C2M 44438553 IC50 = 25 nM T94879 C7RV5Q 44438554 IC50 = 20 nM T94879 CCOJ06 44438555 IC50 = 28 nM T94879 CB93RX 44438557 IC50 = 33 nM T94879 C9AO2Z 44438558 IC50 = 42 nM T94879 C50ZMB 44438560 IC50 = 5 nM T94879 C39ZMJ 44438561 IC50 = 26 nM T94879 CBQN25 44438563 IC50 = 10000 nM T94879 CJH70L 44438564 IC50 = 34 nM T94879 CE4S8J 44438565 IC50 = 51 nM T94879 CK1JU3 44459193 IC50 = 1.288 nM T94879 CZFU59 44459332 IC50 = 43 nM T94879 CJ0Q4D 44459333 IC50 = 2.2 nM T94879 CT39RH 44459469 IC50 = 2.8 nM T94879 CG4AI3 44459482 IC50 = 2.089 nM T94879 CZ6IU2 44459494 IC50 = 6.457 nM T94879 C68RBI 44459495 IC50 = 5.37 nM T94879 CNJ16Q 44459505 IC50 = 4.5 nM T94879 C0FQ1O 44459535 IC50 = 5 nM T94879 CT9R7K 44459542 IC50 = 46 nM T94879 CP97OV 44459564 IC50 = 57.54 nM T94879 C49NWP 44459572 IC50 = 550 nM T94879 C5G2JO 44459598 IC50 = 19.95 nM T94879 C8MBD9 44459599 IC50 = 158.49 nM T94879 C0W4VT 44459622 IC50 = 39.81 nM T94879 C18EJF 44459640 IC50 = 1.8 nM T94879 C7RGD3 44459641 IC50 = 2.089 nM T94879 CQ95TO 44459661 IC50 = 128.82 nM T94879 CRH7N1 44459687 IC50 = 6.31 nM T94879 C8JS2X 44459694 IC50 = 18 nM T94879 CO3F9K 44459713 IC50 = 8.3 nM T94879 CF4C3P 44459717 IC50 = 7 nM T94879 C1W5OG 44459718 IC50 = 21.88 nM T94879 C31SQM 44459720 IC50 = 2.291 nM T94879 CS17XE 44459751 IC50 = 6.761 nM T94879 C85QDR 44459752 IC50 = 13 nM T94879 CI2V6T 44459760 IC50 = 1.096 nM T94879 CJN91Z 44459761 IC50 = 0.8913 nM T94879 CQ01TE 44459776 IC50 = 3.09 nM T94879 C24BGR 44459782 IC50 = 1.514 nM T94879 CB37LV 44459783 IC50 = 6.3 nM T94879 C1V3CW 44459848 IC50 = 3.02 nM T94879 C52JOE 44459875 IC50 = 47.86 nM T94879 CZ1DJ8 44459876 IC50 = 55 nM T94879 CWXV09 44459906 IC50 = 0.3 nM T94879 CJ4L3O 44459907 IC50 = 7.943 nM T94879 CZ0DN5 44572149 IC50 > 10000 nM T94879 C6U8QW 44572150 IC50 > 10000 nM T94879 C9XD8C 44572789 IC50 = 5200 nM T94879 C72XEI 44572984 IC50 > 10000 nM T94879 CIX5Q0 44572985 IC50 > 10000 nM T94879 C7UXN8 44572986 IC50 > 10000 nM T94879 CRBQ49 44572987 IC50 = 6500 nM T94879 C0WXB4 44580020 IC50 = 1.585 nM T94879 CHA63L 44580021 IC50 = 6.31 nM T94879 CX3L1P 44587252 IC50 = 160 nM T94879 CI3K8T 44605342 IC50 = 87100 nM T94879 CV8RY3 45260952 IC50 = 3 nM T94879 CLEU14 45260983 IC50 = 12 nM T94879 C48QSY 45261659 IC50 = 1700 nM T94879 CC5Z7N 45261660 IC50 = 2300 nM T94879 C26IBG 45261674 IC50 = 5000 nM T94879 CTG0D9 45261728 IC50 = 2800 nM T94879 CS7GA3 45264997 IC50 = 760 nM T94879 C3IOB7 45265000 IC50 = 360 nM T94879 CKW39R 45267744 IC50 = 4.571 nM T94879 C9PC5S 45267756 IC50 = 223.87 nM T94879 CR7QN3 45267764 IC50 = 0.3 nM T94879 C1KTZ3 45267771 IC50 = 33.9 nM T94879 C6WLB4 45268626 IC50 = 2.5 nM T94879 CE0U3W 45268639 IC50 = 13.49 nM T94879 CR8JH9 45268646 IC50 = 33.3 nM T94879 CM8OP3 45268652 IC50 = 0.3 nM T94879 CD6A0O 45269469 IC50 = 20.3 nM T94879 CL42XG 45269481 IC50 = 3.467 nM T94879 CRWE76 45269493 IC50 = 0.4 nM T94879 CHN4F0 45269499 IC50 = 2.9 nM T94879 C6DQU1 45269515 IC50 = 534 nM T94879 CB4IO3 45269516 IC50 = 51 nM T94879 CD47UP 45270308 IC50 = 28.18 nM T94879 C4VPC6 45270320 IC50 = 1 nM T94879 CMF3T7 45270338 IC50 = 36.5 nM T94879 C1XZ4Q 45270704 IC50 = 1.21 nM T94879 C89NBL 45270705 IC50 = 1.21 nM T94879 CDWX76 45271142 IC50 = 147.91 nM T94879 C62LVH 45272043 IC50 = 52.5 nM T94879 C0AO8K 45272078 IC50 = 43 nM T94879 CN7GR1 45272848 IC50 = 1.995 nM T94879 C8RZ7H 45272849 IC50 = 2.692 nM T94879 CQ34VM 45272857 IC50 = 3 nM T94879 C5H9RX 45272874 IC50 = 22.4 nM T94879 C7X2VE 45272888 IC50 = 0.9 nM T94879 CN8G9K 45272901 IC50 = 26.7 nM T94879 C2MW1C 45272908 IC50 = 25 nM T94879 C3X7RV 45273795 IC50 = 1.288 nM T94879 C74IXB 45273827 IC50 = 0.3 nM T94879 CLZ39M 45379958 IC50 = 2.38 nM T94879 C98KFA 45486490 IC50 = 1.17 nM T94879 CGA65L 45486496 IC50 = 0.17 nM T94879 CZ8JD0 45486497 IC50 = 0.28 nM T94879 CYF73X 45486498 IC50 = 0.38 nM T94879 C86XSZ 45486501 IC50 = 0.55 nM T94879 CDYO49 45486504 IC50 = 0.06 nM T94879 CNW0I9 45486505 IC50 = 0.71 nM T94879 CWQ6Y5 45486511 IC50 = 16.3 nM T94879 CSG37U 45486513 IC50 = 2.59 nM T94879 CEX01M 45486514 IC50 = 0.32 nM T94879 C58IWJ 45486519 IC50 = 0.25 nM T94879 CE3PK0 45486527 IC50 = 0.68 nM T94879 C1ZYT9 45486549 IC50 = 2.95 nM T94879 CHE56F 45486550 IC50 = 0.34 nM T94879 C84NHX 45486564 IC50 = 0.54 nM T94879 CLMZ68 45486571 IC50 = 4 nM T94879 CB2MG1 45486572 IC50 = 0.32 nM T94879 C0MWV4 45486574 IC50 = 0.88 nM T94879 C9SI3E 45486581 IC50 = 0.36 nM T94879 C51CUF 46193118 IC50 = 640 nM T94879 CTP8R1 46193119 IC50 = 38 nM T94879 CDT4U1 46193239 IC50 = 29000 nM T94879 C0W3LE 46193243 IC50 = 100 nM T94879 CKUN01 46193244 IC50 = 88000 nM T94879 CHU8I7 46193370 IC50 = 2800 nM T94879 C7NC9V 46193371 IC50 = 60 nM T94879 CY49DB 46193372 IC50 = 320 nM T94879 CN05XT 46193373 IC50 = 41000 nM T94879 C1Q6WV 46193374 IC50 = 32000 nM T94879 C60KFT 46193375 IC50 = 50 nM T94879 C2J9IH 46193486 IC50 = 260 nM T94879 CJ86KO 46193489 IC50 = 50 nM T94879 CPYK94 46193490 IC50 = 3400 nM T94879 CHUN05 46193595 IC50 = 40 nM T94879 C5IMB2 46239424 Ki = 6400 nM T94879 CKR9P7 46239425 Ki = 8900 nM T94879 C7SLP0 46239531 Ki = 5000 nM T94879 CI1F5C 46239840 Ki > 100000 nM T94879 C26XVS 46240044 Ki = 17324 nM T94879 CC3UF9 46830325 IC50 = 0.15 nM T94879 CE4JU7 46842025 IC50 = 0.27 nM T94879 CR8JC2 46842169 IC50 = 0.27 nM T94879 CF23CG 46842171 IC50 = 0.27 nM T94879 CWY45O 46842322 IC50 = 4.1 nM T94879 CY9UB1 46842324 IC50 = 0.27 nM T94879 CVP3F6 46886964 IC50 = 0.94 nM T94879 CF49HM 46886965 IC50 = 3.92 nM T94879 CQ91ZP 46887034 IC50 = 2.96 nM T94879 CDI09L 46887035 IC50 = 0.38 nM T94879 C8X6IR 46887483 IC50 = 0.3 nM T94879 C51BJT 46887484 IC50 = 0.86 nM T94879 CB3F2M 46887522 IC50 = 1.84 nM T94879 CVX57Z 46887568 IC50 = 3.28 nM T94879 C3GW8T 46887569 IC50 = 9.79 nM T94879 C13VUK 46888519 IC50 = 0.07 nM T94879 C7G5PM 46888541 IC50 = 0.66 nM T94879 C6NIG0 46888542 IC50 = 1.4 nM T94879 CPM4S1 46888559 IC50 = 5.5 nM T94879 CV53IU 46888560 IC50 = 0.89 nM T94879 C9UY1R 46888576 IC50 = 2.5 nM T94879 CE79JU 46888577 IC50 = 1.2 nM T94879 CQ5B2F 46888578 IC50 = 2.3 nM T94879 C8ITU7 46888595 IC50 = 0.2 nM T94879 C0IQ2C 46888596 IC50 = 2 nM T94879 CS6F1J 46888597 IC50 = 0.087 nM T94879 C7B3ZY 46888631 IC50 = 0.42 nM T94879 C8FW5K 46888632 IC50 = 2.3 nM T94879 C57KWS 46888633 IC50 = 0.35 nM T94879 CS27GK 46888659 IC50 = 0.011 nM T94879 C38INP 46888660 IC50 = 0.07 nM T94879 C6WQ5Y 46888661 IC50 = 1.2 nM T94879 CZ3SO4 46888707 IC50 = 0.19 nM T94879 C02RDT 46888708 IC50 = 0.08 nM T94879 CUN72Y 46888738 IC50 = 0.05 nM T94879 C3P2IN 46933992 IC50 = 11000 nM T94879 CHA5Z0 49821469 IC50 > 1000 nM T94879 C1AYP0 49821627 IC50 > 500 nM T94879 C85AXR 49821714 IC50 > 1000 nM T94879 CZS03D 50902030 Ki > 4274 nM T94879 CH2Z1E 50902289 Ki > 7100 nM T94879 C4HJL2 50902291 Ki > 7950 nM T94879 C6A1IU 50902549 Ki > 2000 nM T94879 C3Y2AV 50903255 Ki > 2000 nM T94879 CN41YJ 50925469 IC50 = 2 nM T94879 CQ3RG5 50925470 IC50 = 7 nM T94879 C2E5JK 50940516 IC50 = 850 nM T94879 CEB5T9 50940517 IC50 = 50 nM T94879 C2C0IA 50940656 IC50 = 850 nM T94879 C4I9OJ 50940659 IC50 = 8750 nM T94879 C6F5RK 50940660 IC50 = 300 nM T94879 C9O4LE 50940680 IC50 = 590 nM T94879 CT3H4X 50940682 IC50 = 4140 nM T94879 CN4S0D 50940686 IC50 = 2310 nM T94879 CT8V2L 50940687 IC50 = 12 nM T94879 CP3G6K 50940690 IC50 = 2300 nM T94879 C7MV1Y 50940692 IC50 = 380 nM T94879 CUM0O5 50940699 IC50 = 730 nM T94879 C9IFA6 50940700 IC50 = 50 nM T94879 C7TF6Q 50940701 IC50 = 1200 nM T94879 CI3AG0 50941259 IC50 = 260 nM T94879 CCUK19 50941260 IC50 = 990 nM T94879 CY37HL 50941261 IC50 = 10 nM T94879 CC0QW5 50941262 IC50 = 1340 nM T94879 C5Q9YU 50941264 IC50 = 3300 nM T94879 C7Y8HK 50941365 IC50 = 270 nM T94879 C8WQX5 50941366 IC50 = 1110 nM T94879 C3NK7Q 50941367 IC50 = 4460 nM T94879 C3QEV9 50941368 IC50 = 290 nM T94879 CA3HQ6 50941461 IC50 = 2040 nM T94879 C8LSY4 50941462 IC50 = 190 nM T94879 C4GBV9 50941463 IC50 = 1260 nM T94879 CYL8N5 50941464 IC50 = 1350 nM T94879 C10WDU 50941465 IC50 = 260 nM T94879 C6YM0P 50941551 IC50 = 1270 nM T94879 C6R4YN 50993785 IC50 = 10000 nM T94879 C0M6XL 50993786 IC50 = 10000 nM T94879 C0OR7K 53248667 IC50 > 100000 nM T94879 CS3R1I 53248669 IC50 = 28900 nM T94879 C30RNE 53248670 IC50 = 6400 nM T94879 C1RJ7M 54580520 IC50 > 400000 nM T94879 CCXF36 54580521 IC50 = 145000 nM T94879 CZG36N 54580522 IC50 > 400000 nM T94879 C0NPM8 54580523 IC50 = 225000 nM T94879 C25VSX 54580524 IC50 > 400000 nM T94879 CBT56Y 54581676 IC50 = 5200 nM T94879 C0MN3D 54582527 IC50 = 156000 nM T94879 C6T1QX 54582528 IC50 = 350000 nM T94879 CP4N1Q 54582529 IC50 > 400000 nM T94879 CW1X3G 54583497 IC50 > 400000 nM T94879 CN96IQ 54585432 IC50 > 400000 nM T94879 CH25CO 54586393 IC50 > 400000 nM T94879 C82LED 54586394 IC50 > 400000 nM T94879 CQ1H3C 54587403 IC50 > 400000 nM T94879 C28GAC 54587404 IC50 > 400000 nM T94879 CFX89L 54587804 IC50 = 5700 nM T94879 CGF65A 54670110 IC50 > 30000 nM T94879 C90ZLC 54670399 IC50 > 30000 nM T94879 CLK61N 56587955 IC50 = 0.1 nM T94879 C4TGL7 56648496 IC50 > 1000 nM T94879 CH6C3L 56648679 IC50 > 10000 nM T94879 CCY79V 56648680 IC50 = 3110 nM T94879 CNE96P 56648857 IC50 > 10000 nM T94879 CX86AQ 56648859 IC50 > 1000 nM T94879 CPC3T4 56654131 IC50 > 10000 nM T94879 C0YD3P 56928304 IC50 > 5000 nM T94879 C8RO6A 56929788 IC50 > 1000 nM T94879 CD52CA 57391118 IC50 = 0.02 nM T94879 C7Y4BX 57391119 IC50 = 1.47 nM T94879 C4PSK2 57391120 IC50 = 0.04 nM T94879 CA1TE7 57391121 IC50 = 0.01 nM T94879 CN60KE 57391196 IC50 = 0.09 nM T94879 CM7N8I 57391197 IC50 = 0.05 nM T94879 C7VXN9 57391198 IC50 = 1.3 nM T94879 C7SC4E 57392888 IC50 = 0.44 nM T94879 CG3DF1 57392948 Ki > 10000 nM T94879 CQT1G9 57392966 IC50 = 1.38 nM T94879 CR28IN 57394623 IC50 = 0.38 nM T94879 CHZ67R 57394624 IC50 = 0.27 nM T94879 CE36TV 57394695 Ki = 24400 nM T94879 CLEY35 57396379 IC50 = 0.64 nM T94879 C7W6TP 57396380 IC50 = 0.05 nM T94879 C80CVX 57396381 IC50 = 0.01 nM T94879 C86YCU 57396469 IC50 = 0.1 nM T94879 C3M6EL 57396470 IC50 = 1.64 nM T94879 CPQ91V 57396471 IC50 = 0.22 nM T94879 CP0AB6 57396472 IC50 = 0.28 nM T94879 CNY5Z8 57398261 IC50 = 0.35 nM T94879 CH57NZ 57398879 IC50 = 15.8 nM T94879 CTYR07 57399826 IC50 = 0.04 nM T94879 CL5UP7 57401597 IC50 = 0.36 nM T94879 C37KMA 57401598 IC50 = 0.13 nM T94879 CHQ79W 57401599 IC50 = 0.02 nM T94879 CWG70K 57401600 IC50 = 0.06 nM T94879 CU5KP3 57401601 IC50 = 0.1 nM T94879 C8GD5N 57402376 IC50 = 8.2 nM T94879 CLU6J0 57403348 IC50 = 2.43 nM T94879 CD73NJ 57403349 IC50 = 0.02 nM T94879 CPA3D1 57403394 Ki = 20800 nM T94879 CEN5Z8 57403417 IC50 = 0.08 nM T94879 CY75FP 57403418 IC50 = 0.05 nM T94879 CA4KZ8 57403419 IC50 = 1.31 nM T94879 C4XMB6 58547809 IC50 > 30000 nM T94879 CEB3G9 58547814 IC50 > 30000 nM T94879 C08QVG 58547833 IC50 > 30000 nM T94879 CFVG67 58547863 IC50 > 30000 nM T94879 CYZA38 58548077 IC50 > 30000 nM T94879 CN57ZH 67426178 IC50 > 10000 nM T94879 CO8C0Z 67453423 IC50 > 2000 nM T94879 CY8J3O 68181896 IC50 = 26000 nM T94879 CUGH78 68654838 IC50 = 1000 nM T94879 CH2X0Z 69394992 IC50 = 2.884 nM T94879 CC43LF 71074083 IC50 = 437 nM T94879 C4P0XT 71092344 IC50 = 4610 nM T94879 C6DAG4 71092519 IC50 = 13900 nM T94879 C2HGI7 71153408 IC50 > 10000 nM T94879 C9GR3L 71153436 IC50 > 10000 nM T94879 CHLQ31 71530755 IC50 = 160 nM T94879 CN8KP5 71575273 IC50 = 0.27 nM T94879 C4GNJ3 71598545 IC50 > 1000 nM T94879 C0M9IA 71666277 IC50 = 21.6 nM T94879 C3O9KX 71666278 IC50 = 0.59 nM T94879 CU0M5P 71666433 IC50 = 0.19 nM T94879 CZC74T 71666437 IC50 = 1.55 nM T94879 C68SDB 71719394 IC50 = 1995.26 nM T94879 CF2W4Z 71738037 IC50 = 240 nM T94879 C95QWN 71765666 IC50 = 17 nM T94879 CZ0G2X 72165213 IC50 > 10000 nM T94879 C7XRY6 72190879 IC50 > 30000 nM T94879 CQ3GD7 72704434 Ki = 630 nM T94879 C9JE6M 75815419 IC50 = 54.3 nM T94879 C65ZBN 76323083 IC50 = 537.03 nM T94879 CZ3P5K 89706867 IC50 = 0.056 nM T94879 CF03DW 90168772 IC50 > 20000 nM T94879 CM6J9K 90168778 IC50 > 20000 nM T94879 C45QVJ 91668196 IC50 = 2300 nM T94879 C1JPD6 91844700 IC50 = 5400 nM T94879 CYQV05 92471958 IC50 = 410 nM T94879 C6TD3W 117685212 IC50 = 337 nM T94879 CVUC27 117685328 IC50 = 1.5 nM T94879 C71BEL 117824219 IC50 = 1.7 nM T94879 CFAG87 117824250 IC50 = 0.059 nM T94879 C62NZT 117824353 IC50 = 64 nM T94879 C3WT5R 117824368 IC50 = 0.29 nM T94879 CGH1Z4 117824420 IC50 = 333 nM T94879 CX12RS 117824489 IC50 = 3.8 nM T94879 CS97IT 117830474 IC50 = 45.2 nM T94879 C60ADH 117830507 IC50 = 57 nM T94879 CMJR74 117830513 IC50 = 0.32 nM T94879 CSCY01 117949009 IC50 = 9800 nM T94879 CYQ74R 118479645 IC50 > 10000 nM T94879 CVYK24 118556943 IC50 > 50000 nM T94879 CM6XW1 118724093 IC50 = 520 nM T94879 C46LFG 118724094 IC50 > 10000 nM T94879 CYM21X 118724095 IC50 = 2900 nM T94879 C4HI1Q 118729758 IC50 = 3000 nM T94879 CKBG19 118729759 IC50 = 3100 nM T94879 C8LRQ7 121370930 IC50 = 110 nM T94879 CRJE23 122185011 IC50 > 30000 nM T94879 CS6M9C 122193679 IC50 > 100000 nM T94879 CVX7U9 127029185 IC50 = 3810 nM T94879 C9OVF8 127029366 IC50 = 5.2 nM T94879 C4UR7D 127038167 IC50 > 1000 nM T94879 C4H2TJ 127038168 IC50 > 1000 nM T94879 CL9JT8 127038169 IC50 = 606 nM T94879 CJPX60 127038509 IC50 = 232 nM T94879 C26EAG 127038511 IC50 = 201 nM T94879 CTM9E4 127038512 IC50 = 279 nM T94879 C6AQ2U 127038513 IC50 = 195 nM T94879 CV1FM0 127038868 IC50 = 228 nM T94879 CADU23 127038869 IC50 = 91.6 nM T94879 CACJ46 132489333 IC50 = 5.6 nM T94879 C2P1IU 134129996 IC50 > 100000 nM T94879 CLE03O 134130328 IC50 > 100000 nM T94879 CSN6J0 134130563 IC50 > 100000 nM T94879 C0A1CZ 134131162 IC50 > 100000 nM T94879 C23CYE 134814217 IC50 = 1.41 nM T94879 CHX5W7 134908214 IC50 = 91200 nM T94879 C1QMI8 135401477 IC50 = 26.92 nM T94879 C1BA7R 135406502 IC50 = 2 nM T94879 CIC0M9 135406542 IC50 = 3 nM T94879 CL6W5K 135406554 IC50 = 5.3 nM T94879 CL6YK2 135406621 IC50 = 1.1 nM T94879 C1LG3R 135406622 IC50 = 27 nM T94879 C9S5CV 135406637 IC50 = 1.4 nM T94879 C17YXR 135406983 IC50 = 5 nM T94879 C41TDB 135413523 IC50 = 3.5 nM T94879 C5JYM4 135415122 IC50 = 3 nM T94879 CN7LX8 135415142 IC50 = 1.5 nM T94879 CJG93Q 135415214 IC50 = 3.2 nM T94879 CQOL86 135417284 IC50 = 30 nM T94879 CG96MZ 135419216 IC50 = 2 nM T94879 COD5W1 135419220 IC50 = 2000 nM T94879 CBA1Q7 135419269 IC50 = 5 nM T94879 CP4HN6 135419318 IC50 = 7 nM T94879 CCXB28 135419329 IC50 = 2 nM T94879 CL8U1V 135419421 IC50 = 3.5 nM T94879 CN1CE4 135423930 IC50 = 2 nM T94879 C1GPZ3 135423938 IC50 = 0.2 nM T94879 C7A2NS 135427992 IC50 = 7.1 nM T94879 C6UFD4 135430871 IC50 = 10 nM T94879 C1Z3WH 135430893 IC50 = 8 nM T94879 CAJU63 135430952 IC50 = 50 nM T94879 CNP87H 135433645 IC50 = 330 nM T94879 C2DAG7 135433829 IC50 = 50 nM T94879 CHD03R 135433867 IC50 = 80 nM T94879 CJ0B6N 135438524 IC50 = 9.5 nM T94879 CJ9IE8 135438525 IC50 = 21 nM T94879 C94RVJ 135438569 IC50 = 0.7 nM T94879 C1A4MY 135439488 IC50 = 100 nM T94879 C0IE4A 135443738 IC50 = 200 nM T94879 C5U1NW 135444771 IC50 = 0.48 nM T94879 CF1U2Y 135451848 IC50 = 0.52 nM T94879 C0DBS7 135452901 IC50 = 1.905 nM T94879 CFKO84 135455980 IC50 = 5.7 nM T94879 CQW8U9 135456038 IC50 = 1 nM T94879 C9LD5N 135456042 IC50 = 2.089 nM T94879 C0BQH8 135456061 IC50 = 10 nM T94879 CA83SQ 135456100 IC50 = 1 nM T94879 C4ZQ1W 135456180 IC50 = 1.3 nM T94879 CM1K9A 135456702 IC50 = 150 nM T94879 C3R8SE 135457869 IC50 = 5200 nM T94879 C6TO5S 135462289 IC50 = 4 nM T94879 CUX8S3 135462319 IC50 = 70 nM T94879 C7HC3R 135462338 IC50 = 2.5 nM T94879 CA8X3R 135462413 IC50 = 1.7 nM T94879 CY3A0S 135462886 IC50 = 2.89 nM T94879 CA9V7D 135463722 IC50 = 10 nM T94879 C4C3JV 135467743 IC50 = 6 nM T94879 CTN73W 135467948 IC50 = 1 nM T94879 CHSI34 135469671 IC50 = 10 nM T94879 CAR9X0 135474505 IC50 = 0.62 nM T94879 CADL53 135475879 IC50 = 40 nM T94879 C3IT7F 135477808 IC50 = 13 nM T94879 C9E5KR 135480166 IC50 = 20 nM T94879 CZ9HT7 135480403 IC50 = 1.7 nM T94879 CJS37E 135482260 IC50 > 101000 nM T94879 CUNL35 135484025 IC50 = 10 nM T94879 C95GLJ 135484081 IC50 = 0.69 nM T94879 CVTR78 135484097 IC50 = 1.04 nM T94879 CKP9T0 135485820 IC50 = 5.3 nM T94879 CUV8L0 135485839 IC50 = 1.1 nM T94879 C23SWA 135485841 IC50 = 1.6 nM T94879 C4ILF7 135487662 IC50 = 1.7 nM T94879 CEHK47 135487696 IC50 = 2.6 nM T94879 CEZ5P3 135487732 IC50 = 5 nM T94879 C18DSI 135489339 IC50 = 34 nM T94879 CHO1Z5 135489408 IC50 = 7 nM T94879 CBW5A9 135491781 IC50 = 3.6 nM T94879 CG82XZ 135491934 IC50 = 18.2 nM T94879 CMNE87 135491938 IC50 = 8.2 nM T94879 CLFQ43 135493551 IC50 = 3 nM T94879 C8L1NK 135494369 IC50 = 3 nM T94879 C7FM8V 135494393 IC50 = 2 nM T94879 C3D4IY 135496441 IC50 = 3 nM T94879 C2MTZ8 135497265 IC50 = 2 nM T94879 CS4NM0 135501101 IC50 = 2 nM T94879 CJ3XM0 135503009 IC50 = 14.7 nM T94879 C86THJ 135503803 IC50 = 1 nM T94879 CN4BY1 135503843 IC50 = 2 nM T94879 C7BM8D 135504134 IC50 = 70 nM T94879 CK0S3E 135505670 IC50 = 0.9 nM T94879 C4ZNY0 135505809 IC50 = 7 nM T94879 C78CIT 135505815 IC50 = 12 nM T94879 CM27YS 135506900 IC50 = 40 nM T94879 CC87SI 135510018 IC50 = 53 nM T94879 CVM2R1 135513834 IC50 = 50 nM T94879 C6GNF4 135513951 IC50 = 0.1 nM T94879 CC9N6X 135513970 IC50 = 1 nM T94879 CL1W4B 135513981 IC50 = 5 nM T94879 CYS04P 135514690 IC50 = 0.9 nM T94879 C4NSC9 135515154 IC50 = 4 nM T94879 C9IU6B 135515212 IC50 = 2.5 nM T94879 CEV79B 135515565 IC50 = 5.5 nM T94879 C0STP6 135518654 IC50 = 2.5 nM T94879 CKDH83 135518785 IC50 = 0.2 nM T94879 C8VT4S 135520162 IC50 = 6.4 nM T94879 CKD97I 135520170 IC50 = 13 nM T94879 CL0HD1 135520500 IC50 = 18 nM T94879 C5EBI4 135525517 IC50 = 44 nM T94879 CD84SI 135528161 IC50 = 35 nM T94879 CYF17I 135528172 IC50 = 3.3 nM T94879 CB6H4I 135528567 IC50 = 13 nM T94879 C6KQV1 135528758 IC50 = 5 nM T94879 CFN34H 135528775 IC50 = 4 nM T94879 CLU8A5 135529022 IC50 = 1.53 nM T94879 C6YF2L 135529725 IC50 = 8 nM T94879 CJIA83 135529861 IC50 = 20 nM T94879 CTX70E 135530119 IC50 = 2.7 nM T94879 CCM89A 135530700 IC50 = 8.5 nM T94879 C43HNQ 135531347 IC50 = 1.1 nM T94879 CV34FU 135532825 IC50 = 5.2 nM T94879 CM3GD7 135532874 IC50 = 10 nM T94879 CGWS52 135532916 IC50 = 2.47 nM T94879 CEF96L 135536692 IC50 = 30 nM T94879 CKC9M0 135536718 IC50 = 40 nM T94879 C6E0BM 135536759 IC50 = 7 nM T94879 CWRQ95 135536783 IC50 = 4 nM T94879 C1Z7AY 135536802 IC50 = 0.8 nM T94879 CSO34W 135536977 IC50 = 0.78 nM T94879 CR0VL3 135543052 IC50 = 3.7 nM T94879 C45LHQ 135543089 IC50 = 2.76 nM T94879 CX4H6D 135544114 IC50 = 9.1 nM T94879 C4ASW0 135544141 IC50 = 0.6 nM T94879 CYE4C5 135544159 IC50 = 8 nM T94879 CW53FT 135545949 IC50 = 0.31 nM T94879 CK5F9W 135546517 IC50 = 1000 nM T94879 C9VKC6 135547908 IC50 = 10.8 nM T94879 C3HTJ7 135548164 IC50 = 3 nM T94879 C2CXY7 135559102 IC50 = 17 nM T94879 C8HW0M 135565273 IC50 = 8.9 nM T94879 C6J2FV 135566412 IC50 = 110 nM T94879 CHDC83 135566745 IC50 = 1.6 nM T94879 C5S7PD 135566746 IC50 > 1000 nM T94879 C3H1QO 135566795 IC50 = 18.2 nM T94879 CN1OH0 135566796 IC50 = 77 nM T94879 C9IJK1 135566935 IC50 = 90.6 nM T94879 C7M1TE 135604959 IC50 = 5 nM T94879 C6I3HM 135678134 IC50 = 20 nM T94879 CCB89G 135723513 IC50 = 20 nM T94879 CZP1J0 135731499 IC50 = 100 nM T94879 C7VBI4 135740146 IC50 = 82 nM T94879 CIQ83H 135744761 IC50 = 300 nM T94879 C97IUH 135750162 IC50 = 37000 nM T94879 CG1AN3 135790070 IC50 = 200 nM T94879 CD5J1S 135790088 IC50 = 1.76 nM T94879 C0M1LQ 135790105 IC50 = 0.31 nM T94879 CH13EW 135832627 IC50 = 4466.84 nM T94879 C31VFB 135832642 IC50 = 4400 nM T94879 C3PO9K 135856789 IC50 = 7560 nM T94879 C7KDO8 135874585 IC50 = 150 nM T94879 C51XVI 135874586 IC50 = 60 nM T94879 CWT6F3 135890114 IC50 = 5.8 nM T94879 C1EP3X 135890118 IC50 = 6.6 nM T94879 C25PUK 135890126 IC50 = 41 nM T94879 CI4DB0 135890131 IC50 = 4.5 nM T94879 CO07ZA 135890143 IC50 = 1.23 nM T94879 CBI80F 135890150 IC50 = 1.61 nM T94879 CQ8CT6 135890151 IC50 = 4 nM T94879 C8I2XR 135890178 IC50 = 1.01 nM T94879 CTX54Z 135896326 IC50 = 1500 nM T94879 CK4X2F 135898900 IC50 = 100 nM T94879 CPNJ62 135898901 IC50 = 50 nM T94879 C43ZKU 135898902 IC50 = 320 nM T94879 CSO02I 135898910 IC50 = 200 nM T94879 C30ZQG 135898911 IC50 = 510 nM T94879 CJQ74U 135898912 IC50 = 38 nM T94879 C4TRA9 135898925 IC50 = 70 nM T94879 CM2T5C 135898926 IC50 = 140 nM T94879 CH5R6Y 135898941 IC50 = 70 nM T94879 CYJ07O 135898942 IC50 = 530 nM T94879 CR30YL 135898943 IC50 = 500 nM T94879 C0MUP5 135898944 IC50 = 310 nM T94879 CT1H3Q 135898959 IC50 = 370 nM T94879 CU3MH0 135964375 IC50 = 381 nM T94879 CI46LV 135964379 IC50 = 1050 nM T94879 C61SDR 135964388 IC50 > 10000 nM T94879 C42FTR 135964389 IC50 = 116 nM T94879 CZ5UD9 135964390 IC50 = 710 nM T94879 CUQ41O 135964394 IC50 = 2100 nM T94879 C7NRJ6 135964396 IC50 = 849 nM T94879 CY6LT4 135964400 IC50 = 4870 nM T94879 C8UT0J 135964407 IC50 = 634 nM T94879 C04IQT 135964410 IC50 = 2160 nM T94879 C98BHJ 135964418 IC50 = 3340 nM T94879 CS4FT5 135964421 IC50 = 80 nM T94879 CO51CW 135964422 IC50 = 146 nM T94879 CC3HS1 135964423 IC50 = 15 nM T94879 C7KI6V 135964424 IC50 = 1330 nM T94879 C1WB6M 135964425 IC50 = 112 nM T94879 CKSO87 135964426 IC50 = 48 nM T94879 CY24DM 135964428 IC50 = 33 nM T94879 CMYW62 135964429 IC50 = 9 nM T94879 CPL92J 135964430 IC50 = 1570 nM T94879 CLX28E 135964433 IC50 = 38 nM T94879 C6D0FX 136026515 IC50 > 10000 nM T94879 CL7BE5 136032221 IC50 = 1.7 nM T94879 C9OQ5U 136032222 IC50 = 2.1 nM T94879 C6OU3Z 136034782 IC50 = 10 nM T94879 CWPB32 136034783 IC50 = 878 nM T94879 C3KCA0 136042216 IC50 = 0.69 nM T94879 CO4FS2 136042217 IC50 = 0.75 nM T94879 C5MCV8 136042218 IC50 = 2.44 nM T94879 C0EZ4B 136042219 IC50 = 0.74 nM T94879 CX1L3V 136042220 IC50 = 0.86 nM T94879 CS32WP 136042221 IC50 = 0.26 nM T94879 C21HJT 136042222 IC50 = 1.27 nM T94879 C4DP9X 136042223 IC50 = 1.83 nM T94879 CMH5B3 136042224 IC50 = 1.36 nM T94879 CMW86G 136042225 IC50 = 1.01 nM T94879 CJ5X4O 136042226 IC50 = 1.66 nM T94879 CM1TU5 136042227 IC50 = 4.35 nM T94879 C4A6JD 136043740 IC50 = 3.1 nM T94879 CS38OR 136044186 IC50 = 0.58 nM T94879 C6LT3U 136053630 IC50 = 0.29 nM T94879 C9OTF5 136053631 IC50 = 0.28 nM T94879 C5ZIU7 136056125 IC50 = 1000 nM T94879 C70DJG 136056126 IC50 = 2.1 nM T94879 C9Q3BW 136056127 IC50 = 81.28 nM T94879 C4U1SF 136056128 IC50 = 954.99 nM T94879 CI8E5F 136056129 IC50 = 780 nM T94879 CJ43ZC 136059652 IC50 = 3 nM T94879 CZT97J 136059653 IC50 = 77 nM T94879 C2DQ4L 136059654 IC50 = 100 nM T94879 CJ1TW7 136059659 IC50 = 80 nM T94879 CE75BO 136059660 IC50 = 100 nM T94879 C58IEH 136059684 IC50 = 1.1 nM T94879 CG6E8F 136059685 IC50 = 7.7 nM T94879 C97HLB 136059686 IC50 = 5.6 nM T94879 CZQ84P 136059687 IC50 = 0.62 nM T94879 CV6PU2 136059688 IC50 = 0.89 nM T94879 C12UMG 136059728 IC50 = 370 nM T94879 C6WH2S 136078534 IC50 = 10 nM T94879 CE51KZ 136079586 IC50 = 4 nM T94879 CRP24A 136087045 IC50 = 417 nM T94879 C7SUX4 136087050 IC50 = 141 nM T94879 C8UF7G 136087052 IC50 = 3300 nM T94879 C6U2FG 136104505 IC50 = 0.18 nM T94879 CB1GP4 136104506 IC50 = 0.28 nM T94879 CIC08H 136104509 IC50 = 0.41 nM T94879 C0LRM5 136104510 IC50 = 0.34 nM T94879 CNRF74 136104512 IC50 = 0.7 nM T94879 C5LXO8 136104513 IC50 = 0.32 nM T94879 C9UK1F 136132272 IC50 = 100 nM T94879 CBO5H3 136132273 IC50 = 50 nM T94879 CPY6I0 136132274 IC50 = 500 nM T94879 CDE2S8 136132275 IC50 = 300 nM T94879 CPL26N 136132276 IC50 = 1 nM T94879 C4ZBT6 136132277 IC50 = 300 nM T94879 CJ9QG1 136132278 IC50 = 5 nM T94879 C23BTX 136132279 IC50 = 20 nM T94879 C1BFD5 136132280 IC50 = 40 nM T94879 C21FVA 136180322 IC50 = 1.5 nM T94879 C41CAD 136180323 IC50 = 1.7 nM T94879 CC42DB 136180324 IC50 = 1.9 nM T94879 CGJX71 136180325 IC50 = 3.4 nM T94879 C0W3NC 136180326 IC50 = 3.9 nM T94879 CYC9Z6 136180327 IC50 = 12 nM T94879 C5EJ0K 136180328 IC50 = 32 nM T94879 CZ1JH2 136180329 IC50 = 14 nM T94879 C9OM5D 136180330 IC50 = 2.6 nM T94879 CMF1V6 136180331 IC50 = 1.6 nM T94879 C01TYU 136180332 IC50 = 16 nM T94879 CXT68L 136180333 IC50 = 13 nM T94879 CY0T8W 136180334 IC50 = 3.3 nM T94879 C1WHX6 136197281 IC50 = 0.83 nM T94879 CQW7T0 136197286 IC50 = 0.62 nM T94879 CPA8E7 136197297 IC50 = 1.21 nM T94879 CS8TV5 136197304 IC50 = 1.7 nM T94879 COTY62 136197323 IC50 = 8.8 nM T94879 C5HIL8 136197357 IC50 = 9.6 nM T94879 CE0F5T 136197398 IC50 = 1.46 nM T94879 CK2FL9 136197415 IC50 = 5.33 nM T94879 CS16YF 136197417 IC50 = 1.86 nM T94879 CN0G6U 136197445 IC50 = 0.92 nM T94879 C8TQ7A 136217455 IC50 = 3300 nM T94879 C4JCZ7 136219297 IC50 = 272 nM T94879 CE32YG 136219298 IC50 = 21.3 nM T94879 CXOM76 136236320 IC50 = 12.6 nM T94879 C65BFU 136236321 IC50 = 58 nM T94879 C96WPH 136236322 IC50 = 8.5 nM T94879 CY2NJ1 136236323 IC50 = 4.8 nM T94879 CUS40O 136236324 IC50 = 13.7 nM T94879 CS9Z1P 136236325 IC50 = 3 nM T94879 CRZ58U 136236326 IC50 = 4.8 nM T94879 C9PIO3 136236327 IC50 = 34.3 nM T94879 CSU3J2 136236328 IC50 = 7.2 nM T94879 C5KF0V 136236329 IC50 > 2000 nM T94879 CDNI42 136236330 IC50 = 312 nM T94879 CI0M5R 136236331 IC50 = 104 nM T94879 CF43SC 136236332 IC50 = 88 nM T94879 CMGK71 136236333 IC50 = 31.5 nM T94879 C9R6HE 136236334 IC50 = 65 nM T94879 C7ZU0K 136236335 IC50 = 71 nM T94879 C2BCV9 136236336 IC50 = 450 nM T94879 CO4S8B 136236337 IC50 > 2000 nM T94879 C6N2KA 136236338 IC50 = 12.5 nM T94879 CN69OZ 136239327 IC50 = 6.2 nM T94879 C63FEW 136239328 IC50 = 29.3 nM T94879 CQZR23 136244112 IC50 = 48 nM T94879 CO9M4H 136244113 IC50 = 10.2 nM T94879 CK6GB7 136244114 IC50 = 74 nM T94879 CF5BV2 136244123 IC50 = 25.5 nM T94879 C5VT4W 136244124 IC50 = 11.1 nM T94879 CZD04T 136244125 IC50 = 2.8 nM T94879 CUQA38 136244132 IC50 = 17.4 nM T94879 CILG36 136286746 IC50 = 3 nM T94879 C39WRP 136286747 IC50 = 3 nM T94879 C7ZX5O 136286761 IC50 = 48 nM T94879 C9SV6G 136645392 IC50 = 65 nM T94879 CANQ56 136645396 IC50 = 53 nM T94879 C9TGH1 136645397 IC50 = 14 nM T94879 C1F7JV 136645401 IC50 = 144 nM T94879 C32LNQ 136645404 IC50 = 149 nM T94879 C4W0IE 136645405 IC50 = 27 nM T94879 CMIU28 136645406 IC50 = 40 nM T94879 C3K2WL 136645410 IC50 = 79 nM T94879 CC1D0X 136645415 IC50 = 20 nM T94879 C02RIK 136645417 IC50 = 12 nM T94879 C8CT0Z 136645422 IC50 = 20 nM T94879 CAWT82 136645431 IC50 = 10 nM T94879 CBZ8Q1 136645433 IC50 = 22 nM T94879 C21EJD 136645435 IC50 = 2 nM T94879 C1KTV3 136645436 IC50 = 36 nM T94879 CK1B9W 136645438 IC50 = 1 nM T94879 C6QOP7 136645441 IC50 = 7 nM T94879 CMZ71T 136645444 IC50 = 10 nM T94879 CL47WS 136645445 IC50 = 3 nM T94879 C64BZR 136645447 IC50 = 44 nM T94879 C7X1UL 136645449 IC50 = 5 nM T94879 CI9ZO7 136645454 IC50 = 13 nM T94879 CA3I8S 136645455 IC50 = 2 nM T94879 CRN16W 136645457 IC50 = 1 nM T94879 CGQ92L 136645458 IC50 = 2 nM T94879 CO5DN2 136645462 IC50 = 2 nM T94879 CRPN39 136645466 IC50 = 11 nM T94879 CL5X3G 136645467 IC50 = 3 nM T94879 C48HNY 136959539 IC50 = 74 nM T94879 C1P8ZW 136959550 IC50 = 5 nM T94879 CKU95F 136966187 IC50 = 17 nM T94879 CFRG19 136985286 IC50 = 15 nM T94879 CE7F4O 136985287 IC50 = 10 nM T94879 CFPT21 136985288 IC50 = 0.5 nM T94879 CBH5Y0 136985291 IC50 = 24 nM T94879 CDAK28 136985292 IC50 = 0.6 nM T94879 CQ9XW7 136985295 IC50 = 122 nM T94879 C1M6NW 136985296 IC50 = 31 nM T94879 CJOA28 136985302 IC50 = 3 nM T94879 C8HG0E 137051684 IC50 = 2.02 nM T94879 CANS59 137136982 IC50 = 47 nM T94879 C5AE3Q 137283418 IC50 = 19 nM T94879 C0KM1X 137288419 IC50 = 2439 nM T94879 C5QIX1 137289788 IC50 = 17 nM T94879 C5X0YR 137289866 IC50 = 7 nM T94879 CU70ZB 137289868 IC50 = 207 nM T94879 CV6AN7 137289892 IC50 = 57 nM T94879 CB14CI 137289900 IC50 = 5 nM T94879 CLY69S 137289946 IC50 = 13 nM T94879 CC5HA4 137290225 IC50 = 121 nM T94879 C4RBC7 137290234 IC50 = 4 nM T94879 CKJ6Q4 137290238 IC50 = 46 nM T94879 CR53GQ 137290273 IC50 = 34 nM T94879 C8DYG6 137290344 IC50 = 13 nM T94879 C9G3JB 137292402 IC50 = 7 nM T94879 C6MXL3 137292504 IC50 = 57 nM T94879 CAZ49O 137300702 IC50 = 4 nM T94879 CGE0J6 137300703 IC50 = 165 nM T94879 CDU43L 137300704 IC50 = 11 nM T94879 CK0QG6 137300705 IC50 = 303 nM T94879 C91IPL 137300706 IC50 = 70 nM T94879 C5UYP8 137300707 IC50 = 5 nM T94879 CHSG63 137300708 IC50 = 23 nM T94879 CX57MR 137300709 IC50 = 39 nM T94879 C54KGS 137300710 IC50 = 10 nM T94879 CQD07Z 137300711 IC50 = 20 nM T94879 C3I1CB 137300712 IC50 = 38 nM T94879 C2N9VT 137348687 IC50 > 10000 nM T94879 C14DWB 137631637 IC50 = 157510 nM T94879 CML1E3 137631792 IC50 > 100 nM T94879 CA92EX 137632005 IC50 = 31 nM T94879 C5HM3W 137632322 IC50 = 17600 nM T94879 C0SGD8 137633727 IC50 = 77 nM T94879 CTRF70 137634642 IC50 > 100 nM T94879 CO7J5T 137635211 IC50 > 100 nM T94879 CF6EZ1 137635781 IC50 > 1000000 nM T94879 CKB51U 137637339 IC50 = 100000 nM T94879 CU17GD 137637935 IC50 = 5.4 nM T94879 C8RG2S 137638853 IC50 > 100 nM T94879 CA3BX6 137639488 IC50 > 100 nM T94879 C49UCG 137642312 IC50 > 100 nM T94879 C8R1GD 137644106 IC50 > 100 nM T94879 CSQ7P5 137644148 IC50 = 16 nM T94879 CM57EI 137646989 IC50 = 3.1 nM T94879 CPLM78 137647044 IC50 = 56 nM T94879 C18JOP 137647693 IC50 = 30 nM T94879 C4V8QP 137648482 IC50 = 50000 nM T94879 CSW42J 137651273 IC50 = 50 nM T94879 CH6EC3 137653604 IC50 > 100 nM T94879 CPK1J0 137654639 IC50 > 100 nM T94879 C93WRT 137655765 IC50 > 100 nM T94879 CDQ8B5 137657724 IC50 > 100 nM T94879 CY57JX 137658794 IC50 = 21 nM T94879 C2ITK1 137660715 IC50 > 100 nM T94879 CJA7I0 137662139 IC50 = 100000 nM T94879 C6KYD7 137700754 IC50 = 4010 nM T94879 CM3UF7 137700779 IC50 > 20000 nM T94879 CPTE92 138319693 IC50 = 0.32 nM T94879 C2QLX3 138393292 IC50 > 5000 nM T94879 CF3B2O 141492937 IC50 = 0.52 nM T94879 CEK54I 141492938 IC50 = 1.2 nM T94879 CMJW70 141492939 IC50 = 3.28 nM T94879 CKB05G 141492943 IC50 = 0.53 nM T94879 CU6A0R 141492944 IC50 = 2.85 nM T94879 CW7NV6 141492945 IC50 = 0.6 nM T94879 C2NW6Y 141492955 IC50 = 0.67 nM T94879 C13PVI 141492968 IC50 = 0.6 nM T94879 C42GOU 141492970 IC50 = 26.9 nM T94879 CGNK49 141492971 IC50 = 0.82 nM T94879 CXN3U7 141492981 IC50 = 86 nM T94879 CZ0M1Y 141492988 IC50 = 1.25 nM T94879 C2T8GE 141492992 IC50 = 6.45 nM T94879 C5XTB1 141492998 IC50 = 2.5 nM T94879 C93ZIQ 141492999 IC50 = 0.39 nM T94879 CUXZ06 141493000 IC50 = 0.97 nM T94879 C7RTX9 141493002 IC50 = 3.14 nM T94879 CQV0B4 141737648 IC50 = 155 nM T94879 C0JV6Y 141737649 IC50 = 39.7 nM T94879 CSOF52 141737655 IC50 = 19.9 nM T94879 C7SRA2 141737657 IC50 = 7.02 nM T94879 CE1H7F 141737660 IC50 = 97.5 nM T94879 CA5UL8 141737663 IC50 = 61 nM T94879 C6ZA7D 141737664 IC50 = 36.9 nM T94879 CMIY07 141737666 IC50 = 21.4 nM T94879 CC61SD 141737667 IC50 = 30.3 nM T94879 C14CZJ 141737668 IC50 = 8.44 nM T94879 CTNG49 141737674 IC50 = 36.4 nM T94879 CJ38IC 141737676 IC50 = 12.7 nM T94879 C1MC5Z 141737681 IC50 = 8.68 nM T94879 CK34HF 141737682 IC50 = 50.2 nM T94879 CQCM72 141737683 IC50 = 177 nM T94879 C2MEL1 141737684 IC50 = 56.4 nM T94879 CTUL23 141737690 IC50 = 5.24 nM T94879 CMW20N 141737696 IC50 = 3.87 nM T94879 CZWD98 141737697 IC50 = 80.2 nM T94879 C7GBH6 141737698 IC50 = 52.5 nM T94879 CVQJ85 141737699 IC50 = 383 nM T94879 CO1C4S 141737703 IC50 = 27.6 nM T94879 CX9N1P 141737704 IC50 = 10.5 nM T94879 C8HEG7 141737705 IC50 = 2.92 nM T94879 C8OWX3 145964082 IC50 = 2.64 nM T94879 C0P7CN 145964738 IC50 = 3.04 nM T94879 CZ1M5C 145964966 IC50 = 1.58 nM T94879 C07GTQ 145966108 IC50 = 0.79 nM T94879 C38QXR 145966233 IC50 = 251.19 nM T94879 CUM0Y5 145968257 IC50 = 6.82 nM T94879 CO4N2T 145968939 IC50 = 2.09 nM T94879 CDHG23 145971317 IC50 = 9.63 nM T94879 CMNV65 145973708 IC50 = 1.05 nM T94879 CC7HN2 145974174 IC50 > 100000 nM T94879 CIFW03 145974279 IC50 = 0.52 nM T94879 CWM49T 145974605 IC50 = 1.63 nM T94879 C2JF3R 145974856 IC50 = 2.64 nM T94879 C8BEH3 145975382 IC50 = 2.38 nM T94879 C5C6NR 145976885 IC50 = 2.37 nM T94879 CTJ6L8 145977069 IC50 = 0.39 nM T94879 C6M5ZW 145977440 IC50 = 19.95 nM T94879 CDB1E7 145977898 IC50 = 4.38 nM T94879 CK1BR0 145978345 IC50 > 100000 nM T94879 CJD7B2 145978603 IC50 = 4.03 nM T94879 CU5VD3 145978669 IC50 = 3.82 nM T94879 C9LGT4 145979889 IC50 = 235 nM T94879 CKZ1Y6 145979895 IC50 = 170 nM T94879 C50DFR 145982956 Ki = 8 nM T94879 CKTF58 145987769 IC50 = 227 nM T94879 CJA1B0 145991631 IC50 = 81.2 nM T94879 CHJ79V 145997874 IC50 = 3390 nM T94879 CM7TX2 148279038 IC50 = 1530 nM T94879 CYPW78 155510908 IC50 = 1.55 nM T94879 C6VZ5O 155514730 IC50 = 1.69 nM T94879 CL8CU6 155521936 IC50 > 200000 nM T94879 CAUO07 155524955 IC50 = 0.54 nM T94879 CT85RG 155530589 IC50 > 200000 nM T94879 CXMU51 155537188 IC50 = 0.79 nM T94879 C1IP4D 155556194 IC50 = 3.9 nM T94879 C2DA1W 155561694 IC50 > 500000 nM T94879 CQ2R0W 155568588 IC50 > 500000 nM T94879 CV07RN 44579973 IC50 = 0.6166 nM T94879 D00REK 5712 IC50 = 31900 nM T94879 D01RLF 105078 IC50 = 794.33 nM T94879 D01TOR 667555 IC50 = 450 nM T94879 D02NWF 2573787 IC50 = 720 nM T94879 D02VRN 6442679 IC50 = 1470 nM T94879 D03BWH 44587253 IC50 = 360 nM T94879 D06NIT 135564899 IC50 = 349 nM T94879 D06TLQ 5488822 IC50 = 1700 nM T94879 D09AUL 10266864 IC50 = 260 nM T94879 D09RKU 46239428 Ki = 9700 nM T94879 D09WUP 25058047 IC50 = 74 nM T94879 D0I6XA 149784 Ki > 200000 nM T94879 D0J0CB 2753 IC50 = 7150 nM T94879 D0J7GF 780643 IC50 = 320 nM T94879 D0O3QI 10356247 IC50 = 4200 nM T94879 D0R6MT 3758 IC50 = 63000 nM T94879 D0S8AV 509245 IC50 = 16230 nM T94879 D0U8YQ 921562 IC50 = 310 nM T94879 D0V1CL 37015 IC50 = 180 nM T94879 D0V4WB 149790 IC50 > 16000 nM T94879 D0W2BI 9799499 IC50 = 700 nM T94879 D0X7SR 10246505 IC50 = 1290 nM T94879 D0YZ0L 44605341 IC50 = 12600 nM T98337 D06OMK 445643 Ki = 79 nM T98337 D02VJY 3037617 IC50 = 8520 nM T98337 D04PGB 445501 IC50 > 100000 nM T98337 CRD1T0 9811664 IC50 > 100000 nM T98337 C9IS6O 9820942 IC50 > 150000 nM T98337 CSN72K 10371065 IC50 = 8360 nM T98337 CF3GI4 10508532 Ki = 600 nM T98337 C5NB9Z 11129344 IC50 > 100000 nM T98337 CTLC58 35027274 IC50 = 3800 nM T98337 C2V6RJ 56962328 IC50 = 3900 nM T98337 CJ46RD 56962330 IC50 = 3900 nM T98337 C1BUW4 57521458 IC50 = 8500 nM T98337 CGU89M 57521460 IC50 > 100000 nM T98337 CKP31Q 57521461 IC50 = 4150 nM T98337 C7D3PN 57521557 IC50 = 15340 nM T98337 CO6T0F 57521558 IC50 = 19300 nM T98337 C2RVN0 57521777 IC50 = 4270 nM T98337 C8PY2R 57521778 IC50 = 4540 nM T98337 C0HOD9 57521879 IC50 = 4180 nM T98337 CS7B2A 57521880 IC50 = 4960 nM T98337 CGP03D 57521881 IC50 = 62800 nM T98337 C9V4QB 57521882 IC50 = 30700 nM T98337 C4C7LK 57522005 IC50 = 11600 nM T98337 C8YI0U 57522006 IC50 > 100000 nM T98337 C0KC6J 57522007 IC50 = 67100 nM T98337 CH89PN 57522008 IC50 = 28500 nM T98337 CG6TK3 57522120 IC50 = 47200 nM T98337 CWQ8J7 57522121 IC50 = 45400 nM T98337 CTCH51 57522237 IC50 = 54050 nM T98337 C8R2IJ 57522238 IC50 = 15780 nM T98337 C1PBX3 57522239 IC50 = 22600 nM T98337 CU5NP7 57522240 IC50 > 100000 nM T98337 C0P3TI 57522347 IC50 > 100000 nM T98337 C6WY9D 57522348 IC50 = 29600 nM T98337 CM7ZV1 57522349 IC50 = 88200 nM T98337 C6FQ4X 57522350 IC50 > 100000 nM T98337 CHVK79 57522455 IC50 > 100000 nM T98337 C73XQS 57522456 IC50 > 100000 nM T98337 C4OJX2 57522457 IC50 = 6200 nM T98337 CGIX69 57522458 IC50 = 16400 nM T98337 CG2SO6 57522567 IC50 = 16100 nM T98337 CR9C3F 57522569 IC50 = 27200 nM T98337 C8SP3L 57522570 IC50 > 100000 nM T98337 CQ3I7G 57522682 IC50 = 18400 nM T98337 C5QM2O 57522683 IC50 = 14700 nM T98337 CE7G2U 57522684 IC50 > 100000 nM T98337 CA4R9I 57522685 IC50 > 100000 nM T98337 C3EP9M 57522800 IC50 > 100000 nM T98337 C46EIF 57522801 IC50 = 66270 nM T98337 CC85GJ 57522802 IC50 > 50000 nM T98337 CCUW31 57522803 IC50 > 50000 nM T98337 CV58SP 57522927 IC50 = 51500 nM T98337 CT58KB 57522928 IC50 = 456 nM T98337 C95OGY 57522929 IC50 > 50000 nM T98337 CZI07G 57522930 IC50 = 2030 nM T98337 C8B9HE 57522931 IC50 = 12300 nM T98337 C7Y9SK 57523063 IC50 = 32730 nM T98337 C4S5KW 57523064 IC50 > 100000 nM T98337 CT4NB0 57523068 IC50 > 100000 nM T98337 C0NUH8 57523069 IC50 > 100000 nM T98337 C2YN0S 57523070 IC50 = 9690 nM T98337 CN1S5R 60123375 Ki = 2700 nM T98337 C2DIM5 70684253 IC50 > 100000 nM T98337 CYQH64 70684260 IC50 = 9660 nM T98337 CG5D2W 70688508 IC50 > 100000 nM T98337 CWDU09 70688522 IC50 = 9130 nM T98337 CWY7C0 70692710 IC50 = 29390 nM T98337 C5MK3W 70694725 IC50 > 100000 nM T98337 CD65LN 70694726 IC50 > 100000 nM T98337 CEZG14 70694756 IC50 > 100000 nM T98337 CU9RN3 70694757 IC50 = 2020 nM T98337 C1Q7UX 71662419 Ki > 100000 nM T98337 CR5Q3M 71662579 Ki > 100000 nM T98337 CJHR74 71662580 Ki > 100000 nM T98337 C8G3VC 71662581 Ki = 7600 nM T98337 COBA89 71662582 Ki > 100000 nM T98337 CK4E7Q 71716537 Ki = 8800 nM T98337 CWY3J5 71716538 Ki = 64800 nM T98337 CCLG13 71716539 Ki = 200 nM T98337 CUD8F9 71717141 Ki = 9800 nM T98337 C7TIC3 71717142 Ki > 100000 nM T98337 C34VNG 71717766 Ki = 1000 nM T98337 CSIY48 71717767 Ki = 51100 nM T98337 C24GAX 71718373 Ki = 1200 nM T98337 CRGS91 71718374 Ki = 2100 nM T98337 CRWB36 71718375 Ki > 100000 nM T98337 C61TIG 71718376 Ki > 100000 nM T98337 CW0T3A 71718980 Ki = 27000 nM T98337 CR9FQ3 71718981 Ki = 18100 nM T98337 CS71CH 71720178 Ki = 13900 nM T98337 C0D6ZR 71720179 Ki = 13800 nM T98337 CK36QR 71720180 Ki > 100000 nM T98337 C9TVZ3 71720822 Ki = 300 nM T98337 CUT2Y6 71720824 Ki > 100000 nM T98337 C9N7TY 71720825 Ki = 23700 nM T98337 C5EMH2 86277875 Ki = 4 nM T98337 C3XNC8 86277887 Ki = 6 nM T98337 C85VMY 91936975 Ki = 700 nM T98337 CCH84L 117967740 Ki = 4900 nM T98337 CXP8S2 117967763 Ki = 800 nM T98337 CEY28F 117967783 Ki = 1500 nM T98337 C46GRQ 117967787 Ki = 140 nM T98337 C2A8EM 117967798 Ki = 7100 nM T98337 CVP4Q3 117967801 Ki = 3400 nM T98337 CWTL26 117967814 Ki = 3400 nM T98337 C5GF3N 117967822 Ki = 3600 nM T98337 C93YQU 117967826 Ki = 62900 nM T98337 CJ26YR 117967829 Ki = 17100 nM T98337 CX51BA 117967835 Ki = 43 nM T98337 C2AF1T 117967843 Ki = 3800 nM T98337 CRCH91 117967851 Ki = 3800 nM T98337 CT3DQ5 117967872 Ki = 10000 nM T98337 C7NTU4 117967885 Ki = 19500 nM T98337 CYS70L 117967909 Ki = 13400 nM T98337 CU86WK 117967913 Ki = 4500 nM T98337 CFA74P 117967937 Ki = 6500 nM T98337 C08BKM 117967939 Ki = 12600 nM T98337 CHN52K 117967946 Ki = 1400 nM T98337 C1ZYL4 117967947 Ki = 4200 nM T98337 CA6ZJ7 117967955 Ki = 13000 nM T98337 C2QZ3D 117967964 Ki = 8700 nM T98337 C07HJM 117967978 Ki = 12000 nM T98337 CSD64M 117968002 Ki = 17800 nM T98337 CTI1X7 117968005 Ki = 1200 nM T98337 CXP8N7 117968006 Ki = 1900 nM T98337 CIS63B 117968011 Ki = 55000 nM T98337 C4LAX1 117968012 Ki = 3200 nM T98337 C58LQV 117968031 Ki = 9100 nM T98337 CF1GO9 117968050 Ki = 36700 nM T98337 CXLE07 117968053 Ki = 3100 nM T98337 CXWU20 117968117 Ki = 2800 nM T98337 CZQB61 117968118 Ki = 4300 nM T98337 C5LK3R 117968129 Ki = 345000 nM T98337 CG65FE 117968136 Ki = 2200 nM T98337 C5O7SB 117968142 Ki = 5000 nM T98337 C5EU1T 117968149 Ki = 7900 nM T98337 CEXT51 117975049 Ki = 1800 nM T98337 CNP23H 122192627 Ki = 110 nM T98337 CEMN03 122192628 Ki = 160 nM T98337 C5ZF3W 122192629 Ki = 4200 nM T98337 C6S7FW 122192630 Ki = 4100 nM T98337 C0K9LY 122192631 Ki = 2000 nM T98337 CE4H8R 122192632 Ki = 2100 nM T98337 CHF0M4 122192633 Ki = 2000 nM T98337 C4A8CV 122192634 Ki = 2500 nM T98337 CK1Y9T 122192635 Ki = 1100 nM T98337 C1MC5U 122192636 Ki = 13000 nM T98337 C1HI5B 122192637 Ki = 17000 nM T98337 C40FKQ 122192638 Ki = 9000 nM T98337 CN6C1I 122192639 Ki > 100000 nM T98337 CC0L6K 127024999 Ki = 5700 nM T98337 C0SKD7 127053468 Ki = 3900 nM T98337 C1P6LO 137642835 Ki = 24.5 nM T98337 C64OBX 145707024 Ki = 230 nM T98337 CRFO70 155516049 Ki = 7800 nM T98337 CGK3T7 155524130 Ki = 810 nM T98337 CPN64O 155525030 Ki = 2600 nM T98337 CQK12X 155526064 Ki = 330 nM T98337 CC21ES 155526980 Ki = 2000 nM T98337 C4O3HP 155529425 Ki = 280 nM T98337 CH3B0K 155535419 Ki = 1300 nM T98337 CO9CS5 155539683 Ki = 28000 nM T98337 CI78TG 155545147 Ki = 3100 nM T98337 CO7S8A 155545716 Ki = 2600 nM T98337 C4AG5E 155551666 Ki = 8200 nM T98337 CP7U4H 155552889 Ki = 2400 nM T98337 CT40BW 155554017 Ki = 490 nM T98337 CKL6H4 155562050 Ki = 650 nM T98337 C4OH7J 155564329 Ki = 1900 nM T13902 CYG60X 512874 Ki = 81.4 nM T13902 CBL1C6 10883540 EC50 = 430 nM T13902 C8C9HM 11132282 EC50 = 22 nM T13902 CB96ZX 24742075 Ki = 64.3 nM T13902 CYL7A6 24825421 EC50 = 90 nM T13902 CI38DG 24825422 EC50 = 12 nM T13902 C5T6WY 24825423 EC50 = 160 nM T13902 CB8EU6 24825424 EC50 = 100 nM T13902 CN5Q0O 24825425 EC50 = 60 nM T13902 CWQU39 24825426 EC50 = 1400 nM T13902 C5EIS2 24825427 EC50 > 10000 nM T13902 CH3YB9 24825428 EC50 = 70 nM T13902 C9NPK4 24825429 EC50 = 320 nM T13902 C7OI1S 24825430 EC50 = 2100 nM T13902 CXRQ34 24825431 EC50 = 31.62 nM T13902 C4WTY2 24825432 EC50 = 230 nM T13902 C9ZDA7 24825433 EC50 > 10000 nM T13902 CLW5C7 24825434 EC50 = 150 nM T13902 CFV48O 24825435 EC50 = 330 nM T13902 C2FKX4 24825436 EC50 = 1000 nM T13902 CV25CA 24825437 EC50 = 30 nM T13902 COM6B8 24825438 EC50 > 10000 nM T13902 CYM47L 24825439 EC50 > 10000 nM T13902 CK4AB0 24825440 EC50 > 10000 nM T13902 CN84ZX 24825441 EC50 = 1200 nM T13902 C4RS1G 52936713 EC50 = 251.19 nM T13902 CA15HU 52936816 EC50 = 398.11 nM T13902 C6BH1V 52936819 EC50 = 1000 nM T13902 CRY03J 52936822 EC50 = 2511.89 nM T13902 CWRU85 52936928 EC50 = 2511.89 nM T13902 CF7M2A 52936929 EC50 = 3162.28 nM T13902 C2GV4R 52936930 EC50 = 5011.87 nM T13902 CAT2L4 52936931 EC50 = 2511.89 nM T13902 COLN94 52936934 EC50 = 794.33 nM T13902 CR6HC7 52937033 EC50 = 100 nM T13902 C2TI8L 52937034 EC50 = 251.19 nM T13902 CCWO80 52937035 EC50 = 316.23 nM T13902 CJ6K7I 52937037 EC50 = 1995.26 nM T13902 CI4Q9R 52937137 EC50 = 1000 nM T13902 CY10CO 52937140 EC50 = 3162.28 nM T13902 C6W5GH 52937141 EC50 = 2511.89 nM T13902 CENW79 52937246 EC50 = 251.19 nM T13902 C7I0MG 52937350 EC50 = 1258.93 nM T13902 CJ3E9B 52937351 EC50 = 794.33 nM T13902 CKC03F 52937353 EC50 = 199.53 nM T13902 CO6AG4 52937354 EC50 = 1584.89 nM T13902 CM7UT9 52937355 EC50 = 158.49 nM T13902 C45YZW 52937356 EC50 = 1258.93 nM T13902 CG98BX 52937447 EC50 = 316.23 nM T13902 CX32GP 52937449 EC50 = 398.11 nM T13902 CING80 52937450 EC50 = 251.19 nM T13902 C68SHU 52937451 EC50 = 1584.89 nM T13902 CHOZ17 52937452 EC50 = 501.19 nM T13902 CL96WV 54580360 EC50 = 251.19 nM T13902 CC67DZ 126673332 Ki = 7000 nM T13902 C16CVG 138857911 EC50 = 600 nM T13902 C0NF4Q 138857912 EC50 = 15 nM T13902 CRFJ45 138857913 EC50 = 13000 nM T13902 CZ93GB 139030532 Ki = 2.1 nM T13902 CE3T1J 145984173 EC50 = 13000 nM T13902 C36QJH 145988910 EC50 = 5000 nM T13902 C97VJP 145990098 EC50 = 400 nM T13902 C0AIB6 155518824 EC50 = 40 nM T13902 C94IEB 155522101 Ki = 2400 nM T13902 CN7HV4 155522503 EC50 = 900 nM T13902 CTR04M 155524650 EC50 = 800 nM T13902 CF3P4T 155527718 EC50 = 1000 nM T13902 C7LHO4 155535510 EC50 = 2000 nM T13902 C91LUA 155539274 EC50 = 9000 nM T13902 CR8AY9 155545328 EC50 = 5000 nM T13902 CG4QF6 155551225 EC50 = 500 nM T13902 C96DYA 155554234 EC50 = 100 nM T13902 CTX5J9 155557666 EC50 = 800 nM T13902 CD8TS3 155558831 EC50 = 3000 nM T13902 CJF3I2 155564002 EC50 = 4000 nM T64213 D0CO6D 71144018 IC50 > 20000 nM T64213 C9F7YI 556143 IC50 = 10 nM T64213 CZN6S9 743974 EC50 > 125892.54 nM T64213 CEFQ61 973047 IC50 = 490 nM T64213 CO19JL 1068397 IC50 = 34 nM T64213 CSXT30 1075105 EC50 = 770 nM T64213 CE0N7K 2124297 IC50 = 4220 nM T64213 CMC2Q6 2877560 IC50 = 10000 nM T64213 CZ1L9C 2898103 IC50 = 31 nM T64213 CPS8X2 11713900 EC50 = 740 nM T64213 C7FBO1 25270198 IC50 > 100000 nM T64213 C23WVS 53361524 IC50 > 10000 nM T64213 CAW4F0 53464379 IC50 = 50 nM T64213 CC21VN 53464543 IC50 = 50 nM T64213 CU78MC 53464607 IC50 = 80 nM T64213 C7I8YR 53465062 IC50 = 10 nM T64213 C5DBC6 53465181 IC50 = 250 nM T64213 CFZQ89 59672648 IC50 = 4930 nM T64213 CIMP91 59673363 IC50 = 930 nM T64213 C0JKR9 71116078 IC50 = 16 nM T64213 CSH8F6 71116172 IC50 = 0.001 nM T64213 CH2E7C 71116460 IC50 = 1.6 nM T64213 C87JXW 71135581 IC50 = 240 nM T64213 C1TQ6W 71135583 IC50 = 140 nM T64213 C5L7HN 71135586 IC50 = 540 nM T64213 CY31NM 71135589 IC50 = 0.001 nM T64213 CSIB17 71136917 IC50 = 74 nM T64213 CN5D4T 71226967 IC50 = 49 nM T64213 CMO71T 71227359 IC50 = 1.8 nM T64213 C51APH 71227580 IC50 = 7.5 nM T64213 C4M9YA 71227675 IC50 = 4.2 nM T64213 CA8Y2J 71227691 IC50 = 14 nM T64213 CO03PX 71227697 IC50 = 1.2 nM T64213 COA09X 71227729 IC50 = 3.1 nM T64213 CXN0D7 71473867 IC50 = 0.001 nM T64213 CX51CS 71474186 IC50 = 1.7 nM T64213 C4D8YT 71474187 IC50 = 5.2 nM T64213 CWA7J3 71474188 IC50 = 1.2 nM T64213 CF50JQ 71474549 IC50 = 5.2 nM T64213 C95VNA 71474551 IC50 = 48 nM T64213 CPG0L8 71491020 IC50 = 0.5 nM T64213 CM34DA 71528444 IC50 = 200 nM T64213 CB8S7P 71528445 IC50 = 5010 nM T64213 CJMG81 71528446 IC50 = 631 nM T64213 CA7MF1 71528447 IC50 = 1000 nM T64213 C6TKZ1 71528448 IC50 = 3980 nM T64213 CCGW28 71528449 IC50 = 2510 nM T64213 C1G7SZ 71528586 IC50 = 1260 nM T64213 CB1XZ5 71528587 IC50 = 126 nM T64213 CX8V9F 71528588 IC50 = 126 nM T64213 CO91MV 71528589 IC50 = 50.1 nM T64213 C9VTG4 71528590 IC50 = 31.6 nM T64213 C15NRD 71528731 IC50 = 12.6 nM T64213 CV4L1C 71528732 IC50 = 15.8 nM T64213 C4PJA7 71528733 IC50 > 10000 nM T64213 C3OT1F 71528734 IC50 = 31.6 nM T64213 C23JVX 71528735 IC50 = 3.2 nM T64213 CW20HQ 71818431 IC50 = 6300 nM T64213 C2L7TX 71818575 IC50 = 12500 nM T64213 CAN5C1 88057277 IC50 = 60 nM T64213 CT4WJ0 90107022 IC50 = 60 nM T64213 CIE3D4 90108382 IC50 = 60 nM T64213 C1EI2P 90665449 IC50 = 2200 nM T64213 C43XPQ 90665450 IC50 = 12.9 nM T64213 CF9CT5 90665451 IC50 = 49.1 nM T64213 C6SU4X 90665452 IC50 = 49.7 nM T64213 CUQK96 90665453 IC50 = 50.5 nM T64213 CSR8D7 90665454 IC50 = 3.4 nM T64213 CXR4H8 90665455 IC50 = 3.6 nM T64213 CJCR26 90665456 IC50 = 3.8 nM T64213 C6C9KP 90665457 IC50 = 4 nM T64213 CJ06SU 91535935 IC50 = 2000 nM T64213 C8Z2ED 117848832 IC50 = 3300 nM T64213 CDNC39 118246723 IC50 > 30000 nM T64213 CMC6G4 121476731 IC50 = 2.4 nM T64213 COR6Q4 121476832 IC50 = 22 nM T64213 C5YP4M 121476835 IC50 = 290 nM T64213 C54XVT 121476884 IC50 = 37 nM T64213 C3UO2A 121476940 IC50 = 200 nM T64213 C9F6PK 121476942 IC50 > 10000 nM T64213 C3TYW2 121476950 IC50 = 240 nM T64213 CD8P1F 121476973 IC50 = 50 nM T64213 C36RBL 121476974 IC50 = 9.5 nM T64213 CZTA14 121476982 IC50 = 29 nM T64213 CL86RI 121477020 IC50 = 35 nM T64213 CK3RB5 121477188 IC50 > 10000 nM T64213 C1XNR3 121513880 IC50 = 420 nM T64213 C58IUP 122189178 IC50 = 8530 nM T64213 CT5C4U 122189179 IC50 = 390 nM T64213 C1RML6 122189180 IC50 = 710 nM T64213 C8HCS3 122189181 IC50 = 2170 nM T64213 CO8M5U 122189182 IC50 > 10000 nM T64213 CU71OA 122189183 IC50 > 10000 nM T64213 C5LZW6 122189184 IC50 = 1320 nM T64213 CDJL98 122189185 IC50 = 2110 nM T64213 CS3R2X 122189186 IC50 = 910 nM T64213 C2BCJ7 122189187 IC50 = 1280 nM T64213 CG25YT 122189188 IC50 = 800 nM T64213 C7MG6P 122189189 IC50 = 260 nM T64213 CF8H0M 122189190 IC50 = 380 nM T64213 C9U6RS 122189191 IC50 = 540 nM T64213 CGFS72 122189192 IC50 = 930 nM T64213 CJZ7Y8 132569635 IC50 = 0.22 nM T64213 CF3D1C 134132776 IC50 = 2.8 nM T64213 CL8FX6 134133585 IC50 = 2.9 nM T64213 CQ2TE9 134133674 IC50 = 6.2 nM T64213 CQ08IP 134133949 IC50 = 32 nM T64213 C2B6MJ 134134519 IC50 = 46 nM T64213 CTJF87 134134782 IC50 = 3.1 nM T64213 C6K7GU 134134874 IC50 = 19 nM T64213 C8S6CT 134135548 IC50 = 530 nM T64213 CS6U7A 134137835 IC50 = 0.57 nM T64213 CROG58 134137935 IC50 = 80 nM T64213 C8IHX2 134138693 IC50 = 11 nM T64213 CFUV82 134141361 IC50 = 4.8 nM T64213 CS1MI5 134141572 IC50 = 1.7 nM T64213 CG80PJ 134141709 IC50 = 24 nM T64213 CN7PO6 134141941 IC50 = 23 nM T64213 CSX9J5 134142444 IC50 = 4.5 nM T64213 C23GVR 134142674 IC50 = 6.7 nM T64213 C84HMG 134142778 IC50 = 32 nM T64213 CBH3N5 134142854 IC50 = 1 nM T64213 CWQL46 134143254 IC50 = 410 nM T64213 C5B0ET 134143719 IC50 = 4300 nM T64213 CT51MF 134144463 IC50 = 6.3 nM T64213 CU7Z6W 134144502 IC50 = 620 nM T64213 CC3YF9 134145287 IC50 = 24 nM T64213 CJ51TH 134145916 IC50 = 3.2 nM T64213 CFQ3K6 134146321 IC50 = 770 nM T64213 C0UAK3 134147888 IC50 = 0.9 nM T64213 CIF84U 134147900 IC50 > 10000 nM T64213 CS24KA 134151107 IC50 = 4.4 nM T64213 C7YIN4 134151570 IC50 = 8.4 nM T64213 C10JCN 134151583 IC50 = 41 nM T64213 CS9M2H 134152318 IC50 = 2.1 nM T64213 C1N0XO 134152649 IC50 = 3.2 nM T64213 CR2F9S 134153899 IC50 = 0.3 nM T64213 CWXZ15 134153919 IC50 > 10000 nM T64213 C80DVZ 134154618 IC50 = 240 nM T64213 C2DIV9 134154947 IC50 = 100 nM T64213 CM2C7B 134155100 IC50 = 1.1 nM T64213 C9S3QG 134155876 IC50 = 37 nM T64213 CU8P2F 134156601 IC50 = 0.36 nM T64213 CUN57J 134156774 IC50 = 620 nM T64213 CFM1G7 134156905 IC50 = 1.8 nM T64213 C8FP7C 134157491 IC50 = 1.9 nM T64213 C24WTD 134157985 IC50 = 6 nM T64213 C1OTG4 134367627 IC50 = 1 nM T64213 C5JV2O 134374891 IC50 = 5 nM T64213 C3TW0A 134374895 IC50 = 3.2 nM T64213 CVLH60 134374993 IC50 = 0.5 nM T64213 CF24PS 134378771 IC50 = 34 nM T64213 C47TLY 134378796 IC50 = 12 nM T64213 CPHO94 137628676 EC50 = 60 nM T64213 C4J3ZS 137632071 IC50 = 0.21 nM T64213 CQ4S0J 137635724 IC50 = 0.65 nM T64213 CG1F7Q 137636243 IC50 = 2 nM T64213 C7AN0Q 137636445 IC50 = 200 nM T64213 C6XVA3 137637570 IC50 = 2000 nM T64213 C5VWH4 137637746 IC50 = 0.62 nM T64213 CC36MB 137638989 IC50 = 500 nM T64213 CP06HM 137639654 IC50 = 2510 nM T64213 CYM4C5 137639667 IC50 = 4.2 nM T64213 C4NIF9 137639683 IC50 = 160 nM T64213 C1XGB3 137639759 IC50 = 64 nM T64213 CZWI69 137639837 IC50 = 1.3 nM T64213 C04ZQU 137640563 IC50 > 25000 nM T64213 CUW2T6 137641026 IC50 = 5010 nM T64213 CS54FI 137641584 IC50 = 40 nM T64213 CISA38 137643086 IC50 = 0.71 nM T64213 C2QP6M 137644050 IC50 = 6.8 nM T64213 CR7W9S 137645621 IC50 = 2000 nM T64213 C7L2QC 137645999 IC50 = 320 nM T64213 CWK5M9 137646962 IC50 = 2.4 nM T64213 CE56RV 137647117 IC50 = 1.3 nM T64213 CKG83O 137647502 IC50 = 0.97 nM T64213 C5G0QR 137647711 IC50 = 1.4 nM T64213 CSJI59 137647785 IC50 = 0.87 nM T64213 CTD69B 137647980 IC50 = 80 nM T64213 CRU69K 137648543 IC50 = 3980 nM T64213 C0T8DE 137649399 IC50 = 60 nM T64213 CKI1J0 137649578 IC50 = 0.39 nM T64213 C5V2WN 137649769 IC50 = 1.8 nM T64213 CJ09RP 137650429 IC50 = 3.7 nM T64213 CXKG32 137650500 IC50 = 3.9 nM T64213 CA17ES 137650754 IC50 = 6.2 nM T64213 C2X4KI 137651468 IC50 = 0.31 nM T64213 CGB1O2 137652110 IC50 = 170 nM T64213 CEC23Z 137652223 IC50 = 1000 nM T64213 CRL59S 137652676 IC50 = 0.5 nM T64213 C6G8IS 137652729 IC50 > 25000 nM T64213 CZOB89 137653593 IC50 = 50 nM T64213 COC3T7 137653869 IC50 = 0.18 nM T64213 CX3JI8 137654148 IC50 = 0.99 nM T64213 CDR68H 137655371 IC50 = 3160 nM T64213 CWH9O5 137657180 IC50 = 6.3 nM T64213 CA6PE5 137657548 IC50 = 100 nM T64213 COLZ09 137657815 IC50 = 500 nM T64213 C36QPL 137659136 IC50 = 1580 nM T64213 CSZT92 137660008 IC50 = 0.29 nM T64213 CW48BQ 137660946 IC50 = 400 nM T64213 C39HPA 137661261 IC50 = 0.19 nM T64213 C4CRB5 137661997 IC50 = 130 nM T64213 CK5GJ8 139300594 IC50 = 175 nM T64213 CYP5F2 139300600 IC50 = 53 nM T64213 CEK6B1 139300630 IC50 = 2.5 nM T64213 CJ02SL 139300726 IC50 = 100 nM T64213 CD9Q0L 139300799 IC50 = 3.8 nM T64213 CK8W0E 139300844 IC50 = 190 nM T64213 CRH14F 139300861 IC50 = 33 nM T64213 C2D9TE 141756938 IC50 = 0.5 nM T64213 CHI60S 141756971 IC50 = 2 nM T64213 C94DWA 141756975 IC50 = 2 nM T64213 C86QVB 141756989 IC50 = 3.2 nM T64213 C9RI2N 141757015 IC50 = 7.9 nM T64213 C53UZY 141757055 IC50 = 0.3 nM T64213 CD05NR 145952261 IC50 = 40 nM T64213 C7Q8VT 145953322 IC50 = 150 nM T64213 C4RD5Z 145954475 IC50 = 1500 nM T64213 CVF6M0 145954552 IC50 = 6300 nM T64213 CE06FU 145955149 IC50 = 50 nM T64213 CCWK87 145956421 IC50 = 150 nM T64213 C5M7JA 145957240 IC50 = 100 nM T64213 CL75MA 145957491 IC50 = 200 nM T64213 CJ1OZ4 145972905 IC50 = 320 nM T64213 C9DO8U 145974540 IC50 = 1000 nM T64213 C7Y6WX 155510800 IC50 = 240 nM T64213 C5ESP7 155512077 EC50 = 10000 nM T64213 CT7JO0 155514099 EC50 = 920 nM T64213 C6TVW5 155515017 IC50 = 290 nM T64213 CJ97CN 155515493 IC50 = 20 nM T64213 CS6UN3 155517309 IC50 = 159 nM T64213 CZ1O0S 155518646 IC50 = 84 nM T64213 CW4J8P 155519095 EC50 > 30000 nM T64213 CE4FD0 155520787 EC50 = 125 nM T64213 CW34OZ 155520969 EC50 = 4700 nM T64213 CZVJ89 155521210 IC50 = 340 nM T64213 CW9RA8 155521362 IC50 = 1700 nM T64213 CQ10LO 155522731 IC50 = 631 nM T64213 CJ2EU3 155523773 EC50 = 1444 nM T64213 C65AUT 155525085 EC50 = 870 nM T64213 CI10UW 155526744 IC50 > 10000 nM T64213 CH0QA6 155526974 IC50 = 240 nM T64213 CT18PY 155527522 IC50 = 0.85 nM T64213 C6IUQ5 155527836 IC50 = 1.9 nM T64213 C1BL2M 155529532 IC50 = 1900 nM T64213 C4FC0I 155529667 IC50 = 310 nM T64213 C9IGK8 155529802 IC50 = 81 nM T64213 CE09AV 155530174 IC50 = 3600 nM T64213 C7CB1N 155530853 IC50 = 3.3 nM T64213 C8QC3R 155530856 IC50 = 32 nM T64213 CF56BN 155531068 EC50 = 12200 nM T64213 CHM17E 155531143 EC50 = 663 nM T64213 C7XU4P 155532190 IC50 = 3800 nM T64213 C5J8SU 155532311 IC50 = 20 nM T64213 C70HOZ 155532522 IC50 = 99 nM T64213 C4X1GY 155532905 IC50 = 25 nM T64213 C72WUI 155533369 IC50 = 1585 nM T64213 C0BH7X 155534103 IC50 = 880 nM T64213 C65PYC 155535183 IC50 > 25000 nM T64213 C36TSC 155536738 IC50 = 40 nM T64213 CP2UV1 155536845 EC50 = 200 nM T64213 C8EQ5U 155538902 IC50 = 45900 nM T64213 CVDF60 155539376 IC50 = 2.5 nM T64213 CBS40J 155540061 EC50 = 910 nM T64213 CW2V3F 155540455 IC50 = 3.5 nM T64213 CH69QA 155541913 IC50 = 22 nM T64213 CAD76Y 155542105 IC50 = 78 nM T64213 CU7I5K 155543594 IC50 = 5200 nM T64213 CPA6K3 155544013 IC50 = 30 nM T64213 CZAM13 155546455 IC50 = 15 nM T64213 C8V5ZC 155546887 IC50 = 730 nM T64213 C7VT8U 155547220 IC50 = 50 nM T64213 C6NTP5 155547945 IC50 = 63 nM T64213 C3W4YN 155548551 IC50 = 1.5 nM T64213 C5MFS0 155549146 IC50 = 11 nM T64213 CJCO06 155550779 IC50 = 820 nM T64213 CU62IK 155551656 EC50 = 670 nM T64213 CJ4FZ7 155554984 IC50 = 51 nM T64213 C8YN0J 155555089 IC50 = 830 nM T64213 CP4KU2 155555477 IC50 = 1800 nM T64213 CGM04A 155555681 IC50 = 144 nM T64213 C2YO0Z 155556366 EC50 > 30000 nM T64213 CWQ6L8 155558548 EC50 = 280 nM T64213 C2N0DM 155562973 IC50 = 310 nM T64213 C74QRJ 155563663 IC50 = 11 nM T64213 CN6ZL9 155564707 IC50 = 1.2 nM T64213 CB6G1D 155565343 IC50 = 84 nM T64213 CVRC68 155566379 EC50 = 2060 nM T64213 C2GP3W 155567128 IC50 = 86 nM T64213 CQ1PK4 155567723 IC50 = 120 nM T64213 CU7ZA1 155568064 IC50 = 96 nM T64213 CU1QT3 155568605 EC50 = 1180 nM T64213 D03HJW 23630211 EC50 = 49 nM T64213 D03LVL 53464483 IC50 = 40 nM T64213 D03OLU 3601086 IC50 = 2300 nM T64213 D0A1UL 49783953 IC50 > 10000 nM T64213 D0B1QM 2742550 IC50 = 29 nM T64213 D0D6MC 1150897 IC50 > 10000 nM T88531 CZN6S9 743974 EC50 > 50118.72 nM T88531 CW2C5H 3007855 EC50 = 3.6 nM T88531 CS6N0M 3395869 EC50 = 81 nM T88531 CR6C3X 3722317 EC50 = 200 nM T88531 CA8G7X 5407221 EC50 = 1100 nM T88531 C4G1TP 9586016 EC50 = 750 nM T88531 CV03NI 76313672 EC50 = 190 nM T88531 C9WES7 76317176 EC50 = 3100 nM T88531 CTQ0J8 76331797 EC50 = 310 nM T88531 C0V5EC 91826086 EC50 = 0.06 nM T88531 CV4CY0 118716400 EC50 = 202 nM T88531 C1B0TF 118716401 EC50 = 11 nM T88531 CW8AH5 118716402 EC50 = 164 nM T88531 C94MPI 118716403 EC50 = 5000 nM T88531 CV8ZA2 118716404 EC50 = 2204 nM T88531 CDP1U2 118716405 EC50 = 600 nM T88531 CZM50U 118716406 EC50 = 22000 nM T88531 C28OWZ 118716407 EC50 > 25000 nM T88531 C4O2IK 118716408 EC50 = 73 nM T88531 CZE4D9 118716409 EC50 = 11 nM T88531 CVX96A 118716410 EC50 = 15 nM T88531 C0T9RJ 118716411 EC50 = 87 nM T88531 CVT81A 118716412 EC50 = 1181 nM T88531 CW45UK 118716413 EC50 = 60 nM T88531 C5LB7A 118716414 EC50 = 25 nM T88531 CKJS72 118716415 EC50 = 13 nM T88531 C4TEZ0 118716416 EC50 = 36 nM T88531 CD02BX 118716417 EC50 = 0.18 nM T88531 C7TYG0 118716418 EC50 = 0.55 nM T88531 C5OHS8 118716419 EC50 = 30 nM T88531 C2JH5T 118716420 EC50 = 0.35 nM T88531 CD7E4C 135411687 EC50 = 240 nM T88531 CSP2W4 135634901 EC50 = 9 nM T88531 CJG4B1 135634945 EC50 = 18 nM T88531 C1APT5 135634948 EC50 = 460 nM T88531 C4U8WO 135893117 EC50 > 10000 nM T88531 CY17RE 137631764 EC50 = 4 nM T88531 C3V4NZ 137633165 EC50 = 3000 nM T88531 C9ZLJ0 137633277 EC50 = 10 nM T88531 C9P1BR 137635316 EC50 = 4 nM T88531 C4UC1Z 137636773 EC50 = 4 nM T88531 CW57DU 137636882 EC50 = 3 nM T88531 CB87SI 137637255 EC50 = 6 nM T88531 CPM64D 137638361 EC50 = 3 nM T88531 CQM3N5 137639471 EC50 = 1 nM T88531 C3D6TJ 137641632 EC50 = 340 nM T88531 CP15JM 137642799 EC50 = 32 nM T88531 C3LHM1 137643474 EC50 = 2 nM T88531 CJ6ZG0 137644264 EC50 = 5 nM T88531 C9B5HG 137644326 EC50 = 10 nM T88531 C7QE2R 137644868 EC50 = 8 nM T88531 CI5B1O 137645445 EC50 = 4 nM T88531 CUYQ58 137646005 EC50 = 4 nM T88531 C5HT9J 137647882 EC50 = 5 nM T88531 C1X6WC 137648191 EC50 = 2 nM T88531 CA5EG0 137648315 EC50 = 5 nM T88531 CNXI18 137649835 EC50 = 16 nM T88531 CUK3N6 137650161 EC50 = 7 nM T88531 C2CNJ7 137654391 EC50 = 4 nM T88531 CJM8Y0 137656189 EC50 = 16 nM T88531 CQ7MO9 137657224 EC50 = 2 nM T88531 C83CYS 137657821 EC50 = 5 nM T88531 C6JL1V 137658295 EC50 = 8 nM T88531 CI5KZ6 137658694 EC50 = 3 nM T88531 CNXE98 137660912 EC50 = 3 nM T88531 CF1DS8 137661197 EC50 = 1.5 nM T88531 CWQ13R 137661496 EC50 = 18 nM T88531 CX1EB4 137662043 EC50 = 3 nM T88531 D0H4UN 73211886 EC50 = 56 nM T88531 D0V6KN 86277841 EC50 = 0.8 nM T73725 D09JEJ 24748573 IC50 = 3.8 nM T73725 D0E3TC 44259 IC50 = 5.52 nM T73725 D03BNU 59604787 IC50 > 10000 nM T73725 D05BVP 3232621 IC50 = 1902 nM T73725 D09CDR 77105816 IC50 = 80 nM T73725 D0CC7E 77105818 IC50 = 150 nM T73725 D0JQ0Z 46916176 IC50 = 584 nM T73725 D0PO8N 117881270 IC50 = 15 nM T73725 CU80LI 3233012 IC50 = 692 nM T73725 CW4C3P 3235048 IC50 > 10000 nM T73725 CGAT36 5327151 IC50 = 498 nM T73725 CR3BS0 12248905 IC50 = 1100 nM T73725 C5VPH9 16129448 IC50 = 211 nM T73725 C7YG1N 24759534 IC50 < 10 nM T73725 CGLQ20 44223952 IC50 = 1327 nM T73725 CR6VH2 44223953 IC50 = 2163 nM T73725 C2IBW0 44223954 IC50 = 2219 nM T73725 CS3Q2Y 44223955 IC50 = 1810 nM T73725 C5M1UN 44223957 IC50 = 3118 nM T73725 CK8G1T 44223965 IC50 = 801 nM T73725 CJ8KD4 44223966 IC50 = 651 nM T73725 CCW0V4 44223967 IC50 = 3594 nM T73725 CF78WD 44223968 IC50 > 10000 nM T73725 CNE30X 44223970 IC50 = 186 nM T73725 CYR45S 44223971 IC50 = 589 nM T73725 CLZ62P 44223973 IC50 = 173 nM T73725 CIXB09 44223974 IC50 = 2725 nM T73725 C2OBX8 44223977 IC50 = 877 nM T73725 C3VRO9 44557921 IC50 > 10000 nM T73725 C3JBN1 44968184 IC50 = 962 nM T73725 CYW79D 44968186 IC50 = 447 nM T73725 C5OYK3 44968199 IC50 = 8510 nM T73725 C2T0EM 44968221 IC50 = 6181 nM T73725 C8NA2J 44968224 IC50 = 1209 nM T73725 CR8DC5 44968225 IC50 = 3331 nM T73725 CV19YK 44968230 IC50 = 889 nM T73725 CD4ZN1 44968231 IC50 = 1648 nM T73725 C16QFN 46172966 IC50 > 10000 nM T73725 CB32ET 46172972 IC50 > 10000 nM T73725 CN26HW 46172980 IC50 = 409 nM T73725 CGH05O 46172984 IC50 = 1092 nM T73725 CLS29B 46872626 IC50 > 10000 nM T73725 C15EJK 46916169 IC50 = 1361 nM T73725 CHG8C4 46916170 IC50 = 414 nM T73725 CI56BA 46916172 IC50 = 195 nM T73725 CZ5DJ4 46916177 IC50 = 301 nM T73725 CXK37B 46916178 IC50 = 1055 nM T73725 CL1GW0 46916179 IC50 = 486 nM T73725 CZ6DK4 46916182 IC50 = 882 nM T73725 CCUG10 46926515 IC50 = 345 nM T73725 C9NC6W 46926516 IC50 = 52 nM T73725 CZ1D2A 46926518 IC50 = 60 nM T73725 C7S6HT 46926519 IC50 = 39 nM T73725 CG1K5A 46926520 IC50 = 1557 nM T73725 CVF48X 46926521 IC50 = 259 nM T73725 C4ULH5 46926522 IC50 = 41 nM T73725 CPE98Z 46926523 IC50 = 20 nM T73725 C6WLX1 46926524 IC50 = 8791 nM T73725 C61LUI 46926526 IC50 > 10000 nM T73725 C0IVD1 46926527 IC50 = 30 nM T73725 CAYI59 49795862 IC50 = 429 nM T73725 C1UQN4 49795863 IC50 = 238 nM T73725 CU8OC0 49795864 IC50 = 1903 nM T73725 C7T5HW 49795865 IC50 = 462 nM T73725 C6N8EY 49795866 IC50 = 190 nM T73725 C7XS1Z 49795867 IC50 = 665 nM T73725 C5EWG8 49855158 IC50 = 4600 nM T73725 CS6N8Z 54581884 IC50 = 8480 nM T73725 CT6XL0 57466811 IC50 = 117 nM T73725 CXJ63M 59603829 IC50 < 10 nM T73725 CQEU96 59603842 IC50 = 14 nM T73725 CW9AE7 60034150 IC50 = 190 nM T73725 C37NKO 67129970 IC50 = 6440 nM T73725 CK80LJ 67130050 IC50 > 10000 nM T73725 CV63UL 67240318 IC50 > 10000 nM T73725 C7GRV2 68755406 IC50 > 10000 nM T73725 C5DGR9 69036886 IC50 = 1012 nM T73725 C21JAS 76853169 IC50 = 1600 nM T73725 CU04XY 77105624 IC50 = 2300 nM T73725 CTIA65 77105820 IC50 = 2800 nM T73725 CKB1P9 77106023 IC50 = 44 nM T73725 CXYW85 77106025 IC50 = 610 nM T73725 C2UDS0 77106026 IC50 = 4000 nM T73725 C97SJD 77106027 IC50 = 3500 nM T73725 CFQ10R 77106028 IC50 = 110 nM T73725 CO14DP 77106030 IC50 = 1100 nM T73725 C9G3PA 77106234 IC50 = 3500 nM T73725 CPD27I 77106235 IC50 = 610 nM T73725 CLOR37 77106236 IC50 = 4600 nM T73725 C2GLD8 77106237 IC50 = 400 nM T73725 C0GYK1 86765296 IC50 = 680 nM T73725 C1HW4B 89735655 IC50 = 110 nM T73725 C2LWZ1 129318964 IC50 = 31 nM T73725 C4Z5MQ 131839619 IC50 = 5 nM T73725 C4QM9O 134397095 IC50 = 34 nM T73725 CQ1K2W 134397387 IC50 = 6 nM T73725 CR08AO 134397388 IC50 = 7 nM T73725 CIN73J 134397390 IC50 = 14 nM T73725 C6I1YX 134397391 IC50 = 163 nM T73725 CQ9D1Z 134397392 IC50 = 17 nM T73725 CUX8N5 134397449 IC50 = 26 nM T73725 CDC39N 134397450 IC50 = 120 nM T73725 C8RN6W 134397451 IC50 = 16 nM T73725 CE1HY2 134397452 IC50 = 26 nM T73725 CIR51J 134397453 IC50 = 11 nM T73725 C72KFM 134397463 IC50 = 28 nM T73725 CT16YX 134397502 IC50 = 26 nM T73725 CI45HZ 134397798 IC50 = 92 nM T73725 CI1E8V 137634241 IC50 > 10000 nM T73725 CDA2N6 137644922 IC50 = 5.3 nM T73725 CZ9BN4 138320062 IC50 = 0.261 nM T73725 C5J2WV 138728749 IC50 = 39 nM T73725 CVU63L 139582016 IC50 = 360 nM T73725 C8PH9S 139582017 IC50 = 1400 nM T73725 C6VB3O 145925651 IC50 >= 5000 nM T73725 CX05ZN 145979845 IC50 = 175 nM T73725 CO1S8D 145986658 IC50 = 910 nM T73725 C2MD1Q 155513187 IC50 > 10000 nM T73725 D00ERW 44444843 Ki > 8753 nM T73725 D06CXU 46926513 IC50 = 23 nM T73725 D0D2FC 2794188 IC50 = 111 nM T73725 D0U3NI 53246941 IC50 = 112 nM T73725 D0UI7U 46926514 IC50 = 231 nM T49526 D00BUR 216327 IC50 > 1000 nM T49526 D02AIN 122678117 IC50 > 33000 nM T49526 D0HZ2E 5311271 Ki = 1060 nM T49526 D0K9IF 71666749 IC50 > 30000 nM T49526 C2KDX3 2464255 EC50 = 1470 nM T49526 CKR9Z3 2464257 EC50 > 30000 nM T49526 CRQ37A 4880560 EC50 = 1690 nM T49526 C8T6YH 8762554 EC50 > 30000 nM T49526 CZM2H8 8881840 EC50 > 30000 nM T49526 CS6FN7 9883254 IC50 = 2600 nM T49526 CD34SB 15982534 IC50 = 35000 nM T49526 CU61HC 16827304 EC50 = 2860 nM T49526 CG26CZ 16862803 EC50 > 30000 nM T49526 C7S9NE 25923464 EC50 > 30000 nM T49526 CI1G2C 26873419 IC50 = 2920 nM T49526 C9L4KT 46205341 IC50 > 333000 nM T49526 CL41FE 46206000 IC50 > 333000 nM T49526 CBM42K 53347890 EC50 = 1160 nM T49526 C3YO2J 53347892 EC50 > 30000 nM T49526 C8ZU0D 53347894 EC50 = 1000 nM T49526 C3O7HM 53347896 EC50 = 1410 nM T49526 C94DCG 53347898 EC50 = 7970 nM T49526 CJ9N3F 53347900 EC50 = 1360 nM T49526 CGU48Z 53347904 EC50 = 4740 nM T49526 CZF4S8 53347906 EC50 = 1710 nM T49526 C09ZWT 53347908 EC50 > 30000 nM T49526 C96ZSQ 53347910 EC50 > 30000 nM T49526 C83WFR 53347912 EC50 > 30000 nM T49526 CTOU65 53347914 EC50 > 30000 nM T49526 C7VX8I 53347916 EC50 = 1030 nM T49526 CZY27H 53347918 EC50 = 420 nM T49526 CW9G6X 53347920 EC50 = 6130 nM T49526 CV73XM 53347922 EC50 = 8160 nM T49526 CC45FS 53347924 EC50 = 1780 nM T49526 CC4J5Y 53347926 EC50 = 1380 nM T49526 C9OR6S 53347928 EC50 > 30000 nM T49526 CBZ0Y3 53347930 EC50 = 810 nM T49526 CU90QI 53347932 EC50 = 880 nM T49526 CP1YA3 53488269 EC50 > 30000 nM T49526 C9TM8Q 53488271 EC50 > 30000 nM T49526 CXG6U4 53488272 EC50 > 30000 nM T49526 CZYL42 53488273 EC50 > 30000 nM T49526 CB0RG1 53488275 EC50 = 890 nM T49526 C8APK2 53488280 EC50 = 1630 nM T49526 C4XKH1 53488282 EC50 > 30000 nM T49526 C9BG8K 53488283 EC50 > 30000 nM T49526 CTDY79 53488284 EC50 = 780 nM T49526 CT6UK4 54765372 EC50 = 4380 nM T49526 CXD82U 54765373 EC50 > 30000 nM T49526 CZD5L7 54765374 EC50 > 30000 nM T49526 C72OFG 54765375 EC50 > 30000 nM T49526 C1JMD5 54765376 EC50 = 12900 nM T49526 CU6IC4 54765377 EC50 = 600 nM T49526 C6C5QV 54765378 EC50 > 30000 nM T49526 CA1I6V 54765379 EC50 > 30000 nM T49526 CK8X1W 54765381 EC50 > 30000 nM T49526 CDK50N 54765382 EC50 = 730 nM T49526 C6QKF9 54765445 EC50 > 30000 nM T49526 CAW2J3 54765446 EC50 = 700 nM T49526 C9VH8O 54765447 EC50 = 2590 nM T49526 CYBF21 54765449 EC50 > 30000 nM T49526 C9B2HV 54765450 EC50 > 30000 nM T49526 CKXT78 54765451 EC50 > 30000 nM T49526 C97QTU 54765453 EC50 > 30000 nM T49526 C36HEY 56947221 EC50 = 27400 nM T49526 C2XWQ6 56947223 EC50 = 1320 nM T49526 CLT4Z1 56947228 EC50 > 30000 nM T49526 C5LUY8 56947229 EC50 > 30000 nM T49526 CPR1W3 56947230 EC50 > 30000 nM T49526 CJA45K 56947232 EC50 > 30000 nM T49526 C2POB1 56947233 EC50 > 30000 nM T49526 C1YK2E 122678192 IC50 > 33000 nM T49526 CJH2V9 137637559 IC50 = 2640 nM T49526 C2KX3V 137661020 IC50 > 3000 nM T49526 CKZT21 155559364 IC50 > 33000 nM T49526 D08ATZ 51351551 EC50 = 49290 nM T49526 D0W2FU 53347902 EC50 = 260 nM T12837 CWU8N7 67338 IC50 = 3000 nM T12837 C0O3TQ 126437 IC50 > 400000 nM T12837 C5N0PM 295976 IC50 = 3100 nM T12837 CWF94O 428849 IC50 = 890 nM T12837 CJ2CX8 582689 IC50 > 65000 nM T12837 CQEF34 1002773 IC50 > 100000 nM T12837 C8G4OE 1192043 IC50 > 100000 nM T12837 CV6LA5 2297580 IC50 = 16600 nM T12837 C89ATQ 2779831 IC50 = 1000 nM T12837 CN0F5E 3014812 IC50 = 7500 nM T12837 C8TOU9 3496505 IC50 > 20000 nM T12837 CH9K1U 5351747 IC50 = 400000 nM T12837 CNK84Q 7128991 IC50 = 105000 nM T12837 CEKH37 10979651 IC50 > 400000 nM T12837 CJ6E7G 11087601 IC50 = 20500 nM T12837 C1ZR6H 11848210 IC50 = 1.2 nM T12837 C4QAH6 15342414 IC50 = 1637 nM T12837 C0M7WQ 22390870 IC50 = 98 nM T12837 CJQ86Y 24827559 IC50 = 8600 nM T12837 CJ4IC6 24962989 IC50 = 80 nM T12837 CA7K9P 43167849 IC50 = 1220 nM T12837 CCLQ46 43187900 IC50 = 5310 nM T12837 C0Y9FH 43199381 IC50 = 200 nM T12837 C7F4DG 44574239 IC50 = 60 nM T12837 CPS2T8 44574240 IC50 = 210 nM T12837 C18PTZ 44574241 IC50 = 310 nM T12837 C4V6OX 44574242 IC50 = 1540 nM T12837 CYZ4G1 44574264 IC50 = 50 nM T12837 CJG7H1 44574265 IC50 = 160 nM T12837 C9KMX6 44574266 IC50 = 50 nM T12837 C9WB3L 44574306 IC50 = 50 nM T12837 CL24UR 44574307 IC50 = 130 nM T12837 C6NE3R 44574308 IC50 = 2200 nM T12837 CQI27O 44574309 IC50 = 400 nM T12837 CJ6L4K 44574374 IC50 = 360 nM T12837 C1RIT4 44574375 IC50 = 2100 nM T12837 C98OJN 44574376 IC50 > 10000 nM T12837 CHI9F3 44574377 IC50 > 10000 nM T12837 C12DMU 44578429 IC50 = 10600 nM T12837 C5GCR8 44578430 IC50 = 29800 nM T12837 C04YVX 44578431 IC50 = 7700 nM T12837 C0WB8T 44578432 IC50 = 230 nM T12837 C8AIP0 44578462 IC50 = 1420 nM T12837 C5N3CJ 44578463 IC50 = 16900 nM T12837 CX4YR8 44578464 IC50 = 160 nM T12837 C3P2UH 44578465 IC50 = 20100 nM T12837 CI0NP8 44578466 IC50 > 30000 nM T12837 CNU74O 44578467 IC50 > 30000 nM T12837 C7ZQW8 44578468 IC50 > 30000 nM T12837 CRSC45 44578469 IC50 = 1320 nM T12837 CI2O0T 44578470 IC50 = 3400 nM T12837 CX95VH 44578502 IC50 = 7100 nM T12837 C92YUQ 44578503 IC50 = 180 nM T12837 CQO7X6 44578504 IC50 = 1100 nM T12837 CZ1F4S 44578505 IC50 = 4300 nM T12837 CZE1J7 44578539 IC50 = 1800 nM T12837 C8GZB2 44578540 IC50 > 50000 nM T12837 CJTR68 44578541 IC50 > 50000 nM T12837 CMQ5N2 44578542 IC50 = 600 nM T12837 CQA74O 45487305 IC50 > 30 nM T12837 CJZ41I 45487306 IC50 > 30 nM T12837 CABH45 45487323 IC50 = 0.12 nM T12837 CD4OH6 45487347 IC50 = 0.26 nM T12837 CEA04X 45487348 IC50 = 2.9 nM T12837 CLP03M 45487354 IC50 = 0.7 nM T12837 CYJ42A 45487360 IC50 = 0.84 nM T12837 CXD72H 45487361 IC50 = 0.41 nM T12837 CD36FG 45487378 IC50 = 17 nM T12837 CA9GE3 45487379 IC50 = 4.6 nM T12837 CWHP79 46867603 IC50 = 30 nM T12837 C70ZYQ 46997620 IC50 = 11100 nM T12837 CUA83Y 50937454 IC50 = 27 nM T12837 CN01BZ 53211571 IC50 > 4700 nM T12837 CKAI31 53361222 IC50 = 8100 nM T12837 CV25JZ 53361223 IC50 = 14400 nM T12837 C0C6YK 53363652 IC50 = 10300 nM T12837 CPU86Z 53363653 IC50 = 15200 nM T12837 C63DVR 53363743 IC50 = 11900 nM T12837 COBL07 53363744 IC50 = 12500 nM T12837 C8QFS7 53363745 IC50 = 12200 nM T12837 CEG3P9 53363834 IC50 = 14800 nM T12837 CW4CD0 53363835 IC50 = 16000 nM T12837 C02ORV 53377508 Ki > 20000 nM T12837 CYM2T4 53868701 IC50 = 32 nM T12837 CPL71I 54596764 IC50 = 116000 nM T12837 C0YR1M 55070650 IC50 > 10000 nM T12837 C72GHW 56642706 IC50 > 100000 nM T12837 CS6Q7R 56642708 IC50 > 100000 nM T12837 CC2O7Y 56746673 IC50 = 13300 nM T12837 C3FUP7 56753262 IC50 = 1900 nM T12837 C7VQ5F 56759179 IC50 > 30000 nM T12837 CN7V5L 56759225 IC50 > 40000 nM T12837 CRI9T6 56759592 IC50 = 600 nM T12837 CJBY70 56951879 Ki > 50000 nM T12837 CD6V9F 58730746 IC50 = 6250 nM T12837 C04KFR 60150359 IC50 = 3000 nM T12837 CQ60CT 62206064 IC50 = 2460 nM T12837 C7RJD3 63155127 IC50 = 3190 nM T12837 CNR16Q 63189585 IC50 > 10000 nM T12837 CQ27KW 64381918 IC50 = 8340 nM T12837 CER5F1 67466175 IC50 > 100000 nM T12837 CO6L5Z 67739618 IC50 = 80 nM T12837 C5QE6A 67988955 IC50 > 50000 nM T12837 C8JTS3 70676140 Ki > 100000 nM T12837 CZL47S 70676141 Ki > 100000 nM T12837 C8KC6O 70676142 Ki > 100000 nM T12837 CAFU69 70686225 IC50 = 100000 nM T12837 CM53OA 72918546 IC50 > 50000 nM T12837 CUP4Q6 76328021 Ki > 50000 nM T12837 CX7V5M 76328022 Ki > 50000 nM T12837 C5P2BM 76331683 Ki > 50000 nM T12837 C8KEM3 91645136 IC50 = 360 nM T12837 C73LWN 92136227 IC50 = 4 nM T12837 CWG18C 118731739 IC50 = 7230 nM T12837 CI1AE0 118731742 IC50 = 5800 nM T12837 C6Y8BM 118731746 IC50 = 21500 nM T12837 CIOL82 122195095 IC50 = 10000 nM T12837 C6KV9H 124081151 IC50 = 50 nM T12837 CP94YL 127031964 IC50 = 27 nM T12837 C9KJ2Q 134130626 IC50 = 149 nM T12837 CV95CT 134131930 IC50 = 3680 nM T12837 CIV51H 134132630 IC50 = 177 nM T12837 C3W8IS 134132824 IC50 = 16 nM T12837 CJ8H7W 134134884 IC50 = 14 nM T12837 CFVI01 134135475 IC50 = 1540 nM T12837 CIY91H 134135786 IC50 = 85 nM T12837 CBJ1S8 134137030 IC50 = 108 nM T12837 CT5I6V 134137361 IC50 = 62 nM T12837 C13UJH 134137680 IC50 = 28 nM T12837 C0C4AO 134138246 IC50 = 53 nM T12837 C4AFS3 134140748 IC50 = 35 nM T12837 CF57RU 134140884 IC50 = 120 nM T12837 CP59XG 134141266 IC50 = 19 nM T12837 C38BUI 134141657 IC50 = 616 nM T12837 CG8PM2 134142051 IC50 = 23 nM T12837 CKGL61 134142579 IC50 = 33 nM T12837 CPS6D3 134144201 IC50 = 18 nM T12837 C2GC5B 134144476 IC50 = 41 nM T12837 C67DQZ 134144962 IC50 = 15 nM T12837 CSY51N 134146326 IC50 = 18 nM T12837 CRY2Z5 134146985 IC50 = 41 nM T12837 C8L6ZH 134148531 IC50 = 15 nM T12837 CEAV71 134149335 IC50 = 42 nM T12837 C5U6TX 134151277 IC50 = 103 nM T12837 C0PIN9 134153830 IC50 = 1070 nM T12837 CMHQ35 134153978 IC50 = 27 nM T12837 C8UX3L 134154872 IC50 = 231 nM T12837 C2OR9A 134155520 IC50 = 17 nM T12837 C54FUD 134155964 IC50 = 28 nM T12837 CXM26R 134156697 IC50 = 22 nM T12837 CF3GA7 134157655 IC50 = 17 nM T12837 CDXJ59 136180348 IC50 = 2600 nM T12837 C93QGH 137633458 IC50 = 69 nM T12837 C4LK1X 137635057 IC50 = 94 nM T12837 C1PMC9 137636992 IC50 = 94 nM T12837 CJ4Q8Z 137638223 IC50 = 223 nM T12837 C13YKS 137638371 IC50 = 130 nM T12837 C8FZG6 137642809 IC50 = 90 nM T12837 C16DLH 137647272 IC50 = 302 nM T12837 C51RHP 137647665 IC50 = 67 nM T12837 C1O5PE 137652170 IC50 = 342 nM T12837 CCO6Z7 137654377 IC50 = 330 nM T12837 CRT8Q3 137655207 IC50 = 63 nM T12837 CK7BA8 137656269 IC50 = 157 nM T12837 C9Z6GL 137659934 IC50 = 144 nM T12837 CB9FM8 137661596 IC50 = 50 nM T12837 CDPN65 137661881 IC50 = 471 nM T12837 CR5D4S 138753329 IC50 = 480 nM T12837 C51ILK 138753330 IC50 = 2000 nM T12837 CE58DF 153041236 IC50 > 100000 nM T12837 CC50SM 155511980 IC50 = 130 nM T12837 CTM72I 155513465 IC50 = 240 nM T12837 C78OZR 155516239 IC50 = 4260 nM T12837 CJQH26 155516447 IC50 = 465 nM T12837 CU04SF 155519144 IC50 = 279 nM T12837 CH5J9U 155520755 IC50 = 6120 nM T12837 C6CY0R 155523571 IC50 = 120 nM T12837 C2LRU6 155523638 IC50 = 1990 nM T12837 C4JEC2 155526486 IC50 = 220 nM T12837 CKNF47 155527838 IC50 = 2310 nM T12837 CTHM63 155528468 IC50 = 11600 nM T12837 C5BUY9 155529011 IC50 = 101 nM T12837 C7C8HI 155529624 IC50 = 21 nM T12837 CBU23P 155531094 IC50 = 2070 nM T12837 C7U9IT 155534335 IC50 = 410 nM T12837 CYMG91 155534360 IC50 = 270 nM T12837 CY8O0Q 155535049 IC50 = 475 nM T12837 CZRU49 155535884 IC50 = 1700 nM T12837 C70HAX 155536607 IC50 = 4480 nM T12837 C0RY3I 155538329 IC50 = 2310 nM T12837 C67JQV 155538900 IC50 > 200000 nM T12837 CO03YQ 155541365 IC50 = 270 nM T12837 CY2W3F 155541904 IC50 = 600 nM T12837 C8LZ6X 155542642 IC50 = 1950 nM T12837 C4UT5G 155542694 IC50 = 785 nM T12837 CYO70M 155543486 IC50 = 3820 nM T12837 CNLE45 155543945 IC50 = 1180 nM T12837 CPXC10 155546110 IC50 = 305 nM T12837 C08EQC 155546573 IC50 = 43 nM T12837 CQ9A0Z 155547391 IC50 = 3490 nM T12837 CHB87K 155547731 IC50 = 658 nM T12837 CKUV39 155549017 IC50 = 37 nM T12837 CM4C9U 155549658 IC50 = 343 nM T12837 C79QNS 155549883 IC50 = 254 nM T12837 CJ8ZI6 155549992 IC50 = 51000 nM T12837 CHPG47 155551515 IC50 = 2050 nM T12837 CVN57A 155552644 IC50 = 5220 nM T12837 C3Q7YP 155558960 IC50 = 900 nM T12837 C3PMG9 155559000 IC50 = 31 nM T12837 CEI8R4 155559940 IC50 = 7980 nM T12837 CU06YI 155562437 IC50 = 165 nM T12837 C8LKQ6 155564730 IC50 = 2610 nM T12837 C81NJP 155565393 IC50 = 772 nM T12837 CTCM91 155566361 IC50 = 530 nM T12837 CF4ZI2 155567058 IC50 = 228 nM T12837 CW56PR 155567067 IC50 = 2130 nM T12837 CVJ62X 155568483 IC50 = 2110 nM T12837 C47PWI 46905055 IC50 > 50000 nM T12837 D02TVQ 71268957 IC50 = 128000 nM T12837 D09CLP 439155 Ki = 400 nM T12837 D0A1CM 5281855 IC50 = 25000 nM T12837 D0BU8W 44219611 IC50 = 0.04 nM T12837 D0Q3FY 44622850 IC50 = 0.07 nM T72458 D0G2XE 6918468 IC50 = 400 nM T72458 D0H7AR 70684954 Ki = 26000 nM T72458 D0LI1C 44469321 IC50 > 30000 nM T72458 D0X9PF 9941379 EC50 = 0.2 nM T72458 CA3ZU6 489667 IC50 = 612 nM T72458 CZN6S9 743974 EC50 > 31622.78 nM T72458 CL04VQ 910537 Ki > 1000000 nM T72458 C0DA9X 2163781 Ki = 161000 nM T72458 CK4YT2 2817655 Ki > 1000000 nM T72458 CB9A2M 2852098 Ki = 118000 nM T72458 C8EPT1 6918707 EC50 = 4 nM T72458 CWZ1O2 6918780 EC50 = 0.44 nM T72458 CY60AZ 6918813 EC50 = 6 nM T72458 C2BQE1 6918814 Ki = 1.8 nM T72458 CK83QR 6918844 Ki = 3.2 nM T72458 C14CGB 6918847 Ki = 6.3 nM T72458 CLV3C7 6918849 IC50 = 0.77 nM T72458 C5U7CS 6918850 Ki = 2.8 nM T72458 C0Q5JL 6918851 IC50 = 8 nM T72458 CRG04O 6918857 Ki = 20 nM T72458 COS6C1 9808720 EC50 = 11 nM T72458 CM02VS 9808801 EC50 = 13 nM T72458 C8IM6O 9851816 Ki = 12.9 nM T72458 CVM3K1 9852314 Ki = 600 nM T72458 CKCF18 9867330 EC50 = 16 nM T72458 CM3Y5H 9893728 IC50 = 9157 nM T72458 CZ5E2C 9915636 Ki = 20.5 nM T72458 CCL2T8 9915813 EC50 = 2600 nM T72458 CFG0W2 9917301 IC50 = 118 nM T72458 CNF37L 9919056 EC50 = 2 nM T72458 C15DES 9924916 Ki = 140000 nM T72458 C7V8AE 9946241 Ki = 42000 nM T72458 CX5CU3 9958649 Ki = 590 nM T72458 C97MRJ 9960253 EC50 = 16 nM T72458 CMU31X 9968756 Ki = 27000 nM T72458 C5F3QU 9969456 Ki = 6400 nM T72458 C5U0JO 9977350 Ki = 180 nM T72458 CG58RO 9983075 Ki = 190 nM T72458 CR6TX4 10004020 IC50 = 52 nM T72458 CC48YG 10008561 EC50 = 6700 nM T72458 CLXA58 10025669 Ki = 25118.86 nM T72458 CRP4X1 10030530 Ki = 6 nM T72458 CL2PE9 10031074 Ki = 2500 nM T72458 C8KI2R 10033237 Ki = 160 nM T72458 CGJ72R 10049407 Ki = 770 nM T72458 C9YQS5 10050686 Ki = 89 nM T72458 CMGB68 10053261 Ki = 6300 nM T72458 CAG52F 10072440 Ki = 920 nM T72458 CSH3Y2 10075878 IC50 = 530 nM T72458 CZ78WX 10077258 EC50 = 13 nM T72458 C7T2XW 10077483 Ki = 4100 nM T72458 CUR4Y1 10077594 Ki = 57 nM T72458 C8MCA1 10077773 Ki = 1.95 nM T72458 C7PV4C 10098133 EC50 = 240 nM T72458 CP5H2J 10098568 IC50 = 260 nM T72458 CW4E8K 10101361 EC50 = 2.17 nM T72458 CSQ60B 10108894 Ki = 16000 nM T72458 C6LVA2 10109225 Ki = 5000 nM T72458 C0DP3Z 10117829 IC50 = 871 nM T72458 C8AQP5 10119206 EC50 = 40 nM T72458 CG1K8Y 10122170 EC50 < 0.1 nM T72458 CFX6U7 10123761 EC50 = 33 nM T72458 C6Y3KL 10128451 IC50 = 16 nM T72458 CF81WV 10132207 Ki = 66000 nM T72458 C0PVS9 10134057 Ki = 6200 nM T72458 CC0ZT7 10137615 Ki = 16000 nM T72458 C86FWN 10141778 IC50 = 16 nM T72458 C2AF5L 10146090 IC50 = 12 nM T72458 CO69QN 10146211 EC50 = 0.58 nM T72458 C51LKY 10146483 EC50 = 65 nM T72458 C03AKT 10155513 Ki = 67000 nM T72458 CPRS08 10157774 Ki = 13000 nM T72458 CXF16O 10158674 Ki = 62000 nM T72458 C97IHD 10159196 Ki = 12000 nM T72458 C1XJM3 10165866 IC50 = 12 nM T72458 CX7WV9 10168556 EC50 = 120 nM T72458 CTD14O 10169912 EC50 = 9 nM T72458 CAB06U 10177247 Ki = 161000 nM T72458 COJ1M5 10178845 Ki = 6800 nM T72458 CV2QX0 10180932 Ki = 12000 nM T72458 C78FGS 10188529 IC50 = 28 nM T72458 C1HMR6 10200110 Ki = 111000 nM T72458 CFZ5I6 10210964 IC50 = 1.9 nM T72458 C8PA3J 10211466 Ki = 73.7 nM T72458 C1VCQ8 10213106 EC50 = 13 nM T72458 CWJ5I0 10225762 Ki = 25000 nM T72458 CH67VW 10230144 IC50 = 30 nM T72458 CF8SA2 10232394 IC50 = 11 nM T72458 CTO7I8 10232787 Ki = 7.3 nM T72458 CFH82K 10239507 IC50 = 11.2 nM T72458 C1OYR8 10255546 Ki = 2600 nM T72458 CSNY06 10257242 EC50 = 25 nM T72458 C6Y1ER 10257541 Ki = 1 nM T72458 C2AL7S 10260053 Ki = 630 nM T72458 CEC2M0 10269187 Ki = 74000 nM T72458 C6T2MU 10270570 Ki = 11000 nM T72458 CX29KB 10282847 IC50 = 1.1 nM T72458 C4SCW2 10283036 Ki = 5.8 nM T72458 CBL5E0 10283067 Ki = 6.4 nM T72458 C01QVJ 10291369 Ki = 26000 nM T72458 CSDX25 10291370 Ki = 7400 nM T72458 CX97KY 10292084 Ki = 33000 nM T72458 C7WDA8 10292876 Ki = 7000 nM T72458 CU17RB 10293285 Ki = 16000 nM T72458 CV3ZJ5 10304463 Ki = 95.6 nM T72458 CU13DH 10304547 IC50 = 0.37 nM T72458 C1E3PC 10304776 IC50 = 1.1 nM T72458 CC0N9A 10304794 Ki = 5.3 nM T72458 CU0CH8 10324857 Ki = 4.3 nM T72458 CE4OK9 10325306 Ki = 0.83 nM T72458 CT9AR6 10325955 EC50 = 14 nM T72458 CO40LC 10348630 EC50 = 227 nM T72458 CSH89D 10369375 Ki = 3.2 nM T72458 C84RZU 10373417 EC50 = 2 nM T72458 C1N3MA 10392968 IC50 = 1900 nM T72458 CJN2I7 10411266 Ki = 340 nM T72458 CNK7M3 10414731 Ki = 80 nM T72458 CPL02I 10463896 EC50 = 6.08 nM T72458 C1GJ2S 10481801 IC50 = 152 nM T72458 CS2EQ0 10481883 Ki = 11 nM T72458 CTEB92 10483153 EC50 = 18 nM T72458 C3NWO8 10484741 EC50 = 59 nM T72458 CICJ50 10864263 IC50 = 469 nM T72458 CBPX36 10864861 EC50 = 8.7 nM T72458 C5SK0I 10874535 IC50 = 597 nM T72458 CM5GF3 10886436 IC50 = 3050 nM T72458 CGIC31 10918643 IC50 = 2081 nM T72458 C52NZB 10928744 IC50 = 193 nM T72458 CP6WR3 10951027 IC50 = 266 nM T72458 CN9D6B 10952071 IC50 = 127 nM T72458 COE81Y 10973172 IC50 = 150 nM T72458 CJKA90 10996121 EC50 = 297 nM T72458 CY3TJ1 10996232 EC50 = 32 nM T72458 CQJF15 11016325 IC50 = 3226 nM T72458 CAL9N7 11017471 Ki = 1.2 nM T72458 C7IJV5 11038873 EC50 = 630 nM T72458 CA2X6S 11050211 IC50 = 238 nM T72458 CHOS10 11061068 IC50 = 0.3 nM T72458 CNP78D 11092487 IC50 = 249 nM T72458 C5H7IP 11092574 IC50 = 364 nM T72458 CO2U6S 11156852 EC50 = 274 nM T72458 C4V9OW 11157584 Ki = 14 nM T72458 CF6T8V 11158829 EC50 = 1995.26 nM T72458 C81JOX 11170774 EC50 = 29 nM T72458 CG64NJ 11179914 EC50 = 490 nM T72458 C3V7DK 11180881 Ki = 15 nM T72458 CHC51K 11181804 Ki = 10.8 nM T72458 CDLG18 11205265 EC50 = 1995.26 nM T72458 C9WTR4 11205266 EC50 = 63.1 nM T72458 CDMB38 11205293 EC50 = 794.33 nM T72458 CLJ83I 11205294 EC50 = 1995.26 nM T72458 C0F8CB 11214733 EC50 = 145 nM T72458 CUC85X 11215553 EC50 = 3.2 nM T72458 CD5SG6 11215758 Ki = 4.8 nM T72458 CF7VQ4 11226756 EC50 = 7 nM T72458 CWLJ34 11237444 Ki = 1300 nM T72458 CR1Q2X 11237928 EC50 = 150 nM T72458 C30NWM 11238126 EC50 = 40 nM T72458 C1T3VM 11249545 Ki = 840 nM T72458 CD5YZ2 11249788 EC50 = 44 nM T72458 C6FBD3 11251566 EC50 = 158.49 nM T72458 C6ETW3 11251567 EC50 = 1258.93 nM T72458 C9LOV4 11251591 EC50 = 251.19 nM T72458 CMI4E5 11251592 EC50 = 79.43 nM T72458 CE2P7Y 11261324 EC50 = 210 nM T72458 CF58GC 11262020 EC50 = 140 nM T72458 C0D1PE 11263072 EC50 = 2.512 nM T72458 CMS1L8 11272336 EC50 = 200 nM T72458 CP9S6F 11273288 EC50 = 2 nM T72458 C07VJD 11274575 IC50 = 158.49 nM T72458 CS2U3A 11286048 IC50 = 1995.26 nM T72458 CS57OX 11295536 EC50 = 71 nM T72458 CQ47NA 11295737 EC50 = 110 nM T72458 CJ7OT2 11296600 EC50 = 3.8 nM T72458 C2PU1F 11296732 Ki = 44 nM T72458 CYH1I3 11297620 EC50 < 0.01 nM T72458 C9XBQ7 11308054 Ki = 29 nM T72458 CYK4F0 11308184 Ki = 77 nM T72458 C97ICV 11309021 IC50 = 794.33 nM T72458 CVE6D9 11309022 EC50 = 794.33 nM T72458 CO0C7R 11330869 Ki = 27 nM T72458 CYUL15 11330992 EC50 = 8 nM T72458 CS7K4R 11341045 Ki = 650 nM T72458 CU6Y1Z 11341046 Ki = 1500 nM T72458 C3RI8D 11341811 EC50 = 34 nM T72458 C4OEC6 11353522 EC50 = 93 nM T72458 CHWO84 11353851 EC50 = 400 nM T72458 CAL3F9 11364326 Ki = 580 nM T72458 C41ZBP 11364343 EC50 = 1300 nM T72458 CYVD37 11364802 EC50 = 44 nM T72458 CEX40J 11366515 EC50 = 630.96 nM T72458 CZ6RU2 11375529 EC50 = 360 nM T72458 C5D1TY 11375764 Ki = 840 nM T72458 C6SN4C 11378005 EC50 = 1258.93 nM T72458 CV7BU3 11378006 EC50 = 1995.26 nM T72458 CR8B4G 11378033 EC50 = 316.23 nM T72458 CUPS87 11387898 EC50 = 150 nM T72458 CMF98X 11398483 Ki = 37 nM T72458 CQ1ZL6 11411962 IC50 = 398.11 nM T72458 CQ7WS5 11421919 Ki = 24 nM T72458 CUTZ31 11445925 EC50 = 398.11 nM T72458 C0GFV8 11456260 EC50 = 48 nM T72458 C3FML2 11468019 Ki = 69.5 nM T72458 C2DNI1 11468666 EC50 = 158.49 nM T72458 C8LN5W 11477853 Ki = 1400 nM T72458 CG5D6C 11480040 IC50 = 3981.07 nM T72458 CPT4K8 11490215 EC50 = 98 nM T72458 CVR0T4 11490658 Ki = 6.3 nM T72458 CY8AJ5 11512024 EC50 = 281.84 nM T72458 CKE15O 11555886 EC50 = 17.9 nM T72458 CF7NS4 11571540 EC50 = 1 nM T72458 CA5GQ7 11592389 EC50 = 151.36 nM T72458 CL87NX 11593230 EC50 = 1 nM T72458 C24UQH 11599302 EC50 = 44.67 nM T72458 CDP3W4 11607111 EC50 = 40 nM T72458 CR0N5C 11613526 EC50 = 707.95 nM T72458 C7F9XQ 11613741 EC50 = 354.81 nM T72458 COLB48 11627577 EC50 = 3235.94 nM T72458 CRE2X6 11635051 EC50 = 537.03 nM T72458 C7JU6O 11635265 EC50 = 177.83 nM T72458 CM2A6K 11636019 Ki = 16 nM T72458 CPM61U 11685018 EC50 = 323.59 nM T72458 C3XN4O 11692334 EC50 = 436.52 nM T72458 C6WAM2 11706338 EC50 = 1000 nM T72458 CWZX95 11730771 IC50 = 1500 nM T72458 C6GMS7 11732821 IC50 > 5000 nM T72458 C3NWA7 11733360 IC50 = 336 nM T72458 C5AZ2R 11753667 EC50 = 21 nM T72458 CIHY70 11753668 EC50 = 44 nM T72458 CH7TQ6 11753695 EC50 = 4.6 nM T72458 C63DVB 11756904 Ki = 64 nM T72458 C59XUF 11757528 EC50 = 710 nM T72458 CHI2W5 11761948 IC50 > 10000 nM T72458 CUL54T 11764499 EC50 = 100 nM T72458 C2SHV7 11786860 EC50 = 12 nM T72458 CD9N5B 11787842 EC50 = 501.19 nM T72458 CQ06HS 11787864 EC50 = 316.23 nM T72458 CMJ3K5 11811937 IC50 = 3829 nM T72458 C0OIV9 11813437 EC50 = 840 nM T72458 C7NL4J 11845272 Ki = 10 nM T72458 C4XF1I 11845276 Ki = 137 nM T72458 CT1F9R 11845438 EC50 = 97 nM T72458 CC42HM 11845440 EC50 = 501 nM T72458 CFKN79 11845444 Ki = 2353 nM T72458 C3JV7M 11845450 EC50 = 2.3 nM T72458 C8WJ6E 11845630 EC50 = 252 nM T72458 CI1VU0 11845804 EC50 = 986 nM T72458 C4V9DO 11845813 EC50 = 291 nM T72458 CSZX65 11846669 EC50 = 14 nM T72458 C5HFB2 11846673 Ki = 90 nM T72458 C25KCW 11846844 EC50 = 39 nM T72458 CO3H9V 11847001 EC50 = 9 nM T72458 CECQ63 11847312 EC50 = 292 nM T72458 C91GMR 11851038 EC50 = 1.02 nM T72458 CT4EC3 11966875 IC50 > 10000 nM T72458 CG15NA 15602927 IC50 = 90 nM T72458 C0E4PU 15603023 IC50 = 60 nM T72458 CI9W3G 15953833 IC50 = 1.5 nM T72458 CAT74W 15953838 EC50 = 177 nM T72458 C2BLT4 16007263 EC50 = 1.7 nM T72458 C54MIL 16007264 Ki = 19 nM T72458 C6XS3N 16007285 Ki = 13 nM T72458 CK3T2B 16038121 EC50 = 1113.1 nM T72458 CYW0B8 16038315 Ki = 6.7 nM T72458 CSM3L8 16038316 Ki = 10 nM T72458 C4N0VF 16046215 Ki = 25 nM T72458 CX68DN 16049796 EC50 > 10000 nM T72458 C8UXP9 16126683 EC50 = 29.7 nM T72458 CPTO16 16132144 EC50 = 0.21 nM T72458 C9YZE5 16133802 EC50 = 0.65 nM T72458 CM8QO6 16721030 IC50 = 19.8 nM T72458 CZU6Q0 16725558 EC50 = 214.5 nM T72458 C4NZ3C 16725559 IC50 = 3.3 nM T72458 CR1DM4 16746686 IC50 = 0.84 nM T72458 C7WHL3 16746823 EC50 = 0.11 nM T72458 C25XZF 17880880 Ki > 1000000 nM T72458 CW58XN 22318631 IC50 = 131 nM T72458 C8BY2K 22318635 IC50 = 40.3 nM T72458 CCQ0V9 22318636 IC50 = 22 nM T72458 CG5SO7 22318639 IC50 = 72.3 nM T72458 C8BFU5 22318643 IC50 = 3590 nM T72458 C6MID9 22318657 IC50 = 303 nM T72458 C9QO2V 22318671 IC50 = 263 nM T72458 CZ1GJ8 23634985 Ki = 35 nM T72458 C6UP8O 23634986 Ki = 9.7 nM T72458 C0RM6I 23635105 Ki = 69 nM T72458 CB45UM 23635106 Ki = 6 nM T72458 CFNQ06 23635107 Ki = 2.8 nM T72458 CPE8L0 23635108 Ki = 2.2 nM T72458 CDC19H 23635109 Ki = 0.6 nM T72458 CHU29W 23635235 Ki = 2.8 nM T72458 CWL5K4 23635236 Ki = 5.7 nM T72458 CVFQ41 23635237 Ki = 5.9 nM T72458 CBW09O 23653113 Ki = 16000 nM T72458 C8KO9M 23661656 Ki = 11 nM T72458 C7DW6E 24180493 EC50 = 4.6 nM T72458 CK2Q5J 24180592 Ki = 3.4 nM T72458 C0QI2D 24180593 Ki = 0.9 nM T72458 C7SMW5 24180646 Ki = 0.9 nM T72458 CC4FM5 24740310 Ki = 890 nM T72458 CGY27Z 24740311 Ki = 260 nM T72458 CE6D9F 24740312 Ki = 6 nM T72458 CU19BT 24740419 Ki = 2.5 nM T72458 C2K1EL 24740535 Ki = 3.2 nM T72458 CTC05L 24740653 Ki = 3.7 nM T72458 CD90WZ 24740655 Ki = 0.59 nM T72458 CUPD43 24741624 Ki = 14 nM T72458 C2S3RO 24741625 Ki = 9.7 nM T72458 C52ZAS 24741961 Ki = 36 nM T72458 CT4I7Z 24741964 Ki = 39 nM T72458 CB47WZ 24764421 IC50 = 19.7 nM T72458 C5TA3W 24774358 IC50 = 160 nM T72458 CO4JK2 24774437 IC50 > 10000 nM T72458 CMB27G 24774521 IC50 = 520 nM T72458 C2TAK6 24774601 IC50 > 1000 nM T72458 C59NIQ 24848934 EC50 = 1.8 nM T72458 C2A1SX 24848995 EC50 = 80 nM T72458 C1EN7W 24857886 IC50 = 7.8 nM T72458 CB9M3F 24873537 Ki = 11 nM T72458 CS0L2N 24882666 Ki = 4200 nM T72458 CP2X4S 24886259 Ki = 6.8 nM T72458 CJ96SC 24886260 Ki = 12.7 nM T72458 CI37TV 24886498 Ki = 27.3 nM T72458 C1M8NX 24886499 Ki = 15.6 nM T72458 CU38LE 24886501 Ki = 75.8 nM T72458 C6IV8J 24886734 Ki = 31.4 nM T72458 C0YV3J 24886735 Ki = 70 nM T72458 CPQ74G 25022598 Ki = 1.1 nM T72458 CG9AV5 25058412 Ki = 8.1 nM T72458 CV07PW 25108215 EC50 = 0.28 nM T72458 CJ5HN6 25128748 EC50 = 37 nM T72458 C3WE0T 25128749 EC50 = 3 nM T72458 CP5TN2 25128751 Ki = 36 nM T72458 CUTA14 25129105 Ki = 6 nM T72458 CPL49Z 25129107 EC50 = 1.2 nM T72458 C4N5DH 25129108 EC50 = 9 nM T72458 CDC2Q6 25129109 EC50 = 1.7 nM T72458 CVSO97 25129453 EC50 = 0.8 nM T72458 CE79VX 25131477 EC50 = 391 nM T72458 C1B7KF 25131478 EC50 = 0.9 nM T72458 CIJ6P4 25132524 EC50 = 31 nM T72458 CY42MT 25132525 EC50 = 83 nM T72458 C9QG3J 25132526 EC50 = 8 nM T72458 CL3JV6 25132864 EC50 = 5 nM T72458 C57QZT 25132866 Ki = 4 nM T72458 CR6YZ2 25132867 EC50 = 25 nM T72458 C8AO5Y 25133207 Ki = 26 nM T72458 C3VGX6 25133208 EC50 = 10 nM T72458 C3KRA8 25133209 EC50 = 2.7 nM T72458 C9U6CQ 25133210 EC50 = 0.9 nM T72458 C74ACT 25133556 EC50 = 1.3 nM T72458 CW7O1N 25133903 EC50 = 167 nM T72458 CG3R0Y 25133907 EC50 = 28 nM T72458 C4SH1P 25211670 Ki = 9.6 nM T72458 CE01RM 25217223 Ki = 416.87 nM T72458 C8O1PH 25217225 Ki = 45 nM T72458 C4HK6C 42630327 EC50 < 0.03162 nM T72458 CU4S6X 44157099 IC50 = 2.5 nM T72458 CBG73U 44158097 EC50 = 43 nM T72458 CIOF26 44158168 IC50 = 0.6 nM T72458 C53LJK 44158169 IC50 = 5.7 nM T72458 CF7X1N 44158255 EC50 = 250 nM T72458 C9UD8I 44158336 EC50 = 200 nM T72458 CF6PT4 44158337 IC50 = 1.5 nM T72458 CHKI60 44265225 Ki > 1000000 nM T72458 CXN2R4 44265309 Ki = 94000 nM T72458 C3EJ1R 44265312 Ki = 161000 nM T72458 CWPT03 44265315 Ki = 24000 nM T72458 CJ1M6N 44265347 Ki = 44000 nM T72458 CEQ6K7 44265351 Ki = 89000 nM T72458 CSL48C 44265374 Ki = 2000 nM T72458 C97AIK 44265472 Ki = 107000 nM T72458 C6DZ4W 44265473 Ki = 8800 nM T72458 CLE96R 44265479 Ki = 68000 nM T72458 CV8GX6 44265487 Ki = 56000 nM T72458 C2CPG9 44265489 Ki = 104000 nM T72458 CLP5G3 44265496 Ki = 2100 nM T72458 C51TPY 44265586 Ki > 1000 nM T72458 CH5WM7 44265588 Ki > 1000 nM T72458 CT89LY 44265589 Ki = 105000 nM T72458 CZS3C7 44265590 Ki = 134000 nM T72458 C3YKG9 44265591 Ki = 56000 nM T72458 C74SBD 44265625 Ki > 1000 nM T72458 CRQ92O 44265626 Ki > 1000 nM T72458 CT2S8I 44265639 Ki = 6800 nM T72458 C18JZD 44265656 Ki = 205000 nM T72458 CZWE24 44265658 Ki = 66000 nM T72458 CD8UC0 44265662 Ki > 1000 nM T72458 C6OU7D 44265665 Ki > 1000 nM T72458 CC28FH 44265672 Ki = 9900 nM T72458 CSK9V6 44265674 Ki > 1000 nM T72458 CS46LN 44265675 Ki > 1000000 nM T72458 C9E0TB 44265681 Ki = 279000 nM T72458 CCGI15 44265707 Ki = 15000 nM T72458 CION54 44265708 Ki > 1000000 nM T72458 C9CM8W 44265711 Ki = 64000 nM T72458 CPUO61 44265713 Ki = 150000 nM T72458 CP1E6X 44265715 Ki = 14000 nM T72458 CRFQ64 44265719 Ki > 1000000 nM T72458 CXUI50 44265722 Ki = 127000 nM T72458 CVEG42 44265727 Ki > 1000 nM T72458 CC4S8V 44265739 Ki > 1000 nM T72458 CG1CH0 44265748 Ki > 1000 nM T72458 C82FPN 44265749 Ki = 139000 nM T72458 C05MIH 44265751 Ki = 30000 nM T72458 CP82FI 44265757 Ki > 1000 nM T72458 CE6A0Z 44265759 Ki > 1000 nM T72458 CPE83Q 44269189 EC50 = 23 nM T72458 CCP5L2 44269214 EC50 = 77 nM T72458 CN5TI2 44269217 EC50 = 2.9 nM T72458 C4M2LJ 44269245 EC50 = 40 nM T72458 C6LD9E 44275119 EC50 = 35 nM T72458 C60GXU 44275121 EC50 = 33 nM T72458 CFIT54 44275175 EC50 = 7 nM T72458 CO7KR8 44275191 EC50 = 37 nM T72458 C72TAL 44275192 EC50 = 15 nM T72458 CA7DX2 44275263 EC50 = 4 nM T72458 CK4E6O 44275264 EC50 = 176 nM T72458 CB4WG5 44275265 EC50 = 10 nM T72458 C3SH7Q 44275312 EC50 = 48 nM T72458 CIA54K 44275371 EC50 = 45 nM T72458 CBS9X6 44275372 EC50 = 7 nM T72458 C5RJ3Z 44275488 EC50 = 6 nM T72458 CBW0I1 44275650 EC50 = 0.9 nM T72458 CO9BJ6 44275654 EC50 = 65 nM T72458 COUM34 44275656 EC50 = 2 nM T72458 CSI8T3 44277299 EC50 = 120 nM T72458 CCGT80 44277300 EC50 = 90 nM T72458 CLG8Y1 44277301 EC50 = 130 nM T72458 C5OHC4 44277696 EC50 = 20 nM T72458 CMU9P1 44278071 EC50 = 180 nM T72458 C9Y7KM 44278193 EC50 = 13 nM T72458 CBWJ71 44278194 EC50 = 24 nM T72458 COS0B2 44278195 EC50 = 35 nM T72458 C8A1GE 44278223 EC50 = 130 nM T72458 CU0J1F 44279606 IC50 > 100000 nM T72458 CEG7U1 44279630 IC50 > 100000 nM T72458 CY9XO5 44279793 IC50 > 100000 nM T72458 CU8PH5 44293516 IC50 = 2.03 nM T72458 C7DZ1Q 44293599 EC50 = 3.38 nM T72458 C57HNX 44307979 IC50 > 10000 nM T72458 C8LZV7 44308004 IC50 > 10000 nM T72458 CFP7W8 44308044 IC50 > 10000 nM T72458 C79WRA 44308214 IC50 > 10000 nM T72458 CT76SR 44308215 IC50 > 10000 nM T72458 COY71H 44314826 EC50 = 0.17 nM T72458 CJAW38 44314951 IC50 > 10000 nM T72458 CA7B1G 44315095 IC50 = 9250 nM T72458 CPX2L1 44315335 IC50 > 10000 nM T72458 C3U0CW 44317053 EC50 = 1420 nM T72458 CKH3J2 44317070 EC50 = 3280 nM T72458 CAW8L7 44317241 EC50 = 20 nM T72458 CK7LG6 44317242 EC50 = 760 nM T72458 CZTI78 44317254 EC50 = 10 nM T72458 CVW5B7 44317276 EC50 = 70 nM T72458 C4ZST8 44317277 EC50 = 4800 nM T72458 C90PCI 44317278 EC50 = 1670 nM T72458 CLO83G 44317279 EC50 = 2500 nM T72458 CQ59BO 44320339 Ki = 1995.26 nM T72458 C6UML0 44322786 EC50 = 21.5 nM T72458 C3CL8S 44322787 EC50 = 6.3 nM T72458 C5SZ6K 44322788 EC50 = 38.5 nM T72458 C27QTD 44322795 EC50 = 1.6 nM T72458 C9HQ8Z 44322812 EC50 = 20.5 nM T72458 C3XED9 44322868 Ki = 220 nM T72458 C8P1HE 44322869 EC50 = 50 nM T72458 CJD5K7 44322895 EC50 = 11.5 nM T72458 CSH73B 44322896 EC50 = 4.6 nM T72458 C3V7PO 44322923 EC50 = 18 nM T72458 CA9F8I 44322924 EC50 = 53 nM T72458 C32ADM 44322957 EC50 = 22.5 nM T72458 CU1R6F 44322958 EC50 = 14.5 nM T72458 CPG80V 44322959 EC50 = 26.5 nM T72458 CJ73UR 44322977 EC50 = 16.5 nM T72458 CW5T8L 44322986 EC50 = 24 nM T72458 CN12SY 44322987 EC50 = 38.5 nM T72458 C8W2GN 44322994 EC50 = 42.5 nM T72458 CEV0F8 44323015 EC50 = 41 nM T72458 CSL38N 44323016 EC50 = 11 nM T72458 CEDS20 44323020 Ki = 57 nM T72458 CI70FV 44323029 Ki = 5 nM T72458 CNB32J 44323031 EC50 = 20 nM T72458 CP9FE1 44323032 EC50 = 13 nM T72458 CCX5N0 44323033 EC50 = 28 nM T72458 C7RT2W 44323034 EC50 = 21.3 nM T72458 CC9E1M 44323212 EC50 = 22 nM T72458 CX7H2C 44323233 Ki = 58 nM T72458 CW49BO 44323234 Ki = 87 nM T72458 C8BID0 44325926 IC50 = 38.7 nM T72458 C9MA4R 44343337 EC50 = 0.019 nM T72458 CD9ER8 44343341 IC50 = 1.8 nM T72458 C46OFK 44343362 EC50 = 0.573 nM T72458 CL8Y3V 44343363 EC50 = 0.018 nM T72458 CCLF38 44347081 Ki = 1300 nM T72458 CT5V4X 44347082 Ki = 3800 nM T72458 C0QW9K 44347105 Ki = 110 nM T72458 CWK01G 44347106 Ki = 58 nM T72458 C4Y2SW 44347107 Ki = 0.28 nM T72458 C60PGA 44347110 Ki = 960 nM T72458 CUEZ31 44347119 Ki = 0.37 nM T72458 CT03JB 44347219 Ki = 0.5 nM T72458 COD7W0 44347220 Ki = 0.26 nM T72458 CNP94O 44347221 Ki = 0.88 nM T72458 CBE37A 44347277 Ki = 4 nM T72458 CIZ30K 44347294 Ki = 4.3 nM T72458 C2YQM4 44347330 Ki = 3700 nM T72458 CX0Z1Y 44347331 Ki = 0.58 nM T72458 CAKI17 44347344 Ki = 0.06 nM T72458 CEIM86 44347370 Ki = 0.57 nM T72458 CS5ID0 44347378 Ki = 420 nM T72458 CDN35X 44347379 Ki = 600 nM T72458 CENG52 44347433 Ki = 1.6 nM T72458 CW1JY7 44347434 Ki = 0.096 nM T72458 C24GLU 44347435 Ki = 0.85 nM T72458 CSD69H 44347750 Ki = 1300 nM T72458 C1A6SC 44347765 Ki = 140 nM T72458 CY2K3L 44347766 Ki = 2000 nM T72458 C7U2KM 44347838 IC50 = 750 nM T72458 CK6FH3 44347927 IC50 = 3300 nM T72458 C2G4RI 44347976 Ki = 300 nM T72458 C9EA0M 44347977 Ki = 310 nM T72458 CN04GT 44347980 Ki = 180 nM T72458 CBW50H 44347987 Ki = 1500 nM T72458 CK93QZ 44347990 Ki = 670 nM T72458 C5BX1H 44348033 Ki = 2500 nM T72458 C27BLZ 44348035 Ki = 1600 nM T72458 CZ6R1G 44348039 Ki = 690 nM T72458 C4OS9M 44348046 Ki = 9300 nM T72458 C9JP8O 44348069 Ki = 270 nM T72458 CCI04W 44348070 Ki = 320 nM T72458 C58SIF 44348144 IC50 = 40000 nM T72458 CA4NE7 44348151 Ki = 620 nM T72458 CY96AB 44348152 Ki = 320 nM T72458 C0F1EA 44348183 EC50 > 10000 nM T72458 CC41MG 44348199 EC50 > 10000 nM T72458 CRSW34 44348200 EC50 = 6.3 nM T72458 CUM7X1 44348844 EC50 = 1000 nM T72458 C9I7PM 44348845 EC50 = 520 nM T72458 C3UWB5 44349006 EC50 = 1100 nM T72458 CT6G1M 44349008 EC50 = 2100 nM T72458 C6E7SA 44349019 EC50 = 24 nM T72458 CH4RT3 44349026 EC50 < 0.1 nM T72458 C6B2XF 44349055 EC50 = 110 nM T72458 CK7V8I 44349056 EC50 = 680 nM T72458 CDI5G1 44349057 EC50 = 470 nM T72458 CEB7L6 44349093 EC50 = 170 nM T72458 C17TCL 44349094 EC50 = 600 nM T72458 CZW0E4 44349105 EC50 = 4400 nM T72458 CC92YX 44349106 EC50 = 440 nM T72458 C84PZR 44349107 EC50 = 690 nM T72458 C8AT4B 44349110 EC50 = 1900 nM T72458 C2ZVP9 44349111 EC50 = 2400 nM T72458 C52OGQ 44349133 EC50 = 380 nM T72458 CZ36XH 44349134 EC50 = 2200 nM T72458 CY21EM 44349151 EC50 = 1600 nM T72458 CHP4U8 44349170 EC50 = 1000 nM T72458 C39SAR 44349173 EC50 = 5.2 nM T72458 C7RSC0 44349183 EC50 = 650 nM T72458 CWT14Q 44349221 IC50 = 3 nM T72458 CZ4M3J 44349222 IC50 = 3.3 nM T72458 CW9A4F 44349223 IC50 = 1.4 nM T72458 C7RMI0 44349224 IC50 = 11 nM T72458 CDW65K 44349226 IC50 = 220 nM T72458 CYHZ68 44349227 IC50 = 9.5 nM T72458 C3K9VR 44349228 IC50 = 19 nM T72458 C7OW3R 44349246 IC50 = 8.9 nM T72458 CBIV27 44349247 IC50 = 4.8 nM T72458 C8AU9D 44349461 EC50 = 530 nM T72458 C26WVI 44349469 IC50 = 13 nM T72458 CNYT90 44349470 IC50 = 32 nM T72458 C2XSM4 44349471 Ki = 2 nM T72458 CU9IJ2 44349593 EC50 = 83 nM T72458 CNB8U7 44349594 IC50 < 0.1 nM T72458 C6XV5P 44357167 IC50 = 12 nM T72458 CWBV76 44357280 IC50 = 22 nM T72458 C39OBA 44357294 IC50 = 18 nM T72458 CRP7I9 44357348 IC50 = 25 nM T72458 CG6HS3 44357406 IC50 = 21 nM T72458 C3TCL0 44357527 IC50 = 14 nM T72458 C3CX9P 44357528 IC50 = 110 nM T72458 CI3TO0 44357547 IC50 = 180 nM T72458 C2MFK4 44357575 IC50 = 90 nM T72458 C4QA0D 44357595 IC50 = 9 nM T72458 CH0XI2 44357626 IC50 = 22 nM T72458 CVZ1T6 44357786 IC50 = 10 nM T72458 C2MG1B 44358565 EC50 = 2.1 nM T72458 C8GKE0 44358566 EC50 = 820 nM T72458 C37KYE 44358608 IC50 = 2755 nM T72458 C7QTS9 44358609 EC50 = 500 nM T72458 CUH68B 44358622 IC50 = 9020 nM T72458 C6E9LI 44358625 IC50 = 5.598 nM T72458 C0WTS6 44358630 IC50 = 98 nM T72458 CN3EM4 44358633 IC50 = 3930 nM T72458 C8XY0P 44358639 IC50 = 2.27 nM T72458 C3TJC8 44358660 IC50 = 130 nM T72458 CM06ZW 44358669 IC50 = 2170 nM T72458 C2S6HF 44358693 IC50 = 2055 nM T72458 CQA6O7 44358695 EC50 > 5000 nM T72458 C81PLU 44358697 EC50 = 4050 nM T72458 CW8E5G 44358698 EC50 = 3060 nM T72458 CU89HD 44358705 EC50 = 260 nM T72458 C2VBG9 44358848 EC50 = 5800 nM T72458 C6RC5L 44358915 IC50 = 1197 nM T72458 CS0C2O 44358917 IC50 = 2990 nM T72458 C9ACB0 44360829 EC50 = 500 nM T72458 CX0ZW3 44361027 IC50 = 108 nM T72458 C2QW1I 44364160 IC50 = 45 nM T72458 CLMA12 44366081 IC50 = 0.23 nM T72458 C2DHN5 44366155 IC50 = 0.51 nM T72458 CYD6R3 44366171 IC50 = 0.5 nM T72458 CO7U1L 44366182 IC50 = 0.48 nM T72458 CL4CY1 44366187 IC50 = 270 nM T72458 C9JN3L 44366213 IC50 = 1.3 nM T72458 C36FMV 44366215 IC50 = 0.087 nM T72458 CS27ZR 44366381 IC50 = 0.16 nM T72458 C61CYL 44372908 EC50 = 77 nM T72458 CWT5B7 44372933 EC50 = 20 nM T72458 C8D1MC 44372942 EC50 = 1150 nM T72458 CEW35X 44372964 EC50 = 45 nM T72458 C2UCY5 44373177 EC50 = 20 nM T72458 CZ42QB 44373197 EC50 = 60 nM T72458 CCB05K 44373198 EC50 = 13 nM T72458 CX92FV 44373317 EC50 = 100 nM T72458 CR40BF 44383343 IC50 = 100 nM T72458 CQCP89 44387680 EC50 = 100 nM T72458 C7F3DV 44390411 EC50 = 4 nM T72458 CN3IE7 44390421 EC50 = 18 nM T72458 C5Y6HU 44390422 EC50 = 63 nM T72458 CR92QC 44390423 EC50 = 60 nM T72458 CEF15X 44390424 EC50 = 27 nM T72458 CP40IU 44391262 Ki = 110 nM T72458 CWO97F 44391271 Ki = 120 nM T72458 C58VDM 44391272 Ki = 160 nM T72458 CZMI04 44391285 Ki = 370 nM T72458 CGL71H 44391286 Ki = 270 nM T72458 C65PWK 44391288 Ki = 36 nM T72458 C9ZV5O 44391289 Ki = 110 nM T72458 CKT64C 44391303 Ki = 140 nM T72458 C1A6TX 44391304 Ki = 22 nM T72458 C07TBF 44391315 Ki = 41 nM T72458 CCV1R7 44391316 Ki = 87 nM T72458 C09FSO 44391379 Ki = 47 nM T72458 C0XPV5 44391380 Ki = 24 nM T72458 CVIE64 44391381 Ki = 120 nM T72458 CQU0T8 44391382 Ki = 10 nM T72458 CK7D6C 44391386 Ki = 52 nM T72458 C2B1EF 44391391 Ki = 56 nM T72458 C36DSN 44391402 Ki = 49 nM T72458 C0WT5A 44391403 Ki = 34 nM T72458 C39BFV 44391404 Ki = 33 nM T72458 CY8DP4 44391405 Ki = 30 nM T72458 CD8HL0 44392514 Ki = 860 nM T72458 CE21OM 44392535 Ki = 1500 nM T72458 C3IHV4 44393417 Ki = 390 nM T72458 C2J1ML 44393418 Ki = 1000 nM T72458 CQ3L0D 44393421 Ki = 1400 nM T72458 C9C7SD 44393430 Ki = 57000 nM T72458 C47HVD 44393441 Ki = 30000 nM T72458 C1OG5U 44393450 Ki = 169000 nM T72458 CX5F8Z 44393808 EC50 = 91 nM T72458 C3P9OV 44393809 EC50 = 36 nM T72458 CQ7ZW3 44393820 Ki = 84 nM T72458 CM1U6O 44393821 Ki = 35 nM T72458 CEX5T7 44393822 Ki = 24 nM T72458 C8NUV7 44393823 Ki = 145 nM T72458 CAT7F3 44393824 EC50 = 2.9 nM T72458 C6V0HU 44393850 EC50 = 40 nM T72458 CH60CQ 44393851 Ki = 49 nM T72458 CFJ6C3 44393862 Ki = 24 nM T72458 CZ2QV6 44393863 Ki = 25 nM T72458 CTM7X6 44393864 Ki = 13 nM T72458 CI8NO6 44393876 EC50 = 90 nM T72458 CI46JK 44393877 Ki = 102 nM T72458 CCV60F 44393885 EC50 = 18 nM T72458 CK2VD1 44393886 Ki = 23 nM T72458 C2IO4E 44393887 Ki = 11 nM T72458 CP8EQ1 44393888 Ki = 12 nM T72458 CR5BI0 44393889 Ki = 33 nM T72458 CN7YD9 44394009 Ki = 90 nM T72458 CS1YM0 44394010 Ki = 66 nM T72458 CKWJ51 44394078 Ki = 53 nM T72458 CK5D8I 44394079 Ki = 27 nM T72458 CT5C0V 44394080 Ki = 14 nM T72458 CM69EP 44394081 Ki = 81 nM T72458 C25TVF 44394093 EC50 = 168 nM T72458 C5K7CG 44394580 EC50 = 123 nM T72458 C08QML 44394581 EC50 = 38.5 nM T72458 C0OMU3 44394582 EC50 = 155 nM T72458 CL3P2Q 44394583 EC50 = 23.7 nM T72458 C5SGR6 44394584 EC50 = 150 nM T72458 CLXA10 44394585 EC50 = 13.7 nM T72458 C48NFW 44394586 EC50 = 68.7 nM T72458 C8GUD1 44394622 EC50 = 59.5 nM T72458 C9O4GM 44394623 EC50 = 4.6 nM T72458 C29ELZ 44394624 EC50 = 5 nM T72458 CP4A0B 44394625 EC50 = 88.5 nM T72458 C94PGA 44394626 EC50 = 159 nM T72458 CF4O9U 44394627 EC50 = 106 nM T72458 CZ37TO 44394654 EC50 = 39.3 nM T72458 CPE65R 44394655 EC50 = 35 nM T72458 C9LKB5 44394656 EC50 = 131 nM T72458 CG1Q8L 44394657 EC50 = 114 nM T72458 CHG12Y 44394658 EC50 = 31.3 nM T72458 C9OTX4 44394659 EC50 = 10.5 nM T72458 CNHD57 44394660 EC50 = 14.5 nM T72458 CHTM92 44394689 EC50 = 29.7 nM T72458 C04RCL 44394690 EC50 = 31.3 nM T72458 CT9D5Y 44394691 EC50 = 21 nM T72458 CHDB95 44394692 EC50 = 30 nM T72458 CHZF38 44394693 EC50 = 20 nM T72458 C9Y6ZI 44394694 EC50 = 121 nM T72458 C06PXF 44394695 EC50 = 82 nM T72458 CJ97VD 44394730 EC50 = 14.1 nM T72458 C1IE7P 44394731 EC50 = 8.5 nM T72458 CLF0X5 44394732 EC50 = 42 nM T72458 C9QR1L 44394733 EC50 = 12 nM T72458 CP1IR5 44394734 EC50 = 135 nM T72458 C2UY8G 44394735 EC50 = 18.7 nM T72458 CTY36S 44394736 EC50 = 27 nM T72458 CR5B6L 44394748 EC50 = 4527 nM T72458 CW13LR 44394749 EC50 = 137 nM T72458 CL3A0O 44394750 EC50 = 446 nM T72458 CIGZ40 44394783 EC50 = 45 nM T72458 C62FUR 44394784 EC50 = 58 nM T72458 CCZ37I 44394785 EC50 = 50 nM T72458 C8RHG3 44394786 EC50 = 96 nM T72458 CQD01R 44394787 EC50 = 185 nM T72458 CO43JY 44394788 EC50 = 146 nM T72458 CCE30Z 44394789 EC50 = 419 nM T72458 C8C6GY 44395416 Ki = 3900 nM T72458 CF3WX5 44395436 Ki = 600 nM T72458 C6ACZ4 44395464 Ki = 1000 nM T72458 CD6BN5 44395465 Ki = 3800 nM T72458 CS5O1J 44395466 Ki = 46 nM T72458 CC3Y5Q 44395503 Ki = 6400 nM T72458 CSAR32 44395513 Ki = 290 nM T72458 CAO42X 44395534 Ki = 5400 nM T72458 C8UY4T 44395535 Ki = 410 nM T72458 CQ7S4C 44395572 Ki = 1000 nM T72458 CSF9I6 44395614 Ki > 10000 nM T72458 C0S9PU 44395615 Ki = 30 nM T72458 C3T1KX 44395646 Ki = 1800 nM T72458 CA8M9V 44395647 Ki = 66 nM T72458 CP1K3Q 44395654 Ki = 38 nM T72458 CG1AR2 44395666 Ki > 10000 nM T72458 C9S6VA 44395667 Ki = 40 nM T72458 CVUQ61 44395681 Ki = 14 nM T72458 C6X2TM 44395869 Ki = 50 nM T72458 C1AN6P 44395899 Ki = 48 nM T72458 CAJM38 44395920 Ki = 140 nM T72458 C5VLQ9 44395948 Ki = 220 nM T72458 C35KSH 44395950 Ki = 26 nM T72458 CLT7X4 44396002 Ki = 41 nM T72458 CCZP29 44396036 Ki = 75 nM T72458 C0IF3K 44396067 Ki = 470 nM T72458 CR8UG7 44396068 Ki = 290 nM T72458 C6QME3 44396069 Ki = 430 nM T72458 C7QF9Y 44396079 Ki = 120 nM T72458 CJ39OH 44396102 Ki = 140 nM T72458 CYS89B 44396114 Ki = 110 nM T72458 C9TU4E 44396120 Ki = 86 nM T72458 C4NZF5 44396125 IC50 = 160 nM T72458 CLG84D 44396126 IC50 = 180 nM T72458 C63TUF 44396140 IC50 = 57.3 nM T72458 CPA70N 44396141 Ki = 210 nM T72458 CC15YA 44396158 Ki = 150 nM T72458 CQR2H1 44396953 Ki = 120 nM T72458 CN1SJ0 44396954 Ki = 270 nM T72458 C87ZDT 44396955 Ki = 340 nM T72458 CTNE47 44396956 Ki = 520 nM T72458 CZ59JV 44396957 Ki = 260 nM T72458 C8D2RU 44396986 EC50 = 238 nM T72458 C6Z9BD 44396987 IC50 = 14 nM T72458 C5OI8Q 44397027 Ki = 23 nM T72458 CZ2C9L 44397028 Ki = 7.6 nM T72458 C98DZS 44397029 Ki = 18 nM T72458 CDZ3O4 44397030 Ki = 8.4 nM T72458 CAZ6R7 44397053 Ki = 260 nM T72458 C34UVG 44397054 Ki = 490 nM T72458 CTF68U 44397079 Ki = 180 nM T72458 CZ7YU4 44397080 Ki = 340 nM T72458 CI8UE5 44397121 Ki = 61 nM T72458 CF6Z4Y 44397122 Ki = 92 nM T72458 CDS5M7 44397123 Ki = 110 nM T72458 CN83XR 44397124 Ki = 45 nM T72458 CI8H6N 44397125 Ki = 22 nM T72458 C6FXK8 44397129 Ki = 210 nM T72458 C4UNI8 44397130 Ki = 240 nM T72458 CK47TL 44397131 Ki = 250 nM T72458 CP9H1C 44397132 Ki = 350 nM T72458 CE1Y6G 44397133 Ki = 400 nM T72458 C7FG4M 44397195 Ki = 230 nM T72458 C9V2RU 44397198 Ki = 6.4 nM T72458 CSV12E 44397199 Ki = 21 nM T72458 CG0FU9 44397216 Ki = 290 nM T72458 C9CF7N 44397220 IC50 = 6 nM T72458 CPI0R3 44397222 Ki = 210 nM T72458 CIS6C5 44397223 Ki = 420 nM T72458 C25TBE 44397224 Ki = 36 nM T72458 C0BUD1 44397225 Ki = 62 nM T72458 CY4G9J 44397226 Ki = 540 nM T72458 CZV64D 44397279 Ki = 220 nM T72458 CU7E3B 44397280 Ki = 60 nM T72458 CXQ0M6 44397281 Ki = 11 nM T72458 CX2OM4 44397282 Ki = 18 nM T72458 CPM68W 44397283 Ki = 12 nM T72458 CX07ID 44397304 Ki = 12 nM T72458 C4ZE3U 44397307 Ki = 220 nM T72458 CV07QL 44397308 Ki = 190 nM T72458 CD81IL 44397337 IC50 = 1000 nM T72458 C32RCI 44397338 EC50 = 470 nM T72458 C5X6SW 44397339 IC50 = 290 nM T72458 C85BWQ 44397355 EC50 = 410 nM T72458 CYUE71 44397356 IC50 = 4.7 nM T72458 C7Z8GI 44397409 IC50 = 3.2 nM T72458 C7TNB6 44397410 EC50 = 61 nM T72458 CK6S9U 44397411 IC50 = 490 nM T72458 C3ODR7 44397412 EC50 = 550 nM T72458 C6XL4E 44397444 IC50 = 3.8 nM T72458 C40IAW 44397445 IC50 = 100 nM T72458 C6F0QR 44397455 IC50 = 0.56 nM T72458 CYF0K3 44397458 IC50 = 750 nM T72458 C8ZIU6 44397459 IC50 = 390 nM T72458 C30ZFY 44397460 IC50 = 160 nM T72458 C49FRZ 44397461 EC50 = 110 nM T72458 CFIQ85 44397534 EC50 = 1100 nM T72458 C4BWN8 44397535 IC50 = 1100 nM T72458 C2O0YK 44397569 EC50 = 210 nM T72458 C21NUS 44397570 EC50 = 680 nM T72458 CSI0J5 44397633 IC50 = 58 nM T72458 CD2ES6 44397651 IC50 = 36 nM T72458 CL6KA2 44397652 EC50 = 110 nM T72458 C78YOV 44397653 EC50 = 550 nM T72458 C3GM2K 44397654 EC50 = 710 nM T72458 C4OUF0 44397655 EC50 = 120 nM T72458 C3J8LY 44397657 EC50 = 200 nM T72458 C8H6EI 44397658 IC50 = 45 nM T72458 CQ6OU7 44397659 EC50 = 750 nM T72458 CIH93R 44397660 EC50 = 430 nM T72458 CKT12I 44397661 IC50 = 950 nM T72458 C1C8WZ 44397698 EC50 = 1100 nM T72458 CSYW04 44397700 IC50 = 17 nM T72458 CZJ60B 44397701 IC50 = 89 nM T72458 CRL32F 44397702 EC50 = 490 nM T72458 CNZ32D 44398259 EC50 = 19.95 nM T72458 C2YWK3 44398340 EC50 = 0.5012 nM T72458 CU7NG4 44400612 Ki = 23 nM T72458 CHGN15 44400658 Ki = 18 nM T72458 CJ36UT 44400660 Ki = 2.4 nM T72458 COM2E6 44400661 Ki = 3.1 nM T72458 C56OUG 44400662 Ki = 2 nM T72458 CTM72F 44400707 Ki = 18 nM T72458 C56BLV 44400708 Ki = 16 nM T72458 CL4A0W 44400709 Ki = 31 nM T72458 CQ8GK5 44400711 Ki = 14 nM T72458 COV9C6 44400768 Ki = 23 nM T72458 CJ4M7S 44400769 Ki = 420 nM T72458 CD4TC0 44400770 Ki = 5700 nM T72458 CO7NM3 44400777 Ki = 2.8 nM T72458 C0E3XG 44400778 Ki = 5 nM T72458 C0OC7A 44400809 Ki = 2.1 nM T72458 COJM70 44400810 Ki = 1.4 nM T72458 CFT4O6 44400811 Ki = 2.4 nM T72458 C5NJQ2 44400812 Ki = 5 nM T72458 CC8SI2 44400813 Ki = 2.9 nM T72458 C3I0DM 44400814 Ki = 1.3 nM T72458 C9SA2Y 44400824 Ki = 2300 nM T72458 C95VUG 44400825 Ki = 1100 nM T72458 C51RXY 44400834 Ki = 94 nM T72458 CAR95M 44400863 Ki = 4.5 nM T72458 C2VI7C 44400864 Ki = 1.7 nM T72458 CQ01GT 44400902 Ki = 3600 nM T72458 CQ16YO 44400903 Ki > 10000 nM T72458 C2MEL4 44400932 Ki = 4.6 nM T72458 C61RQJ 44400934 Ki = 2 nM T72458 C2IJZ5 44400935 Ki = 1.5 nM T72458 CYF7N9 44401275 Ki = 649 nM T72458 CKH54Y 44401285 Ki = 255 nM T72458 C1QM4Y 44401310 IC50 = 6 nM T72458 C1JK9O 44401341 Ki = 2780 nM T72458 CTOS16 44401367 Ki = 109 nM T72458 C3S2XK 44401371 Ki = 376 nM T72458 CH1OX7 44401386 Ki = 1057 nM T72458 CR8GT9 44401392 Ki = 8017 nM T72458 CBQ7N3 44401418 Ki = 667 nM T72458 C1O0YW 44401421 Ki > 50000 nM T72458 CJNH94 44401440 Ki = 138 nM T72458 CGA3W5 44401462 Ki > 50000 nM T72458 CUZJ52 44401513 Ki = 333 nM T72458 CM9W3D 44401520 EC50 = 5 nM T72458 CIQH79 44401522 EC50 = 3 nM T72458 CDSM37 44401524 EC50 = 5 nM T72458 CVN78D 44401528 IC50 = 5 nM T72458 C4R9XD 44401530 EC50 = 7 nM T72458 C9Y0LO 44401553 Ki = 47 nM T72458 C7E3YU 44401573 Ki = 1845 nM T72458 C5LID4 44401581 Ki = 310 nM T72458 C5AQD6 44401585 EC50 = 330 nM T72458 CGNC86 44401587 Ki = 10788 nM T72458 C74QHS 44401592 Ki = 243 nM T72458 CX30HI 44401607 Ki = 226 nM T72458 C1U3NV 44404522 EC50 = 3 nM T72458 CY80DJ 44404523 EC50 = 4 nM T72458 C5DB0V 44404524 EC50 = 6 nM T72458 C1CY7E 44404525 EC50 = 5 nM T72458 CUZ2B7 44404526 EC50 = 2 nM T72458 CNH3C0 44404528 EC50 = 130 nM T72458 C8RKY9 44404529 EC50 = 550 nM T72458 CNZL81 44404538 Ki = 472 nM T72458 CQC38R 44404540 Ki = 467 nM T72458 CKW61M 44404542 Ki = 261 nM T72458 CGT1S0 44404543 Ki = 157 nM T72458 C3LKV0 44404544 Ki = 106 nM T72458 CM2ER9 44404545 Ki = 125 nM T72458 C4MAJ1 44404546 Ki = 190 nM T72458 CVE9L3 44404547 Ki = 50 nM T72458 C72ONL 44404549 Ki = 14 nM T72458 C3F6JI 44404550 Ki = 111 nM T72458 CCF97M 44404560 Ki = 90 nM T72458 CW6UD5 44404561 Ki = 40 nM T72458 CUBW74 44404562 Ki = 130 nM T72458 CP7D1W 44404563 Ki = 110 nM T72458 CU92ZV 44404564 Ki = 40 nM T72458 C6QC2S 44404566 Ki = 150 nM T72458 C35QSF 44404567 Ki = 200 nM T72458 CPF03E 44404568 Ki = 70 nM T72458 CR93UF 44404570 Ki = 70 nM T72458 CKC91E 44404571 Ki = 20 nM T72458 CKY6G8 44404572 Ki = 190 nM T72458 C1TXF6 44404575 Ki = 150 nM T72458 C4IFA0 44404576 Ki = 100 nM T72458 C0FB6W 44404577 Ki = 483 nM T72458 C5EX1D 44404822 Ki = 900 nM T72458 CL8U6X 44404823 Ki = 900 nM T72458 CQMR23 44405360 Ki = 11 nM T72458 CGV7U9 44405361 Ki = 79 nM T72458 C3BP8S 44405362 Ki = 99 nM T72458 CN9FE0 44405364 Ki = 100 nM T72458 CJ95PM 44405365 Ki = 210 nM T72458 CX9E1R 44405366 Ki = 42 nM T72458 C4K9OG 44405368 Ki = 130 nM T72458 CA2D8P 44405374 Ki = 180 nM T72458 CD1U0B 44405375 Ki = 260 nM T72458 CK6S4G 44405376 Ki = 80 nM T72458 CMOH97 44405377 Ki = 120 nM T72458 CK36RZ 44405378 Ki = 140 nM T72458 CFW20E 44405382 Ki = 61 nM T72458 C8GE4Y 44405392 Ki = 280 nM T72458 CVF02W 44405395 Ki = 60 nM T72458 C8A0QP 44405402 Ki = 84 nM T72458 C75WLG 44405403 Ki = 97 nM T72458 CQK5O8 44405425 Ki = 82 nM T72458 CEVF76 44405426 Ki = 16 nM T72458 CSV9Z7 44405443 Ki = 170 nM T72458 CX1RP9 44405450 Ki = 100 nM T72458 C47ZWV 44405526 EC50 = 570 nM T72458 C7VJ2H 44405549 Ki = 140 nM T72458 CA21ST 44405553 Ki = 160 nM T72458 C9JUS5 44405558 Ki = 150 nM T72458 CXYL12 44405561 Ki = 270 nM T72458 CC68NS 44405562 Ki = 230 nM T72458 CUVK05 44405563 Ki = 1000 nM T72458 CF1W2D 44405582 Ki = 130 nM T72458 CH5BW3 44405596 Ki = 210 nM T72458 CVXJ50 44405613 Ki = 110 nM T72458 CB46SC 44405620 Ki = 300 nM T72458 C3NL7Z 44405681 EC50 = 3 nM T72458 C6TE2H 44405769 EC50 = 72 nM T72458 C5W2NU 44405770 EC50 = 5 nM T72458 CU3MJ7 44405773 EC50 = 2 nM T72458 CGMF87 44405785 EC50 = 50 nM T72458 CEH5M3 44405791 EC50 = 90 nM T72458 CRG17F 44405792 EC50 = 2 nM T72458 CA5N2U 44405793 EC50 = 2 nM T72458 CR9GY2 44405794 EC50 = 15 nM T72458 CYW82T 44405802 EC50 = 110 nM T72458 C2B0HL 44405812 EC50 = 5 nM T72458 C6YNC5 44405823 EC50 = 39 nM T72458 CKY6L1 44405825 EC50 = 85 nM T72458 CIY3N6 44405826 EC50 = 3 nM T72458 CH5E4L 44405832 EC50 = 200 nM T72458 CY63HS 44405833 EC50 = 2 nM T72458 CVHQ82 44405835 EC50 = 2 nM T72458 CT9WH8 44405836 EC50 = 2 nM T72458 C7FCD0 44405857 EC50 = 3 nM T72458 CMY9H2 44405858 EC50 = 2 nM T72458 C8AL0J 44405860 EC50 = 2 nM T72458 CL3T6Z 44405879 EC50 = 15 nM T72458 CDR54Z 44405910 EC50 = 2 nM T72458 C0H2SP 44405911 EC50 = 11 nM T72458 C4OM2E 44405913 EC50 = 220 nM T72458 CRMV98 44408154 EC50 = 5.8 nM T72458 CIWX60 44408155 IC50 = 2.1 nM T72458 COG72Y 44408173 EC50 = 5.3 nM T72458 C3CQ4J 44408189 IC50 = 4.3 nM T72458 CW08ZJ 44408190 IC50 = 4 nM T72458 CNWJ27 44408252 EC50 = 16 nM T72458 CH68SP 44408253 EC50 = 14 nM T72458 CCFV91 44408275 EC50 = 8.6 nM T72458 CZ3YG9 44408276 EC50 = 6.1 nM T72458 CAFP51 44408286 EC50 = 2.4 nM T72458 CR8HZ7 44408287 EC50 = 1.3 nM T72458 COC7D2 44408388 EC50 = 15 nM T72458 CJ4N3I 44409103 EC50 = 8 nM T72458 C2NJ0V 44409104 Ki = 13 nM T72458 CKF52N 44409140 EC50 = 160 nM T72458 C5XEI8 44409206 Ki = 76 nM T72458 C9EXZ2 44409337 EC50 = 38 nM T72458 CFT41O 44409338 Ki = 5 nM T72458 CUB1Q2 44409339 EC50 = 20 nM T72458 CK5GO1 44409379 EC50 = 193 nM T72458 CUD19G 44410040 Ki = 0.58 nM T72458 CH1E8N 44410041 Ki = 21 nM T72458 C4Y8LV 44410046 Ki = 26 nM T72458 C61ZVJ 44410175 Ki = 13 nM T72458 C06FAT 44410176 Ki = 2.8 nM T72458 COFW07 44410188 Ki = 5.1 nM T72458 C5QG1S 44410207 Ki = 700 nM T72458 C8F2TJ 44410349 Ki = 26000 nM T72458 CKRP65 44410378 Ki = 110 nM T72458 C6IB1X 44410379 Ki = 14 nM T72458 CL0H4T 44410385 Ki = 690 nM T72458 C48WZD 44410802 Ki = 17.3 nM T72458 C43IKV 44410803 Ki = 10.4 nM T72458 CC8DA0 44412509 Ki = 12 nM T72458 CX60PS 44412510 Ki = 10 nM T72458 C3KB7R 44412511 Ki = 148 nM T72458 C1EOW5 44412512 Ki = 26 nM T72458 CT2N0X 44412513 Ki = 3 nM T72458 C20OFY 44412559 Ki = 3427 nM T72458 C20ZDH 44412560 Ki = 4 nM T72458 CPQJ43 44412561 Ki = 4 nM T72458 CF5G4W 44412572 Ki = 326 nM T72458 C56OPH 44412574 Ki = 3 nM T72458 C9T3YV 44412612 Ki = 2 nM T72458 CSO69M 44412613 Ki = 10 nM T72458 CG23BY 44412626 Ki = 14 nM T72458 CJYM45 44412640 Ki = 13 nM T72458 CEK59C 44412641 Ki = 13 nM T72458 CB6K4I 44412642 Ki = 5 nM T72458 CRD87I 44412646 Ki = 18 nM T72458 CAF4V8 44412647 Ki = 35 nM T72458 CC2QB0 44412665 Ki = 54 nM T72458 CS8EC2 44412676 Ki = 1800 nM T72458 C1QPI3 44412677 Ki = 1500 nM T72458 CXNI74 44412678 Ki = 450 nM T72458 C3UF8S 44412679 Ki = 360 nM T72458 C1VA2R 44412680 Ki = 1000 nM T72458 C3Y0LF 44412681 Ki = 550 nM T72458 CZ3E0A 44412684 Ki = 1800 nM T72458 C65XZU 44412685 Ki = 440 nM T72458 C3GEM5 44412687 Ki = 1100 nM T72458 C57SDW 44412688 Ki = 1300 nM T72458 CLT8W2 44412690 Ki = 1000 nM T72458 CB6H8W 44412691 Ki = 560 nM T72458 C9K3XB 44412711 Ki = 2200 nM T72458 C6GO1C 44412729 Ki = 2600 nM T72458 C0NAS2 44412740 Ki = 1800 nM T72458 CE4QZ5 44412758 Ki = 7 nM T72458 C1K8LS 44412770 Ki = 2800 nM T72458 CX8K7T 44412791 Ki = 1200 nM T72458 CCZP41 44412864 Ki = 1200 nM T72458 CPU13S 44412869 Ki = 21 nM T72458 C9GRF4 44412881 Ki = 1300 nM T72458 CC49LZ 44412884 Ki = 130 nM T72458 C3Q6RO 44412896 Ki = 87 nM T72458 CNP17D 44412897 Ki = 12 nM T72458 CXDA47 44412898 Ki = 8.8 nM T72458 CF73OD 44412909 Ki = 420 nM T72458 CS02LO 44412910 Ki = 480 nM T72458 C6D3MA 44412911 Ki = 15 nM T72458 C7Z8WB 44412912 Ki = 180 nM T72458 CW31RQ 44412930 Ki = 200 nM T72458 CM1J9Q 44412931 Ki = 1500 nM T72458 C4KWB3 44412933 Ki = 1.6 nM T72458 CA9YQ3 44412963 Ki = 710 nM T72458 C0E7QK 44412964 Ki = 520 nM T72458 C0OWN7 44412990 Ki = 750 nM T72458 CA8BU2 44413002 Ki = 310 nM T72458 CJM74H 44413005 Ki = 170 nM T72458 CZX75O 44413056 Ki = 710 nM T72458 CW6ZC0 44413576 EC50 = 10133.6 nM T72458 CG59EP 44413600 Ki = 214.6 nM T72458 CZY3R6 44413602 Ki = 69.6 nM T72458 CJ71PZ 44413604 Ki = 369.9 nM T72458 CPB02M 44413606 Ki = 41.8 nM T72458 CHT0V3 44413652 Ki = 43.9 nM T72458 C0AT2B 44413666 Ki = 68.4 nM T72458 CJY9Q1 44413668 Ki = 5 nM T72458 CN3WD2 44413684 Ki = 100.7 nM T72458 CJQ3N4 44413687 Ki = 46.9 nM T72458 C4T2ES 44413741 Ki = 37.5 nM T72458 C24AUD 44413828 EC50 = 36 nM T72458 C08PBM 44413829 EC50 = 54 nM T72458 CT4FW5 44413830 EC50 = 8 nM T72458 C8IDV1 44413831 EC50 = 457 nM T72458 CZ3Q4T 44413832 EC50 = 515 nM T72458 CV6Z8C 44413842 EC50 = 1617 nM T72458 C4P0LS 44413879 EC50 = 152 nM T72458 C84OJQ 44413880 EC50 = 249 nM T72458 CN7I2S 44413881 EC50 = 254 nM T72458 CF6O4K 44413913 EC50 = 184 nM T72458 CS42BM 44413914 EC50 = 3.7 nM T72458 CN18BL 44413930 EC50 = 14 nM T72458 C4BMF6 44413931 EC50 = 4.3 nM T72458 C9WNH8 44413932 EC50 = 17 nM T72458 CKZ86P 44413938 EC50 = 20 nM T72458 CL2RK9 44413968 EC50 = 1093 nM T72458 CM2J9Z 44413969 Ki = 1712 nM T72458 C34XGB 44413970 Ki = 6666 nM T72458 CA5K6H 44415336 Ki > 10000 nM T72458 CW4FC2 44415337 Ki = 2600 nM T72458 CEU1V2 44415346 Ki = 86 nM T72458 CJ81VG 44415347 Ki = 4000 nM T72458 CDJ81P 44415348 Ki > 10000 nM T72458 CJ3K6S 44415359 Ki = 57 nM T72458 CJ74MF 44415360 Ki = 2500 nM T72458 CS4D9A 44415361 Ki = 350 nM T72458 CW25PK 44415369 Ki = 2800 nM T72458 CIA0T1 44415370 Ki = 1700 nM T72458 C2YMO0 44415377 Ki = 300 nM T72458 CEW9H0 44415384 Ki = 3300 nM T72458 CA8P2G 44415388 Ki = 400 nM T72458 CHC07X 44415398 Ki = 210 nM T72458 CX2WN0 44415405 Ki = 75 nM T72458 CC29YV 44415406 Ki = 74 nM T72458 C7IYH9 44415417 Ki = 110 nM T72458 C0QMO7 44415418 Ki = 94 nM T72458 CV2UY4 44415429 Ki = 690 nM T72458 CY8F9L 44415430 Ki = 1000 nM T72458 CEG71C 44415433 Ki = 140 nM T72458 C01ZBF 44415434 Ki = 170 nM T72458 CHK45T 44415442 Ki = 620 nM T72458 C1B6CI 44415453 Ki = 160 nM T72458 CECU63 44415479 Ki = 25 nM T72458 C6YI9R 44415521 Ki = 490 nM T72458 CKX67G 44415522 Ki = 190 nM T72458 CZ48AF 44415537 Ki = 1400 nM T72458 C84OHY 44415545 Ki = 2100 nM T72458 C2NQ3C 44415546 Ki = 2200 nM T72458 C4ERO9 44415630 Ki = 56 nM T72458 C7Z3YB 44415631 Ki = 1800 nM T72458 C24YUZ 44415659 Ki = 89 nM T72458 C1C2GZ 44415660 Ki = 2400 nM T72458 CGR80P 44415674 Ki = 110 nM T72458 CV0TQ9 44415675 Ki = 360 nM T72458 C6YM0F 44415691 Ki = 2800 nM T72458 CAH6W2 44415692 Ki = 64 nM T72458 CKWO35 44415693 Ki = 18 nM T72458 CT0A3Y 44415706 Ki = 780 nM T72458 C1MG0H 44415707 Ki = 30 nM T72458 C07BZO 44415709 Ki = 1900 nM T72458 CYC49B 44415725 Ki = 4600 nM T72458 C10ZBJ 44415726 Ki = 2300 nM T72458 C5BIZ4 44415727 Ki = 5900 nM T72458 CZ63NT 44415746 Ki = 4900 nM T72458 CBYA87 44415747 Ki = 640 nM T72458 CTEW36 44415748 Ki = 3000 nM T72458 C3F2MN 44415764 Ki = 2600 nM T72458 CQ4C0E 44415765 Ki = 1500 nM T72458 CNR4B5 44415766 Ki = 1600 nM T72458 C9L1FV 44415767 Ki = 92 nM T72458 CM0UP6 44415790 Ki = 4300 nM T72458 CKB35A 44415791 Ki = 2500 nM T72458 CWK5C9 44415809 Ki = 6100 nM T72458 C8Y2QU 44415902 Ki = 820 nM T72458 C3KQ8H 44415912 EC50 = 1.6 nM T72458 CDN97X 44415913 EC50 = 0.3 nM T72458 CAL83K 44415914 EC50 = 0.2 nM T72458 C5CF0M 44415918 EC50 = 2 nM T72458 CXI18W 44415919 Ki = 0.4 nM T72458 C6DH7I 44415920 Ki = 1.3 nM T72458 CIM96K 44415925 Ki = 1100 nM T72458 C1X0OG 44415926 Ki = 5700 nM T72458 C9GO0A 44415940 Ki = 4100 nM T72458 CL95SI 44415941 Ki = 4200 nM T72458 C06CYU 44415956 EC50 = 809 nM T72458 C76IXM 44415961 Ki > 10000 nM T72458 CE24IH 44415965 Ki = 47 nM T72458 C6KGF3 44415966 Ki = 31 nM T72458 CD2A9T 44415972 EC50 = 140 nM T72458 CP0GH2 44415984 Ki = 120 nM T72458 CA7YJ4 44415985 Ki = 920 nM T72458 CHT4E8 44415991 EC50 = 45 nM T72458 CHJ4T5 44416006 Ki = 3100 nM T72458 CV42LA 44416007 Ki = 2200 nM T72458 CPX62S 44416014 EC50 = 18 nM T72458 C6CHM0 44416020 Ki = 2800 nM T72458 CQ7P9R 44416023 Ki = 4500 nM T72458 C4HU5K 44416024 Ki = 4000 nM T72458 CB6Y3A 44416025 Ki = 1500 nM T72458 CITW80 44416043 Ki = 2500 nM T72458 CX12AI 44416044 Ki = 2500 nM T72458 CXNE97 44416045 Ki = 3600 nM T72458 C8A5KJ 44416046 Ki = 2100 nM T72458 C69CUX 44416057 EC50 = 0.34 nM T72458 C56DHI 44416060 EC50 = 1.6 nM T72458 C0LIB3 44416071 Ki = 2900 nM T72458 CZ78QT 44416072 Ki = 2600 nM T72458 C05WHL 44416073 Ki = 2000 nM T72458 C8PA7D 44416074 Ki = 4800 nM T72458 C14XFK 44416075 Ki > 10000 nM T72458 CJI3N4 44416092 Ki = 4400 nM T72458 CK35LI 44416093 Ki = 3800 nM T72458 CS0JZ7 44416094 Ki > 10000 nM T72458 CB2TU4 44416106 EC50 = 0.5 nM T72458 C6Y3SN 44416108 Ki = 4600 nM T72458 CY12SN 44416109 Ki = 3100 nM T72458 CP9T4B 44416122 EC50 = 12 nM T72458 C4FI3Y 44416126 Ki = 2600 nM T72458 C9KLB0 44416135 EC50 = 2.2 nM T72458 C37XPA 44416152 Ki = 5.3 nM T72458 CB3WH4 44416160 Ki = 60 nM T72458 CE32FW 44416161 Ki = 38 nM T72458 C8IFH0 44416162 Ki = 67 nM T72458 CT89FC 44416163 Ki = 160 nM T72458 CC93LB 44416182 Ki = 36 nM T72458 CWF02K 44416183 Ki = 8.8 nM T72458 CI4EV8 44416184 Ki = 80 nM T72458 CWE8T7 44416194 Ki = 71 nM T72458 CE1FA5 44416197 Ki = 6.5 nM T72458 C74NDV 44416200 Ki = 67 nM T72458 CRYG36 44416201 Ki = 16 nM T72458 C53WDB 44416208 Ki = 240 nM T72458 CSM1D2 44416209 Ki = 200 nM T72458 CZ7M5G 44416213 Ki = 12 nM T72458 C0YN8C 44416214 Ki = 1700 nM T72458 CN38JL 44416227 Ki = 230 nM T72458 CD4B9L 44416228 Ki = 120 nM T72458 C1NMV4 44416251 Ki = 92 nM T72458 CF4GR8 44416286 Ki = 5.9 nM T72458 CFKR01 44416298 Ki = 20 nM T72458 CTB6N2 44416299 Ki = 8.1 nM T72458 C9EVI6 44416327 Ki = 9.1 nM T72458 CTZ02S 44416338 Ki = 390 nM T72458 C9AUM3 44416349 Ki = 31 nM T72458 CI1A0C 44416361 Ki = 26 nM T72458 CU7C3F 44416375 Ki = 140 nM T72458 C7SC9P 44417549 IC50 = 1.8 nM T72458 CBCR82 44417551 IC50 = 4.1 nM T72458 CK0P4I 44417552 IC50 = 0.7 nM T72458 CT58RV 44417554 IC50 = 101 nM T72458 C32QEO 44418413 EC50 > 10000 nM T72458 C7FEU6 44418420 EC50 > 10000 nM T72458 CZW07E 44418421 EC50 > 10000 nM T72458 CLQG83 44418430 EC50 = 2.7 nM T72458 C8VG1S 44418431 IC50 = 1.2 nM T72458 C3HPI5 44418437 EC50 > 10000 nM T72458 CMD5N2 44418438 EC50 > 10000 nM T72458 CQE30X 44422937 IC50 = 1600 nM T72458 C6H0NU 44422958 IC50 > 10000 nM T72458 C7I0KW 44422959 IC50 > 10000 nM T72458 C46XOB 44422960 IC50 > 10000 nM T72458 CNM90E 44422961 IC50 > 10000 nM T72458 C2LQW9 44422997 IC50 = 4500 nM T72458 CJM09S 44422998 IC50 = 3600 nM T72458 CI9HF1 44422999 IC50 = 1200 nM T72458 CXH5F8 44423009 IC50 = 590 nM T72458 C3VOD0 44423010 IC50 = 4800 nM T72458 C7UI3W 44423011 IC50 > 5000 nM T72458 CI05BD 44423012 IC50 > 10000 nM T72458 C5EJ3P 44423013 IC50 > 10000 nM T72458 C2NR7G 44423014 IC50 > 10000 nM T72458 C3I2NF 44423359 IC50 = 333 nM T72458 CBDI21 44423373 IC50 = 52.7 nM T72458 CY73KM 44423376 IC50 = 52.2 nM T72458 CB3M0V 44423378 IC50 = 18.3 nM T72458 COZ8M7 44423380 IC50 = 98.6 nM T72458 C9OGJ7 44423382 IC50 = 23.4 nM T72458 C0U7DO 44423384 IC50 = 14.5 nM T72458 C8GO6W 44423420 IC50 = 594 nM T72458 CVSF54 44423421 IC50 = 567 nM T72458 CEH52R 44423422 IC50 = 208 nM T72458 C4MO9L 44423424 IC50 = 218 nM T72458 C02WHJ 44423425 IC50 = 341 nM T72458 CA01NG 44423426 IC50 = 1250 nM T72458 CXA18B 44423427 IC50 = 1870 nM T72458 C17DFM 44423428 IC50 = 1190 nM T72458 C7EM3T 44423429 IC50 = 336 nM T72458 CP8BY0 44423430 IC50 = 105 nM T72458 CB6JP2 44423431 IC50 = 177 nM T72458 CE8U4Y 44423432 IC50 = 147 nM T72458 CV53RU 44423433 IC50 = 241 nM T72458 C40UAO 44423434 IC50 > 10000 nM T72458 C6JZ4Q 44423435 IC50 = 745 nM T72458 C36BEG 44423436 IC50 = 653 nM T72458 C58ZAM 44423437 IC50 = 132 nM T72458 C3KQR1 44423438 IC50 = 2300 nM T72458 C0OA8S 44423439 IC50 = 565 nM T72458 CBI7U4 44423440 IC50 = 159 nM T72458 CMNR76 44423441 IC50 = 296 nM T72458 CF6SQ1 44423442 IC50 = 226 nM T72458 CB46XE 44423443 IC50 = 756 nM T72458 CC3VY2 44423444 IC50 = 36.8 nM T72458 C8RX6Y 44423445 IC50 = 228 nM T72458 CC9GO8 44423446 IC50 = 26 nM T72458 C3S7UM 44423447 IC50 = 82.8 nM T72458 CDP0C8 44423448 IC50 = 47.2 nM T72458 CQCX97 44423449 IC50 = 18 nM T72458 CQ4DG9 44423450 IC50 = 186 nM T72458 C1CZK0 44423451 IC50 = 65.1 nM T72458 C6S4WV 44423452 IC50 = 156 nM T72458 C3J0ZH 44423453 IC50 = 243 nM T72458 CK8TR1 44423454 IC50 = 23 nM T72458 CNB0L9 44423455 IC50 = 33 nM T72458 C8FBW9 44423456 IC50 = 27.1 nM T72458 CV54PE 44423457 IC50 = 11.7 nM T72458 CG45MD 44423458 IC50 = 27.1 nM T72458 CM0K5Y 44423459 IC50 = 24.3 nM T72458 CFLS73 44423460 IC50 = 15.2 nM T72458 CX2T9W 44423461 IC50 = 36.8 nM T72458 C6D1CU 44423462 IC50 = 23.6 nM T72458 CR3XM9 44423463 IC50 = 10.5 nM T72458 C93PXI 44423464 IC50 = 53.2 nM T72458 C1UI9Z 44423465 IC50 = 41.8 nM T72458 C1WX7C 44423466 IC50 = 42.6 nM T72458 C80QNR 44423467 IC50 = 100 nM T72458 CAU4H2 44423468 IC50 = 228 nM T72458 C3Y0VW 44423469 IC50 = 62.8 nM T72458 CW78PM 44423470 IC50 = 85.9 nM T72458 CN07QR 44423471 IC50 = 92.5 nM T72458 CNKS25 44426649 IC50 = 900 nM T72458 CN5RD6 44431510 EC50 > 10000 nM T72458 CF3H8A 44431511 EC50 > 10000 nM T72458 CVB07O 44431512 EC50 = 3200 nM T72458 CY80GN 44431513 IC50 = 1700 nM T72458 COCE51 44431515 EC50 = 2.87 nM T72458 CIM51K 44432885 Ki = 1000 nM T72458 CJN61T 44432891 Ki = 17000 nM T72458 C2W8XE 44432895 Ki = 11000 nM T72458 CI1Y8B 44432897 Ki = 630.96 nM T72458 CV03FK 44432898 Ki = 60 nM T72458 COW1J6 44432899 Ki = 218.78 nM T72458 CC0AJ8 44432900 Ki = 128.82 nM T72458 CLH19Y 44432902 Ki = 51 nM T72458 C4E2AY 44432903 Ki = 11.75 nM T72458 CZ3DA9 44432906 Ki = 7.9 nM T72458 C2C0YT 44432909 Ki = 4.898 nM T72458 CI61RS 44432913 Ki = 32.36 nM T72458 CPBJ64 44432916 Ki = 724.44 nM T72458 CC1FG7 44432917 Ki = 50 nM T72458 CABP12 44432918 Ki > 10000 nM T72458 CRHG83 44432920 Ki = 2290.87 nM T72458 CWF23Z 44432924 Ki = 4.467 nM T72458 CAK9Z8 44432927 Ki = 109.65 nM T72458 CWV84F 44432928 Ki = 7.244 nM T72458 CXPZ80 44432930 Ki = 5 nM T72458 CNM17K 44432931 Ki = 2.692 nM T72458 CV62SP 44432932 Ki = 3.3 nM T72458 CP1G3N 44432933 Ki = 6.457 nM T72458 CDHA64 44432939 Ki = 3.7 nM T72458 C7DZ3N 44432941 Ki = 0.8913 nM T72458 CPG0Z7 44432943 Ki = 2.138 nM T72458 CO7D3R 44432945 Ki = 8.3 nM T72458 CSM8T7 44432946 Ki = 8.71 nM T72458 CGNI61 44432947 Ki = 7.5 nM T72458 CD0ZV7 44432948 Ki = 5.2 nM T72458 C5P1UZ 44432949 Ki = 2.042 nM T72458 CVX47L 44432950 Ki = 1.7 nM T72458 CC06WF 44432951 Ki = 9.7 nM T72458 CHQO21 44432952 Ki = 4.169 nM T72458 CB62YF 44432953 Ki = 14 nM T72458 C2N0MD 44432954 Ki = 33 nM T72458 C0EY7P 44432955 Ki = 17.38 nM T72458 CX3NB9 44432956 Ki = 5.754 nM T72458 C3P5QE 44432957 Ki = 30.9 nM T72458 CXP4J8 44432958 Ki = 77.62 nM T72458 CKNT36 44432959 Ki = 19.95 nM T72458 C0V2US 44432960 Ki = 44.67 nM T72458 CN41MP 44432962 Ki = 3.2 nM T72458 CBRG36 44432963 Ki = 2.9 nM T72458 CL3ZR1 44432964 Ki = 3.89 nM T72458 CDNP90 44432965 Ki = 28 nM T72458 C0L4NV 44432966 Ki = 0.955 nM T72458 CW6V3C 44433158 Ki = 770 nM T72458 C3B7EG 44433262 Ki = 6.4 nM T72458 CPRL53 44433263 Ki = 26 nM T72458 CKX7P2 44433264 Ki = 4.5 nM T72458 CQ91YU 44433265 Ki = 6.2 nM T72458 CJZ3P7 44433266 Ki = 7.9 nM T72458 CRP35K 44433267 Ki = 6.4 nM T72458 CF3J7G 44433268 Ki = 8.7 nM T72458 C3ZIE0 44433269 Ki = 60 nM T72458 CN51TW 44433270 Ki = 1 nM T72458 CQ4X7E 44433271 Ki = 1.5 nM T72458 C4O5HS 44433272 Ki = 3.8 nM T72458 CEA96F 44433273 Ki = 49 nM T72458 CED62W 44433274 Ki = 120 nM T72458 CI29CM 44433275 Ki = 56 nM T72458 CEN1M3 44433276 Ki = 0.95 nM T72458 C9KT3N 44433277 Ki = 1.4 nM T72458 CS2YQ7 44433278 Ki = 140 nM T72458 C27GZL 44433279 Ki = 27 nM T72458 CB29IZ 44433282 Ki = 240 nM T72458 COX3A0 44433283 Ki = 40 nM T72458 CAE5J2 44433284 Ki = 3.8 nM T72458 C9U4FM 44433285 Ki = 2.4 nM T72458 CB6P5W 44433286 Ki = 6 nM T72458 C3R0EA 44433287 Ki = 1 nM T72458 CZN71T 44433288 Ki = 23 nM T72458 CR54CU 44433289 Ki = 7 nM T72458 C1M0JP 44433290 Ki = 0.71 nM T72458 C9ZT8U 44433291 Ki = 26 nM T72458 CI62TG 44433292 Ki = 57 nM T72458 CZ3I4N 44433293 Ki = 2 nM T72458 CZU4D1 44433294 Ki = 1.9 nM T72458 CS5TK4 44433295 Ki = 5 nM T72458 CYH7M2 44433296 Ki = 1.1 nM T72458 C7E4KR 44433297 Ki = 2.6 nM T72458 CPX57U 44433298 Ki = 1.4 nM T72458 CI2PC5 44433299 Ki = 1.5 nM T72458 C89WJP 44433300 Ki = 12 nM T72458 CEJ6Q8 44433378 Ki = 82 nM T72458 CYHD52 44433379 Ki = 390 nM T72458 C16UBL 44433380 Ki = 66 nM T72458 C1ABU5 44433381 Ki = 30 nM T72458 CUX68D 44433382 Ki = 96 nM T72458 CF3GN1 44433383 Ki = 95 nM T72458 C6Z9HA 44433384 Ki = 26 nM T72458 CG9N7V 44433385 Ki = 120 nM T72458 CVB59A 44433386 Ki = 180 nM T72458 CMH6O4 44433387 Ki = 260 nM T72458 C92BPS 44433388 Ki = 67 nM T72458 CC7VN4 44433389 Ki = 110 nM T72458 CTZI97 44433391 Ki = 59 nM T72458 CVX59F 44433392 Ki = 68 nM T72458 CHS4F5 44433406 Ki = 78 nM T72458 CNY6A2 44433407 Ki = 75 nM T72458 CLD9V1 44433409 Ki = 100 nM T72458 CW7SE3 44433411 Ki = 65 nM T72458 CJ20VN 44433413 Ki = 220 nM T72458 C39SZC 44433417 Ki = 31 nM T72458 CAZI23 44433418 Ki = 260 nM T72458 C6JPQ5 44433419 Ki = 250 nM T72458 CEGB56 44433420 Ki = 540 nM T72458 CFL4Z1 44433421 Ki = 350 nM T72458 CUM4N7 44433422 Ki = 160 nM T72458 C06KHC 44433423 Ki = 12 nM T72458 CG6O4A 44433424 Ki = 64 nM T72458 CKG92E 44433425 Ki = 200 nM T72458 CA6Z1R 44433426 Ki = 6.6 nM T72458 CTKI96 44433428 Ki = 12 nM T72458 CW8B6E 44433439 Ki = 8.6 nM T72458 C59IFV 44433441 Ki = 36 nM T72458 CI47FK 44433442 Ki = 15 nM T72458 CHG0X4 44433444 Ki = 18 nM T72458 CLJ9O6 44433445 Ki = 18 nM T72458 CZ7A5U 44433446 Ki = 5.4 nM T72458 C2T3MY 44433448 Ki = 21 nM T72458 C0OZ2S 44433450 Ki = 580 nM T72458 C7H8YL 44433455 Ki = 205 nM T72458 CO13HI 44433475 Ki = 43 nM T72458 C8NU0W 44433478 Ki = 81 nM T72458 CJ2D4S 44433479 Ki = 32 nM T72458 C5X8MW 44433480 Ki = 26 nM T72458 C9OZF5 44433481 Ki = 9.3 nM T72458 CAD9F7 44433482 Ki = 94 nM T72458 CH3KR5 44433483 Ki = 340 nM T72458 CQI17F 44433484 Ki = 98 nM T72458 C68VOP 44433561 Ki = 74 nM T72458 CYCP31 44433562 Ki = 26 nM T72458 CTF0P5 44433563 Ki = 4.5 nM T72458 CZQ3I4 44433564 Ki = 610 nM T72458 CLQI91 44434545 Ki = 39 nM T72458 C6DK3A 44434546 Ki = 1.8 nM T72458 C70WCO 44434547 Ki = 1.8 nM T72458 C2DH7G 44434548 Ki = 1 nM T72458 CHU9Q7 44434549 Ki = 10 nM T72458 C28NVB 44434550 Ki = 0.8 nM T72458 C4KQ0A 44434551 Ki = 26 nM T72458 C9M2BQ 44434552 Ki = 47 nM T72458 CVW3Q1 44434553 Ki = 3.3 nM T72458 CD5G6X 44434554 Ki = 49 nM T72458 CKN63U 44434555 Ki = 2.5 nM T72458 C52DTH 44434556 Ki = 29 nM T72458 C2WS3C 44434557 Ki = 7.5 nM T72458 CX6KL8 44434558 Ki = 6 nM T72458 CA39RJ 44434559 Ki = 3.3 nM T72458 C8HG1P 44434560 Ki = 7.1 nM T72458 C8Z1IM 44434561 Ki = 78000 nM T72458 C5C6IA 44434562 Ki = 0.8 nM T72458 CCP2N5 44434563 Ki = 2.3 nM T72458 C6KPV5 44434568 Ki = 4.5 nM T72458 C2K9TI 44434570 Ki = 106000 nM T72458 CKL0H4 44434572 Ki = 5800 nM T72458 CO0N2A 44434575 Ki = 8.8 nM T72458 CRJN03 44434579 Ki = 38 nM T72458 CKI3L6 44434580 Ki = 21000 nM T72458 CBC27H 44434581 Ki = 10000 nM T72458 C51NSB 44434584 Ki = 4900 nM T72458 CF2S6P 44434587 Ki = 2400 nM T72458 CQ81UI 44434592 Ki = 19000 nM T72458 CP2A4G 44434595 Ki = 9800 nM T72458 CT20IC 44434597 Ki = 164000 nM T72458 CC1H3U 44434598 Ki = 32000 nM T72458 CH17AO 44434599 Ki = 23000 nM T72458 CAID38 44434600 Ki = 81000 nM T72458 CGN1P8 44434601 Ki = 6400 nM T72458 CDV61Y 44434603 Ki = 7000 nM T72458 CZPC57 44434605 Ki = 14000 nM T72458 C5DT7Q 44434611 Ki = 11000 nM T72458 C3MS2D 44434613 Ki = 21000 nM T72458 C5A1GF 44434614 Ki = 16000 nM T72458 CN4D2E 44434616 Ki = 158000 nM T72458 C1B5RV 44434621 Ki = 10000 nM T72458 C5TMA6 44434625 Ki = 222000 nM T72458 C9XG2K 44434631 Ki = 165000 nM T72458 CY2C7G 44434632 Ki = 18000 nM T72458 CQ94YK 44434633 Ki = 5400 nM T72458 CM1NA8 44434634 Ki = 7100 nM T72458 C93NCL 44434635 Ki = 17000 nM T72458 CZ8TO1 44434636 Ki = 6200 nM T72458 CQ06DV 44434637 Ki = 77000 nM T72458 C0SM2J 44434647 Ki = 14000 nM T72458 C9GIF5 44434648 Ki = 9400 nM T72458 CTQ16K 44434649 Ki = 8400 nM T72458 C15MAF 44434650 Ki = 8100 nM T72458 CWD27I 44434651 Ki = 7100 nM T72458 C6X8WB 44434652 Ki = 16000 nM T72458 CWU74N 44434653 Ki = 2300 nM T72458 CXN0M3 44434654 Ki = 59000 nM T72458 CM0VZ8 44434655 Ki = 4700 nM T72458 CP0V1N 44434656 Ki = 99000 nM T72458 CV5Y3N 44434657 Ki = 13000 nM T72458 CVC93Q 44434658 Ki = 21000 nM T72458 CWE1V4 44434659 Ki = 96000 nM T72458 C5WR3A 44434661 Ki = 14000 nM T72458 CJ27QL 44434662 Ki = 6400 nM T72458 C6US7A 44434663 Ki = 5000 nM T72458 C4ZD1B 44434664 Ki = 87000 nM T72458 C03NKU 44434665 Ki = 44000 nM T72458 CJ2AT0 44434666 Ki = 5900 nM T72458 CF41SX 44434682 Ki = 3800 nM T72458 C9IWD4 44434683 Ki = 11000 nM T72458 CJ03PB 44434684 Ki = 3400 nM T72458 CIH0Z6 44434685 Ki = 3700 nM T72458 C4POB8 44434686 Ki = 9800 nM T72458 C1GFE6 44434687 Ki = 7400 nM T72458 C3J7WI 44434688 Ki = 3800 nM T72458 C9Y0BM 44434689 Ki = 17000 nM T72458 CH6LA5 44434690 Ki = 2000 nM T72458 CPRE40 44434691 Ki = 3700 nM T72458 C9O8LX 44434692 Ki = 2400 nM T72458 CE2Z3V 44434693 Ki = 2100 nM T72458 C31LUY 44434694 Ki = 2100 nM T72458 C9C4BN 44434695 Ki = 3700 nM T72458 CF3JX5 44434696 Ki = 1500 nM T72458 CM51SC 44434697 Ki = 2200 nM T72458 CA2FQ4 44434698 Ki = 2700 nM T72458 CTC18P 44434699 Ki = 4300 nM T72458 CQT85W 44434700 Ki = 4500 nM T72458 C8BQ7C 44434701 Ki = 3000 nM T72458 CV2QW3 44434702 Ki = 3400 nM T72458 C9IY3A 44434703 Ki = 2300 nM T72458 CF8J2P 44434704 Ki = 4100 nM T72458 CH7QD5 44434706 Ki = 2100 nM T72458 CT4FO2 44434707 Ki = 1900 nM T72458 C9E4PO 44434709 Ki = 4400 nM T72458 C7LUV2 44434713 Ki = 4100 nM T72458 CR70OD 44434714 Ki = 5600 nM T72458 CA1BF3 44434715 Ki = 4800 nM T72458 C0N4CY 44434753 Ki = 2500 nM T72458 CS1KG4 44434754 Ki = 6400 nM T72458 C2JHP0 44434757 Ki = 3200 nM T72458 CZ43DV 44434758 Ki = 1300 nM T72458 C50PIJ 44434759 Ki = 5600 nM T72458 CKAQ59 44434760 Ki = 2800 nM T72458 CALF38 44434761 Ki = 14000 nM T72458 C17HCY 44434762 Ki = 1500 nM T72458 CX75CS 44434763 Ki = 1900 nM T72458 CNB68V 44434764 Ki = 2300 nM T72458 CZ0R9M 44434765 Ki = 1900 nM T72458 CU9C0K 44434766 Ki = 1600 nM T72458 C8IHB1 44434767 Ki = 2400 nM T72458 C27KYV 44434768 Ki = 2600 nM T72458 CEM27N 44434769 Ki = 5300 nM T72458 CB7A2G 44434770 Ki = 3000 nM T72458 C0Y3IG 44434771 Ki = 3000 nM T72458 CNL2T3 44434772 Ki = 3200 nM T72458 CUW4Y6 44434778 Ki = 3400 nM T72458 CH8WT0 44434780 Ki = 12000 nM T72458 CL9K2D 44434781 Ki = 2600 nM T72458 CJ12GC 44434782 Ki = 9200 nM T72458 CFBX46 44434785 Ki = 7800 nM T72458 C0KB8P 44434787 Ki = 7400 nM T72458 C0M2VI 44434790 Ki = 179000 nM T72458 CH3UV8 44434794 Ki = 149000 nM T72458 C10VDG 44434797 Ki = 179000 nM T72458 CWN02S 44434799 Ki = 150000 nM T72458 C0X1MK 44434821 Ki = 6000 nM T72458 CU1ON8 44434828 Ki = 182000 nM T72458 CBHU73 44434839 Ki = 116000 nM T72458 C20UIF 44434841 Ki = 96000 nM T72458 CA7P5L 44434843 Ki = 3400 nM T72458 CBL2D7 44434845 Ki = 3400 nM T72458 CYE25C 44434847 Ki = 38000 nM T72458 CWE0J6 44434848 Ki = 7700 nM T72458 CB39YP 44434849 Ki = 33000 nM T72458 C0ZV6S 44434850 Ki = 11000 nM T72458 C4U6LJ 44434851 Ki = 7300 nM T72458 CA4M3C 44434853 Ki = 116000 nM T72458 CVGW87 44434854 Ki = 3100 nM T72458 C3G5QO 44434855 Ki = 1200 nM T72458 C2JET5 44434856 Ki = 9200 nM T72458 C2M5VB 44434857 Ki = 16000 nM T72458 CS30KD 44434858 Ki = 25000 nM T72458 C7S1OK 44434859 Ki = 11000 nM T72458 C3AVB5 44434860 Ki = 3200 nM T72458 CZQI93 44434861 Ki = 8400 nM T72458 CC0U5Y 44434862 Ki = 2500 nM T72458 CWTI58 44434863 Ki = 4400 nM T72458 CFOM13 44434864 Ki = 7300 nM T72458 CL97ID 44434865 Ki = 18000 nM T72458 CW93VX 44434867 Ki = 5300 nM T72458 CN36OD 44434868 Ki = 6500 nM T72458 CI09FJ 44434870 Ki = 2100 nM T72458 CZE48F 44434872 Ki = 5700 nM T72458 CXTV37 44434880 Ki = 3700 nM T72458 CQ45JU 44434884 Ki = 3600 nM T72458 C8POL0 44435184 Ki = 44 nM T72458 CZ8H3M 44435220 Ki = 4800 nM T72458 CPM80E 44441633 EC50 = 189 nM T72458 C7XC6E 44441634 IC50 = 1490 nM T72458 CU93IR 44441635 IC50 = 759 nM T72458 CD25AP 44441636 IC50 = 22.2 nM T72458 CQL07M 44441637 EC50 = 827 nM T72458 CIJ89K 44441638 IC50 = 173 nM T72458 CEHV41 44441639 EC50 = 196 nM T72458 C5D6YN 44441641 EC50 = 3.2 nM T72458 CP4TW0 44441642 IC50 = 6 nM T72458 CDC3R8 44441643 EC50 = 21 nM T72458 CU6ZN4 44441644 EC50 = 3.9 nM T72458 CNS4O1 44441645 EC50 = 28.7 nM T72458 CRL83D 44441646 EC50 = 111 nM T72458 C7EQ6Z 44441647 EC50 = 4.9 nM T72458 CHSV38 44441648 EC50 = 157 nM T72458 C3MIO4 44441681 EC50 = 6.5 nM T72458 CV3FT6 44441682 EC50 = 2174 nM T72458 CL93VK 44441683 EC50 = 563 nM T72458 CT3J4B 44441684 EC50 = 10 nM T72458 C3YRT9 44441685 EC50 = 546 nM T72458 CXQ3K8 44441686 EC50 = 151 nM T72458 CCS5T3 44441687 EC50 = 57.8 nM T72458 CHPU36 44441688 EC50 = 84.6 nM T72458 C9DT1C 44441689 EC50 = 1769 nM T72458 CV7BA9 44442899 Ki = 1200 nM T72458 CT3SE2 44442900 Ki = 510 nM T72458 CH8V0J 44442901 Ki = 340 nM T72458 C36JQH 44442902 Ki = 330 nM T72458 C92TFW 44442903 Ki = 310 nM T72458 C8R1KD 44442914 Ki = 300 nM T72458 CKPD40 44442931 Ki = 26 nM T72458 C6XZ1C 44442934 Ki = 38 nM T72458 CP4ZK7 44442941 Ki = 75 nM T72458 C3VJ6X 44442942 Ki = 37 nM T72458 C5PN4K 44442943 Ki = 22 nM T72458 COG72A 44442944 Ki = 130 nM T72458 CV7N5C 44442954 EC50 = 110 nM T72458 CY4E6X 44442956 EC50 = 230 nM T72458 CQ5KH1 44442958 Ki = 390 nM T72458 C7I2UT 44442965 Ki = 11 nM T72458 C45FRV 44442972 Ki = 220 nM T72458 C31FJZ 44442977 Ki = 76 nM T72458 CF6L4W 44442978 Ki = 35 nM T72458 CYMC97 44442981 Ki = 27 nM T72458 C7AD4H 44442985 Ki = 1200 nM T72458 C7Y0HL 44442989 Ki = 690 nM T72458 CYF4D6 44442990 Ki = 140 nM T72458 C6U3VA 44442992 Ki = 100 nM T72458 CUE72J 44442995 Ki = 17 nM T72458 CZ60QW 44442997 Ki = 5.5 nM T72458 C8EL0V 44442998 Ki = 29 nM T72458 C8ZU6S 44442999 Ki = 190 nM T72458 CJZ87H 44443000 Ki = 210 nM T72458 C03CKQ 44443001 Ki = 190 nM T72458 C7JY2F 44443002 Ki = 210 nM T72458 C10XIQ 44443003 Ki = 180 nM T72458 CKT6L8 44443004 Ki = 100 nM T72458 CY7H8L 44443005 Ki = 430 nM T72458 CY0GI2 44443006 Ki = 110 nM T72458 CB8R0W 44443007 Ki = 670 nM T72458 CC63OG 44443008 Ki = 200 nM T72458 CJK49H 44443009 Ki = 2200 nM T72458 C2D0OW 44443010 Ki = 3000 nM T72458 C83IEK 44443011 Ki = 3100 nM T72458 CZLT13 44443012 Ki = 4600 nM T72458 CKW85I 44443013 Ki = 3400 nM T72458 C98VGZ 44443014 Ki = 12 nM T72458 C0W5BQ 44443015 Ki = 25 nM T72458 CAU09V 44443016 Ki = 62 nM T72458 CC4RD1 44443017 Ki = 140 nM T72458 CCW51A 44443018 Ki = 110 nM T72458 C50KLT 44443019 Ki = 24 nM T72458 C7FU9B 44443020 Ki = 30 nM T72458 C47OXH 44443021 Ki = 44 nM T72458 CG7J0H 44443022 Ki = 90 nM T72458 CU5AM8 44443023 Ki = 3.6 nM T72458 CM80SQ 44443024 Ki = 130 nM T72458 C68ESY 44443025 Ki = 52 nM T72458 CZ3K8H 44443026 Ki = 29 nM T72458 C2VCS6 44443027 Ki = 65 nM T72458 CQU1O9 44443028 Ki = 32 nM T72458 CO90XC 44443029 Ki = 27 nM T72458 CGZ71H 44443030 Ki = 2.1 nM T72458 CLT7M0 44443031 Ki = 11 nM T72458 CBYR70 44443032 Ki = 16 nM T72458 CO51HP 44443033 Ki = 1.8 nM T72458 CQ68UV 44443034 Ki = 8.3 nM T72458 CO93SX 44443035 Ki = 0.5 nM T72458 C0WH1X 44443036 Ki = 110 nM T72458 C9IZ0Y 44443037 Ki = 190 nM T72458 C1GJ5L 44443038 Ki = 1800 nM T72458 CF2UI0 44443039 Ki = 2800 nM T72458 CR40SE 44443040 Ki = 1300 nM T72458 C8HOB9 44443041 Ki = 750 nM T72458 CRUJ10 44443042 Ki = 1300 nM T72458 CXI2N5 44443043 Ki = 2700 nM T72458 CM2P9T 44443044 Ki = 1500 nM T72458 C8JA5O 44444425 Ki = 520 nM T72458 CK79AB 44444427 Ki = 4800 nM T72458 C5N4FT 44444429 Ki = 1150 nM T72458 CDWO25 44444430 Ki = 1100 nM T72458 C7B9FO 44444431 Ki = 1700 nM T72458 C6DGU3 44444432 Ki = 220 nM T72458 CTD12E 44444433 Ki = 280 nM T72458 C0V8UC 44444434 Ki = 250 nM T72458 CWGI62 44444435 Ki = 580 nM T72458 C73MYX 44444436 Ki = 320 nM T72458 C2QC4X 44444437 Ki = 420 nM T72458 CHOG98 44444438 Ki = 490 nM T72458 CQ37OR 44444440 Ki = 1200 nM T72458 C02WEC 44444441 Ki = 1200 nM T72458 C92TOP 44444442 Ki = 1100 nM T72458 CDS4U1 44444443 Ki = 320 nM T72458 C6M3VD 44444444 Ki = 550 nM T72458 C9WP5E 44444445 Ki = 950 nM T72458 CUG3B4 44444446 Ki = 360 nM T72458 CL31BQ 44444447 Ki = 840 nM T72458 C0EA1Z 44444448 Ki = 92 nM T72458 CGEZ90 44444449 Ki = 510 nM T72458 C98HTN 44444450 Ki = 230 nM T72458 CFN72H 44444452 Ki = 270 nM T72458 CT69RO 44444454 Ki = 520 nM T72458 CU24DB 44444457 Ki = 240 nM T72458 CYO9U6 44444460 Ki = 190 nM T72458 CL6TV9 44444462 Ki = 1600 nM T72458 CPJI69 44444465 Ki = 1400 nM T72458 C60GBK 44444468 Ki = 450 nM T72458 CQCK08 44444483 Ki = 13 nM T72458 C4ZDW3 44444490 Ki = 47 nM T72458 CB39DL 44444493 Ki = 7.1 nM T72458 CE5CR4 44444495 Ki = 4.7 nM T72458 CBO36Z 44444497 Ki = 11 nM T72458 CIOT60 44444499 Ki = 4.4 nM T72458 C5DWM0 44444500 EC50 = 6.9 nM T72458 C3VL8P 44444502 Ki = 8.9 nM T72458 CD7N9T 44444504 Ki = 7.7 nM T72458 CL17PU 44444505 Ki = 17.3 nM T72458 CDWM65 44444507 Ki = 4.9 nM T72458 C3PST9 44444508 Ki = 47 nM T72458 CIE0P1 44444509 Ki = 10 nM T72458 COS36P 44444510 EC50 = 6.6 nM T72458 C2YX7D 44444511 Ki = 87 nM T72458 CXT65M 44447207 Ki = 810 nM T72458 C7X9AU 44447208 Ki = 280 nM T72458 CVS9K1 44447209 Ki = 130 nM T72458 CY19GE 44447210 Ki = 170 nM T72458 CL03RO 44447211 Ki = 130 nM T72458 CVR68Z 44447212 Ki = 250 nM T72458 COI65T 44447214 Ki = 120 nM T72458 C9PYC4 44447218 Ki = 230 nM T72458 CNJ3I2 44447221 Ki = 38 nM T72458 C9JN4F 44447222 Ki = 170 nM T72458 C4HB7O 44447223 Ki = 190 nM T72458 CT6R7Z 44447224 Ki = 100 nM T72458 CEF6Y1 44447225 Ki = 180 nM T72458 CEK98D 44447226 Ki = 280 nM T72458 CDYL03 44447227 Ki = 71 nM T72458 CW27UZ 44447228 Ki = 260 nM T72458 C8GJI0 44447229 Ki = 290 nM T72458 CY2E8N 44447230 Ki = 180 nM T72458 C3MB7S 44447231 Ki = 330 nM T72458 CS2P5V 44447232 Ki = 200 nM T72458 C8DTJ1 44447233 Ki = 280 nM T72458 CV85GR 44447234 Ki = 74 nM T72458 CG02YX 44447235 Ki = 87 nM T72458 C4APF9 44447236 Ki = 110 nM T72458 CG3W0E 44447237 Ki = 380 nM T72458 CM68RP 44447238 Ki = 37 nM T72458 C60TVF 44447239 Ki = 790 nM T72458 CJ6ZW7 44447240 Ki = 40 nM T72458 CN2X1M 44447241 Ki = 30 nM T72458 CLHT47 44447242 Ki = 28 nM T72458 CYGJ75 44447243 Ki = 410 nM T72458 C9VME8 44447244 Ki = 590 nM T72458 CIS36F 44447245 Ki = 120 nM T72458 CAD46C 44447246 Ki = 1100 nM T72458 CG0L1J 44447247 Ki = 2100 nM T72458 C73SEZ 44447248 Ki = 480 nM T72458 CHO8Y4 44447249 Ki = 43 nM T72458 CG3FA6 44447250 Ki = 10 nM T72458 C0WQO6 44447251 EC50 = 2 nM T72458 C2F7YZ 44447764 Ki = 550 nM T72458 C8MK6X 44447765 Ki = 340 nM T72458 C8Q7FC 44447767 Ki = 98 nM T72458 C8OG4F 44447768 Ki = 96 nM T72458 CE1G2K 44447769 Ki = 190 nM T72458 CM8F0V 44447770 Ki = 110 nM T72458 CS80GC 44447771 Ki = 560 nM T72458 CWN9X8 44447772 Ki = 56 nM T72458 C4A7BL 44447773 Ki = 52 nM T72458 C9MVL5 44447774 Ki = 160 nM T72458 CPL5B2 44447776 Ki = 110 nM T72458 CQ8BE5 44447777 Ki = 11 nM T72458 C6V5UQ 44447778 Ki = 120 nM T72458 C9NXS5 44447779 Ki = 7.2 nM T72458 C8YZ0G 44447780 Ki = 17 nM T72458 CAK75F 44447781 Ki = 53 nM T72458 CVUW60 44447785 Ki = 11 nM T72458 C86ATQ 44447787 Ki = 130 nM T72458 C3V9UN 44447791 Ki = 12 nM T72458 C9O7VQ 44447801 Ki = 94 nM T72458 CU7S8G 44447802 Ki = 74 nM T72458 C5SY1J 44447803 Ki = 18 nM T72458 CCRY28 44447804 Ki = 6.5 nM T72458 CWDG08 44447805 Ki = 190 nM T72458 C0C7VJ 44447806 Ki = 40 nM T72458 C7QT3I 44447807 Ki = 45 nM T72458 C6KPH5 44447808 Ki = 97 nM T72458 CQLZ83 44447809 Ki = 330 nM T72458 C9KNO3 44447810 Ki = 54 nM T72458 C4X7YK 44447811 Ki = 1800 nM T72458 C3L4FZ 44447812 Ki = 78 nM T72458 C4OWP8 44447816 Ki = 180 nM T72458 C5MF9J 44447817 Ki = 79 nM T72458 CFL6R4 44447818 Ki = 92 nM T72458 CXAF32 44447819 Ki = 62 nM T72458 C37AZY 44447820 Ki = 52 nM T72458 C9OBG6 44447821 Ki = 55 nM T72458 CB3KW6 44447822 Ki = 59 nM T72458 CDX4V1 44447823 Ki = 42 nM T72458 CB1GF4 44447824 Ki = 68 nM T72458 C14OSV 44447847 IC50 = 2400 nM T72458 C03AQC 44447849 IC50 = 1500 nM T72458 CR1M0J 44447851 IC50 = 960 nM T72458 CRI7M8 44448436 IC50 = 127.6 nM T72458 C6I4PC 44448477 IC50 = 101.1 nM T72458 C08BMY 44448479 EC50 = 120.5 nM T72458 C2FA5H 44448480 EC50 = 1922 nM T72458 CWB1I0 44448515 IC50 = 28.1 nM T72458 CP35SZ 44448554 IC50 = 22.7 nM T72458 C8TK3Y 44448588 IC50 = 9.8 nM T72458 C0C7KI 44448590 EC50 = 4.6 nM T72458 CMYO10 44448628 IC50 = 37.2 nM T72458 CQHR95 44448629 EC50 = 2.1 nM T72458 C78XDT 44448631 EC50 = 13.4 nM T72458 C8H1UT 44448660 EC50 = 2.8 nM T72458 CCV7B1 44448661 EC50 = 110.8 nM T72458 CL28KE 44448677 IC50 = 82.2 nM T72458 CGZ1F9 44448698 EC50 = 155.6 nM T72458 CYAN15 44449216 EC50 = 565 nM T72458 CTP3D6 44453826 Ki > 100000 nM T72458 C4FV3C 44453850 Ki > 25000 nM T72458 CEI35V 44453902 Ki = 6700 nM T72458 CUPG04 44453903 EC50 > 25000 nM T72458 CBV08D 44455891 Ki = 290 nM T72458 C9L0JY 44455892 Ki = 260 nM T72458 CH1DK5 44455893 Ki = 51 nM T72458 C9GLW5 44455922 Ki = 7.5 nM T72458 CW2PJ8 44455923 Ki = 2050 nM T72458 CAK1U0 44455956 Ki = 470 nM T72458 CF3W1O 44455957 Ki = 560 nM T72458 C92TBV 44455958 Ki = 61 nM T72458 CSVD47 44455996 Ki = 370 nM T72458 CN89EI 44455997 Ki = 3700 nM T72458 CP2EH4 44456027 Ki = 5.3 nM T72458 CH5BY0 44456102 Ki = 1 nM T72458 CI1PL0 44456137 Ki = 2.1 nM T72458 CCW1A3 44456138 Ki = 7.3 nM T72458 CE9VC8 44456183 Ki = 2.2 nM T72458 CD8EJ4 44456184 Ki = 2 nM T72458 C63APB 44456219 Ki = 4.7 nM T72458 CE0P7K 44456222 Ki = 1 nM T72458 CF40UY 44456259 Ki = 5.3 nM T72458 CFD8Z5 44456304 Ki = 4.6 nM T72458 CFD62Q 44456336 Ki = 7.6 nM T72458 C8N0CX 44456368 Ki = 90 nM T72458 CM69AH 44456410 Ki = 7.2 nM T72458 CGLM70 44456416 Ki = 850 nM T72458 C6GL4V 44456460 Ki = 7800 nM T72458 CU7JV8 44456461 Ki = 250 nM T72458 CC64AO 44457043 IC50 = 100 nM T72458 CZ36WX 44457067 IC50 = 60 nM T72458 C4DL5C 44469677 IC50 > 10000 nM T72458 CA5MU1 44562283 Ki = 1700 nM T72458 C27VXC 44562284 Ki = 5800 nM T72458 CA1GN0 44562285 Ki > 10000 nM T72458 C7Z4UN 44562286 Ki = 13 nM T72458 C5CIX6 44562287 Ki = 9.4 nM T72458 C4PR2V 44562288 Ki = 18 nM T72458 C8QL9K 44562289 Ki = 65 nM T72458 C4JKU5 44562323 Ki > 10000 nM T72458 CNF96U 44562324 Ki = 38 nM T72458 COB0Q8 44562361 Ki = 110 nM T72458 C8VGJ4 44562362 Ki = 380 nM T72458 C7B3HD 44562363 Ki = 330 nM T72458 C6JX0A 44562364 Ki = 89 nM T72458 C02QLT 44562365 Ki = 1400 nM T72458 CF5W2K 44562366 Ki = 42 nM T72458 CLFX67 44562367 Ki = 390 nM T72458 CAF74R 44562368 Ki = 110 nM T72458 CHN87Y 44562389 Ki = 3200 nM T72458 C1ZH5L 44562390 Ki > 10000 nM T72458 CA6ZN2 44562391 Ki = 53 nM T72458 CQ8Z5M 44562392 Ki = 83 nM T72458 CKB04G 44562398 Ki = 21 nM T72458 CEQ6Y1 44562399 Ki = 15 nM T72458 C18SIO 44562400 Ki = 120 nM T72458 CSC76I 44562401 Ki = 350 nM T72458 C0SD6C 44562402 Ki = 2 nM T72458 C21YKQ 44562412 Ki = 350 nM T72458 CL6ZR3 44562413 Ki = 1200 nM T72458 CU92FG 44562414 Ki = 24 nM T72458 C93SKQ 44562421 Ki = 33 nM T72458 CA53WV 44562422 Ki = 31 nM T72458 CN3Y7I 44562423 Ki = 26 nM T72458 C5F3XU 44562424 Ki = 110 nM T72458 C9SVX4 44562438 Ki = 91 nM T72458 CCIS23 44562439 Ki = 13 nM T72458 CPSC21 44562440 Ki = 8.3 nM T72458 CTN82A 44562457 Ki = 16 nM T72458 CSVX92 44562458 Ki = 46 nM T72458 CU98AG 44562459 Ki = 21 nM T72458 CQ0I1K 44562460 Ki = 3.2 nM T72458 CY14WQ 44562475 Ki = 2 nM T72458 CQV9B7 44562476 Ki = 1.7 nM T72458 C0VXR6 44562477 Ki = 4.2 nM T72458 C8EQD4 44562478 Ki = 7.7 nM T72458 CAM86F 44562495 Ki = 4.7 nM T72458 CAG1U4 44562496 Ki = 870 nM T72458 C4XFR3 44562497 Ki = 26 nM T72458 CRQW35 44562498 Ki = 110 nM T72458 C7V4WX 44562518 Ki = 29 nM T72458 CXDB43 44562519 Ki = 47 nM T72458 CP98CO 44562520 Ki = 54 nM T72458 CB18VE 44562538 Ki = 66 nM T72458 C8RQE4 44562539 Ki = 66 nM T72458 CF9N1W 44562540 Ki = 32 nM T72458 C94MEZ 44562541 Ki = 23 nM T72458 C0L6BJ 44562558 Ki = 11 nM T72458 CH42ZU 44562559 Ki = 11 nM T72458 CQ3J2B 44562560 Ki = 280 nM T72458 C2L6FI 44562561 Ki = 9 nM T72458 CV79ML 44562593 Ki > 10000 nM T72458 C1WU4Q 44562594 Ki = 560 nM T72458 C0GTB1 44562595 Ki = 230 nM T72458 C5OJ6B 44562596 Ki = 150 nM T72458 CK5WI0 44562597 Ki = 28 nM T72458 C3NSL9 44562598 Ki = 49 nM T72458 C6ILB9 44562599 Ki = 26 nM T72458 CQ8J9K 44569175 EC50 = 2 nM T72458 CL8GU3 44569176 EC50 = 0.9 nM T72458 C97DSW 44577054 Ki = 83 nM T72458 C2FP9E 44577055 Ki = 210 nM T72458 CP56CV 44577056 Ki = 180 nM T72458 C4WP0Z 44577059 Ki = 5.3 nM T72458 CD3T1I 44577060 Ki = 7.5 nM T72458 CQ1M9C 44577061 Ki = 3.1 nM T72458 C6FI8E 44577062 Ki = 4.1 nM T72458 CJ6GZ3 44577063 Ki = 5.4 nM T72458 CHJ6Z1 44577064 Ki = 24 nM T72458 CY4QE9 44577087 Ki = 26 nM T72458 CGF37X 44577088 Ki = 27 nM T72458 CR6Q2S 44577089 Ki = 23 nM T72458 CWOK70 44577090 Ki = 10 nM T72458 C4FSH3 44577091 Ki = 3.4 nM T72458 CF8PL1 44577092 Ki = 1.1 nM T72458 CM6X5S 44577093 Ki = 0.8 nM T72458 CGTV08 44577094 Ki = 3.3 nM T72458 C0YI4V 44577095 Ki = 1.3 nM T72458 CEJ96P 44577510 EC50 = 37 nM T72458 C6Y1BS 44577515 IC50 > 5000 nM T72458 C8B1WR 44577520 IC50 > 1000 nM T72458 C3NSW7 44577523 IC50 > 1000 nM T72458 CR5ZS2 44583562 EC50 = 11 nM T72458 CWFB17 44583567 IC50 = 1.2 nM T72458 CO7X1P 45277088 Ki < 10000 nM T72458 C26EWX 45277089 Ki < 10000 nM T72458 C6X4ER 45277090 Ki < 10000 nM T72458 CH7I1J 45277245 Ki < 10000 nM T72458 CHWX12 46202887 EC50 > 10000 nM T72458 CXM2I4 46202891 EC50 = 53 nM T72458 CM68TW 46202892 EC50 = 108 nM T72458 CCE2L7 46203212 EC50 = 644 nM T72458 C02XLV 46203213 EC50 = 3630 nM T72458 C4N2CP 46203214 EC50 = 11100 nM T72458 CJB6H0 46203215 Ki = 107 nM T72458 CKA84X 46203216 EC50 = 147 nM T72458 CO8H3A 46203515 EC50 = 51 nM T72458 CO95IX 46203516 EC50 = 69 nM T72458 CVW98L 46203517 EC50 = 40 nM T72458 CY12SB 46228659 EC50 > 30000 nM T72458 C10VXP 46228660 EC50 = 338.84 nM T72458 C8XUS4 46228689 EC50 = 794.33 nM T72458 C5FVJ9 46228690 EC50 = 100 nM T72458 CCK7I1 46228725 EC50 > 30000 nM T72458 CD5Q8V 46228726 EC50 = 1071.52 nM T72458 CJ7R0X 46228763 EC50 > 30000 nM T72458 CYD2R3 46228764 EC50 = 1258.93 nM T72458 CQ53EA 46228813 EC50 = 2884.03 nM T72458 CMX28H 46228814 EC50 = 1047.13 nM T72458 C7FAY5 46228815 EC50 = 660.69 nM T72458 C82NVP 46228841 EC50 > 30000 nM T72458 CEDL84 46228842 EC50 > 30000 nM T72458 CP86QH 46228843 EC50 > 30000 nM T72458 C4BD8Z 46228844 EC50 > 30000 nM T72458 CR6PF0 46228845 EC50 > 30000 nM T72458 CCN14H 46228846 EC50 = 165.96 nM T72458 C3T1NY 46228847 EC50 > 30000 nM T72458 COW85F 46228848 EC50 > 30000 nM T72458 CZLY24 46228849 EC50 > 30000 nM T72458 C5VAN7 46228850 EC50 > 30000 nM T72458 C0X9KS 46228888 EC50 > 30000 nM T72458 CDE7N9 46865980 EC50 = 3900 nM T72458 CBI76Q 46884747 IC50 = 89 nM T72458 CQ28TZ 46884748 EC50 = 37.2 nM T72458 CD3E4C 46885323 Ki = 264 nM T72458 CNH0I9 46885324 EC50 = 255 nM T72458 C53CEM 46885325 EC50 = 159 nM T72458 CPKC94 46885326 EC50 = 288 nM T72458 C65EKV 46885366 EC50 = 19 nM T72458 CNW43Y 46885367 EC50 = 55 nM T72458 CE4SF8 46885368 EC50 = 105 nM T72458 C4YX1U 46885369 EC50 = 73 nM T72458 CLY30Q 46885414 EC50 = 81 nM T72458 CV23JL 46885415 EC50 = 32 nM T72458 C7M3HS 46885416 EC50 = 374 nM T72458 CHPS01 46885417 EC50 = 18 nM T72458 C4SVE1 46885480 EC50 = 15 nM T72458 C5QI7J 46885481 EC50 = 5 nM T72458 COU5X2 46885482 EC50 = 6 nM T72458 CU28GA 46885483 EC50 = 4 nM T72458 CG9NJ1 46885523 EC50 = 7 nM T72458 CS90MN 46885524 EC50 = 21 nM T72458 CWI08O 46885525 EC50 = 89 nM T72458 CQ94VM 46885526 EC50 = 82 nM T72458 C90ABZ 46885558 EC50 = 4 nM T72458 C0U7TG 46885559 EC50 = 117 nM T72458 C0MI3C 46885560 EC50 = 243 nM T72458 C50BUQ 46885561 EC50 = 111 nM T72458 CL86JU 46885621 EC50 = 15 nM T72458 CFJ0C1 46885622 EC50 = 220 nM T72458 CX4K9T 46885674 EC50 = 1116 nM T72458 C0Y9NF 46885711 EC50 = 30 nM T72458 C3O5BR 46885712 EC50 = 18 nM T72458 CA82IZ 46885713 EC50 = 347 nM T72458 CG6XN0 46885759 EC50 = 6 nM T72458 CK8D6G 46885760 EC50 = 45 nM T72458 C0C8GN 46885761 EC50 = 62 nM T72458 CY30PG 46885815 EC50 = 46 nM T72458 CEA70O 46885816 EC50 = 126 nM T72458 C6ZUB5 46885817 EC50 = 626 nM T72458 C8LHF6 46885861 EC50 = 962 nM T72458 CAZN09 46885862 EC50 = 130 nM T72458 CWN89S 46885863 Ki = 346 nM T72458 CKQ4X2 46885906 EC50 = 85 nM T72458 C8UTI7 46885907 EC50 = 61 nM T72458 CFC5L1 46885972 EC50 = 69 nM T72458 CUDE25 46885973 EC50 = 91 nM T72458 C3FN1Z 46885974 EC50 = 52 nM T72458 CDH7N3 46886010 EC50 = 257 nM T72458 CO3S1Q 46905544 Ki = 31392 nM T72458 C96XEU 46905545 Ki = 4756 nM T72458 CDY4U0 46911588 EC50 = 2.1 nM T72458 C29LQB 46919520 EC50 = 2.7 nM T72458 CK41RF 46930942 Ki = 1300 nM T72458 CIGV98 46930943 Ki = 350 nM T72458 C8Y2QS 49798104 IC50 = 398.11 nM T72458 C6LEM8 49798106 IC50 = 31.62 nM T72458 C8EG6Y 49798111 IC50 = 1258.93 nM T72458 C24DUW 49798112 IC50 = 251.19 nM T72458 CQS6G8 49798149 IC50 = 200 nM T72458 C1EMQ2 49861348 EC50 = 12 nM T72458 C9QU3G 49862375 EC50 = 5.4 nM T72458 C4WHG2 49862376 EC50 = 10 nM T72458 CPZI97 49862377 EC50 = 6.4 nM T72458 CY7R2T 49862378 EC50 = 9.7 nM T72458 C7GA4I 49862425 EC50 = 19 nM T72458 C1BC2M 49862426 IC50 = 150 nM T72458 C2ZHD1 49862478 EC50 = 19 nM T72458 CN1AJ5 49862662 IC50 = 31.4 nM T72458 CT69NY 49862663 IC50 = 479.2 nM T72458 CW2KQ0 49862664 EC50 = 78.1 nM T72458 C1X3WL 49862665 EC50 = 2.6 nM T72458 CG78ZY 49862736 EC50 = 1.1 nM T72458 C8GVY6 49862737 IC50 = 52.5 nM T72458 C0N8IJ 49862738 IC50 = 6.6 nM T72458 C5MZ9X 49862739 IC50 = 11.9 nM T72458 CBIK17 49862740 IC50 = 44.3 nM T72458 CHX09I 49862741 IC50 = 7.6 nM T72458 CZVN53 49862742 EC50 = 17.1 nM T72458 C8M2TH 49862743 EC50 = 7.4 nM T72458 C9T8SI 49862744 IC50 = 150.7 nM T72458 C8XA3E 49862745 EC50 = 1.5 nM T72458 CEX17U 49862746 IC50 = 3.6 nM T72458 CA2RN4 49862747 IC50 = 2.3 nM T72458 CD5ZR4 49862748 EC50 = 0.6 nM T72458 CPVE31 49862749 EC50 = 3.1 nM T72458 CNY2L7 49862750 EC50 = 0.8 nM T72458 CV6YZ5 49862751 EC50 = 2.9 nM T72458 CFR38H 50899078 EC50 = 0.23 nM T72458 C0QD9I 51346770 Ki = 392 nM T72458 C30PGL 51346771 Ki = 403 nM T72458 CBQN64 52918026 EC50 = 22 nM T72458 CZ8P7W 52940633 EC50 = 14 nM T72458 CZG5F1 52941830 EC50 = 2.4 nM T72458 C5RGD8 52943036 EC50 = 1000 nM T72458 C3XP8F 52943061 IC50 = 1.3 nM T72458 CB71IN 52944242 EC50 = 4.2 nM T72458 CDZ3L2 52945472 IC50 = 1.9 nM T72458 CQN8V6 52947911 IC50 = 9.7 nM T72458 CG5TJ0 53240339 IC50 = 515 nM T72458 CQ7O3U 54584301 IC50 = 16 nM T72458 C8PIL3 54584302 EC50 = 58 nM T72458 CN6F2C 54586246 IC50 = 5.1 nM T72458 CEU0M6 54587278 IC50 = 0.78 nM T72458 CLB28F 56595060 Ki = 330 nM T72458 CF34IC 56659456 EC50 = 0.25 nM T72458 CM94BT 56659465 EC50 = 53 nM T72458 C8BF3M 56659466 EC50 = 0.91 nM T72458 C5V2RD 56659467 EC50 = 1.3 nM T72458 CN41CZ 56659468 EC50 = 4.3 nM T72458 CF3LR1 56662904 EC50 = 0.69 nM T72458 C27DXA 56662925 EC50 = 1.4 nM T72458 CNSK26 56662927 EC50 = 1.9 nM T72458 C8C9IS 56666386 EC50 = 0.37 nM T72458 C3OM7E 56666397 EC50 = 32 nM T72458 CYKJ48 56669816 EC50 = 28 nM T72458 CPT38A 56669817 IC50 = 12 nM T72458 CFU39L 56669819 EC50 = 0.59 nM T72458 CCLJ91 56669820 EC50 = 0.76 nM T72458 C8H9RM 56672278 IC50 = 4900 nM T72458 C2YB1Q 56673302 IC50 = 0.71 nM T72458 C69KAM 56673304 EC50 = 9.9 nM T72458 C1GI2N 56673305 EC50 = 1.1 nM T72458 CE7CI0 56676614 EC50 = 1.2 nM T72458 CJDZ96 56676631 IC50 = 2.5 nM T72458 C7VO5D 56676632 EC50 = 0.8 nM T72458 CJZ5V3 56676633 IC50 = 6.6 nM T72458 CYQ3A6 56676634 EC50 = 307 nM T72458 CA1Q8I 56676635 EC50 = 2.3 nM T72458 C9V7LA 56676638 EC50 = 0.38 nM T72458 CEA19V 56676639 EC50 = 1.1 nM T72458 CLB0G3 56679956 EC50 = 3.8 nM T72458 C47TEG 56679964 EC50 = 12 nM T72458 CAYG58 56679968 EC50 = 1 nM T72458 CP7UR2 56683296 EC50 = 2.9 nM T72458 C9VT6Z 56683297 EC50 = 4.2 nM T72458 CFBT37 56683299 EC50 = 1.6 nM T72458 CZ7WN1 56683300 EC50 = 1.7 nM T72458 CB96KR 56683301 EC50 = 0.98 nM T72458 CTSB57 56850936 Ki = 988 nM T72458 C1U2DB 56851057 Ki = 254 nM T72458 C2WAO4 57634921 EC50 = 2 nM T72458 C4VT5C 57634925 EC50 = 0.47 nM T72458 CKW2T0 57646411 EC50 = 0.04 nM T72458 C8F5XG 57646441 Ki = 0.12 nM T72458 CS2E3H 58658553 EC50 = 6.2 nM T72458 CH1LU3 58777892 Ki = 70 nM T72458 C5P1EC 58777970 Ki = 190 nM T72458 CBM78A 59077913 EC50 = 44 nM T72458 CD1C7S 60168008 Ki = 70 nM T72458 CP6V2L 70681741 Ki = 1800 nM T72458 CPJ3U7 70681742 Ki = 380 nM T72458 C3PS2N 70681743 Ki = 160 nM T72458 CS27GN 70682904 Ki = 36000 nM T72458 C73SKU 70682946 EC50 = 29 nM T72458 CBY2K9 70683600 IC50 = 29 nM T72458 C06RGO 70683847 Ki = 5500 nM T72458 C65FDK 70683848 Ki = 1000 nM T72458 C0O6QG 70685712 IC50 = 20 nM T72458 CCU8P0 70685980 Ki = 900 nM T72458 CAJ5U0 70685981 Ki = 1000 nM T72458 CP7J6R 70688108 Ki = 5500 nM T72458 C3O4SK 70688109 Ki = 6600 nM T72458 CEFQ39 70688110 Ki = 670 nM T72458 CNH4F5 70688111 Ki = 400 nM T72458 CPJ08L 70688853 Ki = 0.33 nM T72458 CU86WQ 70689887 IC50 = 24 nM T72458 CB2X0A 70689888 IC50 = 17 nM T72458 CMKH31 70690145 Ki = 5000 nM T72458 C63ULO 70690146 Ki = 5800 nM T72458 CPM3N9 70690147 Ki = 2600 nM T72458 C2T3GP 70690148 Ki = 6200 nM T72458 C81JGS 70692049 IC50 = 40 nM T72458 C2P3IN 70692050 EC50 = 18 nM T72458 COSQ85 70694364 Ki = 5300 nM T72458 C3G7MZ 70695694 EC50 = 110 nM T72458 C97FOR 70696210 IC50 = 25 nM T72458 C2O7TA 71449047 EC50 = 6.1 nM T72458 CH0F4A 71449048 EC50 > 10000 nM T72458 C1JN2M 71449119 EC50 = 13 nM T72458 CMS5R6 71449140 Ki = 166000 nM T72458 CJPX32 71449204 EC50 = 52 nM T72458 C93FSV 71450911 Ki = 89 nM T72458 C8IXY4 71450912 Ki = 150 nM T72458 CK43RW 71450919 Ki = 500 nM T72458 C6BK5F 71450920 Ki = 3900 nM T72458 CBP20G 71452716 EC50 = 25 nM T72458 CKCN10 71452720 IC50 = 16 nM T72458 C8JMR2 71452721 Ki = 49 nM T72458 C2AGS1 71452731 Ki = 950 nM T72458 CEB0P9 71452732 Ki = 2500 nM T72458 CNPI97 71452733 Ki = 700 nM T72458 CICH01 71452734 Ki = 410 nM T72458 CD94NF 71452735 Ki = 230 nM T72458 CV0J8X 71452824 IC50 = 20 nM T72458 CN4EJ2 71452825 IC50 = 8 nM T72458 CW8OE1 71452826 IC50 = 30 nM T72458 C50LPK 71454491 EC50 = 12 nM T72458 CV4ZM6 71454492 EC50 = 49 nM T72458 C3D7ZL 71454495 Ki = 78 nM T72458 COP19B 71454508 Ki = 150 nM T72458 CN58TM 71454509 Ki = 170 nM T72458 CNB53G 71454510 Ki = 50 nM T72458 CY16AM 71454518 Ki = 15000 nM T72458 CPX03G 71456219 IC50 = 3700 nM T72458 C07WXP 71456220 EC50 > 10000 nM T72458 CQPB08 71456236 EC50 = 16 nM T72458 C05GFW 71456243 Ki = 53 nM T72458 CNRV69 71456245 IC50 = 18 nM T72458 C3NS6M 71456246 EC50 = 740 nM T72458 C3E1NT 71456250 Ki = 1600 nM T72458 C5VH2T 71456251 Ki = 280 nM T72458 CA5GY9 71458041 EC50 = 8 nM T72458 CQZ48M 71458046 Ki = 240 nM T72458 CU17GR 71458055 Ki = 7700 nM T72458 C93UJT 71458056 Ki = 4800 nM T72458 C6WOE4 71458057 Ki = 240 nM T72458 CG89OM 71458058 Ki = 140 nM T72458 C1WR2D 71458059 Ki = 80 nM T72458 C6YR0U 71458117 IC50 > 10000 nM T72458 C3V0DA 71459896 EC50 = 45 nM T72458 CO8C4B 71459937 IC50 = 280 nM T72458 CJ52CU 71459938 IC50 = 22 nM T72458 CS9Y6R 71459941 Ki = 530 nM T72458 CCRG02 71459942 Ki = 180 nM T72458 CU2A1J 71461601 EC50 = 570 nM T72458 CUJS47 71461649 EC50 = 8.6 nM T72458 C3HLD7 71461652 IC50 = 560 nM T72458 C5J2CA 71461656 Ki = 2100 nM T72458 CECQ16 71461657 Ki = 4200 nM T72458 C24GWM 71461662 Ki = 70000 nM T72458 CZ94CM 71461730 IC50 = 0.89 nM T72458 C9E2DM 71717586 IC50 = 4900 nM T72458 CYA8G1 71717886 EC50 = 26 nM T72458 CPH79G 71769787 Ki = 1.8 nM T72458 CMH31J 71769905 Ki = 600 nM T72458 C8KS6E 71770031 Ki = 2.4 nM T72458 CWH6T3 72548703 IC50 = 0.21 nM T72458 CV8K5U 73345513 Ki = 4800 nM T72458 C4IAM6 73345514 Ki = 4.6 nM T72458 CG3H2F 73345549 IC50 = 30 nM T72458 C1A5SK 73345616 IC50 = 74 nM T72458 CI0DV9 73345617 IC50 > 5000 nM T72458 C62DYB 73345878 IC50 = 40 nM T72458 CYMH60 73347015 Ki = 1.5 nM T72458 C31UAJ 73347130 EC50 = 8 nM T72458 C7DYR4 73347133 EC50 = 2 nM T72458 CZ91TE 73347138 IC50 = 570 nM T72458 CK46SP 73347139 IC50 = 4700 nM T72458 CX9LF8 73347140 IC50 = 990 nM T72458 CU1T4A 73347614 Ki = 6 nM T72458 CW8F4U 73348170 EC50 = 0.3 nM T72458 C4SR8Z 73348617 EC50 = 3.3 nM T72458 CK69FV 73348634 EC50 = 3 nM T72458 C6VK5T 73350013 IC50 = 620 nM T72458 CS4I5R 73350057 Ki = 1.01 nM T72458 CI9FS8 73350149 EC50 = 65 nM T72458 CI07CR 73350214 EC50 = 5 nM T72458 CMLR03 73350220 IC50 = 160 nM T72458 CPW67D 73350705 Ki = 0.14 nM T72458 C3EF0P 73351617 Ki = 0.22 nM T72458 CCF87P 73351717 EC50 = 25 nM T72458 CKWH98 73351727 IC50 = 720 nM T72458 CWHE24 73351850 EC50 = 140 nM T72458 C1L7HK 73353100 Ki = 5.7 nM T72458 CJL0D3 73353101 EC50 = 53 nM T72458 CR9N5P 73353187 EC50 = 3162.28 nM T72458 C8C0LW 73353205 IC50 = 4700 nM T72458 CGVC68 73353206 IC50 = 1600 nM T72458 CV27XE 73353216 EC50 = 290 nM T72458 CK2X0G 73353271 IC50 = 3.5 nM T72458 CS3FZ1 73353454 IC50 = 12 nM T72458 CK23FW 73354573 Ki = 2.2 nM T72458 CIEJ89 73354618 Ki = 1.5 nM T72458 CA4MR1 73354641 IC50 = 4 nM T72458 CXZD68 73354698 EC50 = 1995.26 nM T72458 C15BNT 73354704 EC50 = 65 nM T72458 C0ISQ4 73354708 IC50 = 1000 nM T72458 CJS25D 73354709 IC50 > 10000 nM T72458 C7OL2D 73354716 EC50 = 45 nM T72458 C7OT4D 73354780 EC50 = 0.11 nM T72458 CA8MQ1 73354785 IC50 = 230 nM T72458 CB6G1I 73355183 Ki = 150 nM T72458 CAWT96 73355184 Ki = 37 nM T72458 C17PEL 73356313 IC50 = 3.7 nM T72458 CT5UP1 73356732 Ki = 1.7 nM T72458 CR8M0O 73356733 Ki = 1.5 nM T72458 CA4U8O 90643802 EC50 = 0.24 nM T72458 CGBM80 90643803 EC50 = 0.12 nM T72458 CMAX81 90643804 EC50 = 0.26 nM T72458 CI05XM 90643805 EC50 = 0.29 nM T72458 CUJR85 90643806 EC50 = 0.4 nM T72458 C5N1DE 90643807 EC50 = 0.45 nM T72458 C1K0SJ 90643808 EC50 = 0.21 nM T72458 CSL28O 90643809 EC50 = 0.19 nM T72458 C4K7OV 90643810 EC50 = 1.06 nM T72458 CI50KM 90643811 EC50 = 40 nM T72458 CNE2F6 90643812 EC50 = 75 nM T72458 C36YQG 90643813 EC50 = 17 nM T72458 CS03VB 90643814 EC50 = 46 nM T72458 C68MKS 90643815 EC50 = 15 nM T72458 CJZ4V6 90643816 EC50 = 48 nM T72458 CHWK42 90643817 EC50 = 76 nM T72458 C9RH7W 90643818 EC50 = 1.9 nM T72458 CTN29R 90643819 EC50 = 204 nM T72458 CWL31Q 90643820 EC50 > 10000 nM T72458 CY70XF 90643821 EC50 = 5.3 nM T72458 CHV9I8 90643822 EC50 = 195 nM T72458 CAI8R0 90643823 EC50 = 28 nM T72458 CZ07JO 90643824 EC50 = 5.1 nM T72458 CRE52K 90643825 EC50 = 114 nM T72458 C36QSP 90643826 EC50 = 20 nM T72458 COES74 90643827 EC50 = 4.26 nM T72458 C83TIZ 90643828 EC50 = 280 nM T72458 CT7B4I 90643829 EC50 = 7.42 nM T72458 C2S5YA 90643830 EC50 = 24 nM T72458 CWDZ15 90643831 EC50 = 3.6 nM T72458 CD5C0I 90643832 EC50 = 89 nM T72458 CPX3G4 90643833 EC50 = 203 nM T72458 CM0JB7 90643834 EC50 = 2260 nM T72458 CC3T0S 90643835 EC50 = 6.65 nM T72458 C7IB3W 90643836 EC50 = 57 nM T72458 CVK16Q 90643837 EC50 = 9.6 nM T72458 CI64FK 90643838 EC50 = 120 nM T72458 CTU2B7 90643839 EC50 = 640 nM T72458 CKG73H 90643840 EC50 = 40 nM T72458 CM76IZ 90643841 EC50 = 2.6 nM T72458 C2OYM0 90643842 EC50 = 960 nM T72458 C38ZOR 90643843 EC50 = 15 nM T72458 C0K8EC 90643844 EC50 = 160 nM T72458 C8YK4D 90643845 EC50 = 15 nM T72458 CZ7W6Y 90643846 EC50 = 110 nM T72458 C5QDW8 90643847 EC50 = 22 nM T72458 CE2T4B 90643848 EC50 = 250 nM T72458 CKQ84G 90643849 EC50 = 21 nM T72458 CK58AT 90643850 EC50 = 110 nM T72458 CKP10U 90664284 IC50 = 6500 nM T72458 CP1S3T 90664642 EC50 = 82 nM T72458 CR7OX0 90664763 EC50 = 29 nM T72458 CVQ3P5 91971097 IC50 = 3300 nM T72458 C6L8AD 101043841 IC50 = 1300 nM T72458 C1KS2F 101043843 IC50 = 190 nM T72458 CI8PR4 118718122 EC50 = 3.6 nM T72458 CCL46X 118718855 IC50 > 10000 nM T72458 CK6FL5 118718881 EC50 = 14.6 nM T72458 CR13SP 118720353 EC50 = 3.981 nM T72458 CU2D0B 118720354 EC50 = 8.1 nM T72458 C1RU9V 118720355 EC50 = 13 nM T72458 C0WC7Q 118720356 EC50 = 3.7 nM T72458 CCO29V 118720357 EC50 = 24 nM T72458 CQ25BM 118720358 EC50 = 400 nM T72458 CJ3XW9 118720360 EC50 = 1.549 nM T72458 CM24SH 118720361 EC50 = 1.95 nM T72458 CU8DM7 118720362 EC50 = 2.138 nM T72458 C2SNQ7 118720363 EC50 = 1.8 nM T72458 C01ZPV 118720364 EC50 = 1.862 nM T72458 CF2P9J 118720365 EC50 = 4.074 nM T72458 CACO39 118720366 EC50 = 1.95 nM T72458 CI7J4T 118720367 EC50 = 1.585 nM T72458 CSX01G 118720368 EC50 = 1.3 nM T72458 CTJ18H 118720369 EC50 = 1.4 nM T72458 C76NQJ 118720370 EC50 = 1.698 nM T72458 CQ80IN 118720371 EC50 = 82 nM T72458 C4D9HL 118720372 EC50 = 236 nM T72458 CKP1Q6 118720373 EC50 = 188 nM T72458 C71OYW 118720374 EC50 = 11 nM T72458 C8ME0B 118735099 EC50 = 0.3 nM T72458 CK17XF 118735100 IC50 = 6.5 nM T72458 C1O7GU 118735101 EC50 = 0.3 nM T72458 CBTC79 118735102 EC50 = 227 nM T72458 C1O3GL 118735103 IC50 = 200 nM T72458 CAP67E 122178151 IC50 = 70 nM T72458 C65WMB 122184498 IC50 = 2.4 nM T72458 CH9L8O 122184499 IC50 = 18.2 nM T72458 CAQ17N 122184571 IC50 = 16.2 nM T72458 CK48WX 122184572 IC50 = 6.35 nM T72458 CF9PO7 122184573 IC50 = 1390 nM T72458 C3FBZ9 122184574 IC50 = 65.9 nM T72458 CCP0X7 122184575 IC50 = 111 nM T72458 C7OBX1 122184576 IC50 = 1010 nM T72458 CU73AF 122184577 EC50 = 2400 nM T72458 CGB7F4 122184578 IC50 = 134 nM T72458 CB7HZ8 122184579 IC50 = 59.4 nM T72458 C9HE4L 122184580 IC50 = 32.2 nM T72458 C9MJT7 122184581 IC50 = 244 nM T72458 C20NAY 122184582 EC50 = 35.5 nM T72458 CH1B8W 122184631 IC50 = 98 nM T72458 CLXB63 122184632 IC50 = 1700 nM T72458 CIJ14O 122184633 EC50 = 5 nM T72458 CDSR31 122184634 EC50 = 197 nM T72458 CL28BX 122184635 IC50 = 100 nM T72458 CYOR02 122184636 EC50 = 138 nM T72458 C09LFS 122184637 EC50 = 1570 nM T72458 C5CDX9 122184638 EC50 = 946 nM T72458 C64BPZ 122184639 IC50 = 99.9 nM T72458 CEDT39 122184640 EC50 = 1000 nM T72458 CLB43S 122184641 EC50 = 6590 nM T72458 CN4L5U 122184908 EC50 = 0.8 nM T72458 CG0U7B 122184909 EC50 = 152 nM T72458 CZ4HW7 122184910 IC50 = 0.5 nM T72458 C6KW7J 122184911 EC50 = 840 nM T72458 CK3VM5 122184912 EC50 = 1110 nM T72458 C0AFH9 122184913 EC50 = 485 nM T72458 CNBA05 122184914 EC50 = 1450 nM T72458 CARC80 122194229 Ki = 0.14 nM T72458 C80KPB 127046235 EC50 = 0.67 nM T72458 CE63JM 127046977 EC50 = 1.1 nM T72458 CI7TE9 127047209 EC50 = 5.5 nM T72458 C5GX7N 127047475 EC50 = 0.57 nM T72458 C28UAD 127047853 EC50 = 1.2 nM T72458 C9CYP2 127047913 EC50 = 2 nM T72458 C1SF3V 127048118 EC50 = 0.95 nM T72458 CGKE81 132938008 IC50 = 7.5 nM T72458 C7CLU6 133053557 EC50 = 280 nM T72458 CKV0P6 136024005 Ki = 7 nM T72458 CJNF06 137631599 EC50 = 19.95 nM T72458 COM8N7 137631628 IC50 > 1000 nM T72458 CW9P1D 137633115 EC50 = 128 nM T72458 CF2NA9 137633806 EC50 = 1.4 nM T72458 CTD90C 137634090 EC50 = 3800 nM T72458 CPL59T 137635422 EC50 = 1.8 nM T72458 CM1H6A 137636428 EC50 = 677.5 nM T72458 CU4KL7 137636677 EC50 = 602.56 nM T72458 CVC3Q2 137636965 EC50 = 524.81 nM T72458 CK2CZ3 137637026 EC50 = 3.2 nM T72458 CME01A 137637283 EC50 = 0.34 nM T72458 C6TKX9 137637656 EC50 = 2.8 nM T72458 C2FEA6 137638725 EC50 = 6.166 nM T72458 CH17TL 137638778 EC50 = 1.4 nM T72458 CKR14I 137639770 EC50 = 2.1 nM T72458 CHB9X0 137640703 EC50 = 501.19 nM T72458 CBL5Z9 137641157 EC50 = 87.1 nM T72458 CCPD94 137641398 EC50 = 120.23 nM T72458 CTN96O 137642298 EC50 = 71 nM T72458 CGP0V3 137643023 EC50 = 184.6 nM T72458 CAT50J 137643076 EC50 = 178 nM T72458 C5R2TI 137643266 IC50 = 20 nM T72458 CE0YF4 137643385 EC50 = 317.9 nM T72458 C68AYB 137644225 EC50 = 12.7 nM T72458 CJ1I7B 137645567 EC50 > 100000 nM T72458 CKES17 137646333 EC50 = 46773.51 nM T72458 CT18GM 137646617 EC50 = 1047.13 nM T72458 CV5RX4 137647009 EC50 = 6.4 nM T72458 CY7K4J 137647538 EC50 = 114.82 nM T72458 C10VFY 137648144 EC50 = 7.6 nM T72458 C5X7AK 137648344 EC50 = 200 nM T72458 CSF97J 137649543 EC50 = 257.7 nM T72458 CIV6Z7 137649910 EC50 > 3000 nM T72458 CF3VP0 137651074 IC50 = 5 nM T72458 CH62TM 137653176 EC50 > 3000 nM T72458 CF5Z2W 137653739 EC50 = 0.2 nM T72458 CKX3Q9 137653925 EC50 = 1737.8 nM T72458 C12DIK 137655051 Ki = 0.79 nM T72458 CMO01K 137655905 EC50 = 3090.3 nM T72458 CKL0Y8 137656033 EC50 = 112.3 nM T72458 C5WHL4 137656521 EC50 = 11.4 nM T72458 C5FI6X 137657633 IC50 = 45 nM T72458 COS0A1 137658158 EC50 = 147.91 nM T72458 CS1PR7 137659394 EC50 = 478.63 nM T72458 CHB32J 137659790 EC50 = 467.74 nM T72458 CQ7S0L 137659949 EC50 = 21000 nM T72458 C2XLI7 137660671 EC50 = 229.09 nM T72458 C98FVD 137660993 EC50 = 27.54 nM T72458 C4CFP9 137661893 EC50 > 3000 nM T72458 CCZ72V 137662147 EC50 = 2.3 nM T72458 C2WC5J 145948876 IC50 = 950 nM T72458 CUC3S2 145948912 EC50 = 220 nM T72458 C8D7OM 145964017 EC50 = 3.2 nM T72458 CAT7W0 145964349 Ki = 29 nM T72458 CCK75J 145964837 EC50 = 6.7 nM T72458 CS73TM 145966364 EC50 = 1000 nM T72458 CHU51B 145966490 EC50 = 5.3 nM T72458 CJO1Y6 145966716 EC50 = 270 nM T72458 C9RA7Q 145967155 IC50 = 71 nM T72458 CICD84 145971389 EC50 = 150 nM T72458 C97DEG 145971673 EC50 = 720 nM T72458 CEV4F6 145972289 IC50 = 100 nM T72458 C9NRU8 145973779 IC50 = 59 nM T72458 CYD0J5 145973975 IC50 = 73 nM T72458 CR2NQ5 145975465 EC50 = 6.7 nM T72458 CKP26E 145976444 EC50 = 18 nM T72458 C7UJ8Q 145976863 EC50 = 120 nM T72458 CMS17N 145977650 EC50 = 10 nM T72458 CJ28PL 145980198 EC50 = 133 nM T72458 C0S1IN 145980719 EC50 = 928 nM T72458 CEZU78 145980838 IC50 = 2.1 nM T72458 CF34MX 145988152 EC50 = 36 nM T72458 C39KYZ 145988867 EC50 = 280 nM T72458 C7WF3R 145989222 EC50 = 17 nM T72458 C50ZLS 145990599 EC50 = 407 nM T72458 CDQZ25 145994283 IC50 = 10 nM T72458 CE3CN7 155527254 EC50 = 0.03 nM T72458 CX9B4Y 155531854 EC50 = 1.9 nM T72458 C3Q8AU 155532197 EC50 = 5.9 nM T72458 CA5R2L 155532232 IC50 = 14300 nM T72458 C0P7XR 155536962 IC50 = 19300 nM T72458 C6K3AW 155544852 IC50 = 32.2 nM T72458 CQZ7X1 155546131 IC50 = 2700 nM T72458 C7IS0X 155548853 IC50 = 250 nM T72458 CD3J2E 155551202 IC50 = 15700 nM T72458 C20BJD 155551699 EC50 = 4.7 nM T72458 C7C3QR 155551846 EC50 = 0.06 nM T72458 C2SFV9 155561116 IC50 = 1016 nM T72458 CCUT09 155563057 EC50 = 1.9 nM T72458 C1AE7Z 155566718 IC50 = 22000 nM T72458 CR08PO 24858629 IC50 > 1000 nM T72458 D00HAJ 73347136 IC50 = 13000 nM T72458 D00TSX 11672424 IC50 = 100 nM T72458 D00VYC 44400370 EC50 = 0.27 nM T72458 D00XMP 14364677 Ki = 700 nM T72458 D01HTX 11707715 IC50 = 600 nM T72458 D01VMU 44445082 EC50 > 2000 nM T72458 D02JVA 44408515 IC50 = 77 nM T72458 D02MPZ 11535237 EC50 = 2000 nM T72458 D03AZC 25078192 EC50 = 0.16 nM T72458 D04BOG 11629290 IC50 = 150 nM T72458 D04YZZ 44445083 IC50 = 330 nM T72458 D05LLI 11498895 EC50 = 130 nM T72458 D05WNC 11520823 IC50 = 34 nM T72458 D05XRI 44400401 EC50 = 0.26 nM T72458 D05ZUX 44207909 Ki >= 1000 nM T72458 D06PNU 44409257 EC50 = 10 nM T72458 D06RTP 11700730 EC50 = 16 nM T72458 D07DWH 44400402 EC50 = 0.28 nM T72458 D07IBF 44400322 EC50 = 0.54 nM T72458 D07RRN 44406884 Ki = 0.71 nM T72458 D07SFD 44408443 EC50 = 174 nM T72458 D07SRW 10258635 IC50 = 1100 nM T72458 D07UXW 44408400 IC50 = 170 nM T72458 D08DND 44445084 IC50 = 930 nM T72458 D08EBV 44406905 EC50 = 3.2 nM T72458 D09HHW 9842665 IC50 = 103 nM T72458 D09LHF 44413535 EC50 = 16.4 nM T72458 D09OMI 44400400 EC50 = 0.1 nM T72458 D09PDT 24774519 IC50 = 430 nM T72458 D09UUC 46877881 Ki = 190 nM T72458 D09XCH 44400371 EC50 = 5.24 nM T72458 D0A8ME 44400398 EC50 = 0.3 nM T72458 D0B8GR 44413876 EC50 = 5.7 nM T72458 D0B9NH 44408399 EC50 > 10000 nM T72458 D0C7VI 44400369 EC50 = 0.24 nM T72458 D0D8YP 763557 Ki = 2000 nM T72458 D0F6GX 44409240 EC50 = 44 nM T72458 D0GN9K 24774602 IC50 > 10000 nM T72458 D0L1MJ 11700739 IC50 = 16 nM T72458 D0M2QK 44413536 EC50 = 15.4 nM T72458 D0M4EF 11593084 EC50 = 3000 nM T72458 D0N6AS 44158031 EC50 = 200 nM T72458 D0N6KO 9938402 Ki = 0.05 nM T72458 D0P4GI 11629326 IC50 = 1000 nM T72458 D0QW4A 24774356 IC50 = 777 nM T72458 D0R0BY 44400320 EC50 = 0.06 nM T72458 D0R5KO 44413537 Ki = 670 nM T72458 D0T2RY 9948320 Ki >= 1000 nM T72458 D0U1UZ 44413577 EC50 = 1578 nM T72458 D0U5KM 11093672 EC50 = 0.93 nM T72458 D0U6XP 16724004 EC50 = 5700 nM T72458 D0V1JT 9875763 EC50 = 1.25 nM T72458 D0V5YV 44413592 Ki = 4420 nM T72458 D0VD7R 44408408 IC50 = 2700 nM T72458 D0W1SM 44408413 EC50 > 10000 nM T72458 D0WG8P 44400321 EC50 = 0.12 nM T72458 D0WI8M 44445085 IC50 = 300 nM T72458 D0X1YL 25078242 EC50 = 0.92 nM T72458 D0XQ5U 24774438 IC50 > 1000 nM T72458 D0YB7F 92432 EC50 < 0.03162 nM T72458 D0Z1QU 10098971 Ki = 7.9 nM T72458 D0ZD3M 44400399 EC50 = 0.79 nM T16514 D01XNB 4594 Ki = 3400 nM T16514 D03ZFG 5282054 IC50 = 0.19 ug.mL-1 T16514 D04AIT 5280445 IC50 = 62500 nM T16514 D0KL4J 5029 Ki = 5900 nM T16514 D0T6XX 4679 Ki = 4100 nM T16514 D0T9TJ 3034010 Ki = 280 nM T16514 D05TPI 72276 IC50 > 100000 nM T16514 D0U2BH 65064 IC50 = 51970 nM T16514 D0E4WF 439176 Ki = 1500000 nM T16514 C2KJI7 3883 Ki = 5300 nM T16514 CJ0I1N 13792 Ki = 30000 nM T16514 CTHE54 122841 IC50 = 49100 nM T16514 C0WR5N 145691 Ki = 140000000 nM T16514 CCG98V 165114 Ki = 500000 nM T16514 C5Q1JX 182232 IC50 > 1000000 nM T16514 C3FJQ1 485186 IC50 = 91070 nM T16514 CZYL67 2292609 Ki = 380 nM T16514 CMP0Z5 4782471 IC50 = 1140 nM T16514 CE6K3P 5281635 IC50 = 40980 nM T16514 CH01XT 5281656 IC50 = 17850 nM T16514 CJC35O 5282800 IC50 = 100000 nM T16514 CY0CO2 5495925 IC50 = 24830 nM T16514 C51EUJ 7873335 IC50 >= 50000 nM T16514 CG2V5K 7873337 IC50 = 1100 nM T16514 C75GIM 9881506 IC50 = 59000 nM T16514 C9XI1C 9977422 IC50 > 1000 ug.mL-1 T16514 CHZ2D5 9995235 IC50 > 50 ug.mL-1 T16514 C8MXH4 10000563 IC50 > 50 ug.mL-1 T16514 CS7FC2 10020330 IC50 > 50 ug.mL-1 T16514 CTVI84 10040478 IC50 > 50 ug.mL-1 T16514 CNQH21 10040479 IC50 = 2.1 ug.mL-1 T16514 C1PK2F 10044646 IC50 > 1000 ug.mL-1 T16514 CNX5Z8 10085202 IC50 > 50 ug.mL-1 T16514 CUM0N6 10087016 IC50 = 4.6 ug.mL-1 T16514 C9P3CS 10087923 IC50 > 50 ug.mL-1 T16514 C51CUM 10092378 Ki = 30000 nM T16514 C64XGK 10176955 IC50 > 50 ug.mL-1 T16514 CVFJ46 10246217 IC50 > 50 ug.mL-1 T16514 CWI1H5 10266601 IC50 > 50 ug.mL-1 T16514 C5LRW4 10298511 IC50 = 3300 nM T16514 CV6IH8 10354980 IC50 > 50 ug.mL-1 T16514 CVF7Z2 10359032 IC50 = 6.8 ug.mL-1 T16514 C0M2RF 10404949 IC50 > 50 ug.mL-1 T16514 C5MUE3 10422346 IC50 > 50 ug.mL-1 T16514 CQ2LZ5 10466563 IC50 > 50 ug.mL-1 T16514 CJW43Z 10469992 IC50 > 50 ug.mL-1 T16514 C5X7YI 11050315 IC50 > 50 ug.mL-1 T16514 C24UPE 11529878 IC50 > 50 ug.mL-1 T16514 CO96XN 11541428 IC50 = 160 nM T16514 CWQ56J 11543533 Ki = 2500 nM T16514 CZ5N3C 11722353 IC50 > 50 ug.mL-1 T16514 CQY8H4 11724126 IC50 > 50 ug.mL-1 T16514 C7X6DR 11777194 IC50 > 50 ug.mL-1 T16514 CT5D2I 14378645 IC50 = 60200 nM T16514 C45BLU 15081407 IC50 = 31000 nM T16514 C1PJ8I 15788084 Ki = 100000 nM T16514 CO04TC 16046225 IC50 = 25400 nM T16514 CWR7N5 19910294 IC50 = 8590 nM T16514 C19EMT 23649126 IC50 = 160 nM T16514 C9QBC6 25096732 IC50 = 56100 nM T16514 CNCT63 25096734 IC50 = 71700 nM T16514 C06NHT 38390838 IC50 = 50000 nM T16514 CE7B0W 44290695 Ki = 220000 nM T16514 C1QYT0 44388272 IC50 > 50 ug.mL-1 T16514 C0E3PC 44388283 IC50 > 50 ug.mL-1 T16514 CM27AK 44388295 IC50 > 50 ug.mL-1 T16514 C86TYF 44415373 IC50 > 15000 nM T16514 CC3HM1 44415374 IC50 > 15000 nM T16514 C09HMK 44415477 IC50 > 15000 nM T16514 CJA30S 44415496 IC50 > 15000 nM T16514 CF5L3P 44415497 IC50 > 15000 nM T16514 C1VXO4 44415510 IC50 > 15000 nM T16514 CX5KA8 45266261 Ki = 2500000 nM T16514 C3I7XR 51346964 IC50 = 79 nM T16514 CHQW27 52914172 IC50 = 200 nM T16514 CO5AR4 52914173 IC50 = 300 nM T16514 CQCV94 52945061 IC50 = 49160 nM T16514 CIF69A 52948815 IC50 = 14760 nM T16514 CULB62 54706679 IC50 = 19 nM T16514 CYVU49 54712162 IC50 = 136 nM T16514 CQS8R7 54720260 IC50 = 52 nM T16514 CK0IP7 54720261 IC50 = 54 nM T16514 CV4W0R 54720262 IC50 = 194 nM T16514 CS2G5M 54720263 IC50 = 728 nM T16514 CQ9D3F 54720264 IC50 = 68 nM T16514 CR0S7K 54720274 IC50 = 4164 nM T16514 C16TFJ 54720277 IC50 = 734 nM T16514 CJ9A8U 54720280 IC50 = 127 nM T16514 CCG95F 54737895 IC50 = 402 nM T16514 CR0D3L 54737897 IC50 > 15000 nM T16514 C6N2UI 54737898 IC50 > 15000 nM T16514 C7BE1N 54737901 IC50 = 207 nM T16514 CY0F7L 54737905 IC50 = 101 nM T16514 CRWP39 54737909 IC50 > 15000 nM T16514 C6GPH3 54737911 IC50 = 1294 nM T16514 C2KJS4 56658153 IC50 = 1500 nM T16514 CP7IJ5 56658154 IC50 = 580 nM T16514 CK19VO 56661663 IC50 = 420 nM T16514 C0ED9O 56665072 IC50 = 400 nM T16514 CG24JD 56665073 IC50 = 280 nM T16514 C04ZAH 56668685 IC50 = 480 nM T16514 CI51ES 56672028 IC50 = 310 nM T16514 CBYM16 56672029 IC50 = 290 nM T16514 C6NOF0 56675407 IC50 = 1300 nM T16514 C25VNE 56675408 IC50 = 700 nM T16514 CVOA13 56675409 IC50 = 2400 nM T16514 C6W2ZV 56675410 IC50 = 270 nM T16514 CSR3L6 56675411 IC50 = 910 nM T16514 CD5WP7 56678752 IC50 = 1500 nM T16514 CQK16D 56678753 IC50 > 10000 nM T16514 C89BAK 56678754 IC50 = 190 nM T16514 C6XC1K 56678755 IC50 = 530 nM T16514 C2PYZ9 56678756 IC50 > 3000 nM T16514 C53YIK 56678879 IC50 = 420 nM T16514 C54EIB 56682065 IC50 = 2000 nM T16514 C60CNB 56682066 IC50 = 1400 nM T16514 C9U0SZ 56944776 IC50 = 13 nM T16514 C0E2CB 57330203 IC50 = 6 nM T16514 CD3IC4 57519517 IC50 = 15.8 nM T16514 C15LHR 67353959 IC50 = 3 nM T16514 C5IR7A 68288172 IC50 = 430 nM T16514 CQPC84 68288211 IC50 = 40 nM T16514 CXZ9N7 68288384 IC50 = 17 nM T16514 C38ZAK 68288699 IC50 = 85 nM T16514 CK07RI 68288711 IC50 = 70 nM T16514 C9NFH0 68288836 IC50 = 980 nM T16514 C8D6XN 68288941 IC50 = 590 nM T16514 CYF20R 68288944 IC50 = 130 nM T16514 CN38EO 68288981 IC50 = 35 nM T16514 C8NJ1R 68288986 IC50 = 107 nM T16514 C7EP2D 68289020 IC50 = 60 nM T16514 C6BAD8 68289174 IC50 = 60 nM T16514 CO8X9D 68289184 IC50 = 70 nM T16514 C2HJB7 68289227 IC50 = 870 nM T16514 CVRK70 69081490 IC50 = 251 nM T16514 C64OIV 69085357 IC50 = 10 nM T16514 C6O8MS 69166563 IC50 = 50 nM T16514 CCN1K2 70355043 IC50 = 7.9 nM T16514 C3L7MO 70872230 IC50 = 300 nM T16514 C3O8YN 70872278 IC50 = 480 nM T16514 CK56QA 70873969 IC50 = 990 nM T16514 CU0D8S 71460623 IC50 = 10000 nM T16514 CRH37A 71511821 IC50 = 20 nM T16514 CGU2I3 71541605 IC50 > 50000 nM T16514 C5KQG0 71541606 IC50 > 50000 nM T16514 CN6RQ2 71719838 IC50 = 45 nM T16514 CDC29F 72188556 IC50 = 10 nM T16514 C7B2VH 73332466 IC50 = 28 nM T16514 C6ZPL7 73388616 IC50 = 51 nM T16514 CT3N0M 73388705 IC50 = 22 nM T16514 CF40TL 86272214 IC50 = 110 nM T16514 CMDX07 86272688 IC50 = 12 nM T16514 CHU42Z 86272922 IC50 = 3100 nM T16514 CE4A7B 86273159 IC50 = 11 nM T16514 C3WIN2 86273160 IC50 = 10 nM T16514 CWI9H2 86273162 IC50 = 11 nM T16514 CR4O3Z 86273403 IC50 = 110 nM T16514 C0R2KW 86273408 IC50 = 33 nM T16514 C39ZJT 86273883 IC50 = 26 nM T16514 CG40JA 86275336 IC50 > 5000 nM T16514 C4J8CB 86275339 IC50 = 1800 nM T16514 CW0I7F 86275791 IC50 = 350 nM T16514 C1DAT5 86275793 IC50 = 35000 nM T16514 C7U8LK 86275794 IC50 = 50000 nM T16514 CDF60C 89993363 IC50 = 1380 nM T16514 C7H0RS 89993436 IC50 = 32 nM T16514 CP97LB 89993468 IC50 = 41 nM T16514 CCTW25 89993534 IC50 = 550 nM T16514 C9Z3RV 89993608 IC50 = 69 nM T16514 CW2ND1 89993632 IC50 = 33 nM T16514 CUPS02 89993706 IC50 = 23 nM T16514 CRK0M7 89993860 IC50 = 25 nM T16514 C1GH7D 90001554 IC50 = 46 nM T16514 CMUT58 117631954 IC50 = 54 nM T16514 CDV34G 117632261 IC50 = 57 nM T16514 CZK4A6 117632449 IC50 = 69 nM T16514 CPY70A 117992529 IC50 = 360 nM T16514 C8L2AI 117992579 IC50 = 300 nM T16514 CBO57F 117992669 IC50 = 160 nM T16514 CYQ6V8 117992803 IC50 = 460 nM T16514 C29DCG 117992846 IC50 = 1100 nM T16514 CU73WN 117992892 IC50 = 8510 nM T16514 C5EDL1 117992950 IC50 = 33100 nM T16514 CYD3W2 117992981 IC50 = 250 nM T16514 C6GP4I 117992993 IC50 = 590 nM T16514 C7B8NO 117993006 IC50 = 460 nM T16514 COT7W6 117993116 IC50 = 8710 nM T16514 CW82PK 117993126 IC50 = 790 nM T16514 CIK64W 117993152 IC50 = 120 nM T16514 CT09BE 117993175 IC50 = 8910 nM T16514 C1FUZ4 117993412 IC50 = 130 nM T16514 C54FAV 117999149 IC50 = 83 nM T16514 CZT69Y 117999157 IC50 = 30 nM T16514 CC5GD8 117999160 IC50 = 20 nM T16514 CCO89U 117999164 IC50 = 42 nM T16514 C8VLN5 117999171 IC50 = 50 nM T16514 COZ8I6 117999184 IC50 = 200 nM T16514 CN6LZ9 117999235 IC50 = 20 nM T16514 C8PMK6 117999267 IC50 > 10000 nM T16514 C9Y1PD 117999287 IC50 = 300 nM T16514 C5OKI2 118125364 IC50 = 5888.44 nM T16514 CI47HU 118125371 IC50 = 56.23 nM T16514 C9X0KR 118125374 IC50 = 47.86 nM T16514 CZCA13 118125376 IC50 = 490 nM T16514 CP91UC 118125426 IC50 = 160 nM T16514 CYWI47 118125430 IC50 = 41 nM T16514 CC7I0K 118125439 IC50 = 177.83 nM T16514 CH7S8X 118125468 IC50 = 140 nM T16514 CDC75Z 118125490 IC50 = 30.2 nM T16514 C8OPS5 118125499 IC50 = 93.33 nM T16514 C83ZWH 118144180 IC50 = 93 nM T16514 CYI51F 118621498 IC50 = 32 nM T16514 C2OY4N 118621507 IC50 = 97 nM T16514 CFKI50 118621601 IC50 = 90 nM T16514 CUO5I1 118621602 IC50 = 142 nM T16514 CVM6E7 118621647 IC50 = 61 nM T16514 CB5JZ9 118621761 IC50 = 16 nM T16514 CH74OR 118621798 IC50 = 310 nM T16514 C4S1HV 122192508 IC50 = 6 nM T16514 CMNB15 122197394 IC50 = 28700 nM T16514 CY0QH7 122197395 IC50 = 23100 nM T16514 C34DEV 122197396 IC50 = 29700 nM T16514 C9XV2S 122197397 IC50 = 32600 nM T16514 CUT65O 132503175 IC50 = 1500 nM T16514 C1JB6Y 135407178 IC50 > 50 ug.mL-1 T16514 C8T1FY 135410225 IC50 = 4 ug.mL-1 T16514 C75VLC 135432847 IC50 = 5.7 ug.mL-1 T16514 CWK90L 135449011 IC50 > 50 ug.mL-1 T16514 CJD80P 135457983 IC50 > 50 ug.mL-1 T16514 CP8HN9 135488223 IC50 = 8.4 ug.mL-1 T16514 CTH2W0 135503576 IC50 = 2.8 ug.mL-1 T16514 CX8Y7I 135517312 IC50 = 41 ug.mL-1 T16514 CKU80W 135518065 IC50 > 50 ug.mL-1 T16514 CM1HF2 135526950 IC50 > 50 ug.mL-1 T16514 CQK2T3 135535916 IC50 = 8.7 ug.mL-1 T16514 CW0S7A 136102470 IC50 = 49.2 ug.mL-1 T16514 C61AJU 136102471 IC50 > 50 ug.mL-1 T16514 C2NC9L 137633752 IC50 = 3110 nM T16514 CEJO70 137634807 IC50 = 4810 nM T16514 CDT67V 137637200 IC50 = 160 nM T16514 CMSA73 137639962 IC50 = 3980 nM T16514 C1KN9L 137640079 IC50 = 5550 nM T16514 CNVZ89 137640673 IC50 = 3170 nM T16514 C0EY3T 137643629 IC50 = 2610 nM T16514 CWOY74 137647871 IC50 = 8370 nM T16514 CNFP69 137658811 IC50 = 12600 nM T16514 CJQ6B7 137659959 IC50 = 1190 nM T16514 C01KBD 137661456 IC50 = 9560 nM T16514 CZI19P 145960543 IC50 = 590 nM T16514 C19AFT 145961063 IC50 = 170 nM T16514 CW9NJ4 145961301 IC50 = 450 nM T16514 C3AEW6 145962120 IC50 = 36 nM T16514 CG8B1R 145962440 IC50 = 79 nM T16514 CKFR42 145962726 IC50 = 300 nM T16514 C63PUQ 145963234 IC50 = 28 nM T16514 D01WTQ 5495929 IC50 = 40640 nM T16514 D05IWY 5464078 IC50 = 1240 nM T16514 D06PRC 5281650 IC50 = 5540 nM T16514 D09CLP 439155 Ki = 150000 nM T16514 D0B5GC 11349 IC50 > 100000 nM T16514 D0PO8E 6137 Ki > 150000000 nM T16514 D0QP7C 54737894 IC50 = 1403 nM T59604 D02NEH 178024 EC50 = 0.1995 nM T59604 D0BV3J 9804938 IC50 = 22.9 nM T59604 D01HLO 58438464 Ki = 6.607 nM T59604 D05UYQ 15984937 EC50 > 1000 nM T59604 D0LI1C 44469321 IC50 > 30000 nM T59604 D0O1LU 9827407 IC50 = 62.9 nM T59604 D0UO4B 216208 EC50 = 0.9 nM T59604 D0W9VW 11526696 EC50 = 27 nM T59604 D0XH9B 9810101 EC50 = 3 nM T59604 D09TGZ 6918297 IC50 = 15.9 nM T59604 D0A1KU 11683187 Ki = 4400 nM T59604 D0B3CY 121879 Ki = 63 nM T59604 C7Q3IT 328912 IC50 = 1700 nM T59604 CE16YX 753168 IC50 = 8200 nM T59604 C25ZHX 1221269 IC50 = 250 nM T59604 CL5WT1 1744826 IC50 = 180 nM T59604 C1MJA8 2814760 IC50 > 10000 nM T59604 CD2K4M 3153998 Ki = 870 nM T59604 CQ9ZP3 3153999 Ki = 280 nM T59604 C6LAW3 3154000 Ki = 1320 nM T59604 CJ3K0S 3154005 Ki = 2030 nM T59604 CY4I3A 3174463 Ki = 1290 nM T59604 C7QC1D 3180629 Ki = 1370 nM T59604 C0YXV3 3676358 IC50 = 100 nM T59604 CIB78P 5311280 IC50 = 750 nM T59604 CWX3C4 9804743 IC50 = 1.2 nM T59604 C36UOT 9805090 EC50 = 3 nM T59604 CYP42T 9807597 EC50 = 1 nM T59604 C3Q9FN 9827234 EC50 = 10 nM T59604 C91MIV 9848305 EC50 = 986 nM T59604 C75TME 9849592 EC50 = 72 nM T59604 CK0E8G 9868878 EC50 = 7.6 nM T59604 C74HBN 9870965 EC50 = 11.7 nM T59604 C8PFZ1 9875705 EC50 = 1.585 nM T59604 C8BRO3 9876514 Ki = 5 nM T59604 CDB32K 9890375 EC50 = 14 nM T59604 C4BCX8 9890504 EC50 = 1 nM T59604 CPX3E7 9917957 EC50 = 0.34 nM T59604 C8M7BX 9919153 Ki = 6 nM T59604 CMTS32 9950632 EC50 = 30 nM T59604 C4L8RA 9956908 IC50 = 16 nM T59604 C3LV1I 9987037 EC50 = 19.6 nM T59604 CJ7N9H 10005618 EC50 = 3 nM T59604 CSP71U 10006735 EC50 = 6.3 nM T59604 C5X9KF 10026738 EC50 = 16.6 nM T59604 C25PLS 10029990 EC50 = 5 nM T59604 C3JS1K 10032659 EC50 = 7.95 nM T59604 CG2E6X 10100708 EC50 = 69.2 nM T59604 CI0DX4 10118326 EC50 = 1.8 nM T59604 C1Z0XT 10143731 EC50 = 39 nM T59604 C0S8EM 10166594 EC50 = 2.3 nM T59604 CDUZ27 10186158 IC50 = 25.6 nM T59604 C5MRA2 10207327 IC50 = 58 nM T59604 C0O4KL 10209618 EC50 = 7.3 nM T59604 CR5IU4 10210658 EC50 = 16.98 nM T59604 CE3VR7 10253999 Ki = 220 nM T59604 C8RX9I 10280020 EC50 = 0.73 nM T59604 C1E9MX 10323604 EC50 = 1.096 nM T59604 CF27UE 10345516 EC50 = 0.7943 nM T59604 C76XZR 10346217 Ki > 5000 nM T59604 CO16JV 10415000 EC50 = 2.8 nM T59604 CKG7P1 10415364 IC50 = 32 nM T59604 CWM6U8 10506325 EC50 = 6 nM T59604 CP12CV 10530303 IC50 > 10000 nM T59604 CFY90H 10553921 EC50 = 0.7943 nM T59604 CS60ON 10600702 EC50 = 7.5 nM T59604 CO9VJ3 10602640 EC50 = 5 nM T59604 CMW0Z9 10625750 EC50 = 1.585 nM T59604 CL1PH2 10626337 EC50 = 1.995 nM T59604 CW34CO 10699268 IC50 = 55 nM T59604 C9I5HK 10738173 IC50 > 10000 nM T59604 CD91XJ 10745533 EC50 = 18 nM T59604 COU2W4 10746435 IC50 > 2000 nM T59604 C9G2BH 10791616 EC50 = 5 nM T59604 C5Q2WC 10839304 IC50 > 10000 nM T59604 CS8A4G 10864048 IC50 = 185 nM T59604 CPC62E 10907396 IC50 = 337 nM T59604 C5JZW0 10918326 IC50 = 20.1 nM T59604 CTD32I 10929048 IC50 = 228 nM T59604 CS9T3E 10984260 IC50 = 807 nM T59604 CX2S0A 10984270 IC50 = 59.8 nM T59604 CZ0MB4 10994861 IC50 = 807 nM T59604 C06SQO 11016748 IC50 = 16.9 nM T59604 C7PCL0 11114279 IC50 = 213 nM T59604 CSF5J2 11124146 IC50 = 16.2 nM T59604 C6RDO8 11134880 IC50 = 391 nM T59604 C9O4AY 11145720 IC50 = 167 nM T59604 C9ZWB1 11154001 IC50 = 56 nM T59604 CL85TY 11154823 IC50 = 2.8 nM T59604 C19HVQ 11163070 IC50 = 2700 nM T59604 C8C7FK 11166495 IC50 = 83 nM T59604 CQD27L 11176805 IC50 = 67 nM T59604 CVX23I 11178309 IC50 = 70 nM T59604 CX52ZC 11179347 IC50 = 6.9 nM T59604 CB5J8R 11190594 IC50 = 2.8 nM T59604 C9B7QL 11211892 IC50 = 72 nM T59604 C1IQU2 11221946 IC50 = 310 nM T59604 CAG74M 11225576 IC50 = 0.3 nM T59604 CE59SF 11248021 IC50 = 34 nM T59604 C9VA4H 11256439 IC50 = 160 nM T59604 C5QEH2 11258291 EC50 = 40 nM T59604 CTH56E 11281346 IC50 = 50 nM T59604 CIG85H 11282247 IC50 = 19 nM T59604 CZ12BJ 11306502 EC50 = 0.46 nM T59604 CI28KO 11314908 IC50 = 221 nM T59604 CXT20O 11327400 IC50 = 86 nM T59604 CVU6P9 11328064 IC50 = 120 nM T59604 C1H5CL 11328920 IC50 = 2 nM T59604 C5M3ZN 11329138 IC50 = 29 nM T59604 C7Y8VZ 11337482 IC50 = 11 nM T59604 C5A7VJ 11339816 IC50 = 1.5 nM T59604 C7QV2P 11340044 IC50 = 5.8 nM T59604 CI2TD8 11340329 IC50 = 7 nM T59604 C85DMO 11349789 IC50 = 66 nM T59604 C3FID2 11351838 IC50 = 10 nM T59604 C79PWN 11353414 EC50 = 1.5 nM T59604 C23YMZ 11373823 IC50 = 126 nM T59604 CX21SG 11410373 IC50 = 0.4 nM T59604 C5ZH0O 11430392 IC50 = 4.2 nM T59604 C4EL7T 11430583 IC50 = 37 nM T59604 C38KZA 11431274 IC50 = 0.4 nM T59604 C02SXV 11441978 IC50 = 11 nM T59604 CH8IF2 11442040 IC50 = 88 nM T59604 C41XHB 11452801 IC50 = 18 nM T59604 CV0M3Q 11453509 IC50 = 7.7 nM T59604 C6IJ8W 11454617 IC50 = 2.5 nM T59604 CJS58R 11455251 IC50 = 137 nM T59604 CF81ZH 11476589 IC50 = 0.8 nM T59604 C09NWX 11503585 IC50 = 308 nM T59604 CA6BI9 11508639 IC50 = 300 nM T59604 CB7VA3 11517629 IC50 = 37 nM T59604 CSB20C 11523411 IC50 = 110 nM T59604 CDOF50 11525404 EC50 = 10 nM T59604 CG3AZ5 11531313 IC50 = 550 nM T59604 CYO8E0 11532288 EC50 = 15.85 nM T59604 CGS1J2 11537683 IC50 = 110 nM T59604 C5F8WZ 11537800 IC50 = 57 nM T59604 C3ROC9 11538533 IC50 = 7 nM T59604 C6Z4IU 11538534 IC50 = 9.8 nM T59604 CU4AY2 11539587 IC50 = 492 nM T59604 CD2TQ8 11539588 IC50 = 861 nM T59604 CLG67J 11539642 EC50 = 2.512 nM T59604 C17VJD 11554351 EC50 = 39.81 nM T59604 CGY7Z8 11556936 IC50 = 8530 nM T59604 C87NYP 11556937 IC50 = 15700 nM T59604 CPK5I8 11568561 IC50 = 600 nM T59604 CTWI32 11576186 EC50 = 15.85 nM T59604 CI3LV0 11576960 IC50 = 98 nM T59604 CJ1RE7 11577349 IC50 = 10 nM T59604 CZY1F4 11582836 IC50 = 410 nM T59604 CR87OJ 11583811 IC50 = 2.9 nM T59604 CP07SD 11584048 EC50 = 0.7943 nM T59604 C2PS0V 11605061 EC50 = 39.81 nM T59604 C8LS5D 11605333 IC50 = 5.7 nM T59604 C83JXN 11605822 IC50 = 25 nM T59604 C3Q0JA 11606121 IC50 = 4900 nM T59604 CL9E5D 11612155 IC50 = 6.3 nM T59604 CAX29H 11617435 IC50 = 290 nM T59604 CO0X6G 11618705 IC50 = 53 nM T59604 C0PE7U 11626181 IC50 = 319 nM T59604 C2Z5OD 11633712 EC50 = 100 nM T59604 C3UW1I 11646276 IC50 = 9.2 nM T59604 CEA68R 11649239 IC50 = 18 nM T59604 C8JQ6X 11649248 IC50 = 39 nM T59604 C7A6DM 11654867 IC50 = 3350 nM T59604 C5X9KU 11655355 IC50 = 320 nM T59604 C6YW9T 11655578 IC50 = 780 nM T59604 CCYT36 11662746 EC50 = 63.1 nM T59604 CF0WK6 11663710 IC50 = 8 nM T59604 CL14RB 11669486 IC50 = 41 nM T59604 CF14EQ 11676995 IC50 = 110 nM T59604 C4MRC3 11677781 IC50 = 19 nM T59604 C42VAZ 11683469 IC50 = 2.4 nM T59604 C8VTS6 11690097 IC50 = 3.7 nM T59604 C61WEI 11692087 IC50 = 6 nM T59604 CE0F1A 11697618 IC50 = 280 nM T59604 C3X4IJ 11699004 IC50 = 57 nM T59604 CM9WV4 11712108 EC50 = 6.31 nM T59604 CW34HT 11712151 IC50 = 1.2 nM T59604 CQL7H2 11713497 IC50 = 9 nM T59604 CGZ57K 11731384 IC50 = 116 nM T59604 CVS7D5 11751384 IC50 = 343 nM T59604 CBK20C 11827047 IC50 = 22.7 nM T59604 C9XI4T 11846463 IC50 = 11 nM T59604 CWP0B9 11846624 IC50 = 109 nM T59604 CCUF60 11846625 IC50 = 249 nM T59604 CF6D4C 11846627 IC50 = 2270 nM T59604 C5D4KB 11846628 IC50 = 1670 nM T59604 CJ3AT5 11846629 IC50 = 391 nM T59604 CD4VX3 11846630 IC50 = 3080 nM T59604 CWSA56 11846799 IC50 > 1000 nM T59604 CQ9FO0 11846800 IC50 > 10000 nM T59604 C6C8DJ 15481181 EC50 = 3 nM T59604 CJ3SG7 15481185 EC50 = 3.981 nM T59604 C9STQ7 15481188 EC50 = 3 nM T59604 COA2U1 15945877 IC50 = 11 nM T59604 COZU71 15949382 IC50 = 54 nM T59604 C20CRP 16040587 EC50 = 100 nM T59604 C8ZP3G 16041292 EC50 = 501.19 nM T59604 CR0JL5 16112909 IC50 = 660 nM T59604 CJB54V 16112910 IC50 = 560 nM T59604 CD85OU 16112911 IC50 = 750 nM T59604 CA5D3X 16113002 IC50 = 38 nM T59604 COF94S 16113003 IC50 = 5.6 nM T59604 CQ59HR 16113122 IC50 = 154 nM T59604 C8MU4Z 16113124 IC50 = 828 nM T59604 C6K7IZ 16113245 IC50 = 4.5 nM T59604 C96CEF 16113246 IC50 = 8 nM T59604 C2ZGY6 16113248 EC50 = 7.7 nM T59604 C6TGZ4 16113370 IC50 = 29 nM T59604 CDC6B4 16113371 EC50 = 6 nM T59604 CRV2T0 16113372 IC50 = 28 nM T59604 CMSC45 16113468 IC50 = 108 nM T59604 CUJ3A6 16113469 IC50 = 80 nM T59604 CBW76F 16113471 IC50 = 100 nM T59604 CB0J6E 16113472 IC50 = 200 nM T59604 CBU67D 16113474 IC50 = 850 nM T59604 C9IQZ5 16113577 EC50 = 15 nM T59604 CG3H1E 16113578 IC50 = 220 nM T59604 CQ8Z4O 16113579 IC50 = 125 nM T59604 CTI61R 16113580 EC50 = 4 nM T59604 C3OGV4 16113581 IC50 = 120 nM T59604 C7H2GA 16113582 IC50 = 1700 nM T59604 CL98BH 16113583 IC50 = 580 nM T59604 CIQ6S3 16113584 IC50 = 2200 nM T59604 CD85FI 16113585 IC50 = 1000 nM T59604 C95IGA 16113691 IC50 = 15 nM T59604 C0A6WM 16113692 EC50 = 49 nM T59604 C4YLV6 16113693 EC50 = 18 nM T59604 CJ0D5P 16113694 IC50 = 140 nM T59604 C2T4OR 16113695 IC50 = 6 nM T59604 CJ43OU 16113710 EC50 = 5.4 nM T59604 C85YDF 16113796 IC50 = 120 nM T59604 CFQP15 16113797 IC50 = 150 nM T59604 C7U9GO 16113798 IC50 = 150 nM T59604 C6JU3V 16113799 IC50 = 83 nM T59604 CR63OJ 16113800 EC50 = 45 nM T59604 CQ02OX 16113902 IC50 = 11 nM T59604 CVO4T3 16113903 IC50 = 150 nM T59604 C9KMB0 16113904 IC50 = 12 nM T59604 CY29UJ 16113905 IC50 = 145 nM T59604 CFR8D6 16113906 EC50 = 140 nM T59604 C6OXS9 16114008 IC50 = 56 nM T59604 CFY8I0 16114009 IC50 = 130 nM T59604 CF16SW 16114010 IC50 = 55 nM T59604 CY2W6P 16114011 EC50 = 210 nM T59604 CJ4I2K 16114012 IC50 = 170 nM T59604 CM1LX9 16114096 IC50 = 0.5 nM T59604 C5U8PQ 16114097 EC50 = 5.3 nM T59604 CD9C6M 16114098 EC50 = 12 nM T59604 CO1QH0 16114099 IC50 = 28 nM T59604 C7IHG1 16114181 IC50 = 140 nM T59604 C58OIJ 16114183 IC50 > 1000 nM T59604 C4GV2E 16114184 IC50 = 173 nM T59604 CEH6N4 16114289 IC50 = 7 nM T59604 CRT04N 16114290 EC50 = 11 nM T59604 C1DS8N 16114292 IC50 = 0.3 nM T59604 CHQ5N8 16114403 IC50 = 23 nM T59604 CI0PQ3 16114404 IC50 = 32 nM T59604 CE4ZJ1 16114514 EC50 = 9.9 nM T59604 C3N6GQ 16114530 IC50 = 195 nM T59604 CFR8P6 16114531 IC50 = 240 nM T59604 CF0AE8 16114532 IC50 = 96 nM T59604 CSF23I 16134923 IC50 = 0.25 nM T59604 CSK20B 16202767 IC50 = 840 nM T59604 CHV75A 16203236 IC50 = 570 nM T59604 C5D0OB 16203237 EC50 = 23 nM T59604 CRTW49 16203238 EC50 = 41 nM T59604 C6KMR5 16203349 IC50 = 550 nM T59604 C9BHK2 16203569 IC50 = 62 nM T59604 C7U5FV 16203571 IC50 > 1000 nM T59604 CSH9C8 16203918 IC50 = 440 nM T59604 C8QC3F 16203930 IC50 = 110 nM T59604 C6UBC9 16204021 IC50 = 400 nM T59604 CPHM06 16204037 IC50 = 410 nM T59604 CE7Q6B 16204131 IC50 > 1000 nM T59604 CTQD10 16204133 IC50 > 1000 nM T59604 CIQU08 16204145 IC50 = 500 nM T59604 C4R7IG 16204226 IC50 = 470 nM T59604 CS28IM 16204229 IC50 = 700 nM T59604 CS70IJ 16204237 IC50 = 640 nM T59604 CZX82H 16204239 IC50 = 300 nM T59604 CD9A5X 16204241 IC50 = 310 nM T59604 C4SJB9 16204336 IC50 > 1000 nM T59604 CQD54B 16204343 IC50 = 640 nM T59604 CB7RM8 16204433 IC50 > 1000 nM T59604 C1D9TP 16752684 EC50 = 0.1585 nM T59604 C4AZ3J 16752689 EC50 = 125.89 nM T59604 CV46HZ 20600693 EC50 = 0.85 nM T59604 CXS09R 22862436 EC50 = 5 nM T59604 CWR42Q 22867441 EC50 = 0.6 nM T59604 CX8W0F 22888352 EC50 = 2 nM T59604 CXLY27 22888359 EC50 = 9.8 nM T59604 C4QSI5 22888379 EC50 = 19.7 nM T59604 CR01IA 22888395 EC50 = 7.6 nM T59604 CD5Y1W 22888424 EC50 = 3.4 nM T59604 C9XC7B 22888425 EC50 = 5.6 nM T59604 COJ8D5 22888428 EC50 = 14.4 nM T59604 CLYK60 22888433 EC50 = 4.9 nM T59604 CM1D8Q 22888474 EC50 = 0.46 nM T59604 C5X3IN 22888475 EC50 = 1.4 nM T59604 CZ3JV2 22888476 EC50 = 0.49 nM T59604 CL2XZ6 22888486 EC50 = 12 nM T59604 C7H6MC 23631026 EC50 = 6.5 nM T59604 CQ1M3P 23631387 IC50 = 52 nM T59604 CHU29W 23635235 Ki = 680 nM T59604 C5NO7V 23648232 IC50 = 759 nM T59604 CO2KQ7 23648233 IC50 > 1000 nM T59604 CCV54W 23648234 IC50 > 1000 nM T59604 CL3KB7 23648235 IC50 > 1000 nM T59604 CCER83 23648236 EC50 = 279 nM T59604 C0PJ1C 23648242 IC50 = 350 nM T59604 C0OPG8 23648244 EC50 = 2.5 nM T59604 C2EBF7 23648245 IC50 = 16 nM T59604 CNFQ62 23648246 IC50 = 130 nM T59604 C6EGQ3 23648249 EC50 = 2.3 nM T59604 CD0G8V 23648250 EC50 = 15 nM T59604 CAUC58 23649669 EC50 = 1.9 nM T59604 C73PIU 23656300 IC50 = 134 nM T59604 C8KO9M 23661656 EC50 = 4100 nM T59604 CU4T8D 23730225 EC50 = 3 nM T59604 CE3UN2 23730226 EC50 = 5.5 nM T59604 CD5U2Z 23730227 EC50 = 14.6 nM T59604 C1KX8D 23730228 EC50 = 3.8 nM T59604 C1YFU5 23730339 EC50 = 10.1 nM T59604 CK40WD 23730340 EC50 = 82.5 nM T59604 C4M6IA 23730341 EC50 = 3.3 nM T59604 CU7PS4 23730342 EC50 = 7.9 nM T59604 C69RSP 23730343 EC50 = 9.5 nM T59604 CG6TP5 23730458 EC50 = 45.3 nM T59604 CK2Q5J 24180592 Ki = 460 nM T59604 C7SMW5 24180646 EC50 = 79 nM T59604 C60NCW 24755624 EC50 = 0.7943 nM T59604 CU9B7S 24803347 EC50 = 3.981 nM T59604 C09HSR 24894012 EC50 = 0.27 nM T59604 C0P5DO 25010378 EC50 = 0.2 nM T59604 CHX91V 25022503 EC50 = 1.18 nM T59604 CCTG60 25022506 EC50 = 3.981 nM T59604 CMU30E 25022640 EC50 = 0.4 nM T59604 CK0X9U 25032438 Ki = 15 nM T59604 CY6DL8 25098836 EC50 = 2 nM T59604 CV9KH6 25190330 IC50 > 10000 nM T59604 CN35SM 25190383 Ki = 44 nM T59604 CH8RI6 25195191 EC50 > 5011.87 nM T59604 C62QAO 25195192 EC50 > 5011.87 nM T59604 CML1Y2 25211977 EC50 = 4 nM T59604 C3SYE2 25227441 IC50 = 0.078 nM T59604 C83ATJ 25260745 IC50 = 0.43 nM T59604 CZ49UK 25260749 IC50 = 0.31 nM T59604 C89RDC 25260900 IC50 = 2.9 nM T59604 CNR21Q 25260901 IC50 = 6.7 nM T59604 C3JB4O 25261382 IC50 = 1.3 nM T59604 C0BZJ4 25262608 IC50 = 44 nM T59604 CU64LE 25262771 IC50 = 27 nM T59604 C9AQI6 25262772 IC50 = 83 nM T59604 CAT4S5 42624368 IC50 > 2000 nM T59604 CW07AM 44235473 IC50 = 2770 nM T59604 CA1S7F 44281449 EC50 = 2.291 nM T59604 C6TEG2 44281450 EC50 = 4.467 nM T59604 C4DL8B 44281466 EC50 = 14.13 nM T59604 CM2PN4 44293091 EC50 = 21.88 nM T59604 CNT64H 44293557 EC50 = 10 nM T59604 CNDR48 44301387 EC50 = 378.1 nM T59604 C8BYR7 44301389 EC50 = 68.2 nM T59604 CC6XA2 44301462 EC50 = 448.5 nM T59604 C8RVG9 44301510 EC50 = 72 nM T59604 CPY84C 44301512 EC50 = 432.2 nM T59604 C35FWU 44336274 IC50 = 0.2 nM T59604 C7RNU6 44340007 Ki = 18 nM T59604 CY3KR2 44340008 Ki = 0.34 nM T59604 CS2V6M 44340268 Ki = 0.45 nM T59604 CNP5Q7 44357681 IC50 = 7.1 nM T59604 C53YHV 44368295 IC50 = 13.2 nM T59604 CE1V6K 44378837 IC50 = 67 nM T59604 CATD24 44378979 IC50 = 960 nM T59604 C9PZX8 44378981 IC50 = 200 nM T59604 C3MI5R 44378986 IC50 = 340 nM T59604 CK02CW 44379034 IC50 = 340 nM T59604 CF75ZD 44379072 IC50 = 1400 nM T59604 C2TR3U 44379301 IC50 = 3500 nM T59604 CKX5P3 44379303 IC50 = 48 nM T59604 CR40BF 44383343 IC50 = 190 nM T59604 CH20JT 44389131 IC50 = 4100 nM T59604 C0A3JZ 44389151 IC50 = 1900 nM T59604 CRP5G3 44389167 IC50 = 6300 nM T59604 CJD5A3 44389168 IC50 = 2200 nM T59604 CUND20 44389186 IC50 = 4000 nM T59604 CC59YF 44389187 IC50 = 18500 nM T59604 CC7B0N 44389192 IC50 = 860 nM T59604 CDX43V 44389215 IC50 = 6000 nM T59604 C7IT1W 44389216 IC50 = 4500 nM T59604 CG4IP9 44389221 IC50 > 10000 nM T59604 C8S2FN 44389222 IC50 > 10000 nM T59604 CS32WV 44389243 IC50 = 7500 nM T59604 C14EAB 44389248 IC50 = 3100 nM T59604 C6H5JB 44389249 IC50 > 10000 nM T59604 CV2LI4 44389262 IC50 = 1200 nM T59604 CAYW89 44389268 IC50 > 10000 nM T59604 CNU50S 44389271 IC50 > 100 nM T59604 C9HM6U 44389278 IC50 > 10000 nM T59604 CB7XS3 44389283 IC50 = 4700 nM T59604 CU57FZ 44390840 IC50 = 1.6 nM T59604 CRWC94 44390849 IC50 = 0.02 nM T59604 CMSQ24 44390860 IC50 = 15 nM T59604 C8P3CZ 44390862 IC50 = 0.24 nM T59604 C0LN3A 44390869 IC50 = 83 nM T59604 CXI52Q 44390871 IC50 = 4.2 nM T59604 C1E5LM 44390881 IC50 = 160 nM T59604 CJ7EY2 44390888 IC50 = 116 nM T59604 C56AGM 44390889 IC50 = 77 nM T59604 CYD1Q9 44390901 IC50 = 106 nM T59604 CEGR27 44390905 EC50 = 21 nM T59604 C85VNO 44390906 EC50 = 257 nM T59604 CMSB67 44390914 EC50 = 3.4 nM T59604 C76FQD 44390922 EC50 = 6.4 nM T59604 CPLC95 44390980 EC50 < 5 nM T59604 CD5O4B 44390986 EC50 = 2.1 nM T59604 CYLP68 44390996 EC50 = 1.5 nM T59604 CPMY25 44390997 EC50 = 41 nM T59604 CZYL89 44391002 EC50 = 20.9 nM T59604 CTNM61 44391003 EC50 = 17.8 nM T59604 CFXO86 44391007 EC50 = 190 nM T59604 CUX58C 44391008 EC50 = 19.6 nM T59604 C9TWS4 44391010 EC50 = 2.4 nM T59604 CJ8G3Y 44391015 EC50 = 45 nM T59604 CE90XM 44391020 EC50 = 27 nM T59604 C4RCW7 44391021 EC50 = 9.2 nM T59604 CBE9S6 44391024 EC50 = 9 nM T59604 CR1KY8 44391027 EC50 = 26.7 nM T59604 C4BZ3X 44391028 EC50 = 257 nM T59604 CVD75K 44391032 EC50 = 4.3 nM T59604 C3MG7O 44391035 EC50 = 43 nM T59604 CCL8I5 44391038 EC50 = 13.1 nM T59604 CDC4G0 44391039 EC50 = 0.66 nM T59604 CQ8GA6 44391040 EC50 = 21 nM T59604 C0R6JA 44391041 EC50 = 7.3 nM T59604 C0G2HS 44391048 EC50 = 219 nM T59604 CUTM09 44394833 IC50 = 15 nM T59604 C13ITZ 44394913 IC50 = 714 nM T59604 C0R3PY 44394930 IC50 = 162 nM T59604 C85FXK 44394947 IC50 = 47 nM T59604 CPI02V 44394974 IC50 = 29 nM T59604 CN76GO 44394982 IC50 = 3 nM T59604 C6R8ZF 44395002 IC50 = 139 nM T59604 CQ3SF5 44395020 IC50 = 103 nM T59604 CHB16Y 44396269 Ki = 1180 nM T59604 C32LQZ 44396306 Ki = 1920 nM T59604 C6VMK1 44396320 Ki = 910 nM T59604 CBJ45U 44396377 Ki = 1170 nM T59604 CNMA04 44396381 Ki = 1150 nM T59604 C6K1UW 44396384 Ki = 2630 nM T59604 C8JL9Z 44409455 IC50 = 690 nM T59604 CFEN21 44409536 IC50 = 1 nM T59604 CVS16R 44409611 IC50 = 137 nM T59604 CEU2B7 44409661 IC50 = 14 nM T59604 CLG34S 44409666 IC50 = 21 nM T59604 C85OXL 44409667 IC50 = 36 nM T59604 C42SDG 44409672 IC50 = 2.7 nM T59604 C0UEZ5 44409673 IC50 = 3.4 nM T59604 CB26CT 44409678 IC50 = 187 nM T59604 CE3P5U 44409679 IC50 = 3430 nM T59604 C6Z4TD 44409683 IC50 = 316 nM T59604 CL5QG4 44409684 IC50 = 5.5 nM T59604 CXP53Z 44409756 IC50 = 1.5 nM T59604 CT3EZ2 44409757 IC50 = 10 nM T59604 CID79S 44409758 IC50 = 5.4 nM T59604 CTH5F1 44409761 IC50 = 2480 nM T59604 CUA64R 44409762 IC50 = 354 nM T59604 C4P7RB 44409763 IC50 = 38 nM T59604 C75DFK 44409764 IC50 = 96 nM T59604 CY7H4Q 44409767 IC50 = 601 nM T59604 C7H9NR 44409770 IC50 = 66 nM T59604 CVP0N3 44409771 IC50 = 283 nM T59604 CLFC80 44409775 IC50 = 32 nM T59604 C20LGI 44409776 IC50 = 10 nM T59604 CBJ25N 44409785 IC50 = 57 nM T59604 CD84BX 44409801 IC50 = 11 nM T59604 CN5M7P 44409802 IC50 = 19 nM T59604 C8EDJ9 44409809 IC50 = 6 nM T59604 CXP6Z1 44409810 IC50 = 82 nM T59604 C5KD8R 44409821 IC50 = 2 nM T59604 CSGL98 44409831 IC50 = 180 nM T59604 CMU4O8 44409832 IC50 = 634 nM T59604 CGFX78 44409839 IC50 = 279 nM T59604 CJHO48 44409840 IC50 = 13 nM T59604 C9RMI5 44409864 IC50 = 69 nM T59604 CB3L8E 44409865 IC50 = 34 nM T59604 CPIF36 44409867 IC50 = 700 nM T59604 C3XY1N 44409868 IC50 = 248 nM T59604 C5BI1G 44409871 IC50 = 186 nM T59604 C28HBI 44409872 IC50 = 3250 nM T59604 C7TGZ8 44409946 IC50 = 41 nM T59604 CPHK59 44409975 IC50 = 69 nM T59604 CMFX65 44409979 IC50 = 192 nM T59604 CRXW67 44409980 IC50 = 244 nM T59604 CYW24G 44409989 IC50 = 38 nM T59604 CIM85O 44409990 IC50 = 5.2 nM T59604 CCHW29 44409994 IC50 = 19 nM T59604 C1Y9BM 44409998 IC50 = 7.5 nM T59604 C5Y6ZL 44410003 IC50 = 61 nM T59604 CE3AK8 44410007 IC50 = 65 nM T59604 CHS4P3 44410008 IC50 = 380 nM T59604 C5O2EZ 44410012 IC50 = 151 nM T59604 CY90GP 44410013 IC50 = 276 nM T59604 CM8NS3 44411584 EC50 = 4.786 nM T59604 CX8UH6 44411632 EC50 = 5.6 nM T59604 C7IF5J 44411634 EC50 = 2.089 nM T59604 CM5W7O 44411718 EC50 = 10 nM T59604 C4XRF0 44411720 EC50 = 8.5 nM T59604 C0EJN5 44411745 EC50 = 2 nM T59604 C4XQN6 44411753 EC50 = 2.692 nM T59604 CD67ZN 44411902 EC50 = 8.5 nM T59604 C8T3EY 44411905 EC50 = 6 nM T59604 CIWC39 44411913 EC50 = 57 nM T59604 CWQC39 44411920 EC50 = 1.3 nM T59604 C74FRH 44421230 IC50 = 520 nM T59604 CZXM91 44433201 IC50 > 1000 nM T59604 C0BAW6 44433202 IC50 > 1000 nM T59604 CO8MG3 44434007 EC50 = 43 nM T59604 CB8TW6 44434008 EC50 = 55 nM T59604 CKE95S 44434009 EC50 = 42 nM T59604 CBX24U 44434010 EC50 = 30 nM T59604 CPDS49 44434011 EC50 = 51 nM T59604 CHJD74 44434012 EC50 = 27 nM T59604 CBL0Q1 44434015 EC50 = 59 nM T59604 CH9T4L 44434016 EC50 = 49 nM T59604 CS5F1U 44434018 EC50 = 200 nM T59604 CV98TX 44434050 EC50 = 99 nM T59604 CTK43V 44434051 EC50 = 1120 nM T59604 CZCP60 44434052 EC50 = 259 nM T59604 CVBI34 44434053 EC50 = 116 nM T59604 CEKD38 44434054 EC50 = 868 nM T59604 CG0SE7 44434055 EC50 = 390 nM T59604 CR6K8O 44434056 EC50 = 426 nM T59604 C4SFH9 44434073 EC50 = 67 nM T59604 CA71NP 44434074 Ki = 2660 nM T59604 CEX1G5 44434076 EC50 = 147 nM T59604 C7XAT2 44434078 EC50 = 546 nM T59604 C4GZ7L 44434080 EC50 = 17 nM T59604 CN89OI 44434083 EC50 = 12 nM T59604 CDX6Z2 44434086 EC50 = 517 nM T59604 C17XZF 44434109 EC50 = 14 nM T59604 CM50KA 44434110 EC50 = 107 nM T59604 CRJB42 44434111 EC50 = 4 nM T59604 C93WND 44434112 EC50 = 150 nM T59604 C1RW8J 44434113 EC50 = 20 nM T59604 CG5BQ6 44434114 EC50 = 3170 nM T59604 CPW7T6 44434118 EC50 = 75 nM T59604 CM9S2J 44434119 EC50 = 347 nM T59604 C1IYT7 44434120 EC50 = 10 nM T59604 CVX30L 44434121 EC50 = 35 nM T59604 C47WIA 44434122 EC50 = 1860 nM T59604 CYP14C 44434123 EC50 = 29 nM T59604 CG5HP6 44434124 EC50 = 1520 nM T59604 C4G7MZ 44436807 IC50 = 138 nM T59604 C0V5AB 44436812 IC50 = 113 nM T59604 C1IZJ3 44436813 IC50 = 275 nM T59604 CHY84U 44436816 EC50 = 256 nM T59604 CBK90A 44436817 IC50 = 175 nM T59604 CE6HN1 44436828 IC50 = 9.5 nM T59604 C91XJV 44436829 IC50 = 32 nM T59604 CLK31M 44436831 IC50 = 44 nM T59604 C7YOX1 44436832 IC50 = 490 nM T59604 CV3KT1 44436833 IC50 > 1000 nM T59604 CB9Y1W 44436842 IC50 = 53 nM T59604 C4ON6U 44436850 EC50 = 1.6 nM T59604 C9FI7B 44436857 EC50 = 6.1 nM T59604 CGW4J7 44436868 IC50 = 468 nM T59604 C5XF8N 44436876 EC50 = 14 nM T59604 C9HWR1 44436881 IC50 = 255 nM T59604 CS49IW 44436882 EC50 = 183 nM T59604 C0B3MG 44436883 EC50 = 8.7 nM T59604 C3YWE7 44436884 EC50 = 12 nM T59604 CF7IT3 44436885 IC50 = 32 nM T59604 CRWI83 44436886 EC50 = 19.6 nM T59604 CAIF68 44436887 EC50 = 143 nM T59604 C1VO4A 44436888 IC50 = 6 nM T59604 CTKA41 44436889 IC50 = 18 nM T59604 C2HRY9 44436917 IC50 = 375 nM T59604 CTE08W 44437953 EC50 = 6.026 nM T59604 CU7W5D 44437955 EC50 = 1 nM T59604 CC8L3E 44437963 EC50 = 77 nM T59604 C4YDC1 44437966 EC50 = 30 nM T59604 CD25BO 44437969 EC50 = 30 nM T59604 C8J1OH 44437971 EC50 = 18 nM T59604 CE2S0F 44437979 EC50 = 0.28 nM T59604 CM8AY5 44444556 EC50 = 158.49 nM T59604 CW9LC3 44444557 EC50 = 125.89 nM T59604 CXYK84 44444558 EC50 = 39.81 nM T59604 C5GHI6 44444559 EC50 = 0.5012 nM T59604 CVL75O 44444560 EC50 = 31.62 nM T59604 CH8N6W 44444562 EC50 = 5.012 nM T59604 C2L6RI 44444563 EC50 = 0.1995 nM T59604 CA0EX4 44444564 EC50 = 19.95 nM T59604 CE4W5D 44444565 EC50 = 2.512 nM T59604 C6RI1A 44444566 EC50 = 3.162 nM T59604 CE5RN2 44444568 EC50 = 3.981 nM T59604 C7L8OG 44444570 EC50 = 63.1 nM T59604 C4YI8W 44444571 EC50 = 0.7943 nM T59604 CY5QN2 44444572 EC50 = 10 nM T59604 C15MKG 44444574 EC50 = 15.85 nM T59604 CE24TG 44445591 IC50 = 108 nM T59604 C4K1JA 44445592 IC50 = 11 nM T59604 CXS78T 44445593 IC50 = 60 nM T59604 C6RLF1 44445594 IC50 = 1.8 nM T59604 C0OB9Q 44445595 IC50 = 1.1 nM T59604 C4O3TW 44445596 IC50 = 33 nM T59604 C6WI0J 44445597 IC50 = 67 nM T59604 CVC8D2 44445598 IC50 = 49 nM T59604 C8BHU7 44445599 IC50 = 1.9 nM T59604 C8CQS1 44445600 IC50 = 0.7 nM T59604 CVDM94 44445601 IC50 = 105 nM T59604 CA7N0D 44445602 IC50 = 160 nM T59604 CS6JW0 44445603 IC50 = 58 nM T59604 CRT76Q 44445604 IC50 > 1000 nM T59604 CF9J8O 44445605 IC50 = 220 nM T59604 CDK82Q 44445606 IC50 = 34 nM T59604 C49ITN 44445607 IC50 = 120 nM T59604 CE8L5D 44445608 IC50 = 51 nM T59604 C96PSH 44445609 IC50 = 96 nM T59604 CWIY32 44445610 IC50 = 7.9 nM T59604 C7OD1G 44445611 IC50 = 3 nM T59604 C6H2AN 44445612 IC50 = 61 nM T59604 CH8O1Q 44445613 IC50 = 700 nM T59604 CSQ18J 44445614 IC50 = 480 nM T59604 CZW47S 44445615 IC50 = 29 nM T59604 CW08EF 44445616 IC50 = 76 nM T59604 C0YMX6 44445617 IC50 = 270 nM T59604 CH35WJ 44445618 IC50 = 177 nM T59604 CL5SN1 44445619 IC50 = 80 nM T59604 C1K4HU 44445620 EC50 = 16 nM T59604 CM09WI 44445621 IC50 > 1000 nM T59604 C3FJX6 44445622 IC50 = 112 nM T59604 C18GVK 44445624 IC50 = 140 nM T59604 C9C2VA 44445625 IC50 = 18.5 nM T59604 CL7VY1 44445626 IC50 = 5 nM T59604 C5W0YR 44445627 IC50 = 14 nM T59604 CPT7N8 44445628 IC50 = 89 nM T59604 C2H8TW 44445629 IC50 = 300 nM T59604 CP1QF3 44446137 IC50 = 140 nM T59604 C2WYK3 44446140 IC50 > 1000 nM T59604 CE3G4V 44446143 IC50 > 1000 nM T59604 C7WZ6E 44446148 IC50 = 450 nM T59604 C3UM2W 44446150 IC50 > 1000 nM T59604 CP73DI 44446152 IC50 > 1000 nM T59604 CCON73 44446154 IC50 > 1000 nM T59604 C9TY3J 44446157 IC50 = 450 nM T59604 C7ZNF8 44446175 IC50 = 800 nM T59604 C6J4VA 44446177 EC50 = 32 nM T59604 C19UPX 44446178 EC50 = 88 nM T59604 CYE3V6 44446187 EC50 = 75 nM T59604 C5TF6G 44446188 EC50 = 1580 nM T59604 CRHA84 44446189 EC50 = 24 nM T59604 C9WB8K 44446190 EC50 = 24 nM T59604 CHQI08 44447839 EC50 = 0.42 nM T59604 C57ZXB 44447840 EC50 = 1.6 nM T59604 CN7P0S 44447841 EC50 = 0.61 nM T59604 CF7ED5 44447842 EC50 = 6.75 nM T59604 C3V1TO 44447843 EC50 = 0.72 nM T59604 CB4YK8 44447844 EC50 = 1.79 nM T59604 C9LCW5 44447845 EC50 = 34 nM T59604 CHW3R7 44447846 EC50 = 3.1 nM T59604 C5XNV0 44447848 EC50 = 33.2 nM T59604 C24VRW 44447850 EC50 = 1.26 nM T59604 C87OWH 44447852 EC50 = 0.51 nM T59604 C5RFG7 44447853 EC50 = 1.11 nM T59604 CBF75I 44447854 EC50 = 1.66 nM T59604 C5PNS2 44447855 EC50 = 0.34 nM T59604 CK1QX4 44447856 EC50 = 1.04 nM T59604 C4ZC3O 44447857 EC50 = 0.45 nM T59604 CUT47D 44449864 EC50 = 3 nM T59604 CZU9Y0 44449891 EC50 = 0.9 nM T59604 C13VTX 44449922 EC50 = 2.9 nM T59604 C1AQ4F 44449923 EC50 = 105 nM T59604 CC0FR8 44449924 EC50 = 521 nM T59604 C0V8JF 44449955 EC50 = 0.2 nM T59604 CIX4J9 44449956 EC50 = 3.1 nM T59604 C0O9SE 44449987 EC50 = 0.2 nM T59604 C3NQW9 44449988 EC50 = 0.7 nM T59604 CA67EK 44450015 EC50 = 1.3 nM T59604 C40TMA 44450016 EC50 = 0.6 nM T59604 C5XJE2 44450017 EC50 = 1.8 nM T59604 CKP79S 44450044 EC50 = 40 nM T59604 CN0C2P 44450045 EC50 = 27 nM T59604 CG5FL6 44450046 EC50 = 3.3 nM T59604 C0SD3B 44450070 EC50 = 204 nM T59604 C6S8YR 44450071 EC50 = 140 nM T59604 CCUH90 44450100 EC50 = 8.4 nM T59604 C9JZX1 44450101 EC50 = 0.64 nM T59604 C4SCA9 44450102 EC50 = 11 nM T59604 C3DG5S 44450103 EC50 = 4.1 nM T59604 CM3LC9 44450104 EC50 = 1.4 nM T59604 C0LOA1 44450105 EC50 = 33 nM T59604 CU1I0E 44450132 EC50 = 4.4 nM T59604 C61EIS 44450133 EC50 = 14.7 nM T59604 C9Y4QK 44450134 EC50 = 32 nM T59604 CF4WP5 44450135 EC50 = 23 nM T59604 C0H1PK 44450137 EC50 = 70 nM T59604 C45JKU 44450169 EC50 = 26 nM T59604 CL5I7Z 44452749 EC50 = 0.3981 nM T59604 C8EX9A 44452750 EC50 = 1.995 nM T59604 CV52TF 44452776 EC50 = 125.89 nM T59604 C6C9KF 44452777 EC50 = 39.81 nM T59604 C8R3DW 44452778 EC50 = 794.33 nM T59604 CX4RI1 44452806 EC50 = 100 nM T59604 C6N7KC 44452825 EC50 = 39.81 nM T59604 CXJ24Q 44452826 EC50 = 39.81 nM T59604 CIF7L4 44452827 EC50 = 630.96 nM T59604 CM3SB0 44452885 EC50 = 100 nM T59604 CTY80L 44452887 EC50 = 158.49 nM T59604 CWNM19 44452929 EC50 = 19.95 nM T59604 CCZF71 44452932 EC50 = 1.995 nM T59604 C6M5SL 44453070 EC50 = 316.23 nM T59604 CN54QX 44453097 EC50 = 316.23 nM T59604 CZL3X4 44453123 EC50 = 0.5012 nM T59604 CV13SO 44454060 EC50 = 0.8 nM T59604 C56TGO 44454092 EC50 = 19 nM T59604 C8L7PU 44454117 EC50 = 0.5 nM T59604 CZ6K7I 44454302 EC50 = 23 nM T59604 CPM4W2 44454303 EC50 = 0.3 nM T59604 C3O4BS 44454304 EC50 = 19 nM T59604 C83YHV 44454337 EC50 = 0.4 nM T59604 C30CSY 44454338 EC50 = 19 nM T59604 CZ21VY 44454367 EC50 = 0.6 nM T59604 C46EKP 44454368 EC50 = 302 nM T59604 CTJ75W 44454397 EC50 = 2470 nM T59604 C2B4SN 44454398 EC50 = 27 nM T59604 C1PGK4 44454399 EC50 = 22 nM T59604 CDF7M8 44454432 EC50 = 150 nM T59604 CSX29M 44560945 EC50 = 0.9 nM T59604 C5QLC6 44570698 EC50 = 19.95 nM T59604 CHD4F5 44570699 EC50 = 3.981 nM T59604 C9KD1J 44570700 EC50 = 1.995 nM T59604 CX86AU 44570702 EC50 = 2.512 nM T59604 CQ5X3W 44570761 EC50 = 31.62 nM T59604 C2Z3HJ 44570762 EC50 = 316.23 nM T59604 C4D0AV 44570763 EC50 = 1 nM T59604 C17ONP 44570764 EC50 = 0.3162 nM T59604 C84LHN 44570765 EC50 = 0.3981 nM T59604 CE15GU 44570920 EC50 = 7.943 nM T59604 CWF7R1 44570921 EC50 = 15.85 nM T59604 C61CHS 44570922 EC50 = 398.11 nM T59604 CPAI69 44570923 EC50 = 31.62 nM T59604 CTN23G 44570960 EC50 = 0.2512 nM T59604 CP46TB 44570961 EC50 = 3.162 nM T59604 C53BQS 44570962 EC50 = 0.05012 nM T59604 C9ZW2M 44570963 EC50 = 0.1585 nM T59604 C37FQE 44570964 EC50 = 15.85 nM T59604 CUZ8G1 44570965 EC50 = 1.259 nM T59604 C5HZ8J 44570966 EC50 = 0.5012 nM T59604 CG58BJ 44570967 EC50 = 5.012 nM T59604 CKS86A 44571002 EC50 = 0.1995 nM T59604 C2B7WE 44571003 EC50 = 6.31 nM T59604 C3AWE9 44571004 EC50 = 10 nM T59604 CJB06H 44571005 EC50 = 7.943 nM T59604 C6JB2C 44576254 IC50 > 1000 nM T59604 C5TF9Y 44576256 IC50 = 0.25 nM T59604 CD3T1I 44577060 Ki = 240 nM T59604 CVS6Q8 44579640 EC50 = 4000 nM T59604 C6D3LJ 44579641 EC50 = 2000 nM T59604 CCY9F0 44579643 EC50 = 90 nM T59604 C2ZJM0 44579686 EC50 = 4000 nM T59604 CHY2F7 44579752 EC50 = 14000 nM T59604 CVH40U 44579753 EC50 > 10000 nM T59604 C5AHW3 44579754 EC50 > 10000 nM T59604 CDT3M9 44579755 EC50 = 900 nM T59604 CC8AI0 44579756 EC50 = 7 nM T59604 C0MH7I 44579774 EC50 >= 10 nM T59604 C4WN7B 44579775 EC50 = 40 nM T59604 C87QLB 44579776 EC50 = 80 nM T59604 CE9U6O 44579777 EC50 = 150 nM T59604 C2YS5Q 44579778 EC50 = 50 nM T59604 CPM02Q 44579801 EC50 = 220 nM T59604 C5U4QZ 44579802 EC50 = 10 nM T59604 CC5PZ6 44579803 EC50 = 260 nM T59604 CNH16J 44579804 EC50 = 60 nM T59604 C4HIN8 44579805 EC50 = 20 nM T59604 CG2JM1 44579821 EC50 = 140 nM T59604 CY5V2L 44579822 EC50 = 90 nM T59604 C7P8JA 44579823 EC50 = 3 nM T59604 C15AZN 44579824 EC50 = 120 nM T59604 CERM69 44579840 EC50 = 20 nM T59604 CKB1J3 44579841 EC50 = 30 nM T59604 CO3J8L 44579842 EC50 = 1260 nM T59604 CA7W8Q 44579843 EC50 = 90 nM T59604 C34IHS 44579844 EC50 >= 10 nM T59604 C4CA5O 44579857 EC50 = 200 nM T59604 CDE7M9 44579858 EC50 = 50 nM T59604 CNM2G5 44579859 EC50 >= 10 nM T59604 C69CYU 44579860 EC50 = 250 nM T59604 CB79UF 44579861 EC50 = 120 nM T59604 CAG89V 44579879 EC50 = 140 nM T59604 C78VMJ 44579880 EC50 = 30 nM T59604 CB01KP 44579881 EC50 = 780 nM T59604 CT2H0M 44579882 EC50 = 40 nM T59604 C4Y5HF 44579883 EC50 = 120 nM T59604 C7NZY6 44579906 EC50 = 1200 nM T59604 C6C1JT 44579907 EC50 = 20 nM T59604 CLR28I 44579908 EC50 = 1500 nM T59604 C6NB2S 44579909 EC50 = 180 nM T59604 CL7VA5 44579919 EC50 = 2000 nM T59604 CH85UT 44579958 EC50 = 1000 nM T59604 CD5KM4 44579959 EC50 = 600 nM T59604 CNZ5W9 44579995 EC50 > 10000 nM T59604 CBTA01 44579996 EC50 = 2000 nM T59604 CGN8D7 44579998 EC50 > 10000 nM T59604 C4L7TJ 44580028 EC50 = 5000 nM T59604 C79IVU 44580029 EC50 > 10000 nM T59604 CXJY26 44580030 EC50 = 440 nM T59604 C9Q5LO 44580031 EC50 = 330 nM T59604 CMX14O 44580032 EC50 = 9000 nM T59604 C4AMJ8 44582533 IC50 = 55000 nM T59604 C7KBO6 44582534 IC50 = 889000 nM T59604 CQI0D4 45102707 EC50 > 10000 nM T59604 CSEP-69 45102708 EC50 > 1000 nM T59604 C7FSM2 46865987 IC50 = 12.2 nM T59604 CTEA12 46880461 IC50 = 25 nM T59604 CK8A1O 46880462 IC50 = 12 nM T59604 C9KDP4 46880463 IC50 = 640 nM T59604 CEQ6V4 46880495 IC50 = 280 nM T59604 CISM52 46880496 IC50 = 68 nM T59604 C8ZSM3 46880497 IC50 = 6500 nM T59604 CODR73 46880498 IC50 = 46.5 nM T59604 CHJ5Y6 46880566 IC50 = 77 nM T59604 CE9PG2 46880567 IC50 = 147 nM T59604 C01PGO 46880568 IC50 = 6 nM T59604 CS7L4X 46880569 IC50 = 26 nM T59604 C0PXY7 46880628 IC50 = 9.1 nM T59604 CD37LU 46880629 IC50 = 2.1 nM T59604 CUY89F 46880630 IC50 = 4.1 nM T59604 C4P6XS 46880631 IC50 = 2.9 nM T59604 CJ53KF 46880672 IC50 = 7 nM T59604 CYJC08 46880673 IC50 = 136 nM T59604 C1RI9O 46880674 IC50 = 64 nM T59604 CJ5LO0 46880675 IC50 = 17.7 nM T59604 COT5L9 46880724 IC50 = 14.3 nM T59604 C8TW5J 46880725 IC50 = 9 nM T59604 CMUZ29 46880726 IC50 = 20 nM T59604 CMS56Q 46880727 IC50 = 13 nM T59604 CA1V5O 46880770 IC50 = 37.2 nM T59604 CE1OL2 46880771 IC50 = 33.7 nM T59604 CEXW19 46880772 IC50 = 12.7 nM T59604 CE57JN 46880773 IC50 = 42.2 nM T59604 CT1S6C 46880811 IC50 = 143 nM T59604 C6OX9Z 46880812 IC50 = 65 nM T59604 CB1VX9 46880813 IC50 = 244.6 nM T59604 C6CS2B 46880814 IC50 = 123 nM T59604 C6PCS9 46880844 IC50 = 338.7 nM T59604 CJOU53 46880845 IC50 = 42 nM T59604 C2EFB5 46880846 IC50 = 31 nM T59604 C0LJP6 46882103 IC50 = 108 nM T59604 CX1KS6 46882104 IC50 = 310 nM T59604 CB67WR 46882105 IC50 = 444 nM T59604 CH5T9E 46882106 IC50 = 625 nM T59604 CR2C3J 46882152 IC50 = 429 nM T59604 C3KSB8 46882153 IC50 = 682 nM T59604 C39QLM 46882154 IC50 = 5615 nM T59604 C2QM9K 46882155 IC50 = 1649 nM T59604 C43CSF 46882156 IC50 = 846 nM T59604 CE9Z1W 46882196 IC50 = 474 nM T59604 CJ9GQ6 46882197 IC50 = 241 nM T59604 CA18GZ 46882198 IC50 = 97 nM T59604 C6OY8D 46882199 IC50 = 263 nM T59604 C0AU3L 46882236 IC50 = 128 nM T59604 CNZI39 46882237 IC50 = 138 nM T59604 C4YUO1 46882238 IC50 = 161 nM T59604 CGTQ20 46882239 IC50 = 69 nM T59604 CMEL41 46882270 IC50 = 77 nM T59604 CFL3C6 46882271 IC50 = 14 nM T59604 CAVT63 46882272 IC50 = 8 nM T59604 C0IF2Y 46882273 IC50 = 28 nM T59604 CIGP20 46882302 EC50 > 1000 nM T59604 CJG6E9 46882303 EC50 > 1000 nM T59604 CW2Z0V 46882305 IC50 = 16 nM T59604 C9IDW2 46882306 IC50 = 21 nM T59604 C20XKF 46882307 IC50 = 2 nM T59604 C69AMR 46882349 EC50 > 10000 nM T59604 CFZV45 46882350 EC50 > 1000 nM T59604 CSF43I 46882393 EC50 > 1000 nM T59604 CB3QV6 46882394 EC50 = 3.981 nM T59604 C01GKH 46882395 EC50 = 3.981 nM T59604 CX7D3V 46882396 EC50 = 19.95 nM T59604 C4BH9E 46882458 EC50 = 79.43 nM T59604 CJ69NR 46882460 EC50 > 1000 nM T59604 C3FA8G 46882519 EC50 > 10000 nM T59604 CF8IJ2 46882520 EC50 = 79.43 nM T59604 CQN87I 46882521 EC50 = 1584.89 nM T59604 C56ULO 46882522 EC50 = 158.49 nM T59604 CRZ95W 46882582 EC50 = 630.96 nM T59604 CX72IN 46882583 EC50 > 10000 nM T59604 CHS14B 46882671 EC50 > 1000 nM T59604 C2OU8F 46882673 EC50 > 10000 nM T59604 CP84OR 46882710 EC50 > 10000 nM T59604 CPFM68 46882711 EC50 > 10000 nM T59604 CC05XO 46882712 EC50 > 10000 nM T59604 CL3EI9 46882713 EC50 > 10000 nM T59604 CZ15LN 46882714 EC50 > 1000 nM T59604 CD24US 46882752 EC50 > 1000 nM T59604 CAN69D 46882753 EC50 > 1000 nM T59604 C0RQA4 46882754 EC50 > 1000 nM T59604 CBXT24 46882756 EC50 > 1000 nM T59604 C4DLJ2 46882763 IC50 = 40 nM T59604 CH6G4Q 46882766 IC50 = 272 nM T59604 C39WEJ 46882794 EC50 > 1000 nM T59604 CTJ41Q 46882795 EC50 > 1000 nM T59604 C4OZ1U 46882796 EC50 > 1000 nM T59604 CDK0Q3 46882797 EC50 > 1000 nM T59604 CMC4E5 46882804 IC50 = 46 nM T59604 CCUI47 46882805 IC50 = 30 nM T59604 C3NSG9 46882807 IC50 = 1715 nM T59604 C4OQ6D 53248756 Ki = 22 nM T59604 C28QUB 53373577 Ki = 3.311 nM T59604 CC8Q1D 53390181 IC50 = 12.59 nM T59604 CV0P1K 53390538 IC50 = 30.2 nM T59604 CZ0WI6 53391301 IC50 = 37.15 nM T59604 C7XZ1I 54458823 EC50 = 3 nM T59604 CP1W5M 56926173 EC50 = 68 nM T59604 C30RQU 56926461 Ki = 6 nM T59604 C9IEJ8 56942098 IC50 = 4 nM T59604 C6AZ3E 56942099 Ki = 8 nM T59604 CCF90X 56942242 Ki = 0.8 nM T59604 C2AT0L 56942243 Ki = 2 nM T59604 C7ZF9T 56942244 Ki = 12 nM T59604 CX3L9I 56942385 Ki = 46 nM T59604 CVE3F7 56942387 IC50 = 43 nM T59604 CO9KV2 56942388 Ki = 17 nM T59604 CM7PW5 56942535 Ki = 46 nM T59604 CW4QD9 57345597 Ki = 2 nM T59604 CBQK82 57345598 Ki = 3.1 nM T59604 C3REK0 57345599 Ki = 0.2 nM T59604 CX49PE 57345600 Ki = 0.16 nM T59604 CI9UT0 57391292 Ki = 3.1 nM T59604 CH67TI 57391293 Ki = 0.4 nM T59604 C78LTO 57391294 Ki = 3.4 nM T59604 CGB71E 57393073 Ki = 0.1 nM T59604 CRE41N 57394797 Ki = 6.6 nM T59604 CS41PI 57394881 Ki = 0.05 nM T59604 C3D4AH 57394882 Ki = 5 nM T59604 CKDZ14 57398339 Ki = 0.9 nM T59604 CSA36Q 57398340 Ki = 0.01 nM T59604 CE5JQ8 57398341 Ki = 0.2 nM T59604 C7NE4P 57398342 Ki = 0.26 nM T59604 C8Y4UJ 57398343 Ki = 1.9 nM T59604 C8CG2S 57399248 Ki = 1 nM T59604 C18OVS 57400002 Ki = 0.01 nM T59604 CJO70A 57400003 Ki = 2.6 nM T59604 CL2IT5 57401797 Ki = 1.7 nM T59604 CKA34L 57401798 Ki = 6.7 nM T59604 CM15JF 57401799 Ki = 0.3 nM T59604 CGS82D 57401800 Ki = 0.5 nM T59604 CF0CA4 57401801 Ki = 0.6 nM T59604 C53DGY 57401802 Ki = 1.5 nM T59604 C8VI1X 57401803 Ki = 0.27 nM T59604 CX6JR2 57422673 IC50 = 23 nM T59604 CD40CR 57422686 IC50 = 0.15 nM T59604 CRI4K2 57422687 IC50 = 0.29 nM T59604 C6JZ4C 57422688 IC50 = 0.67 nM T59604 CR8S3Q 57422690 IC50 = 0.53 nM T59604 CYSA42 57422692 IC50 = 0.33 nM T59604 CO85NH 57422695 IC50 = 3.9 nM T59604 CTS3E6 57422696 IC50 = 15 nM T59604 CW92IZ 57422697 IC50 = 120 nM T59604 C43BGV 57422730 IC50 = 13 nM T59604 CO1KA7 57422749 IC50 = 65 nM T59604 C2IO0J 57422760 IC50 = 8.7 nM T59604 CSF86Y 57422761 IC50 = 8.6 nM T59604 CJO7S5 57422768 IC50 = 0.48 nM T59604 C03XVS 57422776 IC50 = 5.1 nM T59604 CK1BZ0 57422789 IC50 = 1.3 nM T59604 C59DSI 57422791 IC50 = 8.8 nM T59604 CKMP13 57422792 IC50 = 0.31 nM T59604 CBY54J 57422793 IC50 = 0.62 nM T59604 C2U1VH 57422817 IC50 = 0.77 nM T59604 CH9ZJ5 57785733 IC50 = 0.69 nM T59604 C39VTY 57785737 IC50 = 4.2 nM T59604 CY3NF5 57797614 IC50 = 11 nM T59604 CZ6Q9X 57797640 IC50 = 2 nM T59604 C54DIC 58438451 Ki = 10.47 nM T59604 CPI4W9 58438460 Ki = 12.88 nM T59604 C9UK7P 58438475 Ki = 6.31 nM T59604 CBCA81 58438487 Ki = 9.12 nM T59604 C1FM5N 59446099 IC50 > 10000 nM T59604 CV52YE 59446101 IC50 = 1200 nM T59604 C0V5UB 59446102 IC50 > 10000 nM T59604 C9S1IF 59446103 IC50 > 10000 nM T59604 CS92LO 59446104 IC50 > 10000 nM T59604 C3KB2O 59446107 IC50 = 1340 nM T59604 CQE13H 59446108 IC50 > 10000 nM T59604 C8PKR2 59446111 IC50 > 10000 nM T59604 CS3JD0 59446113 IC50 > 10000 nM T59604 CRJ38P 59446116 IC50 = 51000 nM T59604 C0INX9 59446117 IC50 > 10000 nM T59604 CL50PI 59446120 IC50 = 771 nM T59604 C2G6QX 59446121 IC50 > 10000 nM T59604 CHZQ39 59446122 IC50 > 10000 nM T59604 C3OG9S 59446123 IC50 > 10000 nM T59604 CHNR24 59446125 IC50 > 10000 nM T59604 CP07SK 59446126 IC50 > 10000 nM T59604 CZIC40 59446128 IC50 > 10000 nM T59604 CA0W9Q 59446130 IC50 = 19500 nM T59604 C6QMA8 59446134 IC50 > 10000 nM T59604 CX5Y1T 59446135 IC50 = 808 nM T59604 C7OCA4 59446138 IC50 = 723 nM T59604 CU03SE 59446139 IC50 = 11200 nM T59604 CRQB10 59446141 IC50 = 3740 nM T59604 C29SIX 59446142 IC50 > 10000 nM T59604 CA03QR 59446143 IC50 = 45000 nM T59604 C7IPK4 59446145 IC50 = 568 nM T59604 CU17OY 59446146 IC50 > 10000 nM T59604 CTYL12 59446149 IC50 > 10000 nM T59604 C7OB4H 59446150 IC50 = 3250 nM T59604 CP42MS 59446154 IC50 = 8170 nM T59604 CLV4J8 60165265 IC50 = 38 nM T59604 CYH80K 60194838 IC50 > 10000 nM T59604 CD8S1Q 60194839 IC50 > 10000 nM T59604 CG28AQ 60195018 IC50 = 3860 nM T59604 C5CXK6 60195019 IC50 = 3610 nM T59604 C2GWS0 60195020 IC50 = 5410 nM T59604 C9QK5Y 60195112 IC50 = 1170 nM T59604 CZ7MK5 60195113 IC50 = 4550 nM T59604 CV6XG5 60195114 IC50 = 85600 nM T59604 C45OTP 60195115 IC50 > 10000 nM T59604 CP4RF0 60195284 IC50 = 16100 nM T59604 CW51MB 60195285 IC50 = 465 nM T59604 CX7M6C 60195286 IC50 = 729 nM T59604 CXQ0J6 60195379 IC50 = 1640 nM T59604 C2FPA0 60195645 IC50 > 10000 nM T59604 C4NEG2 60195731 IC50 > 10000 nM T59604 C2YO0F 66601728 IC50 = 7 nM T59604 CT9B1S 66788278 IC50 = 2 nM T59604 C78XLS 66813470 IC50 = 200 nM T59604 C4UP0J 67405379 Ki = 3.981 nM T59604 C7M8VC 67406334 Ki = 4.571 nM T59604 CPV39L 67406727 Ki = 9.2 nM T59604 CU32ZC 67407161 Ki = 15.49 nM T59604 C3GSR6 67407808 Ki = 9.12 nM T59604 CWY79V 67408128 Ki = 7.413 nM T59604 C3BHE6 67410074 Ki = 15.49 nM T59604 C8LM1Q 67457995 EC50 = 0.6 nM T59604 CM3PW8 70681018 IC50 = 3 nM T59604 CMDT94 70681019 IC50 = 79 nM T59604 CY0IK4 70681020 IC50 = 196 nM T59604 C87FCB 70681021 IC50 = 2.5 nM T59604 C5D2MP 70681022 IC50 = 16.5 nM T59604 CN4G3U 70681025 IC50 > 10000 nM T59604 C3J9KZ 70682036 Ki = 14 nM T59604 CKSP64 70682037 IC50 = 4.6 nM T59604 C16WKZ 70683143 IC50 = 28 nM T59604 CHPA96 70683144 IC50 > 10000 nM T59604 CAKY84 70683149 IC50 = 50 nM T59604 CD5TR3 70684154 IC50 = 231 nM T59604 C79PIV 70684155 Ki = 27 nM T59604 C97XVQ 70685218 IC50 = 171 nM T59604 C4O8XG 70685219 IC50 = 4.1 nM T59604 CK8A6W 70685225 IC50 = 3 nM T59604 C1P4OY 70686292 IC50 = 25 nM T59604 CJ2UM8 70686293 Ki = 14 nM T59604 C8RP9Q 70687379 IC50 = 143 nM T59604 CL1WU4 70687380 IC50 = 8 nM T59604 C5QG9Y 70687383 IC50 = 6 nM T59604 CS0HG6 70688404 IC50 = 211 nM T59604 CN7RS4 70689440 IC50 = 7 nM T59604 CGRS90 70689441 IC50 = 20 nM T59604 CCI32L 70690449 Ki = 20 nM T59604 C1AC0G 70691550 IC50 = 0.2 nM T59604 CF8I9T 70691551 IC50 = 1 nM T59604 C8ZI6D 70691552 IC50 = 2.5 nM T59604 C27NFD 70692600 Ki = 14 nM T59604 C8ST6F 70692601 Ki = 11 nM T59604 COI36G 70692602 Ki = 114 nM T59604 CKSH84 70692603 Ki = 25 nM T59604 CM3T7V 70693640 IC50 = 26 nM T59604 CH8GC3 70693641 IC50 = 12 nM T59604 C5LQ9B 70693643 IC50 > 10000 nM T59604 CB4F0R 70693644 IC50 = 7 nM T59604 CG5QA4 70694647 IC50 = 2980 nM T59604 CLK3G6 70694648 Ki = 52 nM T59604 CBX49P 70694649 Ki = 23 nM T59604 C93XHS 70695747 Ki = 4.4 nM T59604 CG0QY5 70695748 IC50 = 314 nM T59604 C62ZQG 70695749 IC50 = 313 nM T59604 CAH70F 70696687 Ki = 152 nM T59604 CI62QY 70696688 Ki = 17 nM T59604 C94JEF 70696689 Ki = 206 nM T59604 CK2T6G 71449740 IC50 = 220 nM T59604 CC6Z0B 71449752 IC50 > 10000 nM T59604 CXZ4K1 71449753 IC50 = 2540 nM T59604 C4BT1J 71449838 EC50 = 168.6 nM T59604 CHNV45 71449843 EC50 > 1000 nM T59604 CZBF56 71451551 IC50 = 129 nM T59604 C7A5LH 71451563 IC50 = 24 nM T59604 CSQF84 71451564 IC50 = 251 nM T59604 CL8V0U 71451652 EC50 > 1000 nM T59604 C0IBC7 71452183 Ki = 100 nM T59604 CN08XO 71453389 IC50 > 10000 nM T59604 CWK3J2 71453390 IC50 = 38 nM T59604 C1XR4A 71453391 IC50 = 25 nM T59604 CTIF57 71453392 IC50 = 110 nM T59604 CY7CZ1 71453404 IC50 = 47 nM T59604 C5KO6D 71453405 IC50 = 700 nM T59604 CTME20 71453485 EC50 = 624.4 nM T59604 CR2F8D 71453488 EC50 = 6.7 nM T59604 C7WR4T 71453489 EC50 = 2.8 nM T59604 C5J9NH 71455085 IC50 = 64 nM T59604 CURV69 71455104 IC50 > 10000 nM T59604 C7IX2J 71455105 IC50 = 140 nM T59604 CK3OR6 71455106 IC50 = 525 nM T59604 CU8BM9 71455196 EC50 > 1000 nM T59604 C5GBY7 71455197 EC50 = 9.4 nM T59604 CBN67Z 71456897 IC50 = 1 nM T59604 CD2RP7 71456910 IC50 = 110 nM T59604 CU30QE 71456984 EC50 = 183.7 nM T59604 CD3X1J 71456992 EC50 = 5.7 nM T59604 C39NDE 71458746 IC50 = 1160 nM T59604 COF8H7 71458747 IC50 = 213 nM T59604 CUJ34O 71458847 Ki = 31.3 nM T59604 CH8UP0 71458848 EC50 = 240.9 nM T59604 C2REN0 71458849 Ki = 22.1 nM T59604 C5FG2U 71458850 EC50 = 96.8 nM T59604 CHT38B 71458859 EC50 = 13.1 nM T59604 CFT7E2 71460564 IC50 = 1470 nM T59604 CEW73V 71460565 IC50 = 1180 nM T59604 CY3R0Z 71460566 IC50 > 10000 nM T59604 CW7EY5 71460576 IC50 = 1390 nM T59604 CDXZ12 71460577 IC50 = 273 nM T59604 CU6M4L 71460578 IC50 = 111 nM T59604 C3OLW2 71460658 Ki = 34.9 nM T59604 C1OPU6 71460659 EC50 = 2.1 nM T59604 CCV93Y 71460664 EC50 = 119.6 nM T59604 CT79JP 71460665 EC50 = 498.1 nM T59604 CVJY40 71462272 IC50 = 239 nM T59604 C1UQO9 71462273 IC50 = 47 nM T59604 C8Q0SD 71462274 IC50 = 2780 nM T59604 CE7J5X 71462275 IC50 > 10000 nM T59604 COLZ61 71462276 IC50 > 10000 nM T59604 C9W5VI 71462373 EC50 > 1000 nM T59604 CEO4H0 71462380 EC50 = 124.1 nM T59604 CK7Z6F 71462381 EC50 = 17.9 nM T59604 C6Y4WM 71462382 EC50 = 161.3 nM T59604 CE2BA8 71716660 EC50 = 0.7943 nM T59604 CEX25Q 72190449 Ki = 275.42 nM T59604 C79XFZ 72190450 IC50 = 1096.48 nM T59604 C7NYG0 72190451 Ki = 25.12 nM T59604 C6PE7F 72190452 Ki = 1380.38 nM T59604 CN4D2K 72191050 Ki = 27.54 nM T59604 CL1A6K 72191051 Ki = 16.22 nM T59604 C4J7PB 73346226 Ki = 3630.78 nM T59604 CUR4F2 73346227 Ki < 20892.96 nM T59604 C2B1GF 73347725 IC50 = 15.85 nM T59604 CCI07X 73350118 IC50 = 12 nM T59604 CBX06Q 73350846 Ki = 25118.86 nM T59604 C2TK7H 73352329 Ki = 1122.02 nM T59604 C93IHF 73352330 Ki < 29512.09 nM T59604 CL8T4U 73355325 Ki = 1698.24 nM T59604 CD63YS 73356869 Ki < 30199.52 nM T59604 CB4Y7R 89768546 IC50 = 6500 nM T59604 C4OP6C 90644553 Ki = 10.47 nM T59604 CF0MJ8 90644554 Ki = 69.18 nM T59604 CG4E8W 90665845 IC50 = 0.12 nM T59604 C1S7YU 90665846 IC50 = 1.5 nM T59604 C8B1RN 90665847 IC50 = 0.28 nM T59604 CCQ67W 90665848 IC50 = 16 nM T59604 C2DF8V 90665849 IC50 = 59 nM T59604 CGB7U8 90665850 IC50 = 1.1 nM T59604 C67YNO 90665851 IC50 = 1.1 nM T59604 C2E6NI 90665852 IC50 = 12 nM T59604 C97PUB 90666011 IC50 = 7.3 nM T59604 CU9OP3 90666012 IC50 = 1.6 nM T59604 C8O2ZM 90666013 IC50 = 1.8 nM T59604 C3ND7I 90666014 IC50 = 32 nM T59604 CSJE46 90666015 IC50 = 44 nM T59604 CN31ZU 90666016 IC50 = 4000 nM T59604 C6W4GH 90666017 EC50 = 1.3 nM T59604 C0D5FT 90666018 IC50 = 6.1 nM T59604 CMX8H0 90666019 IC50 = 370 nM T59604 CK8V1H 90666020 IC50 = 23 nM T59604 CTY8Q0 90666021 IC50 = 7.6 nM T59604 CF03DJ 90666022 IC50 = 120 nM T59604 C2O3UE 90666023 IC50 = 15 nM T59604 C4AP0G 90666024 IC50 = 5.1 nM T59604 CV3J8C 90666025 IC50 = 5 nM T59604 CD48KA 90666026 IC50 = 40 nM T59604 C7EIY6 90666027 IC50 = 1.7 nM T59604 C89PMV 90666028 IC50 = 120 nM T59604 CM2H6G 90666029 IC50 = 2.7 nM T59604 C9G5KP 90666030 IC50 = 5.7 nM T59604 C6NIZ9 90666031 IC50 = 1.6 nM T59604 CPVX39 90666032 IC50 = 12 nM T59604 C0U5BY 90666033 IC50 = 200 nM T59604 C45OBZ 90666034 IC50 = 60 nM T59604 C5WQN4 90666035 IC50 = 980 nM T59604 C85AMH 90666036 IC50 = 500 nM T59604 CKF14A 90666037 IC50 = 190 nM T59604 CM7ED5 90666038 IC50 = 52 nM T59604 CU2T3C 90666039 IC50 = 0.91 nM T59604 C59YXE 90666040 IC50 = 4.8 nM T59604 C6QZL4 90666041 IC50 = 11 nM T59604 CY35OV 90666042 IC50 = 27 nM T59604 C0V5EC 91826086 IC50 > 30000 nM T59604 CXV5R4 118709470 IC50 = 210 nM T59604 CE08TK 118709471 IC50 = 76 nM T59604 CK21QD 118709472 IC50 = 4700 nM T59604 C9ECO8 118709473 IC50 > 10000 nM T59604 C4P0SO 118709502 IC50 = 0.24 nM T59604 CI6FA2 118709503 IC50 = 0.57 nM T59604 CYK5M2 118709504 IC50 = 33 nM T59604 C70QKY 118709505 IC50 = 0.92 nM T59604 CCDV59 118709506 IC50 = 0.4 nM T59604 CT87MK 118709507 IC50 = 7.2 nM T59604 C80ORL 118718706 EC50 = 440 nM T59604 CFP2D9 118722878 IC50 = 6.31 nM T59604 CY9MF7 118725954 Ki = 49 nM T59604 C1W9RO 118725955 Ki > 50 nM T59604 C0T8AU 118725956 Ki = 6.4 nM T59604 C76QKE 118725957 Ki > 50 nM T59604 CPY60A 118725958 Ki = 166 nM T59604 CN21JF 118725959 Ki > 50 nM T59604 C4C2OQ 118725960 Ki = 13 nM T59604 C9LG8K 118725961 Ki = 4 nM T59604 C6KD7W 118725962 Ki = 263 nM T59604 CKQT19 118725963 Ki = 127 nM T59604 CAQ80I 118725964 Ki = 139 nM T59604 C2QS3P 118725965 Ki = 20 nM T59604 CSFY18 118725966 Ki = 28 nM T59604 CR2NZ9 122178176 EC50 = 6 nM T59604 C1Q0GC 122178177 EC50 = 189.2 nM T59604 CT5QV3 122178178 EC50 = 63.1 nM T59604 CK3W1J 122178179 EC50 = 29 nM T59604 CJ3YC7 122178180 EC50 = 60.2 nM T59604 C0DKP8 122178182 EC50 > 1000 nM T59604 C92LNJ 122178184 EC50 = 316.23 nM T59604 CKJ1U0 122178185 EC50 = 251.19 nM T59604 C3LKE9 122178186 EC50 = 99.9 nM T59604 CE0WR2 122178187 IC50 = 77.62 nM T59604 C4XDU8 122178188 EC50 = 39.81 nM T59604 C5Q7WR 122178189 IC50 = 70.79 nM T59604 CZV5P9 122178599 IC50 > 1000 nM T59604 CJ8CE4 122178600 IC50 = 122 nM T59604 C7YJ1F 122178601 IC50 = 88 nM T59604 CW3M9R 122178602 IC50 = 193 nM T59604 CU2I3P 122178603 IC50 = 130 nM T59604 CU48DB 122178604 IC50 = 380 nM T59604 CKWJ12 122178605 IC50 = 8.8 nM T59604 C6FN0V 122178606 IC50 = 2.1 nM T59604 C1HG6X 122178607 IC50 = 4.6 nM T59604 CTF3L2 122178608 IC50 = 3.4 nM T59604 CL31JE 122178609 IC50 = 2 nM T59604 CTIU14 122178610 IC50 = 6 nM T59604 C4A8XV 122178611 IC50 = 108 nM T59604 C1UB6L 122178612 IC50 = 79 nM T59604 C1GY8B 122178613 IC50 = 65 nM T59604 CLB32A 122178614 IC50 = 230 nM T59604 CIO35B 122178615 IC50 = 82 nM T59604 CJS9X1 122178616 IC50 = 100 nM T59604 CCH92O 122180014 IC50 = 84 nM T59604 CZ1C2A 122180015 IC50 = 150 nM T59604 C84EGT 122180016 IC50 = 260 nM T59604 CH4CF5 122180017 IC50 = 11 nM T59604 C9C6OK 122180018 IC50 = 36 nM T59604 CJ7OV3 122180019 IC50 = 180 nM T59604 C2E3MQ 122180020 IC50 = 24 nM T59604 CFG0I3 122180021 IC50 = 6.9 nM T59604 CA9P7Z 122180022 IC50 = 47 nM T59604 C0GD4B 122180023 IC50 = 7.2 nM T59604 CC7TK9 122180024 IC50 = 5.4 nM T59604 CRN0L6 122180025 IC50 = 42 nM T59604 C3HU8Z 122180026 IC50 = 0.96 nM T59604 CNZ3M0 122180027 IC50 = 0.23 nM T59604 CK49AE 122182043 IC50 = 0.39 nM T59604 CT0R6V 122182046 IC50 = 0.42 nM T59604 C7RLI5 122182047 IC50 = 0.3 nM T59604 CY8DA3 122182189 IC50 = 3 nM T59604 CBHG71 122182190 IC50 = 0.44 nM T59604 C87ASV 127045651 Ki > 1000 nM T59604 CAL12J 127045834 Ki > 1000 nM T59604 C2A3GB 127045858 IC50 = 3 nM T59604 CHPL37 127045859 Ki = 3 nM T59604 COK5L4 127046472 EC50 = 70 nM T59604 CO4A9F 127046473 Ki = 8 nM T59604 C36DRS 127046806 Ki = 154 nM T59604 C1MOG4 127046807 Ki = 62 nM T59604 CKQ0Y6 127046808 Ki > 1000 nM T59604 CHSJ34 127046956 IC50 = 2 nM T59604 C80BUK 127046957 IC50 = 4 nM T59604 CXT70M 127047362 IC50 = 130 nM T59604 CD42FM 127047363 Ki > 1000 nM T59604 C06JWX 127047409 EC50 = 170 nM T59604 CAO45B 127047523 Ki = 3 nM T59604 CZA7Y9 127047525 EC50 = 0.8 nM T59604 C27NXH 127047654 Ki = 62 nM T59604 C51JYG 127047655 IC50 = 7 nM T59604 C1C3JS 127048038 IC50 = 115 nM T59604 C26YTW 127048059 Ki = 2.5 nM T59604 C3JDM0 127048060 Ki = 17 nM T59604 C2TGW6 127048061 EC50 = 82 nM T59604 CZ2RL1 145948708 Ki = 50 nM T59604 C2OCP4 145948725 Ki = 2 nM T59604 C27NUT 145949381 EC50 = 25 nM T59604 C54ACE 145949595 EC50 = 19.95 nM T59604 CAB18Y 145949755 EC50 = 12.59 nM T59604 C6P9QW 145949880 IC50 = 501.19 nM T59604 C91DXZ 145950201 IC50 = 63.1 nM T59604 C8N5JL 145950261 EC50 = 125.89 nM T59604 C76GPL 145950336 EC50 = 0.1 nM T59604 CMP8T0 145950877 EC50 = 23 nM T59604 C6LXA0 145950963 EC50 = 158.49 nM T59604 CU81XO 145950987 EC50 = 50.12 nM T59604 C3YMF2 145951150 EC50 = 3 nM T59604 CAF83G 145952396 EC50 = 158.49 nM T59604 C0JZA8 145952404 EC50 = 251.19 nM T59604 C30MRB 145952740 EC50 = 15 nM T59604 C8QJW2 145953016 EC50 = 19 nM T59604 CHG09C 145953855 EC50 = 31.62 nM T59604 C25NVO 145954311 IC50 = 1260 nM T59604 CAW62C 145955250 EC50 = 125.89 nM T59604 C90KIG 145955718 EC50 = 251.19 nM T59604 CZ7IP5 145956026 EC50 = 5 nM T59604 C1J0BV 145956061 EC50 = 1.259 nM T59604 C9K4AQ 145956415 EC50 = 250 nM T59604 CR9DQ8 145956659 EC50 = 47 nM T59604 CFG2A0 145956753 EC50 = 236 nM T59604 CQVJ40 145957075 EC50 = 2.512 nM T59604 CU80KI 145957404 EC50 = 125.89 nM T59604 CASL75 145957443 IC50 = 184 nM T59604 CFZJ34 145957574 EC50 = 1.585 nM T59604 CG40FJ 145958317 EC50 = 25.12 nM T59604 CF0V3H 145958487 EC50 = 7 nM T59604 CWT43A 145958774 EC50 = 226 nM T59604 C4DMP9 145959007 EC50 = 39.81 nM T59604 CY75UJ 145959787 EC50 = 36 nM T59604 C03WXR 145961213 EC50 = 19.95 nM T59604 CF7GE0 145962494 EC50 = 10 nM T59604 CEY3A6 145974293 EC50 = 19.95 nM T59604 CN70VQ 145975725 EC50 > 7700 nM T59604 CWO02C 145979268 EC50 = 439 nM T59604 C3XBR0 145979819 EC50 = 484 nM T59604 C3QNO0 145980333 EC50 = 298 nM T59604 CV85ZH 145980382 EC50 = 29.4 nM T59604 C35FBK 145981196 EC50 = 483 nM T59604 C06LYT 145981343 EC50 = 2164 nM T59604 CD5NG2 145981687 EC50 = 40.7 nM T59604 CNIJ28 145981794 EC50 = 67 nM T59604 C9XC3S 145982096 IC50 > 30000 nM T59604 CM2HZ8 145982683 EC50 > 30000 nM T59604 C06VYC 145984632 EC50 = 363 nM T59604 CB0LX5 145986080 EC50 = 73 nM T59604 C8M9ZU 145986461 EC50 = 1276 nM T59604 CIL85G 145986870 EC50 = 85.7 nM T59604 CA6OW1 145987684 IC50 = 192 nM T59604 CYKQ65 145988286 EC50 = 70 nM T59604 CB4IN0 145988557 EC50 = 117 nM T59604 CXU4N1 145988582 IC50 = 2005 nM T59604 CJ5K7A 145988647 EC50 = 634 nM T59604 CRM2K5 145988894 EC50 = 51 nM T59604 CQ2N4K 145989762 EC50 > 30000 nM T59604 CG78YI 145989916 IC50 = 1300 nM T59604 CJ38OD 145990051 IC50 = 2367 nM T59604 CU3H4A 145990956 IC50 = 919 nM T59604 C58ETM 145991389 IC50 = 2330 nM T59604 C3PVM4 145991797 IC50 = 4010 nM T59604 CPX20Q 145991822 IC50 = 1130 nM T59604 C1DZK8 145991945 EC50 = 937 nM T59604 C7K8NJ 145992125 EC50 = 121 nM T59604 CD2V3K 145992142 EC50 = 189 nM T59604 CT57AZ 145992253 EC50 = 96 nM T59604 C6GEP2 145992835 EC50 = 84.8 nM T59604 CI4VH0 145992854 IC50 = 148 nM T59604 C3I8LB 145993313 EC50 = 970 nM T59604 CB2T3U 145993528 EC50 = 10.6 nM T59604 C15OAH 145993628 IC50 = 106 nM T59604 C02SLN 145993758 IC50 = 1510 nM T59604 C7ZU8A 145994050 EC50 = 194 nM T59604 CEP45Z 145994299 IC50 = 2700 nM T59604 C1PY8C 155526063 Ki = 3.4 nM T59604 C9JM2W 155529391 Ki = 2.7 nM T59604 CLQ4R5 155537651 Ki = 3.05 nM T59604 CAV10C 155540883 Ki = 1.26 nM T59604 C15KZH 155551597 Ki = 6.45 nM T59604 C2W8HU 155557019 EC50 = 2.5 nM T59604 CG7X4P 155561671 Ki = 55 nM T59604 CXC5Q2 46905972 EC50 = 3 nM T59604 D01LKO 44576255 IC50 = 540 nM T59604 D02NZI 9890863 IC50 = 4 nM T59604 D07JZB 44576248 IC50 = 12 nM T59604 D07QLZ 44576252 IC50 = 14 nM T59604 D08GTH 10190715 IC50 = 530 nM T59604 D09QPV 44576253 IC50 = 120 nM T59604 D0C3OY 25091011 Ki = 76.7 nM T59604 D0G8TL 44576249 IC50 = 58 nM T59604 D0J2YB 23631116 Ki = 4 nM T59604 D0L3AP 44576251 IC50 = 60 nM T59604 D0L3EP 25124566 IC50 = 3.981 nM T59604 D0PQ7A 44576250 IC50 = 210 nM T59604 D0U2QP 46882764 IC50 = 4300 nM T59604 D0XR6A 44576247 IC50 = 2.6 nM T59604 D0ZG7W 11441554 IC50 = 7 nM T94255 C8CUS5 1295523 IC50 = 400 nM T94255 CW59YI 2264067 IC50 = 1500 nM T94255 C4WI8K 2950887 IC50 = 1600 nM T94255 CEK6B1 139300630 IC50 > 10000 nM T94255 C4S7LQ 155514237 IC50 = 1300 nM T94255 C7X1EI 155519256 IC50 = 2800 nM T94255 CRO0K3 155530772 IC50 = 5900 nM T94255 C3C9GI 155535515 IC50 = 4700 nM T94255 CG23CH 155556141 IC50 = 4900 nM T94255 CY1JZ0 155564517 IC50 = 3600 nM T94255 D0G2MU 10229 IC50 = 29000 nM T67272 D0RA5Q 72172 IC50 = 0.81 ug.mL-1 T67272 D0U2JP 4369359 IC50 > 100000 nM T67272 D07SDQ 969516 IC50 = 15500 nM T67272 D0F2JS 15547703 IC50 = 680 nM T67272 D0T2IQ 443600 IC50 = 0.32 ug.mL-1 T67272 CKN1L3 20479 Ki = 10000 nM T67272 C0V9WL 73324 IC50 > 100 ug.mL-1 T67272 C8X2GZ 76808 IC50 = 1000000 nM T67272 CG48YC 97710 Ki = 27500 nM T67272 CP1JX4 124031 IC50 = 15 ug.mL-1 T67272 CKWA31 125415 Ki = 17000 nM T67272 C01SOJ 130013 Ki = 19 nM T67272 C2QHX5 182612 Ki = 53000 nM T67272 C6JM7L 182750 IC50 = 30 ug.mL-1 T67272 CV0J8H 182751 IC50 = 41.7 ug.mL-1 T67272 CGT6C5 276114 IC50 = 93.7 ug.mL-1 T67272 C7FP6H 277936 IC50 = 800000 nM T67272 CDBF98 281242 Ki = 10600 nM T67272 CNM0P3 391527 IC50 = 101400 nM T67272 CW10CK 439518 Ki = 200 nM T67272 CESM72 439530 IC50 = 41000 nM T67272 C5RO7V 469541 IC50 = 20 nM T67272 C0TYO2 477693 IC50 = 10.3 ug.mL-1 T67272 C7G3CT 477696 IC50 > 100 ug.mL-1 T67272 C4TRL6 721814 IC50 > 100 ug.mL-1 T67272 CO3KZ2 741570 IC50 = 84.7 ug.mL-1 T67272 CE28KQ 850934 IC50 = 6.7 ug.mL-1 T67272 C0L7TD 1235479 IC50 = 5.4 ug.mL-1 T67272 C6L1VE 1551321 Ki = 167 nM T67272 C2HQJ7 2302144 IC50 = 29.5 ug.mL-1 T67272 C3MR8Q 2817201 Ki = 2010 nM T67272 C59OKR 4330464 IC50 = 12400 nM T67272 CY36MH 4369380 Ki > 10000 nM T67272 CK8VJ3 5311145 Ki = 430000 nM T67272 CAQP85 5713154 Ki = 5950 nM T67272 C7AZE5 6930803 IC50 = 38400 nM T67272 CYQ8J7 9849506 IC50 = 28 nM T67272 C2DMP6 9861924 IC50 = 3.5 ug.mL-1 T67272 CFMG63 9886974 IC50 = 11.4 ug.mL-1 T67272 C30OXI 9990739 Ki = 3850 nM T67272 C5Q6BJ 9995375 IC50 > 100 ug.mL-1 T67272 CYH3C6 10061400 IC50 = 17.8 ug.mL-1 T67272 CV7SK8 10064801 IC50 = 309200 nM T67272 CWU9N2 10198228 IC50 > 100 ug.mL-1 T67272 C27AJQ 10245523 IC50 = 1000000 nM T67272 C0JD8Z 10333136 IC50 = 29 ug.mL-1 T67272 CTZQ69 10347030 IC50 = 1345 nM T67272 CK8T4C 10381531 IC50 = 4.3 ug.mL-1 T67272 C79UAO 10381586 IC50 > 100 ug.mL-1 T67272 C6GWB8 10401570 IC50 = 0.9 ug.mL-1 T67272 CL3H9I 10491923 IC50 = 16 ug.mL-1 T67272 CJ2RK6 10492044 IC50 = 70.7 ug.mL-1 T67272 C3YS4K 10659346 IC50 = 49.5 ug.mL-1 T67272 CN5KG9 10661540 IC50 = 9.6 ug.mL-1 T67272 C1LSP2 10779050 IC50 > 100 ug.mL-1 T67272 CD2GP9 10784566 IC50 > 100 ug.mL-1 T67272 C04XQH 10850290 IC50 = 54.3 ug.mL-1 T67272 C3ODA7 10945796 Ki = 1015 nM T67272 CN5H0B 10970861 Ki = 7.2 nM T67272 C5OPG0 11127644 Ki = 0.79 nM T67272 C10KPB 11142955 Ki = 2 nM T67272 CIOY84 11723708 IC50 = 15 ug.mL-1 T67272 CI2OP1 11942810 IC50 = 122500 nM T67272 CO0W1G 12749378 IC50 = 500000 nM T67272 C7RI2M 13168364 IC50 = 20 nM T67272 C29UOD 13226135 IC50 = 310000 nM T67272 CC9DK6 13384604 IC50 = 30400 nM T67272 CCX02R 13491256 IC50 = 25 nM T67272 C9F5CM 13491267 IC50 = 40 nM T67272 CF19DX 13509139 Ki = 341 nM T67272 CYV1F7 13784835 IC50 > 100 ug.mL-1 T67272 CP8L5J 14104451 IC50 = 38600 nM T67272 C94FPE 14434173 IC50 = 44.1 ug.mL-1 T67272 CT3L5Q 14542146 Ki = 660000 nM T67272 CP4OT8 14542149 Ki = 79000 nM T67272 CC17MK 15078261 Ki = 20 nM T67272 CW9ER1 15159715 IC50 = 30 nM T67272 CWNE58 15159721 IC50 = 21 nM T67272 CO1F2B 15342195 IC50 = 1000000 nM T67272 CE1P6J 15719279 Ki = 2500 nM T67272 CD28WR 15719282 Ki = 10500 nM T67272 CYR87Z 15719283 Ki = 18000 nM T67272 C4Y1HP 15849848 Ki = 7420 nM T67272 CB6WK0 16121107 Ki = 80000 nM T67272 CZQ8O9 16121199 Ki = 100000 nM T67272 CT01PQ 16739331 IC50 > 100000 nM T67272 C7YJZ5 17748252 IC50 = 3100 nM T67272 C9J8IN 18445902 IC50 = 53800 nM T67272 CYR08N 19366756 Ki = 8 nM T67272 C7GDU9 20038035 IC50 > 100 ug.mL-1 T67272 CF4VL0 21120524 Ki = 120 nM T67272 C8JSI4 23628284 IC50 > 100000 nM T67272 CFP01R 24828743 Ki = 100 nM T67272 C9LUM1 24828881 Ki = 27.54 nM T67272 CY9W8O 24860300 IC50 > 100000 nM T67272 C1CMY7 24884567 IC50 = 1800 nM T67272 C0VL7B 24890303 Ki = 52.48 nM T67272 C4R6BZ 24901452 Ki = 500 nM T67272 CTJU08 24975348 Ki = 1000 nM T67272 CIO26D 25022463 IC50 = 48500 nM T67272 CYZ2J7 25141282 IC50 = 21700 nM T67272 CP0YF8 25146956 IC50 = 81800 nM T67272 C12AVL 25146957 IC50 = 71300 nM T67272 C10MBE 25146958 IC50 = 24100 nM T67272 CIUY75 25146959 IC50 = 68400 nM T67272 C5MG9N 25146960 IC50 = 149300 nM T67272 C83IOD 25147056 IC50 = 74800 nM T67272 C1IA0W 25147057 IC50 = 135300 nM T67272 CB3W1I 25147058 IC50 = 161800 nM T67272 CC35MZ 25147059 IC50 = 196400 nM T67272 CO5H9V 25147060 IC50 = 232700 nM T67272 CM20ZC 25147061 IC50 = 29800 nM T67272 C2KZ0T 25147062 IC50 = 62200 nM T67272 C5RMI2 25147153 IC50 = 98400 nM T67272 C43YCQ 25147154 IC50 = 51400 nM T67272 CPQW89 25147155 IC50 = 121500 nM T67272 CQ3I6B 25147156 IC50 = 46600 nM T67272 C2LHR1 25147157 IC50 = 70600 nM T67272 CA34UT 25147158 IC50 = 121700 nM T67272 C3R0DB 25147159 IC50 = 72300 nM T67272 CV4ZE9 25147248 IC50 = 82600 nM T67272 C73HYI 25147249 IC50 = 137300 nM T67272 CV14TY 25147250 IC50 = 33500 nM T67272 CUW8X2 25147251 IC50 = 56100 nM T67272 C0Z7NX 25147252 IC50 = 96600 nM T67272 CU1KO6 25147352 IC50 = 78400 nM T67272 C7RS3Y 25195667 IC50 = 8000 nM T67272 C7IHC9 44207184 IC50 = 120000 nM T67272 C12CDQ 44254309 Ki = 512.86 nM T67272 C8EI1G 44254310 Ki = 181.97 nM T67272 CD3L0N 44254402 Ki = 8.511 nM T67272 CHT0Z1 44254404 Ki = 218.78 nM T67272 CW7LB9 44254495 Ki = 50.12 nM T67272 C5FDC2 44254496 Ki = 12.59 nM T67272 CR01EW 44256381 IC50 = 800 nM T67272 CUBV96 44276209 Ki = 4500 nM T67272 C34DUK 44276215 Ki = 2300 nM T67272 C9CUN1 44276216 Ki = 1900 nM T67272 C0Q1WI 44276218 IC50 = 75000 nM T67272 C32JVB 44276289 Ki = 45000 nM T67272 C79TMD 44276303 Ki = 210 nM T67272 C4JB1Z 44276401 Ki = 25000 nM T67272 CQX6J3 44276410 Ki = 35 nM T67272 CV5MC9 44276625 Ki = 7300 nM T67272 CHP16B 44276842 Ki = 2700 nM T67272 CQP05Z 44283812 IC50 = 1000000 nM T67272 C52KDH 44283814 IC50 = 1000000 nM T67272 CZT7Y3 44283829 IC50 = 3400 nM T67272 CUOI41 44283840 IC50 = 5000 nM T67272 CJ72SM 44283849 IC50 = 1000000 nM T67272 C36NHS 44283851 IC50 = 1000000 nM T67272 CK6ZW2 44283857 IC50 = 3800 nM T67272 C3PQR5 44283863 IC50 = 1000000 nM T67272 C0UG6P 44283886 IC50 = 1000000 nM T67272 C1YQM9 44283908 IC50 = 85000 nM T67272 CZG67T 44283924 IC50 = 146000 nM T67272 CE4NA8 44283925 IC50 = 2900 nM T67272 CT0O3D 44284085 IC50 = 783000 nM T67272 C6SFV4 44284086 IC50 = 1000000 nM T67272 CN9A8Q 44284101 IC50 = 2400 nM T67272 C7K8JV 44323547 IC50 = 1628 nM T67272 CRAI45 44323558 IC50 = 28000 nM T67272 CW2GK4 44344567 Ki = 11 nM T67272 CS75VD 44360285 Ki = 24000 nM T67272 C4QON9 44368427 IC50 = 10.2 ug.mL-1 T67272 C8FB1S 44368725 IC50 = 38.2 ug.mL-1 T67272 CE83AK 44368726 IC50 > 100 ug.mL-1 T67272 CW9BG0 44368735 IC50 > 100 ug.mL-1 T67272 C37TIM 44368736 IC50 = 40.5 ug.mL-1 T67272 C1U4IX 44458314 IC50 = 20 nM T67272 CRTB46 44458322 IC50 = 20 nM T67272 C5XS9L 44481133 IC50 = 23700 nM T67272 C3PYH7 44481390 IC50 = 64300 nM T67272 C38HFR 44481392 IC50 = 28800 nM T67272 CRC8F9 44481394 IC50 = 30800 nM T67272 CPJI36 44481396 IC50 = 23300 nM T67272 C9SG6K 44481398 IC50 = 38100 nM T67272 C0G2AC 44481400 IC50 = 18900 nM T67272 CFI01J 44481402 IC50 = 42000 nM T67272 CZ4KP3 44481661 IC50 = 16900 nM T67272 C3B9EX 44481663 IC50 = 41000 nM T67272 CO5D8W 44481665 IC50 = 21500 nM T67272 CY3KS0 44481667 IC50 = 15800 nM T67272 CXRA28 44481669 IC50 = 22100 nM T67272 C0M5WT 44481671 IC50 = 16600 nM T67272 C1EGD7 44481673 IC50 = 11300 nM T67272 CC5NV2 44481931 IC50 = 15400 nM T67272 CY5QH7 44481933 IC50 = 16900 nM T67272 CDCT90 44481935 IC50 = 9400 nM T67272 CQUL08 44481937 IC50 = 10900 nM T67272 CVM9E2 44481939 IC50 = 12500 nM T67272 C01YEO 44481941 IC50 = 5300 nM T67272 CJD57G 44481943 IC50 = 9200 nM T67272 C7JK5B 44482208 IC50 = 32100 nM T67272 CH3B9V 44482210 IC50 = 20700 nM T67272 CMQA93 44482214 IC50 = 13200 nM T67272 CRZ9P0 44482218 IC50 = 9700 nM T67272 CZ4H7R 44560401 Ki = 5000 nM T67272 C70AIZ 44560402 Ki = 55000 nM T67272 C63VWA 44560403 Ki = 49000 nM T67272 CRX2G5 44560404 Ki = 17000 nM T67272 CA4IF6 44560405 Ki = 11000 nM T67272 C57LTE 44560406 Ki = 10000 nM T67272 C2F3TI 44560407 Ki = 16000 nM T67272 CC3GY2 44560408 Ki = 20000 nM T67272 C9YE7J 44560409 Ki = 21000 nM T67272 C1OEW5 44560410 Ki = 17000 nM T67272 CU4G1S 44560411 Ki = 13000 nM T67272 C2Y0OT 44560412 Ki > 100000 nM T67272 CG7BQ8 44560457 Ki = 33000 nM T67272 C1RK3C 44560557 Ki > 100000 nM T67272 C42VEQ 44560558 Ki = 69000 nM T67272 C0J6LB 44563970 IC50 = 73700 nM T67272 C3US0I 44569010 IC50 = 24800 nM T67272 C3TAN1 44569011 IC50 = 51200 nM T67272 CF0L2W 44569012 IC50 = 74600 nM T67272 CGI35S 44569013 IC50 = 41400 nM T67272 C8PO5Q 44569024 IC50 = 168600 nM T67272 C52JXP 44569036 IC50 = 43800 nM T67272 CU1NI6 44569037 IC50 = 36400 nM T67272 CS9CH4 44569038 IC50 = 61300 nM T67272 C63ZQK 44569039 IC50 = 47300 nM T67272 C2WE7H 44569040 IC50 = 39500 nM T67272 CO8FB4 44569058 IC50 = 134700 nM T67272 C3K4ED 44569059 IC50 = 53600 nM T67272 CPWR76 44569060 IC50 = 47500 nM T67272 CU39FK 44569061 IC50 = 68900 nM T67272 CR6H0X 44569062 IC50 = 28400 nM T67272 CTWR37 44569063 IC50 = 31600 nM T67272 C6M9SH 44569081 IC50 = 114300 nM T67272 C5RN7U 44569082 IC50 = 33500 nM T67272 CQ9OA7 44569083 IC50 = 26300 nM T67272 CCV74H 44576563 IC50 = 54900 nM T67272 C59TCG 44576564 IC50 = 75800 nM T67272 CMI9S4 44576565 IC50 = 92600 nM T67272 CD8ZI4 44576587 IC50 = 155800 nM T67272 CQ87CS 44576614 IC50 = 173700 nM T67272 CJY2W3 44576615 IC50 = 124300 nM T67272 CL92CH 44576616 IC50 = 150600 nM T67272 CIU84E 44576617 IC50 = 168100 nM T67272 C9ODS1 44576618 IC50 = 134800 nM T67272 C35DWL 44576631 IC50 = 61800 nM T67272 C6ZL1U 44576632 IC50 = 73200 nM T67272 CK09LV 44576633 IC50 = 57800 nM T67272 CFL76T 44576634 IC50 = 82700 nM T67272 CC58GQ 44576635 IC50 = 106700 nM T67272 CZNQ90 44593458 IC50 = 141900 nM T67272 CR3Q4N 44593532 IC50 = 41600 nM T67272 CTWL91 46193025 IC50 = 7300 nM T67272 CMLG10 46882676 Ki = 128.82 nM T67272 CTO1Q8 46882677 Ki = 54.95 nM T67272 C19YDM 46886333 Ki = 53000 nM T67272 C9HPU0 46886351 Ki = 27500 nM T67272 CHE51J 49795928 IC50 = 83000 nM T67272 CS1TY7 49795932 IC50 = 104000 nM T67272 CP9WB0 49840768 Ki = 3588 nM T67272 C51YRX 49840770 Ki = 11100 nM T67272 CJ3Z7V 49840772 Ki = 16800 nM T67272 CS3I8G 49840774 Ki = 7245 nM T67272 C3IT5V 49840844 Ki = 10800 nM T67272 CYBW37 49840846 Ki = 48900 nM T67272 CFEC23 49840848 Ki = 9217 nM T67272 C64XMG 49840850 Ki = 5436 nM T67272 CNU1Q7 49840921 Ki = 11900 nM T67272 C7S9QA 50913428 IC50 = 3000 nM T67272 CO4XE9 50913573 IC50 = 5100 nM T67272 CQ90FE 52941108 Ki = 57000 nM T67272 CU4HK1 52943524 Ki = 5974 nM T67272 C9HRG4 52946764 Ki = 50000 nM T67272 C89EGH 52947188 Ki = 841 nM T67272 CU58OG 53257413 Ki = 4955 nM T67272 C6XY5R 53259047 Ki = 1074 nM T67272 C7AXD8 53259048 Ki = 5413 nM T67272 CX51OK 53259216 Ki = 1571 nM T67272 CBS92H 53259217 Ki = 12000 nM T67272 C8RZW7 53259219 Ki > 100000 nM T67272 C4KZ7R 53259403 Ki > 100000 nM T67272 CA0Q2E 53259404 Ki > 100000 nM T67272 C6FU2G 53259405 Ki > 100000 nM T67272 CLSC37 53261358 Ki = 12000 nM T67272 CXMC12 53261359 Ki = 3283 nM T67272 C3Q4ZR 53261360 Ki = 8345 nM T67272 C48JHC 53320960 IC50 > 1000000 nM T67272 C9QWK0 53322291 IC50 = 300000 nM T67272 CO0X3H 53324937 Ki = 20000 nM T67272 CGP68U 53324939 Ki = 60000 nM T67272 CN12AO 53353383 IC50 > 100000 nM T67272 C51GUC 53354365 IC50 > 100000 nM T67272 CRJ5P9 53354369 IC50 > 100000 nM T67272 C4G2HT 53354470 IC50 > 100000 nM T67272 CFS7N9 53494936 Ki = 11 nM T67272 CN53IO 53792079 Ki = 691 nM T67272 CGF98A 54585162 Ki = 1299 nM T67272 CLP2C1 54753981 IC50 = 32690 nM T67272 CGTV56 56658262 IC50 = 248350 nM T67272 CV46HL 56665195 IC50 = 289950 nM T67272 C3L5SO 56665196 IC50 = 615560 nM T67272 CH4M6V 56665197 IC50 = 66340 nM T67272 CSU81T 56672275 IC50 = 39430 nM T67272 CF75JN 56953635 IC50 = 30000 nM T67272 CQ64IE 56953636 IC50 > 100000 nM T67272 C9RJF3 56953637 IC50 = 500 nM T67272 CM7VP3 56953638 IC50 > 70000 nM T67272 C1BWY5 56953762 IC50 = 54000 nM T67272 C4VJI0 56953763 IC50 = 45000 nM T67272 C7JYZ1 56953764 IC50 = 30000 nM T67272 CH67KO 56953765 IC50 > 100000 nM T67272 CSW96U 56955172 IC50 = 44000 nM T67272 CFG17Q 56955173 IC50 = 65000 nM T67272 C76MEC 56955271 IC50 > 100000 nM T67272 CWGA37 56955272 IC50 = 13500 nM T67272 C28VDY 56955273 IC50 = 500 nM T67272 C1QSV9 56955274 IC50 = 48000 nM T67272 C1T2QI 60144811 IC50 = 420 nM T67272 CI4AV6 70073083 IC50 = 9600 nM T67272 C64XBZ 70681347 IC50 = 37000 nM T67272 C4N3VW 70681348 IC50 > 70000 nM T67272 C5EHM1 70681503 IC50 > 100000 nM T67272 CFP12D 70683616 IC50 = 75000 nM T67272 CYVJ36 70683617 IC50 = 122000 nM T67272 CYD34L 70685541 IC50 = 65000 nM T67272 C1DZ3J 70685542 IC50 = 47000 nM T67272 C4BN0J 70689859 IC50 = 10000 nM T67272 CB4ZL3 70690154 IC50 = 39000 nM T67272 CHM4W5 70692015 IC50 = 64000 nM T67272 CJ3OY4 70692312 IC50 = 22000 nM T67272 C0HFX4 70694371 IC50 = 16000 nM T67272 CFT06N 70696054 IC50 > 70000 nM T67272 C6MW3C 70696243 IC50 = 27000 nM T67272 C2IAG5 70696244 IC50 > 100000 nM T67272 CLE79H 70696450 IC50 = 110000 nM T67272 CA6IB0 71450469 IC50 = 910 nM T67272 CT5J7F 71452300 IC50 = 790 nM T67272 C23NVO 71452301 IC50 = 6900 nM T67272 CU3KE8 71453804 Ki = 1000 nM T67272 C5K8WS 71454094 IC50 = 940 nM T67272 CP2D3C 71454095 IC50 = 1100 nM T67272 C3VQW4 71455829 IC50 = 6400 nM T67272 CKR4D0 71459517 IC50 = 1500 nM T67272 C6UQW4 71461261 IC50 = 3000 nM T67272 C9QE5X 71462985 IC50 = 480 nM T67272 CL0P1Y 71584425 IC50 = 1310 nM T67272 C1BF6E 71584426 IC50 = 530 nM T67272 CMRA35 71584427 IC50 = 610 nM T67272 C6STG3 71584428 IC50 = 700 nM T67272 C42XYH 71584672 IC50 = 650 nM T67272 C2TYL8 71584673 IC50 = 730 nM T67272 CS3T9Q 71602397 IC50 = 3120 nM T67272 CIWZ87 71602398 IC50 = 15160 nM T67272 CJK3H7 71603240 IC50 = 9580 nM T67272 CMJF12 71603241 IC50 = 16190 nM T67272 CY7M2C 71603243 IC50 = 10940 nM T67272 C4M9AB 71603244 IC50 = 97490 nM T67272 C9ZJ2B 71603245 IC50 = 19660 nM T67272 C5OB3M 73348808 IC50 = 12100 nM T67272 C28UIX 73356287 IC50 = 793000 nM T67272 CEM9F5 73672383 IC50 = 65290 nM T67272 CRU02V 74766022 Ki = 0.23 nM T67272 C05HWU 86140993 Ki = 1660 nM T67272 CF35LZ 87495845 Ki = 41100 nM T67272 CUD73A 90645555 Ki > 10000 nM T67272 C0YOU8 90664312 IC50 = 9400 nM T67272 CDQF80 90664420 IC50 = 14100 nM T67272 CYND40 90672013 IC50 = 1100 nM T67272 CG9N2T 90672014 IC50 = 420 nM T67272 C34ALI 94005078 IC50 = 220 nM T67272 C8BNV9 95566324 Ki = 19 nM T67272 CX29SF 97550302 Ki = 19 nM T67272 CDA72U 101882336 Ki = 0.21 nM T67272 CVS60Z 118720629 Ki = 4.8 nM T67272 C4VWL9 118720630 Ki = 2.4 nM T67272 C71CKB 118720631 Ki = 146 nM T67272 CCQ74S 118720632 Ki = 24.2 nM T67272 C8JDP5 118720633 Ki = 1.7 nM T67272 CE9X4G 118720634 Ki = 2.1 nM T67272 CW87DK 118720635 Ki = 1.3 nM T67272 CKIF61 118720636 Ki = 27.8 nM T67272 CJ6MY3 118720637 Ki = 2.1 nM T67272 CP5V7M 118720638 Ki = 0.69 nM T67272 CQ6K5N 118720639 Ki = 1.1 nM T67272 CWL1M3 122195270 IC50 = 85000 nM T67272 CN6UZ5 122195271 IC50 = 20000 nM T67272 C6CV7K 122195272 IC50 > 70000 nM T67272 CHE75Z 122195273 IC50 > 70000 nM T67272 C6RY2A 122195274 IC50 = 22000 nM T67272 C14TSF 122195275 IC50 = 62000 nM T67272 CIE12T 122195276 IC50 = 32000 nM T67272 C4DXT1 122195277 IC50 = 52000 nM T67272 CNV2J7 122195278 IC50 > 100000 nM T67272 C8C0HD 124196349 Ki = 172 nM T67272 CLSB73 124196351 Ki = 497 nM T67272 C7IK1U 124196354 Ki = 71.2 nM T67272 CPU97K 124196355 Ki = 49.1 nM T67272 CUE28O 124196356 Ki = 40 nM T67272 C4FV5U 124196371 Ki = 348 nM T67272 C9Y8LQ 124196373 Ki = 29.1 nM T67272 CWVI53 124196382 Ki = 560 nM T67272 CG46VB 124196383 Ki = 188 nM T67272 C0Z5QW 124196384 Ki = 82.1 nM T67272 CGEJ47 124196385 Ki = 37.3 nM T67272 C8Z1BF 124196387 Ki = 300 nM T67272 C9MPY5 127025893 IC50 = 120 nM T67272 C3TF8V 127037842 IC50 = 280 nM T67272 CUO5V9 127039573 Ki = 118 nM T67272 CM0VT4 127048200 Ki = 37700 nM T67272 CTL4Z8 127048201 Ki = 499 nM T67272 CBQ4S3 127048202 Ki = 275 nM T67272 CC96VU 127048834 Ki = 782 nM T67272 CRCB36 127048872 Ki = 2510 nM T67272 CTY5D4 127049157 Ki = 6040 nM T67272 CF3HO2 127049196 Ki = 13500 nM T67272 C03XKF 127049491 Ki = 391 nM T67272 CFW6M1 127049492 Ki = 5740 nM T67272 CL6D0Z 127049497 Ki = 4450 nM T67272 C4I1RH 127049824 Ki = 397 nM T67272 C2A1MZ 127050130 Ki = 1220 nM T67272 CA4MP3 127050430 Ki = 1110 nM T67272 CJT5R9 127050433 Ki = 3220 nM T67272 C0N2LE 127050745 Ki = 2550 nM T67272 C9GBD2 127051304 Ki = 1490 nM T67272 CLK50R 127051701 Ki = 207 nM T67272 C2BUZ7 127051959 Ki = 357 nM T67272 CK81ME 127051999 Ki = 78 nM T67272 CAC25R 127052273 Ki = 297 nM T67272 C3FMN7 127052612 Ki = 2890 nM T67272 CHA9Q6 127052870 Ki = 65 nM T67272 CJM96B 127053163 Ki = 3290 nM T67272 CLJ9F6 145949706 IC50 = 3200 nM T67272 C25EDJ 145952430 IC50 = 1950 nM T67272 C32LGX 145952863 IC50 = 740 nM T67272 C0MC6U 145955648 IC50 = 870 nM T67272 CQNE67 145956257 IC50 = 270 nM T67272 CN84MC 145956662 IC50 = 5370 nM T67272 CN1CQ3 145957783 IC50 = 1680 nM T67272 CB03UD 145960195 IC50 = 5600 nM T67272 CM2D9J 145961321 IC50 = 6500 nM T67272 CK5P6I 145961499 IC50 = 4800 nM T67272 C4J0HA 145963210 IC50 = 5000 nM T67272 C27HIP 145963359 IC50 = 6900 nM T67272 CZU0S1 145963748 IC50 = 280 nM T67272 CL1DE4 145965106 IC50 = 10200 nM T67272 C38IXU 145966119 IC50 = 190 nM T67272 CP9ZD1 145971617 Ki = 80 nM T67272 C1VOU2 145976275 Ki = 1010 nM T67272 CM7YB8 145998092 Ki = 4.5 nM T67272 CSF69J 155511374 Ki = 131 nM T67272 C3WTA6 155513618 Ki > 1000000 nM T67272 CKZ21H 155513922 Ki = 205 nM T67272 CX2ZT9 155513964 Ki = 604 nM T67272 CF7LE9 155514400 Ki = 442 nM T67272 C8GB3J 155514541 Ki = 277 nM T67272 CUGK20 155515062 Ki = 102 nM T67272 C6LCH3 155515796 Ki = 430 nM T67272 CT2C5J 155517371 Ki = 704 nM T67272 CIGF73 155517640 Ki = 19.2 nM T67272 C4AE5F 155518479 Ki = 978 nM T67272 CA3TM6 155518679 Ki = 111 nM T67272 CG2RF3 155520398 Ki = 8.2 nM T67272 CM1ES6 155523825 Ki = 745 nM T67272 CNF48I 155525687 IC50 = 810 nM T67272 C6G0MI 155528995 Ki = 163 nM T67272 CZ2BF0 155529155 Ki = 185 nM T67272 CI2P4Z 155533156 Ki = 235 nM T67272 C7HJ5U 155534393 IC50 = 620 nM T67272 CZN50A 155535841 IC50 = 990 nM T67272 C8C1EI 155540506 IC50 = 3300 nM T67272 C56KWP 155543532 IC50 = 650 nM T67272 CY02VQ 155546277 Ki = 462 nM T67272 CX1CW7 155547815 Ki = 240 nM T67272 C5I9HJ 155548213 Ki = 158 nM T67272 CH61FB 155550504 Ki = 23.4 nM T67272 CA08LZ 155550520 Ki = 522 nM T67272 CWM3Q7 155550895 Ki = 182 nM T67272 C71FAU 155553065 Ki = 43.1 nM T67272 CK3Q4N 155556136 Ki = 137 nM T67272 CHY95K 155559649 Ki = 366 nM T67272 CRQ4V7 155559773 Ki = 170 nM T67272 CM43NT 155559807 Ki = 4420 nM T67272 C9S2FL 155562411 Ki = 919 nM T67272 C07NIE 155563089 Ki = 119 nM T67272 CMUF64 155565532 Ki = 175 nM T67272 C6J9LE 155567025 Ki = 631 nM T67272 C5UH8A 155567330 Ki = 138 nM T67272 CEO6S0 155568852 Ki = 156 nM T67272 C0VK3G 44344579 Ki = 4.8 nM T67272 C2PVI1 44344594 Ki = 2.9 nM T67272 CHEX85 445715 Ki = 2.62 nM T67272 D04DTE 53259050 Ki = 240 nM T67272 D04QJY 123982 Ki = 7000 nM T67272 D06AFP 11436221 IC50 = 3400 nM T67272 D0A7GO 44309732 Ki = 20000 nM T67272 D0H5BG 53494934 Ki = 0.06 nM T67272 D0I6RL 11723962 IC50 > 100000 nM T67272 D0L3PY 123814 Ki = 56.23 nM T59045 D0R3QY 5665 Ki = 850000 nM T59045 D00BRD 126 IC50 = 4.1 ug.mL-1 T59045 D09SWE 31244 IC50 > 1000000 nM T59045 D0B5YS 1183 IC50 = 17100 nM T59045 D0NH9P 135 IC50 > 1000000 nM T59045 D0X7BT 125 IC50 > 1000000 nM T59045 CY8P0F 227 IC50 > 5000000 nM T59045 C6X9CB 978 IC50 > 1000000 nM T59045 C0F1EW 6271 IC50 = 176000 nM T59045 CLE87P 7419 IC50 > 5000000 nM T59045 CV9N2M 7469 IC50 = 188000 nM T59045 CR0U3Y 115067 IC50 > 1000000 nM T59045 CSJ7V0 277942 IC50 > 5000000 nM T59045 C97XKM 506073 IC50 > 5000000 nM T59045 CR3OI1 571807 IC50 > 5000000 nM T59045 CA6EQ4 1514158 IC50 > 5000000 nM T59045 C4Q6ZR 3000722 Ki = 91000 nM T59045 C7EP1S 7016465 Ki = 13000000 nM T59045 CDY5C8 10011990 Ki = 100000 nM T59045 CHX1O3 10103265 Ki = 125000 nM T59045 CFH15U 10419269 Ki = 2300000 nM T59045 CL7H6I 10419448 Ki = 11000000 nM T59045 C3INT9 12896796 IC50 > 1000000 nM T59045 COG3R4 22247029 IC50 > 5000000 nM T59045 C8OP4K 10351955 Ki = 6300000 nM T59045 C6G5XN 135408704 IC50 > 1000000 nM T59045 C59TVG 44378094 Ki = 9000 nM T59045 D00YEV 5281605 IC50 = 12800000 nM T59045 D03VZF 18169 IC50 = 15500 nM T59045 D07ZBH 97472 IC50 = 15400 nM T59045 D0L7RB 16036927 IC50 = 5480 nM T67818 D01BYB 5957 EC50 = 150 nM T67818 D06ACW 6083 EC50 = 1500 nM T67818 D0S6AE 148197 EC50 > 20000 nM T67818 D0Z7FU 6133 EC50 > 2000 nM T67818 CPQ81V 171069 EC50 = 80 nM T67818 CVC6T8 440210 EC50 = 760 nM T67818 CR8K6U 1188014 IC50 = 140 nM T67818 C3LYX1 1188015 Ki >= 100000 nM T67818 CJX73P 1226686 Ki = 6000 nM T67818 C6P7VU 5311303 IC50 = 320 nM T67818 CIH51L 7283514 Ki = 400 nM T67818 CZW7U2 7283646 IC50 = 25000 nM T67818 C2I5JK 7312981 Ki = 400 nM T67818 C8RM7J 7313032 Ki = 500 nM T67818 CF8KI6 9847505 Ki = 2.5 nM T67818 CRE90Y 9955181 EC50 = 840 nM T67818 C3T8BS 10070925 IC50 = 148 nM T67818 C2F7DR 10098947 EC50 = 2630 nM T67818 CM96ZK 10168108 EC50 > 20000 nM T67818 CI9K1V 10191162 EC50 > 20000 nM T67818 CM4K6R 10303040 EC50 > 20000 nM T67818 CZE5Y1 10482694 EC50 = 80 nM T67818 C2BVH7 10601567 Ki = 17.6 nM T67818 C3L6KW 10994891 EC50 = 52 nM T67818 CJS9C0 11304851 IC50 > 25000 nM T67818 C36FVH 11409030 Ki = 91 nM T67818 C4KTZ9 11496216 Ki = 7.3 nM T67818 CO26HV 11510223 Ki = 31 nM T67818 CHB3C7 11510273 Ki = 16 nM T67818 C3AFT9 11517789 Ki = 26 nM T67818 C7ZR5X 11518174 Ki = 16 nM T67818 C2WS9Q 11531074 Ki = 28 nM T67818 CWZ3D4 11533956 Ki = 390 nM T67818 C12UVD 11541258 Ki = 260 nM T67818 C8PDH3 11549000 IC50 = 5.9 nM T67818 CT74ZJ 11560464 Ki = 7 nM T67818 CHR5C4 11562092 Ki = 4500 nM T67818 CQM17R 11562714 Ki = 300 nM T67818 C1X9UA 11575089 Ki = 172 nM T67818 C7NK4X 11575502 Ki = 36.5 nM T67818 CQIE41 11575842 Ki = 20.3 nM T67818 CMKY61 11583568 Ki = 6.6 nM T67818 CJG3K6 11604868 Ki = 7.6 nM T67818 C4G3BS 11606309 Ki = 13.3 nM T67818 CUD1J5 11611428 Ki = 8 nM T67818 CO23MC 11614523 IC50 < 1000 nM T67818 C8V0QO 11620229 Ki = 690 nM T67818 CYH54P 11626368 Ki = 29.5 nM T67818 CJVD59 11634388 IC50 = 2.2 nM T67818 CX7J8F 11636756 IC50 = 1819700.86 nM T67818 CB5OD0 11640537 Ki = 65 nM T67818 CC2R9X 11642453 Ki = 290 nM T67818 C4U5MH 11648059 Ki = 28 nM T67818 C43BEI 11656611 Ki = 4500 nM T67818 C7D4FT 11662179 Ki = 830 nM T67818 CQ6SG9 11675204 Ki = 7 nM T67818 CG3K2W 11692026 Ki = 11 nM T67818 CEU74V 11698231 Ki = 39 nM T67818 CPC34H 11699502 Ki = 13500 nM T67818 CI71BX 11699791 Ki = 18.6 nM T67818 CRPZ90 11704091 Ki = 11 nM T67818 C7QD0V 11706525 Ki = 20.7 nM T67818 CI2MT7 11706804 Ki = 200 nM T67818 C70OHZ 11711880 Ki = 8.7 nM T67818 C7OFE2 11711909 Ki = 94 nM T67818 CODM63 12000021 EC50 = 1200 nM T67818 C67WNM 13455593 EC50 = 426 nM T67818 CKB09S 16005793 IC50 = 75 nM T67818 C4E8CP 16005795 IC50 = 227 nM T67818 CR6W9O 16216480 EC50 > 20000 nM T67818 C6AQ2L 16738126 Ki = 66 nM T67818 CZ7SX0 23675739 IC50 = 3000 nM T67818 CXZ58T 24799317 EC50 = 4390 nM T67818 CKO7C2 24958669 Ki = 50 nM T67818 C7K0OA 24959029 Ki = 100 nM T67818 C0JSZ6 24959030 Ki = 120 nM T67818 CZ36UC 24959031 Ki = 130 nM T67818 CSI9Q5 24959032 Ki = 250 nM T67818 CSO73E 24959398 Ki = 250 nM T67818 C7O9KD 24959759 Ki = 140 nM T67818 CWC1K6 24959760 Ki = 290 nM T67818 CARU61 24959763 Ki = 30 nM T67818 C76JQO 24960128 Ki = 70 nM T67818 C86PJO 24960131 Ki = 20 nM T67818 C2XB7S 24960132 Ki = 60 nM T67818 C29KLZ 24960493 Ki = 60 nM T67818 CZ48MB 24960497 Ki = 30 nM T67818 CMZ9Y8 25099564 Ki = 150 nM T67818 C54AXC 25169254 Ki = 70 nM T67818 C8YV9Q 40995076 Ki = 100 nM T67818 CVC9D3 44306835 EC50 = 52 nM T67818 CTB6U8 44364208 Ki = 5.1 nM T67818 CB7T0D 44364283 Ki = 12.6 nM T67818 C0UQ9H 44364323 Ki = 35 nM T67818 C7CD3U 44425066 Ki = 540 nM T67818 C5W8JN 44425067 Ki = 650 nM T67818 CMG9D2 44425068 IC50 = 870 nM T67818 CW8BQ9 44425069 IC50 = 93.33 nM T67818 CB2C1L 44425070 Ki = 273 nM T67818 CGKL72 44425071 Ki = 706 nM T67818 C2D1MQ 44439743 EC50 > 20000 nM T67818 CW2U7Z 44439757 EC50 > 20000 nM T67818 C42YBU 44439758 EC50 > 20000 nM T67818 C0IBA3 44439765 EC50 > 20000 nM T67818 CI74KG 44448768 Ki = 5200 nM T67818 CT6N0P 44448802 Ki > 10000 nM T67818 C4U5HR 44448803 Ki = 1800 nM T67818 CP70GV 44448830 Ki > 10000 nM T67818 CO31DG 44448868 Ki > 10000 nM T67818 C4UBN8 44448870 Ki > 10000 nM T67818 CP0BD2 44448871 Ki > 10000 nM T67818 CRM3C1 44448909 Ki > 10000 nM T67818 C5Q1YK 44448911 Ki = 1200 nM T67818 CQF4Z2 44448944 Ki > 10000 nM T67818 C4HF1P 44448945 Ki > 10000 nM T67818 CVA01W 44448974 Ki = 760 nM T67818 CI96JR 44449026 Ki = 120 nM T67818 CERK23 44449075 Ki = 2700 nM T67818 CAD32B 44449077 Ki = 130 nM T67818 CQ2P9F 44449103 Ki = 200 nM T67818 C4ZEH5 44449104 Ki = 180 nM T67818 C7OX1B 44449105 Ki = 560 nM T67818 C40LXK 44449129 Ki > 10000 nM T67818 C8F3AN 44449130 Ki = 700 nM T67818 C2S8MC 44449132 Ki = 7200 nM T67818 C6IV9P 44449164 Ki > 10000 nM T67818 CTF47A 44449165 Ki = 270 nM T67818 CTKW57 44449166 Ki > 10000 nM T67818 C5YI3T 44449191 Ki > 10000 nM T67818 C9YID2 44449195 Ki = 960 nM T67818 CMHK57 44562602 IC50 > 25000 nM T67818 C4VGQ9 44562603 IC50 > 25000 nM T67818 CLJX37 44562653 Ki = 300 nM T67818 CS3DV0 44562758 Ki = 300 nM T67818 COV1S4 44562759 Ki = 500 nM T67818 CRU78M 44562760 IC50 = 6000 nM T67818 CQSC98 44562761 Ki = 100 nM T67818 C3FS9P 44562795 Ki = 400 nM T67818 C2M8EJ 44562796 Ki = 200 nM T67818 C1YGU0 44562797 Ki = 800 nM T67818 C7QN9K 44562836 IC50 > 25000 nM T67818 CUC87A 44562837 IC50 = 10000 nM T67818 CRD29T 44562838 IC50 > 25000 nM T67818 C4M6UO 44562839 IC50 > 25000 nM T67818 C8IKO9 44563234 IC50 > 25000 nM T67818 CV69BH 44563235 Ki = 100 nM T67818 CZD86A 46228890 EC50 = 420 nM T67818 C4U6LZ 46228892 EC50 = 460 nM T67818 CWR97Z 46228944 EC50 = 11 nM T67818 CI83JW 46229259 EC50 = 1.89 nM T67818 CQNZ48 46241018 IC50 = 4900 nM T67818 CVP5D0 46241232 IC50 = 29000 nM T67818 CPZ83K 46911434 IC50 = 1600 nM T67818 CF4DN0 46911436 IC50 = 300 nM T67818 CL2U0Q 46911481 Ki = 600 nM T67818 CU0XK3 49797754 Ki = 640 nM T67818 C0IC7Y 49797755 Ki = 760 nM T67818 C6K2YC 49797777 IC50 = 15800 nM T67818 C1D8NS 49797778 IC50 = 5000 nM T67818 CTQ4H0 49798096 IC50 > 25000 nM T67818 C0ICW7 49798097 Ki = 2500 nM T67818 CNZ54V 49798145 Ki = 400 nM T67818 C36ALC 49798146 IC50 > 25000 nM T67818 CPV84E 49798147 IC50 > 25000 nM T67818 C30CIT 49856886 EC50 = 300 nM T67818 C2O6TI 49856888 EC50 >= 30000 nM T67818 CJGE25 49857082 EC50 = 30000 nM T67818 CKI5H9 51032193 IC50 = 10200 nM T67818 CR98BF 53350233 IC50 = 2.5 nM T67818 CP87YH 53350234 Ki = 12 nM T67818 CJ2RM6 56673378 EC50 = 9000 nM T67818 C1I4YV 59128840 Ki = 70 nM T67818 CYQ3S9 59128841 Ki = 21 nM T67818 CKP5V0 59128886 Ki = 207 nM T67818 C1U8JL 59128890 Ki = 11 nM T67818 CI5P7T 59128900 Ki = 12 nM T67818 CRS58Y 59128945 Ki = 435 nM T67818 CL2VD6 59128964 Ki = 45 nM T67818 C3SYF6 59128997 Ki = 31 nM T67818 CY3JA1 59129000 Ki = 1500 nM T67818 CSHK27 59129016 Ki = 410 nM T67818 CPC0R9 59129017 Ki = 2900 nM T67818 CI8U6F 59129057 Ki = 7 nM T67818 CI3LA5 59129071 Ki = 25 nM T67818 CK36PG 59129092 Ki = 59 nM T67818 C94KLF 59129106 Ki > 36000 nM T67818 CX5J7S 59129109 Ki = 186 nM T67818 CUIW36 591291