TTD Target ID TTD Drug/Compound ID Pubchem CID Activity T34562 CANH78 17280 IC50 = 3270000 nM T34562 C27IRS 197934 IC50 = 1280000 nM T34562 CBJ36Y 639433 IC50 = 564130 nM T34562 CF2BD8 907361 IC50 = 21370 nM T34562 C5NQG3 940069 IC50 = 31410 nM T34562 CJGB43 941230 IC50 = 40000 nM T34562 CEX1K9 10243765 IC50 = 19050 nM T34562 C5I4SX 10402002 IC50 = 28980 nM T34562 C2JY8F 15388819 IC50 = 3000 nM T34562 C8G9AL 16756850 IC50 > 10000 nM T34562 C0SDW6 127025482 Ki = 2390 nM T34562 CK7L8U 127027355 IC50 = 23700 nM T34562 CH6ON2 127027684 IC50 = 625710 nM T34562 C7ST9X 127028306 IC50 = 317310 nM T34562 CN86IR 127028327 IC50 = 3333300 nM T34562 CHU16M 127028328 IC50 = 2064200 nM T34562 CV03TZ 127028660 IC50 = 237500 nM T34562 CBE6M2 127028661 IC50 = 627000 nM T34562 C5P3GA 127029548 IC50 = 8760 nM T34562 C1ZP4G 130431469 IC50 > 10000 nM T34562 CMA35H 130431481 IC50 > 10000 nM T34562 D0S9LT 12793 IC50 = 3250000 nM T34562 D0T0YI 378 IC50 = 18500000 nM T25464 D06OMK 445643 IC50 = 14.8 nM T25464 D0G7UX 5284373 IC50 = 183 nM T25464 C12CHL 4470793 Ki > 300000 nM T25464 C6YF5L 9918081 Ki > 3000 nM T25464 CC30ZA 10305301 Ki > 200000 nM T25464 C9TQ7U 11105029 IC50 = 2.8 nM T25464 C7WJF0 15546641 IC50 = 7.2 nM T25464 CU2A6K 44306123 IC50 = 7.32 nM T25464 C7WNM2 44306124 IC50 = 4.17 nM T25464 C86EOZ 44306135 IC50 = 8.65 nM T25464 C8T5NI 44306145 IC50 = 14 nM T25464 CUH17I 44306155 IC50 = 8.7 nM T25464 C6OQ4D 44306156 IC50 = 5.85 nM T25464 CN58YR 44306157 IC50 = 7.25 nM T25464 C8N7QZ 44306253 IC50 = 4.93 nM T25464 CD8O6N 44306280 IC50 = 7.91 nM T25464 C68IRQ 44306324 IC50 = 3.96 nM T25464 CBI4S6 44373943 IC50 > 5000 nM T25464 CQX6L4 44374010 IC50 = 348 nM T25464 C4I9DK 44374019 IC50 = 742 nM T25464 CBH09L 44374020 IC50 = 363 nM T25464 C89QDY 44374110 IC50 = 890 nM T25464 CQ65HS 44374127 IC50 > 5000 nM T25464 CJ9G7T 44374128 IC50 = 1539 nM T25464 C4XI8B 44374132 IC50 = 581 nM T25464 CYO20C 44374169 IC50 = 636 nM T25464 C1G6CI 44374400 IC50 = 840 nM T25464 CS30FH 49863381 IC50 = 140 nM T25464 C3YI2V 49863382 IC50 = 89 nM T25464 CS48JU 49863383 IC50 = 49 nM T71367 D0E3TC 44259 IC50 = 0.57 nM T71367 D00SDR 90054634 IC50 = 330 nM T71367 D0HK8C 90054733 IC50 = 121 nM T71367 D0L2FW 90054621 IC50 = 546 nM T71367 CA3C5S 3685259 IC50 < 5000 nM T71367 CACS26 11561968 Ki > 1000 nM T71367 CU0E8O 11690457 Ki > 1000 nM T71367 CJ21EH 13626914 IC50 = 94 nM T71367 C5VPH9 16129448 IC50 = 892 nM T71367 CGD89T 27126517 IC50 = 861 nM T71367 CC71QJ 27666048 IC50 > 100000 nM T71367 C61HBG 45102725 IC50 = 4200 nM T71367 CLS29B 46872626 IC50 > 10000 nM T71367 C5BZV3 57958821 IC50 = 381 nM T71367 C1MR8Q 60097495 IC50 > 1000 nM T71367 C37NKO 67129970 IC50 > 10000 nM T71367 CK80LJ 67130050 IC50 = 9430 nM T71367 CV63UL 67240318 IC50 > 10000 nM T71367 C7GRV2 68755406 IC50 > 10000 nM T71367 C7D2UQ 69463478 IC50 = 189 nM T71367 CVIA91 71553085 IC50 = 120 nM T71367 C1TR3O 71553152 IC50 = 2480 nM T71367 CDJY72 71568837 IC50 = 1600 nM T71367 C8CAG7 71578921 IC50 > 10000 nM T71367 C6P5YH 71657853 IC50 = 1.4 nM T71367 CKRS82 71678791 IC50 = 18 nM T71367 C7ROZ1 71679297 IC50 = 46 nM T71367 C9JTE7 71679299 IC50 = 16 nM T71367 C9RQW2 71679784 IC50 = 32 nM T71367 CHR3P5 71679785 IC50 = 15 nM T71367 CK1HR0 71679949 IC50 = 41 nM T71367 CF7R0Y 71682057 IC50 = 8000 nM T71367 CZM67T 72703518 IC50 = 150 nM T71367 C84AEF 72705109 IC50 = 77 nM T71367 CBK47T 72705487 IC50 = 132 nM T71367 CVF5P0 73603034 IC50 = 5700 nM T71367 C3SJQ2 76336279 IC50 > 100000 nM T71367 CI6NL9 77068235 IC50 = 8 nM T71367 C7RO1U 86703926 IC50 = 60 nM T71367 C97DVA 89729987 IC50 = 401 nM T71367 C2O4JR 89730033 IC50 = 3.5 nM T71367 C4UY2V 89730039 IC50 = 1.6 nM T71367 CB7Y0S 89730041 IC50 = 3.7 nM T71367 CQM98T 89730047 IC50 = 3.7 nM T71367 CC97QK 90054623 IC50 = 689 nM T71367 C93YPW 90054630 IC50 = 1700 nM T71367 CX0WH7 90054720 IC50 = 297 nM T71367 C9CRM6 90054726 IC50 = 423 nM T71367 CJX51L 90054730 IC50 = 225 nM T71367 CRF7M2 90054734 IC50 = 387 nM T71367 CEO7I0 90054986 IC50 = 58 nM T71367 CIZ2T6 90055028 IC50 = 351 nM T71367 C3ZV1C 90655985 IC50 = 5840 nM T71367 CE9KY0 90655986 IC50 = 2120 nM T71367 C6JIP7 91664348 IC50 = 4000 nM T71367 C18QYF 105539853 IC50 = 19.95 nM T71367 CBZ59D 118701008 IC50 = 3.7 nM T71367 C9CUL3 118711764 IC50 = 1600 nM T71367 CZH6E4 118711841 IC50 = 150 nM T71367 CYL46R 118711842 IC50 = 70 nM T71367 C2OK7E 118711843 IC50 = 710 nM T71367 CR8B9H 118711844 IC50 = 160 nM T71367 C5VDI0 118711845 IC50 = 840 nM T71367 C92TDH 118711846 IC50 = 300 nM T71367 C37IZJ 118711847 IC50 = 640 nM T71367 C8XFB1 118711848 IC50 = 130 nM T71367 COM51H 118711849 IC50 = 180 nM T71367 C7CB6W 118711850 IC50 = 10 nM T71367 CPNM74 118711851 IC50 = 70 nM T71367 C48DCS 118711852 IC50 = 10 nM T71367 CX8CL3 118711853 IC50 = 11000 nM T71367 CZV53F 118711854 IC50 = 19000 nM T71367 C2LT9G 118711855 IC50 = 37000 nM T71367 C0VBS5 118711856 IC50 = 7000 nM T71367 C0IJF5 118711857 IC50 = 23000 nM T71367 C7JV3C 118711858 IC50 = 3000 nM T71367 C4LJ6U 118711859 IC50 = 10000 nM T71367 C0QDO9 118711860 IC50 = 6000 nM T71367 CK0W1O 118711861 IC50 = 1000 nM T71367 C9XBL5 118711862 IC50 = 2000 nM T71367 CT3IS4 118711863 IC50 = 2000 nM T71367 C26EOM 118711864 IC50 = 1000 nM T71367 C9AGI1 118711865 IC50 = 2000 nM T71367 C2SQ6P 118711866 IC50 = 2000 nM T71367 C5GPJ9 118711891 IC50 = 2000 nM T71367 C76KYO 118711892 IC50 = 6000 nM T71367 CKBQ72 118711893 IC50 = 3000 nM T71367 CEU0S4 118711894 IC50 = 5000 nM T71367 CK63ES 118711895 IC50 = 10000 nM T71367 C92ZJE 118711896 IC50 = 8000 nM T71367 C2JA8B 127025153 IC50 = 600 nM T71367 CVUE54 127025154 IC50 = 84 nM T71367 C6W1UY 127025155 IC50 = 64 nM T71367 CLIP96 127026999 IC50 = 96 nM T71367 CEBO19 127027293 IC50 = 46 nM T71367 C5CUO0 127027294 IC50 = 248 nM T71367 CYS8L4 127027295 IC50 = 270 nM T71367 C39LPD 127027304 IC50 = 20 nM T71367 C3E7FZ 127028834 IC50 = 410 nM T71367 CJX04U 127029806 IC50 = 1509 nM T71367 CWVN31 127029807 IC50 = 1722 nM T71367 C9TZ7D 127034994 IC50 = 48 nM T71367 CE7M4J 127036775 IC50 = 14.9 nM T71367 CP89UZ 127036952 IC50 = 13 nM T71367 CX3Z7Q 134136970 IC50 > 100000 nM T71367 C82XFJ 134139661 IC50 > 100000 nM T71367 CKB1J9 134144378 IC50 = 44000 nM T71367 COF17E 134147249 IC50 = 5600 nM T71367 C60OFR 134154014 IC50 > 100000 nM T71367 CY4D8I 135566504 Ki = 812.4 nM T71367 CG3UZ1 135927974 Ki > 1000 nM T71367 CWGA76 137530158 IC50 = 12.59 nM T71367 CI1E8V 137634241 IC50 > 10000 nM T71367 C2E4DP 139592531 IC50 = 158.49 nM T71367 CZ7YS0 146027031 IC50 = 19.95 nM T71367 C2MD1Q 155513187 IC50 > 10000 nM T71367 CE7TI4 155521619 IC50 = 7943.28 nM T71367 CPW4H0 155531070 IC50 = 19952.62 nM T71367 CONB81 155557716 IC50 = 3981.07 nM T71367 D0NY6U 86703914 IC50 = 17 nM T71367 D0O6OH 71553154 IC50 = 18 nM T86928 D04AIT 5280445 IC50 = 500 nM T86928 D0K8KX 5280343 IC50 = 550 nM T86928 D0R3JB 4212 IC50 = 660 nM T86928 D09JEJ 24748573 IC50 = 3 nM T86928 D0B9BU 6918454 EC50 = 100 nM T86928 D0WS1V 448991 IC50 > 10000 nM T86928 C2OAV0 7328982 EC50 = 1600 nM T86928 CQVZ16 44123806 IC50 = 710 nM T86928 C1O6NR 44123807 IC50 = 480 nM T86928 C91MBN 44123808 IC50 = 820 nM T86928 CX08MT 44590715 IC50 = 2610 nM T86928 CVK4W9 44590746 IC50 = 2600 nM T86928 CO1UP9 44590747 IC50 = 5870 nM T86928 C3QRL8 44590749 IC50 = 2500 nM T86928 C4MY0L 44590794 IC50 = 8600 nM T86928 CLPU05 44590795 IC50 = 1520 nM T86928 C1CQS8 44590796 IC50 = 1100 nM T86928 C1MR8Q 60097495 IC50 > 10000 nM T86928 CPL8X0 139593287 EC50 = 6000 nM T86928 C7UNX2 145991479 IC50 < 1000 nM T86928 C2MD1Q 155513187 IC50 > 10000 nM T86928 C4PL1X 155536605 IC50 = 45100 nM T86928 CT9D0Q 155547691 IC50 = 18230 nM T86928 C2G8TU 155550182 IC50 = 1650 nM T86928 C1ACW9 155552233 IC50 = 8070 nM T86928 CDXK27 155562302 IC50 = 850 nM T86928 C6ICJ5 155562508 IC50 = 21990 nM T86928 CV74OB 155566389 IC50 = 4400 nM T86928 CGSU30 155566872 IC50 = 17750 nM T86928 D00RIX 5280443 IC50 = 800 nM T86928 D00YEV 5281605 IC50 = 10000 nM T86928 D01UYI 5281607 IC50 = 9000 nM T86928 D02DML 5281707 IC50 = 200 nM T86928 D07OAT 456214 IC50 > 10000 nM T86928 D0CP3M 5149739 IC50 = 930 nM T86928 D0G3TK 5280863 IC50 = 400 nM T86928 D0LH4L 10154 IC50 = 700 nM T86928 D0MF5Y 5281614 IC50 = 350 nM T86928 D0NJ4H 5281670 IC50 = 10000 nM T86928 D0O1YH 1694 IC50 = 1600 nM T86928 D0T3PW 5281672 IC50 = 900 nM T59102 D00STL 644241 IC50 = 71 nM T59102 D01PZD 5329098 IC50 = 68 nM T59102 D03ZBT 11626560 IC50 > 1000 nM T59102 D07POC 176870 IC50 = 12200 nM T59102 D08CDI 208908 IC50 = 8500 nM T59102 D09GDD 11167602 IC50 = 1.5 nM T59102 D09KTS 24821094 IC50 > 1000 nM T59102 D0AZ3C 5291 IC50 = 72 nM T59102 D0E6XR 3062316 Ki < 10 nM T59102 D0G6QF 3081361 IC50 = 1100 nM T59102 D0H0EQ 24826799 IC50 = 1.2 nM T59102 D0J9ZR 4477 IC50 > 100000 nM T59102 D0R0MW 5329102 IC50 = 2 nM T59102 D0W5HK 216239 IC50 = 37 nM T59102 D00UZR 5330286 IC50 > 10000 nM T59102 D02UFQ 11620908 IC50 > 10000 nM T59102 D03AND 11656518 IC50 = 6 nM T59102 D08HOM 46207586 IC50 = 3 nM T59102 D0A1AQ 5329099 IC50 = 50 nM T59102 D0D1GF 42642645 IC50 = 9.4 nM T59102 D0E3TC 44259 IC50 = 0.6 nM T59102 D0HS5V 11234052 IC50 > 6000 nM T59102 D0M0XB 10302451 IC50 > 5000 nM T59102 D0M9QZ 11485656 IC50 = 60 nM T59102 D0O0LS 25141092 IC50 > 10000 nM T59102 D0O6WV 24794418 IC50 > 500 nM T59102 D0P6DJ 151194 IC50 = 490 nM T59102 D0T2ER 24767976 IC50 = 13 nM T59102 D0Z6MT 16662431 IC50 = 4 nM T59102 D03BNU 59604787 IC50 > 3500 nM T59102 D0JY1I 42613483 IC50 = 3900 nM T59102 D06GBK 2048 IC50 = 6200 nM T59102 D0H4GI 10275001 IC50 = 406 nM T59102 D0IT6Q 3038522 IC50 = 26 nM T59102 D0L5YF 5329032 IC50 = 3400 nM T59102 D0T3ME 156422 IC50 = 6200 nM T59102 C63WLY 89644 IC50 > 10 ug.mL-1 T59102 C5JE2Z 104860 IC50 = 7.6 ug.mL-1 T59102 C6Y9CV 151193 IC50 = 490 nM T59102 CI1NA5 159926 IC50 > 10 ug.mL-1 T59102 CYBA43 177458 IC50 > 10 ug.mL-1 T59102 C32HFB 396514 IC50 = 2000 nM T59102 C4MNG8 445840 IC50 = 5000 nM T59102 C75EDQ 644355 IC50 = 100 nM T59102 C5HPF3 644356 IC50 = 20 nM T59102 C9D7UY 727518 IC50 > 100000 nM T59102 CXB5A2 964113 IC50 > 100000 nM T59102 CDB17F 1538822 IC50 = 24200 nM T59102 CZ2B4M 2358462 IC50 > 100000 nM T59102 CXA1L7 2365265 IC50 > 100000 nM T59102 CEF62M 2379240 IC50 = 33100 nM T59102 CKT64G 2396126 IC50 > 10000 nM T59102 CFVK40 3008950 IC50 > 50000 nM T59102 CD8UW1 3008956 IC50 = 17000 nM T59102 CCD93P 3008957 IC50 > 50000 nM T59102 CU64VM 3008958 IC50 > 50000 nM T59102 C8F0KM 3008959 IC50 > 50000 nM T59102 CV8R9Z 3008960 IC50 > 50000 nM T59102 C8EZ6O 3008961 IC50 > 50000 nM T59102 CX95SU 3008962 IC50 = 8900 nM T59102 C9B2MN 3008963 IC50 > 50000 nM T59102 C9E7BW 3008964 IC50 > 50000 nM T59102 CGK91Q 3008965 IC50 = 14700 nM T59102 CCN9D5 3142817 IC50 = 1000 nM T59102 CY28LS 5293755 IC50 > 100000 nM T59102 CFW19M 5329009 IC50 = 3000 nM T59102 C9I7WT 5329100 IC50 = 60 nM T59102 CMWB28 5329101 IC50 = 17 nM T59102 CGX50J 5329104 IC50 = 5 nM T59102 C2VX0H 5329105 IC50 = 0.5 nM T59102 CK71MQ 5329106 IC50 = 1 nM T59102 CL0Q4S 5329107 IC50 = 3 nM T59102 C6YRH8 5329108 IC50 = 2 nM T59102 CFP59Y 5329109 IC50 = 1 nM T59102 C0JW3Y 5329134 IC50 = 2110 nM T59102 CO7J2A 5329135 IC50 = 620 nM T59102 CQ4TP5 5329136 IC50 = 8290 nM T59102 CXQC42 5329137 IC50 = 11300 nM T59102 CT94JS 5329138 IC50 = 140 nM T59102 CNH06M 5329139 IC50 = 4190 nM T59102 CRY4Z2 5329140 IC50 = 5980 nM T59102 CAPE50 5329141 IC50 = 1400 nM T59102 CFU58A 5329142 IC50 = 160 nM T59102 C5Q8XK 5329143 IC50 = 170 nM T59102 C8PX4D 5329144 IC50 = 650 nM T59102 C6USQ5 5329145 IC50 = 2780 nM T59102 C56LWT 5329146 IC50 = 3650 nM T59102 CZ16MN 5329147 IC50 = 1210 nM T59102 CAN16I 5329148 IC50 = 1530 nM T59102 CG4NC2 5329149 IC50 = 550 nM T59102 CIW70H 5329150 IC50 = 110 nM T59102 C5FT6A 5329151 IC50 = 230 nM T59102 CB0N4L 5329152 IC50 = 940 nM T59102 COFP24 5329153 IC50 = 680 nM T59102 CGWD98 5329154 IC50 = 5460 nM T59102 C4PD0K 5329156 IC50 = 11500 nM T59102 C0RWT8 5329157 IC50 = 1030 nM T59102 C3MU5S 5329158 IC50 = 3460 nM T59102 CN6O4R 5329159 IC50 = 70600 nM T59102 CG68DI 5329160 IC50 > 100000 nM T59102 CYR7V0 5329161 IC50 = 13900 nM T59102 C9BXE2 5329162 IC50 = 94010 nM T59102 CY4V5Z 5329163 IC50 = 240 nM T59102 CI64YA 5329164 IC50 = 4 nM T59102 C2ZV0O 5329165 IC50 < 780 nM T59102 CAB53L 5329166 IC50 = 20 nM T59102 CTW9R8 5329167 IC50 = 19300 nM T59102 C8A3TJ 5329168 IC50 = 40 nM T59102 CVTD82 5329169 IC50 = 680 nM T59102 CQ5WK1 5329170 IC50 = 870 nM T59102 CNC9T7 5329171 IC50 = 5430 nM T59102 C6L0UW 5329229 IC50 > 20000 nM T59102 C1DBV6 5329230 IC50 > 20000 nM T59102 CLKM80 5329231 IC50 > 20000 nM T59102 CTQ18A 5329232 IC50 > 100000 nM T59102 CM5KG6 5329233 IC50 > 20000 nM T59102 CQG6R2 5329234 IC50 > 20000 nM T59102 CJ3A9I 5329235 IC50 > 100000 nM T59102 CPS7X1 5329236 IC50 > 100000 nM T59102 CAN60T 5329237 IC50 > 20000 nM T59102 CY15JP 5329238 IC50 > 20000 nM T59102 C41UBI 5329239 IC50 > 20000 nM T59102 C6VQ9F 5329240 IC50 > 20000 nM T59102 C8WS5K 5329241 IC50 > 20000 nM T59102 CI26UN 5329242 IC50 > 20000 nM T59102 C6PJ2R 5329243 IC50 > 20000 nM T59102 C0OKB7 5329244 IC50 = 20000 nM T59102 C78ZNL 5329245 IC50 > 20000 nM T59102 CWL5S4 5329246 IC50 = 20000 nM T59102 C4X3OE 5329248 IC50 = 5620 nM T59102 CK8FH6 5329249 IC50 > 20000 nM T59102 CN5B6C 5329250 IC50 > 20000 nM T59102 CQ0B6E 5329251 IC50 > 10000 nM T59102 C4KO3N 5329252 IC50 > 100000 nM T59102 C6MZF8 5329253 IC50 > 20000 nM T59102 C9NBG7 5330546 IC50 = 70 nM T59102 CS3A8F 5331081 IC50 > 20000 nM T59102 CG4W8K 5331082 IC50 > 20000 nM T59102 CD4C2A 5331083 IC50 > 20000 nM T59102 C6AT8V 5331084 IC50 > 20000 nM T59102 CJVS23 5331085 IC50 > 20000 nM T59102 CZ29FN 5331086 IC50 > 20000 nM T59102 CYL78A 5331087 IC50 > 20000 nM T59102 CJ87XR 5331088 IC50 = 2100 nM T59102 CFB3K7 5331089 IC50 = 18000 nM T59102 C9WY1O 5331090 IC50 > 20000 nM T59102 C9ZK3D 5331091 IC50 > 20000 nM T59102 C6RJC8 5331092 IC50 = 1100 nM T59102 C0IOY8 5331093 IC50 = 1400 nM T59102 CMD08O 5331094 IC50 = 1100 nM T59102 CDQ3M7 5359485 IC50 = 0.89 ug.mL-1 T59102 C54BYP 5360741 IC50 = 1.8 ug.mL-1 T59102 CD65JT 5427216 IC50 > 100000 nM T59102 CPB95V 5427224 IC50 > 100000 nM T59102 C61NCL 5482344 IC50 = 1800 nM T59102 CDK3J0 5703619 IC50 = 0.4 nM T59102 CA6L5V 5707304 IC50 > 100000 nM T59102 C43YGE 5713379 IC50 > 100000 nM T59102 CT8U7I 5874584 IC50 = 8390 nM T59102 CM8LW9 6036100 IC50 > 100000 nM T59102 C6L5HS 6419386 IC50 = 2800 nM T59102 C3CQW0 6419387 IC50 = 1000 nM T59102 CWOA63 6419388 IC50 = 2000 nM T59102 CZVU64 6419389 IC50 = 1400 nM T59102 C9FN4B 6419390 IC50 = 800 nM T59102 CN53YW 6419391 IC50 = 4000 nM T59102 C17NWJ 6419392 IC50 = 600 nM T59102 C13IRC 6419393 IC50 = 2000 nM T59102 C4FLE9 6419394 IC50 = 800 nM T59102 C4GHT0 6419395 IC50 = 4000 nM T59102 C8SAQ1 6419396 IC50 > 10000 nM T59102 CP71CL 6419397 IC50 > 10000 nM T59102 CQ3S8L 6450842 IC50 = 3700 nM T59102 C2N0IR 6477203 IC50 = 12800 nM T59102 CW5YJ2 6536705 IC50 > 100000 nM T59102 C2OL7K 9796455 IC50 = 353 nM T59102 CI80BK 9803350 IC50 = 2500 nM T59102 C9TAL6 9826308 IC50 = 160 nM T59102 CWVH12 9828619 IC50 = 50 nM T59102 CX10KR 9828962 IC50 = 170 nM T59102 CE5X8J 9844744 IC50 = 490 nM T59102 CSAY10 9845576 IC50 = 1500 nM T59102 C6A9HS 9871170 IC50 = 97 nM T59102 C3CI1J 9872659 IC50 = 20 nM T59102 CUZ07T 9884745 IC50 > 100000 nM T59102 CHF7G5 9890746 IC50 = 90 nM T59102 CXA5C8 9893493 IC50 > 2000 nM T59102 CZ25GL 9894619 IC50 = 70 nM T59102 C3EUB4 9911005 IC50 = 240 nM T59102 C24JTF 9911313 IC50 = 13300 nM T59102 C1Y3MH 9915808 IC50 = 90 nM T59102 C6HP3L 9948410 IC50 > 100000 nM T59102 C7T9DJ 9950440 IC50 > 30000 nM T59102 CO4N3Q 9995374 IC50 > 100000 nM T59102 C5WF7J 10007113 IC50 = 300 nM T59102 CY90DN 10023010 IC50 = 5 nM T59102 CJ95HR 10041745 IC50 = 12 nM T59102 CG57EC 10047098 IC50 = 13400 nM T59102 CUJR40 10062694 EC50 = 6 nM T59102 C1JUF8 10073832 IC50 > 2000 nM T59102 CIV15Q 10113978 IC50 = 84 nM T59102 C5WCL2 10117540 IC50 = 216 nM T59102 C5KHX2 10118413 IC50 = 50 nM T59102 C46DHW 10119600 IC50 = 230 nM T59102 CRNC72 10120038 IC50 = 90 nM T59102 C4VW8P 10121424 IC50 = 40 nM T59102 CYQ01B 10121530 IC50 = 30 nM T59102 CR5D2N 10121709 IC50 = 1 nM T59102 C5X7LQ 10121737 IC50 = 20 nM T59102 C3XW0Y 10122339 IC50 = 2.4 nM T59102 C6IA4L 10143909 IC50 = 77 nM T59102 C7X5LY 10145209 IC50 = 110 nM T59102 CL89XT 10165712 IC50 = 2 nM T59102 C76XOL 10166902 IC50 = 10 nM T59102 C1Y7HR 10167597 IC50 = 36 nM T59102 CR5Y7O 10168074 IC50 = 0.4 nM T59102 CJH54G 10186893 IC50 = 1430 nM T59102 C3ER4N 10187285 IC50 < 4 nM T59102 CM26BU 10187537 IC50 = 140 nM T59102 CA03YO 10187699 IC50 = 1010 nM T59102 CUG37L 10187829 IC50 = 335 nM T59102 C8T7RC 10188599 IC50 = 265 nM T59102 C6FB3Q 10188863 IC50 = 5040 nM T59102 C0N3HC 10189022 IC50 = 50 nM T59102 C6G2RK 10189131 IC50 = 20 nM T59102 CD4C9B 10207679 IC50 = 70 nM T59102 CZU79W 10208916 IC50 = 320 nM T59102 C4G2AD 10209993 IC50 = 9 nM T59102 CZJ78I 10210309 IC50 = 145 nM T59102 CBFZ09 10210632 IC50 = 99 nM T59102 C5YCN2 10215023 IC50 = 66000 nM T59102 C95ZXY 10226609 IC50 = 800 nM T59102 CB83CI 10228726 IC50 = 10 nM T59102 C18DRH 10229841 IC50 = 710 nM T59102 CD7J3O 10231458 IC50 = 20 nM T59102 CL9N2E 10231519 IC50 = 100 nM T59102 CAE03L 10231813 IC50 < 4 nM T59102 CPD6Z9 10236164 IC50 > 100000 nM T59102 CX15BI 10246728 IC50 = 3 nM T59102 C1WL8B 10251852 IC50 > 500000 nM T59102 CH30RC 10253133 IC50 = 1400 nM T59102 CBI47E 10264222 IC50 > 100000 nM T59102 C6DC8Q 10275163 IC50 = 3300 nM T59102 CD2IE3 10278606 IC50 = 920 nM T59102 CH5DQ0 10280082 IC50 = 140 nM T59102 C65JZS 10296462 IC50 = 1250 nM T59102 CVO54Z 10300451 IC50 > 20000 nM T59102 C63DPY 10301981 IC50 = 10 nM T59102 CO90LX 10302121 IC50 = 216 nM T59102 CC4G8B 10302519 IC50 < 4 nM T59102 C2T3WU 10302586 IC50 = 168 nM T59102 C4FP8M 10303591 IC50 < 4 nM T59102 C5CBF9 10320381 IC50 = 6600 nM T59102 C97YDQ 10344304 IC50 = 510 nM T59102 CZV0G7 10359698 IC50 = 16 nM T59102 CQB9H7 10389422 IC50 = 11000 nM T59102 CLAX64 10413508 IC50 = 11000 nM T59102 CQ43JU 10426229 IC50 = 17500 nM T59102 CU8JP3 10432698 IC50 = 1100 nM T59102 C95LYF 10457505 IC50 = 530 nM T59102 C7PLI5 10478569 IC50 > 2000 nM T59102 CJ5M1D 10482445 IC50 = 8000 nM T59102 CJWH60 10489322 IC50 > 100000 nM T59102 C5SVT4 10537949 IC50 > 100000 nM T59102 CGAW17 10562306 IC50 = 85400 nM T59102 C6AJI9 10562777 IC50 = 25500 nM T59102 CE5L6D 10587839 IC50 > 100000 nM T59102 CM8N6L 10593765 IC50 = 24500 nM T59102 CI30LZ 10613858 IC50 > 100000 nM T59102 CH6Z3L 10635478 IC50 = 65500 nM T59102 CB97UD 10636005 IC50 > 100000 nM T59102 C2UWA0 10658651 IC50 = 41700 nM T59102 C5L0IX 10663368 IC50 > 100000 nM T59102 C9Z7XH 10663503 IC50 = 49900 nM T59102 CH1G6P 10682457 IC50 > 100000 nM T59102 C54UAK 10728035 IC50 = 2800 nM T59102 CXSH91 10753550 IC50 = 18200 nM T59102 CVPW04 10755069 IC50 > 100000 nM T59102 C3WR0Q 10779668 IC50 > 100000 nM T59102 CF5T1H 10783444 IC50 > 100000 nM T59102 CX1DH7 10862508 IC50 = 6720 nM T59102 CU8P7M 10862866 IC50 = 2000 nM T59102 C54VTR 10863323 IC50 = 720 nM T59102 C43CLE 10863395 IC50 = 440 nM T59102 CD8M0L 10863993 IC50 = 8180 nM T59102 C71JKT 10873266 IC50 > 30000 nM T59102 C16FCD 10874104 IC50 = 18200 nM T59102 CY7E1M 10874618 IC50 = 160 nM T59102 CU92JA 10875187 IC50 = 1.4 nM T59102 CSTP13 10875630 IC50 = 26 nM T59102 C6QV1L 10885200 IC50 = 9420 nM T59102 C8TDN1 10885583 IC50 = 2210 nM T59102 C70PLZ 10885776 IC50 = 6500 nM T59102 CI4XR0 10885830 IC50 = 20 nM T59102 CRN57U 10895433 IC50 = 2570 nM T59102 CJSX79 10896366 IC50 = 4690 nM T59102 C0BN9J 10896386 IC50 = 150 nM T59102 CJ4P5T 10905857 IC50 = 850 nM T59102 CM5IA4 10906467 IC50 = 210 nM T59102 CO21NS 10907015 IC50 = 80 nM T59102 CB0MK5 10907225 IC50 = 150 nM T59102 C2IOU4 10907383 IC50 = 2810 nM T59102 CC3P6X 10907564 IC50 = 520 nM T59102 CJUI34 10917610 IC50 = 510 nM T59102 CCB49T 10917872 IC50 = 1040 nM T59102 C4WJ2T 10918068 IC50 = 715 nM T59102 C62LQW 10918358 IC50 = 290 nM T59102 C4OX0I 10918469 IC50 = 662 nM T59102 CS0BJ5 10928229 IC50 = 110 nM T59102 C1DS2G 10929540 IC50 = 440 nM T59102 C7MTO0 10929814 IC50 = 2970 nM T59102 CY0J9W 10951558 IC50 = 53 nM T59102 CJE7Y2 10961232 IC50 > 10000 nM T59102 C94GTN 10963029 IC50 = 5000 nM T59102 CBT4S3 10963044 IC50 = 29 nM T59102 CAC02X 10963192 IC50 = 500 nM T59102 CKD72X 10972606 IC50 = 9210 nM T59102 CL89QG 10973305 IC50 = 100 nM T59102 CPY51V 10983215 IC50 = 30 nM T59102 CCN5F8 10984279 IC50 = 3230 nM T59102 C9ELG2 10984685 IC50 = 222 nM T59102 CAP7E6 10995060 IC50 = 305 nM T59102 CB5AD7 11004892 IC50 = 230 nM T59102 C53QCD 11006148 IC50 = 177 nM T59102 C0LK2Q 11006502 IC50 = 494 nM T59102 CC87FE 11015336 IC50 = 1210 nM T59102 C71TOQ 11015640 IC50 > 30000 nM T59102 CY3B6O 11015880 IC50 = 330 nM T59102 C4F8ZN 11026804 IC50 > 30000 nM T59102 CDQ0H4 11027671 IC50 = 178 nM T59102 C59LQM 11027750 IC50 = 100 nM T59102 C4GLS2 11036639 IC50 = 11100 nM T59102 C9NYE2 11037955 IC50 = 290 nM T59102 CT5V2C 11039013 IC50 = 813 nM T59102 CL3FG7 11039428 IC50 = 0.4 nM T59102 CJ05CL 11048367 IC50 = 80 nM T59102 CWVC81 11049206 IC50 = 2310 nM T59102 C5V9DI 11049316 IC50 = 5590 nM T59102 CD9GY6 11049581 IC50 = 1260 nM T59102 C04QKG 11069972 IC50 = 2060 nM T59102 CXDA03 11070177 IC50 > 30000 nM T59102 CB7ND4 11071122 IC50 = 290 nM T59102 C0HM8T 11071223 IC50 = 160 nM T59102 CYG8V1 11071546 IC50 = 335 nM T59102 CV4R8X 11081103 IC50 = 740 nM T59102 CM04HI 11081393 IC50 = 60 nM T59102 CKX3Z5 11081446 IC50 = 220 nM T59102 C4G2AF 11091152 IC50 = 5360 nM T59102 CEB97L 11112669 IC50 = 1260 nM T59102 C4YUN5 11112927 IC50 > 30000 nM T59102 CQDC05 11113190 IC50 = 190 nM T59102 CYH21N 11113218 IC50 > 30000 nM T59102 CDZ80M 11114435 IC50 = 582 nM T59102 C5MAN7 11124388 IC50 = 300 nM T59102 C6HQ2L 11133954 IC50 = 480 nM T59102 CM9QT3 11143981 IC50 = 9960 nM T59102 C9KES6 11144730 IC50 = 790 nM T59102 CTJ9U3 11145086 IC50 = 1410 nM T59102 CU5DO2 11145515 IC50 = 20 nM T59102 C0D8CT 11155618 IC50 = 180 nM T59102 C7CNO9 11156466 IC50 = 100 nM T59102 CMJ31L 11156812 IC50 = 20 nM T59102 CBDS75 11157185 IC50 = 90 nM T59102 CP16ND 11168221 IC50 = 80 nM T59102 CL8Y4F 11177747 IC50 = 270 nM T59102 CWIT81 11178110 IC50 = 150 nM T59102 CCAG52 11179181 IC50 = 70 nM T59102 CK7B4X 11190431 IC50 > 30000 nM T59102 CBG94A 11191231 IC50 = 40 nM T59102 C7BHE0 11200526 IC50 = 4590 nM T59102 C09YIQ 11202821 IC50 > 30000 nM T59102 C65JPE 11212551 IC50 > 30000 nM T59102 C50JAG 11223943 IC50 = 1440 nM T59102 CN6BC7 11226164 IC50 > 30000 nM T59102 C87WCG 11226298 IC50 = 1390 nM T59102 CYA59I 11235645 IC50 > 30000 nM T59102 C0E1ML 11236566 IC50 = 140 nM T59102 C1QAS6 11237612 IC50 = 190 nM T59102 CH2VD7 11245435 IC50 > 30000 nM T59102 CGL6R0 11249274 IC50 = 200 nM T59102 CUV15L 11249319 IC50 > 30000 nM T59102 CKRA10 11258984 IC50 > 10000 nM T59102 C9F6KW 11260252 IC50 = 180 nM T59102 CC93YJ 11260253 IC50 > 30000 nM T59102 C6ZD4C 11270126 IC50 > 30000 nM T59102 CKI25P 11272815 IC50 = 70 nM T59102 CJW65Q 11273677 IC50 > 30000 nM T59102 C3IU8T 11281396 IC50 = 1300 nM T59102 C28XHQ 11282038 IC50 = 620 nM T59102 CZX0K9 11283270 IC50 = 550 nM T59102 C9I8AN 11293184 IC50 > 30000 nM T59102 C7I9TG 11293913 IC50 = 310 nM T59102 CIXK95 11295243 IC50 = 640 nM T59102 CYFT17 11295612 IC50 = 780 nM T59102 CNF7V4 11304951 IC50 > 30000 nM T59102 CVCE09 11305002 IC50 = 2700 nM T59102 CEN1J8 11306433 IC50 > 30000 nM T59102 C5PW1K 11306478 IC50 > 30000 nM T59102 CJ3N8G 11316908 IC50 > 30000 nM T59102 C41RWG 11318423 IC50 = 330 nM T59102 CVQ1Y0 11318736 IC50 = 20 nM T59102 C9G4YJ 11325945 IC50 > 30000 nM T59102 C2WKC3 11330812 IC50 > 30000 nM T59102 C15ZLJ 11340108 IC50 = 100 nM T59102 C4ICB0 11341503 IC50 = 650 nM T59102 C9K3LZ 11350308 IC50 = 1540 nM T59102 CV3K6Q 11351606 IC50 > 10000 nM T59102 C1LT5J 11352217 IC50 > 30000 nM T59102 CU18NY 11352407 IC50 = 3260 nM T59102 C24LHS 11353568 IC50 = 21000 nM T59102 C1UD0O 11372879 IC50 > 30000 nM T59102 CM4UY7 11373369 IC50 = 170 nM T59102 C25ZCN 11374110 IC50 = 130 nM T59102 C6EGP9 11374800 IC50 = 90 nM T59102 C8TLG4 11396174 IC50 = 380 nM T59102 CL19HT 11397589 IC50 = 810 nM T59102 C41NOY 11409644 IC50 = 80 nM T59102 CEG81P 11419763 IC50 = 130 nM T59102 C9IQP7 11419787 IC50 > 30000 nM T59102 C3NBZ9 11420151 IC50 = 6080 nM T59102 CMAI17 11420386 IC50 = 10200 nM T59102 CREQ51 11429654 IC50 = 96 nM T59102 CVQC06 11429694 IC50 > 30000 nM T59102 C9WEH6 11432198 IC50 = 60 nM T59102 C7AI2V 11432911 IC50 > 2000 nM T59102 C17WNX 11443611 IC50 = 90 nM T59102 C3SKT6 11443633 IC50 = 80 nM T59102 COF7Z1 11443718 IC50 > 30000 nM T59102 C6I2ER 11455034 IC50 = 100 nM T59102 CX5L2B 11464443 IC50 = 10300 nM T59102 CD3P4Q 11465678 IC50 = 390 nM T59102 CT34RJ 11466063 IC50 = 290 nM T59102 C6M9NC 11477626 IC50 > 2000 nM T59102 CEB29T 11490006 IC50 > 30000 nM T59102 C46JFZ 11494322 IC50 = 33 nM T59102 C9K8RE 11496022 IC50 = 137 nM T59102 CY72AM 11496228 IC50 = 659 nM T59102 C5UEK0 11510816 IC50 = 110 nM T59102 CG3BZ9 11517980 IC50 = 4 nM T59102 CFQ42U 11525980 IC50 = 23 nM T59102 CL7X4Q 11530963 IC50 = 1867 nM T59102 CID2P7 11536421 IC50 = 54 nM T59102 C6IOJ4 11546085 IC50 = 310 nM T59102 CF28TK 11565353 IC50 = 217 nM T59102 CZ1H0X 11569258 IC50 = 5500 nM T59102 CRL95F 11569396 IC50 = 1 nM T59102 CO9KP5 11583459 IC50 > 10000 nM T59102 CB91RQ 11589811 IC50 = 40 nM T59102 CM65QP 11590120 IC50 = 3 nM T59102 C69FYK 11604142 Ki = 200 nM T59102 CEG5W8 11608830 IC50 = 9 nM T59102 C8IKG5 11616255 IC50 = 458 nM T59102 CCB3X0 11617740 IC50 = 6220 nM T59102 CSM62L 11626920 IC50 = 31 nM T59102 CK34LS 11632737 IC50 = 200 nM T59102 C7W3TE 11633427 IC50 = 10 nM T59102 C5R6DG 11634086 IC50 > 800 nM T59102 C8V0YT 11639969 IC50 = 1200 nM T59102 CZM9K1 11675974 IC50 = 410 nM T59102 C3M1CF 11682291 IC50 = 5420 nM T59102 CCX2F5 11682611 IC50 = 0.4 nM T59102 C8AEX7 11687971 IC50 = 151900 nM T59102 CHG14R 11688408 IC50 = 55 nM T59102 CZY05V 11719421 IC50 = 6 nM T59102 CUB2N6 11719537 IC50 = 5 nM T59102 C9P0VD 11729539 IC50 = 550 nM T59102 CBL38T 11730367 IC50 = 260 nM T59102 C4PE0D 11730369 IC50 = 1140 nM T59102 C3DVE0 11730809 IC50 = 370 nM T59102 CCQO28 11731042 IC50 = 871 nM T59102 C23STH 11731130 IC50 = 601 nM T59102 CSLC27 11731197 IC50 = 50 nM T59102 C5NLG6 11732326 IC50 = 3180 nM T59102 CU54IA 11732691 IC50 > 30000 nM T59102 C2M7ZD 11733137 IC50 = 1240 nM T59102 C67FZJ 11734285 IC50 = 400 nM T59102 CT49LJ 11734851 IC50 = 12 nM T59102 CU9BR4 11749848 IC50 > 30000 nM T59102 C0QV3M 11752083 IC50 = 10900 nM T59102 CAS0V7 11752632 IC50 = 290 nM T59102 CP7AH3 11755812 IC50 = 7700 nM T59102 CRW2H3 11762328 IC50 = 21600 nM T59102 CRI64Z 11762329 IC50 = 1200 nM T59102 CJI7T6 11763085 IC50 = 76 nM T59102 C61QXW 11785508 IC50 > 30000 nM T59102 CEOH20 11813259 IC50 = 943 nM T59102 C89SNG 11813434 IC50 > 30000 nM T59102 C4V8PJ 11813761 IC50 = 110 nM T59102 C1CI6M 11826385 IC50 = 440 nM T59102 CEUB71 11826832 IC50 = 1470 nM T59102 C9EV8H 11827121 IC50 = 3110 nM T59102 C72RZN 11827714 IC50 = 720 nM T59102 C14MZC 11827841 IC50 = 6750 nM T59102 CDZ1I3 11989153 IC50 = 637 nM T59102 CM50UH 12000646 EC50 = 170 nM T59102 CI39TK 12004372 IC50 = 10700 nM T59102 CDGF78 15282555 IC50 = 3300 nM T59102 C7LB4I 15949613 IC50 = 96 nM T59102 C9TU1O 16046126 IC50 > 1000 nM T59102 CW2XK6 16050925 IC50 = 110 nM T59102 C9JK2M 16059071 IC50 > 2000 nM T59102 CW6UJ9 16059338 IC50 > 1000 nM T59102 CH7MS6 16059729 IC50 > 42000 nM T59102 CFKE48 16064750 IC50 = 1 nM T59102 CQG45C 16109001 IC50 = 1940 nM T59102 C5VPH9 16129448 IC50 = 5270 nM T59102 C0V8FB 16730091 IC50 = 2 nM T59102 CA24TE 16730092 IC50 = 5 nM T59102 CGX61W 22041319 IC50 = 10 nM T59102 CYP32E 22707343 IC50 = 540 nM T59102 CFO6J5 22707344 IC50 = 10700 nM T59102 CWXO86 22707354 IC50 = 1320 nM T59102 C8JD2X 22707384 IC50 > 750 nM T59102 CAG61Z 22707433 IC50 = 2880 nM T59102 C20RYA 22707442 IC50 = 1380 nM T59102 CNR0O7 22707450 IC50 = 5160 nM T59102 CEOV57 22707452 IC50 > 100 nM T59102 CPO51J 22707462 IC50 = 6250 nM T59102 CGR94W 22707466 IC50 = 500 nM T59102 C3H1VE 22707498 IC50 = 1160 nM T59102 CDI35F 22707517 IC50 > 30000 nM T59102 C6MBW9 22707526 IC50 = 970 nM T59102 CQ3TW0 22707568 IC50 = 29700 nM T59102 CB29GC 22707603 IC50 = 350 nM T59102 C2UO3S 22707619 IC50 > 30000 nM T59102 CM5R8B 22707669 IC50 = 1120 nM T59102 C7G6NJ 22707741 IC50 = 5170 nM T59102 C9QLP0 23133323 IC50 = 1100 nM T59102 CG12OL 23518511 IC50 > 20000 nM T59102 CRX0Q6 23625758 IC50 = 780 nM T59102 C2RV3U 24180608 IC50 > 30000 nM T59102 C3X1WH 24742411 IC50 = 2 nM T59102 CS78XJ 24742412 IC50 = 3 nM T59102 C2KA6G 24742584 IC50 = 4 nM T59102 CN9GC8 24742586 IC50 = 10 nM T59102 CHU49V 24757938 IC50 < 1 nM T59102 C0D2PA 24758868 IC50 = 20 nM T59102 C3K5YO 24758982 IC50 = 7 nM T59102 CYU0Z8 24758983 IC50 = 6 nM T59102 CJL67N 24759089 IC50 = 4 nM T59102 C2APK8 24759090 IC50 = 9 nM T59102 C5CRF6 24759091 IC50 = 6 nM T59102 CA8U7X 24759094 IC50 = 4 nM T59102 CRB89L 24759205 IC50 = 1 nM T59102 C13JUP 24759314 IC50 = 5 nM T59102 CCPS81 24764502 IC50 > 35000 nM T59102 C9B2TF 24880043 IC50 = 150 nM T59102 CFK2B9 24882503 IC50 = 1400 nM T59102 C43HWQ 24883287 IC50 > 10000 nM T59102 C8DA5Q 24883334 IC50 > 10000 nM T59102 C4V9GH 24894117 IC50 = 11000 nM T59102 CJH19T 24894883 IC50 = 45000 nM T59102 CB5TP8 24894992 IC50 = 38000 nM T59102 CF4N9X 24895100 IC50 = 40000 nM T59102 CY8L7E 24896769 IC50 > 10000 nM T59102 CN13JF 24899915 IC50 = 1.3 ug.mL-1 T59102 CBWR97 24899916 IC50 = 1.8 ug.mL-1 T59102 C9F2JD 24899917 IC50 > 10 ug.mL-1 T59102 C64MTI 24900160 IC50 = 5.8 ug.mL-1 T59102 CO2I6Q 24900161 IC50 > 10 ug.mL-1 T59102 C5FD1A 24937369 IC50 = 5300 nM T59102 C4KG0Y 25022599 IC50 > 1000 nM T59102 CRO0Y8 25022735 IC50 = 90000 nM T59102 C72AJM 25022736 IC50 > 500000 nM T59102 CQ27UI 25113814 IC50 = 10 nM T59102 C2IHY0 25114266 IC50 = 5 nM T59102 CP8S9W 25116064 IC50 = 11 nM T59102 CTV54O 25123227 IC50 = 14 nM T59102 C1IYN7 25127854 IC50 = 5.9 nM T59102 CKD14B 25127856 IC50 = 19 nM T59102 CJBX60 25128180 IC50 = 8.3 nM T59102 CC5SD9 25128181 IC50 = 21 nM T59102 CIG4H0 25178539 IC50 = 4200 nM T59102 C4GI6J 25178540 IC50 = 6700 nM T59102 CL0Z1F 25181502 IC50 = 830 nM T59102 COB9G8 25181586 IC50 = 2800 nM T59102 C8YLD6 25194331 IC50 = 5 nM T59102 CXC9B3 25194865 IC50 = 9 nM T59102 C1I0VS 25194866 IC50 = 3 nM T59102 C9OZN3 25194867 IC50 = 30 nM T59102 C6FGQ1 25206346 IC50 = 91 nM T59102 CXNW87 25207322 IC50 = 8 nM T59102 C8IJB9 25218207 IC50 = 40300 nM T59102 C2TXC6 25218656 IC50 > 2000 nM T59102 CVM13K 42596931 IC50 = 100 nM T59102 CU53WB 42596953 IC50 = 2500 nM T59102 C7GIQ3 42625508 IC50 = 4600 nM T59102 CVZ83M 42625582 IC50 = 2700 nM T59102 C5MD9E 42625892 IC50 = 7300 nM T59102 CJ5U1X 42639664 IC50 = 6.4 ug.mL-1 T59102 CEL61X 44229839 IC50 > 10000 nM T59102 C4NWP5 44246325 IC50 > 200000 nM T59102 C2EW0I 44246326 IC50 = 118000 nM T59102 CSD8T0 44246327 IC50 > 200000 nM T59102 CMKF08 44246328 IC50 > 200000 nM T59102 CAO87V 44246329 IC50 > 200000 nM T59102 CLU2V3 44246330 IC50 = 17400 nM T59102 CHZ6Q1 44269004 IC50 = 10 nM T59102 CY6WC0 44299236 IC50 = 13000 nM T59102 C3RG0C 44299304 IC50 = 2300 nM T59102 CJM26I 44299321 IC50 = 4700 nM T59102 C9UGL3 44299325 IC50 = 10000 nM T59102 CJEZ96 44299338 IC50 = 9000 nM T59102 C8XGN5 44299339 IC50 = 5100 nM T59102 CNH34G 44299354 IC50 = 5600 nM T59102 C82MSD 44299360 IC50 = 18000 nM T59102 CSY8A3 44321301 IC50 > 100000 nM T59102 CCG2M5 44321317 IC50 = 60400 nM T59102 CY9ED1 44321395 IC50 > 100000 nM T59102 C5U1CR 44321686 IC50 > 10000 nM T59102 CETY53 44321717 IC50 = 66000 nM T59102 CV60ME 44321734 IC50 = 13800 nM T59102 C61OFE 44332377 IC50 > 1000 nM T59102 CI2NP3 44332378 IC50 = 160 nM T59102 CHKA01 44332616 IC50 = 820 nM T59102 CYAU21 44349046 IC50 = 409 nM T59102 CWFI13 44349291 IC50 = 564 nM T59102 C18OEK 44349292 IC50 = 50 nM T59102 C8XZ0Q 44349293 IC50 = 292 nM T59102 CYV2D7 44368815 IC50 = 357 nM T59102 CG6NE0 44394479 IC50 = 450 nM T59102 C6QL8A 44394480 IC50 = 970 nM T59102 C1BQ6T 44394484 IC50 = 240 nM T59102 CZ10CS 44394568 IC50 = 3590 nM T59102 CUF85K 44394571 IC50 = 400 nM T59102 CHO52Q 44394593 IC50 = 1010 nM T59102 CHCY97 44394612 IC50 = 2930 nM T59102 C7AB5H 44394617 IC50 = 350 nM T59102 C8M2PH 44394619 IC50 = 90 nM T59102 C58FRU 44394632 IC50 = 460 nM T59102 CB5S0R 44394633 IC50 = 220 nM T59102 CGLU71 44394634 IC50 = 10 nM T59102 CDU4J7 44394635 IC50 = 10 nM T59102 C4ZS5C 44394664 IC50 = 1150 nM T59102 C4ADU7 44394665 IC50 = 1400 nM T59102 C79BHS 44394670 IC50 = 180 nM T59102 CM0GF2 44394673 IC50 = 920 nM T59102 CF31RW 44394679 IC50 = 5 nM T59102 C53PUJ 44394680 IC50 = 280 nM T59102 C2JT4Q 44394704 IC50 = 770 nM T59102 C15GEC 44394709 IC50 = 1060 nM T59102 C6AEU0 44394722 IC50 = 5 nM T59102 C1GNQ7 44394737 IC50 = 4090 nM T59102 C2OAX3 44394745 IC50 = 510 nM T59102 C9RBN1 44394760 IC50 = 20 nM T59102 C6SRC1 44394772 IC50 = 1540 nM T59102 C70JWY 44394773 IC50 = 430 nM T59102 CPT6I0 44394781 IC50 = 3760 nM T59102 CLDS93 44394803 IC50 = 420 nM T59102 C81CTG 44394822 IC50 = 70 nM T59102 CRA0U1 44394842 IC50 = 2000 nM T59102 C0O8HG 44394845 IC50 = 630 nM T59102 C5PD3W 44394846 IC50 = 3090 nM T59102 C97CVT 44394847 IC50 = 100 nM T59102 CLT7U8 44394848 IC50 = 550 nM T59102 CD4U9G 44394849 IC50 = 590 nM T59102 CH8D0U 44394850 IC50 = 3420 nM T59102 CGOD34 44394853 IC50 = 2370 nM T59102 C6QNI1 44394865 IC50 = 80 nM T59102 CE8HO9 44394869 IC50 = 60 nM T59102 C43HND 44394870 IC50 = 100 nM T59102 C1L0SE 44394874 IC50 = 31700 nM T59102 CSE64J 44394875 IC50 = 370 nM T59102 C0XSD5 44394876 IC50 = 800 nM T59102 CW1QA3 44394898 IC50 = 13400 nM T59102 CFC1S9 44394899 IC50 = 160 nM T59102 C6GFO1 44394903 IC50 = 2130 nM T59102 CARP42 44394904 IC50 = 5190 nM T59102 CCT0R3 44394905 IC50 = 100 nM T59102 C8VJ2E 44405089 IC50 = 17 nM T59102 C8K4AL 44407237 IC50 > 50000 nM T59102 CUA18B 44407238 IC50 = 7600 nM T59102 C04HFE 44407248 IC50 > 50000 nM T59102 CR3O1C 44407275 IC50 = 15900 nM T59102 C70BFV 44407276 IC50 = 10200 nM T59102 CMH7W6 44407277 IC50 = 8700 nM T59102 C8W5YG 44447872 IC50 = 6 nM T59102 CUB12D 44449577 IC50 = 389 nM T59102 C3ZBV8 44450546 IC50 = 920 nM T59102 CLK0W7 44453682 IC50 > 1000 nM T59102 C0LY6E 44552561 IC50 = 6100 nM T59102 C7KRU3 44552562 EC50 = 2000 nM T59102 CYV71I 44555430 IC50 = 12.3 nM T59102 CJ1X9V 44565013 IC50 > 10000 nM T59102 CN2Q3D 44565014 IC50 = 1100 nM T59102 CM2GN3 44565015 IC50 > 10000 nM T59102 CV91YE 44572385 IC50 = 2600 nM T59102 C3CB2K 44572429 IC50 = 7800 nM T59102 CM2Q8J 44572430 IC50 = 5200 nM T59102 CAN4B0 44572431 IC50 = 1100 nM T59102 CMAT21 44572489 IC50 = 71000 nM T59102 CU1SY9 44572490 IC50 = 8700 nM T59102 CSD74G 44572491 IC50 = 13000 nM T59102 CA9WO3 44572537 IC50 = 47000 nM T59102 C06SLW 44572538 IC50 = 28000 nM T59102 CY8TG3 44572539 IC50 = 11000 nM T59102 C1JR4C 44572540 IC50 = 40000 nM T59102 CZ0PA9 44572581 IC50 = 2100 nM T59102 CD9VR5 44572582 IC50 = 13000 nM T59102 CG5UK0 44572584 IC50 = 11000 nM T59102 CMX32U 44572633 IC50 = 6200 nM T59102 C5WOE2 44586449 IC50 = 11800 nM T59102 C0VF8M 44586450 IC50 > 50000 nM T59102 C4K7NP 44586451 IC50 > 50000 nM T59102 C1JNR5 44586452 IC50 = 13700 nM T59102 C6T8UP 44586490 IC50 > 500000 nM T59102 CU95NI 44586526 IC50 = 100400 nM T59102 CBK9R3 44586527 IC50 > 500000 nM T59102 CA18IW 44586528 IC50 > 500000 nM T59102 C0YSZ2 44586577 IC50 = 77400 nM T59102 C8M5KI 44611919 IC50 = 22.8 nM T59102 C4KWJ3 45379956 IC50 > 50000 nM T59102 C2CU0B 45380067 IC50 > 50000 nM T59102 C6E2SC 45482700 IC50 > 10000 nM T59102 CZXH74 45482750 IC50 > 10000 nM T59102 CNI92D 46182735 IC50 = 230 nM T59102 CUA97D 46209401 IC50 = 120 nM T59102 C8YPN0 46225596 IC50 > 10000 nM T59102 C34JTS 46225597 IC50 = 5100 nM T59102 CGD73B 46225598 IC50 = 9100 nM T59102 C3E0PU 46225599 IC50 = 10000 nM T59102 CRDY89 46225610 IC50 = 3600 nM T59102 C0JMT8 46225611 IC50 > 10000 nM T59102 CF0D5J 46225612 IC50 = 1400 nM T59102 CFVO38 46225632 IC50 = 8700 nM T59102 CLZ1O6 46225634 IC50 = 4400 nM T59102 C07VDX 46225635 IC50 = 3800 nM T59102 CT70DX 46225640 IC50 = 7900 nM T59102 CJUF68 46225641 IC50 = 7700 nM T59102 C6AJ5N 46225647 IC50 = 3400 nM T59102 C2WCV1 46225648 IC50 = 9900 nM T59102 CBS96A 46225649 IC50 > 10000 nM T59102 C38BFC 46225657 IC50 = 2100 nM T59102 CD0A6F 46225658 IC50 > 10000 nM T59102 C1B3KS 46225663 IC50 = 2100 nM T59102 CU46XI 46225664 IC50 = 8000 nM T59102 CO3HS2 46225665 IC50 > 10000 nM T59102 C2UV1S 46225666 IC50 = 8200 nM T59102 CX5B1G 46225667 IC50 = 9200 nM T59102 C2Q9OH 46225668 IC50 > 10000 nM T59102 CM14FH 46225680 IC50 > 10000 nM T59102 CQS96E 46225681 IC50 > 10000 nM T59102 CJIK35 46225682 IC50 = 3800 nM T59102 C8S4QA 46225688 IC50 = 6700 nM T59102 C2P9QO 46228508 IC50 = 1550 nM T59102 C6E5PY 46228822 IC50 = 7490 nM T59102 C3T8AM 46228951 IC50 = 2390 nM T59102 CYZV41 46231219 IC50 = 2667 nM T59102 C7J5UP 46231220 IC50 = 858 nM T59102 CC96GZ 46231221 IC50 = 900 nM T59102 C9H4YO 46233889 IC50 = 49 nM T59102 CRT34L 46235770 IC50 = 27 nM T59102 CFR1C6 46845026 IC50 > 300000 nM T59102 C7NUY3 46847552 IC50 > 1000 nM T59102 CE3WH9 46865125 IC50 > 200000 nM T59102 C45LYT 46865445 IC50 > 200000 nM T59102 C1XEY4 46866615 IC50 > 200000 nM T59102 CF6K3E 46866616 IC50 > 200000 nM T59102 CA57MX 46886970 IC50 = 24600 nM T59102 CRGH62 46886971 IC50 = 183100 nM T59102 C68AGR 46886972 IC50 > 300000 nM T59102 CP32GW 46886973 IC50 > 300000 nM T59102 C48JWD 46886974 IC50 > 300000 nM T59102 C7H3MD 46887038 IC50 = 174900 nM T59102 C40NOR 46887039 IC50 = 43000 nM T59102 C7I4SB 46887074 IC50 = 182000 nM T59102 CI5QX2 46887110 IC50 = 171300 nM T59102 C0Q7NG 46887111 IC50 = 220400 nM T59102 CU15AN 46887112 IC50 = 110100 nM T59102 CD90BV 46887113 IC50 = 142200 nM T59102 CH3O9K 46887255 IC50 = 8500 nM T59102 C7NUT3 46887298 IC50 > 500000 nM T59102 CWV65D 46887299 IC50 > 500000 nM T59102 CH5BZ6 46887300 IC50 = 192400 nM T59102 C20UCB 46887348 IC50 > 500000 nM T59102 C0KEG5 46887349 IC50 > 500000 nM T59102 CY59RB 46887397 IC50 = 104200 nM T59102 C0WYM1 46898022 IC50 = 10000 nM T59102 CB92VU 46912443 IC50 = 2800 nM T59102 CU6HC7 46912444 IC50 = 34800 nM T59102 C8A4KU 46912445 IC50 > 500000 nM T59102 CNOS56 46912446 IC50 = 1300 nM T59102 CV38NE 46912546 IC50 > 500000 nM T59102 CQLT07 46913878 IC50 < 1000 nM T59102 CHSF07 49806372 IC50 > 1000 nM T59102 CVS85M 49831162 IC50 = 58 nM T59102 CR58WT 49840391 IC50 = 3 nM T59102 CA2J6U 49840467 IC50 = 13 nM T59102 CB0S2P 49842666 IC50 = 9200 nM T59102 C0NA9U 49842670 IC50 > 100000 nM T59102 CAI20B 49842778 IC50 = 21000 nM T59102 CRA74I 49842779 IC50 = 42000 nM T59102 CF91RS 49843531 IC50 > 10000 nM T59102 CE7D2J 49855568 IC50 = 3300 nM T59102 CFD9P3 49855569 IC50 = 1100 nM T59102 C1AU5N 49855758 IC50 = 2300 nM T59102 CIFK93 49855759 IC50 = 4000 nM T59102 CK48OJ 49855760 IC50 = 2300 nM T59102 CZI3M1 49855761 IC50 = 3900 nM T59102 CRPZ58 49855949 IC50 = 2500 nM T59102 CTU0K3 49855950 IC50 = 2700 nM T59102 CF85NL 49855951 IC50 = 4700 nM T59102 CF7YS9 49855952 IC50 = 1000 nM T59102 CJU38G 49855953 IC50 = 1800 nM T59102 CD2K4R 50908681 Ki > 1000000 nM T59102 C2Y6QS 50938552 IC50 > 10000 nM T59102 C9NYP4 51036677 IC50 > 10000 nM T59102 C4WRY3 51037112 IC50 > 10000 nM T59102 CRI28Z 51037948 IC50 > 10000 nM T59102 C4R7IM 52941368 IC50 = 71700 nM T59102 C7BY6M 52942956 IC50 > 200000 nM T59102 CA62KU 52944152 IC50 = 88200 nM T59102 CQV34K 52945403 IC50 > 200000 nM T59102 C97XZA 52946619 IC50 > 200000 nM T59102 CE0X5U 52947574 IC50 = 348000 nM T59102 CD9S4I 52947801 IC50 > 200000 nM T59102 CA6IL3 52947802 IC50 > 200000 nM T59102 C2KAJ4 52948634 IC50 > 500000 nM T59102 C0A1GQ 52949915 IC50 > 500000 nM T59102 C09SDH 53257410 IC50 > 10000 nM T59102 CZY0J7 53323592 IC50 > 100000 nM T59102 CNPM14 53341082 IC50 > 3000 nM T59102 C0SWH5 53348216 IC50 > 40000 nM T59102 CBK9Q6 53357848 IC50 > 10000 nM T59102 C8NA4L 53384644 IC50 > 30000 nM T59102 CVG90B 53389651 IC50 > 10000 nM T59102 C0JMY7 54673975 IC50 = 50500 nM T59102 C8AB1J 54759606 Ki = 19 nM T59102 CQ17GA 56640518 IC50 > 200000 nM T59102 CG20VK 56640520 IC50 > 200000 nM T59102 CZ9C8M 56640588 IC50 > 200000 nM T59102 CH0D7P 56640590 IC50 > 200000 nM T59102 C9DX3J 56649281 IC50 = 26 nM T59102 CR50TJ 56835147 IC50 = 2788 nM T59102 CI5ZJ7 56835161 IC50 > 100000 nM T59102 C2ML5S 56837168 IC50 = 518 nM T59102 CCW89V 56932477 IC50 = 185 nM T59102 CR3FK5 56932525 IC50 = 8 nM T59102 CY36EG 56945171 IC50 = 49 nM T59102 C4OG7H 56945172 IC50 = 93 nM T59102 CH0QA3 56945173 IC50 = 190 nM T59102 CM0NQ5 56945174 IC50 = 1100 nM T59102 CXKF03 56945175 IC50 = 550 nM T59102 CE07AQ 56945176 IC50 = 1600 nM T59102 CU86KC 56945272 IC50 = 23 nM T59102 C9SX7F 56945273 IC50 = 27 nM T59102 CG7VH5 56945274 IC50 = 72 nM T59102 C6WU4V 56945277 IC50 = 19 nM T59102 C7U9SL 56951304 IC50 > 50000 nM T59102 C0GQ9I 56951305 IC50 > 300000 nM T59102 C5YT6A 56951306 IC50 = 8920 nM T59102 CB03EH 56951307 IC50 = 193200 nM T59102 CP58NG 56954518 IC50 = 5 nM T59102 CAK91L 56955954 IC50 > 3600 nM T59102 C4YFJ5 57384105 IC50 = 1500 nM T59102 CV9RW5 57384106 IC50 = 1800 nM T59102 C4WE9B 57391179 IC50 = 10 nM T59102 CY10TP 57391180 IC50 = 6 nM T59102 CR4T2Y 57391283 IC50 = 129100 nM T59102 CU3DM9 57391295 IC50 > 1000 nM T59102 CBL74E 57392425 IC50 = 44300 nM T59102 CU7J9C 57393063 IC50 = 2 nM T59102 CD4HS3 57393074 IC50 = 9 nM T59102 CS60KL 57393075 IC50 > 2000 nM T59102 CWMT98 57394785 IC50 > 1000 nM T59102 CG18LI 57394786 IC50 = 34200 nM T59102 CEDP89 57394787 IC50 = 129300 nM T59102 C9PY4Q 57394798 IC50 = 10 nM T59102 C3F9VS 57394799 IC50 = 700 nM T59102 CP6W4C 57394879 IC50 > 500000 nM T59102 CVR13L 57394880 IC50 > 500000 nM T59102 CA4Q3Y 57395925 IC50 = 145900 nM T59102 C4CN6V 57396453 IC50 = 10 nM T59102 CCT58R 57396454 IC50 > 200 nM T59102 CXA5Z9 57396541 IC50 = 2 nM T59102 CPAH35 57396542 IC50 = 4 nM T59102 CUGP85 57396545 IC50 = 212400 nM T59102 CY8U1Q 57396557 IC50 = 0.9 nM T59102 CBUP96 57396646 IC50 = 159600 nM T59102 CWV96N 57398329 IC50 = 3 nM T59102 C8K1WJ 57398330 IC50 = 0.3 nM T59102 CXJ68F 57398331 IC50 = 229600 nM T59102 CBK02S 57399984 IC50 = 1 nM T59102 CNU4I7 57399985 IC50 = 2 nM T59102 CD9KF3 57399986 IC50 = 2 nM T59102 C0BA7P 57401686 IC50 = 20 nM T59102 CH56JP 57401785 IC50 = 3 nM T59102 C7YMG1 57401804 IC50 = 300 nM T59102 C20ZAX 57401805 IC50 = 4 nM T59102 C15YQW 57401806 IC50 = 20 nM T59102 CY5TJ9 57401807 IC50 = 4 nM T59102 C4L0SA 57401808 IC50 = 0.4 nM T59102 C4J0OD 57403506 IC50 = 0.8 nM T59102 CN0M3Z 57403518 IC50 = 300 nM T59102 CZSM95 57412684 IC50 > 10000 nM T59102 CN53XW 57428969 IC50 = 57.3 nM T59102 CE59QS 57505507 IC50 = 5.5 nM T59102 C8P6RD 57505528 IC50 = 15 nM T59102 C8R4FE 57991377 IC50 = 125.4 nM T59102 CH7L5N 58172700 IC50 = 768.4 nM T59102 C4V7FY 58191950 IC50 = 16000 nM T59102 CPCA29 58191961 IC50 = 70000 nM T59102 C7HF1L 58191965 IC50 = 7200 nM T59102 C8LWY9 58191997 IC50 = 28000 nM T59102 C4IBV1 59375998 IC50 = 12.7 nM T59102 CV8Q2D 59376002 IC50 = 89.9 nM T59102 CL3ND8 59376009 IC50 = 7.6 nM T59102 CC2AF9 59376012 IC50 = 19.4 nM T59102 CR7CG3 59376014 IC50 = 22.7 nM T59102 C60RIS 59376021 IC50 = 41.6 nM T59102 CT3Q5G 59376025 IC50 = 21.3 nM T59102 C97YSI 59376026 IC50 = 64.8 nM T59102 CEH5X6 59376027 IC50 = 40.1 nM T59102 C79EBT 59376032 IC50 = 40.7 nM T59102 C06DNI 59376037 IC50 = 12.1 nM T59102 C0XM7N 59376046 IC50 = 118.4 nM T59102 C70WCP 59376053 IC50 = 15.6 nM T59102 C5IHG9 59376058 IC50 = 18 nM T59102 CTK90V 59376059 IC50 = 260.3 nM T59102 C7ZY5I 59376061 IC50 = 101.4 nM T59102 CFT69X 59376062 IC50 = 70.3 nM T59102 C7D0BF 59376072 IC50 = 13.2 nM T59102 CD0RP7 59376074 IC50 = 62.1 nM T59102 C3HXC7 59376075 IC50 = 19.3 nM T59102 CAY6H8 59376079 IC50 = 13.3 nM T59102 CCX2W0 59376082 IC50 = 160.6 nM T59102 CLH49Z 59790029 IC50 = 1 nM T59102 C9QRX3 60098131 IC50 = 310 nM T59102 CSZA16 60155724 IC50 > 3600 nM T59102 CU79HD 60202383 IC50 = 243 nM T59102 C9ZCT2 62705065 IC50 > 1000 nM T59102 CK6WO0 66552478 IC50 < 10000 nM T59102 C37NKO 67129970 IC50 > 10000 nM T59102 CK80LJ 67130050 IC50 > 10000 nM T59102 CA63QI 67219716 IC50 > 5000 nM T59102 CV63UL 67240318 IC50 > 10000 nM T59102 C7GRV2 68755406 IC50 > 10000 nM T59102 CCS20X 69063773 IC50 = 3 nM T59102 CEB12M 70681395 IC50 = 3 nM T59102 CH27DE 70681409 IC50 = 2 nM T59102 CN29RI 70681410 IC50 = 5 nM T59102 CG93IE 70683519 IC50 = 0.3 nM T59102 CXSN14 70685622 IC50 = 6 nM T59102 CL24MP 70687766 IC50 = 0.2 nM T59102 C51DHN 70689791 IC50 = 3 nM T59102 C6ITV3 70689792 IC50 = 0.9 nM T59102 CMLY63 70689816 IC50 = 0.5 nM T59102 C08ASR 70689830 IC50 = 4 nM T59102 C4TF3G 70691955 IC50 = 5 nM T59102 CTWD94 70691956 IC50 = 50 nM T59102 CIK5N2 70691957 IC50 = 10 nM T59102 C8RZP3 70691958 IC50 = 5 nM T59102 C0XRC9 70691981 IC50 = 3 nM T59102 C9RT8C 70693982 IC50 = 0.7 nM T59102 C2X1KJ 70694006 IC50 = 0.4 nM T59102 C54VLD 70694007 IC50 = 0.2 nM T59102 C6O3SM 70696108 IC50 = 50 nM T59102 CEBO91 71452977 IC50 > 10000 nM T59102 C9DIK2 71512060 IC50 = 2102 nM T59102 C6HF8S 71521082 IC50 = 35400 nM T59102 C9Z3AI 71521083 IC50 > 5000 nM T59102 C5OBF0 71525245 IC50 > 500000 nM T59102 CJX73B 71525246 IC50 > 500000 nM T59102 CCN90I 71525247 IC50 = 331500 nM T59102 CY6JA9 71525248 IC50 > 500000 nM T59102 CGQJ60 71525249 IC50 > 500000 nM T59102 CMKD15 71525283 IC50 = 89700 nM T59102 C3OJ6R 71525284 IC50 > 500000 nM T59102 CP5Q2U 71525285 IC50 = 430100 nM T59102 CZ8N0J 71525286 IC50 > 500000 nM T59102 CG31MI 71525287 IC50 > 500000 nM T59102 CRX81Q 71575642 IC50 = 408 nM T59102 CGK76E 71583411 IC50 > 200000 nM T59102 CB5WX0 71583412 IC50 > 200000 nM T59102 CI8K3T 71583527 IC50 = 196200 nM T59102 C6FGI0 71583528 IC50 > 200000 nM T59102 C3QGE7 71583529 IC50 = 172200 nM T59102 CS9HX7 71583530 IC50 = 70600 nM T59102 CQTZ32 71583531 IC50 > 200000 nM T59102 C0G5RS 71583532 IC50 > 200000 nM T59102 CVEY46 71583533 IC50 = 170800 nM T59102 CX6TR7 71583634 IC50 > 200000 nM T59102 CR15QP 71583635 IC50 = 196200 nM T59102 CZ31PU 71583657 IC50 > 10000 nM T59102 CU1IL6 71741204 IC50 > 100000 nM T59102 CN1GA3 71741327 IC50 > 100000 nM T59102 COS5D7 71741328 IC50 > 100000 nM T59102 C8PWZ0 71741329 IC50 > 100000 nM T59102 CT4XR9 71741332 IC50 > 50000 nM T59102 C4Q6FE 71815105 IC50 = 86.9 nM T59102 CJ9OX6 71815106 IC50 = 176.7 nM T59102 CCKL45 72191698 IC50 = 395.7 nM T59102 C60TUV 72737208 IC50 > 10000 nM T59102 CJ3WA6 72737404 IC50 > 10000 nM T59102 C8SIL6 73349435 IC50 = 1.42 nM T59102 CVNW01 73386831 IC50 > 1000 nM T59102 C2PAK9 73438493 IC50 = 1055 nM T59102 CBAT06 76071144 IC50 = 1083 nM T59102 CH8W7D 77461036 IC50 > 1000 nM T59102 CA65HB 78319164 IC50 = 20 nM T59102 CCJ43A 86302281 IC50 > 10000 nM T59102 CB5NJ4 86302541 IC50 = 4.6 nM T59102 CPG3A5 86302574 IC50 > 30000 nM T59102 C08WGI 86566799 IC50 = 16.3 nM T59102 C5S3YB 90645165 IC50 = 92.3 nM T59102 C6Q4DH 90645475 IC50 = 29.9 nM T59102 C89HTB 90645476 IC50 = 56.5 nM T59102 C9ASG1 90645478 IC50 = 27.1 nM T59102 COY53U 90645479 IC50 = 16.2 nM T59102 C48OSQ 90645480 IC50 = 23.1 nM T59102 CL8GW5 90645481 IC50 = 66.1 nM T59102 CL7SC6 90645482 IC50 = 28.3 nM T59102 CI3OD6 90645484 IC50 = 63.5 nM T59102 CX29IY 90655145 IC50 > 10000 nM T59102 C96DTL 90682879 IC50 = 21.9 nM T59102 CI97DL 102431709 IC50 = 19000 nM T59102 C09MIG 102431710 IC50 = 1500 nM T59102 C5HRO7 102431711 IC50 = 1400 nM T59102 CTGP06 117996541 IC50 > 10000 nM T59102 CY7BI2 118706214 IC50 > 10000 nM T59102 C2IN3C 118710236 IC50 = 8.1 nM T59102 CF2YR1 118710237 IC50 = 1.54 nM T59102 C4AHL2 118711367 IC50 = 5800 nM T59102 C46QUT 118717614 IC50 > 200000 nM T59102 CJC34Y 118717615 IC50 > 200000 nM T59102 CFEP93 118717616 IC50 > 200000 nM T59102 CEC4H0 118717617 IC50 > 200000 nM T59102 CU2TG3 118717618 IC50 > 200000 nM T59102 C5OL0W 118717619 IC50 > 200000 nM T59102 C3KLI5 118723185 IC50 = 500 nM T59102 C5UZ9X 118723186 IC50 = 4000 nM T59102 C3XV6L 118723187 IC50 > 100000 nM T59102 CLD41J 118723188 IC50 > 100000 nM T59102 C0H9YD 118723189 IC50 = 5000 nM T59102 CP8FW0 118723190 IC50 = 13000 nM T59102 CCV0H1 118723191 IC50 = 13000 nM T59102 C1J7QE 118723192 IC50 = 12000 nM T59102 CMHV05 118723193 IC50 = 32000 nM T59102 CRQY80 118723194 IC50 = 300 nM T59102 CVZM84 118723195 IC50 = 1000 nM T59102 CP8Z6I 118723196 IC50 = 14000 nM T59102 CI6HB3 118723197 IC50 = 56000 nM T59102 CVGE25 118723198 IC50 = 2000 nM T59102 C78BAF 118723199 IC50 = 9000 nM T59102 C02HAD 118723200 IC50 = 3000 nM T59102 CDAN63 118723201 IC50 = 26000 nM T59102 CL6T5K 118723202 IC50 = 1000 nM T59102 CDQ92V 118723203 IC50 = 8000 nM T59102 CV0B6M 118723204 IC50 = 2000 nM T59102 CX4E1N 118723205 IC50 = 1000 nM T59102 C8BU5O 118723206 IC50 = 2000 nM T59102 C2G1TN 118723207 IC50 = 7000 nM T59102 C1JO0D 118723208 IC50 = 22000 nM T59102 CYXF26 118723209 IC50 = 31000 nM T59102 C7JYP8 118723210 IC50 = 800 nM T59102 CV6HJ8 118723211 IC50 = 5000 nM T59102 CI6QA2 118723212 IC50 = 100 nM T59102 C3XKJ9 118723213 IC50 = 2000 nM T59102 CU1B5W 118723214 IC50 = 19000 nM T59102 CD5HK1 118723215 IC50 = 8000 nM T59102 CU06YS 118723216 IC50 > 100000 nM T59102 CWYF91 118729842 IC50 = 40.4 nM T59102 CR54XL 118729843 IC50 = 66.1 nM T59102 CF3X9J 118729844 IC50 = 166.3 nM T59102 CT3Q6C 118729845 IC50 = 50.1 nM T59102 C1QWK6 118729846 IC50 = 24.6 nM T59102 CWUA61 118729847 IC50 = 25 nM T59102 C63CDP 118729848 IC50 = 73.2 nM T59102 C1WB7L 118729849 IC50 = 198 nM T59102 C8A7ZT 118729850 IC50 = 58.2 nM T59102 C9WDF4 118729851 IC50 = 84 nM T59102 CT08EZ 118729852 IC50 = 132 nM T59102 C08KEM 122179540 IC50 = 2000 nM T59102 CG0RP7 122179547 IC50 = 2200 nM T59102 C1A0SQ 122179548 IC50 = 4600 nM T59102 C4X7SD 122192466 IC50 = 1982 nM T59102 CNX0Q2 122193763 IC50 = 850 nM T59102 CWV0C3 122193764 IC50 = 2120 nM T59102 CSG98Y 122193765 IC50 = 2820 nM T59102 CCLQ75 122193769 IC50 = 320 nM T59102 CXDR48 122193770 IC50 = 570 nM T59102 CPA8C5 122193773 IC50 = 2300 nM T59102 CY30FL 123752658 IC50 = 5.5 nM T59102 C8KXV1 127025843 IC50 > 1000 nM T59102 C1XD6R 127029809 IC50 = 526.5 nM T59102 CI1E5W 127029864 IC50 = 4.57 nM T59102 CKS28E 127034802 IC50 = 64.2 nM T59102 CKX40V 127037812 IC50 = 223.9 nM T59102 C70RUP 127038480 IC50 > 10000 nM T59102 C3WCN8 127041777 IC50 > 10000 nM T59102 CC58IQ 127043948 IC50 = 120 nM T59102 CHK16Q 127045929 IC50 > 1000 nM T59102 CY3J0C 127047591 IC50 > 1000 nM T59102 CF5D2Y 129318936 IC50 = 6115 nM T59102 C0FM1R 130196825 IC50 = 392 nM T59102 CUO0C5 132156633 IC50 > 10000 nM T59102 C6OMB1 132204257 IC50 = 606 nM T59102 C6ROQ3 132546210 IC50 = 80 nM T59102 CJ04HZ 132585195 IC50 < 1 nM T59102 CERS64 132937256 IC50 = 26197 nM T59102 CN9SD7 132942957 IC50 = 51.4 nM T59102 CMP2S9 132942958 IC50 = 62.2 nM T59102 CN35SO 134146628 IC50 > 1000 nM T59102 CIK38Q 134229735 IC50 = 63.4 nM T59102 CYL5V1 134694986 IC50 > 30000 nM T59102 CLCO61 135398510 EC50 = 51 nM T59102 CN5T7W 135400982 IC50 = 12 nM T59102 CVJ07T 135402853 IC50 = 70 nM T59102 CBK6I2 135407156 IC50 = 30 nM T59102 CMVS34 135410282 IC50 = 10 nM T59102 CUT52Q 135421574 IC50 = 19000 nM T59102 CK9D4A 135428921 IC50 = 4500 nM T59102 C8X5SV 135433815 IC50 = 20 nM T59102 CNZ04G 135453357 IC50 = 4 nM T59102 CS63IO 135476717 IC50 = 65 nM T59102 C2MAC7 135536640 IC50 > 100000 nM T59102 CW08GF 135674125 IC50 = 70 nM T59102 CLS64T 135674129 IC50 = 0.9 nM T59102 C54ABM 135674133 IC50 = 0.3 nM T59102 CM7YH4 135674136 IC50 = 5 nM T59102 C1WSO7 135674140 IC50 = 130 nM T59102 CA0Y7V 135674142 IC50 = 5 nM T59102 CM90FP 135674144 IC50 = 0.9 nM T59102 C3CP1X 135674147 IC50 = 0.3 nM T59102 CBSV42 135674149 IC50 = 5 nM T59102 C1NTB0 135674153 IC50 = 2 nM T59102 CID0W9 135674167 IC50 = 0.1 nM T59102 C1DL9J 135674173 IC50 = 30 nM T59102 CO89UX 135674193 IC50 = 8 nM T59102 C2H3XB 135926086 IC50 = 2 nM T59102 C7BES6 135926087 IC50 = 2 nM T59102 CNTK81 135926088 IC50 = 7 nM T59102 CQ64OH 135926089 IC50 = 39 nM T59102 CXG7O4 135926090 IC50 = 0.1 nM T59102 CN4FG3 135926091 IC50 = 14 nM T59102 C7NZU3 135926094 IC50 > 25000 nM T59102 CL6HQ4 135926104 IC50 = 1 nM T59102 CE37KQ 135926113 IC50 = 0.7 nM T59102 C1ZRT7 135926114 IC50 = 1 nM T59102 CU5W2V 135926115 IC50 = 7 nM T59102 C1D3EW 135926116 IC50 = 0.6 nM T59102 C2PAV1 135971426 IC50 = 10000 nM T59102 CHA4N2 136013680 IC50 > 10 nM T59102 CLN6Y8 136026516 IC50 > 100000 nM T59102 CG1R7B 136087060 IC50 = 7000 nM T59102 C5QZ4H 136126664 IC50 = 1100 nM T59102 CB8RX0 136126665 IC50 = 0.2 nM T59102 CZ7EX0 136183413 IC50 = 3200 nM T59102 CDT7E4 136211077 IC50 > 1000 nM T59102 C9RE8D 136215817 IC50 = 530.6 nM T59102 C1YUD0 136219394 IC50 > 10 nM T59102 CIU8W3 136254389 IC50 > 10 nM T59102 C35MBU 136299423 IC50 = 45 nM T59102 C0W8KA 136299435 IC50 = 4.3 nM T59102 C5G4ES 136299436 IC50 = 3.2 nM T59102 C83OXU 137007054 IC50 = 12000 nM T59102 CCM42D 137249694 IC50 = 14.3 nM T59102 C25ERN 137631967 IC50 = 1 nM T59102 CFUY16 137633842 IC50 > 200000 nM T59102 CNX0F9 137634126 IC50 = 106.2 nM T59102 CHC70D 137634143 IC50 = 3.26 nM T59102 CI1E8V 137634241 IC50 = 5190 nM T59102 C85WBP 137634338 IC50 = 9 nM T59102 CAD3C5 137634686 IC50 = 45.52 nM T59102 CS23KQ 137635618 IC50 = 90100 nM T59102 C5JD9N 137635898 IC50 = 10.3 nM T59102 CK5Y3P 137635915 IC50 = 65.24 nM T59102 C06JRX 137637094 IC50 > 10 nM T59102 CU24QC 137638448 IC50 = 90.3 nM T59102 CO9D4W 137639407 IC50 = 31.36 nM T59102 C3UBE2 137639638 IC50 > 200 nM T59102 CU8YX6 137643005 IC50 = 58200 nM T59102 C2T6FV 137644825 IC50 = 29.79 nM T59102 C1DK0P 137651391 IC50 = 1 nM T59102 C5F3LP 137651946 IC50 = 83.17 nM T59102 CQUY83 137652218 IC50 > 200000 nM T59102 C9JT1N 137655519 IC50 = 60500 nM T59102 C9TEU1 137655771 IC50 = 27.11 nM T59102 CKVO51 137657233 IC50 = 30.2 nM T59102 CV5H3Z 137657932 IC50 > 100 nM T59102 CQMB10 137658515 IC50 = 197 nM T59102 C7IVT9 137658762 IC50 > 200 nM T59102 CQE9M4 137661156 IC50 = 67.85 nM T59102 CM0N3T 137661420 IC50 = 7.2 nM T59102 CT43IF 137661858 IC50 = 8.1 nM T59102 CIWG23 138393067 IC50 = 88 nM T59102 C07EKN 138454794 IC50 = 2075 nM T59102 C5LQU9 138479230 IC50 = 673.6 nM T59102 CSRI06 138547901 IC50 > 1000 nM T59102 CUXO19 138617501 IC50 > 1000 nM T59102 C6AK0N 139030518 IC50 = 97 nM T59102 C34CKN 141523354 IC50 = 19.46 nM T59102 CB3Z1W 145949428 IC50 = 180 nM T59102 CCM27G 145949662 IC50 = 64.6 nM T59102 CVJS01 145949677 IC50 = 12 nM T59102 CWQA26 145949916 IC50 = 34.3 nM T59102 CYF32C 145950953 IC50 = 15 nM T59102 CRXJ25 145951211 IC50 = 91 nM T59102 C4LBC0 145951650 IC50 = 116.2 nM T59102 CR9LH4 145952520 IC50 = 92.7 nM T59102 CC72WG 145953067 IC50 = 7800 nM T59102 C60XZR 145953297 IC50 = 19 nM T59102 CSLC73 145953358 IC50 = 44.2 nM T59102 CAL30B 145953560 IC50 = 15 nM T59102 C0V8SM 145954139 IC50 = 25 nM T59102 CDRQ06 145955547 IC50 = 45.5 nM T59102 C8VN1Y 145955561 IC50 = 27 nM T59102 C2O9XD 145955651 IC50 = 91.7 nM T59102 C1IX5N 145956333 IC50 = 22 nM T59102 C6ZNJ1 145956488 IC50 = 34 nM T59102 CLZH04 145956490 IC50 = 39 nM T59102 C5VSC7 145956704 IC50 = 177 nM T59102 CY69RH 145956768 IC50 = 49.2 nM T59102 CIW0V9 145956964 IC50 = 241.6 nM T59102 CB74GR 145957221 IC50 = 24 nM T59102 CB1MI9 145957910 IC50 = 4.5 nM T59102 CS47UF 145958497 IC50 = 14 nM T59102 CRVO52 145960991 IC50 > 500 nM T59102 CV4M1Z 145961849 IC50 = 60.7 nM T59102 C9PKU6 145963750 IC50 = 5.3 nM T59102 CTUF34 145966712 IC50 = 111 nM T59102 C4OD9Q 145967187 IC50 = 214.5 nM T59102 CNVT54 145971746 IC50 = 61 nM T59102 C3Q4XM 145972183 IC50 = 13 nM T59102 C71ZJX 145972445 IC50 = 135.1 nM T59102 CG8R0P 145972697 IC50 = 1.5 nM T59102 C74TYP 145975351 IC50 = 482.1 nM T59102 CCS92I 145982511 IC50 = 510 nM T59102 CWE21T 145982588 IC50 = 3250 nM T59102 CC12YA 145982666 IC50 = 57.8 nM T59102 CF4BO8 145982785 IC50 = 28.9 nM T59102 CM6ZS7 145982824 IC50 = 63 nM T59102 CZ3CG9 145982825 IC50 = 1260 nM T59102 CF28AU 145983389 IC50 = 42.6 nM T59102 CRL19G 145983447 IC50 = 40 nM T59102 C48UZH 145983504 IC50 = 2230 nM T59102 C8BZC5 145983753 IC50 = 20 nM T59102 CD5L8O 145983778 IC50 > 200 nM T59102 CNK7I9 145984104 IC50 = 3520 nM T59102 C4C2OM 145984258 IC50 = 8 nM T59102 C9DHL3 145984282 IC50 = 3780 nM T59102 CVT02P 145984555 IC50 = 20 nM T59102 CHW8E5 145984671 IC50 = 1230 nM T59102 CYG42V 145984818 IC50 > 200 nM T59102 CFS7D5 145984941 IC50 > 200 nM T59102 C05IMJ 145984942 IC50 = 38.9 nM T59102 C9Q5VI 145985608 IC50 = 820 nM T59102 CA2TW8 145985737 IC50 = 290 nM T59102 CS9C8J 145986155 IC50 > 200 nM T59102 C1Y5MO 145987062 IC50 = 1.81 nM T59102 CI85EU 145998085 IC50 = 1013 nM T59102 C2MD1Q 155513187 IC50 > 10000 nM T59102 C86HPW 155518524 IC50 = 81000 nM T59102 CU6Z5O 155520650 IC50 = 150 nM T59102 CY6NE1 155523855 IC50 = 100 nM T59102 CRP7Q6 155525519 IC50 = 110 nM T59102 CTD5R7 155528337 IC50 = 450 nM T59102 CLEJ03 155529517 IC50 = 230 nM T59102 CS69CA 155532132 IC50 = 25.3 nM T59102 C3NZO0 155533789 IC50 = 90 nM T59102 C2DJ0A 155534253 IC50 = 2010 nM T59102 C37RFQ 155534994 IC50 = 1590 nM T59102 CE46SL 155540854 IC50 > 30000 nM T59102 C5O4JM 155540856 IC50 > 30000 nM T59102 C7SF2C 155547229 IC50 = 356 nM T59102 C6URZ7 155550475 IC50 = 1820 nM T59102 CGVU70 155554426 IC50 > 30000 nM T59102 CUA73V 155555832 IC50 = 330 nM T59102 C8L6PM 155561965 IC50 = 3790 nM T59102 C81JZW 155563388 IC50 = 390 nM T59102 CM23DI 155565660 IC50 = 1290 nM T59102 CK10HA 155568167 IC50 = 3640 nM T59102 CBWO68 49800164 IC50 = 28 nM T59102 D00ATA 5908088 IC50 = 12000 nM T59102 D00GVV 5329155 IC50 = 920 nM T59102 D02BXJ 46864270 IC50 = 2.6 nM T59102 D04FNY 25195216 IC50 = 40 nM T59102 D05NKG 16760286 IC50 = 316.23 nM T59102 D05WTI 11550535 IC50 = 317 nM T59102 D06QWO 14824655 IC50 > 10 ug.mL-1 T59102 D07IHM 9823787 IC50 > 10000 nM T59102 D07OSK 6419834 IC50 = 4000 nM T59102 D09HVH 135566652 IC50 > 10 nM T59102 D09LPL 5329103 IC50 = 3 nM T59102 D09QBA 23378546 IC50 > 10000 nM T59102 D09TNR 9850161 IC50 = 69 nM T59102 D0A1CM 5281855 IC50 = 1300 nM T59102 D0A4XJ 5289418 IC50 = 510 nM T59102 D0BW4G 10907042 IC50 = 130 nM T59102 D0C2GE 67161540 IC50 = 1.3 nM T59102 D0D6MH 11617559 IC50 > 10000 nM T59102 D0EE6A 6398883 IC50 = 640 nM T59102 D0G3SZ 6918469 IC50 = 5.9 ug.mL-1 T59102 D0H1OK 11562302 Ki = 2090 nM T59102 D0HE0E 5941540 IC50 = 5100 nM T59102 D0I3XZ 11601743 IC50 = 171 nM T59102 D0L3FK 5289419 IC50 > 10000 nM T59102 D0M4QA 56935577 IC50 = 10.1 nM T59102 D0R2WK 16038120 IC50 = 3220 nM T59102 D0U3WQ 9817165 IC50 = 90 nM T59102 D0UN9O 3385203 IC50 = 1000 nM T59102 D0X1RH 16051023 IC50 = 420 nM T59102 D0XS9E 5330535 IC50 = 90 nM T59102 D0YE1X 9927943 IC50 = 30 nM T59102 D0YZ7H 9797370 IC50 = 3 nM T59102 D0Z7TM 22273644 IC50 > 2000 nM T85272 D03DAP 3356 IC50 = 209000 nM T85272 D04OSE 4485 IC50 = 96000 nM T85272 D08YIN 1727 IC50 = 89000 nM T85272 D0OB1J 39186 IC50 = 144000 nM T85272 D0U5CE 1548943 IC50 = 29000 nM T85272 D0K9IF 71666749 IC50 > 30000 nM T85272 C29SPL 5867 EC50 = 33000 nM T85272 C6HA8E 5388709 IC50 > 30000 nM T85272 C8W2QA 6439099 IC50 > 30000 nM T85272 C8NM2I 11538313 EC50 = 7000 nM T85272 CA5W9R 11618060 EC50 = 1200 nM T85272 CLT3Z7 11695929 EC50 = 1700 nM T85272 CW9V0Y 13088125 EC50 = 6000 nM T85272 C8JA3E 13703975 EC50 = 4300 nM T85272 C91QFN 25019282 IC50 = 2660 nM T85272 CQSZ72 90675942 IC50 > 30000 nM T85272 CTBD74 90675943 IC50 > 30000 nM T85272 CM12LR 102597975 IC50 > 30000 nM T85272 CQJ49Y 122187245 IC50 = 0.0067 nM T85272 CSW57U 122187246 IC50 = 0.0077 nM T85272 C98BUE 122187247 IC50 = 0.0034 nM T85272 CVT7A6 122187248 IC50 = 0.0027 nM T85272 CI9ZH1 122187249 IC50 = 0.0078 nM T85272 CHJ75V 122187250 IC50 = 0.0095 nM T85272 C20TPX 122187251 IC50 = 0.0028 nM T85272 CQ17ZP 122187252 IC50 = 0.011 nM T85272 C2XUA5 122187253 IC50 = 0.308 nM T85272 CQTJ57 122187272 IC50 = 0.0078 nM T85272 CX2YG6 122187273 IC50 = 0.0181 nM T85272 C4CLN5 122187274 IC50 > 3.333 nM T85272 CF5M8V 122187275 IC50 = 0.49 nM T85272 C24MEW 122187276 IC50 > 3.333 nM T85272 CI7VL5 122187277 IC50 > 3.333 nM T85272 COX2P3 122187278 IC50 = 0.014 nM T85272 CY9RL0 122187279 IC50 = 0.02 nM T85272 CT5B4D 122187280 IC50 = 0.028 nM T85272 C42SZA 122187281 IC50 = 1.8 nM T85272 C6S3XG 122187282 IC50 = 0.0018 nM T85272 C0YG3Z 122187283 IC50 = 0.0057 nM T85272 C1F5PE 122187284 IC50 = 0.0023 nM T85272 C26VHJ 122187285 IC50 = 0.0049 nM T85272 C24JCI 122187286 IC50 = 0.0083 nM T85272 CW4SU9 122187287 IC50 = 0.001 nM T85272 CT0GS6 122187288 IC50 = 0.007 nM T85272 CCO3Y2 122187289 IC50 = 3.279 nM T85272 C1ENW4 122187290 IC50 = 0.046 nM T85272 CFH36G 122187291 IC50 = 0.0172 nM T85272 C3CY5N 122187292 IC50 = 0.004 nM T85272 CY69QI 122187293 IC50 = 0.0027 nM T85272 C05WQZ 122187294 IC50 = 0.003 nM T85272 C1LW9V 122187295 IC50 = 0.0195 nM T85272 CBMT85 122187296 IC50 = 0.0018 nM T85272 C8AKN9 122187297 IC50 = 0.0154 nM T85272 CDM71F 122187298 IC50 = 0.055 nM T85272 CCM08N 122187299 IC50 = 0.0038 nM T85272 C7V2TW 122187300 IC50 = 0.0028 nM T85272 C81QSJ 122187301 IC50 > 3.333 nM T85272 C1IPG9 122187302 IC50 = 0.0324 nM T85272 C0RE2W 122187303 IC50 > 3.333 nM T85272 C9JDM3 122187304 IC50 > 3.333 nM T85272 C5QXR6 122187305 IC50 = 0.0087 nM T85272 C50RMQ 122187306 IC50 = 0.0018 nM T85272 C5Z9PU 122187307 IC50 = 0.07 nM T85272 CT0V4W 122187308 IC50 > 3.333 nM T85272 CX06CZ 122187309 IC50 = 0.008 nM T85272 CK9T7F 122187310 IC50 = 0.59 nM T85272 CC2LE0 122187311 IC50 = 0.0036 nM T85272 CS34VD 122187312 IC50 = 0.002 nM T85272 CIU9T5 122187313 IC50 = 0.0031 nM T85272 CS8QW7 122187314 IC50 = 0.0042 nM T85272 CID97N 122187315 IC50 = 0.458 nM T85272 CZ08GP 122187316 IC50 = 0.0026 nM T85272 C0P6IC 122187317 IC50 > 3.333 nM T85272 CY7M0F 122187318 IC50 = 0.005 nM T85272 CQZK10 122187319 IC50 = 0.0033 nM T85272 C62FDT 122187320 IC50 = 0.0024 nM T85272 C3QZY1 122187321 IC50 = 0.0044 nM T85272 C8B4YL 122187322 IC50 = 0.005 nM T85272 CWV12K 122187323 IC50 = 0.0527 nM T85272 CWVP15 122187324 IC50 = 2.342 nM T85272 CEW35A 122187325 IC50 = 0.0017 nM T85272 CP43GQ 122187326 IC50 = 0.0021 nM T85272 CH46BC 122187327 IC50 = 0.04 nM T85272 C6KW2B 122187328 IC50 = 0.004 nM T85272 C87MGD 122187329 IC50 = 0.0028 nM T85272 C0U9QN 122187330 IC50 = 0.0335 nM T85272 CH4G1L 122187331 IC50 = 0.075 nM T85272 C4ZR9M 122187332 IC50 = 0.266 nM T85272 CM8A1Y 122187333 IC50 = 0.174 nM T85272 CU3IE9 122187334 IC50 = 0.005 nM T85272 CYN12K 122187335 IC50 = 0.0051 nM T85272 CDE52G 122187336 IC50 = 0.74 nM T85272 CZH25J 122187337 IC50 = 0.011 nM T85272 CQP1R4 122187338 IC50 = 0.6 nM T85272 C3QS0A 122187339 IC50 = 9.5 nM T85272 CAFO71 122187340 IC50 = 0.015 nM T85272 CNYJ15 122187341 IC50 = 29.26 nM T85272 CY62QW 122187342 IC50 = 13.22 nM T85272 CCV2G0 122187343 IC50 > 33.33 nM T85272 C0Z8JH 122187344 IC50 = 0.014 nM T85272 CVT8Z7 122187345 IC50 = 0.847 nM T85272 C2YI7W 122187346 IC50 = 0.214 nM T85272 CO7MU2 122187445 IC50 = 0.002 nM T85272 C8QN9Z 122187446 IC50 = 0.0068 nM T85272 C09YUX 122187447 IC50 = 0.005 nM T85272 C8I6TF 122187448 IC50 = 0.0022 nM T85272 CR68ZK 122187449 IC50 = 0.0035 nM T85272 CTY96B 122187450 IC50 = 0.0053 nM T85272 C4WG0M 122187451 IC50 = 0.0182 nM T85272 CLS4H7 122187452 IC50 = 0.0014 nM T85272 CM23CQ 122187453 IC50 = 0.76 nM T85272 CJF8X1 122187454 IC50 > 3.333 nM T85272 C54PSK 122187455 IC50 = 0.005 nM T85272 CGS5Q1 122187456 IC50 = 0.0014 nM T85272 CW0MH4 122187457 IC50 = 0.0011 nM T85272 CXAV52 122187458 IC50 = 0.0034 nM T85272 C3D8EQ 122187459 IC50 = 0.446 nM T85272 CBUT59 122187460 IC50 = 0.005 nM T85272 C1XL3M 122187461 IC50 = 0.004 nM T85272 CBS95M 122187462 IC50 = 0.005 nM T85272 CY79JC 122187463 IC50 = 0.0037 nM T85272 CAY0P4 122187464 IC50 = 0.006 nM T85272 CRQ98D 122187465 IC50 = 0.006 nM T85272 CXP98T 122187466 IC50 = 0.0042 nM T85272 C5TJU8 122187467 IC50 > 3.333 nM T85272 CP7C2I 122187468 IC50 = 0.028 nM T85272 CKC0L8 122187469 IC50 = 0.305 nM T85272 CV3T2C 122187470 IC50 = 0.011 nM T85272 CN5OQ2 122187471 IC50 = 0.0009 nM T85272 CI0J4A 122187472 IC50 = 0.0274 nM T85272 CM14KC 122187473 IC50 = 0.0157 nM T85272 COFI26 122187474 IC50 = 0.0489 nM T85272 CTXG58 122187475 IC50 = 0.0102 nM T85272 CZWG59 122187476 IC50 > 3.333 nM T85272 C1TVY5 122187477 IC50 = 0.0033 nM T85272 CS6FK8 122187478 IC50 > 3.333 nM T85272 CJC21F 122187479 IC50 = 0.0262 nM T85272 C3ZE4Y 122187480 IC50 > 3.333 nM T85272 CS0U8H 122187481 IC50 > 3.333 nM T85272 CY0NV5 122187482 IC50 = 0.0091 nM T85272 C8SHE5 122187483 IC50 = 1.018 nM T85272 CHYI14 122187484 IC50 = 2.42 nM T85272 CEH14V 122187485 IC50 > 3.333 nM T85272 CG98KU 122187486 IC50 = 0.0032 nM T85272 C3P8WN 122187487 IC50 = 0.0061 nM T85272 C9MJ2K 122187488 IC50 = 0.0061 nM T85272 C7J0YH 122187489 IC50 = 0.0044 nM T85272 C4NYT7 122187490 IC50 = 0.04 nM T85272 CMT25I 122187491 IC50 = 0.0015 nM T85272 CQEV80 122187492 IC50 = 0.0076 nM T85272 CY07HP 122187493 IC50 = 1.2 nM T85272 CD0EU3 122187494 IC50 = 0.0256 nM T85272 CQZ0R1 122187495 IC50 = 0.032 nM T85272 CZU4N2 122187496 IC50 = 0.0073 nM T85272 CITK91 122187497 IC50 = 0.0059 nM T85272 C69JKA 122187498 IC50 = 0.0042 nM T85272 C6R5CY 122187499 IC50 = 0.029 nM T85272 CM87YE 122187500 IC50 = 0.0045 nM T85272 CP4GJ7 122187501 IC50 = 0.051 nM T85272 CB14ES 122187502 IC50 = 0.004 nM T85272 CEGB98 122187503 IC50 = 0.042 nM T85272 CU61JG 137651545 IC50 = 13000 nM T85272 CW9P6A 145964460 IC50 > 30000 nM T85272 CQR49Z 145965116 IC50 > 30000 nM T85272 CR6L2G 145967358 IC50 > 30000 nM T85272 CHXE25 145978207 IC50 > 30000 nM T85272 D06PZZ 5413 IC50 = 30000 nM T85272 D08BMM 6312649 IC50 > 30000 nM T85272 D0R9CF 11302540 IC50 = 250 nM T96736 CR57DL 50803848 IC50 = 35000 nM T96736 CP79TH 52931882 IC50 = 2580 nM T96736 CPE79U 52931883 IC50 = 3280 nM T96736 C9LGO3 52931939 IC50 = 2620 nM T96736 C92SRX 52931998 IC50 = 1510 nM T96736 C5F1IT 52932001 IC50 = 2050 nM T96736 CWFG81 52932003 IC50 = 1680 nM T96736 C65DNB 52932059 IC50 = 1240 nM T96736 C06LVX 53363853 IC50 = 2090 nM T96736 C3QGZ1 53364100 IC50 = 3000 nM T96736 CXYI14 71681394 IC50 = 9200 nM T96736 COBN97 71681395 IC50 = 10000 nM T96736 CR5BQ2 71681396 IC50 = 31000 nM T96736 C6E8TM 71681562 IC50 = 9900 nM T96736 C7ITA6 71681563 IC50 = 27000 nM T96736 C9KP1U 71681564 IC50 = 26000 nM T96736 CE6P5O 71681565 IC50 = 33000 nM T96736 CH4F1V 71681566 IC50 = 33000 nM T96736 CA2GQ5 71681720 IC50 = 35000 nM T96736 CP8UN5 71681721 IC50 = 43000 nM T96736 C6O8VG 71681722 IC50 = 51000 nM T96736 C3WU8P 71681723 IC50 = 67000 nM T96736 CA68PI 71681724 IC50 = 78000 nM T96736 C0TKW7 71682046 IC50 = 1500 nM T96736 CGJ18W 71682047 IC50 = 1600 nM T96736 CGMO97 71682048 IC50 = 2300 nM T96736 C4QA6W 71682049 IC50 = 5600 nM T96736 CY63JH 71682050 IC50 = 6100 nM T96736 C2QH9Y 71682204 IC50 = 8100 nM T96736 CS45BO 71682205 IC50 = 11000 nM T96736 CE87JT 71682206 IC50 = 12000 nM T96736 C5KR2M 71682207 IC50 = 12000 nM T96736 CKG6I5 71682208 IC50 = 26000 nM T96736 C4MDP1 71682354 IC50 = 30000 nM T96736 C1H9AY 71682355 IC50 = 32000 nM T96736 CB9J7C 71682356 IC50 = 32000 nM T96736 C0X4DB 71682357 IC50 = 66000 nM T96736 CPQ8K0 71682358 IC50 = 76000 nM T96736 CM82DF 71682662 IC50 = 21000 nM T96736 C5XR3L 71682663 IC50 = 7400 nM T96736 C96MSZ 71682815 IC50 = 10000 nM T96736 C0IE1G 73349029 IC50 = 4700 nM T96736 D0I3KR 71681561 IC50 = 5300 nM T96736 D0Y9BU 46190808 IC50 = 9800 nM T86808 CL2Q6J 44178077 IC50 > 100000 nM T86808 C0BQC4 44586265 IC50 = 2200 nM T86808 C2IML9 58580486 IC50 = 460 nM T86808 D0K1NM 20541332 IC50 > 100000 nM T55398 D0OB0F 5328940 IC50 = 574 nM T55398 D03LWG 53235510 IC50 > 10000 nM T55398 D07EHV 44814409 IC50 > 10000 nM T55398 D07NUL 118414016 IC50 = 2 nM T55398 D0E3TC 44259 IC50 = 4.21 nM T55398 D0T3ME 156422 IC50 > 30000 nM T55398 CGEW10 1247796 IC50 = 2200 nM T55398 CJ3U9Y 2728161 IC50 = 55000 nM T55398 CF6WI5 2824236 IC50 = 2800 nM T55398 C1KY3I 4455946 IC50 = 12000 nM T55398 CRC65X 9863786 IC50 > 30000 nM T55398 C5UG6X 10114595 Ki = 0.48 nM T55398 C8K9HL 10142476 Ki = 0.42 nM T55398 C4RNU9 10184123 Ki = 0.5 nM T55398 CN37YZ 10207985 Ki = 0.34 nM T55398 C8BHJ3 10226185 Ki = 8.2 nM T55398 C78SMB 10227510 Ki = 2.8 nM T55398 CXN06I 10227557 Ki = 2.8 nM T55398 C0SR5Y 10278151 Ki = 0.7 nM T55398 CBOP58 11293798 Ki > 10000 nM T55398 C26BZX 11362471 Ki > 10000 nM T55398 CWXB93 11397177 Ki > 10000 nM T55398 CTG83F 11539329 Ki > 9900 nM T55398 CACS26 11561968 Ki > 4000 nM T55398 CMIL86 11590363 Ki > 9900 nM T55398 C9T6SC 11640926 Ki > 9900 nM T55398 CU0E8O 11690457 Ki = 1900 nM T55398 CB0AP2 11705863 Ki > 4000 nM T55398 CE2VU0 11987888 Ki = 1.2 nM T55398 CFPW41 16007116 Ki > 9900 nM T55398 CST43D 21899140 Ki = 6.5 nM T55398 CM4F0B 21899142 Ki = 1.3 nM T55398 CT46EH 21899147 IC50 = 8000 nM T55398 C7YG1N 24759534 IC50 = 210 nM T55398 CIN29Y 24801862 IC50 = 400 nM T55398 CZ12SD 24801863 IC50 = 3000 nM T55398 CZJ9P4 24857834 IC50 = 70 nM T55398 C3E5XY 24857850 IC50 = 420 nM T55398 CLZ23U 24951610 IC50 = 1100 nM T55398 C2KY1G 25094210 IC50 = 167 nM T55398 CGT1W6 25144294 IC50 = 56 nM T55398 CU7VR0 25144732 IC50 = 8 nM T55398 C6BWZ8 25145145 IC50 = 1000 nM T55398 CA75YC 25169380 IC50 = 6 nM T55398 CC3BU0 25169381 IC50 = 4 nM T55398 CFB65H 25169382 IC50 = 6 nM T55398 CRXS80 25169384 IC50 = 9 nM T55398 CC71QJ 27666048 IC50 > 100000 nM T55398 CTA08W 41420877 IC50 = 2000 nM T55398 CO6HU7 44178069 IC50 = 1142 nM T55398 C8KNA3 44219632 Ki > 4000 nM T55398 C0VIX4 44219633 Ki = 2300 nM T55398 CZH6G2 44412152 IC50 > 30000 nM T55398 C1OQP6 44412156 IC50 = 1500 nM T55398 CJR94S 44412164 IC50 > 30000 nM T55398 COZ5X9 44412166 IC50 = 25000 nM T55398 CU7Q3F 44412167 IC50 = 4000 nM T55398 CU0T2G 44412174 IC50 = 1000 nM T55398 C0V4FU 44412178 IC50 = 550 nM T55398 CIF5C1 44412201 IC50 = 1000 nM T55398 CCY3L4 44412220 IC50 = 20000 nM T55398 CR7Y9K 44412242 IC50 = 30000 nM T55398 C4UOZ2 44412243 IC50 = 6000 nM T55398 CGJ61S 44412251 Ki = 4500 nM T55398 C18ZMY 44412252 IC50 = 800 nM T55398 CM6X1B 44412253 IC50 = 2000 nM T55398 C6TN3O 44412266 IC50 = 1000 nM T55398 CD2W6N 44412267 IC50 = 2000 nM T55398 CRB74Z 44412281 IC50 = 400 nM T55398 C0R2LO 44412325 IC50 = 30000 nM T55398 CA0MI2 44412326 IC50 = 400 nM T55398 CH7M4G 44412327 IC50 = 1000 nM T55398 C35CLR 44412343 IC50 = 150 nM T55398 C7XE0D 44412352 IC50 = 4000 nM T55398 CUV9B8 44412391 IC50 = 6500 nM T55398 CH6F7D 44412392 IC50 = 2000 nM T55398 CG3LU0 44412407 IC50 = 30000 nM T55398 CZ16BF 44412434 IC50 = 4000 nM T55398 CA48QG 44412435 IC50 = 3000 nM T55398 C20AUC 44412442 IC50 = 500 nM T55398 C6N1MJ 44412480 IC50 = 3000 nM T55398 C6O0TZ 44412492 IC50 = 6500 nM T55398 CRK51G 44448764 IC50 = 39 nM T55398 CKI6S2 44448795 IC50 = 6900 nM T55398 C1HB0N 44448797 IC50 = 313 nM T55398 C7GA2S 44448798 IC50 = 3030 nM T55398 CTGL39 44448828 IC50 = 225 nM T55398 CSAH90 44448865 IC50 = 1300 nM T55398 CDWX21 44448867 IC50 = 914 nM T55398 CXV8T5 44448904 IC50 = 497 nM T55398 C3DP0G 44448905 IC50 = 8100 nM T55398 CAQ4T1 44448906 IC50 = 433 nM T55398 CO7Y6K 44448908 IC50 = 1134 nM T55398 COY50K 44448910 IC50 = 1085 nM T55398 CL28QE 44448912 IC50 = 10 nM T55398 CVQ74G 44448939 IC50 = 49 nM T55398 CIUF03 44448940 IC50 = 1156 nM T55398 C28SLH 44448941 IC50 = 5 nM T55398 C47GQS 44448942 IC50 = 263 nM T55398 CCV97Y 44448943 IC50 = 166 nM T55398 CHCN76 44448970 IC50 = 2 nM T55398 C3YM1B 44448971 IC50 = 63 nM T55398 C4S5TP 44448972 IC50 = 112 nM T55398 CV5F0Q 44448973 IC50 = 7 nM T55398 CX8PM6 44448975 IC50 = 3 nM T55398 CH61MQ 44449000 IC50 = 8 nM T55398 C3C2TM 44449002 IC50 = 181 nM T55398 CT3B1M 44449003 IC50 = 208 nM T55398 CE07NB 44449025 IC50 = 15 nM T55398 C5X0LI 44449050 IC50 = 1 nM T55398 CZ3V1X 44449078 IC50 = 35 nM T55398 C0SQE3 44449102 IC50 = 216 nM T55398 CK6E5J 44449122 IC50 = 95 nM T55398 CT7U9G 44449126 IC50 = 7 nM T55398 C37YOA 44449160 IC50 = 487 nM T55398 CXL76B 44449162 IC50 = 535 nM T55398 CSRC92 44449189 IC50 = 1880 nM T55398 CQ5I9D 44449190 IC50 = 126 nM T55398 C3DU4B 44449218 IC50 = 19 nM T55398 C64YUV 44449221 IC50 = 545 nM T55398 C1G4DC 44449335 IC50 = 710 nM T55398 C0CR1V 44449336 IC50 = 660 nM T55398 C1W9XR 44449364 IC50 = 1600 nM T55398 CMC7U0 44449365 IC50 > 10000 nM T55398 C2DCP7 44449366 IC50 > 10000 nM T55398 CP6R3S 44449367 IC50 > 10000 nM T55398 C6IHR2 44449391 IC50 = 3400 nM T55398 CJ68ZB 44449392 IC50 = 160 nM T55398 CZJ8U5 44449393 IC50 = 350 nM T55398 CZYR60 44449394 IC50 = 1200 nM T55398 C2SO6L 44449424 IC50 > 10000 nM T55398 CEGF72 44449425 IC50 > 10000 nM T55398 CBA80K 44449426 IC50 = 700 nM T55398 CUY8W6 44449427 IC50 = 2800 nM T55398 CRWG12 44449486 IC50 = 2400 nM T55398 CF0V1N 44449548 IC50 = 3700 nM T55398 C24SWN 44449549 IC50 = 8900 nM T55398 CD6XC0 44449584 IC50 = 4800 nM T55398 C9TR0X 44449617 IC50 = 1000 nM T55398 C3V7EY 44449647 IC50 = 800 nM T55398 CWB60J 44449650 IC50 > 10000 nM T55398 C6DHC9 44450171 IC50 = 7300 nM T55398 C3DQJ6 44450195 IC50 = 7200 nM T55398 CYH6P3 44520205 IC50 = 340 nM T55398 COV31Z 44586245 IC50 = 200 nM T55398 CE3V0Z 44586278 IC50 = 1189 nM T55398 CC5W9J 44586319 IC50 = 456 nM T55398 C8WPI5 44586320 IC50 = 1934 nM T55398 CZI08B 46175395 IC50 = 170 nM T55398 C35UQP 46175482 IC50 = 240 nM T55398 CF0OV6 46175578 IC50 = 1060 nM T55398 CRC37F 46176531 IC50 > 20000 nM T55398 CY3HW5 46224684 IC50 > 10000 nM T55398 COTJ39 46863083 IC50 = 1100 nM T55398 CLS29B 46872626 IC50 > 10000 nM T55398 C1Q8AW 49824621 Ki = 38.5 nM T55398 CAZQ43 51003133 IC50 = 380 nM T55398 CC24GM 52913874 IC50 = 21 nM T55398 CXA03W 52920796 IC50 = 640 nM T55398 CEQN27 52936621 Ki > 1000 nM T55398 C6OTY5 53251320 IC50 = 26000 nM T55398 CE8OY2 53317913 IC50 = 8 nM T55398 C0SWH5 53348216 IC50 > 40000 nM T55398 C8ZRE3 53356518 IC50 > 50000 nM T55398 C8NA4L 53384644 IC50 > 30000 nM T55398 C1XS2J 54760383 IC50 > 10000 nM T55398 C5KR6N 56595558 Ki = 43 nM T55398 COI9U2 56595687 Ki = 420 nM T55398 C2AM6B 56595688 Ki = 1200 nM T55398 CFY2I4 56595689 Ki = 160 nM T55398 CAM8E1 56595690 Ki = 440 nM T55398 CN5EV7 56595691 Ki = 36 nM T55398 C6ET0W 56595693 Ki = 78 nM T55398 CTR10F 56658543 Ki = 340 nM T55398 C9MJG4 56929824 IC50 = 430 nM T55398 C0UDY9 57401151 IC50 = 7500 nM T55398 COY07J 57519810 IC50 <= 5000 nM T55398 C0PA3D 57519811 Ki = 50 nM T55398 CO75VX 58056108 Ki = 1.7 nM T55398 CSN35V 58056134 Ki = 790 nM T55398 C8CG6L 58056265 Ki = 52 nM T55398 CVQ2U4 58056270 Ki = 610 nM T55398 C8GFI0 58056341 Ki = 2 nM T55398 C9MIL7 58450666 IC50 = 1800 nM T55398 C9HUB2 58570982 IC50 = 240 nM T55398 C6BPR2 58985201 IC50 > 30000 nM T55398 CT3EW2 59292007 IC50 > 1000 nM T55398 CP9A8T 59503659 IC50 = 1219 nM T55398 C1MA6J 59503711 IC50 = 1423 nM T55398 CX29EU 59503744 IC50 = 873 nM T55398 CXJ63M 59603829 IC50 = 64 nM T55398 CQEU96 59603842 IC50 = 23 nM T55398 COH62U 60097413 IC50 > 10000 nM T55398 C1MR8Q 60097495 IC50 > 10000 nM T55398 CK6WO0 66552478 IC50 < 10000 nM T55398 CUF20T 66554581 IC50 = 80 nM T55398 CZ92KC 66554752 IC50 = 2100 nM T55398 CF7RQ2 66554923 IC50 = 280 nM T55398 CMS6L3 66554926 IC50 = 180 nM T55398 CU1DM5 66555095 IC50 = 220 nM T55398 CVQW04 66555265 IC50 = 59 nM T55398 C53YWX 66555955 IC50 = 99 nM T55398 CSL0F3 66555956 IC50 = 170 nM T55398 COS5Q9 66555957 IC50 = 44 nM T55398 C7N3DE 66557142 IC50 < 100 nM T55398 C08DXU 66557143 IC50 < 100 nM T55398 COU2C4 66664636 Ki = 8 nM T55398 CV63UL 67240318 IC50 > 10000 nM T55398 C80HMA 68115414 IC50 = 1500 nM T55398 CW23JE 68241353 IC50 = 470 nM T55398 CK9E0Y 68327832 IC50 = 7 nM T55398 CU26SP 68327847 IC50 = 150 nM T55398 CPG75C 68327866 IC50 = 85 nM T55398 CE41YS 68327879 IC50 = 180 nM T55398 CA47UH 68328137 IC50 = 410 nM T55398 C5Z7QJ 68328146 IC50 = 2400 nM T55398 C8OAS6 68328387 IC50 = 27 nM T55398 C3QE9V 68328415 IC50 = 390 nM T55398 CI4HV8 68328491 IC50 = 2 nM T55398 C9HZG1 68328492 IC50 = 40 nM T55398 CC6F8D 68328504 IC50 = 47 nM T55398 C43RXO 68328520 IC50 = 310 nM T55398 CB2OM0 68328789 IC50 = 61 nM T55398 CRM6L5 68357884 IC50 = 5 nM T55398 CZG9X7 68357894 IC50 = 13 nM T55398 C2B1TC 68357902 IC50 = 370 nM T55398 CYI75G 68678653 IC50 = 24400 nM T55398 C5DGR9 69036886 IC50 = 10000 nM T55398 CV0QP3 70947961 Ki = 11 nM T55398 CKT60L 71455860 Ki > 9900 nM T55398 C6T1LM 71506869 IC50 < 50 nM T55398 CE5XR2 71612615 IC50 = 1.8 nM T55398 C5RZ7I 72709739 IC50 = 100 nM T55398 CV3I1N 72943654 IC50 < 100 nM T55398 CIT2V7 72945768 IC50 = 100 nM T55398 CX1UE8 72945946 IC50 = 100 nM T55398 CM94EG 72945952 IC50 > 30000 nM T55398 CZNM96 73053607 IC50 < 100 nM T55398 C25UCH 73053622 IC50 < 100 nM T55398 C1RO3T 73053624 IC50 < 100 nM T55398 CX75YR 73352604 IC50 = 3.981 nM T55398 C8JTD0 73442848 IC50 = 138 nM T55398 CE5CX0 73442898 IC50 = 300 nM T55398 COU3K5 73669498 IC50 = 113 nM T55398 CS2QC6 73669499 IC50 = 204 nM T55398 C7LER5 73669500 IC50 = 3452 nM T55398 C5C4SU 73669664 IC50 = 1140 nM T55398 CF0C4R 73669837 IC50 = 42000 nM T55398 CYO3D1 73669840 IC50 = 2570 nM T55398 C0FH9Y 73670011 IC50 = 1000 nM T55398 C5WLK7 73670169 IC50 = 410 nM T55398 CTG6S3 73670172 IC50 = 333000 nM T55398 C40BHZ 73670173 IC50 = 228000 nM T55398 CJKB83 73670174 IC50 = 11 nM T55398 CF42WG 73670176 IC50 = 4700 nM T55398 C62MPO 73670344 IC50 = 1081000 nM T55398 CW1VG7 73670345 IC50 = 3012000 nM T55398 CJF7Y5 73670346 IC50 = 104 nM T55398 CZU1A0 73670347 IC50 = 24 nM T55398 CCUH57 73670348 IC50 = 16 nM T55398 C82COK 73670350 IC50 = 18 nM T55398 CD23NU 73670513 IC50 = 6000 nM T55398 C1LPW5 73670673 IC50 = 1000 nM T55398 CLO61M 73670847 IC50 = 89 nM T55398 C6T4WZ 73670848 IC50 = 94 nM T55398 CF7TD8 73670850 IC50 = 530 nM T55398 CT3L4F 73670851 IC50 = 932 nM T55398 CN4B8K 75202037 IC50 = 1.5 nM T55398 CFL54M 75204288 IC50 = 1.8 nM T55398 CYJ4C6 76955703 IC50 < 100 nM T55398 CSH9R0 77847460 IC50 < 100 nM T55398 CQ2SU8 78673832 IC50 > 30000 nM T55398 CE0W9R 78673833 IC50 > 30000 nM T55398 C1HW4B 89735655 IC50 = 3000 nM T55398 C89YHN 90134560 IC50 = 5.3 nM T55398 C2CY5A 90154381 IC50 = 3.6 nM T55398 CGTN69 90154630 IC50 = 1.9 nM T55398 C5S0DF 90154917 IC50 = 3.5 nM T55398 CZTM62 90155093 IC50 = 5.6 nM T55398 CAL0O9 90155375 IC50 = 13 nM T55398 CI5GF8 90155577 IC50 = 300 nM T55398 CSC20O 90271946 IC50 = 20 nM T55398 CWA46G 90271957 IC50 < 100 nM T55398 CC1S2P 90272141 IC50 = 71 nM T55398 CM2LJ5 90275527 IC50 = 2400 nM T55398 CNX5V4 91844450 IC50 = 1193000 nM T55398 C0Y8ZK 91933875 IC50 > 1000 nM T55398 CA1K0F 91938073 IC50 = 1.3 nM T55398 CAU45T 91971978 IC50 > 30000 nM T55398 C0YSX8 117826679 IC50 = 4300 nM T55398 CWA8X7 117871492 IC50 = 2197 nM T55398 CI40BM 117871555 IC50 = 3649 nM T55398 CU1V7Y 117871558 IC50 = 187 nM T55398 CQ6E2O 117871721 IC50 > 20000 nM T55398 CTS35E 117871724 IC50 = 3452 nM T55398 CE7X1L 117871750 IC50 = 212 nM T55398 C6MG7L 117871760 IC50 = 730 nM T55398 C0A4XC 117871929 IC50 = 74 nM T55398 CV4B2W 117871992 IC50 = 307 nM T55398 CY60JR 117872182 IC50 = 401 nM T55398 C3VJ0I 117872205 IC50 = 542 nM T55398 CY5JF0 117872250 IC50 = 187 nM T55398 COIM28 117872315 IC50 = 190 nM T55398 C7PM6F 117872316 IC50 = 1100 nM T55398 C63OVX 117872321 IC50 = 653 nM T55398 CT4AZ2 117872334 IC50 = 1100 nM T55398 C6X8VS 117872368 IC50 = 191 nM T55398 CR0JN8 117872469 IC50 = 128 nM T55398 CBOI97 117872492 IC50 = 478 nM T55398 CO6BH7 117872621 IC50 = 1449 nM T55398 CD8J9G 117872890 IC50 = 1605 nM T55398 CQ5S7L 117872990 IC50 = 285 nM T55398 CD6EA9 117873013 IC50 = 2677 nM T55398 C9OA4U 117873033 IC50 = 101 nM T55398 CL6QV4 117873045 IC50 = 261 nM T55398 CDO5I6 117873092 IC50 = 106 nM T55398 CP89EY 117873164 IC50 = 2 nM T55398 C8QB3S 117873179 IC50 = 1582 nM T55398 CWG60S 117873194 IC50 = 2725 nM T55398 CT3B6F 117873210 IC50 = 683 nM T55398 C08YAE 117885624 IC50 = 12 nM T55398 C2V1RC 117885639 IC50 = 830 nM T55398 CS9J3N 117885675 IC50 = 155 nM T55398 CJ8I7U 117885678 IC50 = 12 nM T55398 CK1A0N 117885680 IC50 = 11900 nM T55398 CYP9O7 117885688 IC50 = 12 nM T55398 C4ECT8 117885692 IC50 = 2107 nM T55398 CYN4S1 117885705 IC50 = 3 nM T55398 C2ABD1 117885712 IC50 = 852 nM T55398 CF6UT1 117885715 IC50 = 373 nM T55398 C3VN9K 117885730 IC50 = 7 nM T55398 CZ8P4J 117885751 IC50 = 4 nM T55398 C9R3WU 117885753 IC50 = 6008 nM T55398 C1HND8 117885755 IC50 = 9510 nM T55398 CS72RV 117885758 IC50 = 216 nM T55398 C6Z3NJ 117885766 IC50 = 44 nM T55398 CKU6S4 117885912 IC50 = 8 nM T55398 C1E2DK 118072831 IC50 < 100 nM T55398 C1ZR5E 118173110 IC50 = 33 nM T55398 CV5Q9X 118388894 IC50 = 4381 nM T55398 CT9RU4 118413945 IC50 = 1.3 nM T55398 C36CUE 118414094 IC50 = 0.5 nM T55398 C69QWZ 118414114 IC50 = 29.5 nM T55398 C7J6RO 118414128 IC50 = 4.8 nM T55398 CLWJ18 118414336 IC50 = 7.6 nM T55398 CSQV50 118414357 IC50 = 840 nM T55398 CUJ9O2 118414389 IC50 = 0.1 nM T55398 CF2D3K 118414391 IC50 = 2836 nM T55398 C5XRA6 118414397 IC50 = 23.9 nM T55398 CHL38K 118414437 IC50 = 5.9 nM T55398 CFM20Z 118414536 IC50 = 0.3 nM T55398 CW3IC5 118414671 IC50 = 4.6 nM T55398 C3N5SA 118414693 IC50 = 12.1 nM T55398 CIH2O7 118414733 IC50 = 3.7 nM T55398 C51HAN 118414780 IC50 = 2.7 nM T55398 C0O3SN 118424414 IC50 = 2.4 nM T55398 CUN8Y5 118424424 IC50 = 0.6 nM T55398 COH1T4 118453721 IC50 = 6 nM T55398 CR7DJ0 118453722 IC50 = 55 nM T55398 CK1Z7I 118462026 IC50 = 4 nM T55398 COB6M3 118475320 IC50 = 2 nM T55398 CX2GE1 118475349 IC50 = 250 nM T55398 CZBA29 118641364 IC50 <= 100 nM T55398 CX58DI 118716791 IC50 > 30000 nM T55398 CD9X2B 118716796 IC50 > 30000 nM T55398 C2YJ0O 118716797 IC50 > 30000 nM T55398 CL3UO9 118716798 IC50 > 30000 nM T55398 C71BAM 118716799 IC50 > 30000 nM T55398 CU4EL6 118716806 IC50 > 30000 nM T55398 C5FK7T 118719435 IC50 = 0.36 nM T55398 CA2NJ8 118719437 IC50 = 0.24 nM T55398 CEFG28 118719438 IC50 = 2.8 nM T55398 CL1N2T 118719440 IC50 = 0.32 nM T55398 CCJ0X7 118719442 IC50 = 2.6 nM T55398 CJ2IZ0 118719443 IC50 = 2.2 nM T55398 CIV1H2 118719446 IC50 <= 100 nM T55398 CHT6K9 118728811 Ki > 4000 nM T55398 CUA3Y2 118728812 Ki > 4000 nM T55398 CDQ78G 118728813 Ki > 4000 nM T55398 CZ6XL7 118728814 Ki > 4000 nM T55398 CMO67K 118728815 Ki > 4000 nM T55398 CR2M0Q 118728816 Ki > 4000 nM T55398 C62SCL 118728817 Ki > 4000 nM T55398 CSB30C 118728819 Ki > 4000 nM T55398 CV7XU8 118728820 Ki = 2700 nM T55398 C3J1EX 118728821 Ki > 4000 nM T55398 CIWB78 118728822 Ki > 4000 nM T55398 CP18SE 118728823 Ki = 3300 nM T55398 CM42CA 118728824 Ki > 4000 nM T55398 C9Q7CL 118728825 Ki > 4000 nM T55398 CCR3S0 118728826 Ki > 4000 nM T55398 CNJK97 118729800 IC50 > 20000 nM T55398 C14CYV 118729801 IC50 = 5190 nM T55398 CNP64R 118729802 IC50 > 20000 nM T55398 CP3U7F 118729803 IC50 = 6850 nM T55398 CQ4Z2H 118729804 IC50 > 20000 nM T55398 CQ92UP 118729805 IC50 > 20000 nM T55398 CX9BS1 118729806 IC50 > 20000 nM T55398 C7WFP3 118729807 IC50 > 20000 nM T55398 C3MUB5 118729808 IC50 > 20000 nM T55398 CHDF03 118729809 IC50 > 20000 nM T55398 C6AW4N 118729810 IC50 > 20000 nM T55398 CBWY74 118729811 IC50 = 1140 nM T55398 CN1KS6 118729812 IC50 > 20000 nM T55398 C36BLM 118729813 IC50 = 403000 nM T55398 C4R1EI 121254788 IC50 = 10 nM T55398 C0XU9Y 121255032 IC50 = 7400 nM T55398 CNQ6Z2 121255052 IC50 = 16 nM T55398 CS64MC 121255054 IC50 = 300 nM T55398 CM1W3K 121255069 IC50 = 16 nM T55398 CYDF91 121255074 IC50 = 9 nM T55398 CDQ48W 121255075 IC50 = 19 nM T55398 CZTX30 121256083 IC50 = 12 nM T55398 CJY83B 121258892 IC50 = 17 nM T55398 CTPB07 121262387 IC50 = 32 nM T55398 CUL6H1 121262551 IC50 = 35 nM T55398 C7X1BQ 121493987 IC50 = 38 nM T55398 C30ILY 122180370 IC50 = 690 nM T55398 CK6YL8 122181591 IC50 = 110 nM T55398 CZFT46 122181592 IC50 = 150 nM T55398 COJ93A 122181593 IC50 = 9200 nM T55398 C3EN9U 122181594 IC50 = 2 nM T55398 CWL8R2 122181623 IC50 = 95 nM T55398 CJD5F2 122181624 IC50 = 20 nM T55398 C8C5TR 122181625 IC50 = 8 nM T55398 CT2BY5 122181626 IC50 = 0.3 nM T55398 CYEG26 122181627 IC50 = 14 nM T55398 C06BWF 122181628 IC50 = 6 nM T55398 CEN5P0 122181629 IC50 = 0.8 nM T55398 C6W4PS 122181630 IC50 = 0.3 nM T55398 C1Z0EK 122181631 IC50 = 0.2 nM T55398 CY4HG7 122181632 IC50 = 2 nM T55398 CW74UE 122181633 IC50 = 6 nM T55398 CV87TR 122181634 IC50 = 62 nM T55398 C92TUX 122181635 IC50 = 160 nM T55398 CSD5U0 122181636 IC50 = 480 nM T55398 CC3FS4 122181637 IC50 = 21 nM T55398 CD83YT 122181638 IC50 = 4 nM T55398 CVQ7H5 122181639 IC50 = 10 nM T55398 CTD2I5 122181640 IC50 = 1 nM T55398 CKJU62 122181641 IC50 = 23 nM T55398 CMQ2R0 122181642 IC50 = 13 nM T55398 C4WZR2 122181643 IC50 = 3 nM T55398 CF2LI0 122181644 IC50 = 3 nM T55398 CMZ95X 122181645 IC50 = 1 nM T55398 CFU63N 122181674 IC50 = 0.5 nM T55398 CF7OC2 122181675 IC50 = 0.5 nM T55398 C76RQM 122181676 IC50 = 6 nM T55398 C8D3JG 122184715 IC50 = 11 nM T55398 C0BLW3 122184716 IC50 = 647 nM T55398 CAQ71B 122191866 IC50 = 470 nM T55398 CO6S2E 122196062 IC50 = 40 nM T55398 C8R7FJ 122196063 IC50 = 5 nM T55398 CJA40H 122196064 IC50 = 1 nM T55398 CV85FQ 122196065 IC50 = 10 nM T55398 CBW67H 122196066 IC50 = 1 nM T55398 C7W5QA 122196067 IC50 = 0.2 nM T55398 CS6AP9 122196068 IC50 = 38 nM T55398 CJO8V9 122196168 IC50 = 3 nM T55398 CVI2P6 122196169 IC50 < 0.5 nM T55398 CO72HB 122196170 IC50 = 2 nM T55398 CA6BO3 122196171 IC50 = 1 nM T55398 CU2XL4 122196172 IC50 = 0.8 nM T55398 CZ3W8X 122196173 IC50 < 0.5 nM T55398 CB21TD 122196174 IC50 = 24 nM T55398 C51YFU 122196175 IC50 = 0.9 nM T55398 CX07CU 122196176 IC50 = 0.4 nM T55398 C2HLK9 122196177 IC50 = 0.2 nM T55398 C84DQM 122196178 IC50 = 0.7 nM T55398 C0DO3U 122196179 IC50 < 0.5 nM T55398 CYMK98 122196180 IC50 = 1 nM T55398 CQ1OM7 122196181 IC50 = 1 nM T55398 CLFH30 122196246 IC50 = 7 nM T55398 C5Z2FM 122196247 IC50 = 25 nM T55398 CTX0M5 122196248 IC50 = 12 nM T55398 C43LHP 122196249 IC50 = 0.4 nM T55398 C6QZE1 123917405 IC50 = 2400 nM T55398 CZEV34 125479776 IC50 = 1200 nM T55398 CR3A1O 125495464 IC50 = 15 nM T55398 CGU28T 126573669 IC50 = 121 nM T55398 C2T8ZA 126573681 IC50 = 146 nM T55398 C4S5LR 126622195 IC50 = 0.2 nM T55398 CH4C5O 126961337 IC50 = 58 nM T55398 CAGL14 126970816 IC50 = 71.9 nM T55398 C31ZLG 127034634 Ki = 7.8 nM T55398 CX3YO4 127034635 Ki = 11 nM T55398 CUS38N 127034643 IC50 = 150 nM T55398 C1C4UV 127034834 Ki = 3.8 nM T55398 CZ7H8F 127035289 Ki = 1.6 nM T55398 CZD87E 127037084 IC50 = 465 nM T55398 CB9Z0V 127038973 IC50 = 234 nM T55398 C1KH4L 129284027 Ki = 30 nM T55398 C6RGX5 129284078 Ki = 2.1 nM T55398 C9VL8H 129284112 Ki = 7.4 nM T55398 CWF79O 129284190 Ki = 14 nM T55398 CBJ6X9 129284195 IC50 = 0.38 nM T55398 C3VK4I 129284254 Ki = 7.3 nM T55398 C4VS8P 129284274 Ki = 35 nM T55398 CK2IL4 129284334 IC50 = 0.19 nM T55398 C96LDG 129284345 Ki = 5.1 nM T55398 CN8WZ2 129284370 Ki = 80 nM T55398 C8VNP1 129284385 IC50 = 7.2 nM T55398 CWA5R2 129284395 Ki = 6.6 nM T55398 CR2YV6 129284442 IC50 = 3.6 nM T55398 C4MG6I 129284483 Ki = 1.1 nM T55398 C9W4CS 129284507 Ki = 6.1 nM T55398 CR94JT 129284517 Ki = 3.5 nM T55398 CF19RT 129284574 Ki = 15 nM T55398 CM2J9U 129284575 Ki = 13 nM T55398 C49BMA 129284616 Ki = 6.1 nM T55398 CO4QV7 129284658 Ki = 1.5 nM T55398 C43SGU 129284679 Ki = 31 nM T55398 CS71NJ 129284701 Ki = 34 nM T55398 CV25CZ 129284859 Ki = 3.2 nM T55398 CM23FX 129297015 Ki = 12 nM T55398 CQO83S 129297033 Ki = 10 nM T55398 C0Z5NP 129297518 Ki = 5.8 nM T55398 C2FU6N 129297531 IC50 = 1.2 nM T55398 CFSC56 129297811 Ki = 3.2 nM T55398 C4NG3W 129298165 IC50 = 0.16 nM T55398 CUOX69 129298210 IC50 = 0.081 nM T55398 CTA06R 129298213 IC50 = 0.32 nM T55398 C96KMC 129298275 Ki = 6.5 nM T55398 C8MXQ4 130274633 IC50 = 7 nM T55398 CK4N0V 130274681 IC50 = 122 nM T55398 C45OHZ 130275697 IC50 = 3 nM T55398 C18QMF 130275783 IC50 = 3 nM T55398 C3WG8E 130276452 IC50 = 8 nM T55398 C9WK5I 130276470 IC50 = 17 nM T55398 CXTZ19 131704459 IC50 = 10 nM T55398 C25WQI 131704460 IC50 > 10000 nM T55398 CY70JL 131839618 IC50 = 6 nM T55398 C4Z5MQ 131839619 IC50 = 5 nM T55398 C2W8TC 131839620 IC50 = 42 nM T55398 C0M7PT 131839621 IC50 = 2 nM T55398 CNF79T 133107904 IC50 = 4 nM T55398 CB0C4Y 133107905 IC50 = 69 nM T55398 CJ43BV 133107906 IC50 = 21.38 nM T55398 C2AN7T 134611886 IC50 > 100000 nM T55398 CY4D8I 135566504 Ki > 1000 nM T55398 C7PJ6X 135566704 IC50 > 30000 nM T55398 C6DP4U 135567024 IC50 = 25 nM T55398 CX3UR8 135567025 IC50 = 19 nM T55398 CPV59N 135685787 Ki = 1500 nM T55398 CG3UZ1 135927974 Ki > 1000 nM T55398 CF1PS8 135934877 Ki = 690 nM T55398 CTRL59 135976660 Ki = 1100 nM T55398 CU0SZ4 136074298 IC50 < 100 nM T55398 CDMS84 136074299 IC50 < 100 nM T55398 CSOR07 136074300 IC50 = 14 nM T55398 CQ84IZ 136180335 Ki > 4000 nM T55398 COLR97 136272332 IC50 = 1487 nM T55398 CS9Z2N 136272346 IC50 = 1688 nM T55398 CX48MU 136272376 IC50 = 11 nM T55398 CYUF15 136272377 IC50 = 78 nM T55398 CL6S3R 136272378 IC50 = 43 nM T55398 C6T7AE 136272379 IC50 = 135 nM T55398 C7Y1QZ 136272387 IC50 = 43 nM T55398 C2V7QH 136272388 IC50 = 27 nM T55398 CN49DR 136272389 IC50 = 490 nM T55398 C7XY1B 136272390 IC50 = 67 nM T55398 COQ3V4 136504460 IC50 = 972 nM T55398 CVPE08 136504461 IC50 = 2429 nM T55398 CB0M7Z 136504482 IC50 = 454 nM T55398 C7ZF1S 136508720 IC50 = 79 nM T55398 CY1Q8P 136508752 IC50 = 85 nM T55398 C5K8ED 136932639 IC50 = 565 nM T55398 C9DF2X 136932640 IC50 = 580 nM T55398 C9IS5M 136983815 IC50 = 121 nM T55398 C9V3KL 136983853 IC50 = 258 nM T55398 CHT7X2 136983871 IC50 = 352 nM T55398 C24BNM 136983876 IC50 = 635 nM T55398 C39FNY 136983894 IC50 = 36 nM T55398 CWL74T 136983918 IC50 = 354 nM T55398 CSJI86 136983949 IC50 = 620 nM T55398 C3R0PB 136984063 IC50 = 450 nM T55398 C5KN9F 136984064 IC50 = 100 nM T55398 CH3M4B 137083628 IC50 > 30000 nM T55398 CJA07O 137083629 IC50 > 30000 nM T55398 C9F8PX 137083630 IC50 = 579 nM T55398 C96CJQ 137348875 IC50 = 360 nM T55398 C8GD6Y 137367179 IC50 = 0.47 nM T55398 CT2FE0 137367190 IC50 = 0.11 nM T55398 C52UFH 137367200 Ki = 210 nM T55398 C3PBN7 137367378 IC50 = 0.026 nM T55398 CZ4VW3 137631374 IC50 = 21 nM T55398 C0U4AO 137631449 IC50 = 10 nM T55398 CN32XA 137631833 IC50 = 82 nM T55398 C90ELI 137631990 IC50 = 730 nM T55398 CSVD52 137632007 IC50 = 20 nM T55398 C0OWI4 137632095 IC50 = 3 nM T55398 CQU8G7 137632864 IC50 = 33 nM T55398 CZH08K 137633516 IC50 = 180 nM T55398 CC9IU4 137634304 IC50 = 5 nM T55398 CYEO71 137634466 IC50 = 5 nM T55398 CQR3H5 137634670 IC50 = 140 nM T55398 CXG74K 137635345 IC50 = 50 nM T55398 CY6TH8 137635761 IC50 = 4.571 nM T55398 CJE35M 137636090 IC50 = 20 nM T55398 C8Z9VW 137637011 IC50 = 3 nM T55398 C1KWC2 137637354 IC50 = 99 nM T55398 CPEI56 137637758 IC50 = 16 nM T55398 CE8AB3 137639678 IC50 = 400 nM T55398 CB6GD5 137639959 IC50 = 47 nM T55398 CB0JI5 137640711 IC50 = 2000 nM T55398 CO1MS6 137641896 IC50 = 14600 nM T55398 CY9QE7 137642189 IC50 = 4.786 nM T55398 CA9DE5 137642519 IC50 = 390 nM T55398 CP6K0U 137642747 IC50 = 120 nM T55398 C47KFJ 137642928 IC50 = 4 nM T55398 C1BK8H 137643835 IC50 = 9 nM T55398 CBA59R 137644862 IC50 = 1300 nM T55398 CP74MV 137644945 IC50 = 75 nM T55398 C7KHW3 137645090 IC50 = 410 nM T55398 CXIN67 137645231 IC50 = 58 nM T55398 C0GYU1 137646905 IC50 = 8 nM T55398 CGU2E5 137648767 IC50 = 840 nM T55398 CQHO93 137649163 IC50 = 3 nM T55398 CBY15N 137649190 IC50 = 56 nM T55398 CX8N6D 137650526 IC50 = 13 nM T55398 C98RIA 137651604 IC50 = 270 nM T55398 C0RUL8 137651621 IC50 = 10 nM T55398 CFX6Y3 137651671 IC50 = 13 nM T55398 C5NUY0 137651713 IC50 = 25 nM T55398 C7BJN4 137652293 IC50 = 170 nM T55398 C5CKI4 137652730 IC50 = 64 nM T55398 CAFG38 137653032 IC50 = 630.96 nM T55398 C8UGS4 137653281 IC50 = 50 nM T55398 CQT9B3 137653599 IC50 = 13 nM T55398 CS6RE8 137654629 IC50 = 50 nM T55398 CNIX25 137655529 IC50 = 1600 nM T55398 C27SVK 137656133 IC50 = 11 nM T55398 CR8Z9G 137656476 IC50 = 2087 nM T55398 CQ0GX8 137657147 IC50 = 40 nM T55398 CLW29O 137657406 IC50 = 9000 nM T55398 C49DOZ 137657630 IC50 = 19 nM T55398 CXS2U8 137658175 IC50 = 34 nM T55398 CO6XD2 137658443 IC50 = 22 nM T55398 CU0ST8 137659008 IC50 = 130 nM T55398 C6Z8YN 137659188 IC50 = 70 nM T55398 CB1XR5 137659870 IC50 = 4 nM T55398 CMZ36T 137659999 IC50 = 730 nM T55398 CK1B4W 137660846 IC50 = 6 nM T55398 CM23OE 137661767 IC50 = 44 nM T55398 CJ0G3C 138376590 Ki = 1.8 nM T55398 CX64WE 138620530 IC50 < 30 nM T55398 C2LHE0 138620547 IC50 < 30 nM T55398 CA63ML 138620560 IC50 < 30 nM T55398 CR0Y8I 138656676 IC50 < 30 nM T55398 CA1I4Y 138656977 IC50 < 30 nM T55398 C72APW 138727769 IC50 = 97.72 nM T55398 C5J2WV 138728749 IC50 = 94 nM T55398 CVU63L 139582016 IC50 = 37 nM T55398 C8PH9S 139582017 IC50 = 4 nM T55398 C45PVO 142501440 Ki = 22 nM T55398 CU12BZ 142501542 IC50 = 0.1 nM T55398 CV1KM9 145979754 IC50 = 77.62 nM T55398 CX05ZN 145979845 IC50 = 22 nM T55398 CY9X5Q 145979885 IC50 = 1190 nM T55398 C9N2XW 145980788 IC50 = 19.5 nM T55398 CNQ67H 145987089 IC50 = 207 nM T55398 C1N9LZ 145987466 IC50 = 446 nM T55398 C9O6WH 145987619 IC50 = 1530 nM T55398 C4QX5P 145987677 IC50 = 44.67 nM T55398 CYS4V9 145990152 IC50 = 234.42 nM T55398 C3T6XI 145991666 IC50 = 1770 nM T55398 CEL5Y6 145991871 IC50 = 738 nM T55398 CP15XW 145992518 IC50 = 33 nM T55398 CSHF19 145992913 IC50 = 602.56 nM T55398 C1N8CA 145993210 IC50 = 671 nM T55398 C12VLN 145993338 IC50 = 87.1 nM T55398 CE9PV2 145993467 IC50 > 10000 nM T55398 CT74QG 145993512 IC50 = 4073.8 nM T55398 C2B4VW 145993656 IC50 = 42 nM T55398 C5H2WU 145993757 IC50 = 16 nM T55398 CHT23F 145993921 IC50 = 804 nM T55398 C6PK4L 146483027 IC50 = 0.078 nM T55398 CMZ4J3 155510495 IC50 < 30 nM T55398 CHX57D 155511560 Ki = 95 nM T55398 CKB64L 155512869 IC50 = 69 nM T55398 C2MD1Q 155513187 IC50 > 10000 nM T55398 C93SNT 155514207 IC50 = 1 nM T55398 C17BHJ 155516763 IC50 = 0.022 nM T55398 C08VAM 155517957 IC50 = 2.5 nM T55398 C8UI7G 155520013 IC50 = 0.29 nM T55398 CCL0S9 155520435 IC50 = 0.099 nM T55398 C7YSD8 155522882 IC50 > 5000 nM T55398 C70GEI 155525183 IC50 > 5000 nM T55398 CWP05R 155527255 Ki = 1.7 nM T55398 CE2YX6 155527737 Ki = 290 nM T55398 CSGV07 155529499 Ki > 8400 nM T55398 CA83QP 155529897 IC50 > 5000 nM T55398 CGDE18 155530136 IC50 > 5000 nM T55398 CSJB85 155530835 Ki = 0.5 nM T55398 CWU8N1 155535119 IC50 = 38 nM T55398 CL5F3C 155537218 Ki = 0.5 nM T55398 CG4LQ2 155539650 Ki = 1.2 nM T55398 C29FDV 155542370 IC50 = 9 nM T55398 C8NOD0 155544794 Ki > 30000 nM T55398 CX9FM8 155548286 IC50 = 2.1 nM T55398 CSJ72Y 155549539 IC50 = 6 nM T55398 CR79JM 155549965 IC50 = 1 nM T55398 CN6O2U 155552158 IC50 > 5000 nM T55398 CM8O9G 155552851 Ki = 170 nM T55398 CWO25P 155555362 Ki = 26 nM T55398 C4Y6BV 155556454 Ki = 6.7 nM T55398 C0WUZ4 155556888 IC50 = 5 nM T55398 C8NMG3 155558108 IC50 > 5000 nM T55398 CWJ08R 155560232 Ki = 0.8 nM T55398 C4IP2Y 155561648 IC50 = 17 nM T55398 C0EBX7 155561943 IC50 = 279 nM T55398 C3D2GP 155562155 IC50 = 21 nM T55398 D00ERW 44444843 Ki > 9921 nM T55398 D00HVA 11624601 Ki > 9900 nM T55398 D02JIL 3572750 IC50 = 4000 nM T55398 D04CFM 86343751 Ki = 1 nM T55398 D04ZIV 58056241 IC50 = 1 nM T55398 D06HVH 54613583 IC50 > 10000 nM T55398 D06WGX 9549184 IC50 > 25000 nM T55398 D09JUD 44449334 IC50 = 20 nM T55398 D0I2FZ 11983295 IC50 = 200 nM T55398 D0J3LR 11634725 Ki > 4000 nM T55398 D0J8VR 25169383 IC50 = 1 nM T55398 D0LY5S 2635761 IC50 = 13600 nM T55398 D0ME9B 46868971 IC50 = 1800 nM T55398 D0Q3NG 11715520 Ki > 9900 nM T55398 D0S7IE 11658882 Ki > 9900 nM T55398 D0T2NE 58056092 IC50 = 8 nM T55398 D0Y2ZC 68115559 IC50 = 7.5 nM T66505 D03EDQ 24776445 IC50 = 5.1 nM T66505 D03LWG 53235510 Ki = 46.5 nM T66505 D04MXN 56846693 Ki = 187.8 nM T66505 D08FDX 24901704 Ki = 41.7 nM T66505 D09BNZ 24775005 Ki = 6 nM T66505 D09UMN 45100669 IC50 < 100 nM T66505 D0D1GF 42642645 Ki = 59.7 nM T66505 D0GD4Q 25027363 IC50 = 1.4 nM T66505 D0M9QZ 11485656 Ki = 87.6 nM T66505 C5V3DJ 1048811 Ki = 50.4 nM T66505 CBVR03 1139102 IC50 = 281 nM T66505 C5W4RP 1300425 IC50 = 89 nM T66505 C0MHW2 2270563 IC50 = 109 nM T66505 C80TKI 2952255 IC50 = 4.4 nM T66505 CFWS91 2953198 IC50 = 91 nM T66505 C1FQR3 3537781 IC50 = 13 nM T66505 CVOH96 3591787 IC50 > 2500 nM T66505 C0LY1H 4269048 Ki = 168.1 nM T66505 CB9I0U 5284329 IC50 = 1500 nM T66505 CK73QZ 6405276 IC50 = 13 nM T66505 CEA26I 6407374 IC50 = 19 nM T66505 C8UB6G 6878030 IC50 = 4.74 nM T66505 CR4Z0H 8440567 IC50 = 1860 nM T66505 C2MJB3 9869236 IC50 = 3420 nM T66505 CLH27B 10392802 IC50 = 140 nM T66505 C1IZR8 10951208 IC50 = 120 nM T66505 CL4BI2 11762419 IC50 = 7520 nM T66505 C2JYM1 18526613 IC50 = 1243 nM T66505 CKU1F2 20875737 IC50 > 5000 nM T66505 C4C9WL 22291085 IC50 = 450 nM T66505 CK6P2Z 24797888 IC50 = 170 nM T66505 CY69VQ 24797889 IC50 = 10 nM T66505 C16WVQ 24797980 IC50 = 240 nM T66505 CZ3EV7 24798071 IC50 = 120 nM T66505 CKYJ26 24905375 IC50 = 8 nM T66505 CN97YF 25065064 IC50 = 724 nM T66505 CEJT74 25065069 IC50 = 2261 nM T66505 CV3R7X 25065678 IC50 = 34 nM T66505 C24YFH 25065681 IC50 = 82 nM T66505 C0HPL9 25065893 IC50 = 185 nM T66505 CJ68BR 25065894 IC50 = 196 nM T66505 CC90KI 25066322 IC50 > 5000 nM T66505 C5UGO6 25066518 IC50 = 112 nM T66505 CGI08J 25066520 IC50 = 95 nM T66505 CYL6V4 25067132 IC50 = 391 nM T66505 CEA5R6 25181471 IC50 < 6 nM T66505 CVPH81 25210551 IC50 = 2700 nM T66505 CI6VC1 25211577 IC50 = 7 nM T66505 CUWT70 25211578 IC50 = 7 nM T66505 CJPE39 25211677 IC50 = 770 nM T66505 CJ0C6Z 25224531 IC50 = 16 nM T66505 C2GBS5 25224707 IC50 = 66 nM T66505 CNX9T4 25226761 IC50 = 1 nM T66505 CUL3B0 25226762 IC50 = 5.8 nM T66505 CCP60F 25226764 IC50 = 12 nM T66505 CC7GX8 25253556 IC50 < 12 nM T66505 C7WZY2 25255940 IC50 = 2.8 nM T66505 CR63VO 44186114 IC50 > 5000 nM T66505 CAU96H 44186115 IC50 = 59 nM T66505 C8I5FZ 44186181 IC50 = 217 nM T66505 CB7K3J 44186182 IC50 > 5000 nM T66505 CBQD07 44186183 IC50 > 5000 nM T66505 C8OLT2 44186184 IC50 = 401 nM T66505 C2EIF1 44186185 IC50 = 230 nM T66505 C9ROY5 44186310 IC50 = 306 nM T66505 CM4SK2 44186312 IC50 = 654 nM T66505 CB5US1 44186313 IC50 = 15 nM T66505 CGR97M 44186314 IC50 = 484 nM T66505 CQ58TU 44186375 IC50 = 67 nM T66505 CJD40V 44186376 IC50 = 21 nM T66505 C3QDF2 44186378 IC50 = 70 nM T66505 CS96ZI 44186429 IC50 = 103 nM T66505 C0L4ES 44186430 IC50 = 25 nM T66505 C1PTH6 44186431 IC50 = 2929 nM T66505 CM8H5Z 44186480 IC50 = 34 nM T66505 C31RVS 44186482 IC50 = 17 nM T66505 C8Z1DQ 44186485 IC50 > 5000 nM T66505 CQT23O 44186526 IC50 > 5000 nM T66505 C6BD5U 44250034 IC50 = 5 nM T66505 CZTH83 44250105 IC50 = 40 nM T66505 C8H9TQ 44395035 IC50 = 3200 nM T66505 C0T2GL 44395101 IC50 = 1100 nM T66505 CY9R4E 44395109 IC50 = 450 nM T66505 C0MT1L 44395257 IC50 > 3000 nM T66505 CF9IW1 44412191 IC50 = 78.4 nM T66505 C1NF9R 44463317 IC50 = 90 nM T66505 CT14KB 44464376 IC50 = 190 nM T66505 CE7J2C 44464620 IC50 = 107 nM T66505 CYJ02G 44464875 IC50 = 80 nM T66505 CYLN29 44517800 IC50 = 31 nM T66505 C3O7TI 44548374 IC50 = 44 nM T66505 C7CJM3 44548378 IC50 = 93 nM T66505 CY9M7W 44549004 IC50 = 40 nM T66505 CRT70E 44591268 IC50 = 30 nM T66505 CQE8H0 44591290 IC50 = 790 nM T66505 C7ZX3O 44591292 IC50 = 1150 nM T66505 C5VUK4 44591325 IC50 = 14 nM T66505 CF1E9T 44591326 IC50 = 340 nM T66505 CVB19K 44591344 IC50 = 32 nM T66505 CMR54E 44591345 IC50 = 55 nM T66505 CPW59G 44591346 IC50 = 210 nM T66505 CO31UZ 44591347 IC50 = 130 nM T66505 CZ2C0W 44610687 IC50 = 380 nM T66505 C4U9EN 44628220 IC50 = 3400 nM T66505 CKM92Y 44628222 IC50 = 2200 nM T66505 CO72KB 44628287 IC50 = 1100 nM T66505 C0YM5V 44628288 IC50 = 1500 nM T66505 CV9A3W 44628450 IC50 = 1200 nM T66505 CMA16F 44628452 IC50 = 1500 nM T66505 CAW8Y9 44628525 IC50 = 320 nM T66505 CK0G2O 44628528 IC50 = 1800 nM T66505 CZY63O 44628618 IC50 = 420 nM T66505 C62FGB 44628620 IC50 = 1300 nM T66505 CPG83O 44628898 IC50 > 2500 nM T66505 CS37ZL 44629065 IC50 = 790 nM T66505 CEX0I1 44629066 IC50 = 1000 nM T66505 CVS96Z 44629067 IC50 = 280 nM T66505 CL9N4Z 44629071 IC50 = 520 nM T66505 CER8Q0 44629155 IC50 = 470 nM T66505 C8XGK2 44629232 IC50 = 510 nM T66505 CDQ47G 44629236 IC50 = 700 nM T66505 CGW6U0 44629295 IC50 = 750 nM T66505 CX1QC4 44629366 IC50 > 2500 nM T66505 CE6B2G 45267515 IC50 = 130 nM T66505 CF8VX0 45267523 IC50 > 10000 nM T66505 CUW4Z0 45267528 IC50 = 70 nM T66505 C0Z3MB 45267540 IC50 = 1800 nM T66505 CUM1G5 45268389 IC50 = 10000 nM T66505 CYU5Q0 45268404 IC50 = 310 nM T66505 CC7H9M 45268408 IC50 = 200 nM T66505 C9VCH6 45268412 IC50 = 100 nM T66505 CS90AD 45269254 IC50 = 3000 nM T66505 CHCB29 45269261 IC50 = 900 nM T66505 CH3NB9 45269264 IC50 = 950 nM T66505 CD0FN3 45270098 IC50 = 1200 nM T66505 CI16LK 45270102 IC50 = 360 nM T66505 CKNH75 45270116 IC50 = 130 nM T66505 CH2F3N 45270117 IC50 > 25000 nM T66505 CRO2M3 45270118 IC50 = 6300 nM T66505 C3PTM6 45270935 IC50 = 720 nM T66505 CN2F0B 45270940 IC50 = 900 nM T66505 CI95MH 45270943 IC50 = 200 nM T66505 C29UPR 45270944 IC50 = 120 nM T66505 CDV71Y 45270956 IC50 = 1400 nM T66505 CGYD64 45271780 IC50 = 10000 nM T66505 CQ9K4Y 45271789 IC50 = 1300 nM T66505 CF12YU 45271790 IC50 = 1200 nM T66505 C2P1MF 45272645 IC50 = 10000 nM T66505 CL1S7X 45272649 IC50 = 10000 nM T66505 CL91PA 45272656 IC50 = 680 nM T66505 CGO7B5 45272667 IC50 > 10000 nM T66505 CB6S7D 45272668 IC50 = 1830 nM T66505 C3C1DS 45273570 IC50 = 330 nM T66505 CES8O2 45273586 IC50 = 150 nM T66505 C1B4AO 45273591 IC50 = 4500 nM T66505 CIQ7M3 45273599 IC50 = 340 nM T66505 CK7XM8 46871826 IC50 = 5.3 nM T66505 CP87LJ 46871827 IC50 = 2.2 nM T66505 CT8FV6 46890873 IC50 = 9.5 nM T66505 CXY13W 46890935 IC50 = 13 nM T66505 C1CIG5 46890990 IC50 = 5.3 nM T66505 CVBK65 46890991 IC50 = 17.3 nM T66505 CIZ8O7 46890992 IC50 = 5.2 nM T66505 C4GR0D 46891044 IC50 = 15 nM T66505 CMT7B2 46891045 IC50 = 10.8 nM T66505 CH1K0L 46891046 IC50 = 20 nM T66505 CY0T2V 46891103 IC50 = 212 nM T66505 CY0A3H 46891104 IC50 = 15 nM T66505 CRW3N1 46891105 IC50 = 20.3 nM T66505 C1V4PY 46891106 IC50 = 110 nM T66505 C2JRG0 46891162 IC50 = 213 nM T66505 C1PC7R 46891163 IC50 = 96 nM T66505 CK6RY3 46891164 IC50 = 3.2 nM T66505 CE46PC 46891165 IC50 = 7 nM T66505 C1JFY6 46891197 IC50 = 11.8 nM T66505 CHQ06G 46891198 IC50 = 3.6 nM T66505 CAYC57 46891199 IC50 = 0.7 nM T66505 CLD87G 46891200 IC50 = 0.4 nM T66505 CVK3A7 46891245 IC50 = 2.3 nM T66505 CQCN85 46891246 IC50 = 7.3 nM T66505 C0NF6E 46891247 IC50 = 10.1 nM T66505 CY89AF 46891248 IC50 = 2.7 nM T66505 C7D9UV 46891298 IC50 = 3.1 nM T66505 CH03ZS 46891299 IC50 = 5.2 nM T66505 CV6MN7 46891300 IC50 = 2340 nM T66505 C59RFZ 46891346 IC50 = 2700 nM T66505 C24DXJ 49840814 IC50 = 4 nM T66505 C2O7ZC 49862152 IC50 = 1870 nM T66505 C9AQO8 49862153 IC50 = 1690 nM T66505 C0AY1M 49862154 IC50 = 20 nM T66505 CSR2H4 49862176 IC50 = 12 nM T66505 CPNL82 49862194 IC50 > 5000 nM T66505 CN0V7S 49862195 IC50 > 5000 nM T66505 CFNZ30 49862196 IC50 = 333 nM T66505 C06TVH 49862197 IC50 = 105 nM T66505 C7H2NL 49862220 IC50 = 19 nM T66505 C0U7CJ 49862221 IC50 = 21 nM T66505 CIUH50 49862222 IC50 > 1000 nM T66505 CZ8GI9 49862236 IC50 = 64.7 nM T66505 C6OQV2 49862237 IC50 = 40.8 nM T66505 C6IW4Q 49862238 IC50 = 8.27 nM T66505 CP1YK8 49862269 IC50 = 3.3 nM T66505 C4HRQ3 49862270 IC50 = 4.8 nM T66505 CCL25Y 49862311 IC50 = 25 nM T66505 C16VMC 49862312 IC50 = 79 nM T66505 C7H5LT 49862313 IC50 = 57 nM T66505 C1J9KL 49862314 IC50 = 8.7 nM T66505 CI0Q6T 49862371 IC50 = 8 nM T66505 C8GS6K 49862372 IC50 > 1000 nM T66505 CB10HZ 49862373 IC50 > 1000 nM T66505 C4FYZ5 49862424 IC50 > 1000 nM T66505 C3QF1T 50768213 IC50 > 2500 nM T66505 CXN52T 50835422 IC50 = 63 nM T66505 CRZL59 53361076 IC50 = 13 nM T66505 C0CE7M 53387030 IC50 = 13 nM T66505 C1RHF7 53387681 IC50 = 5 nM T66505 CTY6C4 53484000 IC50 = 7.2 nM T66505 C13WTO 56658050 IC50 = 46 nM T66505 C8GZD4 56658051 IC50 = 2600 nM T66505 CT62BA 56658169 IC50 = 230 nM T66505 CJDL15 56658170 IC50 = 2000 nM T66505 C30TCQ 56658188 IC50 = 6.4 nM T66505 CV68SR 56658189 IC50 = 48 nM T66505 CL38IE 56658549 IC50 = 180 nM T66505 C4U7WK 56658550 IC50 = 4700 nM T66505 C0G4XL 56658551 IC50 > 2500 nM T66505 C7MBL0 56658552 IC50 > 2500 nM T66505 C75ITF 56658553 IC50 > 2500 nM T66505 C1SH5E 56658575 IC50 = 480 nM T66505 CV2EY4 56658696 IC50 > 2500 nM T66505 CA9KM7 56658697 IC50 = 480 nM T66505 CV6T7E 56658698 IC50 > 2500 nM T66505 CW72LF 56658699 IC50 > 2500 nM T66505 CCA76B 56661560 IC50 = 46 nM T66505 C4H3VZ 56661561 IC50 = 340 nM T66505 CRI23C 56661562 IC50 = 64 nM T66505 C43ICJ 56661679 IC50 = 72 nM T66505 C8D9PR 56662002 IC50 = 15000 nM T66505 C35SAR 56662003 IC50 = 620 nM T66505 CG2U1T 56662004 IC50 = 1000 nM T66505 C9BNK7 56662005 IC50 = 1900 nM T66505 CY26QZ 56662006 IC50 > 2500 nM T66505 CQ41MY 56662174 IC50 = 110 nM T66505 CB4W0O 56662175 IC50 > 2500 nM T66505 CVSD83 56662176 IC50 = 670 nM T66505 C8E5BX 56662793 IC50 = 18 nM T66505 C3PKE1 56663266 IC50 = 3000 nM T66505 CM2O8C 56664980 IC50 = 330 nM T66505 C92THJ 56664981 IC50 = 380 nM T66505 C1ME2L 56665113 IC50 = 37 nM T66505 CAY4Z3 56665494 IC50 = 640 nM T66505 CT9O7X 56665495 IC50 = 6000 nM T66505 CWCK98 56665496 IC50 > 2500 nM T66505 C41XMQ 56665497 IC50 = 2200 nM T66505 CG75HU 56665498 IC50 > 2500 nM T66505 CKA36R 56665499 IC50 > 2500 nM T66505 CKB71O 56665632 IC50 > 2500 nM T66505 CMJ13X 56666699 IC50 = 4600 nM T66505 CX4IC9 56668414 IC50 = 200 nM T66505 CX8Q5Y 56668540 IC50 = 13000 nM T66505 CUFX01 56668541 IC50 = 240 nM T66505 CF7LR5 56668542 IC50 = 32 nM T66505 CI4Q1R 56668557 IC50 = 49 nM T66505 C6KVX4 56668558 IC50 = 27 nM T66505 C2DR5K 56668559 IC50 = 27 nM T66505 CU19OY 56668560 IC50 = 93 nM T66505 CG6JS7 56668711 IC50 = 810 nM T66505 C8W4QB 56668923 IC50 > 2500 nM T66505 CP9U0G 56668924 IC50 = 1000 nM T66505 C02GYK 56668936 IC50 = 45 nM T66505 CMQS94 56669087 IC50 = 1900 nM T66505 C5W8BE 56669674 IC50 = 140 nM T66505 CQJ72G 56669675 IC50 = 100 nM T66505 C51HRV 56669676 IC50 = 15 nM T66505 CR9IJ2 56669677 IC50 = 21 nM T66505 C3IE7S 56671926 IC50 = 530 nM T66505 CYOA69 56671927 IC50 = 390 nM T66505 C5RFI6 56671928 IC50 = 19 nM T66505 CTL7J0 56671929 IC50 = 8 nM T66505 C68YBP 56672043 IC50 = 4900 nM T66505 C4XK3V 56672054 IC50 = 14 nM T66505 CVCW54 56672401 IC50 > 2500 nM T66505 C8CMQ3 56672402 IC50 = 1100 nM T66505 C67POD 56672403 IC50 > 2500 nM T66505 C60FCS 56672404 IC50 > 2500 nM T66505 CK8Y7L 56672544 IC50 = 490 nM T66505 CY8Q6Z 56672545 IC50 = 750 nM T66505 C9O6JQ 56672546 IC50 = 2900 nM T66505 CP0J8E 56672547 IC50 = 1300 nM T66505 COI7L2 56673182 IC50 = 1200 nM T66505 CI9QV5 56675303 IC50 = 790 nM T66505 CO4ND2 56675304 IC50 = 510 nM T66505 CKXE70 56675305 IC50 = 2700 nM T66505 CTE98L 56675306 IC50 = 17000 nM T66505 C5O7WK 56675307 IC50 = 290 nM T66505 CWI58T 56675308 IC50 = 15 nM T66505 CI06FK 56675419 IC50 = 6900 nM T66505 CJEA89 56675420 IC50 = 290 nM T66505 CK57CI 56675440 IC50 = 28 nM T66505 CM5UH2 56675441 IC50 = 33 nM T66505 CY6UA5 56675678 IC50 > 2500 nM T66505 C9C8FG 56675786 IC50 > 2500 nM T66505 CAI9O3 56675787 IC50 > 2500 nM T66505 CSA35C 56675788 IC50 > 2500 nM T66505 CMKQ61 56675800 IC50 = 1600 nM T66505 CK6GW1 56675801 IC50 = 350 nM T66505 CF2GB3 56675802 IC50 = 3 nM T66505 C6IU9P 56675925 IC50 > 2500 nM T66505 CF3R6A 56675926 IC50 = 1500 nM T66505 C04FDY 56675927 IC50 = 2500 nM T66505 C5I4KA 56676509 IC50 = 21 nM T66505 C6RVC4 56676510 IC50 = 230 nM T66505 C41FSK 56676511 IC50 = 19 nM T66505 CO9AX8 56678641 IC50 = 46 nM T66505 CBZ1S6 56678642 IC50 = 180 nM T66505 CL9V4G 56678643 IC50 = 360 nM T66505 CEI80K 56678644 IC50 = 15 nM T66505 CZ9LW6 56678777 IC50 = 79 nM T66505 CWMH38 56679102 IC50 > 2500 nM T66505 CKN39Z 56679103 IC50 > 2500 nM T66505 C0DV4W 56679122 IC50 = 1800 nM T66505 C07JIH 56679237 IC50 > 2500 nM T66505 CR19BZ 56679238 IC50 = 350 nM T66505 C3MI4V 56679239 IC50 = 1700 nM T66505 CC81YD 56679828 IC50 = 430 nM T66505 C03JCI 56679829 IC50 = 1400 nM T66505 CI6UC5 56680279 IC50 = 7800 nM T66505 CDR92Q 56680280 IC50 = 5100 nM T66505 C06HAF 56681960 IC50 = 370 nM T66505 CS30BK 56681961 IC50 = 16 nM T66505 C1Y0MO 56682216 IC50 = 30 nM T66505 CPRT14 56682402 IC50 = 2100 nM T66505 C07GSV 56682403 IC50 > 2500 nM T66505 CDH41P 56682417 IC50 = 760 nM T66505 CGCH03 56682418 IC50 = 25 nM T66505 C3F6TH 56682550 IC50 = 220 nM T66505 CH46PS 56682551 IC50 = 1400 nM T66505 C7BX5M 56682552 IC50 = 340 nM T66505 CN4RZ3 56682553 IC50 = 280 nM T66505 C3L5PZ 56682554 IC50 > 2500 nM T66505 C14GVW 56683156 IC50 = 140 nM T66505 CV85DJ 56683157 IC50 = 42 nM T66505 C6F7RL 56683158 IC50 = 12 nM T66505 C32GXL 56964691 IC50 = 24 nM T66505 C2Q8VL 56964692 IC50 = 41 nM T66505 C27ION 57326206 IC50 = 100 nM T66505 CRJ90X 57326301 IC50 = 180 nM T66505 CH96BW 57326302 IC50 = 820 nM T66505 CL8H5N 57326385 IC50 = 1100 nM T66505 C7SI0M 57326387 IC50 = 29 nM T66505 C61TYN 57326482 IC50 = 130 nM T66505 CF4X2S 57326483 IC50 = 520 nM T66505 CMI5L4 57326484 IC50 = 1800 nM T66505 C32LFE 67374618 IC50 < 16 nM T66505 C46VLA 67374621 EC50 = 15 nM T66505 CLKN38 67375395 IC50 < 19 nM T66505 C5BFR4 67378301 EC50 = 115 nM T66505 CKB37H 67379186 IC50 < 40 nM T66505 C8M9VH 67379418 EC50 = 28 nM T66505 C07NTU 68747277 IC50 = 42 nM T66505 CD9J0Y 68778068 EC50 = 30 nM T66505 CG16HX 68780878 EC50 = 7 nM T66505 CMGA79 70682196 EC50 = 27 nM T66505 CH0T3O 70684298 EC50 = 89 nM T66505 CTCF71 70688555 EC50 = 22 nM T66505 C1Y7FR 70688556 IC50 > 450 nM T66505 CNER46 70690618 EC50 = 21 nM T66505 CTYA67 70692760 EC50 = 8 nM T66505 CFYG52 70694242 IC50 = 110 nM T66505 C45SUB 70694800 EC50 = 17 nM T66505 C95IBJ 70694801 EC50 = 40 nM T66505 C2SWX1 70696850 EC50 = 29 nM T66505 CO58QT 71458712 Ki = 37.9 nM T66505 C0J3TE 76311001 IC50 = 300 nM T66505 C89CXE 76311004 IC50 = 40 nM T66505 CWZE58 76318208 IC50 = 100 nM T66505 C6H5MS 76848956 Ki = 30 nM T66505 C53NWC 86294818 IC50 = 87 nM T66505 CM0A5R 90286184 IC50 = 1800 nM T66505 CIU6F5 90286320 IC50 = 4100 nM T66505 CJ85YQ 90286388 IC50 > 10000 nM T66505 CW6BO1 90286529 IC50 = 910 nM T66505 C0YEV1 90286574 IC50 = 270 nM T66505 C89TEO 90299606 IC50 = 890 nM T66505 C5V3LH 90299611 IC50 = 350 nM T66505 C7LTZ2 90299612 IC50 = 300 nM T66505 C2UV3X 90299614 IC50 = 440 nM T66505 CZ1GP2 90299621 IC50 = 1300 nM T66505 CKD1F0 90299647 IC50 = 690 nM T66505 CFHB98 90644096 IC50 > 25000 nM T66505 CWK6N7 90656290 IC50 = 2700 nM T66505 CK2I6N 90656291 IC50 = 520 nM T66505 CRI41W 90656292 IC50 = 4100 nM T66505 CL29HQ 90656293 IC50 = 790 nM T66505 CD2PB6 90656294 IC50 > 10000 nM T66505 CS8TB7 90656295 IC50 > 10000 nM T66505 CWL3E0 90656296 IC50 = 550 nM T66505 CW7BV0 90656297 IC50 = 1200 nM T66505 CU4NV3 90656298 IC50 = 1500 nM T66505 CP36FA 90656299 IC50 = 420 nM T66505 C6F9NY 90656300 IC50 = 270 nM T66505 COK94Z 90656301 IC50 = 200 nM T66505 CRG6J5 90656302 IC50 = 380 nM T66505 CR4K2D 90656303 IC50 = 270 nM T66505 C9ZU3G 90656304 IC50 = 740 nM T66505 CI7F1H 90656305 IC50 = 960 nM T66505 CVH8R7 90656306 IC50 = 650 nM T66505 C9WDS7 97046899 Ki = 33 nM T66505 CM7LD8 122185868 IC50 = 5.6 nM T66505 CL0ZB6 122185870 IC50 = 10 nM T66505 C9CZ8G 127039132 IC50 = 19 nM T66505 CDVZ38 127039452 IC50 = 42 nM T66505 CILZ74 127048425 IC50 = 373 nM T66505 C0CF8P 127048730 IC50 = 294 nM T66505 C87LZN 127048731 IC50 = 315 nM T66505 C43IVQ 127048732 IC50 = 18 nM T66505 C38MXE 127048733 IC50 = 192 nM T66505 CS57TL 127048734 IC50 = 135 nM T66505 CDT1A0 127049057 IC50 = 352 nM T66505 C92DBP 127049409 IC50 = 326 nM T66505 C8NO0A 127051279 IC50 = 261 nM T66505 CWT20F 127052154 IC50 = 431 nM T66505 CKM9A3 127052181 IC50 = 217 nM T66505 CP7S9A 127052483 IC50 = 92 nM T66505 CCQ86W 127052484 IC50 = 213 nM T66505 C6LU2S 127052485 IC50 = 56 nM T66505 C2CA0W 127053107 IC50 = 456 nM T66505 C2SAG7 127053109 IC50 = 237 nM T66505 CXI0B3 132578555 IC50 > 10000 nM T66505 CY0BT9 136210502 IC50 = 290 nM T66505 CX67HE 136210503 IC50 = 370 nM T66505 CKP6L1 136210504 IC50 = 70 nM T66505 CL47YD 136210505 IC50 = 220 nM T66505 CE1US4 136210506 IC50 = 70 nM T66505 C7OW0J 136210508 IC50 = 160 nM T66505 CL4IW7 136210509 IC50 = 190 nM T66505 CDFZ95 136210510 IC50 = 33 nM T66505 CKS3V1 136210511 IC50 = 5 nM T66505 CKO48T 136210512 IC50 = 110 nM T66505 CE9OD5 136210517 IC50 = 900 nM T66505 CB7AI4 136210518 IC50 = 14 nM T66505 C0TI5R 136244207 IC50 = 640 nM T66505 C9C5MY 145958866 IC50 = 10 nM T66505 CJ8X4A 155515079 Ki = 55 nM T66505 COKI80 155515124 IC50 = 3.9 nM T66505 CTO9C8 155547338 IC50 = 18 nM T66505 CRG7H3 155549835 Ki = 45 nM T66505 C95DIM 155559226 Ki = 28 nM T66505 D03NPX 447077 Ki = 46.2 nM T66505 D05UKJ 442972 Ki = 12.7 nM T66505 D0R8DO 6404568 IC50 = 4237 nM T66505 D0S5OU 73729049 IC50 = 440 nM T41201 CGNU14 10408898 IC50 = 350 nM T41201 CZIY89 11081290 IC50 = 25 nM T41201 CQ4EM2 44344844 IC50 = 40 nM T41201 CCA3Z7 44344899 IC50 = 20 nM T41201 CTPO43 44345020 IC50 = 6 nM T41201 C5KH6G 44345023 IC50 = 5 nM T41201 CL6KF8 44345101 IC50 = 150 nM T41201 C6T5UV 44345102 IC50 = 45 nM T41201 CL32RO 44345105 IC50 = 10 nM T41201 C18KAP 44345106 IC50 = 100 nM T78319 CKUJ53 16217499 IC50 = 6700000 nM T78319 C5D3HE 30980948 IC50 = 14100000 nM T78319 CH8Z3J 73441667 IC50 = 3500000 nM T78319 CG0O3E 90655419 IC50 = 1320000 nM T78319 CR5MK9 90655420 IC50 = 108000 nM T78319 C3CNA9 90655421 IC50 = 65000 nM T78319 CF0EX8 90655422 IC50 = 48000 nM T78319 CGL84T 90655423 IC50 = 36000 nM T78319 D03EPY 7046 IC50 = 27000000 nM T43721 D02ENG 6918651 IC50 > 10000 nM T43721 D05WCI 11670435 IC50 > 10000 nM T43721 D0B5HF 44476893 IC50 > 10000 nM T43721 D0O1ZI 25006684 IC50 > 30000 nM T43721 D0R8IU 24946280 IC50 > 30000 nM T43721 D0T8QB 14982 IC50 = 0.4 nM T43721 D07EBU 135565424 IC50 > 10000 nM T43721 D07FHW 23725123 IC50 > 500000 nM T43721 CDM6C4 92730 IC50 = 400 nM T43721 C7JEN0 94320 IC50 = 750 nM T43721 C2O8KM 101788 IC50 = 490 nM T43721 CFG6D1 111253 IC50 = 329 nM T43721 C8UQT9 1484979 IC50 > 10000 nM T43721 C34FUY 2953793 Ki > 10000 nM T43721 C3B7LM 3146235 IC50 = 8900 nM T43721 CPT5Y6 6918663 IC50 > 200000 nM T43721 C84RBQ 9797661 IC50 > 4000 nM T43721 CY2K5B 9823394 IC50 = 4000 nM T43721 CHV1E3 9975108 IC50 > 4000 nM T43721 CSL50G 9975639 IC50 > 4000 nM T43721 CDZ92L 9998483 IC50 > 4000 nM T43721 CBUP07 10018475 IC50 = 1270 nM T43721 C0I6WB 10040175 IC50 = 3318 nM T43721 CU1W4M 10040176 IC50 = 2006 nM T43721 C4L0HV 10043410 IC50 > 4000 nM T43721 CA4SJ7 10064183 IC50 > 4000 nM T43721 C5LKO8 10085885 IC50 = 1035 nM T43721 CW6KU4 10250720 IC50 = 1300 nM T43721 CO0H7A 10250842 IC50 > 4000 nM T43721 COT1X3 10308303 IC50 > 4000 nM T43721 C2LWK5 10315044 IC50 > 4000 nM T43721 C0QH6L 10335644 IC50 > 4000 nM T43721 C7IUQ6 10335880 IC50 > 4000 nM T43721 CI64PJ 10340916 IC50 > 4000 nM T43721 CL5X6K 10355633 IC50 > 4000 nM T43721 CTLN27 10357519 IC50 > 4000 nM T43721 CTU13Q 10357992 IC50 = 503 nM T43721 CWKP54 10359991 IC50 > 4000 nM T43721 CEO4C7 10360107 IC50 = 613 nM T43721 CUL28X 10380007 IC50 < 4000 nM T43721 CF4NL2 10381554 IC50 = 216 nM T43721 CR4V3G 10402262 IC50 > 4000 nM T43721 C65EQT 10403095 IC50 = 1037 nM T43721 CV8K3E 10446474 IC50 = 4000 nM T43721 CQ9X4Y 10446475 IC50 > 4000 nM T43721 CYI70T 10447474 IC50 = 4000 nM T43721 CS06QG 10452320 IC50 > 100000 nM T43721 CA89WN 10470037 IC50 > 4000 nM T43721 C6LJI0 10473292 IC50 > 4000 nM T43721 CXH39G 10474399 IC50 > 4000 nM T43721 C0C6KD 11190936 IC50 = 122 nM T43721 CD3H7R 11232699 IC50 > 200000 nM T43721 C1PKI0 11257147 IC50 > 200000 nM T43721 CW1T5X 11259177 IC50 = 228 nM T43721 CH12WK 11278558 IC50 > 4000 nM T43721 CP9O5R 11280328 IC50 > 200000 nM T43721 CH85OD 11319723 IC50 = 2350 nM T43721 C8FQ9B 11375180 IC50 = 3950 nM T43721 CS0P1Q 11478969 IC50 = 280 nM T43721 CR4I9H 11484764 IC50 = 290 nM T43721 CN08AP 11495851 IC50 > 10000 nM T43721 CLT1Z9 11502804 IC50 = 6300 nM T43721 C76STL 11504178 IC50 = 21000 nM T43721 C19BYP 11505338 IC50 = 50000 nM T43721 CHW7L1 11510573 IC50 > 100000 nM T43721 CE40MU 11524868 IC50 = 550 nM T43721 C8NP4Y 11526147 IC50 = 3 nM T43721 CG1HB5 11533520 IC50 = 24000 nM T43721 CZE42S 11540388 IC50 = 13000 nM T43721 CN1A6F 11540493 IC50 > 100000 nM T43721 C3LVE2 11545617 IC50 = 30000 nM T43721 CD17CO 11551576 IC50 > 10000 nM T43721 CP8L9K 11552169 IC50 = 23000 nM T43721 CCT0Q7 11552781 IC50 = 18000 nM T43721 CA25ZF 11555218 IC50 = 34000 nM T43721 CJ58XB 11576524 IC50 = 25000 nM T43721 CKF3J6 11604308 IC50 = 16000 nM T43721 CGD7X9 11610822 IC50 = 12000 nM T43721 CDL39R 11613794 IC50 > 30000 nM T43721 C7KBZ4 11618761 IC50 = 5500 nM T43721 CW2XN3 11626362 IC50 = 85000 nM T43721 CXS05L 11627334 IC50 > 10000 nM T43721 CMF3U5 11634114 IC50 > 100000 nM T43721 CDL94B 11649095 IC50 > 100000 nM T43721 CX17LY 11654021 IC50 = 1800 nM T43721 C3B4SN 11655097 IC50 > 20000 nM T43721 C1DJ7W 11655188 IC50 = 26000 nM T43721 C1T6KE 11666874 IC50 = 8300 nM T43721 CFH6G5 11670914 IC50 = 20000 nM T43721 CU5TI1 11676805 IC50 > 100000 nM T43721 CJ13XD 11698697 IC50 = 5300 nM T43721 C26ITU 11699075 IC50 = 27000 nM T43721 CK8BF3 11705872 IC50 > 10000 nM T43721 C4D6YM 11712182 IC50 = 60000 nM T43721 C5AT6X 11722880 IC50 = 1961 nM T43721 CO32UM 11724534 IC50 = 1964 nM T43721 C6TPR1 11739354 IC50 > 4000 nM T43721 C4B5XT 11741200 IC50 > 4000 nM T43721 CB9WI2 11742158 IC50 > 4000 nM T43721 C37IRX 11771845 IC50 = 183 nM T43721 C2XW0P 11853305 IC50 = 6040 nM T43721 C4FKP2 13994830 IC50 > 1000000 nM T43721 CEYW48 15953464 IC50 = 2520 nM T43721 CY3A6Q 15987396 IC50 > 10000 nM T43721 C29ACV 15987476 IC50 > 10000 nM T43721 CS1XM4 16049788 IC50 = 100000 nM T43721 C2T4IM 16222378 IC50 = 30.4 nM T43721 C13TPH 16721119 IC50 > 10000 nM T43721 C2OJC1 16726072 IC50 > 10000 nM T43721 C69QUM 20724870 IC50 = 1174 nM T43721 C51LGI 20724898 IC50 > 4000 nM T43721 CP7JM8 20724899 IC50 > 4000 nM T43721 C31VAH 20724901 IC50 > 4000 nM T43721 CJU3T5 20724903 IC50 > 4000 nM T43721 CLX5A8 20724912 IC50 > 4000 nM T43721 CQ6CF3 20755069 IC50 > 4000 nM T43721 CTRD81 20755103 IC50 > 1000 nM T43721 CD1SR0 22591684 IC50 > 4000 nM T43721 CQ6AO5 22591709 IC50 = 7.5 nM T43721 CWF51V 22591726 IC50 > 4000 nM T43721 CEB47A 24744047 IC50 = 21200 nM T43721 CGR84K 24854349 IC50 > 500000 nM T43721 C6BV8N 24854350 IC50 > 500000 nM T43721 CEW31B 24856362 IC50 > 100000 nM T43721 C7QU2Z 24883422 IC50 = 10000 nM T43721 CLYS75 24889741 IC50 = 20 nM T43721 CVD4K7 24889906 IC50 = 15000 nM T43721 C6EFK9 24889907 IC50 > 30000 nM T43721 C5QD7L 24890069 IC50 = 1600 nM T43721 C9XUC0 24890070 IC50 = 1800 nM T43721 C3A9HI 24890073 IC50 = 90000 nM T43721 C6IHL0 24890239 IC50 = 23000 nM T43721 CEV27L 24895554 IC50 > 10000 nM T43721 C8LYV0 24895658 IC50 > 10000 nM T43721 C2QWU0 24895661 IC50 > 10000 nM T43721 C1G6DM 24895969 IC50 > 10 nM T43721 C59MRG 24896012 IC50 > 10 nM T43721 C6UYQ4 24948172 IC50 > 10000 nM T43721 CJL38O 25065024 IC50 > 10000 nM T43721 C8GR2K 25065025 IC50 = 510 nM T43721 CEMG39 25065027 IC50 > 10000 nM T43721 CB36SV 25065227 IC50 > 10000 nM T43721 C7YH6J 25065230 IC50 > 10000 nM T43721 C9EQ1D 25065231 IC50 > 10000 nM T43721 CU12CJ 25065232 IC50 = 10 nM T43721 CEQF65 25210659 IC50 > 100000 nM T43721 CU7E9B 25265683 IC50 > 10000 nM T43721 CMVE89 42603038 IC50 > 10000 nM T43721 C6VQM9 44143289 IC50 > 100000 nM T43721 CZ58CY 44143291 IC50 > 100000 nM T43721 C8X2ZV 44143292 IC50 > 100000 nM T43721 C1IA7U 44143299 IC50 > 100000 nM T43721 C63STN 44196869 IC50 = 31.2 nM T43721 C7YTM0 44197230 IC50 > 4000 nM T43721 CHA7J4 44250316 IC50 > 1000000 nM T43721 C9S2HX 44402393 IC50 > 200000 nM T43721 C8C2QJ 44402534 IC50 > 200000 nM T43721 CW7IP2 44402550 IC50 > 200000 nM T43721 C0NUI2 44402662 IC50 > 200000 nM T43721 C42FXZ 44418375 IC50 > 100000 nM T43721 CC93VQ 44418376 IC50 = 16000 nM T43721 CP9DO4 44418378 IC50 = 52000 nM T43721 CR7K6S 44418382 IC50 > 100000 nM T43721 C7B6GT 44418383 IC50 > 100000 nM T43721 C1Q8CH 44418384 IC50 > 100000 nM T43721 C7JNH9 44418385 IC50 = 100000 nM T43721 CB58SX 44418389 IC50 = 70000 nM T43721 CGKR51 44418390 IC50 = 49000 nM T43721 CQT37N 44418391 IC50 > 100000 nM T43721 CED27U 44418395 IC50 > 100000 nM T43721 C9L7BU 44418396 IC50 > 100000 nM T43721 C28DBM 44418400 IC50 > 100000 nM T43721 C1KD8E 44418401 IC50 > 100000 nM T43721 CT79UX 44418408 IC50 > 100000 nM T43721 C7RW1O 44418409 IC50 > 100000 nM T43721 C7WQD4 44418433 IC50 > 30000 nM T43721 CV87RE 44418434 IC50 > 30000 nM T43721 CK74ZJ 44418441 IC50 > 30000 nM T43721 C02AMZ 44418445 IC50 > 30000 nM T43721 C7YCN4 44418447 IC50 > 100000 nM T43721 C7AKJ2 44418450 IC50 > 100000 nM T43721 C90QWN 44418451 IC50 = 55000 nM T43721 CA2J1I 44418452 IC50 = 11000 nM T43721 CE1W9Y 44418456 IC50 = 90000 nM T43721 C7R3AT 44418457 IC50 > 100000 nM T43721 C4MVN6 44418458 IC50 = 15000 nM T43721 CXFR60 44418459 IC50 = 100000 nM T43721 CAW7Z2 44418817 IC50 > 100000 nM T43721 CC8ZR0 44418821 IC50 > 100000 nM T43721 CKX95Y 44418852 IC50 > 100000 nM T43721 CF56NG 44418856 IC50 = 56000 nM T43721 CGX84K 44418857 IC50 = 62000 nM T43721 CSP8W1 44419286 IC50 > 30000 nM T43721 CQH6X0 44419304 IC50 = 17000 nM T43721 CBI64W 44419309 IC50 = 14000 nM T43721 C6LOU9 44419313 IC50 = 630 nM T43721 C32WUT 44420153 IC50 > 10000 nM T43721 C14JQE 44420164 IC50 > 10000 nM T43721 C76RGZ 44420166 IC50 > 10000 nM T43721 CINJ57 44420180 IC50 > 10000 nM T43721 CWM5F9 44420181 IC50 > 10000 nM T43721 CLA82E 44420186 IC50 > 10000 nM T43721 C0ET3O 44420190 IC50 > 10000 nM T43721 C3JF5Z 44420196 IC50 > 10000 nM T43721 C64UQO 44420202 IC50 > 10000 nM T43721 CJI76N 44420207 IC50 > 10000 nM T43721 C0T6ML 44420212 IC50 > 10000 nM T43721 C5Y4UB 44420215 IC50 > 10000 nM T43721 C1NCR3 44420232 IC50 > 10000 nM T43721 CQ7B8C 44420233 IC50 > 10000 nM T43721 C0X3PE 44420237 IC50 > 10000 nM T43721 CO4S5M 44420238 IC50 > 10000 nM T43721 CV6P7Y 44420242 IC50 > 10000 nM T43721 C8IH5C 44420243 IC50 > 10000 nM T43721 CZG60J 44420244 IC50 = 50000 nM T43721 CN2B1J 44420246 IC50 > 10000 nM T43721 CG90VX 44420247 IC50 > 10000 nM T43721 C5PU7K 44420248 IC50 > 10000 nM T43721 C7KW0L 44420249 IC50 = 100000 nM T43721 CBL6K2 44420251 IC50 > 10000 nM T43721 CF9N4T 44420252 IC50 > 10000 nM T43721 CVX2Z3 44420253 IC50 > 10000 nM T43721 CX8IQ0 44420257 IC50 > 10000 nM T43721 CN3W4S 44420259 IC50 = 3600 nM T43721 C1YLR4 44420285 IC50 = 65000 nM T43721 CNRY91 44420288 IC50 > 10000 nM T43721 CF23SE 44420291 IC50 > 10000 nM T43721 CE7T4W 44420294 IC50 = 15000 nM T43721 CJ1O7N 44438556 IC50 = 17000 nM T43721 CH0K4M 44438559 IC50 = 3500 nM T43721 CXM65L 44438562 IC50 = 26000 nM T43721 CM01KY 44438566 IC50 = 20000 nM T43721 CFLP12 44438567 IC50 = 12000 nM T43721 CAW10E 44438568 IC50 = 25000 nM T43721 C3IK2C 44438569 IC50 > 100000 nM T43721 C43RLG 44438570 IC50 = 580 nM T43721 CM1Y7N 44438669 IC50 = 15000 nM T43721 CUE3I1 44438670 IC50 = 3300 nM T43721 CQM10L 44438671 IC50 = 15000 nM T43721 CB19EU 44438672 IC50 = 5400 nM T43721 CL4Y3J 44438673 IC50 = 17000 nM T43721 C7ON6I 44438675 IC50 = 65000 nM T43721 C5LN8W 44438676 IC50 > 100000 nM T43721 C8VI7M 44438677 IC50 > 100000 nM T43721 CV12KJ 44438678 IC50 = 21000 nM T43721 CBX9L4 44438679 IC50 = 59000 nM T43721 CF5YU4 44438681 IC50 > 100000 nM T43721 CJ2M3L 44438682 IC50 = 9000 nM T43721 CJB5H3 44443435 Ki > 10000 nM T43721 C3U1WZ 44448872 IC50 > 4000 nM T43721 CZ5A6G 44576636 IC50 > 4000 nM T43721 CHD6G5 44576637 IC50 > 4000 nM T43721 CK67LT 44576651 IC50 > 4000 nM T43721 C9JB2Y 44576672 IC50 > 4000 nM T43721 CMJ91U 44576707 IC50 > 4000 nM T43721 C8D1LU 44576749 IC50 > 4000 nM T43721 CKH1A8 44576750 IC50 > 4000 nM T43721 CN93WV 44576751 IC50 > 4000 nM T43721 CAH82I 44576752 IC50 > 4000 nM T43721 CK5S4W 44576802 IC50 > 4000 nM T43721 C9L3CP 44576803 IC50 > 4000 nM T43721 C2F5RM 44576804 IC50 > 4000 nM T43721 CK41XQ 44576805 IC50 > 4000 nM T43721 CO5YU9 44576846 IC50 > 4000 nM T43721 C4YIR7 44576873 IC50 > 4000 nM T43721 C2HW0I 44576875 IC50 > 4000 nM T43721 COQ7U4 44576945 IC50 > 4000 nM T43721 C18JAM 45269430 IC50 > 1000000 nM T43721 CGPF36 45270351 IC50 > 10000 nM T43721 C83OJH 45271081 IC50 > 1000000 nM T43721 C7O3DH 45271171 IC50 = 2487 nM T43721 CE07FS 45272366 IC50 > 10000 nM T43721 CK65BP 46213656 IC50 > 10000 nM T43721 CHI5S0 46216688 IC50 > 10000 nM T43721 CAX31B 46216689 IC50 > 10000 nM T43721 CN39HK 46229717 IC50 = 268 nM T43721 C4N8DB 46231719 IC50 > 10000 nM T43721 C4WT0Q 46231721 IC50 = 9000 nM T43721 CIX36V 46894126 IC50 = 2.9 nM T43721 CS13YQ 49846481 IC50 > 100000 nM T43721 C6W2XQ 49846838 IC50 > 100000 nM T43721 CA8N9P 52911994 IC50 > 30000 nM T43721 CICZ45 52918012 IC50 > 10000 nM T43721 C4X2WF 52939227 IC50 = 11 nM T43721 CQ6R0S 52939228 IC50 = 33 nM T43721 C1YRT3 52940913 IC50 = 4.9 nM T43721 CSXY62 52941059 IC50 = 7350 nM T43721 C8X4NE 52945350 IC50 = 61.1 nM T43721 CE3AQ9 52945888 IC50 = 458 nM T43721 CO7ZR1 52947102 IC50 = 8650 nM T43721 C2KHL7 52947144 IC50 = 14.5 nM T43721 CJI28A 52950107 IC50 = 2130 nM T43721 CSUK37 53322740 IC50 = 104 nM T43721 CQ7J8E 53322756 IC50 = 194 nM T43721 C6W3JM 53326660 IC50 = 17 nM T43721 CP91BU 53326661 IC50 = 45 nM T43721 C9H5YE 53361128 IC50 > 10000 nM T43721 CN93FS 54580118 IC50 > 4000 nM T43721 CF05VK 54580143 IC50 > 4000 nM T43721 C7FXV6 54580144 IC50 > 4000 nM T43721 C2M8XQ 54580210 IC50 > 4000 nM T43721 C4Q6MO 54580243 IC50 > 4000 nM T43721 CBX17R 54581094 IC50 > 4000 nM T43721 C8O9WK 54581095 IC50 > 4000 nM T43721 CM67RK 54581096 IC50 = 2300 nM T43721 C8ZDF3 54581137 IC50 > 4000 nM T43721 C14YRS 54581213 IC50 > 4000 nM T43721 CQ7GV2 54582134 IC50 > 4000 nM T43721 CZ1B6L 54582135 IC50 > 4000 nM T43721 C07KDH 54582136 IC50 = 3100 nM T43721 CK29GC 54582137 IC50 > 4000 nM T43721 CKGX19 54582164 IC50 > 4000 nM T43721 CWA6Q0 54582242 IC50 > 4000 nM T43721 C07LYE 54582261 IC50 > 4000 nM T43721 CP2N1C 54582262 IC50 > 4000 nM T43721 CM2QX4 54583079 IC50 > 4000 nM T43721 CMKQ26 54583080 IC50 > 4000 nM T43721 C2G7LK 54583125 IC50 > 4000 nM T43721 CL6Z9X 54583126 IC50 > 4000 nM T43721 CGM2W4 54583127 IC50 > 4000 nM T43721 CF42QY 54583128 IC50 > 4000 nM T43721 CWHS39 54583210 IC50 = 4000 nM T43721 CDK5V0 54583231 IC50 > 4000 nM T43721 C5V4DY 54583232 IC50 > 4000 nM T43721 C1JV9N 54583233 IC50 = 1600 nM T43721 CKA9L3 54583234 IC50 > 4000 nM T43721 CZ4YV3 54584081 IC50 > 4000 nM T43721 CHP62C 54584119 IC50 > 4000 nM T43721 CD2QO1 54584120 IC50 = 1300 nM T43721 CCT0B2 54584121 IC50 > 4000 nM T43721 C0VPS6 54584122 IC50 > 4000 nM T43721 C6P5XR 54584196 IC50 > 4000 nM T43721 CY2WM3 54584197 IC50 > 4000 nM T43721 CXNP26 54584198 IC50 > 4000 nM T43721 CWY83C 54584415 IC50 > 4000 nM T43721 CGD4N3 54585028 IC50 > 4000 nM T43721 C8NZ2B 54585029 IC50 > 4000 nM T43721 CHW48S 54585030 IC50 > 4000 nM T43721 CZ8R0S 54585053 IC50 > 4000 nM T43721 C04IZR 54585054 IC50 > 4000 nM T43721 C6GZB9 54585157 IC50 > 4000 nM T43721 C5SHO2 54585992 IC50 > 4000 nM T43721 CJA5Z6 54585993 IC50 > 4000 nM T43721 C4JTZ5 54585994 IC50 > 4000 nM T43721 CKF15E 54586030 IC50 > 4000 nM T43721 CT12RX 54586031 IC50 > 4000 nM T43721 CD6FC5 54586091 IC50 = 1300 nM T43721 CDG95F 54586092 IC50 > 4000 nM T43721 CJ8K1Y 54586966 IC50 > 4000 nM T43721 C51MDN 54586967 IC50 > 4000 nM T43721 CH2F8P 54586968 IC50 > 4000 nM T43721 C61ZTA 54586969 IC50 > 4000 nM T43721 C3Y6HF 54587012 IC50 > 4000 nM T43721 CUF68X 54587090 IC50 = 460 nM T43721 CI1PV5 54587121 IC50 > 4000 nM T43721 C6PSJ3 54587122 IC50 > 4000 nM T43721 C9D1UH 54587123 IC50 > 4000 nM T43721 C82TDJ 54587124 IC50 > 4000 nM T43721 CNQ41E 54590876 IC50 > 10000 nM T43721 C3IAB0 57392785 IC50 = 386 nM T43721 C4I9DE 57408764 IC50 > 100000 nM T43721 CM2DN9 57408765 IC50 = 400 nM T43721 CAI0P1 57418438 IC50 > 100000 nM T43721 C39SNL 57916360 IC50 > 30000 nM T43721 CG16CV 57916503 IC50 > 30000 nM T43721 CG1Y8Z 67464068 IC50 > 10000 nM T43721 CJL0P9 67468231 IC50 > 10000 nM T43721 CM80QX 70687773 EC50 = 2200 nM T43721 CZI43B 70691963 EC50 = 860 nM T43721 CQ5GB9 70691964 EC50 = 720 nM T43721 C3CAB4 71456572 IC50 = 2200 nM T43721 CU24OM 71458421 IC50 > 10000 nM T43721 C0D3IO 71511561 IC50 > 10 nM T43721 C4LAB0 72204152 IC50 = 2200 nM T43721 C17NBW 72204153 IC50 = 2410 nM T43721 CTN6U7 72204155 IC50 = 2690 nM T43721 C0N7EJ 72204340 IC50 = 5850 nM T43721 CS3TL6 72204534 IC50 = 4210 nM T43721 CA5KC4 72204732 IC50 = 6760 nM T43721 C2Q6YJ 72670421 IC50 = 4000 nM T43721 CYAJ36 73345978 IC50 = 1600 nM T43721 CG15WM 73352110 IC50 > 100000 nM T43721 CALM65 73352112 IC50 > 100000 nM T43721 C9WA7F 73353568 IC50 > 100000 nM T43721 CV72YC 73355069 IC50 > 100000 nM T43721 CGR3P5 73355072 IC50 = 228700 nM T43721 C15SEC 73356624 IC50 > 1000000 nM T43721 C2FOM5 73356626 IC50 = 700 nM T43721 CV70BR 73356628 IC50 > 1000000 nM T43721 CWC4Z5 73356629 IC50 > 100000 nM T43721 CPN65E 90643787 IC50 > 30000 nM T43721 CQ23WR 90667215 IC50 > 30000 nM T43721 CFSK10 101911911 IC50 = 25500 nM T43721 CO0H9S 101911912 IC50 = 40700 nM T43721 C91CLR 101911913 IC50 = 299600 nM T43721 C9RBA1 101911914 IC50 = 283600 nM T43721 CMOG09 101911915 IC50 = 11300 nM T43721 CMX6S5 118709259 IC50 > 10000 nM T43721 C7WYI8 127037831 IC50 > 1000000 nM T43721 CI5HA6 127037875 IC50 > 1000000 nM T43721 CP0JV9 127038197 IC50 > 1000000 nM T43721 C4E1LF 127040565 IC50 > 1000000 nM T43721 CTN4E7 127040566 IC50 > 1000000 nM T43721 CB67LT 127040901 IC50 > 1000000 nM T43721 C5P3KE 127040902 IC50 > 1000000 nM T43721 CT5Q1A 127040903 IC50 > 1000000 nM T43721 CW3FN4 127040904 IC50 > 1000000 nM T43721 C9EQX2 127040905 IC50 > 1000000 nM T43721 C32ADQ 127040906 IC50 > 1000000 nM T43721 CYNI06 127041808 IC50 > 1000000 nM T43721 C1ZUD5 127041809 IC50 > 1000000 nM T43721 CCU4H6 127041810 IC50 > 1000000 nM T43721 CZN2A0 127041811 IC50 > 1000000 nM T43721 CCKL17 127042099 IC50 > 1000000 nM T43721 C24EQS 127042100 IC50 > 1000000 nM T43721 CE64CI 127042101 IC50 > 1000000 nM T43721 COR6A5 127042102 IC50 > 1000000 nM T43721 CKM3I9 127042477 IC50 > 1000000 nM T43721 CMP75K 127042478 IC50 > 1000000 nM T43721 CMCP64 127042780 IC50 > 1000000 nM T43721 C4OUL9 127042781 IC50 > 1000000 nM T43721 CGWV92 132053849 IC50 < 100 nM T43721 CT05EL 135399889 IC50 > 10000 nM T43721 C02KAD 135440148 IC50 > 4000 nM T43721 CE0S3Y 135465949 IC50 > 4000 nM T43721 CM7A1J 135492551 IC50 > 4000 nM T43721 C98OIC 135611051 IC50 > 10000 nM T43721 CCQJ43 135611106 IC50 > 10000 nM T43721 C2K9OD 135611129 IC50 > 10000 nM T43721 C4YO9E 135612240 IC50 > 4000 nM T43721 C76MEG 135783319 IC50 > 10000 nM T43721 CMQ2L1 135783320 IC50 > 10000 nM T43721 CE6L4S 135783321 IC50 > 10000 nM T43721 CTAM34 135783322 IC50 > 10000 nM T43721 C7B3JV 135783325 IC50 > 10000 nM T43721 C59KXI 135783328 IC50 > 10000 nM T43721 CKB54L 135783329 IC50 > 10000 nM T43721 C7ZTC5 135783333 IC50 > 10000 nM T43721 C09UQY 135783334 IC50 > 10000 nM T43721 CL5F0J 135783335 IC50 > 10000 nM T43721 CA2ZD0 135857035 IC50 > 10000 nM T43721 CV64MY 135857036 IC50 > 10000 nM T43721 C6IYH3 135967877 IC50 = 35000 nM T43721 C0FO4G 135980568 IC50 = 15 nM T43721 CX3VU1 136000590 IC50 > 4000 nM T43721 CNQ25Z 136021384 IC50 > 10000 nM T43721 C7W4GE 136088954 IC50 > 4000 nM T43721 CT3RN8 136141565 IC50 = 11 nM T43721 CR74OZ 136188845 IC50 > 4000 nM T43721 CWJ0X4 137637923 IC50 = 6261 nM T43721 CDS86M 137656441 IC50 = 9582 nM T43721 C94RSY 137656587 IC50 > 10000 nM T43721 C0DHM9 145952000 IC50 = 100 nM T43721 CC91LF 145952333 IC50 < 100 nM T43721 CDT3Q6 145956314 IC50 = 1000 nM T43721 C09QUS 145958039 IC50 < 100 nM T43721 CV6Q5J 145960157 IC50 = 100 nM T43721 CMVS94 155512106 IC50 > 500000 nM T43721 C1F9PV 155515115 IC50 > 500000 nM T43721 CPO9M4 155520336 IC50 > 500000 nM T43721 CXOU89 155521135 IC50 > 500000 nM T43721 C8WNT0 155521284 IC50 > 500000 nM T43721 CN59WH 155525513 IC50 > 500000 nM T43721 C1D4WM 155537728 IC50 > 500000 nM T43721 CV5KQ0 155543491 IC50 > 500000 nM T43721 CKFU03 155545095 IC50 > 500000 nM T43721 CG19XT 155548236 IC50 > 500000 nM T43721 CB08IM 155548826 IC50 > 500000 nM T43721 C1GC0O 155553184 IC50 > 500000 nM T43721 CEM03Y 155556588 IC50 > 500000 nM T43721 C9E6AM 155561480 IC50 > 500000 nM T43721 COWH25 155562798 IC50 > 500000 nM T43721 CZT7P4 155567250 IC50 > 500000 nM T43721 D00PSW 3630776 IC50 > 3000 nM T43721 D00QOL 11673314 IC50 > 10000 nM T43721 D02KXX 586971 IC50 > 200000 nM T43721 D02WUU 15627039 IC50 > 200000 nM T43721 D03JWH 135450677 IC50 > 10000 nM T43721 D04WVV 10193044 IC50 > 4000 nM T43721 D0A4ZR 135950111 Ki > 10000 nM T43721 D0EU9W 16750524 IC50 > 200000 nM T43721 D0L4VR 636403 IC50 = 170 nM T43721 D0M4PP 4271571 IC50 > 200000 nM T43721 D0P7RN 1483401 IC50 > 200000 nM T43721 D0T3FW 44419251 IC50 > 10000 nM T43721 D0U8IF 10114 IC50 = 1.2 nM T09513 D0A3MV 448014 IC50 > 100000 nM T09513 CH20NR 403176 IC50 = 20 nM T09513 CNG96H 25210579 IC50 > 10000 nM T09513 CE1ZK6 54759168 IC50 > 10000 nM T09513 CL5IR0 135512024 IC50 = 7 nM T09513 D03YVL 5472558 IC50 = 25000 nM T09513 D0Y0ES 3707 IC50 = 100 nM T32880 D06VNK 1110 IC50 = 3000 nM T32880 D01SPD 69669724 IC50 = 280 nM T32880 D03GOO 444972 IC50 = 19000 nM T32880 D03YKE 11256664 IC50 = 591.4 nM T32880 D07KEH 23634441 IC50 = 29 nM T32880 D0N6CS 6914666 IC50 = 70 nM T32880 D00IKR 52912218 IC50 = 14000 nM T32880 D01XZT 24891734 IC50 = 650 nM T32880 D03TPE 97394 IC50 = 14000 nM T32880 D09NCT 53392492 IC50 = 83000 nM T32880 D0QI0J 134204791 IC50 = 15000 nM T32880 CWJ0U1 5312 IC50 = 18000 nM T32880 CMO39B 7493 Ki > 300000 nM T32880 CK23OU 76549 IC50 > 1000000 nM T32880 C8JBE5 94284 IC50 = 8500 nM T32880 C06WZQ 222878 IC50 > 100000 nM T32880 CBZ21G 231363 IC50 > 100000 nM T32880 COS62U 245007 IC50 > 100000 nM T32880 C0MHV8 252439 IC50 = 94000 nM T32880 C3OZ5L 919929 IC50 > 100000 nM T32880 C2OS3W 2238068 IC50 > 100000 nM T32880 CHV8N5 4666803 IC50 > 40000 nM T32880 CGP0X9 6914624 IC50 = 1400 nM T32880 CS7C1Z 8027170 IC50 = 12000 nM T32880 CYJ23Z 10470802 IC50 = 4800 nM T32880 CP76HX 11372202 IC50 = 2400 nM T32880 CM6Q3H 11788622 IC50 > 100000 nM T32880 CDM30S 13770962 IC50 > 1000000 nM T32880 CO03CL 14991438 IC50 = 95000 nM T32880 C9M2AL 16126655 IC50 = 190 nM T32880 CIU0N5 16126706 IC50 = 3900 nM T32880 CI45OC 16126774 IC50 = 3600 nM T32880 CX5VP0 18372521 IC50 = 5300 nM T32880 C52JUB 18372631 IC50 = 4400 nM T32880 CN2HO1 18632368 IC50 = 69700 nM T32880 CDSM62 20816892 IC50 = 4200 nM T32880 C20YQO 22122176 IC50 > 1000000 nM T32880 C92REF 22345738 IC50 = 398000 nM T32880 CCAM68 22959876 IC50 > 100000 nM T32880 CGE7Y9 23260762 IC50 > 1000000 nM T32880 CZ9X6U 24812792 IC50 = 3 nM T32880 CZ8WG7 24831508 IC50 = 22.2 nM T32880 CE9N0S 24891150 IC50 > 100000 nM T32880 CV17FS 24894050 IC50 = 21 nM T32880 C0R7YW 25105470 IC50 = 3 nM T32880 C9TN1M 25105471 IC50 = 3 nM T32880 C9CLE1 25138008 IC50 > 1000000 nM T32880 C8P4AV 25173259 IC50 = 185 nM T32880 C5PJZ9 25173339 IC50 = 44 nM T32880 CIM16Z 25173590 IC50 = 7.8 nM T32880 CP8D4L 25173666 IC50 = 140 nM T32880 CTNC06 25173744 IC50 = 52 nM T32880 C92CGK 25173747 IC50 = 30 nM T32880 C5YWM9 25173822 IC50 = 17 nM T32880 CIF90R 25173824 IC50 = 4.1 nM T32880 C3C0AO 25173900 IC50 = 11 nM T32880 C4TNI3 25206050 IC50 = 1500 nM T32880 CS6N9A 42639237 IC50 = 45500 nM T32880 C2AG1B 42639238 IC50 = 8600 nM T32880 C4LK0F 42639413 IC50 = 700 nM T32880 CY6M3D 42639898 IC50 = 1900 nM T32880 CDE5U3 44419123 IC50 = 46000 nM T32880 CFI5L3 44419124 IC50 = 39000 nM T32880 C0U8JS 44419131 IC50 = 15000 nM T32880 C0Y2EG 44419132 IC50 > 100000 nM T32880 CMD26E 44419133 IC50 = 20000 nM T32880 CLQ71X 44419139 IC50 = 4900 nM T32880 C7MYD0 44419140 IC50 = 6500 nM T32880 C0O3EP 44419147 IC50 = 15000 nM T32880 C5IQT0 44419154 IC50 = 18000 nM T32880 CO8HT3 44419159 IC50 = 15000 nM T32880 CGW2A6 44419160 IC50 = 7300 nM T32880 C6ZYP0 44419165 IC50 = 6800 nM T32880 CB1YA2 44419171 IC50 = 19000 nM T32880 C4QH8U 44419179 IC50 = 10000 nM T32880 CY4NW1 44419252 IC50 = 17000 nM T32880 C6T3AY 44419262 IC50 = 5000 nM T32880 C2FSX3 44419264 IC50 = 14200 nM T32880 C5M4KV 44419265 IC50 = 6800 nM T32880 CE5N3Y 44419266 IC50 = 4600 nM T32880 CQ0IJ2 44419267 IC50 = 7400 nM T32880 C38SEB 44419270 IC50 = 16000 nM T32880 C6OR8X 44419271 IC50 = 4400 nM T32880 C0CW1M 44419272 IC50 = 28700 nM T32880 CQ0A4B 44419273 IC50 = 6000 nM T32880 CVE69C 44419277 IC50 = 9700 nM T32880 C7UOR2 44419278 IC50 = 6100 nM T32880 C1H6FT 44419280 IC50 = 8100 nM T32880 CX43WB 44419281 IC50 = 5900 nM T32880 C0YGE2 44419282 IC50 = 14000 nM T32880 CNR45T 44419283 IC50 = 4100 nM T32880 CE5N6U 44419284 IC50 = 10000 nM T32880 C4UEG7 44419285 IC50 = 3200 nM T32880 CGSN20 44419287 IC50 = 7200 nM T32880 COR69J 44419288 IC50 = 6900 nM T32880 C6NXA4 44419290 IC50 = 5800 nM T32880 C3IW5O 44419297 IC50 = 19000 nM T32880 CAP3T5 44419302 IC50 = 24000 nM T32880 C2X1ZV 44419317 IC50 = 2700 nM T32880 CNV8A6 44419318 IC50 = 580 nM T32880 CS85EJ 44419319 IC50 = 1700 nM T32880 CI2M5C 44419320 IC50 = 2400 nM T32880 C0TIU7 44419321 IC50 = 2400 nM T32880 C1MOH2 44419325 IC50 = 1600 nM T32880 C7KUX4 44419326 IC50 = 1600 nM T32880 C37UJB 44419329 IC50 = 2100 nM T32880 C8SQT3 44419330 IC50 = 2900 nM T32880 C2GTJ8 44419333 IC50 = 1700 nM T32880 C96OKR 44419334 IC50 = 2800 nM T32880 CP42UL 44419336 IC50 = 12000 nM T32880 CPX3V9 44419342 IC50 = 24000 nM T32880 C0B9TD 44419346 IC50 > 100000 nM T32880 C5Z3XD 44462724 IC50 = 1.6 nM T32880 C3CST2 44462748 IC50 = 6.8 nM T32880 CR05QL 44469096 IC50 > 100000 nM T32880 C9MK8J 44469097 IC50 = 12589.25 nM T32880 CK6O8G 44469099 IC50 = 19952.62 nM T32880 CADR40 44469101 IC50 = 25118.86 nM T32880 CBSI48 44469229 IC50 = 50118.72 nM T32880 C4U5RZ 44478798 IC50 = 79.43 nM T32880 CR21XB 44478800 IC50 = 158.49 nM T32880 CXOU61 44481885 IC50 = 1000 nM T32880 CCGJ52 44482164 IC50 = 79.43 nM T32880 CIK17O 44482165 IC50 = 398.11 nM T32880 CBL07Q 44482167 IC50 = 398.11 nM T32880 C42FTP 44482169 IC50 = 316.23 nM T32880 CT15UI 44514766 IC50 = 2.1 nM T32880 CW9OQ6 44568201 IC50 = 72 nM T32880 CF9QX3 44568202 IC50 > 40000 nM T32880 CEQL05 44568203 IC50 > 40000 nM T32880 CVWD50 44568204 IC50 = 1300 nM T32880 CX8B7T 44568205 IC50 = 72 nM T32880 CJ12AH 44568206 IC50 = 98 nM T32880 CC4B5M 44568207 IC50 = 33 nM T32880 CU63MS 44568208 IC50 = 27 nM T32880 C69PMH 44568247 IC50 > 40000 nM T32880 C1M3GY 44568248 IC50 = 400 nM T32880 C3JLM8 44568249 IC50 = 410 nM T32880 CF1E4K 44568250 IC50 = 2300 nM T32880 CX2YE1 44568251 IC50 = 21 nM T32880 CO50XS 44568252 IC50 = 11 nM T32880 C43BDN 44568281 IC50 = 4400 nM T32880 CXR89P 44568282 IC50 = 1700 nM T32880 CVID82 44568283 IC50 > 40000 nM T32880 C9JGC4 44568284 IC50 = 600 nM T32880 CG62EN 44568285 IC50 = 50 nM T32880 CK3SI1 44579681 IC50 = 570 nM T32880 CDAN35 44579682 IC50 = 290 nM T32880 CL9O6W 44579683 IC50 = 320 nM T32880 C1OTW6 44579684 IC50 = 330 nM T32880 CE1KX7 44579685 IC50 = 400 nM T32880 CZF4B8 44579687 IC50 > 40000 nM T32880 C8A3XZ 44579730 IC50 = 2820 nM T32880 C6LQ9S 44579731 IC50 = 5540 nM T32880 CFN49B 44579732 IC50 = 66 nM T32880 CMI6G8 44579733 IC50 > 40000 nM T32880 CBVI46 44579734 IC50 = 730 nM T32880 CVD1W3 44591754 IC50 = 512 nM T32880 C3OL2Y 44591755 IC50 = 230000 nM T32880 C71GJA 44819566 IC50 > 400000 nM T32880 CKD8A7 44819735 IC50 > 400000 nM T32880 C1VH6I 45482712 IC50 = 78000 nM T32880 C0W6RQ 45482725 IC50 > 1000000 nM T32880 C34LSI 45482742 IC50 > 1000000 nM T32880 CK2R4F 45482768 IC50 > 1000000 nM T32880 CIU6F7 45482769 IC50 > 1000000 nM T32880 CJ7OS3 45482772 IC50 = 538000 nM T32880 CX42JP 45482778 IC50 > 1000000 nM T32880 C2HL7F 45486323 IC50 = 21 nM T32880 CUMF70 46899605 IC50 > 100000 nM T32880 C2DBN5 46899607 IC50 > 100000 nM T32880 C3G4QK 46899609 IC50 > 100000 nM T32880 CLK96Z 46899763 IC50 > 100000 nM T32880 CBOM64 46899765 IC50 > 100000 nM T32880 CA56RL 49831102 IC50 = 3 nM T32880 CU63QR 49847377 IC50 = 0.2 nM T32880 CZT4I8 49847378 IC50 = 0.2 nM T32880 CA72PE 49847379 IC50 = 1.6 nM T32880 CC23YW 49847498 IC50 = 55 nM T32880 CJ7H2B 49847753 IC50 = 3.4 nM T32880 C4V7EW 49848258 IC50 = 0.8 nM T32880 C4E2YF 49848485 IC50 = 13700 nM T32880 CWP7L0 49848519 IC50 = 427 nM T32880 CV0PU1 49848649 IC50 = 27 nM T32880 CP8TS6 49848895 IC50 = 0.4 nM T32880 C9COF5 49848896 IC50 = 0.5 nM T32880 CK0B1G 49848897 IC50 = 0.2 nM T32880 CP61VJ 49849002 IC50 = 0.2 nM T32880 C42SBF 49849005 IC50 = 4.3 nM T32880 CBM62Z 49849007 IC50 = 0.4 nM T32880 C05SEW 49849008 IC50 = 0.2 nM T32880 C78SAD 49849115 IC50 = 4.1 nM T32880 CF64IJ 49849120 IC50 = 0.2 nM T32880 CC9EB4 49849122 IC50 = 0.5 nM T32880 C2ORV5 49849123 IC50 = 5.4 nM T32880 CUJ4D6 49870967 IC50 = 100 nM T32880 CX8Z0D 50899320 IC50 = 120 nM T32880 C0HCX8 50916282 IC50 > 400000 nM T32880 C2QG8V 53318573 IC50 = 50118.72 nM T32880 C90UET 53319897 IC50 > 100000 nM T32880 CX7O4F 53319898 IC50 = 79432.82 nM T32880 CS3E2L 53493245 IC50 = 0.7 nM T32880 CRFI05 53493908 IC50 = 0.7 nM T32880 C68OFC 54681699 IC50 = 46 nM T32880 CJO04Q 54739165 IC50 < 50 nM T32880 CT0UM5 54741100 IC50 = 1.5 nM T32880 C28RDF 54746913 IC50 = 4.9 nM T32880 C35JDV 54746961 IC50 = 5.3 nM T32880 CDL06K 54746964 IC50 = 3.1 nM T32880 CK3GC9 54746970 IC50 < 10 nM T32880 C7Q4WV 54747815 IC50 < 10 nM T32880 C2TB1P 54747831 IC50 < 10 nM T32880 CZWR91 54747907 IC50 = 4.1 nM T32880 CT6MD1 54749350 IC50 = 0.65 nM T32880 C9OG0S 54749369 IC50 = 3 nM T32880 CU7S6Y 56656421 IC50 = 50 nM T32880 CMR1X3 56684140 IC50 > 1000000 nM T32880 CE26XI 56684141 IC50 > 1000000 nM T32880 CL8N7V 56964909 IC50 > 1000000 nM T32880 C34DJP 57384236 IC50 = 1.1 nM T32880 CEOC15 57384237 IC50 = 2 nM T32880 CY50WC 57384238 IC50 = 2.3 nM T32880 C7S0ZR 57384239 IC50 = 1.5 nM T32880 C2XN1G 57384481 IC50 = 1.6 nM T32880 CR73IZ 57384482 IC50 = 0.8 nM T32880 CR2M5H 57384483 IC50 = 0.5 nM T32880 CQ72HI 57384749 IC50 = 4.7 nM T32880 C68KGE 57384750 IC50 = 1.9 nM T32880 CA57BP 57384999 IC50 = 0.5012 nM T32880 C5OGF6 57385246 IC50 = 640 nM T32880 CJ8N5F 57385491 IC50 = 680 nM T32880 C2HXQ4 57385492 IC50 = 6600 nM T32880 CFB30C 57385493 IC50 = 2200 nM T32880 CE8A9F 57385494 IC50 = 1200 nM T32880 CHJ8G2 57385495 IC50 = 1000 nM T32880 CMSP14 57385496 IC50 = 7800 nM T32880 CB2Y1U 57385733 IC50 = 370 nM T32880 CH15PS 57385734 IC50 = 2600 nM T32880 CE40ZB 57385735 IC50 = 790 nM T32880 CKO54M 57385736 IC50 > 50000 nM T32880 C5XDF4 57385737 IC50 > 50000 nM T32880 CR7UN3 57385738 IC50 > 50000 nM T32880 C85XSW 57386006 IC50 > 50000 nM T32880 CUL23K 57386007 IC50 = 3040 nM T32880 CJTC03 57386008 IC50 = 440 nM T32880 C9THS0 57386009 IC50 = 15300 nM T32880 CV34YJ 57386010 IC50 > 50000 nM T32880 C0RKZ2 57386011 IC50 > 50000 nM T32880 COI01S 57386263 IC50 > 50000 nM T32880 CUF1Y0 57386264 IC50 = 3100 nM T32880 C2BJT0 57386265 IC50 = 840 nM T32880 CVZ19P 57386266 IC50 = 4700 nM T32880 C3SUV6 57386267 IC50 = 6000 nM T32880 CF0TG4 57386268 IC50 = 3.8 nM T32880 CCR1X8 57386520 IC50 = 98 nM T32880 CQ6JG3 57386521 IC50 = 31 nM T32880 CVK29R 57386523 IC50 = 2.1 nM T32880 C9S8MU 57386524 IC50 = 4.3 nM T32880 CMC8H6 57386782 IC50 = 0.4 nM T32880 CCT5D4 57386783 IC50 = 0.4 nM T32880 CC30XZ 57386784 IC50 = 5 nM T32880 C79BXP 57386785 IC50 = 0.8 nM T32880 CM6DV7 57387028 IC50 = 1 nM T32880 C0GS4F 57387282 IC50 = 0.6 nM T32880 C0TL9C 57387283 IC50 = 2.8 nM T32880 CRV2P5 57387539 IC50 = 0.2 nM T32880 CAU3G9 57387540 IC50 = 0.2 nM T32880 CL2AO8 57387541 IC50 = 0.4 nM T32880 C0XWL8 57387542 IC50 = 0.4 nM T32880 CC4DK0 57387775 IC50 = 1 nM T32880 C8DB9I 57387776 IC50 = 0.8 nM T32880 C2LZ8G 57387778 IC50 = 1200 nM T32880 CUN9V6 57388001 IC50 = 0.7 nM T32880 CV7W0P 57742961 IC50 = 65 nM T32880 CS6Z2D 57983461 IC50 < 100 nM T32880 C2DIK6 57983520 IC50 < 100 nM T32880 CCB65L 59603622 IC50 = 280 nM T32880 COL70Z 67049505 IC50 = 820 nM T32880 CKG14F 67049582 IC50 = 2500 nM T32880 CFM6H7 67049587 IC50 = 220 nM T32880 C3CU9D 67049655 IC50 = 7100 nM T32880 C7AJ1U 67049671 IC50 = 450 nM T32880 C2DPK9 67049808 EC50 = 4700 nM T32880 C3AP9U 67049854 IC50 = 1200 nM T32880 CB3HX6 67049905 IC50 = 1600 nM T32880 C5PM7A 67049973 EC50 = 14000 nM T32880 C4VG9Q 67050041 IC50 = 210 nM T32880 C6UHR9 67050359 IC50 = 730 nM T32880 C92WSG 67050361 EC50 = 13000 nM T32880 C7LBD8 67050367 IC50 = 850 nM T32880 C1N9OY 67050409 EC50 = 5800 nM T32880 C8VM6P 67283460 IC50 = 94 nM T32880 C5RGQ2 68392546 IC50 = 100 nM T32880 CKX41C 69674161 IC50 = 110 nM T32880 C4VU7J 70688210 IC50 = 4.9 nM T32880 CO7H3Q 71133989 IC50 = 2.3 nM T32880 CL3HT1 71449736 IC50 = 6300 nM T32880 CJH86V 71451542 IC50 > 100000 nM T32880 CH38AO 71453382 IC50 > 100000 nM T32880 C2U4AQ 71458738 IC50 = 14200 nM T32880 C1DYB4 71477196 IC50 = 17 nM T32880 C9XGE6 71537024 IC50 < 10 nM T32880 CK34XF 71538425 IC50 < 20 nM T32880 CX74LQ 71545631 IC50 = 18400 nM T32880 CP6WO8 71717922 IC50 = 20 nM T32880 C7Y8SB 71748680 IC50 = 15.85 nM T32880 CC7M4D 72204345 IC50 > 10000 nM T32880 CM41RB 72204346 IC50 > 10000 nM T32880 C9A4KH 72204347 IC50 > 10000 nM T32880 C5MZ7R 72204348 IC50 = 158.49 nM T32880 CA2C1U 72204349 IC50 = 199.53 nM T32880 C4JZ6C 72204350 IC50 = 794.33 nM T32880 CZFG12 72204539 IC50 = 630.96 nM T32880 C8PM1E 72204540 IC50 = 2.512 nM T32880 CT4X1K 72204541 IC50 = 1 nM T32880 CV4EJ6 72204542 IC50 = 79.43 nM T32880 C3X0TL 72204543 IC50 = 1995.26 nM T32880 CZF7R4 72204544 IC50 = 1258.93 nM T32880 CK63AC 72204738 IC50 = 3981.07 nM T32880 CGE63D 72204739 IC50 = 1000 nM T32880 CGR92Y 72204740 IC50 = 3162.28 nM T32880 CIBE51 72204741 IC50 = 398.11 nM T32880 C2C5QX 72204742 IC50 = 3162.28 nM T32880 C4JAC1 72204743 IC50 = 501.19 nM T32880 C3WV2R 72204920 IC50 = 1995.26 nM T32880 C4MO3I 72204921 IC50 = 630.96 nM T32880 C1E4BJ 72204922 IC50 = 7.943 nM T32880 CI0R2O 72204923 IC50 = 31.62 nM T32880 C40BFH 72204924 IC50 = 3.981 nM T32880 CB1G4W 72204925 IC50 = 25.12 nM T32880 C81AQS 72205106 IC50 = 39.81 nM T32880 CK5MI2 72205107 IC50 = 5.012 nM T32880 C35SGD 72205108 IC50 = 15.85 nM T32880 CI0ON6 72205109 IC50 = 50.12 nM T32880 C6LM0T 72205110 IC50 > 10000 nM T32880 CWJG76 72737642 IC50 = 14 nM T32880 C2UFG1 73052701 IC50 = 39 nM T32880 CW64KE 73052704 IC50 = 49 nM T32880 CZU9X4 73052863 IC50 = 13 nM T32880 C4XIZ8 73349624 IC50 = 12589.25 nM T32880 C68RKH 76310231 IC50 = 8500 nM T32880 C89AEL 76310612 IC50 = 0.7 nM T32880 CO1EN3 76317452 IC50 = 278000 nM T32880 CPE6U2 76335997 IC50 > 500000 nM T32880 C7K3JM 89812866 IC50 = 9400 nM T32880 CHVP04 92042841 IC50 = 61 nM T32880 C6NUD0 118718072 IC50 = 41800 nM T32880 CUR10H 118978237 IC50 = 5.8 nM T32880 CI5X2G 118978277 IC50 = 11 nM T32880 CH7WL3 118978299 IC50 = 20 nM T32880 C43IWX 118978308 IC50 = 22.9 nM T32880 C2LBH1 118978321 IC50 = 66 nM T32880 CB3I9Z 118978325 IC50 = 9 nM T32880 CWH4I0 118978339 IC50 = 19 nM T32880 C6XD3H 118978341 IC50 = 5.4 nM T32880 CJE6K4 118978367 IC50 = 7.3 nM T32880 CDBK07 118981498 IC50 = 2.6 nM T32880 CB23LS 118981525 IC50 = 10 nM T32880 C9F6RL 118981536 IC50 = 6.9 nM T32880 CF1E6T 118981546 IC50 = 6.8 nM T32880 C1ABC5 118981554 IC50 = 4.3 nM T32880 CR05OQ 118981555 IC50 = 4.2 nM T32880 CE9U5L 118981600 IC50 = 4 nM T32880 CO5XH7 118981638 IC50 = 4.9 nM T32880 CV84HB 118981731 IC50 = 4.4 nM T32880 CM3VL0 118981967 IC50 = 21 nM T32880 CW89CV 118982285 IC50 = 6.5 nM T32880 C51RST 121245332 IC50 = 3.8 nM T32880 C2LI6C 121245745 IC50 = 8.5 nM T32880 C69YAB 121246676 IC50 = 0.9 nM T32880 C27WIY 121246694 IC50 = 27 nM T32880 C0E7BZ 121246784 IC50 = 1.9 nM T32880 CH4O3R 121246791 IC50 = 1 nM T32880 C71YRT 121246805 IC50 = 5.4 nM T32880 CJU6X7 121246821 IC50 = 2 nM T32880 C1X3HT 121246837 IC50 = 6.1 nM T32880 C2UY6K 121246848 IC50 = 4.2 nM T32880 C5E0SB 121246859 IC50 = 1.8 nM T32880 CE3P9G 121246864 IC50 = 1.5 nM T32880 C6BIK2 121269752 IC50 = 0.62 nM T32880 C6H2YQ 122383780 IC50 = 96000 nM T32880 CT2UZ4 125377518 IC50 > 100000 nM T32880 C5NR3C 129027150 IC50 = 13700 nM T32880 CWO0V4 135566826 IC50 = 2800 nM T32880 CV9J3Z 135737442 IC50 = 195000 nM T32880 CSCH32 135871166 IC50 = 27500 nM T32880 C3Q9KJ 135871167 IC50 = 81000 nM T32880 CJIK12 135871172 IC50 = 2200 nM T32880 CWI9V2 135871182 IC50 = 2100 nM T32880 C39VQA 135871218 IC50 = 700 nM T32880 CF5TV8 135871220 IC50 = 3800 nM T32880 CD6QM3 135871221 IC50 = 800 nM T32880 C2G7XC 135871222 IC50 = 24000 nM T32880 CAJ08Y 135871235 IC50 = 400 nM T32880 C42ISC 135871238 IC50 = 1400 nM T32880 C9DPJ0 135871283 IC50 = 2000 nM T32880 CYVH90 135895253 IC50 = 8 nM T32880 CT57ZH 136069450 IC50 = 0.2 nM T32880 CFT9R3 136069453 IC50 = 0.6 nM T32880 CRPQ42 136069494 IC50 = 2.5 nM T32880 CK8Z3V 136069521 IC50 = 5 nM T32880 CPY1B2 136069522 IC50 = 31 nM T32880 CX0OM4 136069523 IC50 = 11 nM T32880 C6EU4D 136069524 IC50 = 76 nM T32880 CQA2Z1 136069531 IC50 = 9.3 nM T32880 CCH31A 136069532 IC50 = 0.9 nM T32880 CH8GV7 136069561 IC50 = 14 nM T32880 CQ1FS4 136069563 IC50 = 3.9 nM T32880 C97REI 136074309 IC50 = 6000 nM T32880 CN6X7E 136074310 IC50 = 13500 nM T32880 CLV1R6 136074312 IC50 = 5700 nM T32880 CY3Z2V 136074313 IC50 = 1200 nM T32880 CEJ1M9 136074314 IC50 = 3000 nM T32880 CR5IM8 136074315 IC50 = 3400 nM T32880 CX02WY 136074316 IC50 = 2400 nM T32880 CICS75 136074317 IC50 = 7300 nM T32880 CS9C0Q 136074318 IC50 = 3900 nM T32880 CQTB32 136205798 IC50 = 1.1 nM T32880 CV8QP3 136205832 IC50 = 0.2 nM T32880 CB93EM 136205833 IC50 = 0.6 nM T32880 CV1C5I 136986966 IC50 = 2600 nM T32880 CJNU29 137083353 IC50 = 12 nM T32880 C0F8XB 137150345 IC50 = 20 nM T32880 C5UFR2 138319689 IC50 = 62.23 nM T32880 C7RYB5 141508724 IC50 = 248 nM T32880 CI1DE9 141508725 IC50 = 280.6 nM T32880 C5PN8T 141508727 IC50 = 228.2 nM T32880 CE36KV 141508729 IC50 = 418.3 nM T32880 C29GLS 141508732 IC50 = 278.3 nM T32880 C8SW9L 141508738 IC50 = 75.82 nM T32880 C5NJS7 141508739 IC50 = 61.08 nM T32880 C0Q5YG 141508741 IC50 = 308.3 nM T32880 C4QT0G 141508742 IC50 = 759.4 nM T32880 C2XB9I 141508745 IC50 = 418.7 nM T32880 CLK1B4 141508746 IC50 = 419.3 nM T32880 CJ9O3L 141508747 IC50 = 77 nM T32880 CV6N8B 141508748 IC50 = 271 nM T32880 C5SIU2 141508749 IC50 = 67.58 nM T32880 C2JRM3 141508751 IC50 = 231.1 nM T32880 C3WIL6 141508752 IC50 = 375.4 nM T32880 CK2ST8 141508755 IC50 = 418.3 nM T32880 CG0FL4 141508765 IC50 = 52.84 nM T32880 CN8EK0 141508769 IC50 = 579.7 nM T32880 CVMW03 141617793 EC50 = 17000 nM T32880 C2ML4K 141740991 IC50 = 1.9 nM T32880 C15DMN 145955244 IC50 = 16000 nM T32880 CK41QM 145957905 IC50 = 650 nM T32880 CWU6S2 145958372 IC50 = 6500 nM T32880 C7SIP1 145960425 IC50 = 801.4 nM T32880 CID5Y8 145960662 IC50 = 2165 nM T32880 CC9A8D 145960865 IC50 = 3594 nM T32880 CZDC15 145961128 IC50 = 853.8 nM T32880 CVZ8E9 145961326 IC50 = 3086 nM T32880 CEJ90L 145961795 IC50 = 853.8 nM T32880 C9R1SO 145961819 IC50 = 69 nM T32880 CB62WJ 145961830 IC50 = 6995 nM T32880 C4C6NP 145962038 IC50 = 995.8 nM T32880 C2Y7SM 145962118 IC50 = 1507 nM T32880 C6D5GL 145962572 IC50 = 608.2 nM T32880 CPO03J 145962836 IC50 = 5527 nM T32880 CJS57A 145962965 IC50 = 2291 nM T32880 C6YJ5R 155539215 IC50 = 905 nM T32880 COL30E 155540589 IC50 = 63 nM T32880 C5MFJ8 155548449 IC50 = 143 nM T32880 CN7H9B 155554391 IC50 = 70 nM T32880 C0GU8Y 155559177 IC50 > 25000 nM T32880 CG7R3L 155559901 IC50 = 4.8 nM T32880 CGU0A2 155563031 IC50 > 25000 nM T32880 C32NYC 155565735 IC50 > 25000 nM T32880 D07IOY 10365 IC50 = 6100 nM T32880 D08IZY 3080614 Ki = 8000 nM T32880 D08JSE 45102710 IC50 = 100 nM T32880 D0B2WZ 15331 IC50 > 100000 nM T32880 D0R6GQ 1198 IC50 > 10000000 nM T32880 D0WA3E 54685215 IC50 = 22 nM T32880 D0X5US 459617 IC50 = 15000 nM T51487 D02YPG 667484 EC50 = 11000 nM T51487 D06ZII 969472 Ki = 50.1 nM T51487 D07JVL 3016 Ki = 16 nM T51487 D0D5GD 3373 Ki = 3.3 nM T51487 D0F0YZ 4737 IC50 = 1000000 nM T51487 D0L9GG 2118 EC50 = 37 nM T51487 D0T1WN 5732 IC50 = 14 nM T51487 D0A5MC 11712649 IC50 = 330 nM T51487 D0CH7C 57336276 Ki = 985 nM T51487 D0HO2T 23581869 Ki = 0.5 nM T51487 D0S4JK 24771867 IC50 = 490 nM T51487 D0Z9HW 23630026 Ki = 0.5 nM T51487 C7SZ9E 613843 IC50 > 10000 nM T51487 C12NWX 2729103 IC50 > 10000 nM T51487 CO61AF 2820320 IC50 > 10000 nM T51487 C59BWK 2820473 IC50 = 470 nM T51487 C1Z6YU 9821389 Ki = 71 nM T51487 CCX58U 9865233 Ki = 0.73 nM T51487 C1VRB9 9951530 EC50 = 56 nM T51487 CPC3U1 9971547 Ki = 362 nM T51487 CUT5W8 9976743 EC50 = 53 nM T51487 CUSM85 10221761 Ki = 1.3 nM T51487 CBQ4R7 10905261 EC50 = 36 nM T51487 C15NXT 10926766 EC50 = 266 nM T51487 CK1S7J 10927005 EC50 = 107 nM T51487 CWK02D 10936672 EC50 = 135 nM T51487 C09PCZ 10971225 EC50 = 92 nM T51487 CG9Z6N 10991911 EC50 = 17 nM T51487 C7DVK8 11014215 EC50 = 120 nM T51487 CJB1V2 11035207 EC50 = 258 nM T51487 C31EGD 11036467 EC50 = 81 nM T51487 CBV36I 11047145 EC50 = 127 nM T51487 C8B7TF 11067772 EC50 = 95 nM T51487 CNSA17 11143256 EC50 = 136 nM T51487 CCU8G9 11526006 IC50 = 150 nM T51487 CWO70Q 11673720 Ki = 15 nM T51487 CX7G9K 11759134 EC50 = 170 nM T51487 CL4XD0 11783674 EC50 = 18 nM T51487 CB9U0F 11825216 EC50 = 28 nM T51487 CTI32Y 15680235 EC50 < 100 nM T51487 C8SR4O 25187292 IC50 = 46 nM T51487 C6DBS4 25187295 IC50 = 50 nM T51487 CF1B8A 25188671 IC50 = 50 nM T51487 CW97NA 44273000 IC50 = 1 nM T51487 C5KV7A 44364531 EC50 = 208 nM T51487 CZK75V 44364548 EC50 = 118 nM T51487 C0FN6W 44364725 EC50 = 2200 nM T51487 CYE1R8 44364726 EC50 = 41 nM T51487 CE8F3Y 44364734 EC50 = 303 nM T51487 COH5G6 44364735 EC50 = 544 nM T51487 C2VHW7 44364747 EC50 = 133 nM T51487 CZL2P0 44364907 EC50 = 69 nM T51487 CCX08E 44364918 EC50 = 93 nM T51487 C6D3BI 44560284 EC50 = 250 nM T51487 C6J0GP 44561356 IC50 = 580 nM T51487 C9UW4V 44561357 IC50 = 580 nM T51487 CZR6A5 44561358 IC50 > 10000 nM T51487 C4IF7B 44561386 IC50 = 1000 nM T51487 C3GZU0 44576235 EC50 = 11000 nM T51487 C63IYQ 51003493 IC50 = 134 nM T51487 CP8IG3 53317278 IC50 = 64 nM T51487 CP9I6O 53319883 IC50 = 74 nM T51487 CO6P3V 53320033 IC50 = 242 nM T51487 CCZ98L 53321188 IC50 = 67 nM T51487 C8MZR1 53322513 IC50 = 157 nM T51487 CTG2S9 53322514 IC50 > 3000 nM T51487 C29ARN 53323855 IC50 = 1 nM T51487 CBGD06 53323856 IC50 = 94 nM T51487 C9DJP1 53326435 IC50 = 64 nM T51487 CBO9L1 60194848 IC50 = 120000 nM T51487 CU83BZ 60194849 IC50 = 3800 nM T51487 CQ91VU 118278442 Ki = 140 nM T51487 CH0D4J 130439777 Ki = 850 nM T51487 C56XBU 130439778 Ki = 55000 nM T51487 C9N8LW 130439889 Ki = 542 nM T51487 C89LNZ 136118605 IC50 = 479 nM T51487 D06SOQ 6918451 Ki = 0.88 nM T51487 D09IHE 6918583 Ki = 0.8 nM T51487 D0E7PY 11624499 Ki = 174 nM T51487 D0M4CP 5081 EC50 = 1.1 nM T51487 D0O9MG 5311203 Ki = 17 nM T52921 D04CRN 54841 IC50 > 5000 nM T52921 D0CS2F 3955 Ki > 10000 nM T52921 D0PG8O 5360515 Ki > 10000 nM T52921 D0U5FS 3396 Ki = 500 nM T52921 D03TBJ 11848225 Ki = 0.9 nM T52921 D0G2XE 6918468 IC50 = 2200 nM T52921 D0W4YO 16131448 Ki = 0.04898 nM T52921 D0M1YN 5311194 Ki = 0.403 nM T52921 D00ACC 9844019 Ki = 1.12 nM T52921 D08AWI 11430856 Ki > 2000 nM T52921 CBGO28 70419 Ki = 11 nM T52921 C3HB4V 416359 IC50 = 200 nM T52921 CQ6MW0 3655995 EC50 = 174 nM T52921 CLW4B1 5311340 Ki = 8.2 nM T52921 CD49UV 9797246 Ki = 133 nM T52921 CNO0W4 9799433 Ki = 5.22 nM T52921 CYR3O0 9802205 Ki = 50.7 nM T52921 CPG57N 9803475 Ki = 12.9 nM T52921 CX7DO4 9806799 Ki = 4.05 nM T52921 CK6GR9 9816910 IC50 > 5000 nM T52921 CE6NF9 9823363 IC50 = 1.3 nM T52921 C6LGX9 9824268 Ki = 82.4 nM T52921 C7TDX2 9824313 Ki = 46.7 nM T52921 C70KEP 9824565 Ki = 0.5 nM T52921 C06LIG 9825723 Ki = 2.3 nM T52921 CPK4X7 9836463 Ki = 1054 nM T52921 C6Y7NA 9844540 Ki = 2 nM T52921 C0F9RX 9845765 Ki = 7 nM T52921 C8M4HT 9846747 Ki = 2.2 nM T52921 CE2YQ9 9848110 Ki = 2 nM T52921 CKD2H4 9848990 Ki = 77 nM T52921 CLQ6Z8 9866158 Ki = 0.5 nM T52921 CEO0M2 9880173 Ki = 414 nM T52921 CPYK08 9887195 IC50 = 820 nM T52921 CV2G7M 9889948 Ki = 11.8 nM T52921 C1VM4H 9902583 Ki = 692 nM T52921 C5BC4P 9902874 Ki = 39 nM T52921 CX3CM8 9905428 Ki = 1.39 nM T52921 C2TE5X 9922658 Ki = 10 nM T52921 C4NJ0W 9923726 Ki = 125 nM T52921 CIUE54 9924406 Ki = 5.4 nM T52921 C5HN0J 9925137 Ki = 1.1 nM T52921 CZT2J0 9927928 Ki = 18.66 nM T52921 C2U8XH 9932834 Ki = 3.4 nM T52921 C9MK3B 9934232 Ki = 6.8 nM T52921 CUBQ95 9937777 Ki = 2.25 nM T52921 C4FD7V 9947044 Ki = 1.4 nM T52921 CG9ER5 9947155 Ki = 2297 nM T52921 COFT18 9951673 Ki = 4 nM T52921 C3GXH0 9954388 Ki = 5.6 nM T52921 CT8C2X 9958643 Ki = 1.8 nM T52921 CE3CJ4 9969865 Ki = 5102 nM T52921 CAGL19 9997843 Ki = 0.7 nM T52921 CL9QS0 10004950 IC50 = 19 nM T52921 C4N8YE 10020165 Ki = 6 nM T52921 C25DYT 10022859 Ki = 0.52 nM T52921 CFOK60 10042904 Ki = 3.96 nM T52921 CC60VS 10052051 Ki = 505 nM T52921 CV1OU6 10109140 Ki = 4.4 nM T52921 C7YCF1 10109899 Ki = 1 nM T52921 CJNE19 10110916 Ki = 225 nM T52921 C76MVA 10111186 Ki > 10000 nM T52921 CWEC34 10114637 Ki = 4461 nM T52921 C40BMF 10133108 Ki = 51 nM T52921 C2WZ9G 10133332 Ki = 1259 nM T52921 CP1SO7 10134077 Ki = 11 nM T52921 CEG0M4 10134217 Ki = 357 nM T52921 C3ZTU0 10137134 Ki = 225 nM T52921 C83KDV 10137876 Ki = 7.4 nM T52921 C8E9KP 10139672 Ki = 41 nM T52921 CQGE97 10150001 Ki = 94 nM T52921 C76SOW 10150260 Ki = 37 nM T52921 CRC46J 10154739 Ki = 634 nM T52921 CKN3A8 10154848 Ki = 410 nM T52921 CFIL01 10155966 Ki = 2.3 nM T52921 CIO6U3 10156336 Ki = 1239 nM T52921 CP53IB 10156591 Ki = 0.4 nM T52921 CI1U4Z 10156821 Ki = 7.5 nM T52921 CTO0N5 10158555 Ki = 31 nM T52921 CG51TX 10159203 Ki = 11 nM T52921 CWM2X6 10160920 Ki = 18 nM T52921 CB57JZ 10171862 Ki = 78 nM T52921 CDV15J 10172398 Ki = 58 nM T52921 CJN21A 10178311 Ki = 184 nM T52921 CHN4G6 10178563 Ki = 824 nM T52921 C5RO6K 10182346 Ki = 7114 nM T52921 CNZL85 10193971 Ki = 347 nM T52921 CN79QX 10194236 Ki = 31 nM T52921 CWC8L1 10199945 IC50 = 2.5 nM T52921 C12NGT 10199984 Ki = 3454 nM T52921 CH40KY 10202108 Ki = 437 nM T52921 CV1T7R 10202241 Ki > 10000 nM T52921 CYB0H9 10221539 IC50 = 3.3 nM T52921 CM27FK 10225083 Ki = 2 nM T52921 CZ0C5T 10252647 Ki = 66 nM T52921 CH54KF 10260917 EC50 = 0.1585 nM T52921 C8PL7B 10274330 Ki = 33 nM T52921 CR1HX2 10275388 Ki = 4358 nM T52921 CSO8D7 10276738 Ki = 0.38 nM T52921 CDP01X 10286440 Ki = 570 nM T52921 C1FE9H 10286996 Ki = 105 nM T52921 CJ14VU 10291377 Ki = 16 nM T52921 C61OKS 10292091 Ki = 111 nM T52921 CV0T3H 10301207 Ki = 1 nM T52921 C1ENR2 10323169 Ki = 2.3 nM T52921 CD09RQ 10338496 Ki = 110 nM T52921 C0G7RF 10362733 Ki = 4544 nM T52921 C59JAP 10363496 Ki = 2.2 nM T52921 CAYF18 10385808 Ki = 2.6 nM T52921 C95EWP 10395965 Ki = 27 nM T52921 CWK4O1 10406239 Ki = 0.1 nM T52921 CTA8Q0 10407144 Ki = 19.6 nM T52921 CX4TS2 10413540 Ki = 78 nM T52921 CYHC38 10430819 Ki = 0.5495 nM T52921 CZP0C7 10441529 EC50 = 0.302 nM T52921 CZ6I9V 10451761 IC50 = 6.8 nM T52921 CKMN08 10475466 Ki = 4.6 nM T52921 C1DI7F 10500922 Ki = 218 nM T52921 C90DEM 10504545 Ki = 6.8 nM T52921 CDK8W2 10548749 Ki = 5.8 nM T52921 C54EOA 10572810 Ki = 7.3 nM T52921 CD9JB5 10574643 Ki = 2.8 nM T52921 CQ74CO 10593778 Ki = 2.5 nM T52921 CZQ4J6 10596013 Ki = 79.9 nM T52921 CHV5D1 10601891 Ki = 15 nM T52921 CS84IW 10618605 Ki = 2.5 nM T52921 CPC52U 10646744 Ki = 7.2 nM T52921 C10KTE 10646745 Ki = 8.5 nM T52921 CH16SQ 10668903 Ki = 85.6 nM T52921 CMT48G 10669669 Ki = 20.4 nM T52921 CF7SX5 10669670 Ki = 13.2 nM T52921 CP25HJ 10669671 Ki = 37.3 nM T52921 CHC1I4 10697286 Ki = 15.3 nM T52921 C2RN9F 10713623 Ki = 10.2 nM T52921 C8XB3K 10714523 Ki = 1.4 nM T52921 CY36JZ 10715725 Ki = 88.5 nM T52921 CFH5N0 10715726 Ki = 121.2 nM T52921 C48PSE 10718869 Ki = 2.6 nM T52921 CN05WO 10763594 Ki = 0.39 nM T52921 CBC6U3 10765154 Ki = 1.8 nM T52921 CXF9R4 10766007 Ki = 1.8 nM T52921 CDJP34 10783436 IC50 = 6.8 nM T52921 CTR2I0 10788833 Ki = 6.5 nM T52921 CQS8K6 10789513 Ki = 1.8 nM T52921 C9SN6H 10831914 Ki = 369.3 nM T52921 CS3Y4G 10832076 IC50 = 5.9 nM T52921 CMVI50 10832445 Ki = 6.3 nM T52921 CPG23C 10836379 Ki = 20.7 nM T52921 C4IT2B 10837001 Ki = 3.3 nM T52921 C2QIL3 10876990 EC50 = 1 nM T52921 CWJL70 10905740 IC50 = 434 nM T52921 C4TSV6 10927662 Ki = 0.5248 nM T52921 C1TSN4 10928037 Ki = 0.7762 nM T52921 CT5UO7 10937810 Ki = 2.188 nM T52921 CU09AV 10937901 IC50 = 38 nM T52921 CVP6D3 10942284 EC50 = 0.2692 nM T52921 CN7XS4 10948527 IC50 = 340 nM T52921 CSLT97 10949380 IC50 = 283 nM T52921 C9FYG3 10950562 Ki = 1.66 nM T52921 CHK23I 10961428 Ki = 1.66 nM T52921 C2HP7F 10981761 IC50 = 758 nM T52921 C78FTE 10986100 EC50 = 63.1 nM T52921 C8Q6YE 11004121 Ki = 0.4467 nM T52921 CIR4E5 11007758 EC50 = 134.9 nM T52921 C0R2DW 11007770 EC50 = 31.62 nM T52921 C3V7LT 11014751 Ki = 0.6457 nM T52921 CY0S2I 11029698 EC50 = 257.04 nM T52921 CRP95V 11051525 EC50 = 0.2512 nM T52921 C9Z7BY 11115933 EC50 = 1.413 nM T52921 CDU0E5 11123873 Ki = 2.089 nM T52921 CU6PV0 11143820 IC50 = 97 nM T52921 C7HM0O 11152739 Ki = 3.5 nM T52921 C26ENL 11164004 Ki = 15.6 nM T52921 C62WBJ 11165726 Ki = 135 nM T52921 C4COM2 11170657 Ki = 0.05 nM T52921 C3TW2O 11187225 Ki = 4.5 nM T52921 C6EWJ9 11188910 Ki = 4.4 nM T52921 CUBX19 11189444 IC50 > 10000 nM T52921 CTKF50 11191683 IC50 = 5.5 nM T52921 CS5ET8 11212373 IC50 > 10000 nM T52921 C26MVG 11223982 IC50 > 10000 nM T52921 C4QT5Y 11233481 Ki = 15.5 nM T52921 CW1O5V 11256620 Ki = 12 nM T52921 CPBZ36 11274537 Ki > 5000 nM T52921 C4FRH7 11315651 Ki = 1.64 nM T52921 C5DBK1 11326750 Ki = 11 nM T52921 CJM7R5 11327115 Ki = 253 nM T52921 CW7SN4 11329662 Ki = 0.5012 nM T52921 CS1W7V 11338717 IC50 > 10000 nM T52921 CY0SV8 11349939 Ki > 10000 nM T52921 C6UZF7 11371415 Ki = 11.7 nM T52921 C4BZ1C 11372427 Ki = 4.3 nM T52921 CQC4G5 11372671 IC50 = 6150 nM T52921 CT6Z0B 11393860 Ki = 29.3 nM T52921 CGO58L 11406629 IC50 = 3700 nM T52921 CBJ0X5 11407510 IC50 > 10000 nM T52921 CU5GO6 11411841 IC50 = 25.2 nM T52921 CW0E4L 11418847 IC50 > 10000 nM T52921 C9KV1U 11451023 Ki = 5.64 nM T52921 C7UDE8 11461888 Ki = 7.49 nM T52921 CF6DQ2 11462727 Ki = 10 nM T52921 CKIQ83 11463791 IC50 > 10000 nM T52921 CC9TX5 11464294 IC50 > 10000 nM T52921 CMU9K5 11464846 Ki = 0.336 nM T52921 C3BA5F 11480038 Ki = 72 nM T52921 CVQ70S 11480201 Ki = 0.04 nM T52921 C41MEV 11511090 IC50 = 0.22 nM T52921 CZ4OM7 11516508 Ki = 2.2 nM T52921 C2N3BS 11523928 IC50 > 1000 nM T52921 CJE45X 11523929 IC50 > 1000 nM T52921 CL1O0H 11523972 IC50 = 350 nM T52921 CQ30PM 11525624 IC50 = 42 nM T52921 C8TZ9G 11544654 IC50 = 32 nM T52921 CS0B4G 11544795 Ki = 2.4 nM T52921 C3DG8U 11552010 Ki = 10.2 nM T52921 C10BUF 11559590 IC50 > 1000 nM T52921 C5ZR9W 11559820 IC50 = 540 nM T52921 CG6UM9 11561261 IC50 > 1000 nM T52921 CRX48F 11581029 Ki = 18.9 nM T52921 CA35LD 11583008 Ki = 4.6 nM T52921 CVA8L6 11583016 IC50 = 4 nM T52921 C1WBQ5 11597677 IC50 = 83 nM T52921 CY72UC 11602409 Ki = 8.5 nM T52921 C0AOU4 11603249 IC50 = 730 nM T52921 C38FTP 11619363 IC50 = 12 nM T52921 C8RKH0 11619553 IC50 = 8.3 nM T52921 C9WMX4 11624970 Ki = 29.8 nM T52921 C34OQC 11626062 Ki = 1.74 nM T52921 CF6R4S 11632761 IC50 > 1000 nM T52921 C4ZD1X 11633324 IC50 = 7.5 nM T52921 CIY0O4 11639705 IC50 > 1000 nM T52921 CFV5Q1 11661648 IC50 > 1000 nM T52921 CPN46U 11676849 IC50 = 580 nM T52921 C4ULQ7 11710187 IC50 = 23 nM T52921 CE0D1U 11743914 Ki = 116 nM T52921 CV8CF3 11749578 IC50 > 10000 nM T52921 CFRY36 11757207 Ki = 15 nM T52921 CED7I5 11761926 Ki = 0.6607 nM T52921 CCY92E 11768467 EC50 = 7.244 nM T52921 CG9HW8 11795019 Ki = 2.9 nM T52921 CN9M8E 11811722 IC50 = 2420 nM T52921 C8UE5W 11826819 Ki = 2.138 nM T52921 CS7W2V 11848793 Ki = 1.7 nM T52921 CJ34HP 11956520 Ki = 0.19 nM T52921 CA5ZX7 11956918 Ki = 9.4 nM T52921 C14RWU 11967729 EC50 = 10.96 nM T52921 CP1AZ0 11967746 EC50 = 26.3 nM T52921 CF01LM 12986253 Ki = 1.9 nM T52921 C63ASY 12986256 Ki = 120 nM T52921 CAW1M2 15512228 Ki = 0.52 nM T52921 C30CHU 15512229 Ki = 0.2512 nM T52921 C9B5OD 15512233 Ki = 39.81 nM T52921 CX6H8V 15512234 Ki = 1.259 nM T52921 CC5X0L 15512235 Ki = 3.981 nM T52921 CG0CS6 15512236 Ki = 15.85 nM T52921 C53KRM 15512237 Ki = 0.3162 nM T52921 CLA5K8 15512238 Ki = 3.981 nM T52921 C4I5TU 15512239 Ki = 10 nM T52921 CSX74V 15512240 Ki = 1.585 nM T52921 CET25R 15512241 Ki = 5.012 nM T52921 C23GHP 15512242 Ki = 100 nM T52921 C7CNY1 15512243 Ki = 1.585 nM T52921 CZA4J8 15541261 Ki = 23 nM T52921 CE18TP 15586319 Ki = 810 nM T52921 CD7K0Y 15965865 IC50 = 6000 nM T52921 CHN45W 15982524 IC50 = 510 nM T52921 CRX3U8 15982526 IC50 = 680 nM T52921 C6DW5M 15982528 IC50 > 10000 nM T52921 C7Z8OD 15982529 IC50 = 7400 nM T52921 CHO67K 15982530 IC50 = 600 nM T52921 C3B8AG 15982657 IC50 = 880 nM T52921 C4W6CK 15982658 IC50 = 140 nM T52921 CLWI08 15982659 IC50 = 10000 nM T52921 CV1G7O 15982660 IC50 = 83 nM T52921 CG3L8Z 15982661 IC50 = 120 nM T52921 CN64AP 15982791 IC50 = 320 nM T52921 C7KXO3 15982794 IC50 > 10000 nM T52921 CB1CR0 15982795 IC50 = 100 nM T52921 C0PKF1 15982796 IC50 = 10000 nM T52921 C3HL5F 15982797 IC50 = 820 nM T52921 CJY21D 15982932 IC50 > 10000 nM T52921 CJ6W1T 15982933 IC50 < 10000 nM T52921 CK97VS 15982935 IC50 = 250 nM T52921 C8TQ4B 15982937 IC50 = 900 nM T52921 C1PB8H 15982938 IC50 = 1120 nM T52921 CS46QG 15983062 IC50 = 800 nM T52921 CXJ61F 15983063 IC50 = 3600 nM T52921 CIG32A 15983065 IC50 = 10000 nM T52921 CG96OQ 15983067 IC50 = 2750 nM T52921 CA5GL7 16007142 Ki = 4 nM T52921 CDR71P 16043240 IC50 > 10000 nM T52921 C4H2NO 16061455 Ki = 6 nM T52921 C08RXS 16665915 Ki = 800 nM T52921 CS9FW1 16665917 Ki = 290 nM T52921 C1LX0I 16665918 Ki = 18 nM T52921 C6W9BJ 16733371 Ki = 6 nM T52921 C4ORI6 16739256 Ki = 15.1 nM T52921 C1MFJ2 16747695 Ki = 4.1 nM T52921 CG84KV 17858339 IC50 = 320 nM T52921 CWXD07 17858448 IC50 = 4.7 nM T52921 C8AZW7 18441735 IC50 = 15000 nM T52921 C1Y9FT 18782352 Ki = 0.9 nM T52921 CYUG80 18782376 Ki = 10.8 nM T52921 C46DPT 18782378 Ki = 2 nM T52921 C73DWV 18782384 Ki = 14.5 nM T52921 CHAI36 22272877 IC50 = 17 nM T52921 C5VSD6 22272900 IC50 = 17 nM T52921 CB5DY1 22272974 IC50 = 3.9 nM T52921 C1NU9M 22273044 IC50 = 2.1 nM T52921 CX3JY4 22273116 IC50 = 120 nM T52921 CRZ72H 22273255 IC50 = 3100 nM T52921 C8DF5U 22558157 Ki = 12 nM T52921 C1R5PV 22562132 Ki = 5670 nM T52921 CJ8OB0 22562135 Ki = 3592 nM T52921 C0GKU4 22562137 Ki = 20.4 nM T52921 CJ86RS 22725091 Ki = 10 nM T52921 CL7X2U 23383556 Ki = 0.4 nM T52921 COHN67 23383564 Ki = 0.5 nM T52921 C46ZSX 23542099 IC50 = 34 nM T52921 CVLY78 23542106 IC50 = 82 nM T52921 CB9MC8 24735827 Ki = 119 nM T52921 CWP85S 24776395 Ki = 3.1 nM T52921 CVD48X 24776396 Ki = 186 nM T52921 C3WDL8 24776397 Ki = 8.9 nM T52921 CXL4R0 24776398 Ki = 21 nM T52921 CR9I1S 24776399 Ki = 395 nM T52921 CQDJ35 24776400 Ki = 147 nM T52921 C6CX0Z 24776401 Ki = 6.6 nM T52921 CJH18I 24776402 Ki = 12 nM T52921 C27SGI 24776403 Ki = 26 nM T52921 CV5IG2 24776404 Ki = 51 nM T52921 CQ70IW 24776405 Ki = 81 nM T52921 CQ2P5J 24776406 Ki = 136 nM T52921 CYIV42 24776407 Ki = 4.7 nM T52921 CWB06Z 24776408 Ki = 23 nM T52921 C36WQO 24776409 Ki = 42 nM T52921 CUP2C6 24776410 Ki = 90 nM T52921 CC3W7E 24776411 Ki = 130 nM T52921 C3N6GE 24776412 Ki = 65 nM T52921 C2M6BR 24776413 Ki = 92 nM T52921 C8SXV9 24799146 Ki = 180 nM T52921 C1S2NC 24799325 Ki = 104 nM T52921 CLAU56 24799509 Ki = 100 nM T52921 C2VHP0 24799848 Ki = 545 nM T52921 C26ZYM 24800015 Ki = 260 nM T52921 CWV5F4 24800016 Ki = 740 nM T52921 CS01RL 24800107 Ki = 2.1 nM T52921 CL2WB0 24800108 Ki = 0.0858 nM T52921 CY89FP 24800188 Ki = 186 nM T52921 C13MJI 24822630 EC50 = 0.1 nM T52921 C6TWH4 24824635 EC50 = 88 nM T52921 CYM02E 24847114 IC50 = 15 nM T52921 C9O5NZ 24857819 IC50 = 0.65 nM T52921 CN0T1F 24857820 IC50 = 0.66 nM T52921 CS5D1K 24882570 IC50 = 0.033 nM T52921 CQ63PM 24894425 Ki = 17 nM T52921 C2EQR6 24894426 Ki = 0.47 nM T52921 CT9EZ4 24894428 Ki = 1.1 nM T52921 CN1E8M 24894430 Ki = 30 nM T52921 C9USO6 24894431 Ki = 58 nM T52921 C4IDR3 24894531 Ki = 11 nM T52921 CA8E4J 24894533 Ki = 21 nM T52921 C2AU5Y 24894647 Ki = 20 nM T52921 C8JL9I 24894652 Ki = 49 nM T52921 C6AZ9P 24894653 Ki = 25 nM T52921 CC6F9D 24894783 Ki = 51 nM T52921 CDLW86 25001412 Ki = 0.7244 nM T52921 CBIU48 25077447 EC50 = 4.37 nM T52921 CFB8G1 25077910 EC50 = 25 nM T52921 CHWB32 25082025 EC50 = 156 nM T52921 C2FPI9 25084159 EC50 = 22.3 nM T52921 C6HL3Q 25089553 EC50 = 0.1349 nM T52921 CP56DF 25089995 IC50 = 0.471 nM T52921 CF6RA5 25190572 Ki = 84 nM T52921 CPK5D7 25190573 Ki = 34 nM T52921 CON62K 25190574 Ki = 57 nM T52921 C6S3WN 25190575 Ki = 83 nM T52921 CF15AH 25190576 Ki = 53 nM T52921 CBN1Q0 25190577 Ki = 89 nM T52921 CKB72D 25190578 Ki = 234 nM T52921 CZR78G 25190579 Ki = 203 nM T52921 CF2JK0 25190580 Ki = 48.7 nM T52921 CE4R2X 25190581 Ki = 56 nM T52921 CYC6S0 25190582 Ki = 19.5 nM T52921 CE61QB 25190583 Ki = 18.5 nM T52921 C9V8MS 25190584 Ki = 26 nM T52921 C3UV5M 25190585 Ki = 47.8 nM T52921 CKFI42 25190586 Ki = 2.1 nM T52921 C5UQX3 25190587 Ki = 2.55 nM T52921 C5J2WE 25190588 Ki = 8.65 nM T52921 CX84WI 25190589 Ki = 5 nM T52921 C5RUI9 25190590 Ki = 3.5 nM T52921 CQY69C 25190591 Ki = 3.7 nM T52921 C8SEQ2 25190592 Ki = 12.1 nM T52921 C5BS7N 25190593 Ki = 2.15 nM T52921 CE19OU 25190594 Ki = 2.75 nM T52921 CP5ID6 25190595 Ki = 3.8 nM T52921 CO8E4G 25190596 Ki = 3.2 nM T52921 CX87HD 25190597 Ki = 8 nM T52921 CY6CV1 25190598 Ki = 2.3 nM T52921 CW5UP9 25190599 Ki = 0.8 nM T52921 C1C8VK 25190600 Ki = 0.7 nM T52921 CL7Q2F 25190601 Ki = 0.7 nM T52921 CD0H5U 25190602 Ki = 0.5 nM T52921 C8OWC0 25190603 Ki = 0.5 nM T52921 CH06YU 25190604 Ki = 0.6 nM T52921 CEJ25L 25190605 Ki = 0.5 nM T52921 CXD5R8 25190606 Ki = 1 nM T52921 CU6W8O 25190607 Ki = 5.4 nM T52921 CWJB54 25190608 Ki = 4.5 nM T52921 CMHS48 25190609 Ki = 1.7 nM T52921 CBL9S4 25190610 Ki = 2.1 nM T52921 CZ8Y6L 25190611 Ki = 1.6 nM T52921 CL9SN6 25190612 Ki = 1.4 nM T52921 C1MGY3 25190613 Ki = 0.9 nM T52921 CB1G6M 25190614 Ki = 0.9 nM T52921 CJLH27 25190615 Ki = 1 nM T52921 COE65V 25190616 Ki = 0.9 nM T52921 C30VGA 25190617 Ki = 1.5 nM T52921 CO7IV2 25190618 Ki = 0.8 nM T52921 C8Q7WV 25190619 Ki = 0.5 nM T52921 C0G4RJ 25190620 Ki = 6.7 nM T52921 C7X4IV 25190621 Ki = 1.4 nM T52921 CXG8O3 25190622 Ki = 0.5 nM T52921 CD5F6A 25190623 Ki = 0.4 nM T52921 CFUD47 25190624 Ki = 1.3 nM T52921 C15LIW 25190625 Ki = 0.7 nM T52921 C3LEW8 25190626 Ki = 3.6 nM T52921 CIDV61 25190627 Ki = 15.9 nM T52921 CAGS39 25190628 Ki = 1.8 nM T52921 CDS2E6 25190629 Ki = 0.6 nM T52921 CPW19O 25190630 Ki = 12.2 nM T52921 C0SBV7 25207946 Ki = 0.63 nM T52921 C21OJF 25207948 Ki = 0.3 nM T52921 C0P6CS 25207950 Ki = 0.18 nM T52921 CN9I8E 25208095 Ki = 0.2 nM T52921 C5OA1N 25208097 EC50 = 0.02512 nM T52921 C59IKP 25208099 Ki = 0.24 nM T52921 CUNA84 25208101 Ki = 0.15 nM T52921 C2WIG0 25208245 Ki = 0.22 nM T52921 CE4BI6 25208247 Ki = 1.7 nM T52921 CKNE16 25208249 Ki = 0.53 nM T52921 CB04CU 25235412 Ki = 20 nM T52921 CL2Z7J 42629117 EC50 = 14 nM T52921 CWJ2E3 43406622 IC50 > 1000 nM T52921 C49YRK 44143406 IC50 = 350 nM T52921 C3YMQ1 44143407 IC50 = 150 nM T52921 CBFR50 44143408 IC50 = 150 nM T52921 C4BOI0 44143409 IC50 = 75 nM T52921 CRL9K5 44143410 IC50 > 1000 nM T52921 CB4O2Y 44143411 IC50 > 1000 nM T52921 C0JS3Q 44143412 IC50 = 560 nM T52921 C6U7HP 44143413 IC50 = 28 nM T52921 C1TSC2 44143414 IC50 = 530 nM T52921 CAB3T9 44143415 IC50 = 37 nM T52921 CD26LJ 44143416 IC50 > 1000 nM T52921 CG3PW7 44143417 IC50 = 61 nM T52921 CB94OV 44143418 IC50 = 11 nM T52921 COP5W8 44143419 IC50 = 4 nM T52921 CY26BG 44143420 IC50 = 67 nM T52921 C8WLP6 44143421 IC50 = 270 nM T52921 C3S1PL 44143422 IC50 = 13 nM T52921 C05AWH 44143423 IC50 = 33 nM T52921 C4D0YQ 44143424 IC50 = 36 nM T52921 C5CR3I 44143425 IC50 = 72 nM T52921 CQE5U4 44143426 IC50 = 8.2 nM T52921 CZR49E 44143427 IC50 = 7.1 nM T52921 C63RXB 44143428 IC50 = 2.5 nM T52921 C8OH4S 44143429 IC50 = 4.5 nM T52921 CTE6S1 44143430 IC50 = 1.2 nM T52921 CL57VS 44143431 IC50 = 0.52 nM T52921 C2C5QW 44143432 IC50 = 0.72 nM T52921 C6GDL8 44143433 IC50 = 0.81 nM T52921 C3BNV0 44143434 IC50 = 5.7 nM T52921 CXV0B8 44143435 IC50 = 2 nM T52921 CN7HE0 44143436 IC50 = 38 nM T52921 C9CJN0 44143437 IC50 = 0.8 nM T52921 C6INT4 44143438 IC50 = 2.9 nM T52921 CJ46YA 44143439 IC50 = 23 nM T52921 CZ15CE 44143440 IC50 = 630 nM T52921 C0KB7Y 44143441 IC50 = 61 nM T52921 C3RF4I 44143442 IC50 = 27 nM T52921 CE20LQ 44143444 IC50 = 22 nM T52921 CFH9T2 44143445 IC50 = 21 nM T52921 C5NZM3 44143446 IC50 = 1.1 nM T52921 CGSW03 44143448 IC50 = 1.1 nM T52921 CBWD06 44143449 IC50 = 2.1 nM T52921 C2ST5N 44143450 IC50 = 1.4 nM T52921 CF4V5K 44143451 IC50 = 1 nM T52921 CL3R6D 44143452 IC50 = 4 nM T52921 C8IG1V 44143453 IC50 = 0.9 nM T52921 C2Q3DE 44143454 IC50 = 3.7 nM T52921 CZX75A 44143455 IC50 = 0.91 nM T52921 C02YJQ 44143456 IC50 = 1.1 nM T52921 CZV0C7 44143457 IC50 = 1.8 nM T52921 CPQ25W 44181744 Ki = 5 nM T52921 C2XE7Y 44189733 IC50 = 2.3 nM T52921 CGA8R1 44189735 IC50 = 1.9 nM T52921 C50FOG 44189834 IC50 = 2.3 nM T52921 CC63QX 44247589 Ki = 7 nM T52921 CP8Q5B 44248550 Ki = 7 nM T52921 CZNM65 44248674 Ki = 1 nM T52921 CIJF67 44248788 Ki = 272 nM T52921 C9G8KT 44248789 Ki = 34 nM T52921 C9JBR1 44248790 Ki = 22 nM T52921 C5YV0D 44248791 Ki = 14 nM T52921 C1CZ3M 44248792 Ki = 24 nM T52921 CDG15Z 44248915 Ki = 23 nM T52921 C5I7YZ 44248916 Ki = 29 nM T52921 C5T9AP 44248917 Ki = 467 nM T52921 CAY83B 44248918 Ki = 18 nM T52921 CL61MJ 44248919 Ki = 25 nM T52921 C2FLP9 44248920 Ki = 10 nM T52921 C6Q5ZF 44249045 Ki = 9 nM T52921 C0HWG8 44249046 Ki = 9 nM T52921 CHLS96 44249047 Ki = 5 nM T52921 CO4EA3 44249048 Ki = 69 nM T52921 CW6P4Y 44276782 Ki = 89 nM T52921 C9AF6B 44297435 Ki = 28.7 nM T52921 CNP5W1 44297519 Ki = 786 nM T52921 C52MGY 44297539 Ki = 0.49 nM T52921 C9UY4E 44297697 Ki = 535 nM T52921 C8F1ST 44297727 Ki = 189 nM T52921 C7ZYM4 44299404 Ki > 10000 nM T52921 CK6IY4 44315305 Ki = 10 nM T52921 CQ0OK5 44327446 EC50 = 0.7586 nM T52921 CAS38O 44332117 Ki = 4.67 nM T52921 CGZ9N2 44336905 Ki = 191 nM T52921 CYMH75 44337108 Ki = 420 nM T52921 CJ0I6Q 44337123 Ki = 64 nM T52921 CPOX86 44337129 Ki = 7222 nM T52921 CT78UG 44337131 Ki = 14 nM T52921 CO8Y5G 44337163 Ki = 745 nM T52921 CBJ01F 44337212 Ki = 49 nM T52921 C8IJM5 44337229 Ki = 26 nM T52921 C97YKG 44337230 Ki = 1062 nM T52921 C3B4WO 44337231 Ki = 1135 nM T52921 CU8IY3 44337232 Ki = 2532 nM T52921 C3M0QX 44337249 Ki = 680 nM T52921 C0MJL2 44337252 Ki = 1345 nM T52921 CB85KA 44337351 Ki = 94 nM T52921 CI13YG 44337357 Ki = 152 nM T52921 CW2FZ7 44337362 Ki = 198 nM T52921 CJ08FM 44337379 Ki = 30 nM T52921 CIP87K 44337437 Ki = 185 nM T52921 CR62KO 44337452 Ki = 79 nM T52921 C9CIP3 44337459 Ki = 3221 nM T52921 CFA2Q7 44337460 Ki = 684 nM T52921 CZP4K1 44337461 Ki = 2593 nM T52921 CF96JK 44337473 Ki = 367 nM T52921 CX87AS 44337513 Ki = 772 nM T52921 CP1VN3 44337550 Ki = 1016 nM T52921 CZ02BO 44337551 Ki = 34 nM T52921 CS9Z1O 44339374 Ki = 225 nM T52921 C73CSH 44339393 Ki = 153 nM T52921 CF08RA 44339398 Ki > 10000 nM T52921 CFNR91 44339423 Ki = 33 nM T52921 CW56BK 44339424 Ki = 12 nM T52921 C4POK5 44339425 Ki = 135 nM T52921 C03PDA 44339449 Ki = 692 nM T52921 CGI10R 44339450 Ki = 715 nM T52921 C7HIP9 44339463 Ki = 879 nM T52921 CQ24IT 44339491 Ki > 10000 nM T52921 CC1VG7 44339500 Ki = 234 nM T52921 C73QPW 44339504 Ki = 502 nM T52921 CABQ05 44339505 Ki = 1270 nM T52921 C7GRF4 44339525 Ki = 1194 nM T52921 CY85GQ 44339526 Ki = 6520 nM T52921 CZRJ83 44339528 Ki > 10000 nM T52921 CKP7R5 44339529 Ki > 10000 nM T52921 CAD1O4 44339530 Ki = 1106 nM T52921 CIZU20 44339531 Ki > 10000 nM T52921 C2LQO7 44339540 Ki = 307 nM T52921 C7E4MS 44339576 Ki = 47 nM T52921 C2PDT6 44339596 Ki = 102 nM T52921 C34DEN 44339684 Ki = 82 nM T52921 CO3C7M 44339695 Ki = 12 nM T52921 CGY16P 44339707 Ki = 827 nM T52921 CD9ZS8 44342270 IC50 = 1910 nM T52921 C4BK0O 44352743 EC50 = 439 nM T52921 CHX36W 44352744 EC50 = 286 nM T52921 C9RN1Y 44352745 IC50 = 2710 nM T52921 C1GZ8E 44352920 IC50 = 874 nM T52921 CD18TR 44366689 Ki = 2130 nM T52921 CYL95J 44366690 Ki = 35 nM T52921 C7IFR8 44366822 Ki = 34 nM T52921 CL1JV2 44366823 Ki = 44 nM T52921 CX7A3N 44388460 EC50 = 0.06607 nM T52921 CLV18K 44388461 EC50 = 0.1 nM T52921 CK95WL 44388462 EC50 = 0.06761 nM T52921 C5FA4H 44388465 EC50 = 0.4786 nM T52921 CBUS05 44388466 EC50 = 0.2399 nM T52921 CJG21X 44388467 EC50 = 0.2089 nM T52921 CZ7L6C 44388472 EC50 = 5.888 nM T52921 C4WRI8 44388474 EC50 = 0.4074 nM T52921 C5I7AN 44390989 Ki = 12 nM T52921 C2TP3J 44390999 Ki = 620 nM T52921 C9FBO3 44391012 Ki = 1115 nM T52921 C2W7BJ 44391023 Ki = 282 nM T52921 C4BF2U 44391031 Ki = 905 nM T52921 CF49QH 44391052 Ki = 32 nM T52921 C7A8DM 44391062 Ki = 10.8 nM T52921 CTA04B 44391063 Ki = 462 nM T52921 C1WGX6 44391067 Ki = 52 nM T52921 C8Y7OV 44391069 Ki = 218 nM T52921 CT8W3P 44391075 Ki = 1920 nM T52921 CY7OH0 44391079 Ki = 42 nM T52921 CPZ7L8 44391081 Ki = 28 nM T52921 CR5TN7 44391092 Ki = 37 nM T52921 C2DB4N 44391093 Ki = 768 nM T52921 CO2T5M 44391094 Ki = 14 nM T52921 CL79EO 44391099 Ki = 838 nM T52921 C3HTZ1 44391102 Ki = 509 nM T52921 CW76ZY 44391103 Ki = 24 nM T52921 CN1LD9 44391104 Ki = 38.2 nM T52921 CD3QV8 44391111 Ki = 60 nM T52921 CK2HV1 44391119 Ki = 113 nM T52921 C8RDV5 44391124 Ki = 3 nM T52921 C1UDL9 44391133 Ki = 20 nM T52921 CSV6X2 44391134 Ki = 25 nM T52921 CJ9MX1 44391137 Ki = 815 nM T52921 C18SDI 44391138 Ki = 126 nM T52921 C6ZF9E 44391155 Ki = 8.3 nM T52921 CY6T4F 44391156 Ki = 108 nM T52921 CJB0U8 44391157 Ki = 39 nM T52921 C5ZFX2 44394283 Ki = 231 nM T52921 COB70L 44394284 Ki = 40 nM T52921 C5BTZ1 44394320 Ki = 1878 nM T52921 C6DB4X 44394324 Ki = 28.7 nM T52921 C2OV9B 44394344 Ki = 46 nM T52921 C1Y3NV 44394345 Ki = 2614 nM T52921 CCR2U1 44394375 Ki = 83 nM T52921 CQ2O6J 44394381 Ki = 3.9 nM T52921 CTJ2I9 44394405 Ki = 63 nM T52921 CLFU54 44394419 Ki = 187 nM T52921 C0A1OW 44394487 Ki = 5 nM T52921 C61AXY 44394529 Ki = 9535 nM T52921 CRCV49 44394559 Ki = 609 nM T52921 C3YD8C 44395259 Ki > 10000 nM T52921 CR8AF5 44395265 Ki > 10000 nM T52921 CI7GR3 44395286 Ki = 149 nM T52921 CLB5E3 44395291 Ki > 10000 nM T52921 CEX0W2 44395306 Ki = 590 nM T52921 C69ACH 44395319 Ki > 10000 nM T52921 CQO0Y5 44395366 Ki > 10000 nM T52921 C0FUP2 44395387 Ki > 10000 nM T52921 C06LKH 44395410 Ki = 372 nM T52921 C7GP1E 44404646 IC50 = 290 nM T52921 CILB28 44404652 IC50 = 380 nM T52921 C38GAM 44404653 IC50 = 1310 nM T52921 CA58SU 44404670 IC50 = 120 nM T52921 C83PCH 44404679 IC50 = 100 nM T52921 CU0YX9 44404684 IC50 = 2400 nM T52921 CEJ7F8 44404689 IC50 = 2680 nM T52921 CD8M2R 44404693 IC50 = 710 nM T52921 C5X8YK 44404694 IC50 = 470 nM T52921 CODG94 44404695 IC50 = 150 nM T52921 CD79WM 44404698 IC50 = 450 nM T52921 C0BED6 44404699 IC50 = 37 nM T52921 CGA15Y 44404706 IC50 = 10000 nM T52921 C2NHS0 44404707 IC50 > 10000 nM T52921 CJCY60 44404711 IC50 = 1080 nM T52921 CK73OG 44404721 IC50 = 350 nM T52921 CNX5T8 44404731 IC50 = 180 nM T52921 CW9QG2 44406457 IC50 > 10000 nM T52921 CGN73V 44406458 IC50 > 10000 nM T52921 C0J7IK 44406489 IC50 = 6000 nM T52921 C5TIM4 44406497 IC50 = 1000 nM T52921 CBUR32 44406503 IC50 = 10000 nM T52921 C17FYG 44406538 IC50 = 15000 nM T52921 C07CNE 44406539 IC50 = 7000 nM T52921 C5DGV2 44406540 IC50 = 3850 nM T52921 C9Z0ET 44406541 IC50 > 10000 nM T52921 C1L8CG 44406543 IC50 = 10400 nM T52921 CP1OZ6 44406544 IC50 > 10000 nM T52921 CS04TK 44406550 IC50 = 5800 nM T52921 C8HRC9 44406551 IC50 = 15000 nM T52921 CSPE30 44406557 IC50 = 13400 nM T52921 CD7Y0Z 44406585 IC50 > 10000 nM T52921 CC15BY 44406587 IC50 = 10000 nM T52921 C1IM9R 44406603 IC50 = 1000 nM T52921 C3VE8N 44406604 IC50 = 1000 nM T52921 CCI5Z1 44406618 IC50 = 300 nM T52921 C7ES2W 44406621 IC50 = 130 nM T52921 C0SKT9 44406641 IC50 > 10000 nM T52921 C38ABN 44406682 IC50 > 10000 nM T52921 CZ65PF 44406685 IC50 > 10000 nM T52921 CWY76P 44406719 IC50 = 4000 nM T52921 CP5H7S 44406907 IC50 > 1000 nM T52921 CHKO45 44406969 IC50 > 1000 nM T52921 CV4C6R 44406970 IC50 > 1000 nM T52921 C7BNY9 44406975 IC50 > 1000 nM T52921 C0W1EN 44406978 IC50 > 1000 nM T52921 C5U7KF 44406979 IC50 > 1000 nM T52921 CM31XO 44406989 IC50 > 1000 nM T52921 CC0H4U 44406991 IC50 > 1000 nM T52921 CNP5V6 44406994 IC50 > 1000 nM T52921 C3BQ7S 44406995 IC50 > 1000 nM T52921 C92ZTH 44406996 IC50 > 1000 nM T52921 CN82CH 44406997 IC50 > 1000 nM T52921 CX20ZA 44406998 IC50 > 1000 nM T52921 CMRF31 44407013 IC50 = 630 nM T52921 C8RNE9 44407016 IC50 > 1000 nM T52921 CA2OD1 44407020 IC50 = 870 nM T52921 C0OB8F 44407023 IC50 > 1000 nM T52921 C21UFE 44407028 IC50 > 1000 nM T52921 C8GK1Q 44407036 IC50 > 1000 nM T52921 CGO7M0 44407037 IC50 > 1000 nM T52921 C4YW1C 44407038 IC50 > 1000 nM T52921 C4QT3D 44407040 IC50 > 1000 nM T52921 CK84HW 44407043 IC50 > 1000 nM T52921 CZ8D9R 44407044 IC50 = 30 nM T52921 C7QWZ5 44407048 IC50 = 360 nM T52921 CYJ04D 44407049 IC50 > 1000 nM T52921 CJ4A2W 44407050 IC50 > 1000 nM T52921 CU20IA 44407063 IC50 > 1000 nM T52921 C5PDG8 44407065 IC50 > 1000 nM T52921 CGAD30 44407066 IC50 > 1000 nM T52921 CT49JG 44407070 IC50 = 170 nM T52921 C9WJZ5 44407074 IC50 > 1000 nM T52921 CW2CP3 44407078 IC50 > 1000 nM T52921 CL9QK6 44407080 IC50 > 1000 nM T52921 C2S5NT 44407081 IC50 > 1000 nM T52921 C0QB6E 44407084 IC50 = 131 nM T52921 CLG4Y9 44407085 IC50 = 230 nM T52921 CPQ7H2 44407086 IC50 = 290 nM T52921 C0K7ZH 44407091 IC50 > 1000 nM T52921 CM8JK6 44407109 IC50 > 1000 nM T52921 C8R1QN 44407112 IC50 = 340 nM T52921 CEZ4I2 44407113 IC50 > 1000 nM T52921 CA3OW4 44407116 IC50 = 21 nM T52921 CLE6W9 44407119 IC50 > 1000 nM T52921 CK4NE2 44407129 IC50 = 50 nM T52921 CKUT49 44407133 IC50 = 24 nM T52921 COS85F 44407140 IC50 = 330 nM T52921 CAMX28 44407145 IC50 > 1000 nM T52921 CRP3D2 44407146 IC50 > 1000 nM T52921 CZO5R6 44407156 IC50 = 900 nM T52921 C2YME3 44413175 IC50 > 1000 nM T52921 CM7LE4 44413183 IC50 > 1000 nM T52921 C0M9TX 44413184 IC50 > 1000 nM T52921 CFJ64A 44413232 Ki = 970 nM T52921 CNFC81 44413248 Ki > 5000 nM T52921 C0V4FI 44413286 Ki = 550 nM T52921 CS7BI8 44413301 Ki = 81 nM T52921 C1NGS0 44413314 Ki = 94 nM T52921 C5J0BU 44413315 Ki > 5000 nM T52921 CH7E1C 44413329 Ki > 5000 nM T52921 C1OQ0L 44413330 Ki = 2 nM T52921 CKV5S0 44413361 Ki = 52 nM T52921 C5PHK7 44413362 Ki = 62 nM T52921 CSQZ28 44413379 Ki > 5000 nM T52921 CCU2B5 44413384 Ki = 660 nM T52921 CD5SZ9 44413385 Ki = 57 nM T52921 C7GE2K 44413395 Ki > 5000 nM T52921 CCK6Y5 44413396 Ki = 1650 nM T52921 C0FL8K 44413401 Ki = 3500 nM T52921 C6J3HP 44413402 Ki > 5000 nM T52921 CB2OJ9 44413408 Ki = 160 nM T52921 C82VJB 44413413 Ki > 5000 nM T52921 CP31JV 44413414 Ki = 820 nM T52921 C98OQG 44413423 Ki > 5000 nM T52921 CH0DS7 44413441 Ki = 710 nM T52921 CLSK72 44413442 Ki = 10 nM T52921 C6O2VL 44414730 IC50 > 10000 nM T52921 C5Z9VE 44414845 IC50 > 10000 nM T52921 C4LI9Q 44414865 IC50 > 10000 nM T52921 C10OMS 44426811 Ki = 9 nM T52921 C49KAS 44426813 Ki = 41 nM T52921 CJK6Y5 44426815 Ki = 4035 nM T52921 CJ5FC0 44426816 Ki = 295 nM T52921 C4TFP1 44426818 Ki = 1887 nM T52921 CP1Z5J 44426819 Ki = 10000 nM T52921 CP5V8D 44426821 Ki = 8183 nM T52921 C5L4SE 44426822 Ki = 214 nM T52921 C36SCP 44426823 Ki = 323 nM T52921 C72RXV 44426824 Ki = 35 nM T52921 C0S5TE 44426829 Ki = 12 nM T52921 CL1EG2 44426830 Ki = 357 nM T52921 CBFY73 44426831 Ki = 225 nM T52921 CFO9Q6 44426832 Ki = 0.6 nM T52921 C2NFA4 44426833 Ki = 26 nM T52921 COJ48Z 44426834 Ki = 132 nM T52921 CUD42S 44426835 Ki = 5 nM T52921 CKJ90O 44426836 Ki = 11 nM T52921 CZ4R6J 44426837 Ki = 125 nM T52921 CPDE73 44426838 Ki = 9 nM T52921 C53JGK 44426839 Ki = 6753 nM T52921 C7IJY0 44426840 Ki = 6 nM T52921 CJB90W 44426841 Ki = 42 nM T52921 C4Z1FX 44426842 Ki = 21 nM T52921 CK3B6E 44426843 Ki = 3 nM T52921 CD3TB8 44426844 Ki = 439 nM T52921 CF5OJ0 44430021 Ki = 1449 nM T52921 CUQ95Y 44430022 Ki = 16 nM T52921 CZA0E6 44430023 Ki = 1.6 nM T52921 CWX67P 44430033 Ki = 15 nM T52921 C40BHT 44430038 Ki = 0.4 nM T52921 C1QXR6 44430040 Ki = 0.7 nM T52921 CS6Y5Z 44430042 Ki = 0.5 nM T52921 C4CHV5 44430043 Ki = 1.1 nM T52921 CX9P5R 44430044 Ki = 0.5 nM T52921 CA51JN 44430045 Ki = 110 nM T52921 C2G9HQ 44430046 Ki = 674 nM T52921 C8PI4A 44430047 Ki = 9.6 nM T52921 CL1N4D 44430048 Ki = 4.6 nM T52921 C0AYM6 44430049 Ki = 5.5 nM T52921 CMJT74 44430050 Ki = 0.7 nM T52921 C4ZG6A 44430079 Ki = 2 nM T52921 CSNQ43 44430080 Ki = 12 nM T52921 CXV9J7 44430081 Ki = 5.9 nM T52921 CFHY18 44430083 Ki = 1.9 nM T52921 C6SBE1 44430084 Ki = 2.2 nM T52921 CXZ2D3 44430085 Ki = 0.9 nM T52921 CI4X3Z 44430087 Ki = 0.6 nM T52921 C8D0ZX 44431782 Ki = 1273 nM T52921 CT30KJ 44437601 Ki = 3 nM T52921 C1EHS4 44437602 Ki = 2 nM T52921 CX5O0J 44437604 Ki = 5 nM T52921 CWOJ02 44437605 Ki = 3 nM T52921 CK73VO 44437606 Ki = 3 nM T52921 CJ1ST3 44437610 Ki = 0.5 nM T52921 CFH6A5 44437613 Ki = 22 nM T52921 C0M9SC 44437615 Ki = 4 nM T52921 CFN8Z9 44437617 Ki = 6 nM T52921 CTK2S0 44437619 Ki = 1 nM T52921 C4PK1O 44437623 Ki = 5 nM T52921 CP4HR6 44437626 Ki = 4 nM T52921 CA5S2P 44437627 Ki = 46 nM T52921 CKEG06 44437628 Ki = 12 nM T52921 CT7V0O 44437629 Ki = 1595 nM T52921 C45ZTN 44437630 Ki = 10 nM T52921 CQKL94 44437636 Ki = 4 nM T52921 C43URV 44437637 Ki = 3 nM T52921 CJ8L4A 44437638 Ki = 2 nM T52921 CNBQ93 44437639 Ki = 5 nM T52921 C2AV5I 44437640 Ki = 19 nM T52921 CN3R5G 44437641 Ki = 29 nM T52921 C6NA9R 44437642 Ki = 20 nM T52921 CH5RW4 44437643 Ki = 155 nM T52921 C7RIC8 44437644 Ki = 15 nM T52921 C5IL8O 44437645 Ki = 20 nM T52921 CX1S4V 44437646 Ki = 12 nM T52921 CV19NL 44437647 Ki = 29 nM T52921 C02YET 44437648 Ki = 12 nM T52921 CJ2PH5 44437649 Ki = 3 nM T52921 CVH1I9 44437652 Ki = 23 nM T52921 C0ME9B 44437654 Ki = 2 nM T52921 CRKH10 44437656 Ki = 2 nM T52921 CZB4Q9 44438912 Ki = 61.2 nM T52921 CP85QV 44438914 Ki = 824 nM T52921 C7RD2E 44438916 Ki = 14 nM T52921 CNL30S 44438917 Ki = 3.2 nM T52921 C5D4NZ 44438920 Ki = 3.5 nM T52921 CA2LD5 44438921 Ki = 17 nM T52921 C6H7AD 44438922 Ki = 2.4 nM T52921 CRN3W4 44438961 Ki = 1.1 nM T52921 CGYD89 44438962 Ki = 1.5 nM T52921 CZ48KD 44438963 Ki = 36.5 nM T52921 C2EGK7 44438964 Ki = 10.8 nM T52921 COX57F 44438965 Ki = 9 nM T52921 C9S2HB 44438966 Ki = 11.5 nM T52921 C1HF6E 44438967 Ki = 140 nM T52921 C3L7SB 44438968 Ki = 9 nM T52921 CE63GK 44438971 Ki = 249 nM T52921 C8TVI4 44438974 Ki = 6.3 nM T52921 CPHS56 44438975 Ki = 250 nM T52921 CK3Z5G 44438978 Ki = 49 nM T52921 CPA4U5 44438983 Ki = 0.3 nM T52921 C2TKY5 44438988 Ki = 0.8 nM T52921 CL7WN5 44438993 Ki = 2.6 nM T52921 C0A2OM 44439000 Ki = 1.4 nM T52921 CMQA60 44439001 Ki = 8.4 nM T52921 CN4KX9 44449764 IC50 = 31 nM T52921 CWN0C3 44449766 IC50 = 78 nM T52921 CE97XC 44449767 IC50 = 180 nM T52921 C7NKJ3 44449771 IC50 = 140 nM T52921 CRO1B7 44449793 IC50 = 2900 nM T52921 CTMI71 44449822 IC50 = 63 nM T52921 CU6I5Y 44449823 IC50 > 10000 nM T52921 C8QE6N 44449850 IC50 = 8200 nM T52921 CH5MN1 44449851 IC50 = 910 nM T52921 CT39QP 44450085 IC50 = 1.8 nM T52921 C1SQ7M 44450086 IC50 = 20 nM T52921 CGN7O0 44450151 IC50 = 15 nM T52921 CS4DO9 44450180 IC50 = 240 nM T52921 CL5K3J 44450207 IC50 = 2900 nM T52921 CK41RX 44450208 IC50 = 140 nM T52921 CUR83O 44450209 IC50 = 380 nM T52921 C37FVM 44450210 IC50 = 55 nM T52921 CL78ZG 44451517 Ki = 3.548 nM T52921 CG2WD7 44451518 Ki = 21.88 nM T52921 CBK6R5 44451542 Ki = 3.89 nM T52921 CC36BM 44451543 Ki = 2.512 nM T52921 CKB0F9 44451569 Ki = 1.698 nM T52921 C2EJP0 44451572 Ki = 28.84 nM T52921 CYQ53B 44451573 Ki = 1174.9 nM T52921 CGJ3R8 44451592 Ki = 7.943 nM T52921 CAC1G4 44451593 Ki = 17.38 nM T52921 CV26FM 44451594 Ki = 4.898 nM T52921 CKRM60 44451595 Ki = 1.514 nM T52921 C4S0BF 44451619 Ki = 2.399 nM T52921 CAVN40 44451620 Ki = 912.01 nM T52921 C2NCL3 44451621 Ki = 1.202 nM T52921 CHPO59 44451647 Ki = 95.5 nM T52921 C70TSK 44451648 Ki = 11.75 nM T52921 CZ1R2D 44451649 Ki = 0.8913 nM T52921 C5UM1O 44451650 Ki = 1.995 nM T52921 CF4SX9 44451673 Ki = 37.15 nM T52921 C3O8ZP 44451696 Ki = 29.51 nM T52921 C7VLH3 44451724 Ki = 41.69 nM T52921 CYIP73 44451748 Ki = 1.862 nM T52921 C2IS4W 44451777 Ki = 4.898 nM T52921 CST06H 44451779 Ki = 3.311 nM T52921 C4C9TD 44451805 Ki = 4.169 nM T52921 C5RLP6 44451837 Ki = 3.715 nM T52921 CO01GQ 44451872 Ki = 5.888 nM T52921 C7KL9C 44451895 Ki = 9.55 nM T52921 C25JHV 44451918 Ki = 1.413 nM T52921 C4DL5C 44469677 IC50 > 10000 nM T52921 CFAZ41 44517710 IC50 = 5.6 nM T52921 C6T1UX 44551464 EC50 = 3.6 nM T52921 CC01KM 44561020 Ki = 3.7 nM T52921 CY14MD 44561518 Ki = 6 nM T52921 CPO2R3 44570675 Ki = 2.5 nM T52921 CNUJ50 44574003 IC50 = 38 nM T52921 C1T4QN 44574053 IC50 = 16 nM T52921 CW8DR7 44574393 Ki = 1571 nM T52921 C67IZG 44574538 Ki = 3 nM T52921 C5Q4HZ 44574539 Ki = 7.3 nM T52921 C74LHO 44574585 Ki = 2.7 nM T52921 CPL5V1 44574586 Ki = 5.2 nM T52921 C7K4PC 44574587 Ki = 13 nM T52921 C1JPH8 44574588 Ki = 1.9 nM T52921 CNCS12 44574629 Ki = 3.6 nM T52921 CJXE09 44574630 Ki = 14 nM T52921 C2FO5H 44574631 Ki = 3 nM T52921 C5YQ6B 44574632 Ki = 7.4 nM T52921 CD18EP 44574671 Ki = 385 nM T52921 CDS1G8 44574672 Ki = 8 nM T52921 C6ZMS9 44574705 Ki = 6 nM T52921 CDNP82 44574706 Ki = 3151 nM T52921 C13RZI 44574707 Ki = 100 nM T52921 CXQM01 44574708 Ki = 3 nM T52921 CW1GU7 44574743 Ki = 6 nM T52921 CL6UI1 44574744 Ki = 4 nM T52921 CKO8N4 44574745 Ki = 2 nM T52921 CLVU91 44574789 Ki = 11 nM T52921 C5JZK9 44574790 Ki = 5.3 nM T52921 CVZ6K3 44574848 Ki = 31 nM T52921 C1MWD8 44574849 Ki = 40 nM T52921 CA78KV 44574850 Ki = 22 nM T52921 CX1BL6 44574851 Ki = 285 nM T52921 C7YAD5 44574889 Ki = 678 nM T52921 CPH7D4 44574890 Ki = 4.9 nM T52921 CQL2E4 44574891 Ki = 7 nM T52921 C9C3ZJ 44574892 Ki = 10 nM T52921 CLG57R 44574958 Ki = 12 nM T52921 CLMH36 44574962 Ki = 8.2 nM T52921 CAW3R4 44574963 Ki = 11 nM T52921 CAWB12 44575043 Ki = 17 nM T52921 CZO5J4 44575091 Ki = 908 nM T52921 CI6Y7U 44575092 Ki = 142 nM T52921 CO26ZW 44576625 IC50 = 8 nM T52921 CSH8K2 44576626 IC50 = 59 nM T52921 CD0T5K 44576627 IC50 = 18 nM T52921 C4ZCX6 44576628 IC50 = 1.1 nM T52921 CR0LN1 44593575 Ki = 198 nM T52921 CTYR04 44593576 Ki = 19 nM T52921 CDPU87 44596170 EC50 = 94 nM T52921 C45PUQ 45102745 Ki = 0.7 nM T52921 CU8I6T 45263517 Ki = 0.7 nM T52921 CVDQ53 45265789 Ki = 23 nM T52921 C6VZM4 45267505 IC50 = 2.5 nM T52921 CA2MH1 45267506 IC50 = 33 nM T52921 CK16EZ 45267601 IC50 = 28 nM T52921 CR59UW 45267616 IC50 = 200 nM T52921 CY4UA3 45267639 IC50 > 1000 nM T52921 CA2O3N 45268153 Ki = 3 nM T52921 C4F6IO 45268355 IC50 = 4.3 nM T52921 CX3YO5 45268356 IC50 = 17 nM T52921 C7UG6Q 45268498 IC50 = 2.3 nM T52921 C8QG3U 45268503 IC50 = 160 nM T52921 C3YEJ9 45268504 IC50 = 33 nM T52921 C8BPX4 45269032 Ki = 2 nM T52921 CKC09D 45269228 IC50 = 210 nM T52921 CKZ35F 45269347 IC50 > 1000 nM T52921 C06ITN 45269349 IC50 > 1000 nM T52921 C78UOX 45269357 IC50 = 4.7 nM T52921 C4WT5J 45269358 IC50 = 1.4 nM T52921 C3I6YO 45269372 IC50 = 160 nM T52921 CSL62Z 45270082 IC50 = 6.4 nM T52921 C6PRX0 45270174 IC50 = 620 nM T52921 C6GRC1 45270175 IC50 > 1000 nM T52921 CA38NB 45270184 IC50 = 3.7 nM T52921 CVU53F 45270190 IC50 > 1000 nM T52921 CA3S7Q 45270196 IC50 = 530 nM T52921 CY79OE 45270202 IC50 = 540 nM T52921 CVP80J 45270203 IC50 = 500 nM T52921 CC5I8O 45270712 Ki = 71 nM T52921 CM5ZI0 45270907 IC50 = 2 nM T52921 C6P0AZ 45270917 IC50 = 13 nM T52921 CDT5G6 45270928 IC50 = 15 nM T52921 C8KS5V 45271014 IC50 = 850 nM T52921 C2G5XK 45271015 IC50 = 26 nM T52921 CO05CL 45271041 IC50 = 11 nM T52921 CU84PI 45271534 Ki = 2 nM T52921 CP6V4Q 45271862 IC50 = 520 nM T52921 CMGB49 45271885 IC50 = 190 nM T52921 CJGX41 45271896 IC50 > 1000 nM T52921 C6G9DQ 45271902 IC50 = 160 nM T52921 C1UOZ9 45272626 IC50 = 7.8 nM T52921 C0P6GI 45272729 IC50 > 1000 nM T52921 CL0Y5P 45272733 IC50 > 1000 nM T52921 C09HIZ 45272755 IC50 > 1000 nM T52921 CFU9R4 45273531 IC50 = 0.61 nM T52921 CX0N4V 45273537 IC50 = 3.1 nM T52921 CJNO02 45273546 IC50 = 1.4 nM T52921 C3ZPJ5 45273547 IC50 = 12 nM T52921 CGT48R 45273662 IC50 = 130 nM T52921 C91JXR 45273672 IC50 > 1000 nM T52921 C58HQB 45273679 IC50 = 4.5 nM T52921 CS0GA2 45273702 IC50 = 96 nM T52921 C3YHF0 46227961 EC50 = 135 nM T52921 C7LW1S 46227963 Ki = 4.2 nM T52921 C9L6WI 46227966 EC50 = 15 nM T52921 CA2P9C 46879475 Ki = 4082 nM T52921 CH45JY 46879476 Ki = 454 nM T52921 CS2V6N 46879477 Ki = 16 nM T52921 C6R8JO 46879478 Ki = 106 nM T52921 C9URN3 46879536 Ki = 21 nM T52921 C5PW9I 46879537 Ki = 11 nM T52921 CW2N7P 46879538 Ki = 2.9 nM T52921 CGJS91 46879539 Ki = 6.4 nM T52921 C08CHW 46879578 Ki = 28 nM T52921 CNF9D6 46879579 Ki = 2.3 nM T52921 C8UD2Z 46879580 Ki = 0.6 nM T52921 C9E8YP 46879581 Ki = 2.5 nM T52921 C9GB7O 46879627 Ki = 2152 nM T52921 C5VKU0 46879628 Ki = 227 nM T52921 CU2F0K 46879629 Ki = 111 nM T52921 CS7BP4 46879630 Ki = 295 nM T52921 C06NBW 46879667 Ki = 44 nM T52921 C0WY3K 46879668 Ki = 22 nM T52921 C5L7DB 46879669 Ki = 7.7 nM T52921 CSG31K 46879670 Ki = 5 nM T52921 C7P4UE 46879716 Ki = 7.1 nM T52921 CQSI16 46879992 Ki = 470 nM T52921 C16INW 46879993 Ki = 227 nM T52921 C9NR8Q 46880030 Ki = 35 nM T52921 C0O1PU 46880031 Ki = 15 nM T52921 CDY2L8 46880032 Ki = 0.2 nM T52921 CK01VS 46880033 Ki = 1.3 nM T52921 CFXU43 46880088 Ki = 62 nM T52921 CDM4C0 46880089 Ki = 5.2 nM T52921 CA8JU6 46880090 Ki = 5.5 nM T52921 C7LX9B 46880114 Ki = 4.7 nM T52921 CX7RS8 46880115 Ki = 253 nM T52921 C2VS0K 46880116 Ki = 3.5 nM T52921 C18JDU 46880117 Ki = 487 nM T52921 CHN70E 46880151 Ki = 2560 nM T52921 CI5D6H 46880152 Ki = 259 nM T52921 CF0ER7 46880153 Ki = 1118 nM T52921 CU8JO5 46880154 Ki = 471 nM T52921 CR35XL 46880155 Ki = 186 nM T52921 CI6ZA1 46880237 Ki = 29 nM T52921 CID57V 46880238 Ki = 2.7 nM T52921 CG6UO7 46880239 Ki = 18 nM T52921 C31BLP 46880240 Ki = 1050 nM T52921 C3T6NH 49843555 Ki = 1.438 nM T52921 C0TCI3 52915030 IC50 = 31.6 nM T52921 CK6GN5 52915031 IC50 = 28.1 nM T52921 CXF14W 52915032 IC50 = 32.7 nM T52921 CELZ30 52915143 IC50 = 98.9 nM T52921 CR57AK 52915144 IC50 = 308.9 nM T52921 CP29EV 52915145 IC50 = 186.2 nM T52921 C15YXV 52915146 IC50 = 208.6 nM T52921 C45JNG 52915147 IC50 = 141.9 nM T52921 COM38Z 52915266 IC50 = 146.5 nM T52921 COEU73 52915267 IC50 = 154.5 nM T52921 CZK59C 52915268 IC50 = 184.5 nM T52921 C27KOF 52915269 IC50 = 83 nM T52921 CQ71YX 52915270 IC50 = 1115.9 nM T52921 CH56XF 52915389 IC50 = 731.6 nM T52921 C02UBO 52915390 IC50 = 1217.8 nM T52921 CP2M6E 52915391 IC50 = 667.5 nM T52921 CPA43I 52915392 IC50 = 482.9 nM T52921 C5OA9H 52915393 IC50 = 304.6 nM T52921 CA3P2C 52915514 IC50 = 404.7 nM T52921 CK39TQ 52915515 IC50 = 159.6 nM T52921 C98UZW 52915516 IC50 = 799.8 nM T52921 CLAS61 52915517 IC50 = 206.9 nM T52921 C7FDE9 52915518 IC50 = 1106.7 nM T52921 C9YOD2 52915634 IC50 = 246.4 nM T52921 C1ZHF3 52915635 IC50 = 144 nM T52921 CZB67C 52915636 IC50 = 211.6 nM T52921 CE3IS2 52915637 IC50 = 152.9 nM T52921 C8F0TA 52916174 IC50 = 207.3 nM T52921 C4K3NO 52916266 IC50 = 115.7 nM T52921 CPV9S3 52916267 IC50 = 48 nM T52921 CXGN56 52916358 IC50 = 35.6 nM T52921 CO4Q6E 52916359 IC50 = 50.9 nM T52921 CM0KA5 52916360 IC50 = 83.3 nM T52921 CN8L4T 52916470 IC50 = 63.1 nM T52921 C96OUY 52916471 IC50 = 113.6 nM T52921 CC92WA 52916472 IC50 = 82.7 nM T52921 CG91EA 52916597 IC50 = 82.1 nM T52921 CYB6J8 52916598 IC50 = 76.5 nM T52921 CG1F9W 52916599 IC50 = 56.6 nM T52921 C7NO2D 52916712 IC50 = 76.2 nM T52921 CZ3K9S 52916713 IC50 = 71.7 nM T52921 CI32WO 52916714 IC50 = 30.1 nM T52921 C4FZT7 52951674 Ki = 0.231 nM T52921 CS4T2C 52951675 Ki = 0.101 nM T52921 C5VLO1 52951807 Ki = 0.106 nM T52921 CK7I1T 52951808 Ki = 0.137 nM T52921 C0UVH3 52951809 Ki = 0.09 nM T52921 C40BPO 52951810 Ki = 0.15 nM T52921 CF0L7D 52951938 Ki = 4.51 nM T52921 CDAN40 52951939 Ki = 17.1 nM T52921 C89QXK 52951940 Ki = 5.61 nM T52921 COVP24 52951941 Ki = 10.2 nM T52921 CR6B4G 52951942 Ki = 9.08 nM T52921 CSF4G7 52952043 Ki = 5.32 nM T52921 CTU43X 53316968 Ki = 4.54 nM T52921 CCOD69 53316969 Ki = 4.29 nM T52921 CI6CQ0 53319615 Ki = 0.15 nM T52921 C6SY4G 53319616 Ki = 80.5 nM T52921 C3PW1V 53319617 Ki = 4.29 nM T52921 C2EV1S 53322245 Ki = 0.96 nM T52921 C1L8IV 53322246 Ki > 250 nM T52921 C0MD2H 53324890 Ki = 0.73 nM T52921 C5E7LW 53325608 Ki = 4.29 nM T52921 CRZ76L 53326167 Ki = 6.56 nM T52921 CJ46YH 54580478 Ki = 58.88 nM T52921 C35VCH 54580479 Ki = 48.98 nM T52921 CED95R 54581495 Ki = 107.15 nM T52921 CW7FV5 54581497 Ki = 83.18 nM T52921 CWOA13 54583469 Ki > 10000 nM T52921 CE9OC2 54584439 Ki = 60.26 nM T52921 CA4XQ2 54584440 Ki = 1148.15 nM T52921 C8J5OH 54585395 Ki = 58.88 nM T52921 CM3A1U 54585396 Ki = 158.49 nM T52921 CYS7J8 54586351 Ki > 10000 nM T52921 CROS84 54756989 Ki = 18.5 nM T52921 C2ISE6 54756990 Ki = 22 nM T52921 CCN2E8 56658044 Ki = 16 nM T52921 C69VIF 56661555 Ki = 67.8 nM T52921 CDKP63 56664973 Ki = 8.46 nM T52921 C4QM3N 56668405 Ki = 237 nM T52921 CX8F2N 56681954 Ki = 133 nM T52921 C2A4MQ 56681955 Ki = 159 nM T52921 CQY16A 57391870 Ki > 10000 nM T52921 CI5H3N 58268566 Ki = 0.0916 nM T52921 C6Z9JF 58268629 Ki = 0.0892 nM T52921 C6G5TY 60154189 Ki = 7.37 nM T52921 C2ZG0F 60154190 Ki = 9.4 nM T52921 C8MS6N 60154191 Ki = 1.84 nM T52921 CW63KM 60154192 Ki = 5.16 nM T52921 C2QX6R 60154193 Ki > 10 nM T52921 CTCJ21 60154194 Ki > 10 nM T52921 CO4Q8V 60154195 Ki > 10 nM T52921 C80XNK 60154196 Ki > 10 nM T52921 CJ8DW1 60154197 Ki > 40 nM T52921 CD5R7A 60154198 Ki > 40 nM T52921 CY1U7F 60154199 Ki > 40 nM T52921 CXRV52 60154200 Ki = 0.396 nM T52921 CD46EJ 60154264 Ki = 0.114 nM T52921 C98XRD 66911347 Ki = 205 nM T52921 CZ63PG 66986460 Ki = 3.7 nM T52921 CF5I0R 68917692 Ki = 1.26 nM T52921 CPE62M 70682348 Ki > 250 nM T52921 C6KD9C 70682349 Ki > 250 nM T52921 C2PC8W 70682350 Ki > 250 nM T52921 C58AOU 70682351 Ki = 9.84 nM T52921 CH42QP 70682760 Ki = 0.194 nM T52921 C6G0SO 70684433 Ki = 11.6 nM T52921 CZ5B7A 70684434 Ki > 250 nM T52921 CLY56A 70684435 Ki > 250 nM T52921 C8U1PW 70684436 Ki = 13.6 nM T52921 C4ZU7H 70684841 Ki = 0.0902 nM T52921 C6DC8G 70684842 Ki = 0.0672 nM T52921 CWAL85 70686573 Ki > 250 nM T52921 CAFB10 70686574 Ki > 250 nM T52921 CZ6E9M 70686575 Ki > 250 nM T52921 CPD35T 70686907 Ki = 5.32 nM T52921 CI61FE 70688692 Ki > 250 nM T52921 C08OUK 70688693 Ki > 250 nM T52921 CMKZ80 70688694 Ki > 250 nM T52921 CLK7P0 70688695 Ki > 250 nM T52921 C8M4PI 70688696 Ki > 250 nM T52921 C3HAX5 70688697 Ki = 3.79 nM T52921 C7PNH3 70689062 Ki = 0.0373 nM T52921 CA3T1P 70689063 Ki = 0.127 nM T52921 CF7PZ4 70690755 Ki = 5.55 nM T52921 CMNL89 70690756 Ki = 128 nM T52921 CWB17N 70690757 Ki = 26.2 nM T52921 CX5VR6 70690758 Ki = 26.5 nM T52921 C8UYZ6 70690759 Ki > 250 nM T52921 CTB4I1 70690760 Ki = 0.96 nM T52921 CQJ6K3 70691171 Ki = 2.05 nM T52921 CEV6U7 70691173 Ki = 0.248 nM T52921 CY6E2Q 70691339 IC50 > 10000 nM T52921 C3E4FO 70692893 Ki = 101 nM T52921 CV61FR 70692894 Ki = 31.5 nM T52921 C05RKU 70692895 Ki = 286 nM T52921 CLM98A 70692896 Ki > 250 nM T52921 CU60IL 70694933 Ki > 250 nM T52921 CWO5F0 70695375 Ki = 0.169 nM T52921 CJ07AO 70696988 Ki > 250 nM T52921 C4Z0QA 70696990 Ki > 250 nM T52921 CV0P1X 70696991 Ki = 3.03 nM T52921 CFQ8Y9 70696992 Ki > 250 nM T52921 CTO0Y4 70697389 Ki = 0.458 nM T52921 CNE50L 70697390 Ki = 0.124 nM T52921 CG3U7F 70697391 Ki = 0.134 nM T52921 CEOQ43 71229805 Ki = 43.2 nM T52921 CJDR19 71230446 Ki = 44 nM T52921 CM0H5E 71454460 Ki = 22 nM T52921 CBEV63 71461579 Ki = 27.9 nM T52921 C0B7LC 71624265 Ki = 7.63 nM T52921 C7Q9VU 71624266 Ki = 15.26 nM T52921 CD9IO8 71624267 Ki = 212.8 nM T52921 CXZ6E1 71624268 Ki = 9.98 nM T52921 C0O6IR 71624269 Ki = 26.9 nM T52921 CW2G0T 71624270 Ki = 6.53 nM T52921 CBM1C8 71624387 Ki = 12.65 nM T52921 CML7K2 71624388 EC50 = 6.8 nM T52921 C1B9VM 71624389 Ki = 40.28 nM T52921 CWH6T3 72548703 IC50 = 0.98 nM T52921 CC6Q5R 72771081 Ki < 100 nM T52921 C7ZN1K 73345634 Ki = 0.05495 nM T52921 CN5S4A 73350483 Ki = 11.43 nM T52921 COS31U 73354624 Ki = 1700 nM T52921 CJQ25A 76309739 Ki = 4 nM T52921 CC01JG 76309740 Ki = 3 nM T52921 C69JCU 76313421 Ki = 31 nM T52921 CJR57Q 76313422 Ki = 401 nM T52921 CA4IN3 76313423 Ki = 16 nM T52921 CP3HV7 76313424 Ki = 10 nM T52921 CU56FN 76313425 Ki = 10 nM T52921 CPJ4N3 76313426 Ki = 36 nM T52921 C7LV2A 76313427 Ki = 13 nM T52921 CTN6G1 76316935 Ki = 15 nM T52921 C1AW8J 76316936 Ki = 22 nM T52921 CC2AG6 76316937 Ki = 17 nM T52921 CNAE72 76320663 Ki > 1000 nM T52921 CD0PC8 76320664 Ki > 1000 nM T52921 CF83DA 76320665 Ki = 6 nM T52921 C5W1XJ 76320666 Ki = 3 nM T52921 C0MI1G 76324308 Ki = 3 nM T52921 CI2A6W 76324309 Ki = 29 nM T52921 CT9XB8 76324310 Ki = 6 nM T52921 C4QM6R 76324311 Ki = 79 nM T52921 C6AY5S 76327872 Ki = 15 nM T52921 CCR5B1 76327873 Ki = 47 nM T52921 CL58DY 76327874 Ki = 9 nM T52921 CBVL29 76327875 Ki = 19 nM T52921 C64JDN 76327876 Ki = 7 nM T52921 C3G1LA 76327877 Ki = 42 nM T52921 CCN1M9 76331524 Ki = 75 nM T52921 CQ35XY 76331525 EC50 = 14 nM T52921 CDA37E 76335140 Ki = 72 nM T52921 CUZ30G 76335141 Ki = 122 nM T52921 CKZ7T2 76335142 Ki = 10 nM T52921 CQKT47 76335143 Ki = 10 nM T52921 C6K5RY 76335144 Ki = 10 nM T52921 CECO35 76335145 Ki = 12 nM T52921 CLH3X9 81689704 Ki = 80 nM T52921 CGH7J9 86279209 Ki = 3.16 nM T52921 C8HE3B 90306863 Ki = 4630 nM T52921 C1W9QL 90306885 Ki = 75 nM T52921 C1DOG7 90654745 Ki = 0.172 nM T52921 CX3WT1 90654746 Ki = 0.176 nM T52921 CC70MH 90654747 Ki = 0.145 nM T52921 C4ZQD5 90654748 Ki = 0.371 nM T52921 CBV23K 90654749 Ki = 0.114 nM T52921 C87NYV 90654750 Ki = 0.097 nM T52921 C20FOK 90654751 Ki = 0.105 nM T52921 CT91LC 90654752 Ki = 0.185 nM T52921 CT5U7G 90654753 Ki = 0.139 nM T52921 C42GMO 90654754 Ki = 0.0711 nM T52921 CBR5H7 90654755 Ki = 0.0954 nM T52921 C68VLU 90654756 Ki = 0.0648 nM T52921 C8GUX3 90654757 Ki = 0.122 nM T52921 C4Z6KQ 90654758 Ki = 0.0908 nM T52921 C13ACK 90654759 Ki = 0.0939 nM T52921 C7C5BM 90655970 Ki > 10000 nM T52921 CTV50C 90655971 Ki = 2.1 nM T52921 C1S5UB 90655972 Ki = 3.41 nM T52921 CV6A5T 90655973 Ki = 2.99 nM T52921 CL0D4Y 90655974 Ki = 8.63 nM T52921 C51CQN 90655975 Ki = 11.1 nM T52921 C2USA9 90655976 Ki = 76.6 nM T52921 CLKW80 90655977 Ki > 10000 nM T52921 C96DUE 90655978 EC50 = 72.2 nM T52921 C1N5QA 90655979 Ki > 10000 nM T52921 CK9FP8 90656664 Ki = 197 nM T52921 COGW86 90656666 Ki = 105 nM T52921 C9YKV8 90656667 Ki = 187 nM T52921 C3WLH8 90656668 Ki = 396 nM T52921 CP1ZW6 90663949 Ki > 5000 nM T52921 CZ9GL5 90663950 Ki = 45 nM T52921 CFK27M 90663951 Ki > 5000 nM T52921 CBT6F1 90663952 Ki > 5000 nM T52921 C1QAB3 90663953 Ki = 34 nM T52921 C07VRA 101341769 Ki = 39 nM T52921 C4VMI7 101354795 IC50 = 1.67 nM T52921 CBM3Q5 118662014 Ki = 68 nM T52921 CK8Y3E 118662042 Ki = 170 nM T52921 CS81PR 118662074 Ki = 0.8 nM T52921 C8AF6I 118662117 Ki = 29.5 nM T52921 CBJ16O 118662129 Ki = 1510 nM T52921 C4ZP0L 118662159 Ki = 1.6 nM T52921 CR6IU7 118662169 Ki = 2160 nM T52921 C7VE1O 118662183 Ki = 600 nM T52921 C1VR3B 118662189 Ki = 0.7 nM T52921 CG0R6H 118662291 Ki = 2.9 nM T52921 CI17PS 118662309 Ki = 5.8 nM T52921 CCIP14 118662342 Ki = 1.1 nM T52921 CB79UC 118662456 Ki = 2.3 nM T52921 C5LZ8I 118662460 Ki = 0.4 nM T52921 CM8TB4 118705898 Ki = 1300 nM T52921 C80UNO 118705899 Ki = 1500 nM T52921 C6RW0E 118705901 Ki = 880 nM T52921 C20RQZ 118711156 Ki = 1600 nM T52921 CV85YO 118711243 Ki = 5.4 nM T52921 CKUT03 118711485 Ki = 0.5 nM T52921 CI6BM7 118711486 Ki = 2 nM T52921 CMY0F1 118711490 Ki = 0.55 nM T52921 CMRV59 118711491 Ki = 1.1 nM T52921 CTVK82 118717442 IC50 = 1.39 nM T52921 CSIW96 118718262 Ki = 39 nM T52921 C4LM3W 118718263 Ki = 55 nM T52921 C2Q8YU 118718264 Ki = 116 nM T52921 C9BFP5 118718265 Ki = 5 nM T52921 CS14YZ 118718266 Ki = 7 nM T52921 CRBA23 118718267 Ki = 82 nM T52921 C4AS8L 118718268 Ki = 35 nM T52921 CP8I2K 118718269 Ki = 17 nM T52921 C6TGR8 118718270 Ki = 336 nM T52921 C3W1BL 118718271 Ki = 29 nM T52921 CPC23W 118718272 Ki = 24 nM T52921 C2Y4PK 118718273 Ki = 104 nM T52921 C8FC1Q 118718274 Ki = 4 nM T52921 C2BGR0 118718275 Ki = 27 nM T52921 CJZ1F7 118718276 Ki = 34 nM T52921 CCFR52 118718277 Ki = 15 nM T52921 C5O2VC 118718278 Ki = 58 nM T52921 CC0KE5 118718279 Ki = 7 nM T52921 CK1Q9B 118718280 Ki = 20 nM T52921 CB92OV 118718281 Ki = 50 nM T52921 CSK4N3 118718282 Ki = 173 nM T52921 CDBP05 118718283 Ki = 245 nM T52921 CDH69C 118718284 Ki = 670 nM T52921 CLRD02 118718285 Ki = 62 nM T52921 CYI4T2 118718286 Ki = 27 nM T52921 C2F8ZN 118718287 Ki = 99 nM T52921 CA9N0S 118718288 Ki = 11 nM T52921 CVT94Z 118718289 Ki = 6 nM T52921 C1RAX5 118718290 Ki = 10 nM T52921 CKNL94 118718291 Ki = 17 nM T52921 CKN54J 118718292 Ki = 20 nM T52921 CC6U5D 118718293 Ki = 210 nM T52921 C64JUV 118718294 Ki = 70 nM T52921 CICJ78 118718295 Ki = 68 nM T52921 CZMR06 118718296 Ki = 31 nM T52921 C92CER 118718297 Ki = 118 nM T52921 CP23YE 118718298 Ki = 50 nM T52921 COA69M 118718299 Ki = 39 nM T52921 CSW82H 118718300 Ki = 74 nM T52921 C2EGJ8 118718301 Ki = 11 nM T52921 CO5BV4 118718302 Ki = 12 nM T52921 CTF9L6 118722880 Ki = 7.4 nM T52921 CDI8J1 118722882 Ki = 0.5 nM T52921 C3T8YZ 118726261 IC50 = 61 nM T52921 C6I5HS 118726262 IC50 = 4.2 nM T52921 C10BIV 118726263 IC50 = 99.7 nM T52921 CA43CF 118726264 IC50 = 166 nM T52921 CLSG96 118726265 IC50 = 160 nM T52921 CYL40S 118726266 IC50 = 8 nM T52921 CPR0K2 118726267 IC50 = 14 nM T52921 CH9A3M 118726268 IC50 = 26 nM T52921 CEH89Y 118726269 IC50 = 3.9 nM T52921 CT7H2M 118726270 IC50 = 40.9 nM T52921 C1UD6R 118726271 IC50 = 8.8 nM T52921 CRK62Y 118726272 IC50 = 37 nM T52921 CF25IA 118726273 IC50 = 18 nM T52921 CQH1G3 118731120 Ki > 10000 nM T52921 CK0LH7 122179050 Ki = 97 nM T52921 CEY90C 122179051 Ki = 1270 nM T52921 CBP42W 122179052 EC50 = 14 nM T52921 CNCJ68 122179053 EC50 = 7.3 nM T52921 CY96XI 122179055 Ki = 820 nM T52921 C6LDU5 122179056 Ki = 240 nM T52921 C57GMN 122179057 Ki = 56 nM T52921 C0X6AF 122179058 Ki = 56 nM T52921 CS0B3O 122179059 Ki = 26 nM T52921 C09BYL 122179060 Ki = 47.8 nM T52921 CF83LN 122179061 Ki = 62.2 nM T52921 CC73XP 122179063 Ki = 571 nM T52921 C6YQM4 122179064 EC50 = 230 nM T52921 C9WF5T 122179567 EC50 = 323.59 nM T52921 CTA9E8 122179568 EC50 = 158.49 nM T52921 C35HVO 122179584 EC50 = 426.58 nM T52921 CF2W0K 122179586 EC50 = 208.93 nM T52921 CE3LH1 122179587 EC50 = 45.71 nM T52921 CAQ5B0 122409965 Ki = 0.53 nM T52921 C51MTO 124565311 Ki = 0.21 nM T52921 C1YEA7 127030671 Ki > 250 nM T52921 C1HO7F 127033703 Ki = 3.13 nM T52921 CB12AP 127033704 Ki > 250 nM T52921 C4NIU0 127034022 Ki = 5.65 nM T52921 C7ORD8 127034023 Ki = 5.55 nM T52921 CEWM81 127034292 Ki = 3.56 nM T52921 CBOC84 127034554 Ki = 18.1 nM T52921 CXMJ48 127043001 Ki = 27 nM T52921 CFU4H9 127043364 Ki = 47 nM T52921 C30BNK 127043559 Ki = 38 nM T52921 CCSZ68 127044528 Ki = 42 nM T52921 C1EHU5 129188443 Ki = 9.8 nM T52921 CD8FT9 129188454 Ki = 2.17 nM T52921 CC9Z0J 129188459 Ki = 10.3 nM T52921 CG57MT 134563466 Ki = 10.5 nM T52921 CE5RS7 134563496 Ki = 23.6 nM T52921 CAEY19 134563500 Ki = 216 nM T52921 C82SEF 134563650 Ki = 44.7 nM T52921 CC3HK6 134563655 Ki = 0.3 nM T52921 C4U9EM 134563691 Ki = 43.8 nM T52921 CFX37T 134563695 Ki = 129 nM T52921 CPEH72 134563698 Ki = 24.4 nM T52921 CR74XA 134563699 Ki = 31.8 nM T52921 C9PN6I 134578342 Ki = 15.9 nM T52921 CK62WY 134578456 Ki = 9.46 nM T52921 CN0C9Z 134578457 Ki = 1.47 nM T52921 C0HNI9 134578506 Ki = 64 nM T52921 C0JCQ2 134578518 Ki = 136 nM T52921 C1CH3X 135458466 IC50 = 199 nM T52921 CN14XB 136036819 Ki = 5.888 nM T52921 CL14DP 136043756 IC50 = 440 nM T52921 CC1N8P 136043758 IC50 > 1000 nM T52921 CUXY20 136043759 IC50 = 294 nM T52921 C7US0J 136043761 IC50 > 1000 nM T52921 CFLE34 136043762 IC50 > 1000 nM T52921 C0HPR7 136043764 IC50 > 1000 nM T52921 C9WN3S 136043765 IC50 = 580 nM T52921 CB5O8L 136043767 IC50 = 440 nM T52921 CW9HY3 136043768 IC50 > 1000 nM T52921 C8CTV4 136043771 IC50 = 140 nM T52921 CB36GF 136043772 IC50 > 1000 nM T52921 CIZ41F 136043774 IC50 > 1000 nM T52921 CKW90B 136043777 IC50 > 1000 nM T52921 CJL1Y8 136043778 IC50 > 1000 nM T52921 C5KZF8 136043779 IC50 = 58 nM T52921 C2LC8O 136043780 IC50 = 450 nM T52921 C9B0WD 136043781 IC50 = 568 nM T52921 CJM57B 136043782 IC50 = 233 nM T52921 C0A6NT 136043783 IC50 > 1000 nM T52921 C0QTA5 136043784 IC50 > 1000 nM T52921 CRGU10 136043785 IC50 > 1000 nM T52921 COL64J 136043786 IC50 = 120 nM T52921 CV5AJ0 136043787 IC50 > 1000 nM T52921 CH0VN9 136043788 IC50 = 62 nM T52921 C1GJE7 136043789 IC50 > 1000 nM T52921 CC8ZK4 136043790 IC50 = 210 nM T52921 C0QDL8 136043791 IC50 > 1000 nM T52921 CM2I3S 136043792 IC50 = 600 nM T52921 CZ6A5D 136043795 IC50 = 450 nM T52921 C24BXO 136043796 IC50 = 230 nM T52921 CQLF58 136043797 IC50 = 560 nM T52921 C9EF5P 136043798 IC50 > 1000 nM T52921 CEZ83O 136043799 IC50 > 1000 nM T52921 CFZX29 136043800 IC50 = 49 nM T52921 CVFX50 136043807 IC50 > 1000 nM T52921 C5TIE8 136043816 IC50 > 1000 nM T52921 C68CEZ 136043817 IC50 = 450 nM T52921 CCJ02K 136043818 IC50 > 1000 nM T52921 C06YGH 136043819 IC50 = 632 nM T52921 C1XV2U 136043820 IC50 > 1000 nM T52921 C53OLF 136043821 IC50 > 1000 nM T52921 C4NXF8 136043824 IC50 = 410 nM T52921 CX3H8P 146034954 EC50 = 72.44 nM T52921 C85LIH 146034955 EC50 = 7.244 nM T52921 CY5CL2 155521553 Ki = 20.9 nM T52921 CZ1V3B 155523994 IC50 = 0.63 nM T52921 CXH95L 155531153 Ki = 2.27 nM T52921 CTWG84 155533462 Ki = 2 nM T52921 C4RWI6 155536757 Ki = 27 nM T52921 CHJ59D 155537352 Ki = 15.5 nM T52921 C67WLH 155542684 Ki = 23.1 nM T52921 CU83VX 155544763 Ki = 11 nM T52921 CQ0GL3 155569552 Ki = 11 nM T52921 D00BIE 25084507 Ki = 0.34 nM T52921 D00HAJ 73347136 IC50 > 50000 nM T52921 D00LVW 44456141 IC50 = 3.42 nM T52921 D00XZH 44430025 Ki = 433 nM T52921 D00YCW 44426807 Ki = 19 nM T52921 D01CFO 44456028 IC50 = 7.42 nM T52921 D01MUV 10314141 Ki = 62 nM T52921 D01WMU 9820782 Ki = 4 nM T52921 D02NSY 10296561 Ki = 0.2399 nM T52921 D02TPK 44416445 IC50 = 0.0803 nM T52921 D02WBU 44456216 EC50 = 17.7 nM T52921 D03BVN 44456298 EC50 = 23.8 nM T52921 D03PTV 10022129 Ki = 59 nM T52921 D03UJW 22970051 Ki = 23 nM T52921 D04PUK 44426803 Ki = 613 nM T52921 D04WRO 44456337 IC50 = 218 nM T52921 D04ZQX 44426812 Ki = 18 nM T52921 D05NIE 44430036 Ki = 455 nM T52921 D05RII 44413409 Ki = 1140 nM T52921 D05YMD 44455999 IC50 = 21.3 nM T52921 D06MQG 44430018 Ki = 180 nM T52921 D06PHT 10269001 Ki = 13 nM T52921 D06PVO 44426806 Ki = 135 nM T52921 D06RSR 44456187 IC50 = 14.7 nM T52921 D07CIU 9924923 Ki = 55 nM T52921 D07FCB 9925737 Ki = 323 nM T52921 D07NMH 10093682 Ki = 51 nM T52921 D08BAW 44456185 IC50 = 1.86 nM T52921 D08DVV 44430026 Ki = 1147 nM T52921 D08IXN 5497186 Ki = 0.03 nM T52921 D08NDP 25080768 Ki = 0.1 nM T52921 D08QBS 44178080 IC50 = 4.6 nM T52921 D08QBU 44430029 Ki = 1667 nM T52921 D08TFY 10043439 Ki = 17 nM T52921 D08ZDP 44430014 Ki = 9155 nM T52921 D09BYD 20481138 Ki = 11 nM T52921 D09CTG 44416444 IC50 = 0.789 nM T52921 D09FJY 9863568 Ki = 2 nM T52921 D09KBQ 131534 Ki = 2151 nM T52921 D09LRO 44430008 Ki = 23 nM T52921 D09VRT 44426814 Ki = 16 nM T52921 D09XZM 10986104 IC50 = 3.03 nM T52921 D0A1XG 44416268 IC50 > 10000 nM T52921 D0A8NZ 44578000 Ki = 0.27 nM T52921 D0A8ZS 44456217 IC50 = 92.6 nM T52921 D0AC0A 10047612 Ki = 0.253 nM T52921 D0D0UP 10315818 Ki = 48 nM T52921 D0D9BB 10427620 Ki = 313 nM T52921 D0E3RQ 44416159 IC50 = 0.0464 nM T52921 D0F8AX 44430024 Ki = 376 nM T52921 D0F8CV 5462471 Ki > 10000 nM T52921 D0FF6S 16038374 IC50 > 10000 nM T52921 D0G4FA 10384734 Ki = 588 nM T52921 D0G7DF 44426827 Ki = 3 nM T52921 D0HN2M 44430609 Ki = 0.02818 nM T52921 D0IL9H 44430013 Ki = 1745 nM T52921 D0J5JO 44430009 Ki = 27 nM T52921 D0JH5D 44430007 Ki = 34 nM T52921 D0K2NY 44456101 IC50 = 5.67 nM T52921 D0L6QN 10070040 Ki = 24 nM T52921 D0L8YY 10066285 Ki = 5.7 nM T52921 D0M7TP 44456412 IC50 = 14.9 nM T52921 D0NE3U 5485199 IC50 > 10000 nM T52921 D0O7JV 44426810 Ki = 14 nM T52921 D0P3FP 44426808 Ki = 5 nM T52921 D0PN2C 44456140 IC50 = 2.81 nM T52921 D0PR2Q 44456220 EC50 = 27.6 nM T52921 D0Q2PO 25084509 Ki = 0.54 nM T52921 D0Q9TQ 10043898 Ki = 54 nM T52921 D0QH4A 10089987 Ki = 14 nM T52921 D0S2OA 10388166 Ki = 162 nM T52921 D0SE9S 9887077 Ki = 0.3 nM T52921 D0SN6V 44456299 EC50 = 46.5 nM T52921 D0T0GL 44456296 IC50 = 0.66 nM T52921 D0T4ZY 44426817 Ki = 134 nM T52921 D0T9KE 44430016 Ki = 85 nM T52921 D0TJ7R 97333 Ki = 1983 nM T52921 D0U6FM 44456339 IC50 = 21.7 nM T52921 D0V3OY 105104 Ki > 10000 nM T52921 D0VH3M 25088989 Ki = 0.83 nM T52921 D0W3VT 10091033 Ki = 24 nM T52921 D0W7CF 9963005 IC50 = 1.04 nM T52921 D0X4SX 10317947 Ki = 72 nM T52921 D0XX1Y 44426828 Ki = 53 nM T52921 D0Y0IE 44352919 EC50 = 1.97 nM T52921 D0Y2MT 44416158 IC50 = 11.6 nM T52921 D0Y4EW 6324645 EC50 = 0.3236 nM T52921 D0Y5LJ 10336926 Ki = 136 nM T52921 D0Y7KE 44430012 Ki = 1281 nM T52921 D0YM8F 25084510 Ki = 1.79 nM T52921 D0ZE2W 44430028 Ki = 2176 nM T98092 D02EEJ 6479267 Ki = 1.84 nM T98092 D0CE0O 11513676 Ki = 0.34 nM T98092 D0G7UX 5284373 Ki = 2.64 nM T98092 D0M2OY 53259809 Ki = 16800 nM T98092 D08MYL 6473876 Ki = 2.11 nM T98092 CY0Q4V 444384 IC50 = 2000000 nM T98092 CLYE08 497073 IC50 = 6000 nM T98092 C8SG7U 497075 IC50 > 10000000 nM T98092 CAWY91 497076 IC50 = 90000 nM T98092 CC9D3J 497077 IC50 > 10000000 nM T98092 CBMF04 497078 IC50 = 500000 nM T98092 C6KF5Y 1367020 IC50 = 580 nM T98092 CP61UY 2823177 IC50 = 920 nM T98092 CM6OW0 3190778 IC50 = 5.5 nM T98092 CDPT84 4128827 IC50 = 316 nM T98092 C7T6VH 4401642 IC50 = 14 nM T98092 CSQP36 5020377 IC50 = 303 nM T98092 CZ34OX 5116189 IC50 = 5500 nM T98092 C7DIT9 5493631 IC50 = 680000 nM T98092 C35VSF 5493632 IC50 = 1000000 nM T98092 CGN50H 5493634 IC50 = 260000 nM T98092 C8U3AT 5493635 IC50 = 115000 nM T98092 C5I2UC 5493638 IC50 = 280000 nM T98092 CNIC61 6475296 IC50 = 310 nM T98092 C8RA6C 6476061 IC50 = 11.1 nM T98092 CTXB32 6479257 IC50 = 3 nM T98092 CMH26D 6479258 IC50 = 47 nM T98092 C45EVU 6479259 IC50 = 15 nM T98092 CQ1X3C 6479260 IC50 = 61 nM T98092 C1YMW4 6479261 IC50 = 277 nM T98092 CAYZ53 6479262 IC50 = 97 nM T98092 CPCG74 6479263 IC50 = 128 nM T98092 C16CZK 6479264 IC50 = 19 nM T98092 CN1BF8 6479265 IC50 = 165 nM T98092 C8N4YK 6479266 IC50 = 110 nM T98092 CAGX82 6479268 IC50 = 6047 nM T98092 CM36KU 6479269 IC50 = 1572 nM T98092 CJWU53 6479270 IC50 = 882 nM T98092 CRV94O 6479271 IC50 = 959 nM T98092 C03LTJ 10034324 IC50 = 934 nM T98092 CODJ10 10626583 Ki = 795 nM T98092 CO9XA6 10819131 IC50 = 1500000 nM T98092 CF45ID 11516665 IC50 = 20 nM T98092 CGP87C 11531251 IC50 = 951 nM T98092 CSY31B 11559871 IC50 = 748 nM T98092 C6M1ZU 11567780 IC50 = 320 nM T98092 CJ27OG 11588606 IC50 = 140 nM T98092 CN8M2B 11617502 IC50 = 71 nM T98092 CS2Y6M 11631957 IC50 = 60 nM T98092 CX63ZC 11632684 IC50 = 60 nM T98092 CLP34W 11638938 IC50 = 592 nM T98092 CS3YJ8 11660364 IC50 = 640 nM T98092 C37WLM 11675245 IC50 = 528 nM T98092 C3SK8D 11703833 IC50 = 880 nM T98092 C2QN6F 11710570 IC50 = 1437 nM T98092 C73OMC 11717355 IC50 = 458 nM T98092 C89EKB 11718015 IC50 = 499 nM T98092 CUY92Q 13422114 IC50 = 130 nM T98092 CC6XY7 13578707 IC50 = 350 nM T98092 C8KA7W 20415061 IC50 = 460 nM T98092 C31GDL 24814873 IC50 = 14 nM T98092 C2ON4L 25044910 IC50 = 690 nM T98092 CY8HB6 25046022 IC50 = 330 nM T98092 CT2E3I 25098032 IC50 = 590 nM T98092 CK0P2Q 42630203 IC50 = 650 nM T98092 C69CNK 44248910 IC50 > 10000 nM T98092 C46XEC 44248911 IC50 = 103 nM T98092 CS6N9K 44248912 IC50 = 71.2 nM T98092 CHX9S4 44248913 IC50 = 159 nM T98092 CSDG42 44248914 IC50 > 10000 nM T98092 CJT1A8 44249039 IC50 = 364 nM T98092 CVW1T9 44249040 IC50 = 263 nM T98092 CNFI87 44249041 IC50 = 2.59 nM T98092 CW6LT7 44249042 IC50 = 1.52 nM T98092 C7U6PN 44249044 IC50 = 1910 nM T98092 C1HPV8 44249170 IC50 > 10000 nM T98092 CW4AU3 44249173 IC50 = 12.1 nM T98092 CKO3I0 44249174 IC50 > 10000 nM T98092 CL7M2J 44249303 IC50 = 620 nM T98092 C97JUQ 44249304 IC50 > 10000 nM T98092 C0SVJ1 44249305 IC50 = 31.6 nM T98092 CA3K2N 44249306 IC50 > 10000 nM T98092 CBEL85 44249307 IC50 = 370 nM T98092 C5M4VW 44249309 IC50 = 136 nM T98092 CR2K7N 44249310 IC50 > 10000 nM T98092 C57MCG 44249414 IC50 > 10000 nM T98092 CSJD94 44249415 IC50 > 10000 nM T98092 CER54N 44294512 IC50 = 2500000 nM T98092 CKYA61 44294584 IC50 = 850000 nM T98092 C4R1DL 44294708 IC50 > 10000000 nM T98092 CTE19D 44294709 IC50 > 10000000 nM T98092 CT5IJ4 44294814 IC50 = 2800000 nM T98092 C4GLS0 44294838 IC50 = 760000 nM T98092 C5EQ7U 44295020 IC50 = 1300000 nM T98092 CHI01J 44295050 IC50 = 1500000 nM T98092 CS5I9W 44295136 IC50 = 970000 nM T98092 COCG50 44295258 IC50 = 820000 nM T98092 CV7PD8 44341483 IC50 = 48 nM T98092 C5M1FB 44341507 IC50 = 256 nM T98092 CM9L8P 44365970 IC50 = 1500000 nM T98092 C50FPJ 44366040 IC50 = 2500000 nM T98092 C0JKL6 44366208 IC50 = 2600000 nM T98092 C98VGM 44366209 IC50 = 165000 nM T98092 C6PCZ9 44366232 IC50 = 850000 nM T98092 CRES48 44366233 IC50 = 325000 nM T98092 C7AQ3R 44366260 IC50 = 2100000 nM T98092 CS74HY 44366261 IC50 = 970000 nM T98092 CEH4W6 44366303 IC50 = 820000 nM T98092 CF3B2I 44366350 IC50 = 260000 nM T98092 C0I3BR 44366351 IC50 = 760000 nM T98092 C9HQ5S 44366390 IC50 = 2800000 nM T98092 CY89LF 44366391 IC50 = 1300000 nM T98092 CDJ21S 44366404 IC50 = 500000 nM T98092 CPW1A7 44366405 IC50 = 90000 nM T98092 C4SQ1N 44366450 IC50 = 280000 nM T98092 CUI2X6 44366451 IC50 = 6000 nM T98092 CMCP73 44366452 IC50 = 365000 nM T98092 C2LG1F 44366453 IC50 = 115000 nM T98092 C5Q4VN 44393426 Ki = 100 nM T98092 CP57YU 44393427 Ki = 75 nM T98092 CGX7M4 44393512 Ki = 10 nM T98092 CGP76Z 44393513 Ki = 24 nM T98092 CU0RC4 44393514 Ki = 18 nM T98092 CZAD42 44406917 IC50 = 4100 nM T98092 C0FLH5 44582698 IC50 = 740 nM T98092 C0ON5I 44582699 IC50 = 810 nM T98092 CW3R7N 44582757 IC50 = 740 nM T98092 CCV89D 44582780 IC50 = 880 nM T98092 CZM71K 44582804 IC50 = 600 nM T98092 CWF96D 44582805 IC50 = 450 nM T98092 CYN7C5 44582823 IC50 = 160 nM T98092 CW4P8K 44582824 IC50 = 450 nM T98092 CX94NI 45138814 IC50 = 2.4 nM T98092 CN72XD 45269870 IC50 > 10000 nM T98092 CS30FH 49863381 IC50 = 206 nM T98092 C3YI2V 49863382 IC50 = 950 nM T98092 CS48JU 49863383 IC50 = 4.75 nM T98092 CWI47U 50899161 IC50 = 26.6 nM T98092 CHN71J 52940634 IC50 = 31.2 nM T98092 CQ83LE 52940669 IC50 = 22.9 nM T98092 C2H0IK 52940670 IC50 = 46 nM T98092 CPKZ45 52940671 IC50 = 35.2 nM T98092 C7MA9P 52941831 IC50 = 9.12 nM T98092 CH9QA8 52941859 IC50 = 21.4 nM T98092 C97YWD 52945243 IC50 = 26.7 nM T98092 CE05IO 52945473 IC50 = 218 nM T98092 C43LWJ 52945496 IC50 = 140 nM T98092 C3BCG7 52946681 IC50 = 83.5 nM T98092 CR63JF 52946682 IC50 = 22.8 nM T98092 CH8TZ9 52946683 IC50 = 103 nM T98092 C7KW3U 52947912 IC50 = 23 nM T98092 C4KAU1 52947949 IC50 = 662 nM T98092 CGX04A 52947950 IC50 = 65.2 nM T98092 CS90AU 52952820 IC50 = 33.11 nM T98092 CBWK59 53321090 Ki = 106 nM T98092 CNS79R 53344622 IC50 = 2.7 nM T98092 CPD19A 53357115 IC50 = 350 nM T98092 CMYW90 53357116 IC50 = 630 nM T98092 C75LWY 53357117 IC50 = 500 nM T98092 C40GVQ 53357247 IC50 = 360 nM T98092 CC0Y1S 53357248 IC50 = 390 nM T98092 CPM2F7 53357386 IC50 = 330 nM T98092 COP18F 53357507 IC50 = 520 nM T98092 C4P3GC 53357508 IC50 = 420 nM T98092 C4O0YX 53357509 IC50 = 4.1 nM T98092 C96CAE 53357630 IC50 = 450 nM T98092 C8C9ZH 53358962 IC50 = 1.1 nM T98092 C3VJ0N 56668120 IC50 = 2000000 nM T98092 C30PVF 56675024 IC50 = 2600000 nM T98092 CFMP72 56678333 IC50 = 2100000 nM T98092 CFAY29 56678334 IC50 = 165000 nM T98092 CQB1I0 57384849 Ki = 14 nM T98092 CZK8P2 57384850 Ki = 65 nM T98092 CX67HU 57385085 Ki = 4 nM T98092 C6PXU0 57398046 IC50 = 4.9 nM T98092 C6ZK4A 67978739 Ki = 16 nM T98092 C6RT1L 71590783 IC50 = 740 nM T98092 CC0TY2 71590784 IC50 = 810 nM T98092 CH23LT 71596756 IC50 = 550 nM T98092 CZOT97 71596824 IC50 = 380 nM T98092 CC37ZO 71596825 IC50 = 330 nM T98092 C2IJ6X 71596826 IC50 = 460 nM T98092 CSE28O 73333514 Ki = 23 nM T98092 CDF54U 73333515 Ki = 10.7 nM T98092 CKS08Z 73333613 Ki = 12.4 nM T98092 C5FWY3 73333614 Ki = 43.9 nM T98092 C2LR7I 73333729 Ki = 11.8 nM T98092 CQH16I 73333730 Ki = 36.6 nM T98092 CRA39X 73333846 Ki = 57.7 nM T98092 C47PVY 73347049 IC50 = 680000 nM T98092 CKV1A9 73348786 IC50 = 2.3 nM T98092 CIXM26 73353051 IC50 = 16 nM T98092 C5J6GK 122437357 IC50 = 11.2 nM T98092 CUKL46 127038149 IC50 = 10000 nM T98092 CF7KS5 127038150 IC50 = 10000 nM T98092 C6HPE3 127038151 IC50 = 10000 nM T98092 CQC1L7 127038489 IC50 = 940 nM T98092 CI8EO6 127039060 IC50 = 10000 nM T98092 C7NW5Q 127039075 IC50 = 2760 nM T98092 CSU85H 127039831 IC50 = 10430 nM T98092 CA1P8V 127039832 IC50 = 10260 nM T98092 C2JQ4V 127039851 IC50 = 10000 nM T98092 C1DTR2 127039852 IC50 = 1220 nM T98092 CI03BD 127040172 IC50 = 10800 nM T98092 C0OTQ9 127040173 IC50 = 10000 nM T98092 CA75UB 127040174 IC50 = 10000 nM T98092 CC0GN1 127040175 IC50 = 10000 nM T98092 C8PI2G 127041686 IC50 = 10000 nM T98092 CS0EM4 127041788 IC50 = 10330 nM T98092 CE0KL8 127041789 IC50 = 10000 nM T98092 C35DGM 127042320 IC50 = 11620 nM T98092 C2VGI1 136220121 Ki = 64.7 nM T98092 C2ZA8L 137348679 Ki = 7 nM T98092 CY46VP 137637353 Ki = 4.3 nM T98092 D04PGW 6475368 IC50 = 166 nM T98092 D07ABJ 44358392 IC50 = 783 nM T98092 D07IQR 11639129 IC50 = 361 nM T98092 D0P6TX 3663276 IC50 = 754 nM T98092 D0X5JR 11574097 IC50 = 810 nM T52638 D03LWG 53235510 IC50 > 10000 nM T52638 D07EHV 44814409 IC50 > 10000 nM T52638 D0E3TC 44259 IC50 = 12100 nM T52638 C1ZPA9 1292979 IC50 = 623 nM T52638 C1XS2J 54760383 IC50 > 10000 nM T52638 CV63UL 67240318 IC50 > 10000 nM T52638 CM8LU3 122177129 IC50 = 420 nM T52638 CU5V7A 129318960 IC50 = 39 nM T52638 C38TVL 129318961 IC50 = 750 nM T52638 CX48MD 133080583 EC50 = 352 nM T52638 CTR4A0 135383414 IC50 = 95 nM T52638 C8MY4I 137632407 IC50 = 60 nM T52638 CTKX07 137635009 IC50 = 971 nM T52638 CLK3Y7 137635621 IC50 = 106 nM T52638 C0IMX2 137642056 Ki = 32.43 nM T52638 CVR5C8 137654407 IC50 = 2140 nM T52638 CLMT19 137660903 IC50 = 6 nM T52638 C2MD1Q 155513187 IC50 > 10000 nM T52638 D06HVH 54613583 IC50 > 10000 nM T56556 D00YZD 54726191 IC50 = 67000 nM T56556 D04AIT 5280445 IC50 = 8900 nM T56556 D07BSQ 5994 IC50 = 125892.54 nM T56556 D07POC 176870 IC50 = 50000 nM T56556 D09XZB 123631 IC50 = 1100 nM T56556 D0AZ3C 5291 IC50 = 4897.79 nM T56556 D0BP9C 193962 IC50 = 6000 nM T56556 D0J4JM 5770 IC50 = 12600 nM T56556 D0K8KX 5280343 EC50 = 30 nM T56556 D0OB1J 39186 IC50 = 851138.04 nM T56556 D0Q0PR 54675769 IC50 = 104000 nM T56556 D0R0FE 2520 EC50 = 900 nM T56556 D0R3JB 4212 IC50 = 903.8 nM T56556 D0T0KA 4474 IC50 = 16595.87 nM T56556 D01GFX 11640390 EC50 = 104 nM T56556 D02HTD 25167947 IC50 = 1400 nM T56556 D02QWY 24785538 IC50 = 10200 nM T56556 D0CE0O 11513676 IC50 = 2500 nM T56556 D0G7UX 5284373 EC50 = 1750 nM T56556 D0J1HB 23063810 IC50 = 65400 nM T56556 D0L4FS 5280961 IC50 = 6900 nM T56556 D00OWF 5280953 IC50 = 5080 nM T56556 D04RLX 148201 EC50 = 10 nM T56556 D09FGX 119373 IC50 = 400 nM T56556 D0Q7HO 4705 IC50 = 1730 nM T56556 C4DS3F 2361 IC50 = 6050 nM T56556 CQ9MW6 68077 IC50 = 17000 nM T56556 CJ65ZE 72344 IC50 = 4900 nM T56556 CSHM20 73201 IC50 = 8900 nM T56556 CI5UP7 88881 IC50 = 9200 nM T56556 C5ZCH7 97332 IC50 = 1880 nM T56556 CL97OF 97548 IC50 = 1280 nM T56556 CD8L6K 97696 IC50 = 7900 nM T56556 C6I9HU 97860 IC50 = 19000 nM T56556 C3NC7T 114429 IC50 = 11000 nM T56556 C8NLJ2 145659 IC50 = 8300 nM T56556 CNVB16 146013 IC50 = 1280 nM T56556 C4FEY6 147157 IC50 = 3400 nM T56556 C7E5NC 150893 IC50 = 1400 nM T56556 C4J5ZF 185617 IC50 = 10000 nM T56556 CRE67B 265724 IC50 = 1010 nM T56556 CABJ72 276138 IC50 = 1230 nM T56556 C1Q0WH 281852 IC50 = 1690 nM T56556 CPF26C 324081 IC50 = 10700 nM T56556 C4VJH5 324094 IC50 = 16600 nM T56556 CMC10D 324099 IC50 = 9000 nM T56556 CP5B4K 369597 IC50 = 4900 nM T56556 CKC6U2 369599 IC50 = 2800 nM T56556 CO6AM3 378567 IC50 = 17000 nM T56556 CA9IM5 396723 IC50 = 860 nM T56556 CVN3Z5 403923 IC50 = 451 nM T56556 C5YX1H 406017 IC50 = 30000 nM T56556 CHP8G0 406584 IC50 = 960 nM T56556 CWXZ47 406585 IC50 = 15000 nM T56556 CL6QB8 407032 IC50 = 4800 nM T56556 CC1Q8J 409920 IC50 = 6300 nM T56556 C3YG0Z 436659 IC50 > 20000 nM T56556 CWZ14N 468116 IC50 > 20000 nM T56556 CMT3P0 480764 IC50 = 3100 nM T56556 CL6E7C 609712 IC50 = 10000 nM T56556 C14NHZ 624831 IC50 = 12400 nM T56556 C34KNT 631171 IC50 = 2140 nM T56556 CSA18D 651672 IC50 = 940 nM T56556 C90LPE 688666 IC50 = 6500 nM T56556 CMR6U0 693195 IC50 = 2630 nM T56556 CH0DT9 693197 IC50 = 150 nM T56556 C1NZL9 693198 EC50 = 72 nM T56556 CW2U6N 698956 IC50 = 130 nM T56556 C19VMW 698960 EC50 = 72 nM T56556 C65SGT 712193 IC50 = 645 nM T56556 CH6MV7 715632 IC50 = 6380 nM T56556 C2NI7K 718862 IC50 = 890 nM T56556 CNS78D 719277 IC50 = 1150 nM T56556 CST9W8 719279 IC50 = 1480 nM T56556 CEC0X3 719282 IC50 = 2250 nM T56556 CRX4Q5 719284 IC50 = 1930 nM T56556 C6AKG9 735124 IC50 = 8120 nM T56556 C8OB6U 787509 EC50 = 50 nM T56556 C64RUF 877998 EC50 = 70 nM T56556 CXR0P5 917533 IC50 = 15800 nM T56556 C2X8PT 930478 IC50 = 108 nM T56556 CXQ4P8 1183964 IC50 = 944 nM T56556 CB31HC 1186125 IC50 = 362 nM T56556 CM42KO 1187243 IC50 = 107.15 nM T56556 CYT7E4 1214451 EC50 = 13 nM T56556 CCNX23 1361994 IC50 = 216 nM T56556 C35OEM 1413870 IC50 = 28900 nM T56556 CV7F8O 1418188 IC50 = 405 nM T56556 CAXQ59 1424290 IC50 = 2780 nM T56556 C2FL5J 1553837 IC50 = 250 nM T56556 C5RA6J 1566118 IC50 = 166 nM T56556 CQYO27 1597005 IC50 = 10700 nM T56556 C0M7DO 1696333 IC50 = 1340 nM T56556 COAE97 2176800 IC50 = 1060 nM T56556 C6ZFC1 2463411 IC50 = 791 nM T56556 CG3V9C 2549745 IC50 = 224 nM T56556 C2ZDU4 2562583 IC50 = 570 nM T56556 CFC30O 2789499 EC50 = 11 nM T56556 C01JRM 3034694 IC50 = 9300 nM T56556 C69NQO 3627000 EC50 = 58 nM T56556 C72VLI 4022553 IC50 = 196 nM T56556 C43JKM 4271896 IC50 = 3860 nM T56556 CHV3N6 4786429 IC50 = 360 nM T56556 CKG0Q7 4839583 IC50 = 724 nM T56556 CGKX02 4841865 IC50 = 1320 nM T56556 CN35MZ 4970131 IC50 = 11800 nM T56556 C8PN0C 5280682 IC50 = 680 nM T56556 CF6KZ2 5281677 IC50 = 17200 nM T56556 CQ9GX3 5320462 IC50 = 2000 nM T56556 C2TVO1 5328202 IC50 = 1980 nM T56556 C0O4SM 5332516 IC50 = 2630 nM T56556 CI6TE3 5348770 IC50 = 9230 nM T56556 CTO51S 5352005 IC50 = 540 nM T56556 CQL05G 5355469 IC50 = 3000 nM T56556 CTPE71 5355684 IC50 = 3280 nM T56556 CN8GP9 5355845 IC50 = 16200 nM T56556 C9T0DZ 5355846 IC50 = 10500 nM T56556 CW1UM5 5357488 IC50 = 2200 nM T56556 CU29TR 5373259 IC50 = 530 nM T56556 CV7Z2A 5373273 IC50 = 1060 nM T56556 CRW09S 5373997 IC50 = 3090 nM T56556 C09NZD 5380645 IC50 = 31020 nM T56556 C2KZF0 5476176 IC50 = 2400 nM T56556 CO17YB 5702790 IC50 = 1730 nM T56556 CI4U9Z 5711223 IC50 = 12050 nM T56556 CVF14X 5712116 IC50 = 4970 nM T56556 CCAT78 5723044 IC50 = 2190 nM T56556 CR51QS 5729243 IC50 = 22390 nM T56556 CG25KB 5729341 IC50 = 1950 nM T56556 CE0W8M 5730384 IC50 = 7800 nM T56556 CD18KY 5730712 EC50 = 2100 nM T56556 CA9WL4 5797184 IC50 = 18200 nM T56556 C7LKC3 5822497 IC50 = 10720 nM T56556 C29JCA 5909266 IC50 = 3320 nM T56556 CDLV62 5936200 IC50 = 2200 nM T56556 C9DB2C 5953849 IC50 = 850 nM T56556 CG82WY 5978982 IC50 = 2820 nM T56556 CFO1R0 6063342 IC50 = 1910 nM T56556 CP8O7I 6070899 IC50 = 1470 nM T56556 CMC06O 6123891 IC50 = 6440 nM T56556 C90ACD 6199559 IC50 = 9830 nM T56556 CYX45A 6213016 IC50 = 4910 nM T56556 CV91FR 6213967 EC50 = 1250 nM T56556 C6SZW5 6229071 IC50 = 7290 nM T56556 CU3X5P 6229072 IC50 = 9210 nM T56556 CFO9D1 6256073 IC50 = 8700 nM T56556 CX87NG 6475921 IC50 = 12300 nM T56556 COF72V 6919145 IC50 = 910 nM T56556 C0MGV7 7048595 IC50 = 3790 nM T56556 CNH60W 7946188 IC50 = 7220 nM T56556 C0O7PG 9109771 IC50 = 810 nM T56556 CLIG51 9281828 IC50 = 753 nM T56556 C1IPS5 9283400 EC50 = 85 nM T56556 C0D2SZ 9448204 IC50 = 4280 nM T56556 C4CF5U 9448550 EC50 = 512 nM T56556 C40XDF 9880195 EC50 = 14 nM T56556 CHI5S9 9975676 IC50 = 5910 nM T56556 C26IPN 10047854 IC50 = 5700 nM T56556 CY73KI 10322450 IC50 = 4 nM T56556 C7QYK3 10359377 IC50 = 830 nM T56556 C7Z8IW 10379829 IC50 = 4250 nM T56556 C0V5QI 10394010 IC50 = 11000 nM T56556 CT9MP2 10404096 IC50 = 3800 nM T56556 C36PIN 10407830 IC50 = 8190 nM T56556 C78HZG 10495050 IC50 = 6160 nM T56556 CR9SE7 10540319 IC50 = 6370 nM T56556 CEZ2B4 10612087 IC50 = 1940 nM T56556 CIOL78 10699195 IC50 = 16000 nM T56556 CF1UM5 10746774 IC50 = 29000 nM T56556 CI1RC8 10830017 IC50 = 9100 nM T56556 CT8PY0 10899903 IC50 > 20000 nM T56556 CDX92T 11210677 IC50 = 2460 nM T56556 CL1YX5 11246927 IC50 = 3620 nM T56556 C0SO6D 11312797 IC50 = 930 nM T56556 CL3YO1 11537442 IC50 = 700 nM T56556 C2C3WI 11957988 IC50 = 2089.3 nM T56556 C47ZJY 11996857 IC50 = 20000 nM T56556 CR3X7L 12388142 IC50 = 2890 nM T56556 C0KZQ2 12388145 IC50 = 5210 nM T56556 CS4YL1 12511782 IC50 = 2140 nM T56556 CRE67S 12753643 IC50 = 2580 nM T56556 CT24DO 13147509 IC50 = 920 nM T56556 C5VXB4 13147512 IC50 = 3550 nM T56556 C4GZ8Y 13168110 EC50 = 41 nM T56556 C5X4VH 13250463 IC50 > 20000 nM T56556 CM28RZ 13329020 IC50 = 424 nM T56556 C1U9IN 13707046 IC50 = 2890 nM T56556 C5DMA3 14034811 IC50 = 260 nM T56556 CRIH25 14259001 IC50 = 6600 nM T56556 CG0ZK1 14531326 EC50 = 900 nM T56556 C2LA5S 15556477 IC50 = 5680 nM T56556 CJ78CV 15648569 IC50 = 720 nM T56556 CJ5XV3 15965811 IC50 > 100000 nM T56556 C19FNV 15993184 EC50 = 12 nM T56556 CLD92G 15999199 EC50 = 4.7 nM T56556 C0A3IV 16092354 IC50 = 1190 nM T56556 C3TH4N 16092356 IC50 = 689 nM T56556 C7DW6Y 16092357 EC50 = 131 nM T56556 C7TBI5 16339054 IC50 = 15400 nM T56556 CMVW98 16618023 EC50 = 1310 nM T56556 CD04RW 16745324 IC50 = 2500 nM T56556 CN73EP 16805556 IC50 = 4790 nM T56556 CPOZ18 17375361 IC50 = 11200 nM T56556 CX06NR 17412108 IC50 = 16000 nM T56556 C5MOF7 17497142 IC50 = 10400 nM T56556 COG12F 17585222 IC50 = 8680 nM T56556 CPE15U 18004103 IC50 = 14500 nM T56556 CYSV63 19392346 IC50 = 60000 nM T56556 C3UT8G 20239593 IC50 = 170 nM T56556 CJ4Z1L 20646908 IC50 = 20900 nM T56556 C59FWO 20646970 IC50 = 51300 nM T56556 CIZV45 20646979 IC50 = 40000 nM T56556 CB7T2K 20963109 EC50 = 1.2 nM T56556 C2RQF6 21002393 IC50 = 1180 nM T56556 CB50QE 21418982 IC50 = 648 nM T56556 CCJ3M5 22004538 IC50 = 32400 nM T56556 CFI13S 22310708 IC50 = 420 nM T56556 CDQX04 22330280 IC50 = 462 nM T56556 C9IHU3 22330507 IC50 = 1990 nM T56556 C85SLA 23792651 IC50 = 8900 nM T56556 C7TOB4 23906108 IC50 = 1660 nM T56556 CU1G8A 23940255 IC50 = 87.1 nM T56556 CRCA82 23965087 EC50 = 21 nM T56556 CX2UF8 24016488 IC50 = 612 nM T56556 C2XB8M 24017959 IC50 = 183 nM T56556 C3ESV6 24178402 EC50 = 90000 nM T56556 C6AU1C 24204512 IC50 = 790 nM T56556 CU7LR8 24208774 IC50 = 458 nM T56556 CLY6U7 24626581 IC50 = 921 nM T56556 CCPS81 24764502 IC50 = 35000 nM T56556 CKW04J 24807980 EC50 = 7000 nM T56556 CJUW92 24807981 EC50 = 1500 nM T56556 CP8H2D 24807987 EC50 = 58000 nM T56556 C9T7BZ 24808155 EC50 = 75000 nM T56556 C9SMO0 24808156 EC50 = 120000 nM T56556 CW4EM8 24808157 EC50 = 150000 nM T56556 C7UV4H 24808344 EC50 = 500 nM T56556 C9F8CE 24826109 IC50 = 430 nM T56556 C9LXA0 24827935 IC50 = 350 nM T56556 C39SHG 24882446 IC50 = 23988.33 nM T56556 CF1JU8 24978503 IC50 = 230 nM T56556 C60EJI 25113688 EC50 = 73000 nM T56556 CS3ZN9 25195356 IC50 = 350 nM T56556 C2YA4G 25217469 IC50 = 1750 nM T56556 CM80XH 25222999 IC50 = 60 nM T56556 CSRV83 25223000 IC50 = 172 nM T56556 C26ZQR 25223001 IC50 = 632 nM T56556 C0S7AF 25223002 IC50 = 317 nM T56556 CZ4A5K 25223105 IC50 = 858 nM T56556 CKY89F 25223106 IC50 = 1990 nM T56556 CIJU21 25223199 IC50 = 119 nM T56556 CUZ5S9 25223200 IC50 = 183 nM T56556 C03FQV 25223201 IC50 = 552 nM T56556 C8S6UH 25223298 IC50 = 1015 nM T56556 CZQE36 25223299 IC50 = 977 nM T56556 C6O2ZR 25225119 EC50 = 30000 nM T56556 C8W9VD 25249649 IC50 > 10000 nM T56556 C78LKG 26213315 IC50 = 4100 nM T56556 CJPM47 31538107 IC50 = 1350 nM T56556 CI4AK1 39969954 IC50 = 14400 nM T56556 C0X8OT 44221093 IC50 = 10200 nM T56556 C9BNA1 44248179 EC50 = 63.2 nM T56556 C4DBF9 44257640 IC50 = 5900 nM T56556 C2NK1G 44428701 IC50 = 770 nM T56556 C4NCQ7 44428711 IC50 > 20000 nM T56556 CUIG60 44428712 IC50 = 450 nM T56556 CQ6A3K 44428713 IC50 = 560 nM T56556 CNBA28 44428714 IC50 = 1380 nM T56556 C43CIH 44451513 IC50 = 77624.71 nM T56556 CMHP85 44451563 IC50 = 263026.8 nM T56556 C29SBO 44451564 IC50 = 6606.93 nM T56556 C1G2CB 44451590 IC50 = 7585.78 nM T56556 C6NW0Q 44451617 IC50 = 14454.4 nM T56556 C1ENZ0 44451645 IC50 = 44668.36 nM T56556 CB0OL9 44451671 IC50 = 6025.6 nM T56556 CC9LK5 44451719 IC50 = 6025.6 nM T56556 CS4RX9 44451745 IC50 = 7244.36 nM T56556 C9Z4VY 44451773 IC50 = 12882.5 nM T56556 CTP09O 44451801 IC50 = 11481.54 nM T56556 CP69AF 44451832 IC50 = 22908.68 nM T56556 C45VCM 44451857 EC50 = 15000 nM T56556 C4T5UP 44451866 IC50 = 21877.62 nM T56556 CI1Y5L 44451888 IC50 = 64565.42 nM T56556 CP3B8R 44451889 IC50 = 36307.81 nM T56556 C3S5OK 44451912 IC50 = 5011.87 nM T56556 C6M3ZN 44451913 IC50 = 47863.01 nM T56556 C9AOQ4 44562411 IC50 = 15135.61 nM T56556 CLBO81 44565459 IC50 = 9080 nM T56556 C7NRZ8 44565460 IC50 = 6760 nM T56556 CN03BJ 44565480 IC50 = 2610 nM T56556 C38FXL 44565481 IC50 = 58400 nM T56556 CZUI80 44565482 IC50 = 74100 nM T56556 CZT54M 44565509 IC50 = 74100 nM T56556 C4Q2ER 44593438 IC50 = 24547.09 nM T56556 CE6F2U 45272659 IC50 = 22600 nM T56556 COPA25 46227750 IC50 = 10200 nM T56556 COA30H 46227751 IC50 = 630 nM T56556 CLWR13 46227752 IC50 = 500 nM T56556 C54HFY 46232422 IC50 > 100000 nM T56556 C5TJ4Y 46232423 IC50 = 25200 nM T56556 CY2RN7 46232494 IC50 > 100000 nM T56556 CW9J2R 46232495 IC50 > 100000 nM T56556 CO7V0S 46232496 IC50 > 100000 nM T56556 CZ89LA 46232497 IC50 = 15400 nM T56556 C4RUB7 46232498 IC50 = 6400 nM T56556 CR96LU 46232536 IC50 = 18800 nM T56556 C6UW4G 46232537 IC50 = 11100 nM T56556 C5ATF2 46232538 IC50 = 23200 nM T56556 CKXH76 46232539 IC50 > 100000 nM T56556 CXI72Q 46359934 IC50 = 1430 nM T56556 C0L6DC 46359963 IC50 = 60 nM T56556 CD64QE 49816175 IC50 = 1270 nM T56556 C72QDG 49844541 IC50 = 8920 nM T56556 CY4XL9 50806112 IC50 = 1890 nM T56556 C5PHF6 51041756 IC50 = 15500 nM T56556 C5M9DP 51041990 IC50 = 8400 nM T56556 CL29IG 53321447 IC50 = 6500 nM T56556 CPL41H 54341571 IC50 = 13600 nM T56556 C4Z7MF 54580539 IC50 > 100000 nM T56556 C96NWY 54580541 IC50 > 6200 nM T56556 CN30LW 54581539 IC50 > 5000 nM T56556 C6AIG3 54582535 IC50 = 183 nM T56556 CY24RJ 54582627 IC50 = 508 nM T56556 CN38OK 54583506 IC50 > 50000 nM T56556 CLTM38 54586400 IC50 > 50000 nM T56556 CK52PH 54586413 IC50 = 130 nM T56556 CIAU38 54587418 IC50 > 50000 nM T56556 CKZ01T 54587433 IC50 = 390 nM T56556 CB4DX1 54754510 IC50 = 450 nM T56556 CS7XP1 54754512 IC50 = 350 nM T56556 C4WO8B 56681840 IC50 = 270 nM T56556 C1H9ML 56764960 IC50 = 1390 nM T56556 C5EN2Q 56924700 IC50 = 170 nM T56556 CTX1N3 56924701 EC50 = 31 nM T56556 CP1VK5 56951135 IC50 = 16300 nM T56556 C2SF8B 56951136 IC50 = 470 nM T56556 C2KMN3 56951137 IC50 = 180 nM T56556 CAT80Q 56951138 IC50 = 200 nM T56556 CJ8C4Y 56951261 IC50 = 160 nM T56556 C0N9YK 57394942 IC50 = 7260 nM T56556 CTN9Q0 57396989 IC50 = 940 nM T56556 CR8MW5 57398461 IC50 = 1930 nM T56556 C9LPN4 57400130 IC50 = 3210 nM T56556 CW7B0M 57614266 IC50 = 2210 nM T56556 CQZS56 66636984 IC50 = 4100 nM T56556 C5RHD4 66637000 IC50 = 230 nM T56556 C5IT4O 70686509 IC50 = 28200 nM T56556 C9Y1TS 70686876 IC50 = 3270 nM T56556 C9B5TD 70690679 IC50 = 13300 nM T56556 CA1WO9 70696907 IC50 = 4300 nM T56556 CE1QO3 71296003 EC50 = 42 nM T56556 C2YIM8 71449571 IC50 = 5120 nM T56556 C7VGS2 71453183 IC50 = 1530 nM T56556 C1ZHB6 71453184 IC50 = 8220 nM T56556 C6ZOP0 71453185 IC50 = 970 nM T56556 CY5LI4 71454921 IC50 = 7950 nM T56556 C3OLA2 71454922 IC50 = 9350 nM T56556 C5T0NL 71454923 IC50 = 152 nM T56556 C0CIZ8 71458549 IC50 = 5910 nM T56556 CTWA64 71458550 IC50 = 5930 nM T56556 C0U5FJ 71458829 IC50 = 112 nM T56556 CA02ZE 71460396 IC50 = 3750 nM T56556 CZS0L5 71460397 IC50 = 2460 nM T56556 CPQ16X 71462088 IC50 = 6830 nM T56556 C4ZD2W 71492590 IC50 = 207 nM T56556 C0P6IG 71492759 IC50 = 176 nM T56556 C3T8ZF 71560811 EC50 = 18 nM T56556 CFN89Y 71560812 EC50 = 500 nM T56556 C42SMF 71560938 EC50 = 10000 nM T56556 C98LPJ 71560939 EC50 = 1000 nM T56556 CWCJ73 71624433 IC50 = 1100 nM T56556 CN3KI6 71624434 IC50 = 3214 nM T56556 C9RD7L 71624435 IC50 = 760 nM T56556 CGA8B3 71624544 IC50 = 544 nM T56556 C8YT2N 71624545 IC50 = 1461 nM T56556 CI7QT2 71624546 IC50 = 641 nM T56556 CA7P8Q 71624648 IC50 = 1540 nM T56556 C18BKV 71624649 IC50 = 1031 nM T56556 CMA90D 71624650 IC50 = 237 nM T56556 C3KVP8 71624651 IC50 = 591 nM T56556 CB40GR 71624766 IC50 = 943 nM T56556 CEF9J8 71624767 IC50 = 839 nM T56556 C0Z3PN 71682039 EC50 > 100000 nM T56556 CV5Z9M 71682040 EC50 > 100000 nM T56556 C1IZT7 71682041 EC50 > 100000 nM T56556 COV12T 71682195 EC50 > 100000 nM T56556 C3Y4FW 71682196 EC50 > 100000 nM T56556 CLF3I8 71682197 EC50 > 100000 nM T56556 CN6Q3L 71696716 EC50 = 12.3 nM T56556 CQCF98 71724480 EC50 = 29.5 nM T56556 C1PR7Z 71724504 EC50 = 7.2 nM T56556 CA7K8Z 71724506 EC50 = 57.5 nM T56556 CD9KH7 71724532 EC50 = 14.8 nM T56556 CWR2L5 71724556 EC50 = 0.9 nM T56556 C4ODQ2 71724557 EC50 = 160 nM T56556 C7T0UM 71724558 EC50 = 23.6 nM T56556 CUL9E2 71724582 EC50 = 38.7 nM T56556 CNW68B 71724606 EC50 = 371.7 nM T56556 CCZ9B3 71724628 EC50 = 18 nM T56556 C48CAR 72735227 IC50 = 400 nM T56556 CI6E4O 72735228 IC50 = 1550 nM T56556 CXWG13 72735229 EC50 = 3.5 nM T56556 CG7S2T 72735404 IC50 = 240 nM T56556 C2O8IJ 72735405 IC50 = 190 nM T56556 CVZK97 72735406 IC50 = 260 nM T56556 CFL45O 72735407 IC50 = 110 nM T56556 CKF0Q7 72735408 IC50 = 680 nM T56556 C5I7XA 72735580 IC50 = 610 nM T56556 CY20ED 72735581 IC50 = 470 nM T56556 C6D7QV 72735582 IC50 = 320 nM T56556 CR91NX 72735583 IC50 = 1520 nM T56556 CQ5NB6 72950792 IC50 = 426 nM T56556 CF57OZ 73346145 IC50 = 1060 nM T56556 CUX0H5 73346146 IC50 = 4270 nM T56556 C90GUQ 73347669 IC50 = 3070 nM T56556 C7KIJ0 73349189 IC50 = 2440 nM T56556 CC9F2B 73349190 IC50 = 11100 nM T56556 C7DAJ3 73352266 IC50 = 4970 nM T56556 CK3EX6 73355255 IC50 = 2710 nM T56556 CKH8D4 73355256 IC50 = 6120 nM T56556 C7NTB0 73356802 IC50 = 457 nM T56556 CIWH89 73356803 IC50 = 17900 nM T56556 C25AUR 73356804 IC50 = 4840 nM T56556 C8NC1P 76310339 EC50 = 220 nM T56556 CBDY35 76310340 EC50 = 570 nM T56556 CH9B2W 76317551 EC50 = 570 nM T56556 CVN95Y 76317552 EC50 = 530 nM T56556 C2U1VA 76321285 EC50 = 100 nM T56556 C3T5OH 76324898 EC50 = 1670 nM T56556 CCP3L1 76324899 IC50 > 2000 nM T56556 CD4V0F 76328460 IC50 = 250 nM T56556 CZ3P5R 76332141 EC50 = 80 nM T56556 C7ISD3 76335756 EC50 = 500 nM T56556 CPJ5M2 76335757 EC50 = 1270 nM T56556 CZ4SE6 76335758 EC50 = 500 nM T56556 C67ASV 76335759 EC50 = 1110 nM T56556 C5Z3GF 76335761 EC50 = 600 nM T56556 C73WDV 85922974 IC50 > 10000 nM T56556 CRB93S 89784681 EC50 = 69.3 nM T56556 CG71EX 89784708 EC50 = 28 nM T56556 C4ZOX6 89784717 EC50 = 190 nM T56556 C0ZQO6 89784722 EC50 = 32.8 nM T56556 C4U5CZ 89784733 EC50 = 54 nM T56556 CW17YB 89784735 EC50 = 59 nM T56556 C0VD4P 89784742 EC50 = 34.1 nM T56556 CZT7B9 89784751 EC50 = 47 nM T56556 CH70XJ 89784752 EC50 = 24.9 nM T56556 C6MRA2 89784753 EC50 = 24.5 nM T56556 C1JH4L 89784756 EC50 = 230 nM T56556 CN1RD8 89784760 EC50 = 195 nM T56556 C2YB6Q 89784818 EC50 = 54 nM T56556 CSK8X6 89784827 EC50 = 15.5 nM T56556 CENX80 89785043 EC50 = 32.5 nM T56556 CY46QV 89785047 EC50 = 17.5 nM T56556 CQL7T6 89785059 EC50 = 17 nM T56556 CENR59 89785064 EC50 = 235 nM T56556 CVZG56 89785117 EC50 = 86.1 nM T56556 CT43OU 89785127 EC50 = 32 nM T56556 C3FB6Q 89785132 EC50 = 30.5 nM T56556 C4S9WG 89785146 EC50 = 20 nM T56556 CCE95J 89785148 EC50 = 16.5 nM T56556 C9SBA1 89785178 EC50 = 90 nM T56556 CSI51G 89785190 EC50 = 19.7 nM T56556 CGB2P5 89785210 EC50 = 302.5 nM T56556 CTY1H5 89785238 EC50 = 48 nM T56556 CHGX10 89785254 EC50 = 195 nM T56556 CB1FR2 89794901 EC50 = 3.3 nM T56556 C43AXK 89795130 EC50 = 82.5 nM T56556 C70LJV 89795278 EC50 = 242.5 nM T56556 CFU4W2 89795305 EC50 = 152.5 nM T56556 CVB23M 89795326 EC50 = 3.6 nM T56556 CX1W9Z 89795330 EC50 = 0.9 nM T56556 C7XG4U 89795333 EC50 = 111 nM T56556 C7W1TP 89795335 EC50 = 36 nM T56556 CAX9S0 89795337 EC50 = 3.3 nM T56556 COB3Z9 89795340 EC50 = 1.7 nM T56556 C6BW0Q 89795341 EC50 = 15.8 nM T56556 COVK20 90142631 IC50 > 25000 nM T56556 CUHC90 90469229 EC50 = 3600 nM T56556 C05JQB 90469230 EC50 = 2500 nM T56556 C41EMT 90469289 EC50 = 1300 nM T56556 CA1VH0 90469291 EC50 = 2600 nM T56556 C4NX2Q 90469293 EC50 = 2600 nM T56556 C0NW8T 90469355 EC50 = 700 nM T56556 CJK73Q 90655473 EC50 = 700 nM T56556 CFX2C0 90655474 EC50 = 300 nM T56556 CYU3G9 90655475 EC50 = 400 nM T56556 CGWI98 90655476 EC50 = 15 nM T56556 C1D9TM 90655477 EC50 = 1400 nM T56556 C8A9RT 90655478 EC50 = 1100 nM T56556 CHKF72 90655479 EC50 = 2300 nM T56556 CFS75L 90655480 EC50 = 800 nM T56556 CA57QF 90655481 EC50 = 1300 nM T56556 C78PYH 90655482 EC50 = 500 nM T56556 CM1X5R 90655483 EC50 = 1100 nM T56556 CSD17I 90655484 EC50 = 1800 nM T56556 CF4Z8T 91669184 IC50 = 600 nM T56556 C3G6AI 91964346 IC50 = 953 nM T56556 CL15PA 91964352 IC50 = 300 nM T56556 C8BRG2 101876951 EC50 = 200 nM T56556 C24YLQ 101913604 IC50 = 490 nM T56556 CYM1I6 101913605 IC50 = 1600 nM T56556 CQ81YV 101913606 IC50 = 210 nM T56556 C86WSC 117777746 EC50 = 5.2 nM T56556 C9E0BT 117777811 EC50 = 4.1 nM T56556 C9YPJ7 117803128 EC50 = 25.5 nM T56556 C2UY8J 118017356 IC50 = 1700 nM T56556 CP14NL 118017358 IC50 = 1810 nM T56556 C7L8PT 118017419 IC50 = 1700 nM T56556 C7YH4G 118017423 IC50 = 610 nM T56556 C0OQ9P 118716252 EC50 = 4100 nM T56556 CK0H3V 118716255 EC50 = 400 nM T56556 C3VRT8 118716258 EC50 = 1500 nM T56556 CNS3X0 118716259 EC50 = 1300 nM T56556 CS9IV4 118716261 EC50 = 400 nM T56556 C5FD4B 118716262 EC50 = 800 nM T56556 C3BY1A 118716264 EC50 = 600 nM T56556 CLAZ45 118716265 EC50 = 3000 nM T56556 C62JPR 118716267 EC50 = 3400 nM T56556 C6JIC7 118717839 EC50 = 700 nM T56556 CLAF39 118719581 IC50 = 310 nM T56556 CHIB60 118719582 IC50 = 700 nM T56556 CFGK85 118719583 IC50 = 3000 nM T56556 CXO3V7 118719584 IC50 = 20000 nM T56556 CPI2F5 118719585 IC50 = 610 nM T56556 CCI1E7 118737162 IC50 = 184 nM T56556 C0D4GP 118737164 IC50 = 100 nM T56556 C5WYN2 118737166 IC50 = 261 nM T56556 CGT48U 118737167 IC50 = 78.9 nM T56556 CC8Q3G 118737168 IC50 = 118 nM T56556 CNZ06S 118737171 IC50 = 137 nM T56556 C3M9PE 118737173 IC50 = 451 nM T56556 C8O2WM 118737174 IC50 = 11200 nM T56556 C41ROW 118737175 IC50 = 106 nM T56556 C2UZG9 118737176 IC50 = 269 nM T56556 CUSI65 118737177 IC50 = 201 nM T56556 C85ZHJ 118737178 IC50 = 117 nM T56556 CR75MD 118737179 IC50 = 73 nM T56556 CEM28H 118737180 IC50 = 180 nM T56556 C3IH1T 118737181 IC50 = 64.2 nM T56556 C5SRA7 118737182 IC50 = 79.4 nM T56556 CU6EP1 122179376 IC50 = 357 nM T56556 CIL20J 122179390 IC50 = 45 nM T56556 C0OUW1 122179391 IC50 = 38 nM T56556 CRF71Q 122420973 IC50 = 1810 nM T56556 CCE46L 126587406 EC50 = 3.9 nM T56556 CN0LZ6 126739167 IC50 = 2330 nM T56556 CSR0Y7 127028060 IC50 > 100000 nM T56556 C8Z2XI 127028354 IC50 > 100000 nM T56556 C8Q9DG 127028355 IC50 > 100000 nM T56556 CRI72H 127028356 IC50 > 100000 nM T56556 C5A1NO 127028392 IC50 = 9640 nM T56556 CUC9I4 127040367 IC50 > 100000 nM T56556 C0I9VF 127040368 IC50 > 100000 nM T56556 CX9JE1 127040369 IC50 = 34900 nM T56556 CRM9W5 127040370 IC50 = 12000 nM T56556 CJY60W 127042304 IC50 > 100000 nM T56556 CO2P8K 127042305 IC50 = 99700 nM T56556 C56HDS 127042306 IC50 = 37600 nM T56556 CZ0E5J 127042554 IC50 = 230 nM T56556 C90ELS 127042555 IC50 = 230 nM T56556 C87PMI 127042802 IC50 = 87800 nM T56556 CRQ7U8 127042918 IC50 = 36900 nM T56556 C39PWZ 127042920 IC50 = 66600 nM T56556 C21DSU 127042921 IC50 > 100000 nM T56556 C6UZ7C 127042922 IC50 > 100000 nM T56556 CSBM31 127042943 IC50 = 12200 nM T56556 C12BJD 127042944 IC50 = 38200 nM T56556 C42ZKN 127044753 IC50 = 210 nM T56556 CA8P0B 127044754 IC50 = 310 nM T56556 CUF52K 127044901 IC50 = 840 nM T56556 CF3ML0 127044902 IC50 = 680 nM T56556 C7GXK0 127044903 IC50 = 1230 nM T56556 CP1K0B 127044904 IC50 = 390 nM T56556 CO3AX7 127044909 IC50 = 290 nM T56556 C63KNP 127044910 IC50 = 880 nM T56556 CP2U0C 127044913 IC50 = 360 nM T56556 C9SE5Y 127044914 IC50 = 3130 nM T56556 CB4JL3 127044915 IC50 = 1090 nM T56556 C9Z8XO 127045057 IC50 = 1710 nM T56556 C3FG1L 127045064 IC50 = 190 nM T56556 CM1B6D 127045208 IC50 = 1300 nM T56556 CZAL20 127045209 IC50 = 890 nM T56556 C4DH6E 127045210 IC50 = 320 nM T56556 CFX5J3 127045211 IC50 = 460 nM T56556 C5F2BE 127045212 IC50 = 970 nM T56556 CYT62M 127045213 IC50 = 680 nM T56556 C6R5MV 127045214 IC50 = 600 nM T56556 CZBJ54 127048170 IC50 = 8710 nM T56556 C6L0AF 127049502 IC50 = 8240 nM T56556 CK1SN3 127049508 IC50 = 14300 nM T56556 CB9EV4 127049509 IC50 = 6070 nM T56556 C1VP2D 127052887 IC50 = 7680 nM T56556 CG9TE5 127052888 IC50 = 9940 nM T56556 CA7N9R 127052889 IC50 = 4680 nM T56556 CX20OQ 129903920 EC50 = 10 nM T56556 CX48UI 129904103 IC50 = 1200 nM T56556 CK8S4T 132285218 IC50 = 26 nM T56556 C1WG6D 132510852 IC50 = 38 nM T56556 CH3VU5 132510853 IC50 = 29 nM T56556 C5CT0K 132547158 EC50 = 20 nM T56556 C1V7GY 134129908 IC50 = 127 nM T56556 C9VJC1 134129912 IC50 > 10000 nM T56556 CK1TS2 134129976 IC50 = 280 nM T56556 CQ5N3X 134129987 IC50 = 129 nM T56556 C3B1NJ 134130004 IC50 > 10000 nM T56556 CDG0S3 134130015 IC50 = 66.9 nM T56556 C13RTP 134130119 IC50 = 212 nM T56556 CG0NC4 134130126 IC50 = 117 nM T56556 C71PUG 134130154 IC50 = 308 nM T56556 CM40NH 134130306 IC50 > 10000 nM T56556 CCP16R 134130324 IC50 > 10000 nM T56556 C7EVF0 134130371 IC50 = 4390 nM T56556 CR6Z4W 134130497 IC50 = 150 nM T56556 C90RDH 134130514 IC50 = 223 nM T56556 CA7QF6 134130525 IC50 = 319 nM T56556 CZF1D2 134130601 IC50 = 168 nM T56556 CYLW12 134130603 IC50 > 10000 nM T56556 C63NSK 134130669 IC50 = 131 nM T56556 CK15FY 134130999 IC50 = 832 nM T56556 C6LRO0 134131064 IC50 = 208 nM T56556 C36TJZ 134131208 IC50 > 10000 nM T56556 CD69RC 134131216 IC50 = 300 nM T56556 CWP09Q 134131281 IC50 = 96.6 nM T56556 CYT40U 134131325 IC50 > 10000 nM T56556 C1JP2L 134131336 IC50 = 330 nM T56556 C6GIZ2 134131389 IC50 = 251 nM T56556 CB7A2U 134131478 IC50 = 311 nM T56556 CQ8PC9 134131521 IC50 = 679 nM T56556 C1Q0BR 134131558 IC50 = 793 nM T56556 C6QKS0 134131773 EC50 = 540 nM T56556 CDJ2L0 134133476 IC50 = 7100 nM T56556 CVRT47 134134470 IC50 = 4900 nM T56556 CA18ZH 134137512 EC50 = 4350 nM T56556 CJTO68 134140233 EC50 = 340 nM T56556 CQO05X 134141004 IC50 = 7800 nM T56556 C3PIE7 134141342 IC50 = 8900 nM T56556 CPJC31 134144364 EC50 = 380 nM T56556 C9FZI6 134147046 EC50 = 86 nM T56556 CMUK36 134147167 EC50 = 910 nM T56556 C8CIP6 134148609 EC50 = 360 nM T56556 C2Z5LD 134148627 EC50 = 360 nM T56556 CXV6P1 134149485 EC50 = 550 nM T56556 CUBF46 134149834 EC50 = 280 nM T56556 C9Q4YF 134151298 EC50 = 630 nM T56556 C48WKX 134151943 EC50 = 1050 nM T56556 CE14NO 134156590 IC50 = 7400 nM T56556 C4HTR0 134156671 EC50 = 260 nM T56556 CMN2A4 135418331 IC50 = 12800 nM T56556 C41IEM 135659059 IC50 > 20000 nM T56556 CO69BC 135885017 IC50 = 11900 nM T56556 C09BGP 135885019 IC50 = 5900 nM T56556 CV4F5D 137631464 IC50 = 507 nM T56556 COU58A 137631903 EC50 = 116 nM T56556 CL7J6T 137632165 IC50 = 128 nM T56556 CD5VI8 137632443 IC50 = 1267 nM T56556 CV09DQ 137632591 IC50 = 594 nM T56556 CXA82V 137632731 IC50 = 1100 nM T56556 C29XTR 137633043 IC50 = 621 nM T56556 CF73VM 137634351 EC50 = 85 nM T56556 CKCE38 137634438 EC50 = 72 nM T56556 C39YOJ 137634518 IC50 = 4260 nM T56556 CS26GV 137634543 IC50 = 541 nM T56556 CI2K0G 137634736 IC50 = 454 nM T56556 CB0ZJ4 137635897 EC50 = 16 nM T56556 CS3RK1 137636023 IC50 = 628 nM T56556 C54LGH 137636095 EC50 = 16 nM T56556 CI1S9R 137636359 IC50 = 146 nM T56556 C51AGO 137636525 EC50 = 8 nM T56556 CEUR16 137637400 IC50 = 605 nM T56556 CUWZ73 137637797 IC50 = 206 nM T56556 C15FLS 137638403 EC50 = 676 nM T56556 CJ57LP 137638487 EC50 = 141 nM T56556 CFL5V7 137638559 IC50 = 488 nM T56556 C1CAL5 137638992 IC50 = 882 nM T56556 CI3NO0 137639122 IC50 = 1070 nM T56556 CI5Z8K 137639498 EC50 = 47 nM T56556 CTNP09 137639885 EC50 = 4 nM T56556 C8DL5H 137639918 EC50 = 37.1 nM T56556 C5IP1S 137640378 EC50 = 210 nM T56556 C91SBQ 137640534 EC50 = 3 nM T56556 CV3QD9 137641058 EC50 = 13 nM T56556 CI0KU2 137643961 EC50 = 22 nM T56556 C36TRI 137644856 IC50 = 952 nM T56556 CS4Z5B 137644952 IC50 = 283 nM T56556 C9HCB1 137645106 EC50 = 11 nM T56556 CP42GX 137645755 IC50 = 1656 nM T56556 CN3Y8B 137646060 IC50 = 403 nM T56556 C5LFG0 137646752 EC50 = 7 nM T56556 CUP1D3 137646767 EC50 = 32 nM T56556 CTN5H3 137647282 IC50 = 2563 nM T56556 C1FM8R 137647675 EC50 = 4 nM T56556 CV2FL8 137647707 EC50 = 22 nM T56556 CVL5T7 137648146 EC50 = 79 nM T56556 CBL59T 137648334 EC50 = 8 nM T56556 CAU49L 137648335 EC50 = 4 nM T56556 C15MCA 137648533 IC50 = 838 nM T56556 CMR58G 137649090 IC50 = 164 nM T56556 C8UYC1 137649208 EC50 = 5 nM T56556 CX1NH9 137649265 EC50 = 14 nM T56556 CH07EY 137649297 IC50 = 355 nM T56556 C0W1LM 137649303 EC50 = 16 nM T56556 CYP3S6 137649349 IC50 = 325 nM T56556 CZF79C 137649780 IC50 = 1202 nM T56556 CLTE54 137650017 EC50 = 16 nM T56556 C03KMV 137650224 IC50 = 1515 nM T56556 CBAK32 137650656 IC50 = 1380 nM T56556 C5S9OL 137651096 IC50 = 512 nM T56556 C2ZVM8 137651212 IC50 = 1713 nM T56556 CC0H4S 137651220 EC50 = 82 nM T56556 C60QXZ 137651369 EC50 = 9 nM T56556 CM0SC5 137651605 EC50 = 140 nM T56556 C9PE5G 137652835 IC50 = 519 nM T56556 CDZ5I0 137652882 IC50 = 299 nM T56556 CS14NG 137652949 EC50 = 4 nM T56556 CXS2E7 137653095 EC50 = 4 nM T56556 C2B9JN 137653194 IC50 = 472 nM T56556 CN6QH5 137653329 EC50 = 85 nM T56556 C65IAD 137653455 IC50 = 985 nM T56556 C59ZRO 137653532 IC50 = 910 nM T56556 CB1Y8V 137655046 IC50 = 348 nM T56556 C6RP1Z 137655517 IC50 = 354 nM T56556 C89NMB 137655783 IC50 = 1530 nM T56556 C12YJV 137655818 IC50 = 5270 nM T56556 CTV4I1 137655973 IC50 = 122 nM T56556 C0N1TD 137656929 IC50 = 866 nM T56556 COY89M 137657641 EC50 = 145 nM T56556 C5C0KF 137658808 EC50 = 1540 nM T56556 CTO85K 137659047 IC50 = 6400 nM T56556 CB8CJ2 137659409 IC50 = 691 nM T56556 C9HU7R 137659989 IC50 = 325 nM T56556 C8MXN5 137661038 EC50 = 2 nM T56556 C31GEP 137661880 IC50 = 750 nM T56556 CPI3E4 137662036 IC50 = 1630 nM T56556 C7SH6Z 137662093 EC50 = 12 nM T56556 CP1M2F 137662213 IC50 = 2121 nM T56556 CC1QL5 139593871 IC50 = 2130 nM T56556 C5PKZ2 139593897 IC50 = 951 nM T56556 C9USZ1 145949183 EC50 = 4 nM T56556 C3H7QO 145949352 EC50 = 29 nM T56556 C43QGK 145949445 IC50 = 284 nM T56556 CFN6T2 145949660 EC50 = 11 nM T56556 C2X7WS 145950031 IC50 = 44.8 nM T56556 CHB1S3 145950435 IC50 = 57.7 nM T56556 CZRP27 145950520 IC50 = 51.5 nM T56556 CB7KD0 145950545 EC50 = 2 nM T56556 CUB64Y 145950625 EC50 = 690 nM T56556 CNG6V3 145950683 IC50 = 78.7 nM T56556 CK6YR0 145950764 EC50 = 19.5 nM T56556 C07XUY 145950844 IC50 = 61.4 nM T56556 C94HRD 145950874 EC50 = 577 nM T56556 CE4SY2 145950964 IC50 = 1150 nM T56556 CUY09I 145950988 IC50 = 127 nM T56556 CIZ82R 145951128 IC50 = 1040 nM T56556 CR31OX 145951139 IC50 = 336 nM T56556 C4TRJ3 145951213 IC50 = 799 nM T56556 C53MCJ 145951316 IC50 = 65.3 nM T56556 CSYV28 145951611 EC50 = 19 nM T56556 CUD94F 145952004 EC50 = 63 nM T56556 C8Y7ND 145952143 IC50 = 66.3 nM T56556 C5V1MZ 145952691 IC50 = 801 nM T56556 C9O3IC 145952963 IC50 = 1770 nM T56556 C1L4NV 145953000 EC50 = 0.6 nM T56556 CIF74V 145953301 IC50 = 726 nM T56556 C5Z0BT 145953360 IC50 = 33 nM T56556 COSR30 145953465 IC50 = 369 nM T56556 CW97IA 145953788 IC50 = 904 nM T56556 CC3GQ9 145954340 EC50 = 21.8 nM T56556 C21XAV 145954560 EC50 = 1230 nM T56556 C2KBR1 145954586 IC50 = 30.2 nM T56556 CQ7Y6U 145955013 EC50 = 48 nM T56556 C7LP2U 145955206 EC50 = 6 nM T56556 CJ3ET0 145955421 EC50 = 10 nM T56556 CBI96G 145955592 IC50 = 20 nM T56556 C06LAX 145955721 IC50 = 2120 nM T56556 C3CAG9 145955791 IC50 = 221 nM T56556 CM62WT 145956236 IC50 = 120 nM T56556 CHCB46 145956407 EC50 = 4 nM T56556 C6FS8J 145956778 IC50 = 119 nM T56556 CLD32M 145957548 IC50 = 48.2 nM T56556 C8ZAT2 145957575 IC50 = 44.8 nM T56556 CX32LO 145957840 IC50 = 106 nM T56556 C9F8TW 145957857 EC50 = 48.3 nM T56556 CXH7F4 145957934 IC50 = 820 nM T56556 CB5PZ6 145958054 EC50 = 71.2 nM T56556 CB9CF1 145958160 EC50 = 14 nM T56556 CL15OJ 145958265 EC50 = 10 nM T56556 C9QO8G 145958364 IC50 = 16200 nM T56556 CL76TP 145958566 IC50 = 1190 nM T56556 CDH0A1 145958606 IC50 = 642 nM T56556 CD46YZ 145958660 IC50 = 1640 nM T56556 C0T5ZE 145958944 IC50 = 1620 nM T56556 CBQ8K0 145959274 IC50 = 795 nM T56556 CPU4D2 145959408 IC50 = 33.1 nM T56556 C3ZLR8 145959442 IC50 = 84 nM T56556 C2XSC1 145959549 IC50 = 49.1 nM T56556 C4PQ5A 145959673 IC50 = 811 nM T56556 C3C6SA 145959746 EC50 = 34 nM T56556 CIA08G 145959888 IC50 = 101 nM T56556 CVX17O 145960171 EC50 = 5 nM T56556 CYL21E 145960198 IC50 = 570 nM T56556 C2T8PH 145960322 IC50 = 610 nM T56556 CR0J2I 145960997 IC50 = 57.2 nM T56556 CA7RL9 145962283 IC50 = 5310 nM T56556 CBU79J 145964049 IC50 = 501 nM T56556 C1A7DH 145964067 IC50 = 9930 nM T56556 C5YP9J 145964072 IC50 = 6910 nM T56556 C80ESB 145964513 IC50 = 1060 nM T56556 CM5W0B 145964551 IC50 = 733 nM T56556 CNM1G3 145964790 IC50 = 766 nM T56556 C2QI8W 145965708 IC50 = 90 nM T56556 CJRZ24 145966467 IC50 = 445 nM T56556 C4OZH5 145966511 IC50 = 880 nM T56556 CBL6O0 145966757 IC50 = 7670 nM T56556 C4ZA8I 145966835 IC50 = 1550 nM T56556 CVB80Y 145966874 IC50 = 14390 nM T56556 C58UJF 145968465 IC50 = 15800 nM T56556 CTP6I7 145971735 IC50 = 646 nM T56556 CYU1W6 145971955 EC50 = 11 nM T56556 CZ3N8M 145972213 IC50 = 210 nM T56556 CIT6S0 145972309 IC50 = 18500 nM T56556 C6DKL1 145972800 IC50 = 438 nM T56556 C9QW5V 145973127 IC50 = 59 nM T56556 C96ARL 145973335 IC50 = 3230 nM T56556 C65PUC 145973732 IC50 = 6730 nM T56556 CM1UP7 145973867 IC50 = 430 nM T56556 C14UYO 145974134 IC50 = 287 nM T56556 C8K3YC 145974263 IC50 = 130 nM T56556 C1CKI3 145974543 IC50 = 297 nM T56556 CH30BM 145974617 IC50 = 270 nM T56556 CGWT84 145974788 EC50 = 4 nM T56556 C2O0FG 145974893 IC50 = 351 nM T56556 CLZ4D7 145974899 IC50 = 8760 nM T56556 CQ53WA 145974921 IC50 = 1400 nM T56556 CZ4I8A 145975509 IC50 = 61.6 nM T56556 CAF5H4 145975609 IC50 = 9000 nM T56556 CRO97S 145975756 IC50 = 2830 nM T56556 CM05IS 145975969 IC50 = 176 nM T56556 CA3V5K 145976004 IC50 = 15300 nM T56556 CT4C0Y 145976071 IC50 = 23240 nM T56556 C3PU1W 145976134 IC50 = 77.4 nM T56556 CM0DC2 145976272 IC50 = 2720 nM T56556 CZ9EA3 145976337 IC50 = 4080 nM T56556 C7EP8H 145976472 IC50 = 6650 nM T56556 CV9W1U 145976531 IC50 = 39800 nM T56556 COA43R 145976548 IC50 = 190 nM T56556 C6SV1M 145976742 IC50 = 11400 nM T56556 C6W1PJ 145977012 IC50 = 228 nM T56556 CZP74I 145977357 IC50 = 129 nM T56556 CQ6PN4 145977383 IC50 = 8340 nM T56556 CB7WX4 145977891 IC50 = 102 nM T56556 CK89HF 145978336 IC50 = 2130 nM T56556 C3Q8JT 145978355 IC50 = 1130 nM T56556 C53TFX 145978471 IC50 = 259 nM T56556 C4S5RJ 145978614 IC50 = 287 nM T56556 C3FSQ9 145978662 IC50 = 267 nM T56556 CGY0D8 145978682 IC50 = 2360 nM T56556 CL4WJ5 145978764 IC50 = 565 nM T56556 CF8L7A 145979103 EC50 = 22.3 nM T56556 CM6Z4G 145979318 EC50 = 989 nM T56556 CDYJ89 145979389 IC50 = 5400 nM T56556 C3EX7W 145979504 EC50 = 51.7 nM T56556 C24OSG 145979776 IC50 = 8440 nM T56556 C4G7LT 145980033 EC50 = 38.3 nM T56556 CUSP05 145981621 IC50 = 10900 nM T56556 C26OWY 145981942 EC50 = 19.9 nM T56556 C10YDI 145982128 EC50 = 1170 nM T56556 CZ9N5Q 145982445 IC50 = 6950 nM T56556 C3ZG6V 145982714 IC50 = 6630 nM T56556 C13VFZ 145985646 EC50 = 6.4 nM T56556 CU1Z8M 145986566 EC50 = 1390 nM T56556 C37ULP 145986567 IC50 = 10000 nM T56556 C3KFN7 145987093 EC50 = 448 nM T56556 CFU24J 145987833 EC50 = 3.1 nM T56556 CGL02K 145988126 EC50 = 57 nM T56556 C4F5OW 145988257 IC50 = 20100 nM T56556 CCIF35 145989307 IC50 = 12000 nM T56556 CX3YR7 145990226 EC50 = 34.7 nM T56556 CN1V8K 145992500 EC50 = 7.4 nM T56556 CT02XU 145992768 EC50 = 14 nM T56556 CKZA78 145992770 EC50 = 107 nM T56556 C07OTB 145993028 EC50 = 25.2 nM T56556 C65JUT 145993130 EC50 = 10.9 nM T56556 C8WF7P 145993760 IC50 = 6330 nM T56556 C3UC5J 145994097 EC50 = 59.7 nM T56556 CKM79V 145994277 EC50 = 27.1 nM T56556 CF92IR 155510784 EC50 > 100000 nM T56556 C3MZ1E 155511724 EC50 = 2300 nM T56556 CE4C1X 155512695 IC50 = 1630 nM T56556 CC9X1U 155514114 IC50 = 13100 nM T56556 CVZ7D2 155514151 EC50 = 4600 nM T56556 C0AFT8 155514623 EC50 = 2.4 nM T56556 C17AZU 155515244 EC50 = 5100 nM T56556 CUHI07 155515592 IC50 = 994 nM T56556 CH6O3X 155515825 EC50 = 16000 nM T56556 CV9TF6 155516191 EC50 = 2.2 nM T56556 C75VID 155517095 EC50 = 46 nM T56556 C4IS7E 155518051 EC50 = 4500 nM T56556 CLQO05 155518383 IC50 = 202 nM T56556 CCL04Y 155518581 IC50 = 7400 nM T56556 CCK94U 155519382 IC50 = 2570 nM T56556 CA1BD2 155520579 EC50 = 3700 nM T56556 CE50TP 155521906 IC50 = 7270 nM T56556 C97CDW 155522930 IC50 = 20000 nM T56556 CS18PU 155523410 EC50 = 33500 nM T56556 CN6ST7 155523417 EC50 = 1.1 nM T56556 C1V9YM 155523822 EC50 = 3000 nM T56556 CBZ8K4 155524289 IC50 = 513 nM T56556 C4LK0P 155524329 IC50 = 47.3 nM T56556 C86ZPR 155525910 EC50 = 8100 nM T56556 C8C7VA 155525927 EC50 > 100000 nM T56556 C8TQ4G 155526547 EC50 = 13.5 nM T56556 C7WI3R 155526594 IC50 = 1070 nM T56556 CTW8I2 155526857 EC50 = 3800 nM T56556 C41JTR 155528166 EC50 = 5600 nM T56556 C9BGT5 155528240 EC50 = 55.4 nM T56556 C75OQS 155529248 IC50 = 1900 nM T56556 C56AHP 155530068 EC50 = 3.5 nM T56556 CE0F4W 155530435 IC50 = 3669 nM T56556 C2PW4J 155530538 IC50 = 2025 nM T56556 CQZD59 155530897 IC50 = 3948 nM T56556 C1HFX4 155531129 EC50 = 7200 nM T56556 CUL2G4 155531672 EC50 > 1000 nM T56556 C4IW9M 155533366 EC50 = 41000 nM T56556 C9QT4A 155533532 IC50 = 7.98 nM T56556 CRC20Y 155534149 EC50 = 6400 nM T56556 CP9C0M 155534240 EC50 = 1220 nM T56556 C52RYM 155534490 IC50 = 178 nM T56556 CHF7A6 155535686 EC50 = 84 nM T56556 COFC46 155536723 EC50 = 4700 nM T56556 CP3U4C 155536912 EC50 = 46000 nM T56556 CYG84N 155537154 EC50 = 9500 nM T56556 CB1FI9 155537197 EC50 = 793 nM T56556 C2J7TM 155537461 IC50 = 652 nM T56556 CGD47O 155537584 EC50 = 2.1 nM T56556 C8FX4B 155537647 IC50 = 5650 nM T56556 CVES34 155538494 EC50 = 2300 nM T56556 CS4WO9 155538718 IC50 = 10500 nM T56556 CFN41J 155538958 EC50 = 6200 nM T56556 C8WT1F 155539055 IC50 = 1460 nM T56556 CLU37N 155539307 EC50 = 8100 nM T56556 C9VW3C 155539729 IC50 = 31 nM T56556 C70PUH 155540561 IC50 = 335 nM T56556 CL9G5X 155541828 IC50 > 10000 nM T56556 CE0G9A 155542384 IC50 = 1100 nM T56556 C56DUX 155543049 IC50 > 10000 nM T56556 CP93FH 155543149 EC50 = 6800 nM T56556 CJ5Q2K 155543420 IC50 = 10080 nM T56556 C7JUC3 155543680 EC50 = 3800 nM T56556 CYE3M6 155544628 IC50 = 556 nM T56556 C0GVI7 155545772 EC50 = 1800 nM T56556 CQ3S7A 155545818 IC50 > 10000 nM T56556 CMIN20 155545978 IC50 = 846 nM T56556 CDO86V 155546844 IC50 = 1780 nM T56556 CEA2R7 155547184 IC50 = 2900 nM T56556 COM08I 155547388 IC50 = 1320 nM T56556 CDY82R 155549328 EC50 = 4600 nM T56556 C86HEA 155549333 IC50 = 811 nM T56556 C72IFK 155549366 IC50 = 10400 nM T56556 CDFC58 155549450 IC50 = 1230 nM T56556 C53PGC 155550195 EC50 = 446 nM T56556 CWK3L0 155550287 EC50 = 11000 nM T56556 CB8FC1 155550293 EC50 = 4300 nM T56556 C8F3HQ 155550402 IC50 = 2000 nM T56556 CGF1W0 155551433 IC50 = 1920 nM T56556 CP7A5R 155552128 EC50 = 3900 nM T56556 CIF4T8 155553306 EC50 = 2.8 nM T56556 CG9K4Y 155553476 EC50 > 100000 nM T56556 C5QE9O 155553583 IC50 = 1030 nM T56556 CEZ7B1 155554618 EC50 = 6.5 nM T56556 CX6CM0 155554919 EC50 = 64 nM T56556 C2Y9UG 155554959 EC50 = 2300 nM T56556 C7JI4C 155555932 EC50 = 60 nM T56556 C8M0BP 155556108 IC50 = 989 nM T56556 CDAP41 155557648 IC50 = 202 nM T56556 CG0H8N 155557744 EC50 = 3300 nM T56556 CM2J5L 155558116 EC50 = 6400 nM T56556 C27XQN 155558615 EC50 = 7.2 nM T56556 CUNV65 155558919 EC50 = 17.8 nM T56556 C21LPY 155559292 IC50 = 1260 nM T56556 CG6NC7 155560071 EC50 = 4200 nM T56556 C46KOL 155560381 IC50 = 698 nM T56556 CY6UB5 155561091 IC50 = 112 nM T56556 CS2B6P 155561257 EC50 = 97 nM T56556 C6VUX2 155561896 IC50 = 77.3 nM T56556 CX42YD 155562157 IC50 > 10000 nM T56556 CPOI59 155562875 IC50 = 883 nM T56556 CWM67C 155563340 EC50 = 2500 nM T56556 CS0NC2 155563858 IC50 = 805 nM T56556 CJ57SV 155563869 IC50 > 10000 nM T56556 CU1TG6 155564277 IC50 = 7820 nM T56556 CJ4GX0 155564603 IC50 = 1060 nM T56556 C7SMU4 155565022 IC50 = 1100 nM T56556 C6Z2XK 155566234 EC50 = 4700 nM T56556 CAN76P 155566986 EC50 > 100000 nM T56556 C8ZE6S 155567126 IC50 = 4490 nM T56556 CO1LU7 155567143 EC50 = 30.7 nM T56556 C9QA2H 155567258 IC50 = 4780 nM T56556 CHT79A 155568041 EC50 = 5900 nM T56556 CFCV37 155568122 IC50 = 14800 nM T56556 CTV5K3 155568177 EC50 = 24.5 nM T56556 C03SJY 155568508 EC50 = 2 nM T56556 CO08ZV 155568670 EC50 = 5400 nM T56556 CTXV81 155568869 EC50 = 2.4 nM T56556 COQJ76 155569267 IC50 = 1450 nM T56556 D00RIX 5280443 IC50 = 3100 nM T56556 D01UYI 5281607 IC50 = 1500 nM T56556 D02ZRO 735125 IC50 = 1080 nM T56556 D04GYT 15511439 IC50 = 3981.07 nM T56556 D07RSH 631105 IC50 = 5980 nM T56556 D09HIM 22004473 IC50 = 3890.45 nM T56556 D0A4TF 15511440 IC50 = 5011.87 nM T56556 D0E5IP 3795 EC50 = 189 nM T56556 D0G3TK 5280863 IC50 = 4700 nM T56556 D0I7GE 11790 IC50 = 1310 nM T56556 D0NJ4H 5281670 IC50 = 49000 nM T56556 D0S0RK 10680 IC50 = 17000 nM T56556 D0S8CE 15950351 IC50 = 676.08 nM T75907 C79IRE 71620755 IC50 = 360 nM T75907 C7PI9C 71620756 IC50 = 360 nM T75907 CGD70V 71620759 IC50 = 360 nM T75907 CX85HD 71621073 IC50 = 360 nM T75907 CZB46R 71621227 IC50 = 360 nM T75907 CNP1U5 86574151 IC50 = 360 nM T75907 C2LM9W 127026354 IC50 = 30 nM T75907 CRD02W 127026355 IC50 = 280 nM T75907 C6KE3B 127026667 IC50 = 80 nM T75907 CE2PX6 127026668 IC50 = 30 nM T75907 C7VP6A 127026669 IC50 = 10 nM T75907 C1IF8B 127028921 IC50 = 70 nM T75907 C5ZK6J 127029217 IC50 = 50 nM T75907 CZ3DS8 127029218 IC50 = 40 nM T75907 CMR68I 127029233 IC50 = 1 nM T75907 C7ZHE4 127029234 IC50 = 10 nM T75440 D01XOD 54897 Ki = 0.5 nM T75440 D04BNP 5391 IC50 = 62517269.28 nM T75440 D07JVL 3016 IC50 = 123594743.3 nM T75440 D09LDR 4616 IC50 = 55590425.73 nM T75440 D0CP4E 2802 IC50 = 555904257.3 nM T75440 D0E0OG 3958 IC50 = 285759054.3 nM T75440 D0T5WK 4506 IC50 = 100000000 nM T75440 D0W2NM 3380 IC50 = 263026799.2 nM T75440 D0Z5OV 17925 IC50 = 555904257.3 nM T75440 D0Z9VB 31640 IC50 = 10864256.24 nM T75440 D0G4YZ 11653141 Ki = 2.47 nM T75440 D0M2TS 71600087 IC50 = 800 nM T75440 D01LOJ 11595759 Ki = 6.68 nM T75440 D0FR9I 10430788 Ki = 0.188 nM T75440 D0ZK2Q 9841240 Ki = 2.5 nM T75440 D05UXF 6433109 Ki = 6.4 nM T75440 D08AWI 11430856 Ki > 2000 nM T75440 D0K5IQ 9844410 IC50 = 0.92 nM T75440 D0VN4K 1345 IC50 = 1.1 nM T75440 CCH08A 2997 IC50 = 106414301.8 nM T75440 C87SBM 4540 IC50 = 500034535 nM T75440 CWB1Y9 15024 IC50 = 285759054.3 nM T75440 C2B9SE 16795 IC50 = 76913044.03 nM T75440 CC9L3A 19011 IC50 = 2630267.99 nM T75440 CHL67Q 30401 IC50 = 40831938.63 nM T75440 C7H2PJ 65764 IC50 = 2328091.26 nM T75440 CSTD39 75849 IC50 = 25003453.62 nM T75440 CL25FN 76175 IC50 = 2857590.54 nM T75440 CV8O9T 78641 IC50 = 2588212.92 nM T75440 CB0PY6 92294 IC50 = 15381546.4 nM T75440 CJD8Z6 118749 IC50 = 345143739.3 nM T75440 CYOL58 128744 IC50 = 142889395.9 nM T75440 CH2JA9 148760 IC50 = 10423174.29 nM T75440 CIUV59 188298 IC50 = 13335214.32 nM T75440 C1RK6L 520217 IC50 = 666806769.2 nM T75440 CNA35U 528222 IC50 = 454988060.2 nM T75440 CQ8H2P 622885 IC50 = 1614358.56 nM T75440 C89UHQ 5458184 Ki = 0.242 nM T75440 C01SQJ 6603782 Ki = 0.41 nM T75440 CR5NV7 9975396 IC50 = 181970085.9 nM T75440 C48VJA 10264786 IC50 = 27797132.68 nM T75440 CM8L2J 10358803 IC50 = 277971326.8 nM T75440 C8MT4I 10453776 Ki = 3.9 nM T75440 C3QEM9 10469149 IC50 = 263026799.2 nM T75440 CYX7O2 10738832 Ki = 1.6 nM T75440 CR67IU 10833643 IC50 = 11.8 nM T75440 CFJG64 11059058 IC50 = 1040 nM T75440 CR97ZW 11488150 Ki = 2.68 nM T75440 CR6OL3 11780929 Ki = 30.1 nM T75440 CXLW54 11948707 Ki > 10000 nM T75440 CM1T4V 12790028 IC50 = 142889395.9 nM T75440 C50BWX 13292074 IC50 = 47643098.68 nM T75440 CLH94F 13485706 IC50 = 416869383.5 nM T75440 CKZI28 15294055 IC50 = 620 nM T75440 CZ2IS9 16660294 Ki > 10000 nM T75440 C3W8DT 16749353 IC50 > 5000 nM T75440 CCP1J0 20542073 IC50 = 33342641.28 nM T75440 CDJ23A 23275339 IC50 = 2172701.18 nM T75440 CSB68Q 23275675 IC50 = 195884467.4 nM T75440 CWYX46 23275762 IC50 = 35727283.82 nM T75440 C9S0VL 23275763 IC50 = 625172692.8 nM T75440 CHL6M4 23275854 IC50 = 55590425.73 nM T75440 CTG41H 24778289 IC50 > 2000 nM T75440 C54TYJ 24945827 Ki = 0.882 nM T75440 CL6RD3 25140330 Ki = 0.537 nM T75440 CV4ZB3 25140479 Ki = 0.15 nM T75440 CD5V1U 25140760 Ki = 0.86 nM T75440 CIKB38 25208880 Ki = 0.997 nM T75440 C0RWI9 44366034 IC50 = 23280912.58 nM T75440 CFG7O1 44366036 IC50 = 41686938.35 nM T75440 CF72JC 44366089 IC50 = 25003453.62 nM T75440 CG9YJ7 44366116 IC50 = 135207256.3 nM T75440 CQ19LG 44366138 IC50 = 71449632.61 nM T75440 C1X5TW 44366161 IC50 = 188799134.9 nM T75440 C4LPC1 44366162 IC50 = 20417379.45 nM T75440 C8LT0S 44366169 IC50 = 52601726.64 nM T75440 C24VAZ 44366175 IC50 = 3334264.13 nM T75440 C26GHA 44366179 IC50 = 58884365.54 nM T75440 CR2V5W 44366192 IC50 = 833681184.6 nM T75440 CNAU14 44366206 IC50 = 285759054.3 nM T75440 CL7MP2 44366219 IC50 = 333426412.8 nM T75440 C94OVZ 44366228 IC50 = 188799134.9 nM T75440 CSF51U 44366236 IC50 = 243781081.8 nM T75440 CIP40L 44366255 IC50 = 52601726.64 nM T75440 C5TOJ7 46853447 IC50 = 2000 nM T75440 C8ZCU1 50994211 Ki = 1.57 nM T75440 CMJ62D 53245590 Ki = 2540 nM T75440 C49IKC 56671767 Ki = 1.19 nM T75440 C9D8WH 68968012 IC50 = 1.6 nM T75440 C1U2OK 72793912 Ki = 8 nM T75440 C0ZT5N 90644973 Ki = 293 nM T75440 CWE5X6 90656115 IC50 = 350 nM T75440 CLM5N2 90656116 IC50 = 680 nM T75440 CEAH51 118731302 Ki = 0.87 nM T75440 C5X8MN 122186880 Ki = 2897 nM T75440 C7ODW3 122195524 Ki > 900 nM T75440 CEK04Y 122196423 Ki = 28.13 nM T75440 C7ZKE3 122196424 Ki = 224.46 nM T75440 CVLH25 122196425 Ki = 29.11 nM T75440 C2HUV5 122196426 Ki > 10000 nM T75440 C5L9BD 134143752 Ki = 2100 nM T75440 C71PIY 134144970 Ki = 2200 nM T75440 CGS61F 137553161 Ki = 2930 nM T75440 CD7X5J 145951649 Ki = 28.9 nM T75440 CI4F0U 145954243 Ki = 25.4 nM T75440 CUSI97 145954858 Ki = 54.3 nM T75440 CKA9Z4 145958209 Ki = 70 nM T75440 C9ZY4V 145960315 Ki = 31.5 nM T75440 CPN90L 145971987 Ki = 31.6 nM T75440 CCTO46 155512230 Ki > 10000 nM T75440 CV35ZN 155513505 Ki = 3980 nM T75440 CB65EC 155513663 Ki = 96.1 nM T75440 C23PQH 155514371 Ki = 243 nM T75440 CLD73A 155514689 Ki = 1531.3 nM T75440 CWH24L 155517967 Ki = 562.5 nM T75440 CB0JS3 155518392 Ki > 10000 nM T75440 CH4ZC6 155518977 Ki = 53 nM T75440 C8DNZ6 155519967 Ki = 4737.3 nM T75440 CKH8G2 155522433 Ki > 10000 nM T75440 C36DYH 155525138 IC50 = 2.13 nM T75440 CIW07A 155526405 Ki = 3.2 nM T75440 C2UL4X 155526804 Ki > 10000 nM T75440 C1O0IC 155527848 Ki > 10000 nM T75440 C78XNA 155528306 Ki = 385.3 nM T75440 C2XY8U 155531728 Ki = 184.2 nM T75440 CY0H3U 155533272 Ki = 2020 nM T75440 COT9U8 155535203 Ki = 2380 nM T75440 CTD7J5 155537862 Ki = 462.3 nM T75440 C4C9NY 155541492 Ki > 10000 nM T75440 C1LU5B 155541865 Ki = 200 nM T75440 CMT60C 155543832 Ki = 2890 nM T75440 CJS87Q 155545399 Ki = 3170 nM T75440 C1L0SN 155547768 Ki = 200.7 nM T75440 CJ61KL 155547788 Ki = 369 nM T75440 CRY61B 155548339 Ki = 1696 nM T75440 C6IL4E 155548476 Ki = 50 nM T75440 CGL97X 155555425 Ki > 10000 nM T75440 CDL16X 155555765 Ki = 693.8 nM T75440 CBS89O 155556618 Ki = 2020 nM T75440 CLQH75 155558424 Ki = 208.4 nM T75440 CIPF89 155559210 Ki = 214 nM T75440 CAQ4S5 155561301 Ki > 10000 nM T75440 CCOD50 155562467 Ki = 2220 nM T75440 COP4K5 155562523 Ki > 10000 nM T75440 CI12LD 155566336 Ki > 10000 nM T75440 CU9HA1 155566889 Ki > 10000 nM T75440 C13REG 44471685 Ki = 3166 nM T75440 C6VJE1 6603767 Ki = 4.5 nM T75440 C9TZG6 9842567 Ki = 1.4 nM T75440 D06DTT 193319 IC50 = 71449632.61 nM T75440 D0A0ED 132496 Ki = 3.25 nM T75440 D0FF6S 16038374 IC50 > 2000 nM T75440 D0O6JQ 24839733 Ki = 13.6 nM T94621 D03ZBT 11626560 IC50 > 10000 nM T94621 D01NEC 51042438 IC50 = 1 nM T94621 D01ZAQ 25227436 IC50 = 8 nM T94621 D02ZQS 16095342 IC50 = 1350 nM T94621 D09IYM 24905401 IC50 = 402 nM T94621 D0E3TC 44259 IC50 = 6.5 nM T94621 D0I4TH 24788740 IC50 = 18 nM T94621 D0MS3Z 16725726 Ki = 4 nM T94621 D0W3RW 24964624 IC50 = 12 nM T94621 D03BNU 59604787 IC50 > 10000 nM T94621 D0ZE5U 11161844 IC50 = 5 nM T94621 D0T3ME 156422 IC50 > 30000 nM T94621 COYW98 9222 IC50 > 100000 nM T94621 C3XD4Z 139106 IC50 = 135000 nM T94621 C5EH9L 139601 IC50 = 80000 nM T94621 CU73ST 599501 IC50 = 660000 nM T94621 CFC7G1 756695 IC50 = 41000 nM T94621 C1SVD2 2132479 IC50 = 1900 nM T94621 C9ZT2G 2753118 IC50 = 72000 nM T94621 CFY1D0 2974957 IC50 > 10000 nM T94621 CABJ52 3129049 IC50 = 59000 nM T94621 C98ITU 5327109 IC50 = 260 nM T94621 CWN6P7 5702541 IC50 = 590 nM T94621 CG17TN 6914611 IC50 = 6.8 nM T94621 C7E2QK 6914613 IC50 = 257 nM T94621 CIAL53 9819282 IC50 = 23000 nM T94621 CC7Y2O 9828163 IC50 = 220 nM T94621 C8QZD6 9829528 IC50 = 26 nM T94621 C16VXB 9863538 IC50 > 10000 nM T94621 CI0AW6 9871034 IC50 = 2057 nM T94621 C7H8EO 9871171 IC50 = 7356 nM T94621 C18HKQ 9885748 IC50 = 720 nM T94621 CUE4B5 9912061 IC50 > 50000 nM T94621 CU7FH2 9957031 IC50 > 50000 nM T94621 CJX43Z 10055074 IC50 = 359 nM T94621 CEV18B 10128689 IC50 > 50000 nM T94621 C7PK4U 10152003 IC50 = 15700 nM T94621 C4FUG5 10152760 IC50 = 4517 nM T94621 CMO32F 10152761 IC50 = 325 nM T94621 CMR17F 10174144 IC50 > 50000 nM T94621 CLP79V 10196532 IC50 = 388 nM T94621 CI8MW4 10216627 IC50 = 5 nM T94621 C0O8FI 10217663 IC50 = 1179 nM T94621 CY6MJ3 10218178 Ki = 325 nM T94621 CT97JL 10218280 IC50 = 577 nM T94621 C8V6RI 10240275 IC50 = 212 nM T94621 CD3W6Y 10289038 IC50 > 20000 nM T94621 C2LP9A 10289671 IC50 = 300 nM T94621 CT0M7Q 10311653 IC50 = 259 nM T94621 C4MOF8 10312133 IC50 = 144 nM T94621 CAK9U4 10415819 IC50 = 65 nM T94621 CNY45Z 11151075 IC50 = 10 nM T94621 CO48BE 11165629 IC50 = 14 nM T94621 CO2DA6 11165945 IC50 = 10 nM T94621 C53MZX 11168481 IC50 > 50000 nM T94621 C1GYU5 11175137 IC50 = 18000 nM T94621 C3IJ6D 11180030 IC50 > 50000 nM T94621 CPVK21 11180486 IC50 = 1228 nM T94621 CMA1U5 11196322 IC50 = 510 nM T94621 C7BN5E 11225451 IC50 > 50000 nM T94621 CC6V3Z 11225497 IC50 = 529 nM T94621 C1UZC6 11226082 IC50 = 37720 nM T94621 CKB72H 11237628 IC50 = 8141 nM T94621 CL0QN6 11246027 IC50 = 27 nM T94621 C2ON6C 11246455 IC50 = 118 nM T94621 CCF0G6 11249067 IC50 = 2062 nM T94621 C49NET 11256399 IC50 = 204 nM T94621 C3T6XF 11256709 IC50 = 8 nM T94621 C1TCF3 11260243 IC50 > 50000 nM T94621 COHW29 11272514 IC50 > 50000 nM T94621 C9FG0K 11293497 IC50 = 4 nM T94621 CBOP58 11293798 Ki = 1120 nM T94621 CHBC32 11296432 IC50 = 839 nM T94621 CO39LB 11312547 IC50 = 31000 nM T94621 C1KOA4 11325683 IC50 = 39 nM T94621 CPV82H 11341558 IC50 > 50000 nM T94621 C26BZX 11362471 Ki = 3970 nM T94621 C4G3RZ 11364261 IC50 > 50000 nM T94621 COF6V0 11370369 IC50 = 9 nM T94621 C5EP3S 11373564 IC50 = 11 nM T94621 C1LT9H 11374804 IC50 > 50000 nM T94621 CD2P0L 11383042 IC50 = 5 nM T94621 CWXB93 11397177 Ki > 10000 nM T94621 CPFW90 11399527 IC50 = 556 nM T94621 CRC7H2 11407608 IC50 = 29 nM T94621 C6KQ2U 11409661 IC50 > 50000 nM T94621 C4L5TF 11409804 IC50 = 7356 nM T94621 C4OT0X 11417334 IC50 = 10 nM T94621 CCP18F 11430140 IC50 = 6 nM T94621 C1FC5U 11431759 IC50 > 50000 nM T94621 CW53GT 11440050 IC50 = 57 nM T94621 C5H7KT 11453730 IC50 = 3 nM T94621 CI9L2T 11454186 IC50 > 50000 nM T94621 CQS3U5 11454871 IC50 > 50000 nM T94621 CE72WO 11489421 IC50 = 15390 nM T94621 C7XM4C 11504922 IC50 = 59 nM T94621 CPN02A 11513279 IC50 = 27 nM T94621 C38OKZ 11513374 IC50 = 177 nM T94621 C85JUO 11514232 IC50 = 1600 nM T94621 CJ7XT8 11526364 IC50 = 1909 nM T94621 CTM2Q3 11526695 IC50 = 85 nM T94621 CEX8Y5 11527102 IC50 = 44 nM T94621 C5NPU9 11534762 IC50 = 5127 nM T94621 CCJ7Z1 11535873 IC50 = 830 nM T94621 CTG83F 11539329 Ki > 8400 nM T94621 CG84SZ 11540975 IC50 = 1572 nM T94621 CWCN15 11541348 IC50 = 44 nM T94621 CY0JX9 11541985 IC50 = 21 nM T94621 CSCJ29 11542208 IC50 = 229 nM T94621 C2O3DZ 11543058 IC50 = 880 nM T94621 CA8R0K 11547290 IC50 = 928 nM T94621 CX96EC 11549174 IC50 = 22 nM T94621 C3Z8PI 11549180 IC50 = 31 nM T94621 CJEB45 11549190 IC50 = 2106 nM T94621 CJF21M 11549537 IC50 = 297 nM T94621 CN25UD 11556452 IC50 = 99 nM T94621 CACS26 11561968 Ki > 10000 nM T94621 C3WVM7 11564772 IC50 = 180 nM T94621 C4LI8C 11564882 IC50 = 770 nM T94621 C9LDN1 11577612 IC50 = 107.2 nM T94621 CPJZ24 11584546 IC50 = 696 nM T94621 C0SCK2 11585287 IC50 = 8923 nM T94621 CAP6N0 11588244 IC50 = 8 nM T94621 CMIL86 11590363 Ki > 8400 nM T94621 C6C0VR 11592032 IC50 = 1131 nM T94621 C61KCW 11596252 IC50 = 680 nM T94621 CK61VI 11606572 IC50 = 3706 nM T94621 C20IRX 11606613 IC50 = 1304 nM T94621 C7PA8T 11607451 IC50 = 27 nM T94621 CNA3X5 11608401 IC50 = 6900 nM T94621 C3FQP1 11614515 IC50 = 4 nM T94621 CBEG76 11621110 IC50 = 635 nM T94621 C7P8CI 11622815 IC50 = 9500 nM T94621 CP2R3O 11636277 IC50 = 45 nM T94621 C4YWT2 11636404 IC50 = 6 nM T94621 C9T6SC 11640926 Ki > 8400 nM T94621 C2OC8S 11642946 IC50 = 43 nM T94621 CDY01B 11643074 IC50 = 252 nM T94621 C9RLC8 11643116 IC50 = 77 nM T94621 CP0I2U 11643417 IC50 = 25 nM T94621 CPA5Y7 11650332 IC50 = 184 nM T94621 COR9B8 11650399 IC50 = 16 nM T94621 CBW0A4 11660816 IC50 = 250 nM T94621 C87JQN 11663666 IC50 = 281 nM T94621 C7XEV0 11664023 IC50 = 94.4 nM T94621 CESQ80 11670972 IC50 = 239 nM T94621 C43LDG 11671553 IC50 = 73 nM T94621 CTI6U1 11671757 IC50 = 47 nM T94621 CX1GS0 11672017 IC50 = 16 nM T94621 CON70D 11672049 IC50 = 68 nM T94621 C0V7SU 11675388 IC50 = 2.2 nM T94621 CC5B1E 11681688 IC50 = 16 nM T94621 C0Q7ZW 11688053 IC50 = 400 nM T94621 CU0E8O 11690457 Ki > 10000 nM T94621 C81CLV 11693440 IC50 = 138 nM T94621 C95XBF 11695362 IC50 = 430 nM T94621 CPK2W8 11696113 IC50 = 5 nM T94621 C0NRG1 11703456 IC50 = 8 nM T94621 CB0AP2 11705863 Ki > 10000 nM T94621 CG3RQ4 11708454 IC50 = 290 nM T94621 C3B2HN 11708521 IC50 = 3200 nM T94621 CCK3Q5 11712132 IC50 = 1242 nM T94621 CY8U0T 11713130 IC50 = 90 nM T94621 CM49IK 11715597 IC50 = 920 nM T94621 C0TN5D 11738219 IC50 = 200 nM T94621 CJKC74 11750389 IC50 = 17 nM T94621 C9A6KM 11857236 Ki = 2 nM T94621 CA9ST2 11959186 IC50 = 63 nM T94621 CC7M0D 11959190 IC50 = 50 nM T94621 C39VTW 11959283 IC50 = 63 nM T94621 CQ8U1P 11959284 IC50 = 16 nM T94621 C36HDX 11959286 IC50 = 40 nM T94621 CTE96C 11959310 IC50 = 25 nM T94621 CO0A4K 11959314 Ki = 5 nM T94621 C12CRJ 11959377 IC50 = 200 nM T94621 CUWL12 11959378 IC50 = 25 nM T94621 CVPT94 11959513 IC50 = 316 nM T94621 C5LZ9C 11959550 IC50 = 200 nM T94621 C3UVQ2 11959600 IC50 = 79 nM T94621 C1WDQ0 11959682 IC50 = 20 nM T94621 CMW89V 11959683 IC50 = 20 nM T94621 CA6K4Y 11959684 IC50 = 20 nM T94621 C7RNV1 15602982 IC50 = 280 nM T94621 C3P1ED 15602983 IC50 = 34000 nM T94621 C7N6CQ 15604547 IC50 = 21 nM T94621 CSA02I 15979148 IC50 = 14.6 nM T94621 CBE54Y 15979149 IC50 = 6.7 nM T94621 C9YE7I 15979150 IC50 = 2.8 nM T94621 C92FEN 15979151 IC50 = 10.4 nM T94621 C9QO8U 15979276 IC50 = 10 nM T94621 CFPW41 16007116 Ki > 8400 nM T94621 CZK8V6 16043304 IC50 = 23 nM T94621 C9TU1O 16046126 IC50 > 1000 nM T94621 CKV4G1 16079040 IC50 = 20 nM T94621 CBM80K 16091080 IC50 = 47.7 nM T94621 C7Z4LV 16095343 IC50 = 1950 nM T94621 CHR8G4 16122633 IC50 = 20 nM T94621 C51PSY 16122634 IC50 = 5200 nM T94621 C2RNZ0 16657945 IC50 = 9 nM T94621 C94ONJ 16658020 IC50 = 12000 nM T94621 CSR4V7 16658021 IC50 = 3000 nM T94621 C0O6SY 17751068 IC50 = 8.5 nM T94621 CSK49V 17751069 IC50 = 7 nM T94621 C9C5TV 17751819 IC50 = 6 nM T94621 CWK2H5 21103101 IC50 = 274 nM T94621 CA46OM 21103107 IC50 > 50000 nM T94621 CJXU82 21103111 IC50 = 1877 nM T94621 CF9YE6 21103119 IC50 = 332 nM T94621 C5AR9M 21103197 IC50 = 281 nM T94621 CN1O7X 23647016 IC50 > 50000 nM T94621 CJ3EO0 23647017 IC50 = 1755 nM T94621 CH14KD 23647018 IC50 = 45270 nM T94621 CQ5Z0J 23647019 IC50 = 5407 nM T94621 CT7XW8 23647020 IC50 > 50000 nM T94621 C2JTA3 23647573 IC50 = 5 nM T94621 C83PYS 23647592 IC50 = 9 nM T94621 CI90XG 23647594 IC50 = 21 nM T94621 CWE47K 23647595 IC50 = 45 nM T94621 CICB91 23647596 IC50 = 4 nM T94621 C7W0PE 23647597 IC50 = 4 nM T94621 CTI1F7 23647598 IC50 = 6 nM T94621 CSOG98 23647599 IC50 = 19 nM T94621 CJAI42 23647600 IC50 = 51 nM T94621 CUX75S 23647601 IC50 = 37 nM T94621 CUX5O6 23647602 IC50 = 5 nM T94621 CA4LE6 23647603 IC50 = 8 nM T94621 CGS7Q3 23647604 IC50 = 3 nM T94621 CH89JW 23647605 IC50 = 5 nM T94621 CLDV63 23647606 IC50 = 5 nM T94621 C2BHO1 23658108 IC50 = 25 nM T94621 CL8M1D 23658126 IC50 = 5 nM T94621 CC97WO 23658173 IC50 = 70 nM T94621 CSJ34W 24701731 IC50 = 270 nM T94621 C7YG1N 24759534 IC50 = 23000 nM T94621 C7R9TA 24762195 IC50 = 8 nM T94621 CQNP54 24764449 IC50 = 25000 nM T94621 CW3JR8 24783593 IC50 = 14 nM T94621 C05MQY 24783594 IC50 = 35 nM T94621 C93TIM 24786152 IC50 = 12 nM T94621 CSY9Z6 24788164 IC50 = 11 nM T94621 CFR62V 24788432 IC50 = 12 nM T94621 C2JNI3 24788623 IC50 = 17 nM T94621 CMR7F1 24788739 IC50 = 15 nM T94621 CY1ZS7 24803305 Ki = 3 nM T94621 C2ANO6 24804134 Ki = 8 nM T94621 CSH8A5 24804780 Ki = 6 nM T94621 CUTH13 24805273 IC50 = 125 nM T94621 C0AO5R 24828715 IC50 = 110000 nM T94621 C1H2AM 24828716 IC50 = 246 nM T94621 CU9E4W 24828717 IC50 = 12 nM T94621 C5U2ZM 24828854 IC50 = 3 nM T94621 CQ4G2E 24828855 IC50 = 7 nM T94621 C57SYK 24829098 IC50 = 25 nM T94621 C3YLM1 24829099 IC50 = 71 nM T94621 CM5AX9 24829102 IC50 = 25 nM T94621 CY97JK 24829220 IC50 = 7 nM T94621 CT7QD8 24829222 IC50 = 25 nM T94621 C5WS6R 24894100 IC50 = 48 nM T94621 CV5IE4 24963049 Ki = 1 nM T94621 C9YN2Q 24967131 IC50 > 10000 nM T94621 CLJ2N0 24971386 IC50 = 1299 nM T94621 CC7B8W 24971387 IC50 = 1709 nM T94621 CCWV70 24971388 IC50 = 1381 nM T94621 CSE34D 24971389 IC50 = 1160 nM T94621 C5NFP2 24971390 IC50 = 1514 nM T94621 C0B9HE 24971391 IC50 = 17470 nM T94621 CX1U6V 24971392 IC50 = 1792 nM T94621 C3JT8Q 24971393 IC50 = 494 nM T94621 C0PFZ7 24992842 IC50 = 35 nM T94621 CC61ER 24993160 IC50 = 46 nM T94621 CT81XK 24993161 IC50 = 44 nM T94621 CZK9Q1 24993162 IC50 = 5.5 nM T94621 CK0NZ8 24993163 IC50 = 27 nM T94621 CQ9BF6 24993164 IC50 = 15 nM T94621 C71EOU 24993165 IC50 = 90 nM T94621 C1Y3TF 24993166 IC50 = 20 nM T94621 CA9F3Y 25023714 IC50 = 1000 nM T94621 C8Z4PI 25023715 IC50 = 3980 nM T94621 CV96QX 25023716 IC50 = 2340 nM T94621 C5INV4 25023717 IC50 = 2510 nM T94621 CPOH02 25023718 IC50 = 10000 nM T94621 C6F7RD 25023719 IC50 = 2570 nM T94621 C1JEU6 25023729 IC50 = 9 nM T94621 C14NAT 25023731 IC50 = 20 nM T94621 C81XKW 25023732 IC50 = 4 nM T94621 CFH80B 25023733 IC50 = 13 nM T94621 CR8JP7 25023735 IC50 = 13 nM T94621 C4W7LY 25023736 IC50 = 6 nM T94621 CA6QU5 25023737 IC50 = 5 nM T94621 COV3Q4 25061501 IC50 = 9 nM T94621 C8NR9H 25170562 IC50 = 6 nM T94621 CS9LC3 25170563 IC50 = 22 nM T94621 CN8YZ4 25170991 IC50 = 29 nM T94621 CHN5O0 25190977 IC50 = 19 nM T94621 COWB90 25221040 IC50 = 130 nM T94621 CC25TV 25222706 IC50 = 13 nM T94621 C1IG7E 25243798 IC50 > 10000 nM T94621 CH65JV 25243799 IC50 > 10000 nM T94621 CBQO98 42602095 IC50 = 40 nM T94621 CJ61SE 42602096 IC50 = 23 nM T94621 CI42XG 42602097 IC50 = 30 nM T94621 CD2AH4 42602175 IC50 = 24 nM T94621 CSWA85 42602176 IC50 = 46 nM T94621 C1LUN4 42602178 IC50 = 14 nM T94621 C8O3EA 42602260 IC50 = 22 nM T94621 C93NKL 42602264 IC50 = 15 nM T94621 C59CDG 44389260 IC50 = 157 nM T94621 CEP4T0 44422924 IC50 = 10 nM T94621 C0PEK6 44426856 IC50 = 31 nM T94621 COP8A3 44449880 IC50 = 42 nM T94621 CMC82Z 44449900 IC50 = 1476 nM T94621 C3APO5 44449908 IC50 = 210 nM T94621 CA85HS 44449909 IC50 = 981 nM T94621 C4QJK8 44449942 IC50 = 1600 nM T94621 C0ICB5 44449973 IC50 = 280 nM T94621 CE15WY 44449975 IC50 = 900 nM T94621 CEWB75 44450002 IC50 = 260 nM T94621 CDEJ84 44450004 IC50 = 1075 nM T94621 C8OG1V 44517709 IC50 = 1500 nM T94621 C1EVH2 44560678 IC50 = 827 nM T94621 CI58CZ 44560679 IC50 = 224 nM T94621 CC4Z5M 44560681 IC50 = 165 nM T94621 CWOM65 44560715 IC50 = 40 nM T94621 C7YCO3 44560716 IC50 = 80 nM T94621 C5X7PO 44560717 IC50 = 130 nM T94621 COTH35 44560718 IC50 = 84 nM T94621 C6J0ZC 44560719 IC50 = 180 nM T94621 CL0A2D 44560720 IC50 = 140 nM T94621 CR8K0X 44560724 IC50 = 185 nM T94621 CE08JD 44560725 IC50 = 146 nM T94621 CSX84T 44560726 IC50 = 92 nM T94621 C1O0IG 44560727 IC50 = 43 nM T94621 CB7X4S 44560728 IC50 = 192 nM T94621 C94LIO 44560729 IC50 = 190 nM T94621 C3UQ8C 44560730 IC50 = 116 nM T94621 C8OD4F 44560731 IC50 = 225 nM T94621 CLB20U 44560732 IC50 = 230 nM T94621 CGY1X7 44561054 IC50 = 29 nM T94621 CZK43G 44561055 IC50 = 223 nM T94621 C4WLX8 44561056 IC50 = 421 nM T94621 CXC8I3 44561057 IC50 = 23 nM T94621 CS0QZ4 44561058 IC50 = 539 nM T94621 C1QG9P 44561059 IC50 = 3570 nM T94621 C9MTS4 44561060 IC50 = 59 nM T94621 CZ9L8F 44572052 IC50 = 24.1 nM T94621 CIV48S 44572053 IC50 = 483.3 nM T94621 CFVA91 44572054 IC50 = 55.1 nM T94621 CZE8M9 44572055 IC50 = 77.9 nM T94621 C0DJS1 44591843 Ki = 4 nM T94621 CX52YW 44591844 Ki = 4 nM T94621 C1LS6V 44591845 Ki = 16 nM T94621 CSZ5R9 44592438 IC50 = 500 nM T94621 C6X7FC 44592501 Ki = 40 nM T94621 CTS95L 44592502 Ki = 40 nM T94621 CSKZ16 44592503 IC50 = 8 nM T94621 COY57J 44592504 Ki = 0.63 nM T94621 C3CDV8 44592505 Ki = 2 nM T94621 CJK7L8 45141615 IC50 = 19 nM T94621 CUEX28 45141616 IC50 = 84 nM T94621 C7XZI3 45141617 IC50 > 1000 nM T94621 CZC94D 45141618 IC50 = 35 nM T94621 CY8DC7 45141619 IC50 = 16 nM T94621 C5N4FO 45141620 IC50 = 18 nM T94621 CSB9Q2 45141621 IC50 = 69 nM T94621 C9BXC0 45141812 IC50 = 7 nM T94621 CEU36T 45141813 IC50 = 36 nM T94621 CLED29 45141814 IC50 = 14 nM T94621 CC16ZH 45141815 IC50 = 11 nM T94621 CM57PW 45141816 IC50 = 29 nM T94621 CC3R8E 45141817 IC50 = 210 nM T94621 CQ7OZ9 45142021 IC50 = 4.9 nM T94621 C01CFQ 45142022 IC50 = 5.7 nM T94621 C7FS2V 45142023 IC50 = 11 nM T94621 CYBD69 45142024 IC50 = 8 nM T94621 CR37UP 45142025 IC50 = 4 nM T94621 CU2K8B 45142026 IC50 = 25 nM T94621 CE4D3F 45142255 IC50 = 31 nM T94621 CLCU70 45142256 IC50 = 12 nM T94621 CJQ28R 45142257 IC50 = 52 nM T94621 CJIA74 45142258 IC50 = 12 nM T94621 C1V2YL 45142259 IC50 = 58 nM T94621 CQ5SD4 46190876 IC50 = 39 nM T94621 CY3HW5 46224684 IC50 = 4200 nM T94621 CB5H9C 46225574 IC50 = 31 nM T94621 C8M1DT 46225589 IC50 = 6 nM T94621 C60XUQ 46226079 IC50 = 15 nM T94621 C5PCH8 46226080 IC50 = 15 nM T94621 C6UD1Y 46226095 IC50 = 250 nM T94621 C7IF4T 46226096 IC50 = 63 nM T94621 CUDZ46 46226135 IC50 = 6300 nM T94621 C0P4CT 46226136 IC50 = 12 nM T94621 CPH49S 46226137 IC50 = 7 nM T94621 CM5X8B 46226156 IC50 = 15 nM T94621 C64TVL 46226417 IC50 = 25 nM T94621 CLS29B 46872626 IC50 > 10000 nM T94621 C2O8RZ 46886323 IC50 > 1000 nM T94621 CM8RX4 46886549 Ki = 17 nM T94621 C70BLN 46886550 IC50 = 50 nM T94621 CCV96R 46886665 Ki = 39 nM T94621 CJ2E9Q 46929857 IC50 > 25000 nM T94621 CC1Y0M 52941299 IC50 = 4951 nM T94621 CDT94U 52941495 IC50 = 1485 nM T94621 C9UF6K 52941555 IC50 = 433 nM T94621 CYM80Q 52942489 IC50 = 37826 nM T94621 CS09YT 52942516 IC50 = 5027 nM T94621 CQ08WT 52942668 IC50 = 1288 nM T94621 CHW04J 52943916 IC50 = 630 nM T94621 CY8BV4 52944892 IC50 = 707 nM T94621 CEM95A 52946401 IC50 = 5586 nM T94621 CKE3C7 52946402 IC50 = 1067 nM T94621 C3Q4CU 52947490 IC50 = 8362 nM T94621 CR9E1Z 52947590 IC50 = 26500 nM T94621 CE81HA 52950003 IC50 = 279 nM T94621 C3TU8R 52950063 IC50 = 872 nM T94621 C7MC5G 52950205 IC50 = 4371 nM T94621 C8NA4L 53384644 IC50 > 30000 nM T94621 CO6B0E 54583043 IC50 > 10000 nM T94621 C3PGE2 54585958 IC50 > 10000 nM T94621 CV7HJ8 54585959 IC50 > 10000 nM T94621 CPC5D2 56603995 IC50 = 8 nM T94621 CFP56A 56604013 IC50 = 8 nM T94621 CM8JX1 56604907 IC50 = 25000 nM T94621 CN9QD7 56643097 IC50 > 10000 nM T94621 CT4E8R 56832546 IC50 = 3300 nM T94621 CS7U9L 56965952 IC50 = 18 nM T94621 CQ57PE 57345536 IC50 = 3021 nM T94621 CQP7E0 57750290 IC50 = 31 nM T94621 CNBO65 57750312 IC50 = 36 nM T94621 C2F9DS 57750315 IC50 = 159 nM T94621 CZ08KN 57750321 IC50 = 96 nM T94621 CUY8T6 57750329 IC50 = 709 nM T94621 CK4W1L 57750342 IC50 = 30 nM T94621 CM5X9L 57750343 IC50 = 836 nM T94621 CBY5E4 57750369 IC50 = 42 nM T94621 CSI9Y4 57750382 IC50 = 210 nM T94621 C6GH7X 57750391 IC50 = 190 nM T94621 CL7CW0 57750402 IC50 = 130 nM T94621 CA4G5W 57750407 IC50 = 13 nM T94621 CM7XL6 57750408 IC50 = 20 nM T94621 CY4Z8R 57750418 IC50 = 344 nM T94621 C87LKR 58191080 IC50 = 4 nM T94621 CZPF92 58191081 IC50 = 6 nM T94621 CZA32V 58344912 IC50 = 700 nM T94621 CPVF85 58344916 IC50 = 660 nM T94621 CD3LX9 58344922 IC50 = 15 nM T94621 CS8ZY7 58344924 IC50 = 25 nM T94621 C89NVR 58344941 IC50 = 47 nM T94621 CYK74H 58344983 IC50 = 32 nM T94621 CRJ47B 58345005 IC50 = 16000 nM T94621 CIOV02 58345019 IC50 = 800 nM T94621 CY62SG 58345029 IC50 = 30 nM T94621 CM5HE1 58345070 IC50 = 130 nM T94621 CO18NP 58345151 IC50 = 35 nM T94621 CV61YJ 58345169 IC50 = 51000 nM T94621 CW6SC9 58345215 IC50 = 20000 nM T94621 CFLZ87 58345232 IC50 = 24 nM T94621 CYBT41 58345302 IC50 = 80 nM T94621 C4PE7X 58345314 IC50 = 27 nM T94621 C8X3WB 58458198 IC50 = 4177 nM T94621 C20XPF 58458267 IC50 > 2000 nM T94621 CP85TJ 58458278 IC50 = 6 nM T94621 CT79LH 58458379 IC50 = 356 nM T94621 CXJ63M 59603829 IC50 > 100000 nM T94621 CQEU96 59603842 IC50 = 430 nM T94621 CPVD45 59670809 IC50 = 33 nM T94621 C32WHR 59670989 IC50 = 24 nM T94621 CDWQ04 59671004 IC50 = 31 nM T94621 C43HZT 59671085 IC50 = 249 nM T94621 C0BRA5 59671144 IC50 = 66 nM T94621 CEYW16 59671148 IC50 = 10 nM T94621 C50NWX 59671151 IC50 = 3 nM T94621 CZH4W5 59671179 IC50 = 18 nM T94621 C8FY0G 59671180 IC50 = 17 nM T94621 COH62U 60097413 IC50 > 5000 nM T94621 C1MR8Q 60097495 IC50 > 10000 nM T94621 CC3MB4 60155179 IC50 = 9300 nM T94621 C9QB8G 60155270 IC50 = 1900 nM T94621 CM6NF2 60155627 IC50 = 3500 nM T94621 C62SQG 60155628 IC50 = 24 nM T94621 COS39T 60155629 IC50 = 33 nM T94621 CG6XQ3 67161715 IC50 = 477 nM T94621 CNXU89 67162253 IC50 = 311 nM T94621 CV63UL 67240318 IC50 > 10000 nM T94621 CP8OI2 67304551 IC50 = 5300 nM T94621 CY76UR 67305743 IC50 = 4.5 nM T94621 C3UKG8 67312397 IC50 = 3.2 nM T94621 CM6TZ3 67312506 IC50 = 2.5 nM T94621 C5DGR9 69036886 IC50 = 10000 nM T94621 CS8UF1 70675988 IC50 = 6 nM T94621 C2W5BX 70675991 IC50 = 2005 nM T94621 CUJA60 70676312 IC50 = 6 nM T94621 CRBW21 70676316 IC50 = 30 nM T94621 CGX49K 70676464 IC50 = 5 nM T94621 C1IEJ2 70789254 IC50 = 66000 nM T94621 C8T7ZP 70789255 IC50 = 9500 nM T94621 CKT60L 71455860 Ki > 8000 nM T94621 C9DIK2 71512060 IC50 > 10000 nM T94621 CQV96E 71583048 IC50 = 8111 nM T94621 CSPR52 71583049 IC50 = 16498 nM T94621 CNT5F3 71583050 IC50 = 805 nM T94621 CH7I0W 71583051 IC50 = 8578 nM T94621 CXSI14 71718330 IC50 > 100000 nM T94621 C1TM3P 71720141 IC50 > 100000 nM T94621 CJ2T9E 76332983 IC50 > 10000 nM T94621 C1HW4B 89735655 IC50 = 2500 nM T94621 CQCX41 118737057 IC50 > 10000 nM T94621 C9J4ES 135503073 IC50 = 8 nM T94621 CK94UW 136036657 IC50 = 83 nM T94621 CO16JK 136099766 IC50 = 188 nM T94621 C3ZS9L 136099767 IC50 = 284 nM T94621 CLB4O7 136099768 IC50 = 98 nM T94621 CC73PA 138911338 IC50 = 1.2 nM T94621 CSU93V 155077019 IC50 = 0.54 nM T94621 C2MD1Q 155513187 IC50 > 10000 nM T94621 C86HPW 155518524 IC50 = 21000 nM T94621 CL5DR0 155525783 IC50 < 0.64 nM T94621 CHS21A 155553831 IC50 = 14 nM T94621 CG95WV 155563831 IC50 = 2.8 nM T94621 CEIW13 155566807 IC50 = 79 nM T94621 D00ERW 44444843 Ki = 4800 nM T94621 D00HVA 11624601 Ki > 8400 nM T94621 D05APZ 135398501 IC50 = 210 nM T94621 D09FFE 449241 IC50 = 590 nM T94621 D0I1FJ 11393719 IC50 = 741 nM T94621 D0L2WP 46225540 IC50 = 12 nM T94621 D0OX1T 10172943 IC50 = 30 nM T94621 D0Q3NG 11715520 Ki > 8400 nM T94621 D0R2WK 16038120 Ki > 10000 nM T94621 D0S7IE 11658882 Ki > 8400 nM T94621 D0V6GX 11311693 IC50 = 20 nM T59720 C9G0HL 10533268 Ki = 35 nM T59720 C0QN5G 10606215 Ki = 35 nM T59720 C4IZ1Y 10820377 Ki = 35 nM T59720 CA50FN 56662663 Ki = 35 nM T59720 CH3SW7 56679684 Ki = 35 nM T43031 D0E3TC 44259 IC50 = 18.4 nM T43031 C1SVD2 2132479 IC50 = 3500 nM T43031 C18HKQ 9885748 IC50 = 77000 nM T43031 CACS26 11561968 Ki > 2000 nM T43031 CU0E8O 11690457 Ki > 2000 nM T43031 CKV4G1 16079040 IC50 = 500 nM T43031 CL81VC 21100709 IC50 = 11500 nM T43031 CZ3XP5 46926535 IC50 = 2600 nM T43031 C75GBE 49837568 IC50 = 22500 nM T43031 CEQN27 52936621 Ki > 1000 nM T43031 CT4E8R 56832546 IC50 = 14000 nM T43031 C1MR8Q 60097495 IC50 > 1000 nM T43031 CV63UL 67240318 IC50 = 630 nM T43031 CXSI14 71718330 IC50 = 83000 nM T43031 C1TM3P 71720141 IC50 = 83000 nM T43031 CJ2T9E 76332983 IC50 > 10000 nM T43031 C07EKN 138454794 IC50 > 10000 nM T43031 C0BU2E 145954767 IC50 > 10000 nM T43031 C2MD1Q 155513187 IC50 > 10000 nM T43031 D0K0UJ 49837564 IC50 = 170 nM T55922 D05FFR 5351154 Ki > 1000 nM T55922 CD0Y2A 118705586 Ki = 1070000 nM T55922 CD64YM 118725236 Ki = 1207000 nM T55922 C4ZJU9 239269 IC50 > 180000 nM T55922 CL14FJ 240808 IC50 > 180000 nM T55922 C9BOU0 240809 IC50 > 180000 nM T55922 CD3MU4 388060 IC50 > 180000 nM T55922 CG8Y0J 463012 IC50 > 180000 nM T55922 C1EPW6 476291 IC50 = 1500 nM T55922 CWN21X 608203 IC50 > 180000 nM T55922 CHU71V 2766291 IC50 > 180000 nM T55922 C3KV6A 11742879 Ki = 21200 nM T55922 C7HG1T 15218331 Ki = 20600 nM T55922 C1M3XT 19754189 IC50 > 180000 nM T55922 C05HNS 25181313 IC50 = 400 nM T55922 CQ39IJ 25183746 IC50 = 31000 nM T55922 CV90QL 25231313 IC50 = 3000 nM T55922 CTN16A 25231650 IC50 = 4000 nM T55922 C7NB0S 25231818 IC50 = 170 nM T55922 CIF3B2 25231819 IC50 = 440000 nM T55922 CH84SG 25231821 IC50 = 500000 nM T55922 CDS82O 25232183 IC50 = 49 nM T55922 CP1DT0 25233591 IC50 = 88000 nM T55922 C5BL4R 25233958 IC50 = 157000 nM T55922 C2EMK0 29066960 IC50 > 180000 nM T55922 CHB02E 44564175 IC50 = 7 nM T55922 C1L3WI 44564176 IC50 = 86 nM T55922 CE0JM4 44564196 IC50 = 11 nM T55922 CMWC14 44564197 IC50 = 5 nM T55922 CAID84 44564238 IC50 = 15 nM T55922 CFB5I1 44564239 IC50 = 18 nM T55922 CB7U4V 44564271 IC50 = 7000 nM T55922 CS43LM 44564338 IC50 = 70000 nM T55922 C57HRM 44564339 IC50 = 420000 nM T55922 C9Q3ZV 45097405 IC50 > 180000 nM T55922 C8UP6J 56919646 IC50 > 180000 nM T55922 CNI72Y 56919796 IC50 > 180000 nM T55922 C6A4KE 56919816 IC50 > 180000 nM T55922 C8I4ZA 56919856 IC50 > 180000 nM T55922 COU16Q 56920121 IC50 > 180000 nM T55922 CKLS86 56920454 IC50 > 180000 nM T55922 C8B4NQ 56920865 IC50 > 180000 nM T55922 C4T8JN 56921130 IC50 > 180000 nM T55922 C5CHU3 56921153 IC50 > 180000 nM T55922 CZHJ85 56921749 IC50 > 180000 nM T55922 C4U2XL 56921808 IC50 > 180000 nM T55922 COC17L 56922155 IC50 > 180000 nM T55922 C84CMO 56922551 IC50 > 180000 nM T55922 CUB52I 56923076 IC50 > 180000 nM T55922 CFG3V8 61710896 IC50 > 180000 nM T55922 C0Q8VJ 71460033 Ki = 3800 nM T55922 CA5VM1 80647643 IC50 > 180000 nM T55922 CHF61P 80761654 IC50 > 180000 nM T55922 C5JT8K 80768222 IC50 > 180000 nM T55922 C1B3TQ 80768523 IC50 > 63000 nM T55922 CFB2V6 80768610 IC50 > 180000 nM T55922 CGM4L1 100765007 IC50 > 180000 nM T55922 C8AF7O 104032679 IC50 > 180000 nM T55922 CV6FI3 107371081 IC50 > 180000 nM T55922 CW9RE8 113977178 IC50 > 160000 nM T55922 CIZ98T 114563625 IC50 > 180000 nM T55922 CP68ZQ 118725161 Ki = 21200 nM T55922 CUX9J4 118725180 Ki = 19600 nM T55922 CI9ZG7 118725204 Ki = 7200 nM T55922 CTB96Z 118725211 IC50 = 9000 nM T55922 CG8LY5 118725234 Ki = 18000 nM T55922 CI7C4Q 118725235 Ki = 669000 nM T55922 CZ4AP8 118725238 Ki = 478000 nM T55922 CQI0V5 118725241 Ki = 415000 nM T55922 CX13CP 118725243 Ki = 960000 nM T55922 CL3QZ8 118725244 IC50 = 178600 nM T55922 CAQH86 118725250 IC50 = 204800 nM T55922 CMS1X0 137632229 IC50 > 180000 nM T55922 CA6JL1 137632834 IC50 > 180000 nM T55922 CS1V5F 137632899 IC50 > 180000 nM T55922 CVC92M 137634051 IC50 > 180000 nM T55922 C82GYX 137634161 IC50 > 180000 nM T55922 CX84ME 137634646 IC50 > 180000 nM T55922 CT85ZK 137635286 IC50 > 180000 nM T55922 CGWV42 137635709 IC50 > 180000 nM T55922 C0D3HO 137635782 IC50 > 180000 nM T55922 C9ANK4 137635823 IC50 > 180000 nM T55922 CIKN81 137637985 IC50 > 63000 nM T55922 C8LO3S 137638905 IC50 > 180000 nM T55922 C7IWK8 137639930 IC50 > 180000 nM T55922 C6K3NC 137640514 IC50 > 180000 nM T55922 CD9HO6 137641254 IC50 > 21000 nM T55922 CK4NM7 137642459 IC50 > 180000 nM T55922 CT9Z2B 137642510 IC50 > 180000 nM T55922 CP05EG 137642600 IC50 > 63000 nM T55922 CPL3I7 137642845 IC50 = 44000 nM T55922 CF3W1S 137644197 IC50 > 63000 nM T55922 CO2ZG3 137645098 IC50 > 180000 nM T55922 CZ39RI 137645795 IC50 > 180000 nM T55922 CR2G4T 137646814 IC50 > 63000 nM T55922 C5D8MS 137647022 IC50 > 180000 nM T55922 CYA0M8 137648601 IC50 > 180000 nM T55922 C8J6EA 137648725 IC50 > 180000 nM T55922 C5HQ3N 137648979 IC50 > 21000 nM T55922 C4XUM8 137649315 IC50 > 21000 nM T55922 CNK2S4 137650167 IC50 > 180000 nM T55922 CE8ID4 137650445 IC50 > 180000 nM T55922 C9K4XH 137651053 IC50 > 21000 nM T55922 C75RCW 137651145 IC50 > 7000 nM T55922 C4C9DG 137651239 IC50 > 180000 nM T55922 CD23LP 137651376 IC50 > 63000 nM T55922 C03QHT 137651433 IC50 > 180000 nM T55922 C0TO6G 137651822 IC50 > 180000 nM T55922 CQE98H 137652324 IC50 > 180000 nM T55922 CHM69W 137652349 IC50 > 180000 nM T55922 CE57MT 137652443 IC50 > 180000 nM T55922 C46JEQ 137652753 IC50 > 180000 nM T55922 CFCI38 137652950 IC50 > 180000 nM T55922 C4GMS8 137653057 IC50 > 180000 nM T55922 CPZ58N 137653090 IC50 > 21000 nM T55922 CGK5Y1 137653360 IC50 > 180000 nM T55922 CSQF12 137653636 IC50 > 180000 nM T55922 CP8TJ0 137654766 IC50 > 21000 nM T55922 C75NWC 137655212 IC50 > 180000 nM T55922 CR6N5Y 137656925 IC50 > 21000 nM T55922 C9PJD2 137657088 IC50 > 180000 nM T55922 C5Q0YO 137657983 IC50 > 180000 nM T55922 CJ4M7L 137658244 IC50 > 180000 nM T55922 C3RO8E 137659106 IC50 > 180000 nM T55922 C6BN1M 137659420 IC50 > 63000 nM T55922 CBXA79 137659429 IC50 > 63000 nM T55922 CYD2N8 137659438 IC50 > 180000 nM T55922 C71FOJ 137660126 IC50 > 180000 nM T55922 C89UTS 137660314 IC50 > 63000 nM T55922 CPZ9E8 137660942 IC50 > 180000 nM T55922 CD1Y9L 137660985 IC50 > 180000 nM T55922 C4QM7T 137662328 IC50 > 180000 nM T55922 D03OLX 25231309 IC50 = 9000 nM T55922 D0I7IA 25231315 IC50 = 5000 nM T55922 D0P5YR 446204 IC50 = 55 nM T55922 D0YM6B 25231308 IC50 = 600 nM T58130 CN8XM2 5311263 EC50 = 8.1 nM T58130 CLS96Y 6419701 EC50 = 83.18 nM T58130 COZF72 10322404 EC50 = 2.692 nM T58130 C7QRT8 11648176 EC50 = 3.8 nM T58130 CV86RF 44368508 EC50 = 4.898 nM T58130 C85ANH 46213949 IC50 > 8000 nM T58130 CET63X 46223906 EC50 = 3.3 nM T58130 C57TYK 71569053 EC50 = 3.8 nM T58130 CSN3I7 71569056 EC50 = 2.4 nM T58130 CPT5S2 71718248 EC50 = 4.467 nM T58130 CKC4U7 71719457 EC50 = 4.898 nM T58130 C5P1CQ 71720690 EC50 = 3.467 nM T58130 CG65XZ 122191108 Ki = 170 nM T58130 CWQ8Y3 122191544 IC50 = 266 nM T58130 D05TVG 23682233 Ki = 170 nM T58130 D0X0UR 5497152 EC50 = 570 nM T17345 D01KKQ 135400182 IC50 = 21000 nM T17345 D0AO5H 5578 Ki = 0.006 nM T17345 D0C0SK 4993 Ki = 8 nM T17345 D0H0KB 5070 IC50 = 312000 nM T17345 D0M4VM 5320 IC50 = 18000 nM T17345 D0SV8E 126941 Ki = 0.00034 nM T17345 D0Y4GO 135410875 Ki = 7 nM T17345 D0Y7TS 5583 IC50 < 1 nM T17345 D04LBC 213043 IC50 = 8 nM T17345 D09AYQ 54369 Ki = 0.025 nM T17345 D05HCO 177894 Ki = 0.0003 nM T17345 D05AHQ 68916 Ki = 58.88 nM T17345 D06YIB 135436405 IC50 > 100000 nM T17345 D0D2RN 169371 Ki = 0.0018 nM T17345 D0FC5T 21453 IC50 = 530 nM T17345 D0N3XT 57030 IC50 = 1.8 nM T17345 CND0P2 1881 Ki = 4.5 nM T17345 C7OTP8 3439 IC50 = 220 nM T17345 CU2C4N 3534 IC50 = 70000 nM T17345 C8Y3OG 3537 IC50 = 2000 nM T17345 CEJF30 19931 Ki = 1659.59 nM T17345 C1F2TO 25889 Ki = 110 nM T17345 CY85FK 38778 Ki = 77.62 nM T17345 CRV0E5 72468 IC50 = 1000 nM T17345 CZ8JM5 72509 IC50 = 2.7 nM T17345 C87TYO 72934 IC50 = 15 nM T17345 C7SXL6 87152 IC50 = 1040000 nM T17345 CJ19OK 101067 Ki = 9.6 nM T17345 C8OGL7 102185 IC50 = 9400 nM T17345 C1Q8JR 121750 Ki = 7.7 nM T17345 C4HSB8 125843 IC50 = 1.35 nM T17345 CZA4M3 158351 IC50 = 220 nM T17345 CRQ24H 160203 Ki = 22.39 nM T17345 CZM82G 269322 IC50 = 3.9 nM T17345 C82AVZ 275733 IC50 = 3.8 nM T17345 C5JO7S 316019 IC50 = 3000 nM T17345 C3BRV9 317332 IC50 = 2700 nM T17345 CV20SE 324351 IC50 = 4.1 nM T17345 CPI45H 324352 IC50 = 8.6 nM T17345 CWV02U 324357 IC50 = 5.8 nM T17345 CY8C9L 329597 IC50 = 25000 nM T17345 C9GDJ6 353015 Ki = 0.00089 nM T17345 C3QH5B 354441 Ki = 218.78 nM T17345 CE7IH3 354768 IC50 = 19 nM T17345 CHA7L8 360682 Ki = 0.00035 nM T17345 CT64FM 375312 IC50 = 5.8 nM T17345 CC3ZE0 381233 IC50 = 11.6 nM T17345 C7VFS0 381234 IC50 = 11.4 nM T17345 C3F5KM 382165 IC50 = 8.7 nM T17345 CT51LK 393599 Ki = 0.0004 nM T17345 C8WO4J 403898 Ki = 42000 nM T17345 CTO2D8 404585 Ki = 100 nM T17345 C2IZ4Q 405137 Ki = 1800 nM T17345 C0MKV6 405140 Ki = 600 nM T17345 CDC2L4 406510 Ki = 4000 nM T17345 C25WDV 406511 Ki = 4000 nM T17345 C58ZQB 406512 Ki = 3000 nM T17345 CU4O0N 407233 Ki = 93.33 nM T17345 CD27CT 407235 Ki = 70 nM T17345 C5E7QX 429008 IC50 = 740 nM T17345 C6P2YK 444617 IC50 = 8500 nM T17345 CS9OU4 447021 IC50 = 26 nM T17345 CTXS72 447022 IC50 = 2900 nM T17345 C65ECP 448780 Ki = 5200 nM T17345 CT4N6R 456183 Ki = 6 nM T17345 CYC5M0 456204 IC50 = 4.7 nM T17345 CU1IP4 456205 IC50 < 100 nM T17345 C5VDE1 456216 IC50 = 3900 nM T17345 C1GU8M 456245 IC50 = 820 nM T17345 CD83KY 456272 IC50 = 440 nM T17345 CA6RC1 456306 IC50 = 2700 nM T17345 CQ61JH 456893 IC50 = 5 nM T17345 CEQ98S 456897 IC50 = 18200 nM T17345 CI10YF 457336 IC50 = 150 nM T17345 CHUR38 457342 IC50 = 5.5 nM T17345 CB2ZR6 457343 IC50 = 300 nM T17345 CBD80Z 457349 IC50 = 2300 nM T17345 CX4L1I 457350 IC50 = 1000 nM T17345 C7SZQ6 457353 IC50 = 142 nM T17345 C23EKX 457354 IC50 = 5.1 nM T17345 CBDY12 457370 IC50 = 2600 nM T17345 C81HJP 457371 IC50 = 31000 nM T17345 C53LNC 457372 IC50 = 750 nM T17345 CSWJ43 457373 IC50 = 730 nM T17345 CI17EV 457374 IC50 > 10000 nM T17345 C38SDU 457375 IC50 > 10000 nM T17345 CQY5L9 457376 IC50 > 10000 nM T17345 CMI8V4 457377 IC50 > 10000 nM T17345 CM5JA3 459880 IC50 = 370 nM T17345 CFQ2A9 459881 IC50 = 1000 nM T17345 CW1Q3Y 459887 IC50 = 710 nM T17345 C9YRU0 460024 IC50 = 57 nM T17345 CT9FW6 461920 Ki = 10.2 nM T17345 C03TKX 462111 IC50 = 17 nM T17345 CM4T5X 462117 IC50 = 10 nM T17345 C97EVZ 462118 IC50 = 28000 nM T17345 CHI3D7 462119 IC50 = 28000 nM T17345 C08HAR 462121 IC50 = 26000 nM T17345 C4SOE5 462122 IC50 = 27000 nM T17345 CUO54Z 462123 IC50 = 11 nM T17345 CS04OY 462124 IC50 = 25000 nM T17345 C7DI1F 462125 IC50 = 140 nM T17345 C8WYK9 462127 IC50 = 1400 nM T17345 C6NS9C 462129 IC50 = 50 nM T17345 C4AI1C 462134 IC50 = 3.6 nM T17345 C0EH1R 462466 Ki = 42.66 nM T17345 C8YC0H 462467 Ki = 134.9 nM T17345 CAHX06 462469 Ki = 302 nM T17345 CINY32 462582 IC50 = 2400 nM T17345 C8F9IM 462583 IC50 = 3900 nM T17345 C8QJT5 462584 IC50 = 550 nM T17345 CC65NE 462585 IC50 > 10000 nM T17345 CO46NQ 462587 IC50 = 4300 nM T17345 C62CHU 462589 IC50 = 2100 nM T17345 CTO26P 462590 IC50 = 3100 nM T17345 CQ4DV2 462591 IC50 = 2000 nM T17345 CJ4H0N 462592 IC50 = 2600 nM T17345 C0W2ZP 462593 IC50 = 24000 nM T17345 CBM4S2 462594 IC50 = 33000 nM T17345 C5Z4WX 462595 IC50 = 320 nM T17345 CO05RB 462596 IC50 = 180 nM T17345 C7XI6R 462597 IC50 = 3500 nM T17345 CV80TA 462598 IC50 = 4100 nM T17345 CS1AR6 462599 IC50 = 4400 nM T17345 C74WHR 462600 IC50 = 1300 nM T17345 C3HUT1 462601 IC50 = 400 nM T17345 CEW0T1 462602 IC50 = 270 nM T17345 C52FZM 462603 IC50 = 92 nM T17345 C8PC9F 462604 IC50 = 4300 nM T17345 C7ZJP3 462605 IC50 = 9100 nM T17345 CXW5K6 462606 IC50 = 820 nM T17345 C59MPI 462607 IC50 = 30 nM T17345 CK60HY 463731 IC50 = 990 nM T17345 CO3N7T 463890 IC50 = 12 nM T17345 CVK3W9 463891 IC50 = 7.1 nM T17345 CV4Q2D 463908 IC50 = 1200 nM T17345 C0XBM2 464022 IC50 = 590 nM T17345 C9PX5G 464023 IC50 = 500 nM T17345 C87RIT 464024 IC50 = 850 nM T17345 CMN7V4 464028 IC50 = 6100 nM T17345 CLC49E 464033 IC50 = 440 nM T17345 C6Z1YM 464034 IC50 = 420 nM T17345 C4H1FO 464035 IC50 = 36 nM T17345 CC80XF 464040 IC50 = 10 nM T17345 CRF85I 464992 IC50 = 27 nM T17345 CX8Y6N 464994 IC50 = 670 nM T17345 CCD18G 466230 IC50 = 6.7 nM T17345 CIR4Z5 466231 IC50 = 2500 nM T17345 CZI41B 467890 Ki = 87 nM T17345 CQB5F2 467891 Ki = 29 nM T17345 C0HG3Q 467892 Ki = 10 nM T17345 C7EJH4 467893 Ki < 2 nM T17345 CL91XC 467894 Ki = 10 nM T17345 CI8A9R 467895 Ki = 6.4 nM T17345 CT9M6G 467896 Ki < 2 nM T17345 C68DYK 467897 Ki = 24 nM T17345 CS8GB6 467898 Ki = 0.1 nM T17345 C3VY2Z 467899 Ki = 0.4 nM T17345 C4WIB5 467900 Ki = 0.1 nM T17345 CI81OG 467901 Ki = 0.2 nM T17345 CL8X1M 467902 Ki = 0.2 nM T17345 CSMT16 467903 Ki = 30 nM T17345 C45HLJ 467904 Ki = 0.4 nM T17345 CRUW28 467905 Ki = 0.1 nM T17345 CF1M8Q 468708 IC50 = 450 nM T17345 CSO8F0 468709 IC50 > 26000 nM T17345 CRP1D3 468710 IC50 > 25000 nM T17345 CQM7K4 468711 IC50 > 15000 nM T17345 CT6B0K 468712 IC50 > 15000 nM T17345 C92GMA 470175 IC50 = 6.1 nM T17345 CS6A3D 470176 IC50 = 2.8 nM T17345 C41BHZ 470177 IC50 = 5.2 nM T17345 C1BU8E 470179 IC50 = 6.7 nM T17345 CA3U5C 470200 IC50 = 3.7 nM T17345 C1Y2GQ 470201 IC50 = 5.9 nM T17345 C4D2QK 470202 IC50 = 6.1 nM T17345 C0V5MT 470264 IC50 = 120 nM T17345 CLY84S 470265 IC50 = 8 nM T17345 CMT51S 470266 IC50 = 44 nM T17345 C76HNV 470281 IC50 = 69 nM T17345 CQA07O 470284 IC50 = 250 nM T17345 CWV91M 470285 IC50 = 19 nM T17345 C25WGL 470286 IC50 = 4.6 nM T17345 CX5KM2 470287 IC50 = 3.2 nM T17345 CPC2W8 470288 IC50 = 4.1 nM T17345 CGI39U 470317 IC50 = 4 nM T17345 CI81MK 470318 IC50 = 850 nM T17345 C3O4TZ 470332 IC50 = 5300 nM T17345 CMJ5I4 470333 IC50 = 1900 nM T17345 CLM7A5 472826 IC50 = 3400 nM T17345 C0IJ7Q 472845 IC50 = 3.8 nM T17345 CM6FH7 472846 IC50 = 6.2 nM T17345 CQGS78 472847 IC50 = 2 nM T17345 C8NJU3 472848 IC50 = 68 nM T17345 CNBY98 472849 IC50 = 14 nM T17345 CIHZ91 472850 IC50 = 33 nM T17345 C9H4YB 472852 IC50 = 277 nM T17345 C7VGW9 472853 IC50 = 20 nM T17345 CVFX53 472910 Ki = 24.4 nM T17345 CERP02 474750 IC50 = 15 nM T17345 C0SG1N 476032 IC50 = 2459 nM T17345 C1Z6AQ 476042 IC50 = 1526 nM T17345 CY37PZ 476043 IC50 = 942 nM T17345 C74WGU 477890 IC50 = 7300 nM T17345 C3JY5Z 479281 IC50 = 700 nM T17345 CM2GT8 479412 IC50 = 76000 nM T17345 CF3C8Q 479413 IC50 = 13000 nM T17345 C41TQB 479416 IC50 = 530 nM T17345 C59FRQ 479418 IC50 = 160000 nM T17345 CF2JD3 479421 IC50 = 6200 nM T17345 CRB65P 481401 IC50 > 19000 nM T17345 COV85S 482165 IC50 = 1300 nM T17345 C9KOB8 485848 IC50 = 0.0021 nM T17345 C3JX2W 490573 IC50 = 5000 nM T17345 C25VUD 490663 Ki = 96.3 nM T17345 CI74ZT 490664 Ki = 4.3 nM T17345 CEW3B0 490665 Ki = 33 nM T17345 C89KLU 490666 Ki = 310 nM T17345 C7LX8H 490667 Ki = 250 nM T17345 CR1SM3 490668 Ki = 49 nM T17345 CLTA76 504022 IC50 = 5000 nM T17345 CN5CJ7 688803 IC50 = 50000 nM T17345 CQ5E7D 789778 Ki = 9.8 nM T17345 C9JQC0 2437106 IC50 = 500 nM T17345 C7RW2A 2731323 Ki = 130 nM T17345 C67UFD 2737412 IC50 = 580 nM T17345 C5F6EO 3010592 IC50 = 6.8 nM T17345 CG6F5S 3132813 Ki = 6.4 nM T17345 C2IFO1 3145500 IC50 = 1900 nM T17345 CFRL82 5183677 IC50 = 830 nM T17345 CHGZ97 5288461 IC50 = 800 nM T17345 CQ1ZH4 5742617 IC50 = 1216 nM T17345 CQ75AN 5742620 IC50 = 624 nM T17345 CT79NS 5742621 IC50 = 1410 nM T17345 CM59DP 5742624 IC50 = 970 nM T17345 C2N0IR 6477203 Ki = 1600 nM T17345 CYP69H 6482470 IC50 = 10000 nM T17345 CXI43R 9805576 IC50 = 1530 nM T17345 CYZ79K 9846618 IC50 = 8.8 nM T17345 CVWX01 9881905 Ki = 15000 nM T17345 CC36EP 9889551 IC50 = 10000 nM T17345 CP75AV 9898639 IC50 = 18000 nM T17345 C5VZN4 9911146 IC50 = 420 nM T17345 C3GI6F 9931657 Ki = 0.005 nM T17345 CL0P6O 9932276 IC50 = 1000 nM T17345 CIDQ05 9952879 Ki = 0.12 nM T17345 CBQK30 9973530 Ki = 4.2 nM T17345 CG9ZU8 9976735 IC50 > 26000 nM T17345 C2C7WX 9980556 Ki = 0.54 nM T17345 C3FR4N 10004772 IC50 = 125 nM T17345 C7RD2X 10007840 Ki = 0.183 nM T17345 C9A1VX 10019413 Ki = 24 nM T17345 CID95L 10030947 Ki = 0.000014 nM T17345 CN4V0B 10053803 Ki = 0.00041 nM T17345 C04LWZ 10060600 Ki = 1.6 nM T17345 CQI0P1 10060703 IC50 = 20 nM T17345 C37ZPO 10065177 Ki = 977.24 nM T17345 C5THD4 10070986 IC50 = 16 nM T17345 C70FRM 10072852 IC50 = 66 nM T17345 CQ8U6T 10090457 Ki > 5000 nM T17345 CSJY78 10246793 Ki = 36 nM T17345 C8ME5O 10260430 IC50 = 2.5 ug.mL-1 T17345 CGT0H9 10326322 Ki = 0.00011 nM T17345 CKFP04 10403719 Ki = 140 nM T17345 C7KXJ2 10404647 IC50 = 560 nM T17345 C9PRM3 10405166 IC50 = 2.8 nM T17345 CTX6H7 10433577 IC50 = 210 nM T17345 CZD4B0 10456691 IC50 = 21000 nM T17345 CB15AR 10457642 IC50 = 1.3 nM T17345 CHM3X4 10478775 Ki = 3400 nM T17345 CPO4W7 10518330 Ki = 9.8 nM T17345 C12BJE 10522269 Ki = 52 nM T17345 CZ8YM9 10544281 Ki = 75 nM T17345 CM95NE 10565157 Ki = 7.1 nM T17345 CLK5H2 10590469 IC50 = 3185 nM T17345 CG83DM 10608757 Ki = 750 nM T17345 C9WCK2 10634047 Ki = 8.6 nM T17345 CI5SU7 10658874 Ki = 10.5 nM T17345 CBXD51 10682649 Ki = 8.8 nM T17345 CXZL07 10709354 Ki = 13 nM T17345 C41ICW 10719122 IC50 = 3100 nM T17345 C0B7YU 10805231 Ki = 131 nM T17345 CHK35G 10807265 Ki = 19 nM T17345 CMF9L1 10826074 Ki = 3.6 nM T17345 C7XFJ5 10828475 Ki = 11 nM T17345 C3R0FI 10860015 IC50 = 10 nM T17345 C0S6TG 10883066 IC50 = 22000 nM T17345 CYWT73 10884015 IC50 = 100000 nM T17345 C9HR0M 10902858 IC50 = 32000 nM T17345 C8B0FL 10961831 IC50 = 5400 nM T17345 C4ZML2 10981577 IC50 = 85 nM T17345 C9D4VK 10991113 IC50 = 44 nM T17345 C9LPA1 10993870 IC50 = 920 nM T17345 CCQ4P6 11003295 IC50 = 2 nM T17345 C2P3AT 11047021 IC50 = 1300 nM T17345 CZ90JL 11058970 IC50 = 450 nM T17345 C4RBD9 11078421 IC50 = 21 nM T17345 CP5YV0 11099765 IC50 = 27000 nM T17345 CY1A7Q 11102571 IC50 = 7 nM T17345 C9ZWB1 11154001 IC50 > 10000 nM T17345 CO2DY5 11247965 Ki = 0.034 nM T17345 C8Q6ZT 11248313 Ki = 2.1 nM T17345 CIG85H 11282247 IC50 = 300 nM T17345 CI2TD8 11340329 IC50 > 10000 nM T17345 C85DMO 11349789 IC50 = 28000 nM T17345 C4EL7T 11430583 IC50 > 10000 nM T17345 CH8IF2 11442040 IC50 > 10000 nM T17345 C41XHB 11452801 IC50 > 10000 nM T17345 CJS58R 11455251 IC50 > 10000 nM T17345 C03JKV 11478803 Ki = 0.0001 nM T17345 C3ROC9 11538533 IC50 < 10 nM T17345 C6K9EH 11573029 IC50 = 630 nM T17345 C1XJI4 11645134 IC50 = 10700 nM T17345 C71ZQD 11645349 IC50 = 34 nM T17345 CYL01H 11651834 IC50 = 9400 nM T17345 CRUQ79 11673839 IC50 = 98000 nM T17345 C8AEX7 11687971 Ki = 500 nM T17345 C19BQV 11688044 IC50 = 8400 nM T17345 CQ4H5E 11744008 IC50 = 9000 nM T17345 CE7DH6 11783065 IC50 = 30000 nM T17345 CTB69W 11822511 IC50 = 47 nM T17345 CR9GN2 11826533 IC50 = 22000 nM T17345 CWP0B9 11846624 IC50 = 1830 nM T17345 CCUF60 11846625 IC50 = 2300 nM T17345 CW5VO2 12214236 Ki = 56000 nM T17345 CU1CF0 12242319 IC50 = 377000 nM T17345 CML17O 12242320 IC50 = 242000 nM T17345 CZO4H8 12242322 IC50 = 57000 nM T17345 C9AQ3V 12242324 IC50 = 740000 nM T17345 C13ZHJ 12517699 IC50 = 28000 nM T17345 CRSM76 12517700 IC50 = 7000 nM T17345 CSN4H6 12517701 IC50 = 8000 nM T17345 CMT96B 12517702 IC50 = 11000 nM T17345 C32RLQ 12517703 IC50 = 903000 nM T17345 C3G8JV 12517705 IC50 = 168000 nM T17345 CYPT41 12655201 IC50 = 370 nM T17345 CI0Y1T 12655204 IC50 = 58 nM T17345 CUXC87 12803287 IC50 = 340000 nM T17345 C98JXK 13112734 IC50 = 120 nM T17345 CX3Q6D 13112736 IC50 = 49 nM T17345 C8EIC5 13112740 IC50 = 29 nM T17345 C1INA2 13112752 IC50 = 310 nM T17345 C5X3WZ 13112757 IC50 = 44 nM T17345 C84HXC 13170795 IC50 = 14000 nM T17345 CU4O5B 13739857 IC50 = 61 nM T17345 CZLB08 13877973 IC50 = 230 nM T17345 CU8A4L 13877981 IC50 = 1110 nM T17345 CZV23T 13953684 IC50 = 67 nM T17345 CIW97R 13953685 IC50 = 93 nM T17345 CQFS01 13953687 IC50 = 110 nM T17345 C49DCF 13953688 IC50 = 170 nM T17345 C47HUP 13953689 IC50 = 20 nM T17345 C25SRU 13989362 IC50 = 5.3 nM T17345 CHI71Y 13989363 IC50 = 5.4 nM T17345 CRN23J 14083105 IC50 = 72 nM T17345 CS1G8K 14503206 IC50 = 40 nM T17345 CD84TM 14503207 IC50 = 70 nM T17345 CZET95 14560097 IC50 = 3 nM T17345 CAM5O1 14570150 Ki = 0.8 nM T17345 C8XLI9 14570153 IC50 = 66 nM T17345 CM49FY 14570156 IC50 = 110 nM T17345 C46HSO 14570159 IC50 = 14 nM T17345 CEL4B9 14570163 IC50 = 46 nM T17345 C6N4JB 14570319 IC50 = 300 nM T17345 C20TUW 14570320 IC50 = 630 nM T17345 CFQ37R 14570325 IC50 = 1800 nM T17345 CK5JI7 14570338 IC50 = 540 nM T17345 C3B7AQ 14570339 IC50 = 140 nM T17345 C9W4IP 14776576 IC50 = 6.4 nM T17345 C9V3SY 14776579 IC50 = 88 nM T17345 CX4U2T 14776583 IC50 = 57 nM T17345 CU1M4X 14776589 IC50 = 5.3 nM T17345 CWDB20 14776590 IC50 = 5.9 nM T17345 C9EW5Z 14776615 IC50 = 6000 nM T17345 CA4HC9 14776619 IC50 > 20000 nM T17345 CW5C6T 14801655 IC50 = 32 nM T17345 CBKR63 14801660 IC50 = 35 nM T17345 C68YXF 14801666 IC50 = 30 nM T17345 C4UVQ0 14840934 IC50 = 27000 nM T17345 CL5H0X 14840943 IC50 = 35 nM T17345 CORH59 14840958 IC50 = 50 nM T17345 C7VK0C 15021215 IC50 = 1.34 nM T17345 C4D8IR 15523786 Ki = 14.1 nM T17345 CW1QA4 15523787 Ki = 0.107 nM T17345 C6QM7Z 15616236 IC50 = 19000 nM T17345 C8W1DB 15616238 IC50 > 50000 nM T17345 CQ1TU0 16038397 Ki = 9.6 nM T17345 CWKX69 16086910 Ki = 110000 nM T17345 C6V7GN 16086911 Ki = 35000 nM T17345 C3X9DE 16086912 Ki = 3900 nM T17345 C9KZ4H 16086913 Ki = 33000 nM T17345 CTK25X 16086914 Ki = 69000 nM T17345 C7MA5T 16086915 Ki = 13000 nM T17345 CD59VR 16086916 Ki = 35000 nM T17345 C6UX1P 16086917 Ki = 109000 nM T17345 CRWB95 16086918 Ki = 13000 nM T17345 C0RE7Z 16086919 Ki = 12000 nM T17345 C1BYA7 16110323 IC50 = 1460 nM T17345 C4XBM2 16110326 IC50 = 1380 nM T17345 CB36UF 16110328 IC50 = 5710 nM T17345 CS9FR8 16110329 IC50 = 1160 nM T17345 C31SJW 16110337 IC50 = 400 nM T17345 CJ73WY 16110338 IC50 = 1460 nM T17345 C3LHA7 16110339 IC50 = 14300 nM T17345 C8OYD1 16110341 IC50 = 1220 nM T17345 C81MTW 16110344 IC50 = 1380 nM T17345 CZJM43 16732891 IC50 = 2900 nM T17345 CGM38B 16732892 IC50 = 6000 nM T17345 CMC21Z 16732893 IC50 = 5800 nM T17345 C9IG0J 16733029 IC50 = 2700 nM T17345 CHL6F9 16733030 IC50 > 31000 nM T17345 C8X9EC 16733031 IC50 > 31000 nM T17345 CW5SB7 16733033 IC50 > 28000 nM T17345 CM80YI 16733034 IC50 = 5800 nM T17345 CM1I4D 16733035 IC50 > 32000 nM T17345 CP8VS3 16733036 IC50 = 1400 nM T17345 C83VHB 16733162 IC50 = 1400 nM T17345 CED2R5 16733163 IC50 = 2900 nM T17345 CDA8P5 16733164 IC50 = 18000 nM T17345 CXA71B 16733165 IC50 = 32000 nM T17345 CC09RL 19089924 IC50 = 430 nM T17345 CK1P0V 21496446 IC50 = 140 nM T17345 C7B8CR 21705470 IC50 = 83300 nM T17345 C27WPQ 23161237 IC50 = 1100 nM T17345 CE2XM5 23629645 Ki = 800 nM T17345 CT2G9I 23647976 IC50 = 2100 nM T17345 CUSF67 23648073 Ki = 94000 nM T17345 CI2F9K 23648074 Ki = 28000 nM T17345 C4SXQ7 23648075 Ki = 15000 nM T17345 CDUX91 23648076 Ki = 9500 nM T17345 CE4G3V 23729147 IC50 > 125000 nM T17345 C7TLP1 24202945 Ki = 2000 nM T17345 C4S9RX 24202946 Ki = 8000 nM T17345 C6H1RM 24202947 Ki = 8000 nM T17345 C7AXQ6 24203165 Ki = 6000 nM T17345 CUC7I6 24203167 Ki = 4000 nM T17345 CG7RU5 24203941 Ki = 3000 nM T17345 C9BO1H 24203942 Ki = 5000 nM T17345 COCG69 24203943 Ki = 3000 nM T17345 C6S0FC 24204135 Ki = 5000 nM T17345 C2M1JB 24204136 Ki = 11000 nM T17345 C5S8PW 24204221 Ki = 4000 nM T17345 C63PUM 24204222 Ki = 3000 nM T17345 C89JMH 24204223 Ki = 5000 nM T17345 CN13ZR 24204418 Ki = 5000 nM T17345 C1IN2K 24204433 Ki = 3000 nM T17345 C6Y0ZX 24204434 Ki = 7000 nM T17345 CP73JD 24204806 Ki = 5000 nM T17345 C6M5YP 24204807 Ki = 8000 nM T17345 CA3BT0 24204808 Ki = 4000 nM T17345 CEK8R6 24777136 IC50 = 39 nM T17345 C6O5CL 24778299 IC50 = 25 nM T17345 CL7KN4 24950538 IC50 = 2600 nM T17345 C2C4FZ 24950539 IC50 = 3000 nM T17345 C9LY5G 24950540 IC50 = 33000 nM T17345 CPEF92 24950541 IC50 > 30000 nM T17345 CD8QM2 24950542 IC50 = 28000 nM T17345 CX5Q0K 24950543 IC50 > 26000 nM T17345 CH9A4V 24950693 IC50 > 29000 nM T17345 CG6A8V 24950694 IC50 > 15000 nM T17345 C6F2CR 24950695 IC50 > 26000 nM T17345 CX1AR8 24950696 IC50 > 30000 nM T17345 C1PHA0 24950697 IC50 = 16000 nM T17345 CG2B8O 24950698 IC50 = 30000 nM T17345 CX97IY 24950699 IC50 > 28000 nM T17345 C32OJF 24950851 IC50 = 27000 nM T17345 CCY8U4 24950852 IC50 > 29000 nM T17345 C17DAP 24950853 IC50 > 29000 nM T17345 CPDN34 24950854 IC50 > 27000 nM T17345 C2BXV5 25002412 IC50 > 125000 nM T17345 CQ3AV2 25002763 IC50 > 125000 nM T17345 CNBS61 25007427 IC50 = 55200 nM T17345 C1ER2L 25007788 IC50 > 125000 nM T17345 CIB13V 25058133 IC50 = 1280 nM T17345 CZ9L1Y 25093361 IC50 = 1700 nM T17345 COHL97 25093362 IC50 = 1360 nM T17345 C7PUO6 25093363 IC50 = 1250 nM T17345 CZE0Q4 25093364 IC50 = 7200 nM T17345 CGRF64 25093365 IC50 = 1420 nM T17345 CU0M5T 25093366 IC50 = 2770 nM T17345 CMQR72 25093367 IC50 = 3370 nM T17345 COE57Z 25093368 IC50 = 4200 nM T17345 CJV6X5 25093369 IC50 = 1360 nM T17345 C49FRJ 25093370 IC50 = 1380 nM T17345 C6W1TN 25107577 IC50 = 3500 nM T17345 CHU9G1 25107640 IC50 = 1500 nM T17345 C5WV3Q 25107642 IC50 = 5600 nM T17345 C2FU7W 25107643 IC50 = 2500 nM T17345 C5EP2L 25107644 IC50 = 2800 nM T17345 C3YT9V 25107645 IC50 = 2900 nM T17345 CQV0S4 25107646 IC50 = 2600 nM T17345 CO01BE 25138222 IC50 = 3200 nM T17345 CCK4R2 25138223 IC50 = 1300 nM T17345 C7P2RD 25138224 IC50 = 1180 nM T17345 C4VFL0 25138225 IC50 = 57 nM T17345 CR2MW1 25138226 IC50 = 130 nM T17345 CQO1Y3 25138227 IC50 = 360 nM T17345 COB9G8 25181586 IC50 > 33000 nM T17345 CF8EX5 25187895 IC50 = 200 nM T17345 C5BH0D 25187896 IC50 = 290 nM T17345 C3F5HV 25187897 IC50 = 210 nM T17345 CJ51SH 25187898 IC50 = 180 nM T17345 C1J4CH 25195124 IC50 = 750 nM T17345 C4P5UX 25195125 IC50 = 1410 nM T17345 C8IJB9 25218207 IC50 > 31000 nM T17345 C2SY4Z 25243853 Ki = 10000 nM T17345 CS6HE5 42627761 IC50 = 110000 nM T17345 C3C2GH 44123767 IC50 = 2370 nM T17345 C93GYN 44123768 IC50 = 2150 nM T17345 COI2S4 44136999 Ki = 15430 nM T17345 CWH0S1 44137255 Ki = 590 nM T17345 CI0BF4 44201386 IC50 = 19 nM T17345 CZ6DE0 44221143 IC50 = 300 nM T17345 CL8B5Q 44221144 IC50 = 840 nM T17345 CSJ28V 44221145 IC50 = 280 nM T17345 COT01Q 44221146 IC50 = 620 nM T17345 CS14YU 44221147 IC50 = 300 nM T17345 CA64NZ 44221340 IC50 = 600 nM T17345 CK5OL1 44221343 IC50 = 2600 nM T17345 CW0IM7 44221344 IC50 = 260 nM T17345 C0QZ7V 44221345 IC50 = 290 nM T17345 C74PHB 44221346 IC50 = 2200 nM T17345 CW39YO 44221347 IC50 = 350 nM T17345 CBHT60 44221538 IC50 = 260 nM T17345 CN5QV6 44221539 IC50 = 540 nM T17345 C9O1JI 44239402 IC50 = 173 nM T17345 CL13YN 44239406 IC50 = 19.9 nM T17345 C2PA5U 44239552 IC50 = 1790 nM T17345 C4NWP5 44246325 Ki = 2500 nM T17345 C2EW0I 44246326 Ki = 770 nM T17345 CSD8T0 44246327 Ki = 650 nM T17345 CMKF08 44246328 Ki = 12000 nM T17345 CAO87V 44246329 Ki = 5300 nM T17345 CLU2V3 44246330 Ki = 4600 nM T17345 CZ8U9G 44264907 IC50 = 1 nM T17345 CCJ0E5 44272288 IC50 = 27 nM T17345 CZ83VS 44273520 Ki = 776.25 nM T17345 CB9ZO8 44281305 IC50 = 320 nM T17345 C2O1KM 44281312 IC50 = 650 nM T17345 CFB79E 44282924 Ki = 46.2 nM T17345 C8QZ2E 44282925 Ki = 55.7 nM T17345 C51OKF 44282953 Ki = 0.131 nM T17345 C41RVE 44283340 IC50 = 1.5 nM T17345 CTZ9E5 44291963 Ki = 0.00033 nM T17345 C0D1VX 44291964 Ki = 0.0006 nM T17345 CHSF50 44291965 Ki = 0.00035 nM T17345 CDW63J 44292014 Ki = 0.00062 nM T17345 CG4KS0 44292015 Ki = 0.00021 nM T17345 C2DQ9E 44300934 IC50 = 1000 nM T17345 CN9U6W 44300964 IC50 = 420 nM T17345 CEV8X6 44300967 IC50 = 220 nM T17345 C54FJZ 44301716 IC50 = 190 nM T17345 C9JG5P 44308541 IC50 = 4.6 nM T17345 C0LZ8X 44308557 IC50 = 5.7 nM T17345 C7Q4RC 44309078 IC50 = 10.2 nM T17345 C8KST2 44314297 IC50 = 12 nM T17345 CBK5E3 44338827 IC50 = 14 nM T17345 CE14LA 44342970 IC50 = 27 nM T17345 CV6U1R 44343198 IC50 = 600 nM T17345 C6GME8 44346127 IC50 = 200 nM T17345 CN0GE5 44366301 Ki = 0.00019 nM T17345 C05HEV 44366644 IC50 = 18 nM T17345 C8AQ0F 44372902 IC50 = 0.84 nM T17345 C5F0ZB 44378252 Ki = 0.29 nM T17345 CZ7Y4L 44378321 Ki = 9.87 nM T17345 C3W2YH 44378322 Ki = 0.69 nM T17345 CM4Z7A 44421498 Ki = 0.077 nM T17345 CZ4CF9 44424991 IC50 = 2800 nM T17345 C0G4XZ 44523554 IC50 = 382.1 nM T17345 CB3D5L 44529842 IC50 > 100000 nM T17345 CPDY84 44531062 IC50 = 7.6 nM T17345 CN76FA 44568860 IC50 = 20 nM T17345 CPT49L 44582168 IC50 = 560 nM T17345 C0O4GX 44582169 IC50 = 1408 nM T17345 CM67QY 44582180 IC50 = 9340 nM T17345 CPS34N 44654525 IC50 = 2900 nM T17345 CMH39V 45267084 IC50 > 22000 nM T17345 C2V1MK 45267934 IC50 = 110000 nM T17345 CA53OY 45267939 IC50 > 27000 nM T17345 CYGI67 45268817 IC50 > 16000 nM T17345 C9H3DZ 45269661 IC50 > 20000 nM T17345 CE6W3J 45269665 IC50 > 24000 nM T17345 CW82HJ 45270497 IC50 > 28000 nM T17345 CW37YT 45270501 IC50 > 19000 nM T17345 CUNA34 45270504 IC50 > 21000 nM T17345 CGU1K7 45271328 IC50 > 25000 nM T17345 C17OKU 45271331 IC50 > 19000 nM T17345 C9M2ET 45271332 IC50 > 22000 nM T17345 CVGQ38 45272213 IC50 = 813000 nM T17345 CTFO90 45273072 IC50 > 23000 nM T17345 C50PYG 45273073 IC50 > 42000 nM T17345 C70SNR 45481871 IC50 = 1200 nM T17345 CM65ZU 45481878 IC50 = 60 nM T17345 CIGZ82 45481879 IC50 = 2300 nM T17345 CM3BD5 45481892 IC50 = 290 nM T17345 CP82LD 45481893 IC50 = 1580 nM T17345 CD1G7Q 45481939 IC50 = 400 nM T17345 CM1BK5 45481950 IC50 = 88 nM T17345 C1YAE7 46231368 IC50 = 4000 nM T17345 C1PJ2K 46231369 IC50 > 200000 nM T17345 CV38CS 46231370 IC50 > 200000 nM T17345 C5WM1J 46231371 IC50 > 200000 nM T17345 C5D7UV 46231372 IC50 > 200000 nM T17345 C9OER4 46231373 IC50 > 200000 nM T17345 CW0UO4 46231409 IC50 > 200000 nM T17345 C7OG0U 46231410 IC50 > 200000 nM T17345 CU5T7G 46231411 IC50 > 200000 nM T17345 COML63 46231412 IC50 > 200000 nM T17345 CK21OD 46231413 IC50 > 200000 nM T17345 C7Y5MX 46231414 IC50 > 200000 nM T17345 CN3HM6 46844539 Ki = 49.8 nM T17345 C5NOF1 46844540 Ki = 11.8 nM T17345 C9OM6V 46844541 Ki = 13 nM T17345 C2K9SC 46844649 Ki = 188 nM T17345 C6N1YZ 46861681 IC50 = 900 nM T17345 CY3M7K 46861682 IC50 = 1000 nM T17345 CIL1Z3 46886064 IC50 = 2000 nM T17345 CDV7P4 46886065 IC50 = 500 nM T17345 CO6E2M 46886122 IC50 = 500 nM T17345 CVX23N 46886123 IC50 = 800 nM T17345 CE9TL8 46886124 IC50 = 1000 nM T17345 COQ64I 46886125 IC50 = 1000 nM T17345 CPF1G2 46886145 IC50 = 2000 nM T17345 CB4YL0 46886146 IC50 = 2000 nM T17345 CM8B7K 46886147 IC50 = 800 nM T17345 C42TQK 46886148 IC50 = 3000 nM T17345 C5USK9 46886149 IC50 = 700 nM T17345 CCGH29 46886469 IC50 = 4000 nM T17345 C3PZL9 46886489 IC50 = 1000 nM T17345 CF27TO 46886490 IC50 = 3000 nM T17345 C26DLM 46886513 IC50 = 6000 nM T17345 CN4JM7 46886546 IC50 = 3000 nM T17345 CLY37J 46898100 Ki = 34 nM T17345 CQ3E4W 46898103 Ki = 7.6 nM T17345 C9H4WN 46905455 Ki = 9 nM T17345 CF4UK7 46907163 Ki = 24.5 nM T17345 CL14GQ 50992060 Ki = 22.5 nM T17345 CE0VL8 50994805 IC50 = 300000 nM T17345 CJA45X 52914860 IC50 = 90 nM T17345 CV21AI 52914861 IC50 = 100 nM T17345 CT8R2P 52918390 Ki = 1026 nM T17345 C7BY6M 52942956 Ki = 830 nM T17345 CE02NU 52943039 IC50 = 42000 nM T17345 CX24TS 52943277 IC50 = 340 nM T17345 CA62KU 52944152 Ki = 1600 nM T17345 CE37DL 52944456 IC50 = 314 nM T17345 CQV34K 52945403 Ki = 1100 nM T17345 C97XZA 52946619 Ki = 11000 nM T17345 CD9S4I 52947801 Ki = 4300 nM T17345 CA6IL3 52947802 Ki = 1300 nM T17345 C0MQ9Y 53346505 Ki = 1138 nM T17345 C2EGS5 53346506 Ki = 12.2 nM T17345 CAK50X 53346507 Ki = 26.3 nM T17345 COSG28 53346508 Ki = 12 nM T17345 C5U3KJ 53346509 Ki = 11.1 nM T17345 CD60FA 53346510 Ki = 5.8 nM T17345 CX2NV9 53346511 Ki = 4.5 nM T17345 CK72UF 53387838 IC50 > 100000 nM T17345 CXOL35 56595784 Ki = 572 nM T17345 CT45OM 56595785 Ki = 854 nM T17345 C9OW8X 56658455 IC50 > 100000 nM T17345 C1VYN7 56658457 IC50 > 100000 nM T17345 CDWN05 56658459 IC50 > 100000 nM T17345 CEX01L 56659280 Ki = 323 nM T17345 C6UHW8 56659281 Ki = 11.1 nM T17345 C0OSM1 56662749 Ki = 95.6 nM T17345 CO14BL 56665108 IC50 = 155 nM T17345 C6ER2F 56665410 IC50 > 100000 nM T17345 C1KWA9 56665412 IC50 > 100000 nM T17345 C7IX2A 56665414 IC50 > 100000 nM T17345 CPO4V8 56665416 IC50 > 100000 nM T17345 CUPO65 56666113 IC50 > 20000 nM T17345 CDC24L 56666218 Ki = 44.1 nM T17345 C9C7KW 56666219 Ki = 85 nM T17345 CH91WP 56666648 IC50 = 14000 nM T17345 CMHP59 56668551 IC50 = 5330 nM T17345 CQP5U2 56668841 IC50 > 100000 nM T17345 C2F0BA 56668843 IC50 > 100000 nM T17345 CDGX83 56668845 IC50 > 100000 nM T17345 CML5O9 56669623 Ki = 743 nM T17345 C2FBW1 56669624 Ki = 702 nM T17345 CCS0D3 56669625 Ki = 253 nM T17345 CP91XV 56673137 Ki = 20.9 nM T17345 C3JKO4 56673138 Ki = 22.2 nM T17345 COK3Z5 56675436 IC50 = 134 nM T17345 CUQ67O 56675715 IC50 > 100000 nM T17345 C6RCQ7 56676341 IC50 > 20000 nM T17345 C8AQ1O 56676459 Ki = 138 nM T17345 C7T2IG 56676460 Ki = 27.5 nM T17345 COA13E 56676461 Ki = 245 nM T17345 COG17M 56678776 IC50 = 548 nM T17345 C6VS9Y 56679010 IC50 = 21800 nM T17345 CJZ9B0 56679012 IC50 > 100000 nM T17345 C2B0OZ 56679014 IC50 > 100000 nM T17345 C90TMJ 56679774 Ki = 129 nM T17345 C29UVR 56679775 Ki = 10.1 nM T17345 COF0V7 56680536 IC50 = 49.04 nM T17345 CKX0H5 56682332 IC50 > 100000 nM T17345 CLGR37 56682334 IC50 > 100000 nM T17345 CDH01Q 56683111 Ki = 41.1 nM T17345 CRLK58 57381314 IC50 = 289 nM T17345 CZBG69 57381532 IC50 = 599 nM T17345 CRB3F1 57404325 IC50 > 250000 nM T17345 CA6DB4 57404326 IC50 = 50000 nM T17345 CBOX49 59608000 Ki = 4330 nM T17345 CTW7K2 60142113 IC50 = 5960 nM T17345 C7NCS0 60142250 IC50 = 2110 nM T17345 CC1X7M 60142382 IC50 = 1610 nM T17345 C3SH4V 60194459 Ki = 33.6 nM T17345 C25XOP 60199138 Ki = 18.1 nM T17345 C0WYU6 60199139 Ki = 20.2 nM T17345 CSA7P4 66563689 Ki = 47.6 nM T17345 CLJ4S9 66924089 IC50 = 15000 nM T17345 C47NRM 67607115 Ki = 1164 nM T17345 C5C0VZ 67607544 Ki = 1086 nM T17345 C8YM7S 67607902 Ki = 663 nM T17345 CVQW83 67615348 Ki = 320 nM T17345 C23NBA 67889361 Ki = 943 nM T17345 C95DAH 67889364 Ki = 2.9 nM T17345 CG5J2I 70687448 IC50 > 250000 nM T17345 CJAF56 70689505 IC50 > 250000 nM T17345 CZ48NJ 70695829 IC50 = 340 nM T17345 C0OB8G 71307952 IC50 = 57 nM T17345 C7KSO5 71449539 IC50 = 420 nM T17345 CJ6SQ8 71451328 IC50 = 33 nM T17345 CQ5YE6 71451881 Ki = 4680 nM T17345 C2F5XK 71453144 IC50 = 800 nM T17345 CTP47E 71454881 IC50 = 1070 nM T17345 CB1WD6 71456658 IC50 = 32 nM T17345 CSU17Q 71460350 IC50 = 18 nM T17345 C0UXW2 71462049 IC50 = 33 nM T17345 C7FEJ4 71462050 IC50 > 100000 nM T17345 CFP1O3 71463580 IC50 = 150 nM T17345 CKA6Q2 71463581 Ki = 11 nM T17345 C9SU7T 71520360 Ki > 55000 nM T17345 C9M2JK 71520483 Ki > 332000 nM T17345 C5N4XG 71521660 Ki > 110000 nM T17345 CGP9N4 71525312 IC50 = 1300 nM T17345 C3GN0W 71560185 IC50 = 400 nM T17345 CRZK12 71560290 IC50 = 250 nM T17345 CF06NE 71560291 IC50 = 1500 nM T17345 C2SJ7K 71560296 IC50 = 60 nM T17345 CCP40I 71560419 IC50 = 45 nM T17345 CR38HE 71560424 IC50 = 140 nM T17345 C06WSC 71560425 IC50 = 260 nM T17345 CV3A1O 71680871 IC50 = 190 nM T17345 CL5G6W 71680872 IC50 = 3650 nM T17345 CN8E7Q 71680873 IC50 = 250 nM T17345 CLT08Y 71680874 IC50 = 1000 nM T17345 CBW3F2 71680875 IC50 = 3900 nM T17345 CX82PD 71680876 IC50 = 2100 nM T17345 CGR6J5 71680877 IC50 = 5900 nM T17345 C23EQL 71681031 IC50 = 2200 nM T17345 CI9Y4J 71681032 IC50 = 7200 nM T17345 CO4V1J 71681033 IC50 = 2100 nM T17345 CU5IC1 71681034 IC50 = 450 nM T17345 C3I5KR 71681035 IC50 = 3100 nM T17345 CYG8K1 71681036 IC50 = 12 nM T17345 CNT81J 71681037 IC50 = 14 nM T17345 CCS0L2 71681187 IC50 = 4.7 nM T17345 C1X8KC 71681188 IC50 = 4.6 nM T17345 C46UPB 71681189 IC50 = 32 nM T17345 C7A1WK 71681190 IC50 = 340 nM T17345 CTIX90 71681191 IC50 = 5.6 nM T17345 C38MXU 71681192 IC50 = 46 nM T17345 CMJ47I 72771095 Ki = 1101 nM T17345 CZ4D3T 73386686 IC50 = 180 nM T17345 C8HKV5 76308482 IC50 = 3000 nM T17345 CR1SA3 76310814 Ki = 4000 nM T17345 CBH3C5 76311133 Ki = 841 nM T17345 CE8K7X 76314747 Ki > 5000 nM T17345 CWYV16 76314759 Ki = 1607 nM T17345 C9L4RE 76314760 Ki = 2922 nM T17345 CWN21Q 76318014 Ki = 4000 nM T17345 CE9Q3J 76318015 Ki = 200 nM T17345 CFM0V3 76318330 Ki = 749 nM T17345 CY8T3V 76319350 IC50 = 1.3 nM T17345 C17BXW 76319351 IC50 = 8.9 nM T17345 C0WMC2 76319379 IC50 = 10 nM T17345 C1B0TE 76322025 Ki = 723 nM T17345 C7N0YG 76323015 IC50 = 7300 nM T17345 CN7LS9 76325171 IC50 = 100 nM T17345 CL62UB 76325172 IC50 = 500 nM T17345 C2TF7J 76325354 Ki = 6000 nM T17345 CZ5DA3 76325652 Ki > 3000 nM T17345 C3PJ8X 76325653 Ki > 3000 nM T17345 CUC0O5 76325779 IC50 > 1000000 nM T17345 CQYO16 76328899 Ki = 3000 nM T17345 C12PIT 76328900 Ki = 3000 nM T17345 C1W8SP 76329213 Ki = 610 nM T17345 CVS27U 76329214 Ki = 437 nM T17345 CU1N3X 76330211 IC50 = 94 nM T17345 C8CQ5G 76332587 Ki = 3000 nM T17345 CM7X0D 76332864 Ki = 1564 nM T17345 CIAJ89 76336478 Ki = 2299 nM T17345 CYZJ97 76336479 Ki > 5000 nM T17345 C60IHU 76336487 Ki = 170 nM T17345 CJEA39 77461251 IC50 = 1200 nM T17345 CI0BY7 86276188 IC50 = 688 nM T17345 CLN0B2 86276189 IC50 = 625 nM T17345 CMF27J 86577836 IC50 = 172 nM T17345 C9EMA6 86577876 IC50 = 127 nM T17345 CC0F4M 86577948 IC50 = 136 nM T17345 CMV52E 86578029 IC50 = 208 nM T17345 C6F0NA 86578120 IC50 = 477 nM T17345 CUMG18 86578123 IC50 = 170 nM T17345 C4L6CM 86578162 IC50 = 49 nM T17345 C7T4CU 86578197 IC50 = 147 nM T17345 C37MOB 86578230 IC50 = 148 nM T17345 CQ3I8M 86578301 IC50 = 174 nM T17345 CVD2Y7 90666046 IC50 = 2730 nM T17345 CQS9A6 90666047 IC50 = 3100 nM T17345 C1UY6B 90666049 IC50 = 8720 nM T17345 CIG5W1 121493974 Ki = 200.77 nM T17345 CY21HZ 122164615 IC50 = 92 nM T17345 C8QB7N 124080837 IC50 = 511 nM T17345 C9NQ7B 124080838 IC50 = 1372 nM T17345 CW2D6Y 124081250 Ki = 388.62 nM T17345 CS04TC 124081251 Ki = 234.23 nM T17345 CO5MJ2 124220265 IC50 = 45 nM T17345 CE5F7Z 124220266 IC50 = 16 nM T17345 C6WU1A 124220267 IC50 = 41 nM T17345 CRE75U 127031638 IC50 = 30000 nM T17345 CY2W5J 127032512 IC50 > 100000 nM T17345 CCQ0D9 127032513 IC50 = 56400 nM T17345 CJ2Q3G 127032813 IC50 = 2400 nM T17345 CAVH35 127033390 Ki = 5.83 nM T17345 C2J9OY 127033391 IC50 = 700 nM T17345 CWK31L 127033392 IC50 = 300 nM T17345 CO9HL0 127033684 IC50 = 8000 nM T17345 C3HRW8 127033994 IC50 > 100000 nM T17345 CBT27N 127034482 IC50 = 5000 nM T17345 CT2OP4 127034483 IC50 = 7000 nM T17345 C6V8HZ 127034484 IC50 = 20000 nM T17345 CK7AG3 127036397 IC50 = 42000 nM T17345 CU7ZS5 127041310 IC50 = 310 nM T17345 C6ZX0J 127041311 IC50 = 310 nM T17345 C2WOC5 127041312 IC50 = 110 nM T17345 C8FD5L 127041909 IC50 = 2 nM T17345 C5Q2OX 127041910 IC50 = 42400 nM T17345 CD8MQ0 127041911 IC50 = 720 nM T17345 C2ILO0 127041912 IC50 = 320 nM T17345 COL16A 127043134 Ki = 2494.9 nM T17345 CWQ6Y4 127043135 Ki = 346.15 nM T17345 CE2R6W 127043324 Ki = 158.77 nM T17345 CEM63B 127043325 Ki = 376.62 nM T17345 C6BF8K 127045460 Ki = 451.15 nM T17345 C14WFB 129906767 IC50 = 72490 nM T17345 CEWR32 130301107 IC50 = 935 nM T17345 CM7E0A 132574708 IC50 = 52000 nM T17345 C4W5JI 134132161 IC50 = 2500 nM T17345 C32OQG 134133398 IC50 > 10000 nM T17345 C4W7YT 134135190 IC50 = 920 nM T17345 CW84JC 134135508 IC50 = 33.56 nM T17345 CF2T9N 134136051 IC50 > 10000 nM T17345 CI45FO 134136319 IC50 = 36.01 nM T17345 C17NRB 134136557 IC50 > 10000 nM T17345 CW0P8B 134136864 IC50 = 32.49 nM T17345 CS27VL 134138165 IC50 = 7.46 nM T17345 CP5IW7 134138953 IC50 = 9200 nM T17345 CCWD64 134139368 IC50 = 1100 nM T17345 CVZI26 134141070 IC50 = 86.11 nM T17345 CTO84X 134141850 IC50 > 10000 nM T17345 C34GRK 134142208 IC50 = 11.07 nM T17345 C3WXJ9 134143008 IC50 = 2100 nM T17345 CWT7F2 134144326 IC50 = 760 nM T17345 CY1X2T 134144992 IC50 = 6.46 nM T17345 C20VFD 134145574 IC50 = 4.08 nM T17345 C86PJW 134146078 IC50 > 10000 nM T17345 C1KFQ9 134147493 IC50 > 10000 nM T17345 CTHA87 134147818 IC50 = 18.28 nM T17345 CQG73J 134147949 IC50 > 10000 nM T17345 CCZ38F 134148801 IC50 > 10000 nM T17345 C2H7AI 134149549 IC50 = 4200 nM T17345 CQ0B2P 134150774 IC50 = 8.23 nM T17345 CA0J6U 134151081 IC50 = 56.75 nM T17345 C3RTP9 134152596 IC50 > 10000 nM T17345 CL72SR 134153211 IC50 > 10000 nM T17345 C2B4RW 134154165 IC50 = 3.72 nM T17345 CK6CQ1 134154523 IC50 > 75000 nM T17345 C18MPZ 134154991 IC50 = 46.62 nM T17345 C5MA8G 134155232 IC50 > 10000 nM T17345 C31ZAM 134156833 IC50 = 2800 nM T17345 C1IX4T 134812633 IC50 = 308 nM T17345 C0LJE4 134816733 IC50 = 11990 nM T17345 C4SZU6 134816735 IC50 = 15320 nM T17345 C3MKJ4 134816970 IC50 = 3670 nM T17345 CCT84X 135399760 IC50 > 240000 nM T17345 CQ4F8Y 135402053 IC50 = 910 nM T17345 C6AY2U 135403832 IC50 > 20000 nM T17345 C0LTC1 135404992 IC50 = 2100 nM T17345 C9EA3J 135407589 IC50 > 100000 nM T17345 C3MHI2 135427303 IC50 = 640 nM T17345 CSNH87 135431649 IC50 = 2100 nM T17345 CJ51DM 135443603 IC50 = 83 nM T17345 CS0I8R 135469335 IC50 > 95000 nM T17345 CS4M7U 135471854 IC50 = 170 nM T17345 C7YPI6 135481470 IC50 = 330 nM T17345 C7BQ1O 135487985 IC50 = 420 nM T17345 C79OVQ 135488791 IC50 = 11 nM T17345 CPZ72B 135488819 IC50 = 460 nM T17345 C5WV3M 135488820 IC50 = 110 nM T17345 CD40CJ 135502983 IC50 > 26000 nM T17345 C98GZD 135511915 IC50 > 54000 nM T17345 CFH82R 135516724 IC50 > 32000 nM T17345 CLB45I 135543610 IC50 > 62000 nM T17345 CK4FS8 135543796 IC50 = 7000 nM T17345 CV7HQ6 135545795 IC50 = 10000 nM T17345 C8N5QD 135545810 IC50 > 21000 nM T17345 CCF8H5 135545819 IC50 > 80000 nM T17345 C9K8DE 135545856 IC50 = 11000 nM T17345 C9Z4ES 135567027 IC50 > 20000 nM T17345 CE5O9J 135570463 IC50 = 22600 nM T17345 C06IDH 135746097 IC50 > 30000 nM T17345 CGLI18 135749904 IC50 = 120 nM T17345 CQ49YZ 135749905 IC50 > 39000 nM T17345 CBUS79 135749906 IC50 > 37000 nM T17345 C2HZK8 135749907 IC50 > 37000 nM T17345 CD48XU 135749908 IC50 > 35000 nM T17345 C9NZA4 135749909 IC50 > 35000 nM T17345 C0ME1H 135749910 IC50 = 33000 nM T17345 CMVH39 135749911 IC50 > 35000 nM T17345 CR4DU1 135749912 IC50 > 35000 nM T17345 C1H6ZF 135749913 IC50 > 31000 nM T17345 CR5NK7 135749914 IC50 > 24000 nM T17345 C1LV7B 135749915 IC50 > 32000 nM T17345 CQF8P5 135800109 IC50 > 24000 nM T17345 C4IDQ3 135855753 IC50 = 66600 nM T17345 C39FIY 135855754 IC50 = 20300 nM T17345 C0N1LQ 135855759 IC50 = 66600 nM T17345 C6A4QR 135855760 IC50 = 100000 nM T17345 CRV4K7 135855761 IC50 = 10200 nM T17345 CAUV24 135855764 IC50 = 72600 nM T17345 CYAS86 135855765 IC50 = 37300 nM T17345 CTG51U 135887103 IC50 = 4700 nM T17345 CE6TP5 135887104 IC50 = 8500 nM T17345 CY5H4A 135887105 IC50 = 400 nM T17345 CHT2O4 135887106 IC50 = 220000 nM T17345 CWL71S 135887124 IC50 = 2000 nM T17345 CNKW46 135887125 IC50 = 12000 nM T17345 CH1W2S 135887126 IC50 = 210 nM T17345 C6U0PF 135887127 IC50 = 250 nM T17345 COA6S0 135887128 IC50 = 1950 nM T17345 CBO9A7 135887129 IC50 = 320 nM T17345 CFIG79 135887147 IC50 > 1000000 nM T17345 CDA05G 135887148 IC50 > 1000000 nM T17345 CZB8O6 135960753 IC50 = 22000 nM T17345 CZ6C4R 135964391 IC50 > 29000 nM T17345 CUOV62 135964392 IC50 > 34000 nM T17345 CG23QU 135964393 IC50 > 32000 nM T17345 CR5EG8 135964397 IC50 > 28000 nM T17345 C0T2QO 135964404 IC50 > 32000 nM T17345 CD8WY9 135964405 IC50 > 25000 nM T17345 CRXF18 135964411 IC50 > 31000 nM T17345 C87XGZ 135964413 IC50 > 32000 nM T17345 CF1N5G 136002190 IC50 = 750 nM T17345 C3LWJ1 136002235 IC50 = 460 nM T17345 CJ7ES6 136016316 IC50 = 290 nM T17345 C24FWM 136016317 IC50 = 370 nM T17345 C9SMI1 136016318 IC50 = 340 nM T17345 CMG1F8 136016319 IC50 = 300 nM T17345 C1GE3H 136016320 IC50 = 640 nM T17345 C56SPO 136046100 IC50 = 430 nM T17345 CT0NK9 136046104 IC50 > 40000 nM T17345 CA1R9P 136046152 IC50 = 950000 nM T17345 C6CMD5 136046154 IC50 = 1300 nM T17345 CDMI28 136056632 IC50 = 3800 nM T17345 CL8YP6 136056633 IC50 = 530 nM T17345 CZ0JY3 136056634 IC50 = 1500 nM T17345 CMQ87O 136056635 IC50 = 3800 nM T17345 C5X9UG 136078523 IC50 = 650 nM T17345 CTK4I6 136078526 IC50 = 260 nM T17345 CML42R 136092224 IC50 63300 nM T17345 C8O2GN 136109165 IC50 = 100 nM T17345 CALV20 136109177 IC50 = 100 nM T17345 CKI9N0 136136563 IC50 = 3000 nM T17345 CG3OA8 136136566 IC50 = 1400 nM T17345 C7QAB0 136171375 IC50 = 3200 nM T17345 C6XHI1 136171377 IC50 = 280 nM T17345 CVKL45 136171378 IC50 = 300 nM T17345 C23HGZ 136191424 Ki ~ 600 nM T17345 CVY71R 137300720 IC50 > 10000 nM T17345 CWE38X 137491959 IC50 = 12500 nM T17345 CM10NY 137631470 IC50 = 28000 nM T17345 CAZB89 137631503 IC50 = 2250 nM T17345 CWR72A 137632901 IC50 = 19000 nM T17345 CYF76S 137633375 IC50 = 5330 nM T17345 CFUY16 137633842 IC50 > 27000 nM T17345 CNT9K1 137634037 IC50 = 9.2 nM T17345 CZ5B9O 137634433 IC50 = 16900 nM T17345 CPB9Q3 137634556 IC50 = 1260 nM T17345 C0PNW5 137635062 IC50 = 450 nM T17345 CS23KQ 137635618 IC50 > 28000 nM T17345 CF5S9P 137636125 IC50 = 4 nM T17345 C7N6WS 137636390 IC50 > 150000 nM T17345 C53CKY 137636400 IC50 = 853 nM T17345 COE67T 137637328 IC50 > 50000 nM T17345 CL87FM 137638209 IC50 = 108 nM T17345 CA01DG 137638564 IC50 = 3.2 nM T17345 CP8X2O 137639098 IC50 = 290 nM T17345 CL95CK 137639545 IC50 = 6.1 nM T17345 CK6GP0 137640129 IC50 = 14800 nM T17345 C4QHY1 137640582 IC50 = 3610 nM T17345 C8MQ6U 137642178 IC50 = 2.6 nM T17345 C19WKB 137642364 IC50 = 6000 nM T17345 CU8YX6 137643005 IC50 > 27000 nM T17345 CW27XK 137644048 IC50 = 25000 nM T17345 C4N6GR 137644261 IC50 = 36 nM T17345 CT6CI1 137644294 IC50 = 710 nM T17345 C9YX2K 137644352 IC50 = 4000 nM T17345 CA7QW8 137645236 IC50 = 53.4 nM T17345 CSXF17 137645367 IC50 = 2840 nM T17345 CO0U6R 137646091 IC50 = 1400 nM T17345 C4NJB5 137646478 IC50 = 4.2 nM T17345 C83JEY 137646749 IC50 = 13.1 nM T17345 CRU6D2 137647615 IC50 = 5.3 nM T17345 CA7Y9F 137648264 IC50 = 4780 nM T17345 CZGU30 137648786 IC50 = 44 nM T17345 CQED79 137651284 IC50 = 2550 nM T17345 C5V4MO 137651590 IC50 = 14.1 nM T17345 CL1DZ0 137651595 IC50 = 5280 nM T17345 CQUY83 137652218 IC50 > 29000 nM T17345 CB3H5W 137652434 IC50 = 6.4 nM T17345 CSR07T 137654267 IC50 = 3190 nM T17345 CR71UO 137654559 IC50 = 950 nM T17345 C9JT1N 137655519 IC50 > 30000 nM T17345 C5XVK8 137656132 IC50 = 4130 nM T17345 C1M2YZ 137657601 IC50 = 2480 nM T17345 CQJD20 137657673 Ki = 13170 nM T17345 CX2T5K 137658038 IC50 = 35.6 nM T17345 CYV97X 137659199 IC50 = 4340 nM T17345 CO79SP 137659251 IC50 = 1670 nM T17345 CYML31 137659929 IC50 = 59.2 nM T17345 CETP42 137660220 IC50 = 3.4 nM T17345 C8W5GY 137660580 IC50 = 20100 nM T17345 C4UF6M 137660773 IC50 = 4.8 nM T17345 CD6VN2 137660870 IC50 = 9 nM T17345 C7V3LC 137661421 IC50 = 3.9 nM T17345 CFI5E0 137661591 IC50 = 18 nM T17345 CC8QH2 138460007 IC50 = 1090 nM T17345 C9NL0Q 138460276 IC50 = 1430 nM T17345 CL45VQ 145949793 Ki = 530 nM T17345 CX76CQ 145954183 Ki = 1400 nM T17345 C8QO7R 145955925 Ki = 640 nM T17345 CE0VX2 145967688 IC50 = 700 nM T17345 C49HWY 145967911 IC50 = 970 nM T17345 C4Q8MH 145968315 IC50 = 1101 nM T17345 CL72EN 145968368 IC50 = 1400 nM T17345 CK5H1X 145968380 IC50 = 579 nM T17345 C7ILN2 145968384 IC50 = 2730 nM T17345 CKC3W9 145968635 IC50 = 70510 nM T17345 C2V6SX 145968836 IC50 = 2318 nM T17345 CBP38L 145968849 IC50 = 590 nM T17345 C2LD6U 145968997 IC50 = 1917 nM T17345 CZ6LQ5 145969012 IC50 = 7930 nM T17345 C7N8WS 145969103 IC50 = 12290 nM T17345 CR9J7O 145970201 IC50 = 610 nM T17345 C04XEC 145970467 IC50 = 1130 nM T17345 C48KNM 145970614 IC50 = 811 nM T17345 CBXY67 145970730 IC50 = 2530 nM T17345 CT72GK 145970859 IC50 = 60 nM T17345 CIG4X8 145970868 IC50 = 11230 nM T17345 CHC2I0 145971065 IC50 = 2100 nM T17345 CEA95O 145971179 IC50 = 2046 nM T17345 CLY9F6 145988837 IC50 = 1104 nM T17345 CG36PF 145989276 IC50 > 100000 nM T17345 CUP4Z9 151456061 IC50 = 1360 nM T17345 CSL7O9 152598220 IC50 = 1790 nM T17345 C5OVQ3 152617142 IC50 = 347 nM T17345 CI79YB 155510882 IC50 = 1630 nM T17345 CB8J3L 155511255 IC50 = 37.94 nM T17345 C7GFM4 155512559 Ki = 18.41 nM T17345 CGK20J 155513582 IC50 = 819 nM T17345 C6D2CN 155514408 IC50 = 903 nM T17345 CS84IM 155515034 Ki = 555.55 nM T17345 CO9ZD7 155516975 IC50 = 29.29 nM T17345 CPX7N5 155517476 Ki = 23.42 nM T17345 CK8UH6 155518935 Ki = 13.41 nM T17345 C1ZA0M 155520729 IC50 = 1098 nM T17345 CHW46G 155523087 IC50 >= 1000 nM T17345 CUY38N 155523154 Ki = 18.24 nM T17345 CF4JM8 155523234 IC50 = 10 nM T17345 CEA02Z 155527030 Ki = 508.88 nM T17345 CT6S0G 155527248 IC50 = 237 nM T17345 CLO94T 155527394 Ki = 14.36 nM T17345 C3U4ED 155528338 IC50 = 300 nM T17345 C4N5QE 155528668 Ki = 19.55 nM T17345 C8PH3I 155529256 IC50 = 2626 nM T17345 C1GZ7W 155529285 Ki = 21.72 nM T17345 CR0O1S 155529844 IC50 > 30000 nM T17345 C87EWF 155530674 IC50 = 1100 nM T17345 CJ1P8L 155531623 IC50 = 1330 nM T17345 CT40PE 155532707 IC50 = 1800 nM T17345 C5H8LY 155532752 Ki = 32.89 nM T17345 C9OW3C 155533311 Ki = 74.16 nM T17345 C2P4MC 155534197 IC50 = 4125 nM T17345 C51XLA 155539843 Ki = 22.07 nM T17345 CFP3Y7 155540286 IC50 >= 1000 nM T17345 CG1S5K 155542983 IC50 = 65.88 nM T17345 C49SMW 155543062 IC50 = 2253 nM T17345 C0SNO1 155543141 IC50 = 3260 nM T17345 C5GZ1N 155543331 IC50 = 980000 nM T17345 CC20PV 155543847 IC50 = 1808 nM T17345 CP15AX 155544485 Ki = 48.67 nM T17345 C9MU3J 155546590 IC50 = 53.42 nM T17345 C9QN6E 155547319 IC50 = 100 nM T17345 CA4T8J 155548037 IC50 = 541 nM T17345 CNA65G 155549118 IC50 = 5980 nM T17345 CM5F3R 155550798 Ki = 8.72 nM T17345 CKBA16 155550915 IC50 = 973 nM T17345 C4SXE2 155551604 Ki = 32.43 nM T17345 CPV2I5 155552635 IC50 = 210 nM T17345 C2NIY4 155552687 Ki = 34.84 nM T17345 C3U7CK 155552787 IC50 = 1540 nM T17345 C0V2SW 155553051 IC50 = 125000 nM T17345 C1WXN8 155553663 IC50 = 2710 nM T17345 C4PLU8 155554619 Ki = 27.27 nM T17345 CVHM01 155555730 Ki = 12.5 nM T17345 C3KM4N 155556589 IC50 = 48.95 nM T17345 C4WH0C 155557612 Ki = 12.77 nM T17345 C8WB9O 155558582 IC50 >= 1000 nM T17345 CDB7F2 155560431 IC50 > 30000 nM T17345 CMYU10 155561126 Ki = 52.39 nM T17345 CE84AM 155561456 IC50 = 670 nM T17345 CXYW29 155562270 IC50 = 200 nM T17345 CU71YW 155562818 IC50 = 1571 nM T17345 CFM53Y 155563602 IC50 = 1576 nM T17345 CQ97VE 155565527 IC50 = 180000 nM T17345 C6COP9 155565754 IC50 = 1300 nM T17345 CV6WP8 155566484 IC50 = 9.28 nM T17345 C8BGX5 155567131 Ki = 29.05 nM T17345 CWON57 155567297 Ki = 45.97 nM T17345 C8M7LB 155567321 IC50 = 1338 nM T17345 CGMA98 155567948 Ki = 13.59 nM T17345 CUV9H3 155568251 IC50 = 2800 nM T17345 C9S2ON 155568330 IC50 = 468 nM T17345 C5ILH2 155568439 IC50 = 1373 nM T17345 D00IBG 643976 IC50 = 325000 nM T17345 D01HKU 44428667 IC50 = 120 nM T17345 D02ZCP 446244 IC50 = 620 nM T17345 D02ZPZ 6532431 Ki = 1.8 nM T17345 D03DRF 46886486 IC50 = 2000 nM T17345 D04PAW 16216218 IC50 = 250 nM T17345 D05WHM 6917908 IC50 = 4.4 nM T17345 D06DIH 158376 IC50 = 220 nM T17345 D06ERH 637760 IC50 > 100000 nM T17345 D06QEN 467889 Ki = 230 nM T17345 D06UPT 446752 IC50 = 4.3 nM T17345 D07LSP 135438608 IC50 = 1900 nM T17345 D07XLJ 462120 IC50 = 2400 nM T17345 D08GPU 490662 Ki = 2.9 nM T17345 D0B0UI 44428664 IC50 = 70 nM T17345 D0H8AW 291270 IC50 = 23000 nM T17345 D0J4KJ 446245 IC50 = 940 nM T17345 D0JY6J 93114 Ki = 10.4 nM T17345 D0LH5P 100516 IC50 = 4.1 nM T17345 D0ME8Z 24778025 IC50 = 0.39 nM T17345 D0O9YG 9049 Ki = 55.6 nM T17345 D0P9XE 46871716 Ki = 93 nM T17345 D0R4PS 135403648 Ki = 2370 nM T17345 D0S4ZT 46886512 IC50 = 5000 nM T17345 D0Y3TU 334409 Ki = 1 nM T17345 D0Z9QC 135517463 IC50 = 34 nM T17345 D0ZG7W 11441554 IC50 > 100000 nM T77393 C6F2WU 700755 Ki > 1000000 nM T77393 CZS6I0 720519 Ki > 1000000 nM T77393 CJL6Z8 765511 Ki = 323000 nM T77393 CQ2S4B 910123 Ki = 61000 nM T77393 C9AVC3 1006789 IC50 = 25000 nM T77393 C5XG0W 1006800 IC50 = 13620 nM T77393 C36IHN 1006808 IC50 = 24000 nM T77393 C3N7ZL 1006833 IC50 = 9630 nM T77393 CMD15J 1006856 IC50 = 22000 nM T77393 CA1X5I 1025961 IC50 = 22000 nM T77393 C3D1ZK 1266319 IC50 = 38000 nM T77393 CKR60Y 2810167 IC50 = 6000 nM T77393 CU0VC2 2943337 IC50 > 20000 nM T77393 CN9SE0 3308644 Ki = 843000 nM T77393 CAV9I1 3697667 Ki = 8440 nM T77393 C9FT3D 13430822 Ki = 589000 nM T77393 C9CR0M 15561337 Ki = 651000 nM T77393 C6C2JF 16483718 IC50 = 24000 nM T77393 C1XOL3 16487351 IC50 = 22000 nM T77393 CL3C9H 16645214 IC50 = 22000 nM T77393 C78LBG 16645215 IC50 = 30000 nM T77393 C4IAR3 16645216 IC50 = 12970 nM T77393 C6IM7Q 24757930 Ki = 27300 nM T77393 C6XPA0 39845054 IC50 = 48000 nM T77393 CC30IP 39845125 IC50 = 23000 nM T77393 CT4OS9 39845172 IC50 = 13000 nM T77393 CI9N1O 46864279 Ki = 120 nM T77393 CM51WO 46864280 Ki = 20 nM T77393 C81DFP 46866889 Ki = 200 nM T77393 C1U3KE 46867009 Ki = 3 nM T77393 CCKI47 46867010 Ki = 20 nM T77393 CT24XZ 46867121 Ki = 6300 nM T77393 C5WP7S 46867122 Ki = 7300 nM T77393 CM27BD 46867257 Ki < 1 nM T77393 CS6J9I 46889977 Ki = 160 nM T77393 C4DR8T 46889978 Ki = 30 nM T77393 CAJ5E1 46889979 Ki = 90 nM T77393 C8NY4I 46889980 Ki = 160 nM T77393 CK48PC 46889981 Ki = 80 nM T77393 CM5XP9 46889982 Ki = 27000 nM T77393 C0SFR4 46889983 Ki > 50000 nM T77393 C0L7GM 46889984 Ki = 3200 nM T77393 CPE06Y 46889985 Ki > 50000 nM T77393 CZ9VF6 46889986 Ki = 150 nM T77393 CXV0F2 46889987 Ki = 6500 nM T77393 COKG74 46889988 Ki = 1600 nM T77393 CP7E6H 46889989 Ki = 15100 nM T77393 CQTU62 46889993 Ki = 15000 nM T77393 CO7ZX4 46889994 Ki = 9000 nM T77393 C1WP0Q 46889995 Ki = 15600 nM T77393 C52WPZ 53356803 Ki < 1 nM T77393 C5JOC6 54766612 Ki < 1 nM T77393 CBT35C 54766613 Ki < 1 nM T77393 CH1KS7 70679466 IC50 = 338.2 nM T77393 C8IPK7 71586081 IC50 = 0.9 nM T77393 CY1J9L 85721372 IC50 > 20000 nM T77393 CN7F5K 127048565 IC50 = 660.9 nM T77393 C5J6QE 127048926 IC50 = 733.3 nM T77393 C9IK3M 127048927 IC50 = 127.4 nM T77393 CZ9T0Q 127048933 IC50 > 20000 nM T77393 C4DL6C 127048934 IC50 = 11400 nM T77393 CUN7F3 127048935 IC50 > 20000 nM T77393 CH1K3Y 127049251 IC50 = 206.1 nM T77393 CG84YX 127049252 IC50 = 207.2 nM T77393 CO0ZG4 127049253 IC50 = 130 nM T77393 C1IPG6 127049254 IC50 > 20000 nM T77393 CT10RI 127050095 IC50 > 20000 nM T77393 CL5V0S 127050385 IC50 = 1604 nM T77393 CXH7K0 127050386 IC50 = 198.5 nM T77393 C19BTR 127050387 IC50 = 465.7 nM T77393 C7T5WN 127052836 IC50 = 392.6 nM T77393 CC71PB 127052837 IC50 = 103.9 nM T77393 CBI1K8 127052955 IC50 > 20000 nM T77393 CO8X1P 127052956 IC50 > 20000 nM T77393 CR8JM3 127052957 IC50 > 20000 nM T77393 C75QVY 127052958 IC50 > 20000 nM T77393 CX8MA9 127052959 IC50 > 20000 nM T77393 CGY79B 127052960 IC50 > 20000 nM T77393 CQF37D 132580838 IC50 = 46.5 nM T77393 C0LHZ3 132580839 IC50 = 26.4 nM T77393 CN3MY7 134129874 IC50 > 20000 nM T77393 CVZS03 134129880 IC50 = 81.5 nM T77393 CO75BV 134129898 IC50 = 340.8 nM T77393 C15JEQ 134129903 IC50 = 13600 nM T77393 CSMF23 134129955 IC50 = 70.1 nM T77393 C8WNH1 134130001 IC50 > 20000 nM T77393 CZV10G 134130017 IC50 = 102.1 nM T77393 CMLA18 134130074 IC50 = 5800 nM T77393 C6OPH7 134130102 IC50 = 197.6 nM T77393 CZ9X1B 134130118 IC50 > 20000 nM T77393 CYO72F 134130195 IC50 = 47.9 nM T77393 C8M9NP 134130199 IC50 = 285.1 nM T77393 CN0HP5 134130274 IC50 = 104.6 nM T77393 C9DJC5 134130275 IC50 = 1363 nM T77393 C7A3FI 134130278 IC50 = 77.1 nM T77393 C1UR5D 134130359 IC50 > 20000 nM T77393 CL3Z2T 134130407 IC50 = 30.1 nM T77393 CO9BF6 134130408 IC50 = 1553 nM T77393 C9YS8H 134130465 IC50 = 92.5 nM T77393 CB08EV 134130500 IC50 = 62.5 nM T77393 CY24IA 134130560 IC50 = 113.4 nM T77393 C8XUN4 134130570 IC50 = 18.2 nM T77393 CRIW18 134130589 IC50 > 20000 nM T77393 CM5US2 134130592 IC50 = 8.5 nM T77393 CXH06K 134130734 IC50 = 285.3 nM T77393 CB61JP 134130757 IC50 = 7.6 nM T77393 C48BIF 134130903 IC50 > 20000 nM T77393 C5KRU7 134130925 IC50 = 75.8 nM T77393 CZ4J1P 134130945 IC50 = 95.6 nM T77393 CBP5O4 134130958 IC50 = 421.9 nM T77393 CYL7R9 134131003 IC50 = 88.7 nM T77393 CYFW16 134131026 IC50 = 50.2 nM T77393 CIN01V 134131045 IC50 = 15 nM T77393 CBF6E4 134131065 IC50 = 77.9 nM T77393 C4B7MN 134131117 IC50 = 3186 nM T77393 C59JMH 134131257 IC50 = 1093 nM T77393 CHJ39K 134131302 IC50 > 20000 nM T77393 C7GBH3 134131374 IC50 > 20000 nM T77393 C7SKU8 134131410 IC50 = 76 nM T77393 C3O4TN 134131411 IC50 > 20000 nM T77393 CF5S3O 134131548 IC50 = 70 nM T77393 C30GML 134131594 IC50 = 80.4 nM T77393 C56NTH 134135619 IC50 = 483.5 nM T77393 C17JRH 134135674 IC50 > 20 nM T77393 C7PN4W 134135702 IC50 = 263.5 nM T77393 C10RIC 134136312 IC50 = 1171 nM T77393 CCN03X 134137047 IC50 > 20 nM T77393 C3ZA5K 134137967 IC50 > 20 nM T77393 C71GIB 134140087 IC50 = 283.9 nM T77393 CB0NA6 134143014 IC50 = 162.4 nM T77393 C9IGQ2 134143930 IC50 > 20 nM T77393 C2RS6U 134144485 IC50 > 20 nM T77393 C3G6AQ 134145642 IC50 = 433.2 nM T77393 C9AJI4 134145666 IC50 > 20 nM T77393 C72APM 134148078 IC50 = 454 nM T77393 CO57LR 134148875 IC50 > 20 nM T77393 CG74JP 134149023 IC50 > 20 nM T77393 CCMR94 134149266 IC50 > 20 nM T77393 CRMX45 134149901 IC50 > 20 nM T77393 CG78KP 134153992 IC50 = 244.9 nM T77393 CF1KZ5 134155604 IC50 = 58.8 nM T77393 CI3CN5 134157644 IC50 = 811.6 nM T77393 CH1S6B 134364156 Ki = 3.53 nM T77393 C8LV1Q 134364178 Ki = 105 nM T77393 C4MIV7 134369551 Ki = 7540 nM T77393 CK6ZM1 134369552 Ki = 7210 nM T77393 C1OLR0 134369556 Ki = 665 nM T77393 CHNY14 134369557 Ki = 2600 nM T77393 C3LO6E 134369558 Ki = 17600 nM T77393 CLH26P 134369559 Ki = 219 nM T77393 C59CPA 134369560 Ki = 503 nM T77393 CJ3R0T 134369561 Ki = 3130 nM T77393 C12FZJ 134369563 Ki = 3910 nM T77393 C7QFN0 134369568 Ki = 690 nM T77393 CKUR59 134369576 Ki = 1380 nM T77393 C1Y3CD 134369579 Ki = 4130 nM T77393 C4F5BV 134369583 Ki = 1260 nM T77393 CK0JG5 134369594 Ki = 480 nM T77393 C0LKG2 134369619 Ki = 1460 nM T77393 CR6ZE1 134369620 Ki = 148 nM T77393 CYM14L 134369623 Ki = 118 nM T77393 C9Z7GJ 134369629 Ki = 42.5 nM T77393 CN8DO3 134369637 Ki = 27.6 nM T77393 CDVS67 134369647 Ki = 473 nM T77393 C3OE7I 134369648 Ki = 9.89 nM T77393 CLC39Q 134369650 Ki = 22.8 nM T77393 C71NAT 134369652 Ki = 28.9 nM T77393 CH8C7V 134369653 Ki = 76.1 nM T77393 C2C7AZ 134369665 Ki = 13.1 nM T77393 CT61JH 134369666 Ki = 185 nM T77393 CRW1A0 134369668 Ki = 184 nM T77393 CBW56J 134369669 Ki = 95 nM T77393 C6B9RO 134369670 Ki = 51.9 nM T77393 C4F1OP 134369672 Ki = 20.7 nM T77393 C15BUR 134369676 Ki = 2.82 nM T77393 CP46RA 134369681 Ki = 924 nM T77393 C63WBR 134369708 Ki = 16.4 nM T77393 C8B3LO 137349384 Ki = 85200 nM T77393 CSM61B 138319680 Ki = 0.044 nM T77393 CK27NV 138470399 Ki = 9.36 nM T77393 CMTD84 138470404 Ki = 65.1 nM T77393 CMG7V3 138470418 Ki = 2.51 nM T77393 CB24SI 138470423 Ki = 0.902 nM T77393 C8X5US 145981722 Ki = 109000 nM T77393 C9EAI7 145982119 Ki > 125000 nM T77393 CJ23AP 145988536 Ki = 1120 nM T77393 CF0BR7 145989019 Ki = 64000 nM T77393 C0IUB7 145989142 Ki = 117000 nM T77393 C49OYH 145990286 Ki > 125000 nM T77393 CK2C9E 145991249 Ki = 64300 nM T77393 C7YAG8 145992826 Ki = 118000 nM T77393 CX74VN 145992918 Ki = 29700 nM T77393 C2AHW4 145993387 Ki = 4.94 nM T49031 D00UVA 11556711 IC50 = 2.7 nM T49031 D01MML 49867936 IC50 = 8.44 nM T49031 D04AIT 5280445 IC50 = 1300 nM T49031 D0E7PQ 5311 IC50 > 25000 nM T49031 D0K8KX 5280343 IC50 = 2000 nM T49031 D0SH3I 387447 Ki = 0.55 nM T49031 D0T9TJ 3034010 IC50 > 100000 nM T49031 D05KED 53340666 IC50 > 25000 nM T49031 D07SDQ 969516 IC50 = 10000 nM T49031 D0DP0J 92135659 IC50 = 1670 nM T49031 D0F9BT 25067547 IC50 = 10 nM T49031 D0L4FS 5280961 IC50 = 9260 nM T49031 D0N0RN 11347535 IC50 = 22 nM T49031 D0U2BH 65064 IC50 = 86 nM T49031 D0VO0T 24800541 IC50 = 3 nM T49031 D0Y2SW 25183872 IC50 = 3 nM T49031 D0U7OU 3220 IC50 = 1220 nM T49031 CKGX24 7060 IC50 > 25000 nM T49031 C29BVT 11926 IC50 > 25000 nM T49031 CTK25Q 72277 IC50 = 1200000 nM T49031 CPSA65 80458 IC50 = 3000 nM T49031 CNIW58 107905 IC50 = 194 nM T49031 CDZ65K 199472 IC50 = 187 nM T49031 CA6ID2 241903 IC50 = 4580 nM T49031 C9A1KC 282849 IC50 > 25000 nM T49031 CF5T0S 282888 Ki = 2180 nM T49031 CPEL12 336327 IC50 > 100000 nM T49031 C46ZED 434315 Ki = 2120 nM T49031 C7HME8 439246 IC50 = 41600 nM T49031 C3YF4P 462382 IC50 = 1.2 nM T49031 C1MY6Z 490002 Ki = 2.3 nM T49031 CZ0AH3 638278 IC50 = 4880 nM T49031 C2DC6P 684753 Ki = 11500 nM T49031 CS4F8G 688857 IC50 = 5210 nM T49031 C2JU6P 833502 Ki = 10900 nM T49031 CS1P9Y 906456 IC50 = 172200 nM T49031 C2CR9F 1722365 Ki = 2010 nM T49031 C5FC0Z 2215326 IC50 = 3500 nM T49031 CL3KS0 5497183 IC50 = 61 nM T49031 CL9NX1 6610292 IC50 = 160 nM T49031 CK1U3G 6871286 IC50 > 10000 nM T49031 CL4VY9 9874885 Ki = 0.72 nM T49031 C3TDO0 9920246 IC50 = 1900 nM T49031 COK6X9 9960660 Ki < 1 nM T49031 CB2KX5 10032943 Ki = 0.5 nM T49031 CDPZ20 10099985 Ki = 5.7 nM T49031 C56PLQ 10258908 Ki = 0.72 nM T49031 CV25EX 10346881 IC50 = 51090 nM T49031 CO2HE7 10461001 Ki = 38 nM T49031 C5CBI2 10484581 Ki = 0.65 nM T49031 CDW5Y2 10542930 IC50 > 10000 nM T49031 CLU69K 10628969 IC50 = 420 nM T49031 CU8I1N 11243977 EC50 = 10 nM T49031 C1A2IM 11512726 IC50 = 2.9 nM T49031 C31TAR 11520347 Ki = 500 nM T49031 C6B5UF 11520360 IC50 = 52 nM T49031 C3GE9O 11532672 IC50 = 3360 nM T49031 CF2R5T 11534087 IC50 = 17 nM T49031 C61XQZ 11542118 IC50 = 1.5 nM T49031 CV56WA 11548000 IC50 = 6560 nM T49031 CWX6Y7 11549328 Ki = 32 nM T49031 C8MEH4 11549343 Ki = 140 nM T49031 C3BTN5 11556651 IC50 = 2.5 nM T49031 C2OPE1 11556685 IC50 = 2.4 nM T49031 CMH1V5 11563622 IC50 = 570 nM T49031 C8T5DM 11570453 IC50 = 170 nM T49031 C9KS5X 11578303 IC50 = 120 nM T49031 CB1L7I 11583999 IC50 = 260 nM T49031 CETS82 11585586 Ki = 45 nM T49031 CW7Z2P 11585713 IC50 = 2500 nM T49031 CH4RG7 11591941 IC50 > 10000 nM T49031 CFH34R 11598900 IC50 = 21000 nM T49031 CR9VG2 11599767 IC50 = 5.9 nM T49031 CKN7V8 11600122 Ki = 0.51 nM T49031 CO9PW8 11607192 IC50 = 78 nM T49031 CW0T9J 11613973 IC50 = 56000 nM T49031 C9OT1M 11621366 IC50 = 1.1 nM T49031 CX51NM 11636132 IC50 = 540 nM T49031 CB70KR 11636235 IC50 = 10 nM T49031 CLUA24 11636269 IC50 = 1400 nM T49031 CYR86V 11664755 IC50 = 49 nM T49031 CJFM60 11671614 IC50 = 4.3 nM T49031 CZ68VB 11672014 IC50 = 44 nM T49031 CZF9M1 11686028 Ki = 130 nM T49031 CE82UG 11692971 IC50 = 28000 nM T49031 CJE3N7 11693095 IC50 = 6.7 nM T49031 CJ1H4E 11700022 IC50 = 14 nM T49031 CX9D8R 11707332 IC50 = 2300 nM T49031 CF3Y2Q 11714595 IC50 = 49 nM T49031 CLBD57 15479395 IC50 = 220 nM T49031 C8D5OY 16084592 IC50 = 6670 nM T49031 C5RA8E 17480620 Ki = 7550 nM T49031 C7JCW4 21140132 Ki = 4700 nM T49031 C19EMT 23649126 IC50 = 700 nM T49031 CU0FE7 24752894 IC50 > 10000 nM T49031 C9E8MQ 24753965 IC50 = 7190 nM T49031 C7A4VT 24966905 IC50 > 10000 nM T49031 C5RCN7 24966906 Ki = 580 nM T49031 C1LJZ3 24966907 IC50 > 10000 nM T49031 C1MJ0W 25053219 IC50 = 1440 nM T49031 C64CJD 25111344 IC50 > 5000 nM T49031 CG52FR 42601513 Ki = 843 nM T49031 CB8H2Y 42612596 IC50 = 49 nM T49031 CN6D8U 44190246 IC50 = 4.37 nM T49031 CKH7Y0 44190247 IC50 = 1.6 nM T49031 CC8FG3 44191199 IC50 = 1.2 nM T49031 CKM83N 44307872 IC50 = 140 nM T49031 C21GXN 44410779 Ki > 450000 nM T49031 CXS71L 44411047 IC50 = 430 nM T49031 C90ZUI 44411546 IC50 = 2230 nM T49031 CMV46Q 44411707 IC50 = 4320 nM T49031 CP03SX 44411716 IC50 = 4150 nM T49031 CHFA42 44477958 IC50 = 15300 nM T49031 C69XJY 44477959 IC50 = 10000 nM T49031 C7NW5T 44555355 IC50 = 0.08 nM T49031 CN57MC 44583022 IC50 = 10 nM T49031 C9GUZ5 45140224 IC50 = 31 nM T49031 C5GAE4 45140225 IC50 = 3 nM T49031 C9RL7F 46233200 IC50 = 1 nM T49031 CNFQ84 46233201 IC50 = 2 nM T49031 CB57EF 46233202 IC50 = 100 nM T49031 CZ29GM 46233203 IC50 = 200 nM T49031 CQO52J 46233204 IC50 = 130 nM T49031 C4V9JP 46233205 IC50 = 300 nM T49031 C38TWK 46233206 IC50 = 524807460.3 nM T49031 CM81GQ 46864294 IC50 = 2.1 nM T49031 CX1YJ8 49799952 IC50 = 4.26 nM T49031 CHO3X2 49799953 IC50 = 7.63 nM T49031 C3XCL9 49859747 Ki = 2430 nM T49031 CIW0H6 50899478 IC50 = 0.55 nM T49031 C5QU2O 50899571 IC50 = 0.42 nM T49031 C8WD6E 50899573 IC50 = 0.39 nM T49031 CWDL81 52948098 IC50 = 16 nM T49031 C5EQD3 53362657 IC50 = 303.8 nM T49031 C7Q0RA 54455523 IC50 = 514 nM T49031 CV1P6X 56945245 IC50 = 92 nM T49031 CG2D5M 57149553 IC50 = 93 nM T49031 C3QG8L 59127842 IC50 = 1700 nM T49031 CLM1G5 60164712 IC50 > 30000 nM T49031 CGZ89B 65806958 IC50 = 24790 nM T49031 C82JTA 71305068 IC50 = 11600 nM T49031 CQD09I 71495550 Ki = 3744 nM T49031 CR38FB 71543331 Ki = 374.9 nM T49031 C2GAT5 71561597 IC50 = 1500 nM T49031 C62JWN 71561733 IC50 = 13000 nM T49031 CJ9AR2 71561735 IC50 = 5500 nM T49031 CXJP49 71561736 IC50 = 2800 nM T49031 CZ4I1N 71561866 IC50 = 10500 nM T49031 CHG65M 71561867 IC50 = 630 nM T49031 CA5T6O 71561868 IC50 = 2400 nM T49031 C2E9HV 71561869 IC50 = 480 nM T49031 C5FDT2 71561997 IC50 = 93 nM T49031 C2F0BJ 71561998 IC50 = 160 nM T49031 CSG26R 71561999 IC50 = 110 nM T49031 C45HOE 71562349 IC50 = 1200 nM T49031 CSDV65 71562351 IC50 = 1100 nM T49031 CKE98R 71625293 Ki = 101 nM T49031 CA95PY 71625294 Ki = 67 nM T49031 CVD0M7 71625412 Ki = 10.3 nM T49031 C6KP3Q 71625413 Ki = 10.8 nM T49031 CO9HD8 71625414 Ki = 11.4 nM T49031 CB7A3F 71625415 Ki = 10.6 nM T49031 CB24WG 71625416 Ki = 6 nM T49031 C6YL0H 71655218 IC50 = 38 nM T49031 CJ2B4Q 71655219 IC50 = 90 nM T49031 C58CEL 71655220 IC50 = 14 nM T49031 C4E2RB 71655221 IC50 = 5.7 nM T49031 C32PIH 71655289 IC50 = 35 nM T49031 C6BSW5 71655290 IC50 = 130 nM T49031 C19VOE 71655291 IC50 = 200 nM T49031 C6ZCI2 71655292 IC50 = 63 nM T49031 C7BIM2 71655353 IC50 = 29 nM T49031 CY78WU 71655354 IC50 = 230 nM T49031 C5H0IP 71655355 IC50 = 210 nM T49031 CW0Y5L 71655356 IC50 = 130 nM T49031 C8G6CQ 71655357 IC50 = 60 nM T49031 C2B4FJ 71655358 IC50 = 33 nM T49031 C1RYA4 71655419 IC50 = 300 nM T49031 C42YSR 71655420 IC50 = 57 nM T49031 CS3OP6 71655421 IC50 = 41 nM T49031 C7EW4B 71655422 IC50 = 47 nM T49031 C63MDL 71655423 IC50 = 30 nM T49031 CHCW60 71655482 IC50 = 28 nM T49031 C1Z7FJ 71655483 IC50 = 230 nM T49031 CZ0B7D 71655484 IC50 = 79 nM T49031 C75FOB 71655485 IC50 = 25 nM T49031 CQR98T 71655486 IC50 = 10 nM T49031 CM9U4L 71655547 IC50 = 77 nM T49031 CBMY45 71697266 Ki = 1620 nM T49031 CC1EV9 71697268 Ki = 260 nM T49031 CPW74Y 71697269 Ki = 800 nM T49031 CL0Q1G 71697270 Ki = 1450 nM T49031 CX1R7P 71697360 Ki = 300 nM T49031 C69BUX 71697361 Ki = 98 nM T49031 C2X5UT 71697363 Ki = 5900 nM T49031 C0UPY7 71697364 Ki = 440 nM T49031 C92HCM 71697365 Ki = 1340 nM T49031 CIPT74 71697366 Ki = 170 nM T49031 CJ52KP 71717087 Ki = 2.3 nM T49031 C7FLM2 72724741 IC50 = 50 nM T49031 CC65XM 72724804 IC50 = 28 nM T49031 C5IX8L 72724805 EC50 = 332 nM T49031 CK41SO 72724806 IC50 = 330 nM T49031 CR4A1Z 72724807 IC50 = 500 nM T49031 CJG3W2 73897219 IC50 = 63340 nM T49031 C0ER9W 74538726 IC50 = 5700 nM T49031 C1IN8Q 76310070 IC50 = 3380 nM T49031 CNYC80 76313773 IC50 = 1040 nM T49031 C0LU1D 76317291 IC50 = 900 nM T49031 C0U3XB 76317292 IC50 > 10000 nM T49031 CX6O8P 76317293 IC50 > 10000 nM T49031 CF8B7J 76320989 IC50 > 10000 nM T49031 CON57Y 76320990 IC50 > 10000 nM T49031 C3H2UI 76320991 Ki = 1100 nM T49031 CZO5L9 76320992 IC50 = 1660 nM T49031 C9P2HW 76320993 IC50 = 1650 nM T49031 CX5H3D 76320994 IC50 = 670 nM T49031 CP7R9O 76320995 IC50 = 1940 nM T49031 C1U5JY 76328224 IC50 = 1370 nM T49031 CN48JG 76328225 IC50 = 2190 nM T49031 CB89NY 76328226 IC50 = 800 nM T49031 CCF2T7 76328227 IC50 = 750 nM T49031 C4MAE1 76335476 IC50 = 580 nM T49031 CL30YE 76335477 IC50 = 2700 nM T49031 CG5E8R 76335478 IC50 > 10000 nM T49031 CV3S5J 76335479 IC50 = 1570 nM T49031 C4C2HT 76335480 IC50 = 1460 nM T49031 CQAL89 76335481 IC50 = 1660 nM T49031 CGY43C 78425867 IC50 = 2670 nM T49031 C0WA1V 86290925 Ki = 10260 nM T49031 C6FVI5 86302567 Ki = 560 nM T49031 C4T2MX 86302568 Ki = 330 nM T49031 CH1AU3 86302591 Ki = 1480 nM T49031 CNK78C 86302666 Ki = 0.14 nM T49031 CQLZ84 90381790 Ki = 39213 nM T49031 C0U9JN 90645047 Ki = 57 nM T49031 C9VK0E 90645048 Ki = 490 nM T49031 C8K2VQ 90645050 Ki = 85 nM T49031 CEN72L 90645051 Ki = 53 nM T49031 C4RAD1 90645052 Ki = 60 nM T49031 CJH69O 90645053 Ki = 4570 nM T49031 C54TGH 90645054 Ki = 80 nM T49031 C1EB8U 90645055 Ki = 2340 nM T49031 CFPT98 90655054 IC50 = 140 nM T49031 C5JZ8R 90655055 IC50 = 280 nM T49031 C3DWJ2 90655129 Ki = 8030 nM T49031 C5Z8EX 90655130 Ki = 10100 nM T49031 C6C2HX 90655131 Ki = 7670 nM T49031 C24PAH 90655132 Ki = 1450 nM T49031 CIXL21 90655133 Ki = 300 nM T49031 C2X7HV 90665951 IC50 > 1000 nM T49031 CRH4M3 90665952 IC50 > 1000 nM T49031 C5ZA4B 90665953 IC50 = 910 nM T49031 CPJ21F 90665954 IC50 = 50 nM T49031 C3KRH8 90665955 IC50 = 25 nM T49031 C1BA4E 90665956 IC50 = 12 nM T49031 CY80KV 90665957 IC50 = 8.4 nM T49031 CA48LV 90665958 IC50 = 5.4 nM T49031 CYB86O 90665959 IC50 = 22 nM T49031 CW8MS4 90665960 IC50 = 6.8 nM T49031 CQ67SO 90665961 IC50 = 4.8 nM T49031 CN94OJ 90665962 IC50 = 4.7 nM T49031 C2K9LZ 90665963 IC50 = 12 nM T49031 C81TAL 90665964 IC50 = 4 nM T49031 CP5S0X 90665965 IC50 = 3 nM T49031 C8IVK5 90665966 IC50 = 11 nM T49031 C7DL5F 90665967 IC50 = 3.7 nM T49031 C78ZBE 90665968 IC50 = 4 nM T49031 C2AG7C 90665969 IC50 = 3.9 nM T49031 C10CYW 90665970 IC50 = 1.1 nM T49031 CHBL08 90665971 IC50 = 940 nM T49031 CVZO36 90665972 IC50 = 22.6 nM T49031 C5EN3W 90665973 IC50 = 16 nM T49031 C62YEW 90665974 IC50 = 23 nM T49031 CF20ZD 90665975 IC50 = 160 nM T49031 CQE72G 90665976 IC50 = 7.3 nM T49031 CYF9H8 90665977 IC50 = 11.6 nM T49031 CJB32F 98103582 Ki = 17500 nM T49031 CG1IY3 98473743 Ki = 2350 nM T49031 C8NM0U 101553172 Ki = 2120 nM T49031 CG0N1O 101874275 IC50 = 16 nM T49031 CZX37E 102160215 IC50 = 14400 nM T49031 CVC0L7 102236951 IC50 = 93600 nM T49031 CXUQ14 102236952 IC50 = 31900 nM T49031 CHR18W 102579879 IC50 = 23600 nM T49031 C9C5OZ 117607839 IC50 = 782 nM T49031 C9BZ6E 117607841 IC50 = 185 nM T49031 CLHS74 117607901 IC50 = 926 nM T49031 CW9R0U 117607904 IC50 = 688 nM T49031 CKPU97 117607978 IC50 = 6630 nM T49031 C7QST8 117611788 IC50 = 6894 nM T49031 C2QDO6 117611839 IC50 = 54 nM T49031 CO1HJ9 117611880 IC50 = 18226 nM T49031 CZ6C1M 117611892 IC50 = 3620 nM T49031 C9YH1X 117611941 IC50 = 42468 nM T49031 C29AKS 118717990 IC50 = 0.38 nM T49031 CU4O3M 118718077 IC50 = 0.4 nM T49031 CS16DB 118718078 IC50 = 0.22 nM T49031 CK6E3L 118718085 IC50 = 0.34 nM T49031 CRZY67 118736272 IC50 = 290 nM T49031 CPY1S2 118736273 IC50 = 920 nM T49031 C2HWT3 118736382 IC50 = 17190 nM T49031 CY0VM1 118736383 IC50 = 12970 nM T49031 C6X0GY 118736384 IC50 = 13880 nM T49031 CS50HX 118736385 IC50 = 17310 nM T49031 C80ROJ 118736389 IC50 = 660 nM T49031 CIJ3E0 118736391 IC50 = 1630 nM T49031 CYO8P5 118736392 IC50 = 11730 nM T49031 C1DP4N 118899141 IC50 = 76000 nM T49031 CUH45I 118899149 IC50 = 78200 nM T49031 CA83ML 118899158 IC50 = 74870 nM T49031 C7YGZ8 122177663 IC50 = 360 nM T49031 CR80CE 122177664 IC50 = 930 nM T49031 CO0E6T 122189322 Ki = 3231 nM T49031 CG3U9I 122189323 Ki = 743.4 nM T49031 CM68CG 122189324 Ki = 7575 nM T49031 CWN52G 122189325 Ki = 906.2 nM T49031 CH08QC 122189326 Ki = 591.6 nM T49031 CSWG38 122189327 Ki = 951.9 nM T49031 C2ZJK1 122189328 Ki = 2113 nM T49031 CP7I6J 122189329 Ki = 963.1 nM T49031 CY7O0G 122189330 Ki = 1237 nM T49031 CO9E8A 122189331 Ki = 2347 nM T49031 CK7UV3 122189332 Ki = 1140 nM T49031 C8E7MQ 122189333 Ki = 1711 nM T49031 CI46QN 122189334 Ki = 949.8 nM T49031 CZ6LS4 122189335 Ki = 447 nM T49031 CZSI84 122189336 Ki = 385.2 nM T49031 C0OLW2 122204528 IC50 = 900 nM T49031 C90BKO 122520041 IC50 < 10 nM T49031 C3P0QD 122576697 IC50 = 220 nM T49031 C17FZG 127027248 IC50 = 26.24 nM T49031 C0DW3P 127027565 IC50 = 42.61 nM T49031 C6OVL9 127028490 IC50 = 49.5 nM T49031 CCF5E4 127028491 IC50 = 120.2 nM T49031 CV6JZ1 127028492 IC50 = 471 nM T49031 CO4D8I 127028814 IC50 = 24547089.16 nM T49031 C1Y9BP 127028815 IC50 = 3.34 nM T49031 CLB70K 127029400 IC50 = 8.32 nM T49031 C3FR6D 127029685 IC50 = 25.02 nM T49031 C6A1GD 127029686 IC50 = 4.6 nM T49031 CI6S1K 127030040 IC50 = 8.46 nM T49031 C4X7CO 127030041 IC50 = 2.34 nM T49031 C3LRH9 127030042 IC50 = 2.73 nM T49031 CAB69Z 127030043 IC50 = 16.4 nM T49031 CA50HP 127030044 IC50 = 114 nM T49031 C8DA4P 127030315 IC50 = 295120922.7 nM T49031 CQV32H 127030316 IC50 = 1.16 nM T49031 CI6P8J 127030317 IC50 = 1.15 nM T49031 CXQ69J 127030318 IC50 = 6.96 nM T49031 CQJ7F3 127030635 IC50 = 0.76 nM T49031 CZH53T 127030636 IC50 = 1.34 nM T49031 CO7WC6 127030637 IC50 = 2.46 nM T49031 CU0BJ3 127030638 IC50 = 862978547.8 nM T49031 C6Y2XQ 127031260 IC50 = 4.69 nM T49031 CJL9I1 127032443 IC50 = 1.02 nM T49031 CK3BX6 127032447 IC50 = 6.31 nM T49031 CI8RZ2 127032448 IC50 = 8.47 nM T49031 CV76UR 127032449 IC50 = 6.94 nM T49031 CVQ04L 127032450 IC50 = 4.82 nM T49031 CL36HN 127045979 IC50 = 26050 nM T49031 CI7H5T 127045980 IC50 = 23050 nM T49031 CIVH08 127045981 IC50 = 21540 nM T49031 C4ZG2O 127045982 IC50 = 16140 nM T49031 CWN9X5 127046160 IC50 = 14230 nM T49031 CUK8M7 127046161 IC50 = 13760 nM T49031 C4CAH2 127046162 IC50 = 13340 nM T49031 CDR54T 127047437 IC50 = 10250 nM T49031 CNL84P 127047438 IC50 = 17630 nM T49031 C3G7FU 127047439 IC50 = 9880 nM T49031 CED9T0 127047850 IC50 = 11860 nM T49031 C8QSW1 127048158 IC50 = 13800 nM T49031 CD51BP 127048159 IC50 > 25000 nM T49031 CP59LC 127048521 IC50 = 7800 nM T49031 CSLW65 127048522 IC50 > 25000 nM T49031 CADQ63 127048523 IC50 = 18700 nM T49031 C2A0UO 127048524 IC50 = 2300 nM T49031 CX65VA 127048525 IC50 = 21600 nM T49031 C5TS0O 127048526 IC50 > 25000 nM T49031 C3SY6Q 127049154 IC50 = 7600 nM T49031 CE5VT0 127049164 IC50 > 25000 nM T49031 CG9XP1 127049501 IC50 > 25000 nM T49031 CKYV35 127049817 IC50 > 25000 nM T49031 CVY2Q6 127049838 IC50 = 6300 nM T49031 CNX36Z 127049839 IC50 = 5600 nM T49031 COH67Z 127049840 IC50 = 9100 nM T49031 C1B4PE 127049841 IC50 = 5260 nM T49031 CJM29H 127049842 IC50 > 25000 nM T49031 CZIV95 127049843 IC50 = 15600 nM T49031 CDX7J4 127049844 IC50 = 5500 nM T49031 C3JE8G 127049845 IC50 = 6700 nM T49031 CEU1Y3 127050799 IC50 = 19200 nM T49031 CAS65J 127051646 IC50 = 8200 nM T49031 CLU6P9 127051647 IC50 > 25000 nM T49031 C9BFA0 127051648 IC50 > 25000 nM T49031 CMW2S6 127051649 IC50 > 25000 nM T49031 CE25WX 127051650 IC50 = 9900 nM T49031 C5REY7 127051651 IC50 > 25000 nM T49031 C4QXW2 127051652 IC50 > 25000 nM T49031 CL4N3G 127051653 IC50 = 8500 nM T49031 CFC43I 127052871 IC50 = 6100 nM T49031 C8AUE5 127053172 IC50 = 19900 nM T49031 C4YV1I 127053228 IC50 = 208929613.1 nM T49031 CPB1J8 127053229 IC50 = 3.21 nM T49031 CZR14W 127053267 IC50 = 4.18 nM T49031 CX53LM 127053268 IC50 = 1.12 nM T49031 CW3L9P 127053269 IC50 = 5.17 nM T49031 C6W2RO 127053272 IC50 = 524807460.3 nM T49031 C3AZ9G 127053273 IC50 = 5.24 nM T49031 CU8NW9 127053274 IC50 = 6.7 nM T49031 C4O6VG 127053280 IC50 = 162181009.7 nM T49031 C98AVC 127053285 IC50 = 1.26 nM T49031 CH2EP6 127053293 IC50 = 39 nM T49031 C3IVZ5 127053294 IC50 = 14.2 nM T49031 CDS47Y 127053295 IC50 = 17.2 nM T49031 CI2U8S 127053300 IC50 = 3.67 nM T49031 CQ6YW0 127053301 IC50 = 1.46 nM T49031 CT96PH 129047769 IC50 = 1140 nM T49031 CI24DQ 129047778 IC50 = 409 nM T49031 CI2J8F 129047830 IC50 = 110 nM T49031 C7BGS2 129047963 IC50 = 960 nM T49031 C4FRX1 132501288 IC50 = 26300 nM T49031 C34DQH 132501408 IC50 = 18500 nM T49031 CSP91A 132501468 IC50 = 5300 nM T49031 C1IFJ2 132501469 IC50 > 100000 nM T49031 CUT65O 132503175 IC50 = 370 nM T49031 CTQ8E6 132528967 IC50 = 2.4 nM T49031 CFB4V6 132528968 IC50 = 3 nM T49031 CM34ST 132528969 IC50 = 1.4 nM T49031 C5ZWQ8 132528970 IC50 = 4.3 nM T49031 C3WLQ2 134134387 IC50 = 15.7 nM T49031 CLM6F9 134134689 IC50 = 45.7 nM T49031 C5JS7V 134138393 IC50 = 669.9 nM T49031 CJ8ZN5 134139145 Ki = 420 nM T49031 C63QWU 134141164 IC50 = 16.9 nM T49031 C3EKC0 134142355 IC50 = 343.9 nM T49031 CEF0U1 134144291 IC50 = 601.4 nM T49031 CH9PI2 134146604 IC50 = 14.7 nM T49031 C8GH5D 134155148 IC50 = 152.9 nM T49031 C2Z5NM 134155499 Ki = 10980 nM T49031 C3K5UI 134155758 IC50 = 16.6 nM T49031 CH4XU1 134156052 IC50 = 23.7 nM T49031 C52IBY 134823859 IC50 = 394.2 nM T49031 C8VHK7 137632080 IC50 = 2710 nM T49031 CQO35X 137632519 IC50 = 2 nM T49031 CVSF43 137632662 IC50 = 25.7 nM T49031 C2NC9L 137633752 IC50 = 2180 nM T49031 CN78FJ 137633908 IC50 = 50 nM T49031 C08FKI 137634357 IC50 = 75 nM T49031 C3JI7B 137634520 IC50 = 5.5 nM T49031 CEJO70 137634807 IC50 = 510 nM T49031 CM3G2X 137635261 IC50 = 22160 nM T49031 CGPH59 137635270 IC50 > 1000 nM T49031 C40KOA 137635653 IC50 = 0.6 nM T49031 C64VSP 137636270 IC50 = 22290 nM T49031 C3H9XJ 137636488 IC50 = 41 nM T49031 CQP57Z 137636959 IC50 = 1 nM T49031 C3U2JC 137637883 IC50 > 50000 nM T49031 CW8D3F 137638026 IC50 = 197 nM T49031 C1HIY2 137638305 IC50 = 6.6 nM T49031 CNYU52 137639027 IC50 = 1.1 nM T49031 CZO8K2 137639142 IC50 = 5840 nM T49031 CNE56R 137639426 IC50 = 740 nM T49031 C0JQF2 137639470 IC50 = 39400 nM T49031 CG8V1S 137639601 IC50 = 3.8 nM T49031 CMK7O5 137639868 IC50 > 50000 nM T49031 CMSA73 137639962 IC50 = 260 nM T49031 C1KN9L 137640079 IC50 = 510 nM T49031 CVAK38 137640137 IC50 = 0.3 nM T49031 CB94IM 137640658 IC50 = 19600 nM T49031 CNVZ89 137640673 IC50 = 500 nM T49031 CIJ6E3 137640968 IC50 > 1000 nM T49031 C0B1FH 137641544 IC50 = 192.5 nM T49031 C6DF7U 137641807 IC50 > 1000 nM T49031 C0GWD7 137641958 IC50 = 10 nM T49031 CO1L4N 137642007 IC50 = 21.8 nM T49031 CH09CN 137642553 IC50 = 0.0002 nM T49031 C6DJF3 137642709 IC50 = 168 nM T49031 C3AEP5 137642951 IC50 = 99 nM T49031 CSXN16 137643018 IC50 = 44.25 nM T49031 CE0J4N 137643562 IC50 = 7 nM T49031 C0EY3T 137643629 IC50 = 2430 nM T49031 CB85DX 137643715 IC50 = 11.42 nM T49031 CJ6Z5F 137645427 IC50 > 1000 nM T49031 CL09KP 137645698 IC50 = 10 nM T49031 CEB8L5 137646135 IC50 > 50000 nM T49031 C5NF8R 137647268 IC50 = 90 nM T49031 CWOY74 137647871 IC50 = 1380 nM T49031 CC9R2E 137647922 IC50 = 2.6 nM T49031 C0KYZ2 137648206 IC50 = 237 nM T49031 CSF5N6 137648399 IC50 = 10.8 nM T49031 CNA75Z 137648431 IC50 = 8830 nM T49031 C7NYD8 137649498 IC50 > 1000 nM T49031 C19DEP 137649562 IC50 = 1360 nM T49031 C58EXC 137650165 IC50 = 200 nM T49031 CU9EK0 137650556 IC50 = 8.6 nM T49031 C7BUK5 137650655 IC50 = 12 nM T49031 CQ5AJ9 137650783 IC50 = 1.2 nM T49031 C7QW9D 137650914 IC50 = 57 nM T49031 C09QJA 137650983 IC50 = 1 nM T49031 C2NYK9 137651187 IC50 = 3 nM T49031 CCWZ51 137651207 IC50 = 20 nM T49031 CDQ41W 137651497 IC50 = 19.7 nM T49031 C04AZG 137651667 IC50 = 4 nM T49031 C57ZKC 137652515 IC50 = 182 nM T49031 C7R4DB 137653941 IC50 = 22 nM T49031 C8XLU1 137654027 IC50 = 29030 nM T49031 CGSU61 137654406 IC50 = 11.6 nM T49031 C2QMK8 137654413 IC50 = 40 nM T49031 CT08DG 137654519 IC50 = 1.5 nM T49031 CDAE50 137655349 IC50 = 23.17 nM T49031 CUC26W 137655738 IC50 = 20 nM T49031 CV8P6O 137656187 IC50 > 50000 nM T49031 CHV31Y 137656315 IC50 = 3570 nM T49031 CTA1F2 137656425 IC50 = 67 nM T49031 C90JMU 137656505 IC50 = 0.7 nM T49031 CSZ1A5 137657170 IC50 = 2.9 nM T49031 C1Y9RS 137657408 IC50 = 660 nM T49031 C5N2CB 137657727 IC50 > 1000 nM T49031 CNM6C4 137657944 IC50 > 1000 nM T49031 CJU5K7 137658335 IC50 = 110 nM T49031 CNFP69 137658811 IC50 = 2710 nM T49031 C3XE0H 137659182 IC50 = 0.9 nM T49031 CUFT31 137659572 IC50 = 17 nM T49031 CY6A3Q 137659779 IC50 = 18 nM T49031 C9CQ4N 137659903 IC50 = 25.93 nM T49031 CJQ6B7 137659959 IC50 = 3390 nM T49031 CY1S6E 137660489 IC50 = 24.58 nM T49031 C4BMO7 137660514 IC50 = 2 nM T49031 C8MH9V 137660779 IC50 = 18 nM T49031 CL1G7H 137661189 IC50 = 2.4 nM T49031 C01KBD 137661456 IC50 = 570 nM T49031 C1R9BC 137661627 IC50 = 13.3 nM T49031 CI96SM 137661745 IC50 = 1970 nM T49031 C1JH8K 138545006 IC50 > 100000 nM T49031 CLT78F 138545112 IC50 > 100000 nM T49031 C7DZ8K 138545235 IC50 > 100000 nM T49031 C5DJC6 138545265 IC50 = 10000 nM T49031 CIS28V 139209090 IC50 = 1412 nM T49031 CB46AI 139209092 IC50 > 100000 nM T49031 CMNL75 145960420 IC50 = 9.7 nM T49031 CL45BO 145960456 IC50 = 140000 nM T49031 C1W6TO 145960482 IC50 = 92 nM T49031 C0YF7Z 145960612 IC50 = 109 nM T49031 CU1EV5 145960693 IC50 = 126 nM T49031 C01WBE 145960929 IC50 = 335 nM T49031 C5G6LM 145961320 IC50 = 8900 nM T49031 C96AIF 145961391 IC50 > 100000 nM T49031 CI9QB0 145961558 IC50 = 210 nM T49031 CUIF27 145961566 IC50 = 10000 nM T49031 CQE07I 145961835 IC50 = 166 nM T49031 CI9JH6 145961877 IC50 = 6700 nM T49031 C3M4OD 145961898 IC50 = 18000 nM T49031 CBI7V1 145962019 IC50 = 27800 nM T49031 CN1I2C 145962168 IC50 = 69000 nM T49031 C8CSZ0 145962247 IC50 = 125000 nM T49031 CMD9X7 145962389 IC50 = 53 nM T49031 CVEF93 145962537 IC50 = 39000 nM T49031 C35NPT 145962676 IC50 = 192 nM T49031 C97URS 145962850 IC50 = 950 nM T49031 CVB9A4 145963178 IC50 = 36 nM T49031 CPA60M 145963188 IC50 = 65 nM T49031 CM95CN 145963260 IC50 = 155 nM T49031 CUL94O 145963403 IC50 = 275 nM T49031 COA19G 145963426 IC50 > 100000 nM T49031 C2LEB3 145963518 IC50 = 67000 nM T49031 CS6I8T 145964202 IC50 > 8000 nM T49031 CJ3Q5B 145964538 IC50 = 890 nM T49031 CKAS15 145964962 IC50 = 1100 nM T49031 CO83HL 145965095 IC50 > 8000 nM T49031 C15VCH 145966003 IC50 > 8000 nM T49031 C3L5IP 145966472 IC50 = 6300 nM T49031 C40QHP 145969617 IC50 > 8000 nM T49031 CV5NU9 145974241 IC50 = 2100 nM T49031 CQ42KP 145974420 IC50 > 8000 nM T49031 CRUD43 145974971 IC50 = 6100 nM T49031 CZ8H4Y 145975867 IC50 = 370 nM T49031 C38NRV 145976554 IC50 > 8000 nM T49031 CK2B4J 145978094 IC50 = 890 nM T49031 C9BWP4 145979302 IC50 = 2130 nM T49031 CN79HG 145979487 IC50 = 2800 nM T49031 CODE68 145979676 IC50 = 11.6 nM T49031 CEI3U1 145979850 IC50 = 4300 nM T49031 C24WEG 145980281 IC50 = 8.2 nM T49031 CIZU61 145980473 IC50 = 9.8 nM T49031 C35BOY 145980635 IC50 = 7.8 nM T49031 C69MQC 145980644 IC50 = 8.8 nM T49031 C07EJK 145980652 IC50 = 5.7 nM T49031 C5AYC4 145980811 IC50 = 64000 nM T49031 CG6UL0 145980995 IC50 = 1740 nM T49031 C2XPD3 145981337 IC50 = 2.7 nM T49031 C21VNK 145981642 IC50 = 22.8 nM T49031 CB67YT 145981691 IC50 = 1480 nM T49031 C41IRV 145981707 IC50 = 350 nM T49031 C5L8JM 145981943 IC50 = 12.9 nM T49031 CE94FB 145982013 IC50 = 7.7 nM T49031 C4UVP5 145982479 IC50 = 10.2 nM T49031 CLO3P1 145982669 IC50 = 74.86 nM T49031 C4B2NC 145982840 IC50 = 3.53 nM T49031 CL1F8N 145982922 IC50 = 28700 nM T49031 CGB54U 145983051 IC50 = 8.21 nM T49031 CQF0E2 145983505 IC50 = 4.16 nM T49031 CFE52X 145983530 IC50 = 27.75 nM T49031 C7SKN2 145983622 IC50 = 30.78 nM T49031 CG9LA8 145983719 IC50 = 5.89 nM T49031 C7WD8V 145983830 IC50 = 26.79 nM T49031 CSV4F0 145983965 IC50 = 20.44 nM T49031 C8WRQ7 145984091 IC50 = 21.17 nM T49031 C2UV4N 145984105 IC50 = 8.86 nM T49031 CPK4C5 145984357 IC50 = 4.82 nM T49031 C62OHN 145984529 IC50 = 5.26 nM T49031 CQ30LY 145984824 IC50 = 6.74 nM T49031 CF5R2L 145984944 IC50 = 3.22 nM T49031 CNZ16R 145985009 IC50 = 8.11 nM T49031 C16JLE 145985104 IC50 = 1.98 nM T49031 CVZ10A 145985697 IC50 = 42.79 nM T49031 C9G2VJ 145985757 IC50 = 387 nM T49031 C07VUG 145985780 IC50 = 2.31 nM T49031 C69VIS 145985988 IC50 = 593.7 nM T49031 CXBR78 145986043 IC50 = 12.89 nM T49031 C5X3GQ 145986425 IC50 = 6200 nM T49031 CRZE86 145986857 IC50 = 5100 nM T49031 CAJ5K8 145986961 IC50 = 3.6 nM T49031 CIB5Z9 145986993 IC50 = 5 nM T49031 CHWT73 145987085 IC50 = 6800 nM T49031 CM3H4F 145987197 IC50 = 2900 nM T49031 CNZ7R6 145987536 IC50 = 9200 nM T49031 CYBN31 145987734 IC50 = 835 nM T49031 C1EF3B 145988020 IC50 = 7.1 nM T49031 CM1U6F 145988104 IC50 = 15.9 nM T49031 CQIS01 145988427 IC50 = 6000 nM T49031 C4R3HC 145988596 IC50 = 7 nM T49031 CQ7W9S 145988601 IC50 = 13.2 nM T49031 CMW7U5 145989009 IC50 = 35.9 nM T49031 CN8K1E 145989337 IC50 = 3.1 nM T49031 CE16JH 145989568 IC50 = 113 nM T49031 CON2B3 145989641 IC50 = 7.7 nM T49031 CF3OZ9 145989730 IC50 = 18.7 nM T49031 CXG30R 145990249 IC50 = 11300 nM T49031 CWS03B 145991519 IC50 = 9.4 nM T49031 C8G1BT 145991875 IC50 = 10000 nM T49031 C8IL9E 145992200 IC50 = 5100 nM T49031 CBY18W 145992498 IC50 = 1400 nM T49031 CCU34H 145992780 IC50 = 360 nM T49031 C6GHQ9 145993211 IC50 = 22000 nM T49031 C2Q8BT 145993325 IC50 = 7.6 nM T49031 CVN3A5 145993374 IC50 = 6.6 nM T49031 CEVY70 145993649 IC50 = 880 nM T49031 CC24LD 145993770 IC50 = 19.7 nM T49031 CJO08K 145993925 IC50 = 125 nM T49031 C1UC2Z 147001460 IC50 = 77.1 nM T49031 CES1Y7 147009690 IC50 = 52.2 nM T49031 CYUM75 147335182 IC50 = 36.8 nM T49031 CSK1A5 147672609 IC50 = 4.6 nM T49031 CDX0I3 149045896 IC50 = 729 nM T49031 C1YFV0 155510465 IC50 < 10 nM T49031 CX74UV 155510547 IC50 < 10 nM T49031 C2AW9L 155510675 IC50 = 37 nM T49031 CLHB15 155510759 IC50 = 14 nM T49031 C4FH8S 155512766 IC50 = 48.3 nM T49031 C7J5BO 155512794 IC50 = 41.5 nM T49031 CZXI74 155513137 IC50 = 32 nM T49031 CL7I6A 155513548 IC50 = 30.8 nM T49031 C6IB7G 155513571 IC50 = 9 nM T49031 CY56QN 155514326 IC50 = 952 nM T49031 C5J0OF 155514653 IC50 = 253 nM T49031 C8E6ZX 155514792 IC50 = 1400 nM T49031 C0SDO2 155515259 IC50 = 230 nM T49031 CX76LO 155515463 IC50 = 34 nM T49031 CGW2M6 155516032 IC50 > 100000 nM T49031 C53ZEN 155516179 IC50 > 10000 nM T49031 CM3BV8 155516620 IC50 > 100000 nM T49031 CHU0Q9 155516696 IC50 = 111 nM T49031 C4VT1Y 155517101 IC50 = 430 nM T49031 C2BCH9 155517229 IC50 = 248 nM T49031 C6I7SU 155517529 IC50 = 154 nM T49031 CJ6ZU4 155517550 IC50 > 1000 nM T49031 CCB58J 155517652 IC50 = 481 nM T49031 CE95IQ 155518158 IC50 > 100000 nM T49031 CFQZ35 155518266 IC50 = 1410 nM T49031 CW8Z7I 155518578 IC50 = 8100 nM T49031 C5ATN1 155519023 IC50 = 232 nM T49031 C2OQU6 155519126 IC50 > 100000 nM T49031 CEF5D1 155519196 IC50 > 100000 nM T49031 C7FP0V 155519306 IC50 = 395 nM T49031 C5B4HU 155519323 IC50 = 14 nM T49031 CEJ56T 155519405 IC50 = 6700 nM T49031 CH9R4W 155520688 IC50 = 54 nM T49031 COL16B 155520712 IC50 = 8 nM T49031 C4WO3N 155521110 IC50 = 392 nM T49031 CNM0Q9 155521286 IC50 > 10000 nM T49031 CD4OH3 155521410 IC50 = 56 nM T49031 C0S4TP 155521499 IC50 = 30.6 nM T49031 CZKF54 155521690 IC50 = 1300 nM T49031 C8NOH2 155521815 IC50 = 6040 nM T49031 CJZT01 155522109 IC50 = 952 nM T49031 CTDK64 155522147 IC50 = 480 nM T49031 CN60CL 155522148 IC50 = 243 nM T49031 CB0WG8 155522381 IC50 = 2.1 nM T49031 C73DYM 155522560 IC50 = 5907 nM T49031 CQ3OD0 155522579 IC50 = 116 nM T49031 C8GNQ9 155522828 IC50 = 486 nM T49031 CM7ZA2 155523065 IC50 = 99 nM T49031 CW75YK 155523151 IC50 > 100000 nM T49031 CY3UP7 155523507 IC50 = 405 nM T49031 CL0IQ3 155523963 IC50 = 25.5 nM T49031 C94IEH 155524612 IC50 = 922 nM T49031 CZP1E6 155524975 IC50 = 30 nM T49031 CIP3E9 155526380 IC50 = 460 nM T49031 C5R3PX 155526504 Ki = 17 nM T49031 C78BVM 155526764 IC50 = 1130 nM T49031 CVJ70O 155526910 IC50 = 1561 nM T49031 CAC34Y 155527225 IC50 = 1800 nM T49031 COMG30 155527377 IC50 = 579 nM T49031 C6OC8R 155527614 IC50 = 836 nM T49031 CPHX68 155527880 IC50 = 1.5 nM T49031 CWZ17S 155528412 IC50 = 67 nM T49031 CROM71 155528428 IC50 = 436 nM T49031 C3PMD9 155529033 IC50 = 506 nM T49031 CW3G4Z 155529142 IC50 = 920 nM T49031 CCW71B 155529960 IC50 = 100 nM T49031 CYW5R1 155530452 IC50 > 100000 nM T49031 C2MW8Q 155530743 IC50 > 100000 nM T49031 CUP2B4 155531358 IC50 = 39 nM T49031 CIL2D0 155531506 IC50 = 51 nM T49031 CD84AS 155531896 IC50 = 40190 nM T49031 C9SH6Q 155532346 IC50 = 352 nM T49031 CLE8N1 155532865 IC50 = 660 nM T49031 CL9A0E 155532989 IC50 = 20.6 nM T49031 CK28QW 155533771 IC50 = 20 nM T49031 C2TR0X 155533978 IC50 = 50210 nM T49031 CEF08Q 155534115 IC50 > 100000 nM T49031 C9ODL6 155534328 IC50 = 968 nM T49031 CH9GO0 155534453 IC50 = 56.5 nM T49031 CG5E2L 155534840 IC50 = 16 nM T49031 C72EIY 155535051 IC50 = 89 nM T49031 C5G9LX 155535238 IC50 = 113 nM T49031 COZ5V6 155535430 IC50 = 46600 nM T49031 CT3A0N 155536062 IC50 = 14 nM T49031 C20BYW 155536148 Ki = 10.1 nM T49031 C9IL7E 155536781 IC50 = 38.8 nM T49031 C7O0SH 155537082 IC50 = 1111 nM T49031 CP7D4R 155537435 IC50 = 26.8 nM T49031 CCYI81 155537845 IC50 = 29370 nM T49031 C3EF7U 155538548 IC50 = 100 nM T49031 C2S5HL 155538665 IC50 = 52.1 nM T49031 C2NTI6 155538936 IC50 > 100000 nM T49031 CW5U4H 155539000 IC50 = 64.8 nM T49031 C6E1YP 155539344 IC50 > 100000 nM T49031 C69TOB 155539701 IC50 = 57 nM T49031 CLE9Y6 155539965 IC50 = 280 nM T49031 CT2V8E 155540850 IC50 = 4380 nM T49031 CTM03H 155540978 IC50 = 4726 nM T49031 C6RE8V 155540985 IC50 = 36.6 nM T49031 CQE43H 155541095 IC50 > 100000 nM T49031 C0T3CO 155541137 IC50 = 139.6 nM T49031 CNZ5B4 155541377 IC50 = 2000 nM T49031 C6OIY3 155541618 IC50 > 100000 nM T49031 C42XMS 155542291 IC50 = 3 nM T49031 C1K6NV 155542487 IC50 = 259 nM T49031 C41IBR 155542489 IC50 = 2200 nM T49031 CRU73P 155542979 Ki = 4.8 nM T49031 CHJY08 155543004 IC50 > 10000 nM T49031 CH92PY 155543085 IC50 = 1682 nM T49031 CH6X3Q 155543527 IC50 = 26 nM T49031 CTL46N 155543581 IC50 = 64 nM T49031 CB4K6P 155543584 IC50 = 274 nM T49031 C0EG5T 155543676 IC50 < 10 nM T49031 CR7WL1 155544072 IC50 = 35 nM T49031 C13HEG 155544089 IC50 > 10000 nM T49031 CH17XP 155544685 IC50 > 100000 nM T49031 C72ADE 155544797 IC50 = 162.2 nM T49031 CEC78A 155545362 IC50 > 1000 nM T49031 CB4J8F 155545830 IC50 = 162 nM T49031 C7YS2H 155546237 IC50 = 119 nM T49031 C3Q5GS 155546528 IC50 = 17 nM T49031 CV8T2E 155546596 IC50 = 269 nM T49031 C2R3FM 155546808 IC50 = 111.6 nM T49031 C0V4GT 155547050 IC50 = 2 nM T49031 CKY05M 155547055 IC50 = 37090 nM T49031 CBG9C3 155547430 IC50 = 98.2 nM T49031 CNS2J4 155548060 IC50 < 10 nM T49031 CQ0Z4K 155548281 IC50 = 35 nM T49031 C1LJ0G 155548285 IC50 = 257 nM T49031 CA8Z7D 155548324 IC50 = 9120 nM T49031 C8HVD1 155548349 IC50 > 100000 nM T49031 CZB82L 155548494 IC50 = 370 nM T49031 CC5H7R 155548878 IC50 > 100000 nM T49031 C8JC4L 155548940 IC50 = 50 nM T49031 CK4Q0J 155548955 IC50 = 3863 nM T49031 CX27NO 155549084 IC50 > 100000 nM T49031 CP7FQ0 155549178 IC50 > 1000 nM T49031 CIM5K2 155549227 IC50 = 39000 nM T49031 CH35KO 155550346 IC50 = 36 nM T49031 C12LPX 155551071 IC50 = 29 nM T49031 CRV20J 155551193 IC50 = 25 nM T49031 C6BZ4E 155551617 IC50 = 7 nM T49031 CCKN07 155551785 IC50 = 43.1 nM T49031 CX7P8L 155552184 IC50 = 853 nM T49031 CR7Q8D 155552542 IC50 = 2011 nM T49031 CH93MA 155553025 IC50 = 4.9 nM T49031 CBHM14 155553205 IC50 > 100000 nM T49031 C35NJC 155553210 IC50 = 45300 nM T49031 C2VBQ0 155553272 IC50 = 25 nM T49031 CK9FW3 155553273 IC50 = 60.7 nM T49031 CI15FC 155553565 IC50 = 8600 nM T49031 CVJ3E7 155553910 IC50 = 5000 nM T49031 C0DQC5 155554155 IC50 = 34.1 nM T49031 CDI56O 155554254 IC50 = 37.5 nM T49031 C1AIJ3 155554704 IC50 = 82070 nM T49031 C6YP0L 155554916 IC50 > 100000 nM T49031 C9GE3U 155554982 IC50 > 100000 nM T49031 C2IE7D 155555749 IC50 = 12430 nM T49031 CCI45A 155555926 IC50 = 361 nM T49031 C5SZB7 155556059 IC50 < 10 nM T49031 CJ0QX2 155556352 IC50 > 100000 nM T49031 CP58EH 155556856 IC50 = 26050 nM T49031 CW0K5V 155556875 IC50 < 10 nM T49031 CYJ92G 155557164 IC50 < 10 nM T49031 C6YSC7 155557266 IC50 < 10 nM T49031 C9M1NU 155557790 IC50 = 32 nM T49031 CXCF36 155558612 IC50 = 63 nM T49031 C0Z4ET 155558668 IC50 = 540 nM T49031 CK41QD 155558933 IC50 = 3.8 nM T49031 C5AQM2 155559051 IC50 < 10 nM T49031 CMH7V5 155559237 IC50 > 100000 nM T49031 CR3V7P 155559353 IC50 = 2.1 nM T49031 CT97AU 155559419 IC50 < 10 nM T49031 C7O2KR 155559420 IC50 = 638 nM T49031 CJ5UC9 155560661 IC50 = 33 nM T49031 C2GHS4 155561494 IC50 = 2.1 nM T49031 C98PWZ 155561783 IC50 = 1197 nM T49031 C5OM0U 155561976 IC50 = 12 nM T49031 CZJ52C 155562121 IC50 = 70450 nM T49031 CZXL78 155562443 IC50 = 530 nM T49031 CYB71Z 155563262 IC50 = 18 nM T49031 C2USA4 155563322 IC50 = 166 nM T49031 CZ3XY4 155563335 IC50 > 100000 nM T49031 C9CG3Y 155563835 IC50 = 189 nM T49031 C1UR9Y 155564187 IC50 = 118 nM T49031 CY83KQ 155564232 IC50 < 10 nM T49031 C3N8XZ 155564979 IC50 = 12030 nM T49031 C5YCE8 155565509 IC50 = 4 nM T49031 C0XSM3 155565602 IC50 = 44.9 nM T49031 CEAV80 155566012 IC50 = 5000 nM T49031 CV1L3T 155566407 IC50 > 10000 nM T49031 C7HP0L 155566550 IC50 = 770 nM T49031 CU53FD 155566562 IC50 = 49 nM T49031 CK87TX 155566958 IC50 = 21 nM T49031 C2T7GX 155567492 IC50 < 10 nM T49031 CT23WX 155567596 IC50 < 10 nM T49031 C5Z7YC 155567712 IC50 = 750 nM T49031 CG2KN0 155567727 IC50 > 100000 nM T49031 C7UPT8 155567911 IC50 = 127 nM T49031 CR1NB6 155568111 IC50 = 139 nM T49031 C63DVL 155568157 IC50 = 36.8 nM T49031 CIC1Q5 155568323 IC50 = 50.9 nM T49031 CV68GZ 155568757 IC50 = 1070 nM T49031 CUE8B1 155568787 IC50 = 205 nM T49031 C4ZV3Q 155568941 IC50 > 10000 nM T49031 C1I7QW 155568944 IC50 = 346 nM T49031 CL1QZ7 44583044 IC50 = 9 nM T49031 D00RIX 5280443 IC50 = 1800 nM T49031 D01NCW 11534772 IC50 = 460 nM T49031 D01UYI 5281607 IC50 = 4900 nM T49031 D05MDE 11505372 IC50 = 150000 nM T49031 D05VEV 11556056 IC50 = 120 nM T49031 D06NEB 11693148 IC50 = 35 nM T49031 D08AIJ 440735 IC50 = 14600 nM T49031 D09GZQ 11713852 IC50 = 1300 nM T49031 D09IMK 11621748 IC50 = 3.2 nM T49031 D0A5WN 11621347 IC50 = 2.1 nM T49031 D0B3US 11585523 IC50 = 3300 nM T49031 D0G3TK 5280863 IC50 = 10500 nM T49031 D0I0MU 11534625 IC50 = 69 nM T49031 D0K0KT 11621207 IC50 = 6.1 nM T49031 D0K4PY 114829 IC50 > 100000 nM T49031 D0M7BR 5280378 IC50 > 100000 nM T49031 D0Q4MO 23642227 IC50 = 150 nM T49031 D0QY3R 11513217 IC50 = 24 nM T49031 D0RB1V 6419835 IC50 = 124 nM T49031 D0RL4S 11714476 IC50 = 27 nM T49031 D0SY2M 5281708 IC50 > 100000 nM T49031 D0T3PW 5281672 IC50 = 10000 nM T49031 D0W3ON 416002 IC50 = 600 nM T49031 D0Y3TZ 370 IC50 = 7100000 nM T49031 D0Y6HD 90645049 Ki = 51 nM T00926 D0BP9C 193962 IC50 = 8500 nM T00926 D0K8KX 5280343 Ki = 2400 nM T00926 D0O3OS 104850 Ki = 1400 nM T00926 D0R0FE 2520 EC50 = 1925 nM T00926 D0R1RS 3715 IC50 = 12000 nM T00926 D0R3JB 4212 IC50 = 27.5 nM T00926 D0Z3DY 2333 Ki = 190 nM T00926 D02HTD 25167947 IC50 = 14900 nM T00926 D02QWY 24785538 IC50 = 36300 nM T00926 D0G7UX 5284373 EC50 = 1700 nM T00926 D0O2EF 56946615 IC50 > 100000 nM T00926 D0V7UQ 56946834 IC50 = 2500 nM T00926 D02VJY 3037617 IC50 = 5180 nM T00926 D07GTB 16760063 IC50 = 7570 nM T00926 C52MFS 1756 EC50 = 42000 nM T00926 C8C1JP 72343 IC50 = 38320 nM T00926 C5ZCH7 97332 IC50 = 26350 nM T00926 CL97OF 97548 IC50 = 9860 nM T00926 CA3NK8 193841 EC50 = 5100 nM T00926 CR67FB 243037 EC50 > 100000 nM T00926 CABJ72 276138 IC50 = 1760 nM T00926 CM70RQ 285815 IC50 = 16000 nM T00926 CN8ZL4 298546 EC50 = 45000 nM T00926 C7HME8 439246 Ki = 2400 nM T00926 COI2C9 560674 EC50 = 98000 nM T00926 CTF2J0 687260 EC50 > 100000 nM T00926 CH6MV7 715632 IC50 = 8770 nM T00926 C64RUF 877998 IC50 = 15900 nM T00926 CXR0P5 917533 IC50 = 8800 nM T00926 C7D1QN 921567 EC50 > 100000 nM T00926 CK8TP4 1019287 IC50 > 100000 nM T00926 CL27VW 1069464 IC50 = 3900 nM T00926 CXQ4P8 1183964 IC50 = 8130 nM T00926 CQT4J5 2094802 IC50 > 100000 nM T00926 C1A0FV 2298706 EC50 = 9800 nM T00926 CW6SA0 2787558 IC50 > 100000 nM T00926 C8PN0C 5280682 IC50 = 50000 nM T00926 CNI9X4 5281888 Ki = 600 nM T00926 CPHR19 5325373 EC50 > 100000 nM T00926 CJMT13 5325385 EC50 > 100000 nM T00926 C8VZ9T 5325386 EC50 > 100000 nM T00926 C81ZSW 5325387 EC50 = 85000 nM T00926 CTO51S 5352005 IC50 = 50000 nM T00926 CB2U6E 5467200 IC50 = 1100 nM T00926 C0EM5S 6509849 IC50 = 2800 nM T00926 C32UFI 9828452 IC50 = 61 nM T00926 C82UNW 9828532 IC50 = 1800 nM T00926 CI78PM 9848185 IC50 = 1050 nM T00926 C30DJS 9873998 IC50 = 800 nM T00926 CK5L6J 9904482 EC50 = 64000 nM T00926 CHI5S9 9975676 IC50 = 2900 nM T00926 CEG64W 9976758 EC50 = 2800 nM T00926 CDTB42 9979854 IC50 >= 250 nM T00926 CL5ZS9 9980860 IC50 = 650 nM T00926 C2B0CY 10004696 IC50 >= 250 nM T00926 CQI0Z7 10029563 IC50 = 76 nM T00926 C0HN4T 10031184 IC50 = 118 nM T00926 CG3RA9 10046544 IC50 = 1850 nM T00926 C5IQ2D 10047863 IC50 < 250 nM T00926 CK4A1L 10048669 IC50 = 1020 nM T00926 C2ZUK8 10051663 IC50 < 250 nM T00926 CC6U1G 10071405 IC50 >= 250 nM T00926 CSY05M 10072430 IC50 = 38 nM T00926 CO0QB1 10092403 IC50 = 7350 nM T00926 CWJ7R4 10094280 IC50 >= 250 nM T00926 CE6X4R 10221081 EC50 = 49100 nM T00926 C96LOC 10251349 IC50 > 50000 nM T00926 CQT7H4 10320818 IC50 = 65 nM T00926 C3I4DW 10322116 IC50 = 715 nM T00926 CY73KI 10322450 EC50 = 1800 nM T00926 CW6D4S 10333981 IC50 = 10800 nM T00926 CK9SQ7 10344755 IC50 = 533 nM T00926 CXG67L 10345205 IC50 = 500 nM T00926 C7Z4DU 10346312 IC50 >= 250 nM T00926 C7Z8IW 10379829 IC50 = 2870 nM T00926 CAO02N 10383921 IC50 = 789 nM T00926 CQU08N 10388318 IC50 >= 250 nM T00926 C36PIN 10407830 IC50 = 197 nM T00926 C1DYS4 10432300 IC50 = 920 nM T00926 CG40WP 10454772 IC50 = 910 nM T00926 CW4BK0 10455921 IC50 = 138 nM T00926 CE7IT1 10459316 IC50 >= 250 nM T00926 CCS90U 10472817 IC50 = 714 nM T00926 C78HZG 10495050 IC50 = 932 nM T00926 CE1U9A 10517005 EC50 > 100000 nM T00926 CCG5H3 10518339 IC50 = 14500 nM T00926 C8HWT1 10543161 IC50 = 2710 nM T00926 CD2EQ3 10585756 IC50 = 43100 nM T00926 CHE31J 10591449 IC50 > 100000 nM T00926 C58EFZ 10616146 IC50 = 4190 nM T00926 CH1V7U 10708375 IC50 = 20400 nM T00926 C7ANU6 10709061 IC50 = 8290 nM T00926 CH72SE 10709378 IC50 = 18300 nM T00926 CSK86O 10756523 IC50 = 2560 nM T00926 C01KTG 10758537 IC50 = 5970 nM T00926 CQF21J 10776189 IC50 = 26400 nM T00926 CI1RC8 10830017 IC50 = 4060 nM T00926 COHV95 10848828 IC50 = 4460 nM T00926 C53AIX 10850200 IC50 = 43400 nM T00926 C2BXZ1 11156535 IC50 >= 250 nM T00926 CKJ32I 11164648 IC50 = 6350 nM T00926 C5E8LY 11168500 IC50 = 20 nM T00926 C84PJK 11177283 IC50 = 94 nM T00926 C8HF7R 11177641 IC50 = 399 nM T00926 CYQ98P 11179994 IC50 = 138 nM T00926 CN3B9L 11186582 IC50 = 9000 nM T00926 CTBH70 11189272 IC50 = 2800 nM T00926 C8CWV4 11200621 IC50 = 632 nM T00926 C6XUE4 11201011 IC50 = 33 nM T00926 CLT87I 11212921 IC50 = 41 nM T00926 CFD6R7 11213871 IC50 = 48 nM T00926 CD8VO1 11214464 IC50 = 15 nM T00926 C63QRZ 11226516 IC50 = 17 nM T00926 C7PTZ8 11246811 IC50 >= 250 nM T00926 C79PBA 11247947 IC50 = 59 nM T00926 C86MWN 11249529 IC50 = 13.7 nM T00926 COJD26 11258566 IC50 = 2300 nM T00926 CEN76W 11261262 IC50 = 40.9 nM T00926 CI1M9O 11270541 IC50 = 28 nM T00926 CP13GR 11270563 IC50 = 59 nM T00926 C8NL3A 11281999 IC50 = 3440 nM T00926 C4I2ZV 11293873 IC50 = 2710 nM T00926 CY79US 11293906 IC50 = 110 nM T00926 CFX64S 11293909 IC50 = 166 nM T00926 CH7E1O 11293927 IC50 = 147 nM T00926 C1YH6T 11295806 IC50 = 97 nM T00926 CJYA49 11304370 IC50 = 24 nM T00926 CXKY42 11305058 IC50 = 45 nM T00926 CD9SN8 11316308 IC50 = 167 nM T00926 CE4HY2 11318194 IC50 = 88 nM T00926 CL8ZT6 11327691 IC50 = 3150 nM T00926 CY8G5H 11337594 IC50 >= 250 nM T00926 C78BGT 11339085 IC50 = 169 nM T00926 C65ZTX 11350733 IC50 = 820 nM T00926 C8P1QC 11351150 IC50 >= 250 nM T00926 CYZ51K 11359019 IC50 = 8370 nM T00926 C61ARN 11362459 IC50 = 1415 nM T00926 C31PLX 11376266 IC50 = 29 nM T00926 CZ9W0I 11385818 IC50 = 78 nM T00926 C8S3OV 11396606 IC50 = 87 nM T00926 C0G4AF 11408751 IC50 = 120 nM T00926 C13MRQ 11418752 IC50 = 955 nM T00926 CUO79V 11419244 IC50 = 63 nM T00926 C49LBJ 11432257 IC50 = 620 nM T00926 CTK09U 11443156 IC50 = 13 nM T00926 CLB97A 11443942 IC50 = 26.5 nM T00926 CM2J9W 11444700 IC50 < 250 nM T00926 CSK8F9 11453657 IC50 = 190 nM T00926 C19WQH 11454150 IC50 >= 250 nM T00926 CTQS76 11454703 IC50 = 10 nM T00926 C59DBU 11454819 IC50 < 250 nM T00926 CYCB17 11455462 IC50 = 107 nM T00926 C6W0MU 11477947 IC50 = 122 nM T00926 CH0T1B 11488138 IC50 = 27 nM T00926 CJXT34 11751643 IC50 = 67 nM T00926 CXWU95 11752839 IC50 < 250 nM T00926 C9X6DU 11774980 IC50 = 51 nM T00926 CLR59J 11775287 IC50 = 62 nM T00926 C2C3WI 11957988 IC50 > 20000 nM T00926 CG1CU7 12219475 EC50 > 100000 nM T00926 CS4D6C 12405466 EC50 = 15100 nM T00926 C4D7RX 12613559 EC50 = 26500 nM T00926 C6UJA5 13144102 EC50 > 100000 nM T00926 CT0DU8 13633111 IC50 = 20400 nM T00926 CO9ES2 13633119 IC50 = 1210 nM T00926 CJ9Z4M 15290116 EC50 = 72000 nM T00926 CLD92G 15999199 IC50 = 40600 nM T00926 C0A3IV 16092354 IC50 = 3730 nM T00926 CMVW98 16618023 EC50 = 728 nM T00926 CX06NR 17412108 IC50 = 39300 nM T00926 CB7T2K 20963109 IC50 = 7720 nM T00926 CFI13S 22310708 IC50 = 7820 nM T00926 CK4UG1 23323164 IC50 > 100000 nM T00926 C3ESV6 24178402 EC50 = 2800 nM T00926 C60EJI 25113688 EC50 = 9300 nM T00926 C6O2ZR 25225119 EC50 = 2700 nM T00926 C3J8PO 39176758 IC50 > 100000 nM T00926 CG7UZ6 44220872 IC50 = 12300 nM T00926 C8C9MJ 44220873 IC50 = 42600 nM T00926 CSLJ20 44220874 IC50 = 5380 nM T00926 CPIM70 44220875 IC50 = 21600 nM T00926 C01FMP 44220876 IC50 = 16200 nM T00926 C04ZKP 44220877 IC50 = 18300 nM T00926 CY9AW0 44221092 IC50 = 11600 nM T00926 C0X8OT 44221093 IC50 = 4510 nM T00926 C12MDG 44221095 IC50 = 14300 nM T00926 C3MNS1 44221096 IC50 = 27500 nM T00926 C2VWE1 44221097 IC50 = 1230 nM T00926 C9BNA1 44248179 EC50 = 73 nM T00926 CKA6N2 44276937 IC50 = 122 nM T00926 CTOA75 44368818 IC50 = 2020 nM T00926 CPLV23 44368900 IC50 > 10000 nM T00926 C26MFU 44368902 IC50 = 7600 nM T00926 CHO6P8 44368923 IC50 = 400 nM T00926 COWL28 44369026 IC50 = 1330 nM T00926 CDLX46 44369027 IC50 = 1560 nM T00926 C9VXD2 44369028 IC50 = 3840 nM T00926 CT0SK1 44369032 IC50 = 36000 nM T00926 CCD76W 44369044 IC50 = 37000 nM T00926 C1V6QO 44369052 IC50 = 900 nM T00926 CY08UQ 44369067 IC50 = 1000 nM T00926 C0FXA2 44369069 IC50 = 18570 nM T00926 C82JKC 44369082 IC50 = 1500 nM T00926 C0Z4TJ 44369087 IC50 = 15100 nM T00926 CZD46M 44369091 IC50 = 6350 nM T00926 CLIY42 44369110 IC50 = 1000 nM T00926 CTE65O 44369198 IC50 = 7200 nM T00926 C1J6DA 44369228 IC50 = 4500 nM T00926 CKPW47 44369229 IC50 = 3200 nM T00926 CA0PF4 44369232 IC50 > 100000 nM T00926 CU9H3K 44369247 IC50 = 39000 nM T00926 C05EUO 44369260 IC50 = 3330 nM T00926 CGU9Z8 44369264 IC50 = 2910 nM T00926 C5JLT0 44369265 IC50 = 2800 nM T00926 CE32OY 44369278 IC50 = 10000 nM T00926 C40XPZ 44404554 IC50 >= 250 nM T00926 CU97QG 44404555 IC50 < 250 nM T00926 CHX57V 44404558 IC50 < 250 nM T00926 C89BQU 44405535 EC50 = 420 nM T00926 CLV54W 44405572 EC50 = 250 nM T00926 C8A7CS 44405716 EC50 = 640 nM T00926 CM8O3W 44451264 EC50 > 100000 nM T00926 C45VCM 44451857 EC50 = 21000 nM T00926 CG61YX 44542293 EC50 > 100000 nM T00926 CI9VZ6 44542743 EC50 > 100000 nM T00926 C80EVI 44723582 EC50 > 100000 nM T00926 C43FNG 45266957 IC50 = 4180 nM T00926 C8C4ZS 45267881 IC50 = 22800 nM T00926 C8IYJ2 45268774 IC50 = 198000 nM T00926 CUE5Y2 45269621 IC50 = 29100 nM T00926 CJG13Y 45272176 IC50 = 24000 nM T00926 CAPW24 45272182 IC50 = 20700 nM T00926 COA30H 46227751 IC50 > 20000 nM T00926 CLWR13 46227752 IC50 > 20000 nM T00926 CX2EU1 46843551 EC50 = 13000 nM T00926 CON7Q5 46888534 EC50 = 46000 nM T00926 C53NLD 46888535 EC50 = 7610 nM T00926 CWO79T 46899560 EC50 = 12000 nM T00926 CUFI19 46899561 EC50 = 8700 nM T00926 C43WPR 46899562 EC50 = 8000 nM T00926 C2QX3P 46899563 EC50 = 63000 nM T00926 CBWT20 46899565 EC50 = 13600 nM T00926 CHR49C 46899724 EC50 > 100000 nM T00926 CZXN91 46899725 EC50 = 85800 nM T00926 C7ZS6E 46899726 EC50 = 29500 nM T00926 C1H9ML 56764960 IC50 = 22700 nM T00926 C2WYN9 56945196 IC50 > 100000 nM T00926 C7RW8P 56945197 IC50 = 11200 nM T00926 C7LDX6 56945198 IC50 > 100000 nM T00926 C2N8DS 56945199 IC50 > 100000 nM T00926 CN2WF6 56945201 IC50 > 100000 nM T00926 CB7W4E 56945202 IC50 > 100000 nM T00926 CT4BW6 56945299 IC50 > 100000 nM T00926 CTEJ21 56945300 IC50 = 45800 nM T00926 CU2HC7 56945301 IC50 = 40600 nM T00926 CUK5Q9 56945302 IC50 = 38800 nM T00926 C36HTV 56945303 IC50 = 46600 nM T00926 C7X2EU 56945304 IC50 = 44500 nM T00926 C4VNX9 56945305 IC50 = 16300 nM T00926 C1JCB9 56945418 IC50 = 44000 nM T00926 C6UD7F 56945419 IC50 = 32200 nM T00926 C98UJH 56945420 IC50 = 8000 nM T00926 C51PRX 56945421 IC50 = 22000 nM T00926 CES25H 56945422 IC50 = 9500 nM T00926 C2QB4L 56945423 IC50 = 7700 nM T00926 CA6UX7 56945524 IC50 = 74500 nM T00926 C4AVC1 56945525 IC50 = 40600 nM T00926 CC25LY 56945526 IC50 = 75800 nM T00926 C8KLW6 56945527 IC50 = 37900 nM T00926 C6ZSA3 56945528 IC50 = 30000 nM T00926 C2IAL8 56945529 IC50 = 28000 nM T00926 CP6G0O 56945530 IC50 > 100000 nM T00926 C27RQI 56946614 IC50 > 100000 nM T00926 CK1ZU5 56946616 IC50 = 23600 nM T00926 C73GCK 56946617 IC50 > 100000 nM T00926 CL8Z0F 56946723 IC50 = 23300 nM T00926 CIQ64Z 56946724 IC50 = 17200 nM T00926 CXMK07 56946726 IC50 > 100000 nM T00926 CRY4C6 56946727 IC50 = 80000 nM T00926 CV29FO 56946728 IC50 > 100000 nM T00926 CI69QT 56946831 IC50 > 100000 nM T00926 CDPU29 56946832 IC50 > 100000 nM T00926 C69ELZ 56946833 IC50 = 6100 nM T00926 CH7M4O 56946835 IC50 > 100000 nM T00926 CP1VK5 56951135 IC50 > 200000 nM T00926 C1XCE9 57393400 IC50 > 100000 nM T00926 CJXP74 71061793 EC50 > 100000 nM T00926 CA2N0L 71062020 EC50 = 31800 nM T00926 C0QGU2 71062093 EC50 = 33200 nM T00926 C5T0NL 71454923 IC50 = 11180 nM T00926 C4ZD2W 71492590 IC50 = 418 nM T00926 C0P6IG 71492759 IC50 = 434 nM T00926 CV9QS7 71524587 EC50 > 100000 nM T00926 C7JIG6 71524588 EC50 > 100000 nM T00926 C1EY6B 71524589 EC50 = 14700 nM T00926 C4LPZ3 71524590 EC50 = 3200 nM T00926 C60ZQJ 71524591 EC50 = 8800 nM T00926 CGV8F5 71525288 EC50 > 100000 nM T00926 CO9ZJ3 71560809 EC50 > 100000 nM T00926 C0E6OM 71560810 EC50 > 100000 nM T00926 C3T8ZF 71560811 EC50 > 100000 nM T00926 CFN89Y 71560812 EC50 > 100000 nM T00926 C42SMF 71560938 EC50 > 100000 nM T00926 C98LPJ 71560939 EC50 > 100000 nM T00926 CG8DU1 71618156 EC50 > 100000 nM T00926 C0Z3PN 71682039 EC50 > 100000 nM T00926 CV5Z9M 71682040 EC50 > 100000 nM T00926 C1IZT7 71682041 EC50 > 100000 nM T00926 COV12T 71682195 EC50 > 100000 nM T00926 C3Y4FW 71682196 EC50 > 100000 nM T00926 CLF3I8 71682197 EC50 > 100000 nM T00926 CN6Q3L 71696716 EC50 = 113 nM T00926 CQCF98 71724480 EC50 = 151 nM T00926 C1PR7Z 71724504 EC50 = 140 nM T00926 CA7K8Z 71724506 EC50 = 217 nM T00926 CD9KH7 71724532 EC50 = 250 nM T00926 CWR2L5 71724556 EC50 = 220 nM T00926 C4ODQ2 71724557 EC50 = 425 nM T00926 C7T0UM 71724558 EC50 > 1000 nM T00926 CUL9E2 71724582 EC50 = 238.3 nM T00926 CNW68B 71724606 EC50 = 616.7 nM T00926 CCZ9B3 71724628 EC50 = 230 nM T00926 C48CAR 72735227 IC50 = 14090 nM T00926 CQ5NB6 72950792 IC50 = 21800 nM T00926 CF57OZ 73346145 IC50 = 19000 nM T00926 CK3EX6 73355255 IC50 = 27500 nM T00926 C7NTB0 73356802 IC50 = 15100 nM T00926 CRB93S 89784681 EC50 = 301.7 nM T00926 CG71EX 89784708 EC50 = 175 nM T00926 C4ZOX6 89784717 EC50 = 670 nM T00926 C0ZQO6 89784722 EC50 = 171 nM T00926 C4U5CZ 89784733 EC50 = 208 nM T00926 CW17YB 89784735 EC50 = 272 nM T00926 C0VD4P 89784742 EC50 = 114 nM T00926 CZT7B9 89784751 EC50 = 135 nM T00926 CH70XJ 89784752 EC50 = 193 nM T00926 C6MRA2 89784753 EC50 = 87 nM T00926 C1JH4L 89784756 EC50 = 243.3 nM T00926 CN1RD8 89784760 EC50 = 333.3 nM T00926 C2YB6Q 89784818 EC50 = 137 nM T00926 CSK8X6 89784827 EC50 = 233.3 nM T00926 CENX80 89785043 EC50 = 103 nM T00926 CY46QV 89785047 EC50 = 172.3 nM T00926 CQL7T6 89785059 EC50 = 99 nM T00926 CENR59 89785064 EC50 = 263 nM T00926 CVZG56 89785117 EC50 = 78 nM T00926 CT43OU 89785127 EC50 = 133.8 nM T00926 C3FB6Q 89785132 EC50 = 219 nM T00926 C4S9WG 89785146 EC50 = 650 nM T00926 CCE95J 89785148 EC50 = 184 nM T00926 C9SBA1 89785178 EC50 = 246.7 nM T00926 CSI51G 89785190 EC50 = 225 nM T00926 CGB2P5 89785210 EC50 = 276.3 nM T00926 CTY1H5 89785238 EC50 = 155 nM T00926 CHGX10 89785254 EC50 = 292.7 nM T00926 CB1FR2 89794901 EC50 = 441.7 nM T00926 C43AXK 89795130 EC50 = 750 nM T00926 C70LJV 89795278 EC50 > 1000 nM T00926 CFU4W2 89795305 EC50 = 760 nM T00926 CVB23M 89795326 EC50 = 245 nM T00926 CX1W9Z 89795330 EC50 = 165 nM T00926 C7XG4U 89795333 EC50 = 950 nM T00926 C7W1TP 89795335 EC50 = 475 nM T00926 CAX9S0 89795337 EC50 = 457.5 nM T00926 COB3Z9 89795340 EC50 = 180 nM T00926 C6BW0Q 89795341 EC50 = 137.7 nM T00926 CUHC90 90469229 EC50 = 11900 nM T00926 C05JQB 90469230 EC50 = 7000 nM T00926 C41EMT 90469289 EC50 = 3900 nM T00926 CA1VH0 90469291 EC50 = 12400 nM T00926 C4NX2Q 90469293 EC50 = 6600 nM T00926 C0NW8T 90469355 EC50 = 5200 nM T00926 C8BRG2 101876951 EC50 = 1100 nM T00926 C0H9DF 101891699 EC50 = 23000 nM T00926 CXHQ89 102340685 IC50 = 4280 nM T00926 CJ7VI3 102340686 IC50 = 6260 nM T00926 CS1P5K 102340687 IC50 = 3380 nM T00926 C93SXK 102340688 IC50 > 100000 nM T00926 C86WSC 117777746 EC50 = 255 nM T00926 C9E0BT 117777811 EC50 = 135 nM T00926 C9YPJ7 117803128 EC50 = 579 nM T00926 C5GUV9 118708511 IC50 = 5800 nM T00926 CQLK93 118708512 IC50 > 100000 nM T00926 C5F8LY 118708513 IC50 = 13600 nM T00926 CL8H6M 118708514 IC50 > 100000 nM T00926 CCT4I2 118708515 IC50 > 100000 nM T00926 C7GI8W 118708516 IC50 > 100000 nM T00926 CE7Q3U 118708517 IC50 > 100000 nM T00926 C31MGA 118708518 IC50 > 100000 nM T00926 CKV6P1 118708519 IC50 > 100000 nM T00926 C1MJ4N 118708520 IC50 > 100000 nM T00926 C7WFJ3 118708521 IC50 = 2200 nM T00926 CVK89G 118708522 IC50 > 100000 nM T00926 C7G3ZV 118708523 IC50 = 94500 nM T00926 CG8S9M 118708524 IC50 = 15800 nM T00926 C9T4KE 118708525 IC50 = 11100 nM T00926 CG3LK4 118708526 IC50 = 8130 nM T00926 C42ETW 118708527 IC50 = 23600 nM T00926 C0OQ9P 118716252 EC50 = 41400 nM T00926 C3VRT8 118716258 EC50 = 5200 nM T00926 C4Z2DS 118719365 EC50 = 10000 nM T00926 CU6EP1 122179376 IC50 = 322 nM T00926 CIL20J 122179390 IC50 = 142 nM T00926 C0OUW1 122179391 IC50 = 141 nM T00926 CCE46L 126587406 EC50 > 1000 nM T00926 CZG92F 127028059 IC50 = 11300 nM T00926 CSR0Y7 127028060 IC50 > 100000 nM T00926 C8Z2XI 127028354 IC50 = 19800 nM T00926 C8Q9DG 127028355 IC50 = 20800 nM T00926 CRI72H 127028356 IC50 = 22700 nM T00926 C58QBI 127028357 IC50 > 100000 nM T00926 C6AIP3 127028358 IC50 > 100000 nM T00926 CG46ES 127028359 IC50 = 30100 nM T00926 CRP9U1 127028361 IC50 = 53300 nM T00926 CUC9I4 127040367 IC50 = 18500 nM T00926 C0I9VF 127040368 IC50 = 5500 nM T00926 CX9JE1 127040369 IC50 = 8300 nM T00926 CRM9W5 127040370 IC50 = 1800 nM T00926 CJY60W 127042304 IC50 = 58300 nM T00926 CO2P8K 127042305 IC50 = 26700 nM T00926 C56HDS 127042306 IC50 = 8300 nM T00926 CRI0X9 127042307 IC50 > 100000 nM T00926 CK4J8D 127042801 IC50 = 7300 nM T00926 C87PMI 127042802 IC50 = 13200 nM T00926 CRQ7U8 127042918 IC50 = 10900 nM T00926 CDL84X 127042919 IC50 > 100000 nM T00926 C39PWZ 127042920 IC50 = 38000 nM T00926 C21DSU 127042921 IC50 = 6800 nM T00926 C6UZ7C 127042922 IC50 > 100000 nM T00926 CSBM31 127042943 IC50 = 12100 nM T00926 C12BJD 127042944 IC50 = 18800 nM T00926 CZBJ54 127048170 IC50 = 1010 nM T00926 CO93BJ 127048171 IC50 = 8980 nM T00926 C6L0AF 127049502 IC50 = 636 nM T00926 CK1SN3 127049508 IC50 = 1070 nM T00926 CB9EV4 127049509 IC50 = 2500 nM T00926 C7PF5I 127050480 IC50 = 623 nM T00926 C59EXD 127050481 IC50 = 876 nM T00926 CUO40Y 127050796 IC50 = 910 nM T00926 C7MJ5X 127050797 IC50 = 586 nM T00926 CT6A2G 127050798 IC50 = 2360 nM T00926 C6V7JZ 127051981 IC50 = 418 nM T00926 C4P0LG 127051982 IC50 = 821 nM T00926 C5CX0B 127051983 IC50 = 200 nM T00926 CBQL62 127051984 IC50 = 340 nM T00926 C0FOG1 127051985 IC50 = 866 nM T00926 C1VP2D 127052887 IC50 = 9410 nM T00926 CG9TE5 127052888 IC50 = 643 nM T00926 CA7N9R 127052889 IC50 = 981 nM T00926 C6ZK3C 135449697 EC50 > 100000 nM T00926 CD2NR8 136110930 IC50 = 95000 nM T00926 C1EB8Q 136236384 EC50 > 100000 nM T00926 CI0KU2 137643961 IC50 = 15900 nM T00926 CHCB46 145956407 IC50 = 44200 nM T00926 C1F4LH 145971569 IC50 > 1000 nM T00926 CK61NI 145973976 IC50 > 1000 nM T00926 CF8L7A 145979103 EC50 = 298 nM T00926 C3EX7W 145979504 EC50 = 170 nM T00926 C4G7LT 145980033 EC50 = 95 nM T00926 C26OWY 145981942 EC50 = 156 nM T00926 C13VFZ 145985646 EC50 = 53 nM T00926 C4A1LN 145985882 EC50 = 38000 nM T00926 CI38SJ 145987174 EC50 = 28900 nM T00926 CFU24J 145987833 EC50 = 103 nM T00926 CGL02K 145988126 EC50 = 205 nM T00926 CX3YR7 145990226 EC50 = 200 nM T00926 CZRB08 145990960 EC50 = 62000 nM T00926 CN1V8K 145992500 EC50 = 208 nM T00926 CT02XU 145992768 EC50 = 121 nM T00926 CKZA78 145992770 IC50 = 12500 nM T00926 C07OTB 145993028 EC50 = 111 nM T00926 C65JUT 145993130 EC50 > 1000 nM T00926 C3UC5J 145994097 EC50 = 207.3 nM T00926 CKM79V 145994277 EC50 = 155.8 nM T00926 C5VRT4 155511477 IC50 > 100000 nM T00926 C1L0WJ 155511549 IC50 = 20000 nM T00926 CE4C1X 155512695 IC50 = 5800 nM T00926 C0AFT8 155514623 EC50 > 1000 nM T00926 CH6O3X 155515825 EC50 = 5080 nM T00926 CV9TF6 155516191 EC50 > 1000 nM T00926 C4IS7E 155518051 EC50 = 2200 nM T00926 CLQO05 155518383 IC50 = 9680 nM T00926 CA1BD2 155520579 EC50 = 12700 nM T00926 C8WFN9 155522227 IC50 > 100000 nM T00926 C8V3OE 155522345 IC50 > 100000 nM T00926 CQK86M 155522385 IC50 > 100000 nM T00926 CS18PU 155523410 EC50 = 5600 nM T00926 CN6ST7 155523417 EC50 > 1000 nM T00926 C86ZPR 155525910 EC50 = 4400 nM T00926 C8TQ4G 155526547 EC50 > 1000 nM T00926 C9BGT5 155528240 EC50 > 1000 nM T00926 C75OQS 155529248 IC50 = 2980 nM T00926 C3O4FR 155529325 IC50 > 100000 nM T00926 C56AHP 155530068 EC50 = 181.4 nM T00926 C9F3YI 155530680 IC50 = 44000 nM T00926 C6I0LU 155531567 IC50 = 18000 nM T00926 CUL2G4 155531672 EC50 > 1000 nM T00926 CJ5X8R 155532908 IC50 = 322 nM T00926 C4IW9M 155533366 EC50 = 5800 nM T00926 C9QT4A 155533532 IC50 = 85100 nM T00926 CHF7A6 155535686 EC50 > 1000 nM T00926 C28CPM 155536187 IC50 = 3600 nM T00926 CQC9E5 155536529 IC50 > 100000 nM T00926 CGM43D 155536878 IC50 = 40000 nM T00926 CYG84N 155537154 EC50 = 7300 nM T00926 C2J7TM 155537461 IC50 = 17300 nM T00926 CGD47O 155537584 EC50 > 1000 nM T00926 CNS83Y 155538210 IC50 = 33000 nM T00926 CVES34 155538494 EC50 = 1900 nM T00926 CLU37N 155539307 EC50 = 3000 nM T00926 CXN6C4 155539538 IC50 = 31000 nM T00926 CL6QG0 155542981 IC50 = 73000 nM T00926 C7JUC3 155543680 EC50 = 4500 nM T00926 C1HI5E 155550141 IC50 > 100000 nM T00926 CB8FC1 155550293 EC50 = 3500 nM T00926 C8B3LI 155551011 IC50 = 3700 nM T00926 CX43TI 155551742 IC50 = 41000 nM T00926 CIF4T8 155553306 EC50 > 1000 nM T00926 CEZ7B1 155554618 EC50 = 137 nM T00926 CX6CM0 155554919 EC50 = 530 nM T00926 CU9P0W 155555392 IC50 = 18000 nM T00926 C7JI4C 155555932 EC50 = 348.3 nM T00926 C27XQN 155558615 EC50 = 212 nM T00926 C8ATZ5 155558917 IC50 = 53000 nM T00926 CUNV65 155558919 EC50 > 1000 nM T00926 CFRS42 155559312 IC50 > 100000 nM T00926 CG6NC7 155560071 EC50 = 10100 nM T00926 CE6C4X 155562808 IC50 > 100000 nM T00926 CWM67C 155563340 EC50 = 2800 nM T00926 C6Z2XK 155566234 EC50 = 3700 nM T00926 CO1LU7 155567143 EC50 > 1000 nM T00926 C7KFG6 155567619 EC50 = 3900 nM T00926 CTV5K3 155568177 EC50 > 1000 nM T00926 C03SJY 155568508 EC50 = 139.3 nM T00926 CTXV81 155568869 EC50 > 1000 nM T00926 C0K1HQ 155569340 IC50 = 12900 nM T00926 D00RFY 5281612 IC50 = 3000 nM T00926 D00RIX 5280443 Ki = 2400 nM T00926 D01FGM 5280666 IC50 = 3000 nM T00926 D07NAY 5281692 Ki = 5000 nM T00926 D0G3TK 5280863 Ki = 2400 nM T00926 D0I7GE 11790 IC50 = 11300 nM T00926 D0T3PW 5281672 Ki = 2400 nM T17967 D03GFC 16741245 EC50 = 80 nM T17967 CHGI09 6597 IC50 = 9000000 nM T17967 CMC1D0 12892 Ki = 176 nM T17967 C6NQ9Y 1116656 IC50 = 3800 nM T17967 CHK89E 6102763 IC50 = 2000 nM T17967 C19DIZ 7178516 EC50 = 5200 nM T17967 CI5FC0 7178544 EC50 = 3800 nM T17967 CG7X9S 7178546 EC50 = 1100 nM T17967 CC28SV 16414363 IC50 = 10900 nM T17967 CHK6P1 16424570 IC50 = 5200 nM T17967 CKQY13 28361735 IC50 = 10500 nM T17967 C28NIL 29255080 IC50 = 1500 nM T17967 C80ODY 67932020 Ki = 1070 nM T17967 CXIN84 72376511 IC50 = 570 nM T17967 CELO13 72376512 EC50 = 456 nM T17967 C47XUW 86280454 IC50 = 65 nM T17967 CI7HO1 97281116 IC50 = 2500 nM T17967 CK6QG0 117972799 IC50 = 206 nM T17967 CUE2B5 118155888 IC50 = 1177 nM T17967 C2SA5C 118155890 IC50 = 416 nM T17967 C5CJ3D 118155894 IC50 = 154 nM T17967 C5Y8GW 118155895 IC50 = 432 nM T17967 C75WOG 118155906 IC50 = 195 nM T17967 C2OW7X 118155909 IC50 = 1196 nM T17967 C4QI2B 124201642 Ki = 2170 nM T17967 CRHZ85 124390110 IC50 = 7.8 nM T17967 C3FC0O 126200721 IC50 = 5900 nM T17967 C0VN5E 134561057 IC50 = 580 nM T17967 C46MPX 134561154 IC50 = 72 nM T17967 CKQ63N 134561155 IC50 = 58 nM T17967 C5X0YD 134561193 IC50 = 1514 nM T17967 CMQ04B 134561196 IC50 = 156 nM T17967 C30MTB 134561301 IC50 = 357 nM T17967 CHME32 134561302 IC50 = 67 nM T17967 C7WTU8 134561303 IC50 = 221 nM T17967 CR3V2E 134561305 IC50 = 65 nM T17967 CO3V2F 134561468 IC50 = 767 nM T17967 C8W3YG 136087021 IC50 = 1126 nM T17967 C0BUJ9 136249185 IC50 = 2600 nM T17967 CMO6K1 137636150 IC50 = 1657 nM T17967 CKU8P4 137638606 IC50 = 629 nM T17967 CAP1D8 137641886 IC50 = 1610 nM T17967 CS3KF0 137642154 Ki = 150 nM T17967 C7KIS8 137645507 IC50 = 1346 nM T17967 CSA49E 137646868 IC50 = 91 nM T17967 CI5TH3 137653481 Ki = 702 nM T17967 C7RB8J 137653507 Ki = 1330 nM T17967 C5XEM7 137655013 IC50 = 565 nM T17967 C0AZR8 137656816 IC50 = 68 nM T17967 C3SV7G 137659540 Ki = 1278 nM T17967 C9LP0W 137660248 IC50 = 4371 nM T17967 CHQ86U 149832647 IC50 = 140 nM T17967 CL6T4P 149986651 IC50 = 10 nM T17967 C24DWX 150179460 IC50 = 302 nM T17967 C7BM5V 150226583 IC50 = 126 nM T17967 CDO4W3 150362366 IC50 = 373 nM T17967 CJ17UR 150426809 IC50 = 18 nM T17967 CMS4L6 150703157 IC50 = 1620 nM T17967 C7J0AF 150821022 IC50 = 772 nM T17967 C1Z5DA 151004457 IC50 = 98 nM T17967 C02NBO 151026196 IC50 = 133 nM T17967 C0Q9PK 151406722 IC50 = 193 nM T17967 CY8OK4 151698036 IC50 = 110 nM T17967 C2RVC3 151777753 IC50 = 252 nM T17967 CKR2T1 151835909 IC50 = 113 nM T17967 CTI5R1 151961601 IC50 = 1455 nM T17967 CC3ME1 152131905 IC50 = 8 nM T17967 CAR6N3 152143591 IC50 = 132 nM T17967 C79SKI 152618834 IC50 = 184 nM T17967 C49BFR 155510663 IC50 = 2040 nM T17967 COH17B 155516961 IC50 > 10000 nM T17967 CRK41X 155523490 IC50 = 2660 nM T17967 C8K4NL 155527038 IC50 = 9910 nM T17967 CCG7K6 155528322 IC50 = 64 nM T17967 CNY40T 155534218 IC50 = 1960 nM T17967 CM20ZB 155534260 IC50 = 503 nM T17967 C8EH6M 155538895 IC50 = 95 nM T17967 C7BTJ9 155554053 IC50 = 8590 nM T17967 CA18GY 155563372 IC50 = 1660 nM T17967 C6Y5IM 155567964 IC50 = 7220 nM T89565 CV7IN2 104934 Ki = 210 nM T89565 C1KR5B 5327301 Ki = 98000 nM T89565 C37TKL 5327302 Ki = 12000 nM T89565 C64ZMN 5327304 Ki = 22000 nM T89565 C3IZ2W 5327307 Ki = 23000 nM T89565 C16DTL 5327308 Ki = 24000 nM T89565 C4O3QY 5327309 Ki = 63000 nM T89565 C3GUM7 5327310 Ki = 36000 nM T89565 CLAC59 9828058 Ki = 81 nM T89565 CDX7A4 10963183 Ki = 32000 nM T89565 CDT9G3 11467504 IC50 = 0.81 nM T89565 CJ57OA 14585243 Ki = 47 nM T89565 C8D5TB 44364680 Ki = 11000 nM T89565 C86ORE 44459987 IC50 = 13489.63 nM T89565 CDY2W5 49796910 IC50 = 0.2 nM T89565 CGY3W2 71471109 IC50 > 100000 nM T89565 CANH70 71716242 IC50 = 35200 nM T89565 C40WIR 71718085 IC50 = 750 nM T89565 CU75VK 71719897 IC50 = 19500 nM T89565 CBV6F1 71720507 IC50 = 560 nM T89565 CWM2E8 133081971 IC50 = 2980 nM T89565 CID3N6 134134572 Ki = 48 nM T89565 CV0R3B 134135432 Ki = 24 nM T89565 C3D7LQ 134136688 Ki = 59 nM T89565 CBY95D 134138690 Ki = 41 nM T89565 CG3EI1 134145896 Ki = 34 nM T89565 CI9X3K 134147411 Ki = 16 nM T89565 CP16IA 134148745 Ki = 111 nM T89565 CPE90G 134149983 Ki = 34 nM T89565 CBE39C 134151245 Ki = 135 nM T89565 CY0LD4 134152014 Ki = 59 nM T89565 C3K5HR 134153309 Ki = 28 nM T89565 CWQT79 134156687 Ki = 99 nM T89565 D0Y5IQ 44255320 IC50 = 5000 nM T50269 D00KHM 16362 EC50 = 1700 nM T50269 D01AZG 5073 EC50 = 320 nM T50269 D03YGR 156419 EC50 = 320 nM T50269 D09GDD 11167602 EC50 = 1800 nM T50269 D0A9YA 6918296 EC50 = 330 nM T50269 D0GQ7K 4046 EC50 = 2500 nM T50269 D0JC9N 60164 EC50 = 1300 nM T50269 D0K5WS 5280795 EC50 = 400 nM T50269 D0M8AB 750 EC50 = 94000 nM T50269 D0N6RF 65999 EC50 = 3200 nM T50269 D0P1FO 16078 EC50 = 1300 nM T50269 D0U5FS 3396 EC50 = 1200 nM T50269 D0Z5IU 1548887 EC50 = 380 nM T50269 D0Y2HR 2247 EC50 = 4200 nM T50269 C3O9AG 439709 EC50 = 12589.25 nM T50269 C8HZF2 783663 IC50 = 76 nM T50269 C9H1CE 5390854 EC50 = 590 nM T50269 C4SWU6 6324617 IC50 = 1700 nM T50269 C3W8ZK 17758335 IC50 > 100000 nM T50269 CH9J0Y 24846186 Ki = 67 nM T50269 COX8D7 44408895 IC50 > 100000 nM T50269 CR6CE1 44408940 IC50 > 100000 nM T50269 COY01R 44420834 IC50 = 3162.28 nM T50269 CE30WA 44420835 IC50 = 7400 nM T50269 C0DIM8 44420839 IC50 > 100000 nM T50269 CYE94N 44420840 IC50 > 100000 nM T50269 C59CNH 44420842 IC50 > 100000 nM T50269 C6N3DU 44420843 IC50 > 100000 nM T50269 C6Q1OE 44420847 IC50 > 100000 nM T50269 CKHC34 44420848 IC50 > 100000 nM T50269 C52YKX 44420851 IC50 > 100000 nM T50269 C23CLN 44420852 IC50 > 100000 nM T50269 C2NF6H 44420854 IC50 > 100000 nM T50269 CW2TL6 44420856 IC50 > 100000 nM T50269 C3XV2H 44420857 IC50 > 100000 nM T50269 CG30DJ 44420862 IC50 > 100000 nM T50269 C3AYZ8 44420865 IC50 > 100000 nM T50269 CVS4Z1 44420866 IC50 > 100000 nM T50269 CKG6M0 44420867 IC50 > 100000 nM T50269 CCB95G 44420868 IC50 > 100000 nM T50269 CYX7A3 44420870 IC50 > 100000 nM T50269 COH12C 44420871 IC50 > 100000 nM T50269 C9X7JH 44420872 IC50 > 100000 nM T50269 CR8HG1 44420875 IC50 > 100000 nM T50269 C19QZY 44420876 IC50 > 100000 nM T50269 CSZ5F4 44420878 IC50 = 2400 nM T50269 C6ZG0M 44420879 IC50 > 100000 nM T50269 C3IU8N 44420880 IC50 > 100000 nM T50269 CW80SJ 44420881 IC50 = 3981.07 nM T50269 CV8C2B 44420885 IC50 = 7943.28 nM T50269 CPBM16 44420891 IC50 = 3162.28 nM T50269 CYG93V 44427853 IC50 > 100000 nM T50269 C3C2OK 44427854 IC50 > 100000 nM T50269 C8Y9FW 44427856 IC50 > 100000 nM T50269 C19LSU 44427858 IC50 > 100000 nM T50269 C1FY4M 44427860 IC50 > 100000 nM T50269 CC2BE1 44427862 IC50 > 100000 nM T50269 CW95BM 44427864 IC50 > 100000 nM T50269 C3XJ4Z 44427866 IC50 > 100000 nM T50269 C84GXL 44427868 IC50 > 100000 nM T50269 C8CPX2 44427870 IC50 > 100000 nM T50269 CS17TJ 44427872 IC50 > 100000 nM T50269 CDL67C 44427876 IC50 > 100000 nM T50269 C9B6ER 44427877 IC50 > 100000 nM T50269 C15UHM 44427879 IC50 > 100000 nM T50269 CCAV10 44427881 IC50 > 100000 nM T50269 CXRV71 44427883 IC50 > 100000 nM T50269 CKX81C 44427885 IC50 > 100000 nM T50269 CG71DA 54467154 IC50 = 6900 nM T50269 C6DQT3 71450923 IC50 = 501.19 nM T50269 C2HUL4 90659973 IC50 > 100000 nM T50269 CO9ZU7 99118914 Ki = 40 nM T50269 CFW2V1 118195533 EC50 = 0.0012 nM T50269 CHM30C 118195560 EC50 = 0.06 nM T50269 C3HMN2 118195567 EC50 = 0.43 nM T50269 C8DSH5 118195581 EC50 = 0.00016 nM T50269 CKDM68 123133764 EC50 = 32 nM T50269 CPV2O3 132547348 EC50 = 327 nM T50269 CTN47D 135753560 IC50 = 8800 nM T50269 C8H3QG 135753564 IC50 > 200000 nM T50269 CLE71N 137631631 IC50 = 109 nM T50269 CL2X3J 137631882 IC50 = 690 nM T50269 C4L8SF 137635401 IC50 = 260 nM T50269 C1YE3F 137637510 IC50 = 720 nM T50269 CS41FM 137639832 IC50 = 4590 nM T50269 CKR79P 137644791 IC50 = 165.96 nM T50269 CVL25O 137645081 IC50 = 245.47 nM T50269 C3DZ4I 137650620 IC50 = 49 nM T50269 CDP0F7 137654599 IC50 = 220 nM T50269 C5QN0I 137655067 IC50 = 380.19 nM T50269 CU8FI4 137656578 IC50 = 75 nM T50269 CF1C3T 137657339 IC50 = 51.29 nM T50269 CRZY05 155519552 Ki = 741 nM T50269 CF27SE 155541454 Ki = 91 nM T50269 D04IEW 9909368 IC50 = 1900 nM T50269 D0H0BD 441071 Ki = 23 nM T50269 D0M4ZK 44420890 IC50 = 5011.87 nM T50269 D0X3TL 44420886 IC50 = 6200 nM T67710 D02CII 76943386 EC50 = 0.02 nM T67710 D03NHS 76283707 EC50 = 4100 nM T67710 CA6P1K 11963968 Ki = 0.912 nM T67710 CA4WI0 12001598 Ki = 707.95 nM T67710 CNF70V 16220269 IC50 = 68000 nM T67710 CH3KU5 23626097 Ki = 2818.38 nM T67710 CF1V4U 23626240 Ki = 3388.44 nM T67710 C5K7RJ 23626241 Ki = 562.34 nM T67710 C7O1ZX 23626243 Ki = 676.08 nM T67710 CS2FX3 23626399 Ki = 288.4 nM T67710 C0ZIC4 23626400 Ki = 154.88 nM T67710 CSI39A 23626402 Ki = 70.79 nM T67710 C0XE1Q 23626403 Ki = 3.802 nM T67710 CUTB14 23626557 Ki = 13.18 nM T67710 C5TJF3 23626558 Ki = 50.12 nM T67710 C0LNV5 23626559 Ki = 20.42 nM T67710 C27CIX 23626560 Ki = 6.761 nM T67710 CXU8E9 23626561 Ki = 3.548 nM T67710 C7JG9E 23626730 Ki = 1.445 nM T67710 C5N9AK 23626731 Ki = 1.82 nM T67710 CF8X4T 23626732 Ki = 6.761 nM T67710 C3B8PO 23626733 Ki = 616.6 nM T67710 CF4NW8 23626734 Ki = 8.71 nM T67710 CVO15W 23626891 Ki = 6.607 nM T67710 CB3D4J 23626894 Ki = 83.18 nM T67710 CU75YI 25118026 IC50 = 9400 nM T67710 CC9G1A 44270419 EC50 = 7.9 nM T67710 CS9AC3 44270511 EC50 = 4.4 nM T67710 C02OVQ 44270512 EC50 = 5.5 nM T67710 CC1OX8 44270513 EC50 = 9.1 nM T67710 CN3D6A 44428088 Ki < 100000 nM T67710 CPY82C 44428090 Ki = 933.25 nM T67710 CRS3H8 44428091 Ki = 380.19 nM T67710 C4FXJ3 44428092 Ki = 112.2 nM T67710 CN6WS7 44584917 EC50 = 32 nM T67710 CH14QN 44584920 EC50 = 13 nM T67710 CJR45V 44584921 EC50 = 0.06 nM T67710 CXSB17 44584922 EC50 = 0.15 nM T67710 CQS1U6 45485585 EC50 > 10000 nM T67710 C5XME6 49838154 EC50 > 1000000 nM T67710 C09VXY 49840922 EC50 = 1122 nM T67710 CPX2V6 49841000 EC50 = 0.2 nM T67710 CU3J0E 50908590 EC50 = 2.4 nM T67710 C24IPZ 56841901 EC50 = 0.07 nM T67710 C6Y8QI 66815925 EC50 > 1000000 nM T67710 CM8BP9 66817107 EC50 = 26000 nM T67710 C6IP4J 66817215 EC50 = 32000 nM T67710 CVCF27 66817553 EC50 = 33000 nM T67710 CAX82O 66817788 EC50 = 12000 nM T67710 C6CM8L 76283959 EC50 = 3600 nM T67710 C4WM1Z 137631923 EC50 = 19 nM T67710 C9XVZ4 137634846 EC50 = 0.51 nM T67710 CHV35B 137634885 EC50 = 0.26 nM T67710 CWA3V8 137635204 EC50 = 1.12 nM T67710 CIN0J6 137635394 EC50 = 0.08 nM T67710 CB64NJ 137636149 EC50 = 0.15 nM T67710 CP59IE 137636311 EC50 = 0.51 nM T67710 C7KQ9X 137637857 EC50 = 0.29 nM T67710 C6ZXO0 137637950 EC50 = 3 nM T67710 CLW1R3 137639371 EC50 = 14.57 nM T67710 CUZP78 137639372 EC50 = 0.13 nM T67710 C7O9IM 137639587 EC50 = 18.69 nM T67710 C05BRV 137640122 EC50 = 0.52 nM T67710 CT9B3U 137640833 EC50 = 0.34 nM T67710 C1O3FE 137641949 EC50 = 0.4 nM T67710 CSY1M3 137642287 EC50 = 0.14 nM T67710 C93LST 137642401 EC50 = 4.98 nM T67710 C3V6MW 137642849 EC50 = 0.12 nM T67710 C12BTY 137643019 EC50 = 0.34 nM T67710 CDR83Q 137643296 EC50 = 1.8 nM T67710 CQIU59 137645140 EC50 = 0.71 nM T67710 C71AOQ 137650056 EC50 = 11.51 nM T67710 C89VPB 137651582 EC50 = 0.18 nM T67710 C4A9EI 137652688 EC50 = 9.74 nM T67710 CL41NK 137654722 EC50 = 0.36 nM T67710 CV6G8Y 137657562 EC50 = 1.84 nM T67710 CRNM53 137657563 EC50 = 167 nM T67710 C79QHV 137657564 EC50 = 0.44 nM T67710 CN6V0J 137657565 EC50 = 0.83 nM T67710 CE0J2B 137657566 EC50 = 0.79 nM T67710 CQ8J3B 137657687 EC50 = 0.32 nM T67710 C5Q7KC 137657688 EC50 = 0.65 nM T67710 C38QDU 137657689 EC50 = 4.13 nM T67710 C5PM6C 137659455 EC50 = 0.48 nM T67710 CE5MN9 137659482 EC50 = 0.06 nM T67710 C3BK4S 137659489 EC50 = 2.59 nM T67710 C0ZJN1 137659716 EC50 = 0.17 nM T67710 C4TH5F 137660321 EC50 = 9.84 nM T67710 C8WFK3 137660410 EC50 = 0.27 nM T67710 CCT8K0 139035050 IC50 = 90 nM T67710 CDXQ89 145964425 EC50 = 67000 nM T67710 C60ZAH 145975286 EC50 = 50000 nM T67710 C9MJG6 145975813 EC50 > 1000000 nM T67710 CL3X2U 155513348 EC50 = 4600 nM T67710 C26GUZ 155518374 IC50 = 6800 nM T67710 CXZ5W0 155521869 IC50 > 100000 nM T67710 CB7Z3X 155522420 IC50 = 3500 nM T67710 CX2TS6 155522839 IC50 = 7600 nM T67710 CN5D9T 155526572 IC50 = 6100 nM T67710 C8LAP0 155529306 IC50 > 100000 nM T67710 CAE4T8 155533095 EC50 = 3600 nM T67710 CKW9P0 155536792 EC50 = 2.5 nM T67710 CTQ9U5 155536860 IC50 = 14000 nM T67710 C2I0PA 155540108 IC50 = 14000 nM T67710 CHM51V 155542161 EC50 = 5300 nM T67710 C2BHW9 155543526 IC50 = 38000 nM T67710 CGT23X 155546261 IC50 = 730 nM T67710 C59QIA 155547998 IC50 = 2300 nM T67710 C38KWY 155550447 IC50 = 4100 nM T67710 CGS61H 155551285 IC50 = 44000 nM T67710 CQ7ZP6 155553639 EC50 = 4600 nM T67710 C65GPR 155553648 EC50 > 100000 nM T67710 C6GAF5 155555773 IC50 = 4000 nM T67710 CFNP14 155557308 IC50 = 45000 nM T67710 CHDB02 155558265 IC50 = 23000 nM T67710 CGVN45 155559611 IC50 = 180 nM T67710 CTQ3H1 155560902 IC50 = 16000 nM T67710 C4DQ3V 155567876 EC50 > 100000 nM T68698 D0H1OL 135398635 Ki = 1472000 nM T68698 D0I7BL 65269 Ki = 110 nM T68698 D0I7TN 23190 IC50 = 4000 nM T68698 D0R2QS 72968 IC50 = 0.004 ug.mL-1 T68698 CY1P2C 72501 Ki = 4 nM T68698 CRG3J6 73651 Ki = 12 nM T68698 CI8KD2 97627 Ki = 410 nM T68698 C2CG8M 98567 Ki = 1930 nM T68698 CGF69C 99920 Ki = 3.3 nM T68698 C3BU7T 147104 Ki = 110 nM T68698 CHT80Q 275945 Ki = 22000 nM T68698 C8I2PG 358177 IC50 = 31 nM T68698 C3J5VD 402194 IC50 < 20000 nM T68698 CRU2Q9 443234 Ki = 39 nM T68698 CVQW71 451935 IC50 = 1000 nM T68698 C72EKO 469184 IC50 = 7600 nM T68698 CY0ZN2 472632 IC50 = 0.2 ug.mL-1 T68698 CA2U7Y 472655 IC50 > 10 ug.mL-1 T68698 C67BXW 481083 IC50 > 10 ug.mL-1 T68698 CJL5D2 489877 IC50 = 0.87 ug.mL-1 T68698 CLRY91 489878 IC50 = 3760 nM T68698 CLO12U 490351 Ki = 41 nM T68698 CJ2L8F 490432 IC50 = 123000 nM T68698 C5L8GI 490433 IC50 = 76000 nM T68698 CE9J3U 501516 Ki = 5020 nM T68698 C58AMW 501517 Ki = 27 nM T68698 CHNA61 501518 Ki = 586 nM T68698 C12AIT 501519 Ki = 22 nM T68698 C8T0YV 501520 Ki = 67600 nM T68698 CB4HR1 512554 IC50 > 10 ug.mL-1 T68698 CKIL63 512555 IC50 = 195 nM T68698 CTF70X 512656 IC50 > 10 ug.mL-1 T68698 CL24RG 512657 IC50 > 10 ug.mL-1 T68698 C1AU9I 512658 IC50 > 10 ug.mL-1 T68698 CL74IO 1362195 Ki = 1700 nM T68698 C13DGU 5358592 IC50 = 40 nM T68698 COLD86 6439007 Ki = 330 nM T68698 CX58IU 6450949 Ki = 125 nM T68698 CSB29R 6474190 IC50 = 90700 nM T68698 CW7NE1 6476927 IC50 = 8 nM T68698 CZR3N8 9816781 IC50 = 75020 nM T68698 CB01OK 9840103 Ki = 16000 nM T68698 CRAI41 9993207 Ki = 7900 nM T68698 C2SKW5 9997450 Ki = 134 nM T68698 CW21OU 10015023 IC50 = 7670 nM T68698 C3DI6E 10061387 Ki = 39 nM T68698 C4VB3K 10243225 Ki = 8800 nM T68698 CHG3J9 10400519 Ki = 273 nM T68698 C2FV5L 10422910 IC50 = 18 nM T68698 CNR64H 10655770 IC50 = 930 nM T68698 CR6A7V 11380460 IC50 = 12680 nM T68698 CJ8QH3 11537088 Ki = 17000 nM T68698 CV0F5A 11564784 Ki = 500 nM T68698 CTMK84 11615884 IC50 > 100000 nM T68698 CXEG94 11777524 Ki = 4500 nM T68698 C2RE5C 11779405 Ki = 110 nM T68698 CX35EZ 12097487 IC50 = 36460 nM T68698 C6IX0V 12769724 IC50 = 100000 nM T68698 C4SD3B 13712019 IC50 = 28000 nM T68698 CEC2K8 13939857 Ki = 35 nM T68698 CW0E2J 14134370 Ki = 160 nM T68698 CU06ED 14134371 IC50 = 1230 nM T68698 CB35KG 14134372 Ki = 200 nM T68698 C45LBI 14134395 IC50 = 950 nM T68698 CF9SO7 14134396 Ki = 200 nM T68698 CPJ92T 14134397 Ki = 170 nM T68698 C5YGX9 14134400 Ki = 90 nM T68698 CYGP51 14134401 Ki = 166 nM T68698 CCF8Z2 14134506 IC50 = 80 nM T68698 CFRL70 16075366 IC50 = 180 nM T68698 CZ03BO 21152084 Ki = 43400 nM T68698 CY07FB 25244925 Ki = 2600 nM T68698 C97ZIN 44189703 IC50 = 1.5 nM T68698 CL4K0U 44278585 Ki = 0.5 nM T68698 CYP2V1 44373339 IC50 > 100000 nM T68698 CS4NG1 44396071 IC50 > 100000 nM T68698 C7ZMI0 44396095 IC50 > 100000 nM T68698 C6BN5P 44396175 IC50 = 97270 nM T68698 CCW9P4 44432644 IC50 = 28940 nM T68698 CS2EY3 44450578 IC50 = 163000 nM T68698 C5JM9A 44450579 IC50 > 500000 nM T68698 CNI6X4 44451567 IC50 = 47200 nM T68698 CI3VJ8 44551468 IC50 = 400 nM T68698 CT8I2H 44561305 Ki = 12400 nM T68698 CVS3O8 44561306 Ki = 20300 nM T68698 C6BG4W 45110892 IC50 = 2.2 nM T68698 C7GN9D 45110893 IC50 = 36 nM T68698 CB5IQ2 45110895 IC50 = 98 nM T68698 CG5RZ9 45111029 IC50 = 4827 nM T68698 C5H3VJ 45111030 IC50 = 189 nM T68698 C36LBT 45111031 IC50 = 9.4 nM T68698 C50EYM 45111032 IC50 = 41 nM T68698 CJA7Q8 45111033 IC50 = 2.7 nM T68698 CL8NW5 45111034 IC50 = 1223 nM T68698 CYAQ84 45111036 IC50 = 28 nM T68698 C7RM9B 46174640 IC50 = 1.3 nM T68698 CZL10R 46874055 Ki = 94.6 nM T68698 CXH9E4 46874068 Ki = 4000 nM T68698 CY41AR 46874106 Ki = 67000 nM T68698 C3DB1E 46874218 Ki = 3100 nM T68698 CN59VL 46874243 Ki = 681 nM T68698 C0HY4G 46874757 Ki = 111 nM T68698 CS32QG 46874759 Ki = 101 nM T68698 C3F2PG 46874761 Ki = 10000 nM T68698 C0NLW6 46875043 Ki = 13700 nM T68698 C0DI9E 46875054 Ki = 45000 nM T68698 CD3C8F 46875063 Ki = 16000 nM T68698 CMGN58 46875065 Ki = 10000 nM T68698 CD28UB 46875621 Ki = 1100 nM T68698 CPHC63 46875632 Ki = 1700 nM T68698 CJ6EL3 46875710 Ki = 770 nM T68698 C19BFH 46875728 Ki = 48500 nM T68698 CE5O4A 46875732 Ki = 570 nM T68698 C8T2JI 46875733 Ki = 710 nM T68698 C7B8QH 46875922 Ki = 3600 nM T68698 CCE7X6 46875931 Ki = 3900 nM T68698 C2VZR9 46876033 Ki = 1300 nM T68698 CGJ03W 46876073 Ki = 96 nM T68698 CZ50WH 46876160 Ki = 3800 nM T68698 CY4L3V 46876365 Ki = 360 nM T68698 CTV70J 46876373 Ki = 570 nM T68698 CKB03R 46876407 Ki = 320 nM T68698 CH81PT 46877209 Ki = 75000 nM T68698 C5NFH6 46877212 Ki = 50000 nM T68698 C1O4WI 46877256 Ki = 750000 nM T68698 CWM2L0 46877257 Ki = 3200 nM T68698 C8IWQ3 46877302 Ki = 105000 nM T68698 CLG04P 46877303 Ki = 19000 nM T68698 C81YJV 46877310 Ki = 550 nM T68698 CJ23FN 46877328 Ki = 4000 nM T68698 CKE16H 46877337 Ki = 118500 nM T68698 CM4CG5 46877338 Ki = 96000 nM T68698 C0HQ5A 46877339 Ki = 17000 nM T68698 C6IRP9 46886640 IC50 > 250000 nM T68698 CW0Y4H 49797674 Ki = 19800 nM T68698 C8GU9B 51003093 IC50 = 60170 nM T68698 CM8WE3 51003094 IC50 > 1000000 nM T68698 C7M3KT 51003095 IC50 > 1000000 nM T68698 C46DIL 51003096 IC50 > 1000000 nM T68698 CZK6B3 53318848 IC50 > 1000000 nM T68698 CC6GR8 57522307 IC50 = 910 nM T68698 C0Z8LK 68364288 IC50 = 2300 nM T68698 CIX13E 73351185 Ki = 1900 nM T68698 C8H9WC 73352895 Ki = 800 nM T68698 CPHB93 90644119 IC50 > 10000 nM T68698 CWP2F5 90644120 IC50 = 2100 nM T68698 C28IXS 90644121 IC50 > 10000 nM T68698 C8INM3 90644122 IC50 = 672 nM T68698 C7ZQA6 90644123 IC50 = 878 nM T68698 C4Y6KI 90644124 IC50 = 1960 nM T68698 CD2X0B 90644125 IC50 = 976 nM T68698 CS3KR7 91824125 Ki = 1.5 nM T68698 C4F3MG 118710205 IC50 = 530 nM T68698 C1PIQ5 118710206 IC50 = 380 nM T68698 C6TMO4 118710207 IC50 = 340 nM T68698 C7IDP1 118710208 IC50 = 970 nM T68698 CG5M1W 118710209 IC50 = 8780 nM T68698 CN29AS 118710210 IC50 = 11360 nM T68698 C0RW1F 118710211 IC50 > 100000 nM T68698 C87EMG 118710212 IC50 = 17000 nM T68698 CMWO70 118710213 IC50 = 2700 nM T68698 C39PRU 118710214 IC50 = 52 nM T68698 CT9PF2 118710215 IC50 = 81 nM T68698 CV51BZ 118710216 IC50 = 530 nM T68698 C5YR2F 118710217 IC50 > 100000 nM T68698 CGT1A9 118710218 IC50 = 4600 nM T68698 CM64LA 118710219 IC50 = 230 nM T68698 CKP9S8 118710220 IC50 = 890 nM T68698 CBW08J 118710221 IC50 = 13 nM T68698 CLAB80 118710222 IC50 = 200 nM T68698 CD01LY 118710223 IC50 = 49 nM T68698 C7HJ8B 118710224 IC50 = 44 nM T68698 C5J7EQ 118710225 IC50 = 330 nM T68698 C01AOB 118710226 IC50 = 320 nM T68698 COMR26 118710227 IC50 = 130 nM T68698 C3AY7W 118710228 IC50 = 70 nM T68698 C91TJV 118710229 IC50 = 60 nM T68698 C1S0YD 118710230 IC50 = 49 nM T68698 C29JSZ 118710231 IC50 = 1200 nM T68698 CI8Z4P 118710232 IC50 = 1500 nM T68698 C34ARU 118710233 IC50 = 110 nM T68698 CR26QJ 118710234 IC50 = 600 nM T68698 CVL4C5 118710235 IC50 = 150 nM T68698 CEW89M 118718118 Ki = 224 nM T68698 CY4DU7 122178501 IC50 > 100000 nM T68698 CGY0N1 122178503 IC50 > 100000 nM T68698 CD98QW 122178504 IC50 > 100000 nM T68698 CX8FW7 122178506 IC50 > 100000 nM T68698 CA98UV 122183895 IC50 = 640 nM T68698 CQ0LA3 122183896 IC50 > 100000 nM T68698 CK6J3X 122183897 IC50 > 100000 nM T68698 CNOV-65 122183898 IC50 = 70 nM T68698 CQM0H1 122183899 IC50 = 60 nM T68698 C6JAU8 122183900 IC50 = 49 nM T68698 CMU94S 122183901 IC50 = 1200 nM T68698 CTU42V 122183902 IC50 = 1500 nM T68698 C0SZO2 122183903 IC50 = 110 nM T68698 CHM13L 122183904 IC50 = 600 nM T68698 C80TRM 122183905 IC50 = 150 nM T68698 CI8WG9 122183915 IC50 = 8.5 nM T68698 CP1FW4 135398641 Ki = 925000 nM T68698 CP4M0E 135976391 Ki 128000 nM T68698 C8WD3Z 135976393 Ki = 422000 nM T68698 CZD50N 137090971 IC50 > 100000 nM T68698 CJW84E 137090972 IC50 > 100000 nM T68698 C5ZM8O 137628302 IC50 > 10000 nM T68698 CW0C4P 155517779 IC50 > 3700 nM T68698 CNP67J 155524359 IC50 > 100000 nM T68698 CKN0W4 155530574 IC50 > 100000 nM T68698 CI2OR3 155531848 IC50 = 4390 nM T68698 CAE5R9 155536819 IC50 > 100000 nM T68698 CZXU90 155538219 IC50 > 100000 nM T68698 CTM53Z 155543643 IC50 > 100000 nM T68698 CKWS45 155544569 IC50 > 100000 nM T68698 CDU83I 155549525 IC50 = 760 nM T68698 CKP82O 155553203 IC50 = 1060 nM T68698 C09CGT 155568198 IC50 > 100000 nM T68698 C0I9OP 155568822 IC50 > 100000 nM T68698 D02XPR 73124 IC50 = 280 nM T68698 D02YYQ 23661679 IC50 = 7530 nM T68698 D0D2MS 11737492 IC50 = 15700 nM T68698 D0F5AJ 126704 Ki = 160 nM T68698 D0O2CM 498018 IC50 = 480 nM T68698 D0X3MK 73087 IC50 = 440 nM T04689 D0T8GD 89594 EC50 = 180000 nM T04689 D09ADT 119380 EC50 = 411000 nM T04689 CUI25G 115224 IC50 = 120000 nM T04689 CY1XN7 7446712 IC50 = 1000 nM T04689 C74CBS 9794141 EC50 = 34000 nM T04689 C0Z5RS 9859386 IC50 = 6000 nM T04689 CLWT60 9882021 EC50 > 100000 nM T04689 CDH4J3 10130527 IC50 = 11000 nM T04689 C6LB2N 10130752 IC50 = 8000 nM T04689 CIQ12L 11701287 Ki = 944 nM T04689 CY7F5O 15389735 EC50 > 1000000 nM T04689 CQ03LX 21290600 IC50 = 81000 nM T04689 CW2R4M 23624283 IC50 = 3981.07 nM T04689 CC1SF7 49863118 IC50 = 794.33 nM T04689 CJ34EQ 53483935 IC50 = 4200 nM T04689 CLH24J 56663402 IC50 > 10000 nM T04689 CU7OP3 56666825 IC50 > 10000 nM T04689 CY01LS 56666826 IC50 > 10000 nM T04689 CCP40B 56666827 IC50 > 10000 nM T04689 CVT85Q 56670262 IC50 = 7800 nM T04689 C7XK8I 56677105 IC50 = 5500 nM T04689 C02AZR 56677106 IC50 > 10000 nM T04689 CL45WN 57345320 IC50 > 30000 nM T04689 CV2J9A 57663655 IC50 = 6309.57 nM T04689 CU3D9N 73388373 EC50 = 19952.62 nM T04689 CI14LP 145949343 IC50 = 11300 nM T04689 CGW92C 145952721 IC50 > 30000 nM T04689 D0R4RN 1204 IC50 = 160 nM T33966 CSD1A3 125874 Ki = 200 nM T33966 CX7U8V 444797 Ki = 450 nM T33966 CF5A3T 9837547 IC50 > 50000 nM T33966 CHI95J 9926432 IC50 = 1400 nM T33966 CM1A0D 9943447 IC50 = 6400 nM T33966 CVK4L6 10418061 IC50 = 3900 nM T33966 C6FQ0R 10465893 IC50 = 1700 nM T33966 CT7IR8 12110710 IC50 > 100000 nM T33966 CFQW82 18955956 Ki = 207000 nM T33966 CYT07N 21575382 IC50 = 0.007 ug.mL-1 T33966 CG0M4T 21575383 IC50 = 3.4 ug.mL-1 T33966 C4UDA1 21606664 IC50 = 0.0052 ug.mL-1 T33966 CR1BW2 21606665 IC50 = 0.0076 ug.mL-1 T33966 C14ZMJ 24768537 Ki = 150 nM T33966 C7J1DP 24774575 Ki = 15000 nM T33966 CP2LY7 25033280 Ki = 17000 nM T33966 C4YKQ1 25033281 Ki = 22000 nM T33966 CA9D6R 25209871 IC50 = 0.12 ug.mL-1 T33966 C46SPD 44374719 Ki = 6500 nM T33966 C0NI9F 44374736 Ki = 5820 nM T33966 CFPX72 44374737 Ki = 4950 nM T33966 CPRQ07 44374750 Ki = 1200 nM T33966 C9RPC6 44374765 Ki = 1160 nM T33966 C1CPB2 44374994 Ki = 980 nM T33966 CXTF63 44374995 Ki = 560 nM T33966 CGD91Y 44374996 Ki = 5900 nM T33966 C4UBK7 44374998 Ki = 320 nM T33966 CG75AN 44377126 Ki = 1200 nM T33966 C6SV1C 44387258 IC50 = 1100 nM T33966 C06HJB 44446952 Ki = 11000 nM T33966 CNK7X5 44446953 Ki = 35000 nM T33966 CEB78N 44446954 Ki = 11000 nM T33966 CMO78A 44446956 Ki = 530 nM T33966 CV6H2M 44446957 Ki = 350 nM T33966 CF4KE1 44446959 Ki = 3600 nM T33966 CW9C0E 44446960 Ki = 7200 nM T33966 CQB5M0 44446963 Ki = 9900 nM T33966 C94POY 44446965 Ki = 5000 nM T33966 CBX2U9 44446967 Ki = 2300 nM T33966 CRZ6B3 44446968 Ki = 14000 nM T33966 CY9O4I 44446969 Ki = 8900 nM T33966 C4PQ7D 44446970 Ki = 1600 nM T33966 C96KIY 44446972 Ki = 5000 nM T33966 CK1EM5 44446974 Ki = 4600 nM T33966 C4V6RZ 44446975 Ki = 16000 nM T33966 CBL9E6 44446976 Ki = 1900 nM T33966 CVYX54 44446979 Ki = 3300 nM T33966 CAI9Z6 44446980 Ki = 4600 nM T33966 C86KVP 44446984 Ki = 11000 nM T33966 CYQN96 44452011 Ki = 2080 nM T33966 CFOM52 44452012 Ki = 790 nM T33966 CJ8G5P 44452013 Ki = 68000 nM T33966 CZI4H9 44452015 Ki = 62600 nM T33966 CC2IS3 44454957 Ki = 12000 nM T33966 C1ESI2 44454959 Ki = 12000 nM T33966 C8L0MV 44454960 Ki = 12000 nM T33966 CBG6T0 44454987 Ki = 15000 nM T33966 CN7UW3 44455013 Ki = 8900 nM T33966 CC5L7S 44455015 Ki > 50000 nM T33966 C6KDT1 44455016 Ki = 9300 nM T33966 CF4ML7 44455018 Ki = 14000 nM T33966 CZI6S1 44455047 Ki = 1700 nM T33966 C3UF6E 44455406 Ki = 5000 nM T33966 CJG71N 44455407 Ki = 32000 nM T33966 C0IR5W 44455428 Ki = 17000 nM T33966 C62KSV 44455429 Ki > 50000 nM T33966 CR9WL2 44455430 Ki = 11000 nM T33966 CXD0Q4 44558923 IC50 = 0.022 ug.mL-1 T33966 C48QBD 45101440 Ki = 160 nM T33966 CP43WZ 45484707 Ki = 430 nM T33966 C2Q9OC 45484717 Ki = 31000 nM T33966 C85MBH 112499885 Ki = 0.087 nM T33966 C2L8SI 112499886 Ki = 0.107 nM T33966 CS49EB 112499887 Ki = 0.04 nM T33966 CG9SC3 145949929 Ki = 289000 nM T33966 C8H1FK 145950532 Ki = 294000 nM T33966 CH02KU 145955234 Ki = 56000 nM T33966 CA6QF8 145956086 Ki = 413000 nM T33966 CZH6P7 145956217 Ki = 238000 nM T33966 CF01VH 145974566 Ki = 60400 nM T33966 CU65CB 155511784 Ki = 0.08 nM T33966 CFG96J 155514645 Ki = 5.9 nM T33966 CF64GH 155518335 Ki = 0.07 nM T33966 CY0H2S 155519530 Ki = 3.1 nM T33966 CA49SR 155523686 Ki = 1.7 nM T33966 C5X4TD 155524117 Ki = 0.1287 nM T33966 C4F1EB 155538870 Ki = 0.3 nM T33966 CD81NB 155547411 Ki = 1.2 nM T33966 D06LNX 3858 IC50 = 400 nM T33966 D0N4RO 44377139 Ki = 310 nM T06792 D00UVA 11556711 IC50 = 2420 nM T06792 D0SH3I 387447 IC50 = 3 nM T06792 D0DP0J 92135659 IC50 = 1840 nM T06792 D0VO0T 24800541 IC50 = 1 nM T06792 CLU69K 10628969 IC50 = 440 nM T06792 CU0FE7 24752894 IC50 = 104 nM T06792 CN62YJ 46850523 IC50 = 140 nM T06792 CEV5D1 49859748 IC50 = 10600 nM T06792 C3QG8L 59127842 IC50 = 36 nM T06792 C82JTA 71305068 IC50 = 21500 nM T06792 C45HOE 71562349 IC50 > 10000 nM T06792 CGY43C 78425867 IC50 = 1850 nM T06792 CC0OF1 101874274 IC50 = 300 nM T06792 CG0N1O 101874275 IC50 = 7100 nM T06792 CL50TR 101874276 IC50 = 7300 nM T06792 C0RY3V 101874277 IC50 = 6200 nM T06792 CVHC29 101874278 IC50 > 100000 nM T06792 C4VHU6 101874279 IC50 > 100000 nM T06792 C9C5OZ 117607839 IC50 = 3530 nM T06792 CLHS74 117607901 IC50 = 223 nM T06792 CW9R0U 117607904 IC50 = 0.623 nM T06792 C7QST8 117611788 IC50 = 51 nM T06792 CO1HJ9 117611880 IC50 = 140 nM T06792 C9YH1X 117611941 IC50 = 112 nM T06792 CO6E0B 118709670 IC50 = 170 nM T06792 C8WMH3 118709671 IC50 = 68 nM T06792 CZ8GE0 118709672 IC50 = 96 nM T06792 CZ70XF 118709673 IC50 = 67 nM T06792 C7C9PZ 118709674 IC50 = 220 nM T06792 CS05KF 118709675 IC50 = 22 nM T06792 C17ZTF 118709676 IC50 = 34 nM T06792 C0WZ3V 118709677 IC50 = 66 nM T06792 C14VLB 118709678 IC50 = 87 nM T06792 CO5CU1 118709679 IC50 = 42 nM T06792 C1RA9C 118709680 IC50 = 130 nM T06792 C9BWP4 145979302 IC50 = 5700 nM T06792 CN79HG 145979487 IC50 = 3500 nM T06792 CEI3U1 145979850 IC50 = 4800 nM T06792 CG6UL0 145980995 IC50 = 4000 nM T06792 CB67YT 145981691 IC50 = 16100 nM T06792 C41IRV 145981707 IC50 = 14000 nM T06792 CL1F8N 145982922 IC50 = 13000 nM T06792 C5X3GQ 145986425 IC50 = 12600 nM T06792 CRZE86 145986857 IC50 = 45000 nM T06792 CHWT73 145987085 IC50 = 8900 nM T06792 CM3H4F 145987197 IC50 = 4300 nM T06792 CNZ7R6 145987536 IC50 = 12500 nM T06792 C1EF3B 145988020 IC50 = 23800 nM T06792 CQIS01 145988427 IC50 = 7310 nM T06792 CE16JH 145989568 IC50 = 52000 nM T06792 CXG30R 145990249 IC50 = 21000 nM T06792 C8IL9E 145992200 IC50 = 10320 nM T06792 CBY18W 145992498 IC50 = 2770 nM T06792 C6GHQ9 145993211 IC50 = 59000 nM T06792 CEVY70 145993649 IC50 = 24600 nM T06792 CJO08K 145993925 IC50 = 8800 nM T06792 C8E6ZX 155514792 IC50 > 10000 nM T06792 CX76LO 155515463 IC50 > 10000 nM T06792 C53ZEN 155516179 IC50 > 100000 nM T06792 CM3BV8 155516620 IC50 > 100000 nM T06792 CE95IQ 155518158 IC50 > 100000 nM T06792 CNM0Q9 155521286 IC50 > 100000 nM T06792 CZKF54 155521690 IC50 > 10000 nM T06792 CB0WG8 155522381 IC50 = 743.5 nM T06792 C8GNQ9 155522828 IC50 > 25000 nM T06792 CW75YK 155523151 IC50 > 100000 nM T06792 CAC34Y 155527225 IC50 = 3100 nM T06792 CUP2B4 155531358 IC50 = 415 nM T06792 C2NTI6 155538936 IC50 > 100000 nM T06792 C6OIY3 155541618 IC50 > 100000 nM T06792 C12LPX 155551071 IC50 > 10000 nM T06792 CBHM14 155553205 IC50 > 100000 nM T06792 C35NJC 155553210 IC50 > 10000 nM T06792 CI15FC 155553565 IC50 > 10000 nM T06792 CVJ3E7 155553910 IC50 > 100000 nM T06792 C6YP0L 155554916 IC50 > 100000 nM T06792 C5Z7YC 155567712 IC50 > 10000 nM T06792 C4ZV3Q 155568941 IC50 > 10000 nM T06792 D0Q4MO 23642227 IC50 = 287 nM T01943 D04AIT 5280445 IC50 = 5000 nM T01943 D0K8KX 5280343 IC50 = 1500 nM T01943 D0L4FS 5280961 IC50 = 7000 nM T01943 D0U2BH 65064 IC50 = 400 nM T01943 CY0AL9 72279 IC50 = 30000 nM T01943 CNIW58 107905 IC50 = 400 nM T01943 CDZ65K 199472 IC50 = 600 nM T01943 CN7AQ6 15958429 IC50 = 14 ug.mL-1 T01943 CZR73C 16072317 IC50 = 12.5 ug.mL-1 T01943 C20YLR 22600366 IC50 = 0.58 ug.mL-1 T01943 C15VRN 44412009 IC50 = 40000 nM T01943 C6XHE9 49770727 IC50 = 12 ug.mL-1 T01943 CG4H0W 71768351 IC50 > 100000 nM T01943 CMAP17 71768352 IC50 = 16300 nM T01943 CW0T6G 72703050 IC50 > 100000 nM T01943 CPZO91 72703242 IC50 > 100000 nM T01943 CQ2IU6 72703243 IC50 = 90000 nM T01943 C0B3KS 72703244 IC50 = 13000 nM T01943 CE6HI7 72703245 IC50 = 28000 nM T01943 CJ12BK 72703246 IC50 = 10000 nM T01943 CESN04 73347724 IC50 > 100000 nM T01943 D01KKU 5281894 IC50 = 20000 nM T01943 D02TVS 985 IC50 > 100 ug.mL-1 T01943 D0MF5Y 5281614 IC50 = 2000 nM T01943 D0NJ4H 5281670 IC50 = 8000 nM T01943 D0RB1V 6419835 IC50 = 400 nM T01943 D0S9YX 5280373 IC50 = 8000 nM T01943 D0SY2M 5281708 IC50 = 30000 nM T01943 D0T3PW 5281672 IC50 = 2000 nM T19229 D01KKQ 135400182 IC50 = 99.5 nM T19229 D02LWU 148121 IC50 = 57 nM T19229 D0SV8E 126941 IC50 = 121 nM T19229 D0Y4GO 135410875 IC50 = 13.2 nM T19229 CPM3L5 67092576 IC50 > 1000 nM T19229 CTK64O 67092918 IC50 > 1000 nM T19229 C87FBU 135455948 IC50 = 80.2 nM T19229 CF8D5O 135465664 IC50 > 1000 nM T19229 C9Z4ES 135567027 IC50 = 5.21 nM T19229 C14LTO 135567028 IC50 = 43.4 nM T19229 CF39AI 135567029 IC50 = 3.34 nM T19229 C8N7ES 135567030 IC50 = 41.5 nM T19229 CGM2V5 135567031 Ki = 420 nM T19229 CFE2O7 135567034 IC50 = 40 nM T19229 C8KVP5 135567035 IC50 = 6.51 nM T19229 CSQX75 135567163 IC50 = 87.4 nM T19229 CQF8P5 135800109 IC50 = 9.71 nM T19229 C6XK3M 135862924 Ki = 100 nM T19229 CL8VN5 136015502 IC50 = 312 nM T19229 CR7UY3 136044173 IC50 > 1000 nM T19229 C0Q5FI 136044174 IC50 > 1000 nM T19229 CGX68Y 136044175 IC50 > 1000 nM T19229 C4C9FN 136044176 IC50 > 1000 nM T19229 CIPD35 136044177 IC50 > 1000 nM T19229 CZG8W6 136059167 IC50 = 30.4 nM T19229 CZC95Y 136059168 IC50 > 1000 nM T19229 CG2ID9 136059169 IC50 > 1000 nM T19229 C2WH0S 136059178 IC50 > 1000 nM T19229 CB3GL7 136059191 IC50 > 1000 nM T19229 CCHG08 136059192 IC50 > 1000 nM T19229 C4Q1HF 136180345 IC50 = 141 nM T19229 CDC83K 136180346 IC50 = 57.4 nM T19229 CF7NW6 136180347 IC50 > 1000 nM T19229 CPH52E 137150145 IC50 > 1000 nM T19229 C9XD1M 137150146 IC50 = 747 nM T19229 CHDB56 137150160 IC50 = 48.6 nM T19229 CUF8R1 155515541 IC50 = 207 nM T19229 CMKA64 155517044 IC50 = 81.7 nM T19229 CCL3Y9 155518053 IC50 = 20.4 nM T19229 C91SVN 155519837 IC50 = 57.5 nM T19229 CO7BN6 155524531 IC50 > 1000 nM T19229 CT70WU 155530762 IC50 = 5.01 nM T19229 CX42MF 155532591 IC50 = 267 nM T19229 CFU98A 155534971 IC50 = 88.5 nM T19229 C4K2RU 155538415 IC50 > 1000 nM T19229 C27BIX 155539477 IC50 > 1000 nM T19229 C6S7OC 155548982 IC50 = 3.82 nM T19229 CX3K8F 155549935 IC50 = 4.57 nM T19229 CJ0MK5 155554671 IC50 = 67 nM T19229 CYQ0I9 155555353 IC50 = 109 nM T90987 CJS23I 9868333 Ki = 7800 nM T90987 CY08WJ 10322755 Ki = 7800 nM T90987 C8C5AV 11294179 Ki > 1000 nM T90987 CZB81D 44395506 IC50 = 79 nM T90987 C52ESR 66559934 IC50 > 50000 nM T90987 C57ARI 66560021 IC50 > 50000 nM T90987 CU58DB 66560022 IC50 > 50000 nM T90987 C16RDM 66560389 IC50 > 50000 nM T90987 C8RZG9 66560479 IC50 > 50000 nM T90987 CKW2Q5 71453375 IC50 > 50000 nM T90987 D0H6CK 10160968 Ki = 776 nM T06569 D00STL 644241 Ki = 461 nM T06569 D01MUR 68844 Ki = 0.9 nM T06569 D02PJA 24841 Ki = 810000 nM T06569 D03QGM 5355 Ki = 0.8 nM T06569 D03RTS 2662 Ki = 94 nM T06569 D03UOT 785 Ki = 521000 nM T06569 D05OFX 219078 Ki = 412 nM T06569 D05UYW 5284549 Ki = 10 nM T06569 D07HBX 338 Ki = 11900 nM T06569 D07INV 3295 Ki = 43 nM T06569 D07VDZ 5284627 Ki = 45 nM T06569 D09NIA 2732 Ki = 1347 nM T06569 D09VAZ 5565 Ki = 43000 nM T06569 D0AZ3C 5291 Ki = 392 nM T06569 D0AZ8C 5213 Ki = 9700 nM T06569 D0C2II 4100 Ki = 10 nM T06569 D0C8FX 3005837 Ki = 2410 nM T06569 D0E1SW 1986 Ki = 11 nM T06569 D0H8FH 3702 Ki = 1606 nM T06569 D0J4GO 3038 Ki = 79 nM T06569 D0J7RK 36811 Ki = 9470 nM T06569 D0K0OZ 5702160 Ki = 98.2 nM T06569 D0K1QD 3998 Ki = 4800 nM T06569 D0K8KX 5280343 Ki = 6170 nM T06569 D0L4JT 5333 Ki = 941 nM T06569 D0L6DA 119607 Ki = 572 nM T06569 D0OT0O 44561 Ki = 1810000 nM T06569 D0PQ3G 3440 Ki = 245 nM T06569 D0SH3I 387447 Ki = 4380 nM T06569 D0U5QK 1983 Ki = 658000 nM T06569 D0Y2IZ 5560 Ki = 2459 nM T06569 D0Z3EI 6038 Ki = 33 nM T06569 D04IIU 216468 Ki = 47 nM T06569 D05NJI 5287541 Ki = 653 nM T06569 D06PII 5356 Ki = 134 nM T06569 D08BXT 1102 Ki = 1410 nM T06569 D0L6HN 996 Ki = 208000 nM T06569 D0U3EP 445154 Ki = 8070 nM T06569 D0V0UK 82267 Ki = 0.07 nM T06569 D03SLR 445858 Ki = 8450 nM T06569 D0NH9P 135 Ki = 5700 nM T06569 D0LD9S 1103 Ki = 990 nM T06569 CI0WH9 72 Ki = 4720 nM T06569 CUT2V4 260 Ki = 730000 nM T06569 COV5W3 402 Ki = 710000 nM T06569 CSZ43B 540 Ki = 690000 nM T06569 C97QXH 767 Ki = 690000 nM T06569 C39CTO 768 Ki = 70000 nM T06569 C1QDT0 781 Ki = 890000 nM T06569 CAD4R0 798 Ki = 3630 nM T06569 CW0R2L 944 Ki = 760000 nM T06569 CQV86E 1100 Ki = 14200000 nM T06569 C8W7BZ 1118 Ki = 9900000 nM T06569 CU12QE 1203 Ki = 4910 nM T06569 C5L7VX 2871 Ki = 2230 nM T06569 CJ2F6P 5056 Ki = 8630 nM T06569 CDJ4K6 5987 Ki = 0.09 nM T06569 CUP2F4 7043 Ki = 234700 nM T06569 C1CVT7 7121 Ki = 24420 nM T06569 C6NC4O 7414 Ki = 5100 nM T06569 CJKY76 7420 Ki = 3170 nM T06569 CIU0C8 7519 Ki = 234700 nM T06569 CUG8B9 11418 Ki = 402300 nM T06569 CCPT31 11419 Ki = 427100 nM T06569 CUA0L6 14917 Ki = 600000 nM T06569 C3NG2U 24529 Ki = 820000 nM T06569 CFM9L6 24530 Ki = 70000 nM T06569 C4OU6D 35703 Ki = 82300 nM T06569 C1N6SE 61127 Ki = 29138 nM T06569 CE5RZ1 76509 Ki = 780 nM T06569 CX47BZ 78479 Ki = 53000 nM T06569 CEC01M 97598 Ki = 12840 nM T06569 CN19UT 129695 Ki = 110 nM T06569 CUX39B 132037 Ki = 3410 nM T06569 CVB67D 134560 Ki = 73 nM T06569 CD2HC7 138614 Ki = 405600 nM T06569 C8AO0Z 165323 Ki = 114 nM T06569 C1QOB5 284045 Ki = 382473 nM T06569 CT3ZU4 388776 Ki = 1100 nM T06569 CH21KA 389641 Ki = 104000 nM T06569 C6CQO3 389642 Ki = 114000 nM T06569 CNPZ40 394897 Ki = 765 nM T06569 C4TD8M 2388085 Ki > 10000 nM T06569 C21FUI 2801263 Ki = 3790 nM T06569 CE2GR3 2900806 Ki = 109000 nM T06569 CI8JY0 5172475 Ki = 740 nM T06569 C9L8AX 6537802 Ki = 41 nM T06569 C65FRB 6852128 Ki = 136 nM T06569 CKCM96 7463376 Ki = 8580 nM T06569 CDCP43 7766335 Ki = 420 nM T06569 CY47OI 9998322 Ki = 24 nM T06569 CWM01R 10059806 Ki = 13692 nM T06569 CD58EL 10083644 Ki = 730 nM T06569 C58IYR 10366827 Ki = 590 nM T06569 C3HBY6 10375558 Ki = 4150 nM T06569 C73KXU 10586607 Ki = 6700 nM T06569 C9TSQ6 10632698 Ki = 43100 nM T06569 C8C6ER 11069133 Ki = 41 nM T06569 C39IDU 11183936 Ki = 12010 nM T06569 CHC42Y 11245700 Ki = 654 nM T06569 CA6T0Z 11322287 Ki = 11660 nM T06569 CXB86F 11579563 Ki = 12530 nM T06569 CDU79V 11637531 Ki = 10820 nM T06569 CX4W3J 11701693 Ki = 9870 nM T06569 CV7HN1 11795548 Ki = 65 nM T06569 CMPA32 12066940 Ki > 500000 nM T06569 CB15KR 12066941 Ki > 500000 nM T06569 CREV05 12140130 Ki = 12430 nM T06569 CHOG93 14611919 Ki = 2650 nM T06569 C8PER5 15938557 Ki > 500000 nM T06569 CC0Z4V 16119626 Ki = 510 nM T06569 C6SFI8 18268734 Ki > 10000 nM T06569 C61KUX 21726402 Ki = 9680 nM T06569 C54IUM 21778115 Ki = 17830 nM T06569 C27BJH 21778117 Ki = 17430 nM T06569 C9U4TE 22313850 Ki = 1230 nM T06569 CICR37 23426698 Ki = 38190 nM T06569 CPN2T5 25392418 Ki > 10000 nM T06569 C82MRL 44144383 Ki = 25 nM T06569 CI3O9B 44395149 Ki = 147 nM T06569 CZ4DF9 44399462 Ki = 76 nM T06569 CD5MJ6 44399571 Ki = 59 nM T06569 C2T7MB 44399654 Ki = 749 nM T06569 C8E0MV 44552472 Ki = 9210 nM T06569 CKG53H 44552473 Ki = 1920 nM T06569 C17XAJ 44552559 Ki = 4170 nM T06569 CF0KQ8 44581932 Ki = 73 nM T06569 C23MVW 45269009 IC50 = 35700 nM T06569 C0RG8K 45269749 Ki > 100000 nM T06569 CV5RQ3 45484187 Ki = 4300 nM T06569 CTG20B 45485271 Ki = 100 nM T06569 CK4U0V 45485283 Ki = 5600 nM T06569 CHE08Y 46225608 Ki = 10230 nM T06569 CIE2H3 46225609 Ki = 9640 nM T06569 CF42NR 46225631 Ki = 7610 nM T06569 C0ZG3L 46225639 Ki = 7960 nM T06569 CGW1I5 46225644 Ki = 7840 nM T06569 CEOQ06 46225645 Ki = 8310 nM T06569 CR0WO3 46225646 Ki = 8540 nM T06569 CC2BL5 46225656 Ki = 8980 nM T06569 CW52PZ 46225672 Ki = 4950 nM T06569 CXJ1C9 46225673 Ki = 4310 nM T06569 C93AIR 46899573 Ki = 156000 nM T06569 CJ0R2O 46911381 Ki = 921 nM T06569 CF89ML 53307609 Ki = 29670 nM T06569 C0NUM6 53386724 Ki = 980 nM T06569 C54FGU 53386866 Ki = 543 nM T06569 CRI54V 53386867 Ki = 1035 nM T06569 CUX7S4 53386868 Ki = 814 nM T06569 CIJ9V0 56684131 Ki = 8140 nM T06569 CH52DA 56921864 Ki = 8950 nM T06569 CUR32K 57334711 Ki = 480 nM T06569 C2CD1R 57334712 Ki = 470 nM T06569 C1K0DM 57334713 Ki = 470 nM T06569 CP7YR5 57345662 Ki = 8 nM T06569 C13FJU 57392368 Ki = 510 nM T06569 CY5G4Z 57395885 Ki = 960 nM T06569 C5RX6H 57396029 Ki = 5240 nM T06569 CP75OF 57397664 Ki = 158592 nM T06569 CUAG84 57397836 Ki = 765300 nM T06569 CW43HV 57397837 Ki = 5590 nM T06569 C1MCW8 57399336 Ki = 919182 nM T06569 C2CAM1 57399491 Ki = 4810 nM T06569 C2J7GW 66572313 Ki = 35450 nM T06569 C7J5RN 66573254 Ki = 45360 nM T06569 CQR91N 70692438 Ki = 28170 nM T06569 CWJ0Q8 70696540 Ki = 11143 nM T06569 CXJ16H 71450117 Ki = 8055 nM T06569 CB8JA3 71455488 Ki = 9340 nM T06569 C02UHX 71455489 Ki = 7116 nM T06569 CICJ97 71457274 Ki = 9280 nM T06569 CMHG14 71521493 Ki = 6200 nM T06569 CHN53G 71521494 Ki = 7700 nM T06569 CZJ5M6 71521495 Ki = 7900 nM T06569 CFBE53 71521496 Ki > 100000 nM T06569 CME27W 71521497 Ki = 8100 nM T06569 C24XWU 71521575 Ki = 8800 nM T06569 CJF68W 71521576 Ki > 100000 nM T06569 CX82JD 72696463 Ki = 130 nM T06569 COCV73 72696591 Ki = 1388 nM T06569 C5KHD7 72696592 Ki = 220 nM T06569 C4FBA6 72696593 Ki = 274 nM T06569 CO1JM5 72696594 Ki = 167 nM T06569 CUF61Q 72696595 Ki = 148 nM T06569 CO1JT3 73054728 Ki = 857 nM T06569 CDGZ03 101879106 Ki > 120 nM T06569 CY6ER7 101879108 Ki > 120 nM T06569 C0D1SQ 118724328 Ki > 120 nM T06569 C89YTC 118724329 Ki > 120 nM T06569 CBT87C 118724330 Ki > 120 nM T06569 C49AWZ 118724331 Ki > 120 nM T06569 CH1N0C 122193189 Ki = 560 nM T06569 C19HVL 122193190 Ki = 740 nM T06569 C5TQJ1 122193251 Ki = 540 nM T06569 C8XCL0 122193252 Ki = 470 nM T06569 CIX41M 138393379 Ki > 10000 nM T06569 CBOM51 138753317 Ki > 10000 nM T06569 COP4Q6 155516517 Ki = 9192 nM T06569 CAG9L4 155517430 Ki = 2440 nM T06569 CP49HE 155520274 Ki = 7428 nM T06569 CTJ3I7 155530506 Ki = 7218 nM T06569 CT5NG1 155534179 Ki > 10000 nM T06569 CVU5P6 155535355 Ki > 10000 nM T06569 C8RV6T 155541805 Ki > 10000 nM T06569 CU1NE7 155549031 Ki > 10000 nM T06569 CWB82E 155555878 Ki > 10000 nM T06569 CH5VU6 155568899 Ki > 10000 nM T06569 D00IUB 13019 Ki = 13700 nM T06569 D00RNZ 910172 Ki = 93100 nM T06569 D00XJA 711717 Ki = 65200 nM T06569 D00YEF 148885 Ki = 1414 nM T06569 D01BUB 94952 Ki = 90600 nM T06569 D01STY 9861037 Ki = 1024 nM T06569 D02DBP 5054 Ki = 550000 nM T06569 D02QGI 273 Ki = 740 nM T06569 D03NBX 637308 Ki = 770 nM T06569 D03ZMQ 323 Ki = 2000 nM T06569 D04CVC 4687472 Ki = 96 nM T06569 D04NSN 169682 Ki = 813 nM T06569 D05QUG 45485279 Ki > 500000 nM T06569 D05TLB 11117301 Ki = 795 nM T06569 D05WQF 637540 Ki > 1000000 nM T06569 D05XZM 10081162 Ki = 6680 nM T06569 D06DYP 234562 Ki = 44500 nM T06569 D06TPF 1057 Ki = 520 nM T06569 D07MTM 403 Ki = 23500 nM T06569 D07QJJ 289 Ki = 606000 nM T06569 D07TAJ 914298 Ki = 6600 nM T06569 D09JPC 16402 Ki = 720 nM T06569 D09PWX 8739 Ki = 887 nM T06569 D09QHC 7370 Ki = 2970 nM T06569 D09WSJ 19772348 Ki = 1334 nM T06569 D09WVV 8111 Ki = 11500 nM T06569 D0A0YX 5143 Ki = 935 nM T06569 D0A1CM 5281855 Ki = 7060 nM T06569 D0A6HS 6852129 Ki = 103 nM T06569 D0AU0M 637542 Ki = 6720 nM T06569 D0C7LR 313 Ki = 720000 nM T06569 D0D4OV 20043772 Ki = 1020 nM T06569 D0D6UR 12394434 Ki > 500000 nM T06569 D0E8CC 18794 Ki = 93 nM T06569 D0EJ9B 66827 Ki = 0.82 nM T06569 D0G0FJ 11206245 Ki = 1090 nM T06569 D0G3BI 25090 Ki = 54700 nM T06569 D0H3NS 10752 Ki = 76300 nM T06569 D0L5TZ 20195365 Ki = 9300 nM T06569 D0LU4S 156219 Ki = 13000 nM T06569 D0M3PO 69561 Ki = 955 nM T06569 D0M6RM 7365 Ki = 13.9 nM T06569 D0N1AW 45485270 Ki = 1300 nM T06569 D0NN3Q 78105 Ki = 1275 nM T06569 D0OI1H 72894 Ki = 772 nM T06569 D0OT5L 1631814 Ki = 7400 nM T06569 D0P6AM 3526523 Ki = 4680 nM T06569 D0Q7DJ 10742 Ki = 7550 nM T06569 D0R4WJ 16129778 Ki = 17800 nM T06569 D0R7QY 127676 Ki = 1860 nM T06569 D0RB0D 44268050 Ki > 500000 nM T06569 D0TY8X 31036 Ki = 86 nM T06569 D0U4BB 10748 Ki = 5500 nM T06569 D0V9EN 689043 Ki = 7330 nM T06569 D0VD7H 84724 Ki = 798 nM T06569 D0X5HL 15107 Ki = 640 nM T06569 D0X6IE 4422372 Ki = 55 nM T06569 D0Y3TZ 370 Ki = 6130 nM T06569 D0YU8J 1502014 Ki = 1097 nM T06569 D0Z1HY 67136 Ki = 608 nM T06569 D0ZC3W 6269 Ki = 1582 nM T03529 D07XOD 2733079 IC50 = 11000 nM T03529 CCI13U 11536910 IC50 = 20400 nM T03529 CN8LG9 13171484 IC50 = 37000 nM T03529 CXC3W5 20377108 IC50 = 28400 nM T03529 C3PDB6 20377110 IC50 = 122000 nM T03529 CI3Q2W 25125116 IC50 = 312000 nM T03529 C5NER0 25125122 IC50 = 7100 nM T03529 CGF7A0 25125458 IC50 = 12800 nM T03529 CS1RD3 25125461 IC50 = 7600 nM T03529 CJ4I7C 25125799 IC50 = 31600 nM T03529 CM6EV5 70681820 IC50 = 7500 nM T03529 CUYZ39 70681821 IC50 = 5600 nM T03529 C9BP5R 70681822 IC50 = 5200 nM T03529 CP6E4R 70681828 IC50 = 16400 nM T03529 CBHO57 70681829 IC50 = 11800 nM T03529 COQC31 70681830 IC50 = 17500 nM T03529 CUF80Q 70681831 IC50 = 15700 nM T03529 CXU67P 70681832 IC50 = 119000 nM T03529 C45NUH 70681833 IC50 = 70600 nM T03529 CV91MS 70681834 IC50 = 194000 nM T03529 CDN0C4 70683924 IC50 = 39800 nM T03529 CH2PL3 70683932 IC50 = 9900 nM T03529 C8E4JH 70683933 IC50 = 7700 nM T03529 CA27DC 70683934 IC50 = 98000 nM T03529 CUC9K6 70686055 IC50 = 17200 nM T03529 C48CLJ 70686056 IC50 = 12300 nM T03529 C59QXF 70688191 IC50 = 21300 nM T03529 C3S9IJ 70688192 IC50 = 11600 nM T03529 C1S3IH 70690203 IC50 = 11400 nM T03529 CJ5PK6 70690208 IC50 = 56000 nM T03529 CL0JW1 70692374 IC50 = 16200 nM T03529 CNW8O1 70692382 IC50 = 13200 nM T03529 CM2KW1 70692383 IC50 = 8400 nM T03529 C04XZL 70694433 IC50 = 6200 nM T03529 CD5O8R 70694437 IC50 = 9500 nM T03529 CTLH58 70696507 IC50 = 10900 nM T03529 C3TV8N 70696508 IC50 = 18700 nM T03529 D05AMQ 6539137 IC50 = 83500 nM T03529 D0M5DR 57330144 IC50 = 36100 nM T97822 D03RTS 2662 IC50 = 89 nM T97822 D0GY5Z 2244 IC50 = 15000 nM T97822 D0R1RS 3715 IC50 = 10 nM T97822 D0U2FN 71321 IC50 = 6500000 nM T97822 D05WPQ 6438354 IC50 = 3200 nM T97822 D09QRO 55390 IC50 = 10000 nM T97822 D0DP8P 47795 IC50 = 5800 nM T97822 D0JY4Y 443292 IC50 > 100000 nM T97822 D0N1SU 133021 IC50 = 160 nM T97822 D0O8ZE 5059 IC50 = 5300 nM T97822 D0S8YL 3969 IC50 = 44000 nM T97822 CH0L7P 71697 IC50 = 950000 nM T97822 CI5D9O 92656 IC50 = 100 nM T97822 CV7L0G 112230 IC50 = 100000000 nM T97822 CT2XZ0 116545 IC50 = 7079457.84 nM T97822 CAT4E3 129615 IC50 = 3388441.56 nM T97822 CCJ76H 512829 IC50 = 9000 nM T97822 CE2BC3 512830 IC50 = 14000 nM T97822 C16VBD 512831 IC50 = 12000 nM T97822 CT7E6Y 573683 IC50 > 800000 nM T97822 CZ0AH3 638278 IC50 = 130000 nM T97822 C6EVL8 854057 IC50 = 3467368.5 nM T97822 CQM64G 3037018 IC50 = 800 nM T97822 COH1C4 3052566 IC50 = 446683.59 nM T97822 C82IPJ 3052567 IC50 = 912010.84 nM T97822 C4VBK3 3253091 IC50 = 50000 nM T97822 CU86JL 4618600 IC50 = 40000 nM T97822 C4M1JC 5709318 IC50 = 44000 nM T97822 COQ7T3 5973690 IC50 = 63000 nM T97822 C3G7DT 6365297 IC50 = 4200 nM T97822 C40FZG 6366698 IC50 = 1300 nM T97822 C02AQY 6366699 IC50 ~ 1000 nM T97822 CWK1F9 6438990 IC50 = 110 nM T97822 C62UOZ 6439221 IC50 = 780 nM T97822 CHQ4Z3 6439222 IC50 = 1300 nM T97822 COC86Q 6439421 IC50 = 390 nM T97822 CLJ91K 6439912 IC50 = 260 nM T97822 C82TEX 7515046 IC50 < 10000 nM T97822 CUS6L8 9822795 IC50 = 30 nM T97822 C5C9ET 10042219 IC50 > 100000 nM T97822 C9T7YV 10063338 IC50 > 100000 nM T97822 CBL7R3 10220019 IC50 = 400 nM T97822 C2WE0I 10246235 IC50 = 9600 nM T97822 C20BTQ 10313997 IC50 = 5500 nM T97822 C8EQI3 10334136 IC50 > 100000 nM T97822 CC1UF0 10335738 IC50 > 100000 nM T97822 C25MYB 10425738 IC50 > 100000 nM T97822 CPR7J0 10469807 IC50 = 12589254.12 nM T97822 C6JI5F 10492615 IC50 > 300000 nM T97822 C0NRO9 10513373 IC50 = 570000 nM T97822 CK0OL2 10704667 IC50 = 27000 nM T97822 CUOI16 10729548 IC50 = 26000 nM T97822 C8IBM2 10801359 IC50 = 250000 nM T97822 CC8S6O 10801786 IC50 = 37000 nM T97822 CDZ94R 10826230 IC50 = 29000 nM T97822 CGLQ72 11723348 IC50 > 100000 nM T97822 CH9VC8 13245625 IC50 > 10000 nM T97822 CRA87I 13556944 IC50 = 14125375.45 nM T97822 C0P5AK 13914227 IC50 > 100000 nM T97822 C49OGE 13914253 IC50 > 100000 nM T97822 C4U3RD 14006855 IC50 = 5000 nM T97822 C6EZ0K 14312565 IC50 > 10000 nM T97822 C2X8PQ 14416570 IC50 = 34 nM T97822 C5PT1G 14416572 IC50 670 nM T97822 C1SG0F 14416576 IC50 = 10000 nM T97822 CRYI80 14416580 IC50 = 610 nM T97822 C27NOS 14416585 IC50 < 10000 nM T97822 C6BP2F 14416587 IC50 < 1000 nM T97822 CER87K 14762923 IC50 = 13803842.65 nM T97822 CGYF09 14762938 IC50 = 501187233.6 nM T97822 CX9AH8 14762939 IC50 = 501187233.6 nM T97822 CU3OT4 14762940 IC50 = 165958690.7 nM T97822 CXT3B5 14762942 IC50 = 100000000 nM T97822 CNZ45J 14762943 IC50 = 91201083.94 nM T97822 CL2A1E 14762944 IC50 = 91201083.94 nM T97822 C78IHC 14762948 IC50 = 50118723.36 nM T97822 CBL2O8 14762951 IC50 = 14791083.88 nM T97822 C8NKZ7 14762954 IC50 = 7079457.84 nM T97822 C4PS0F 14771889 IC50 < 10000 nM T97822 CV41BE 14771890 IC50 = 3100 nM T97822 CCX7K5 14771891 IC50 = 1400 nM T97822 CG57JP 14771892 IC50 = 1300 nM T97822 C91VJM 14771893 IC50 = 230 nM T97822 C0EMA5 14771894 IC50 < 1000 nM T97822 CZ4WJ2 14771895 IC50 = 730 nM T97822 CV5YH8 14771896 IC50 < 10000 nM T97822 C3HNQ2 14771897 IC50 < 10000 nM T97822 CH0TC9 14771898 IC50 < 10000 nM T97822 CX3N7Z 14771899 IC50 = 11000 nM T97822 CX7VA0 14771900 IC50 < 10000 nM T97822 CZC2D4 14771901 IC50 < 10000 nM T97822 CTY60Q 14771902 IC50 < 10000 nM T97822 C0D5OC 14771903 IC50 = 1500 nM T97822 CS3V5C 14771904 IC50 < 10000 nM T97822 CNH5M1 14771905 IC50 = 3200 nM T97822 CXN94C 14771906 IC50 = 510 nM T97822 CY2HF8 14771907 IC50 = 1400 nM T97822 CP5M9A 14771908 IC50 = 190 nM T97822 CI3XK7 14771909 IC50 < 10000 nM T97822 C8NTK2 14771910 IC50 = 750 nM T97822 C8H6XA 14771911 IC50 = 2500 nM T97822 CK53TR 14771912 IC50 < 1000 nM T97822 C10DIY 14771913 IC50 < 1000 nM T97822 C2F9TX 14771915 IC50 = 1100 nM T97822 C83VPQ 14771916 IC50 = 710 nM T97822 CA0C7U 14771917 IC50 = 1000 nM T97822 CK0AR5 14771918 IC50 < 1000 nM T97822 C8SRH6 14771919 IC50 > 10000 nM T97822 CCS9Y4 14771920 IC50 > 10000 nM T97822 C47LJK 14771921 IC50 > 10000 nM T97822 C9OWP0 14771922 IC50 = 1300 nM T97822 C1Z6FX 14771923 IC50 = 780 nM T97822 CHI8M3 14771924 IC50 < 10000 nM T97822 C4JX5S 14771927 IC50 = 590 nM T97822 CRGJ45 14771928 IC50 < 10000 nM T97822 C7L2ZJ 14771929 IC50 = 400 nM T97822 CXAG49 14771930 IC50 < 1000 nM T97822 C54ITL 14771931 IC50 = 110 nM T97822 CC4LM1 14771932 IC50 < 10000 nM T97822 CU6TO3 14771933 IC50 < 10000 nM T97822 C08CRZ 14771934 IC50 = 630 nM T97822 CA3D5U 14771935 IC50 = 1000 nM T97822 CZU2H5 14771936 IC50 = 300 nM T97822 C3B0LX 14771937 IC50 < 10000 nM T97822 CRT9E4 14771938 IC50 > 10000 nM T97822 C18DXV 14977360 IC50 = 71000 nM T97822 CD8YK4 15256755 IC50 = 140000 nM T97822 C53TQI 19044744 IC50 > 100000 nM T97822 CGPW68 19044748 IC50 > 100000 nM T97822 CLN6S5 19044753 IC50 > 100000 nM T97822 CR1W2E 19934882 IC50 > 100000 nM T97822 CF30ID 23275601 IC50 = 66069344.8 nM T97822 CUC36F 23680215 IC50 = 9772372.21 nM T97822 CN6F4H 23680216 IC50 = 4365158.32 nM T97822 C2JUV4 23680221 IC50 = 17782794.1 nM T97822 CHY73S 23680224 IC50 = 524807460.3 nM T97822 C7HV8Y 23680227 IC50 = 70794578.44 nM T97822 CZV8U1 23680228 IC50 = 4677351.41 nM T97822 C54NWH 23680229 IC50 = 741310241.3 nM T97822 CNU43B 23680230 IC50 = 891250938.1 nM T97822 C8A9UV 23689693 IC50 = 562341325.2 nM T97822 CJ1Z9S 44315480 IC50 = 794328234.7 nM T97822 C7UG4F 44315519 IC50 = 15135612.48 nM T97822 C8FEV0 44319113 IC50 = 25000 nM T97822 C1ZH6U 90664380 IC50 > 100000 nM T97822 C5T4EQ 131801158 IC50 = 23 nM T97822 C6JF0E 135616214 IC50 = 2500 nM T97822 CH4YE6 135987613 IC50 > 10000 nM T97822 CFNO28 145950339 IC50 = 34 nM T97822 CG37FR 145950583 IC50 = 27 nM T97822 CCN16Y 145952805 IC50 = 44 nM T97822 C2FVO7 145953074 IC50 = 38 nM T97822 C19TPY 145958203 IC50 = 50 nM T97822 C1BLR8 145959460 IC50 = 33 nM T97822 CUXQ13 145971245 IC50 = 41 nM T97822 C8U9TX 145971276 IC50 = 28 nM T97822 D00GBX 71751 IC50 = 5.7 nM T97822 D01TOR 667555 IC50 = 50000 nM T97822 D05EMX 14076674 IC50 = 10000000 nM T97822 D06VWH 11758240 IC50 = 2 nM T97822 D08GOT 13752584 IC50 = 4897788.19 nM T97822 D09AUL 10266864 IC50 = 51000 nM T97822 D0EW3L 5281222 IC50 = 120000 nM T97822 D0M6UM 129265 IC50 = 22000 nM T97822 D0P1LP 7090 IC50 = 12000 nM T97822 D0U0YE 14762941 IC50 = 165958690.7 nM T97822 D0U2YL 131820 IC50 = 36000 nM T97822 D0U8YQ 921562 IC50 = 14000 nM T23673 D00STL 644241 IC50 = 1100 nM T23673 D05ROI 44462760 IC50 = 150 nM T23673 D09GDD 11167602 IC50 = 1.5 nM T23673 D0E6XR 3062316 IC50 = 164 nM T23673 D0R0MW 5329102 IC50 > 10000 nM T23673 D0W5HK 216239 IC50 = 3 nM T23673 D0Y9EW 42611257 IC50 = 48 nM T23673 D03AND 11656518 IC50 = 19 nM T23673 D04AHQ 71721540 IC50 = 42 nM T23673 D0B9BU 6918454 IC50 = 12 nM T23673 D0E3TC 44259 IC50 = 130 nM T23673 D0F5JZ 24180719 Ki = 3.3 nM T23673 D0M6BD 16719221 IC50 = 56 nM T23673 D0N8RV 9868037 IC50 = 41 nM T23673 D0T4QA 90456533 IC50 = 0.2 nM T23673 D03BNU 59604787 IC50 > 3500 nM T23673 D02YAQ 6603857 IC50 = 49000 nM T23673 D0A9KI 9863367 IC50 > 50 nM T23673 D0F8DL 176155 IC50 = 330 nM T23673 D0T3ME 156422 IC50 = 1400 nM T23673 CB37VR 5034 IC50 = 77 nM T23673 C1YNB7 447721 IC50 > 1000 nM T23673 C73DGZ 656907 IC50 > 1000 nM T23673 CXJ40G 667570 IC50 = 1300 nM T23673 C3OKI4 1228884 IC50 = 1300 nM T23673 C1SVD2 2132479 IC50 = 6500 nM T23673 CVE5C7 2807754 IC50 = 6800 nM T23673 CK2QF5 4163701 IC50 = 17000 nM T23673 C2N9KR 5353919 IC50 = 9 nM T23673 C3G5DZ 9797863 IC50 = 6700 nM T23673 C1A0GW 9798540 IC50 = 1100 nM T23673 CR6T9K 9800910 IC50 = 11000 nM T23673 CNJE78 9811391 IC50 = 1500 nM T23673 CJ7TP1 9818992 IC50 = 4000 nM T23673 C5TVQ1 9819877 IC50 = 230 nM T23673 C1F0PU 9819906 IC50 = 3100 nM T23673 CY52NF 9819987 IC50 = 1200 nM T23673 C8Y9EF 9820630 IC50 = 2000 nM T23673 C1E2DV 9826083 IC50 > 10000 nM T23673 CSQ85J 9827373 IC50 = 700 nM T23673 CP1KY2 9827920 IC50 = 100 nM T23673 C36KUT 9842995 IC50 = 6000 nM T23673 C8UY4X 9844334 IC50 = 6600 nM T23673 C65RQN 9849174 IC50 = 6 nM T23673 C41QWA 9857146 IC50 = 5800 nM T23673 C1W4JG 9872939 IC50 = 400 nM T23673 C45ENX 9883939 IC50 = 3000 nM T23673 CVW95E 9884589 IC50 = 4900 nM T23673 C9KO2G 9884742 IC50 = 7600 nM T23673 CSZ72R 9884877 IC50 = 3700 nM T23673 C18HKQ 9885748 IC50 = 24000 nM T23673 CJ4QV2 9885993 IC50 = 470 nM T23673 CXTE43 9905562 IC50 = 3000 nM T23673 CG47NJ 9906915 IC50 = 6000 nM T23673 C5GE7T 9917045 IC50 = 880 nM T23673 C24UQF 9927821 IC50 = 11000 nM T23673 C5NE6S 9928371 IC50 = 8000 nM T23673 CJT0A3 9929998 IC50 = 7700 nM T23673 C3V6WA 9930407 IC50 = 500 nM T23673 CQ64LI 9935852 IC50 = 695 nM T23673 C61KBJ 9943464 IC50 = 7200 nM T23673 C5ZVD1 9949990 IC50 = 5000 nM T23673 C60EDC 9950128 IC50 = 1700 nM T23673 CW2N9R 9950282 IC50 = 590 nM T23673 CI4BL2 9950385 IC50 = 120 nM T23673 C30RGW 9950906 IC50 = 11000 nM T23673 C3MSR9 9950907 IC50 = 8100 nM T23673 C48ITV 9951822 IC50 = 1900 nM T23673 C2W3AV 9995236 IC50 > 100000 nM T23673 C26QHZ 10005638 IC50 > 10000 nM T23673 CBL7Y0 10127660 IC50 = 53 nM T23673 C0SB5R 10128380 IC50 = 88 nM T23673 CO2E8Y 10128955 IC50 = 73 nM T23673 C30ULG 10128960 IC50 = 410 nM T23673 CABY28 10129238 IC50 = 160 nM T23673 C4V8FQ 10151557 IC50 = 13 nM T23673 C9ZN8M 10151709 IC50 = 61 nM T23673 CS89XI 10152022 IC50 = 300 nM T23673 CLY75M 10173949 IC50 = 130 nM T23673 C6MYH8 10175138 IC50 = 160 nM T23673 C50CXW 10195382 IC50 = 50 nM T23673 C25XBS 10195523 IC50 = 330 nM T23673 C52OSM 10195599 IC50 = 26 nM T23673 C6T3MD 10196590 IC50 = 70 nM T23673 C5E7HJ 10217017 IC50 = 1 nM T23673 C1E6OC 10217682 IC50 = 2300 nM T23673 CE31PD 10218746 IC50 = 210 nM T23673 CLV62C 10238782 IC50 = 460 nM T23673 C2TO8Y 10239830 IC50 = 82 nM T23673 C5WCZ2 10269141 IC50 = 20000 nM T23673 CKF79I 10289214 IC50 = 110 nM T23673 CY6UR3 10289414 IC50 = 100 nM T23673 C26OJV 10289677 IC50 = 150 nM T23673 C3I0MT 10289813 IC50 = 230 nM T23673 CMF93A 10293379 IC50 = 12000 nM T23673 C59HOA 10310634 IC50 = 130 nM T23673 CIO14B 10311595 IC50 = 27 nM T23673 CSAJ01 10311596 IC50 = 170 nM T23673 CZKA14 10311642 IC50 = 44 nM T23673 CSR83F 10311959 IC50 = 63 nM T23673 C17NJQ 10312001 IC50 = 140 nM T23673 CRIA28 10312314 IC50 = 60 nM T23673 CIS0N3 10323382 IC50 = 3500 nM T23673 CA8B5T 10390073 IC50 = 2100 nM T23673 CD47LT 10522840 IC50 = 2600 nM T23673 CN2TU0 10526792 IC50 = 1000 nM T23673 C9Q5ON 10546780 IC50 = 1400 nM T23673 CXN40D 10565927 IC50 = 380 nM T23673 CGSD37 10567785 IC50 = 135 nM T23673 C8E3NI 10568528 IC50 = 90 nM T23673 CFP95Y 10591281 IC50 = 750 nM T23673 CW1L8E 10591928 IC50 = 110 nM T23673 C2JVA6 10595034 IC50 = 20 nM T23673 CJ2O7T 10601190 IC50 = 4500 nM T23673 C16KBG 10637813 IC50 = 5000 nM T23673 C0QC5K 10638921 IC50 = 23 nM T23673 C46ERK 10639924 IC50 = 210 nM T23673 CLSA43 10663963 IC50 = 2100 nM T23673 CTA89W 10664281 IC50 = 610 nM T23673 CK4EW1 10664282 IC50 = 56 nM T23673 CD94OB 10665884 IC50 = 320 nM T23673 CWM72U 10666557 IC50 = 1600 nM T23673 C2UFM7 10711296 IC50 = 950 nM T23673 C1FZ3L 10757716 IC50 = 3000 nM T23673 C29ITE 10829679 IC50 = 86 nM T23673 CKZ95C 10829684 IC50 = 80 nM T23673 C81JVA 10833164 IC50 = 2500 nM T23673 CP6K0I 11155829 IC50 = 210 nM T23673 CSK2W9 11166166 IC50 = 580 nM T23673 CXC91Z 11167118 IC50 = 76 nM T23673 CT1K6D 11167921 IC50 = 180 nM T23673 CZKL03 11190042 IC50 = 120 nM T23673 CGS76Q 11224163 IC50 = 200 nM T23673 C2W5RC 11235063 IC50 > 30000 nM T23673 C6QLP2 11235672 IC50 = 110 nM T23673 C8YQ6T 11235899 IC50 = 170 nM T23673 CH73GV 11258258 IC50 = 480 nM T23673 C2XQC6 11259227 IC50 = 280 nM T23673 CJ69GI 11283035 IC50 = 80 nM T23673 CC1K4L 11294093 IC50 = 490 nM T23673 CQ8CM9 11305234 IC50 = 140 nM T23673 C72GHB 11318236 IC50 = 230 nM T23673 CNFT61 11364677 IC50 = 340 nM T23673 CD57AN 11373388 IC50 = 190 nM T23673 CV24KW 11407374 IC50 = 360 nM T23673 C8W5UG 11407870 IC50 = 250 nM T23673 CFHN02 11407902 IC50 = 340 nM T23673 COT0F6 11418292 IC50 = 480 nM T23673 CP0WH6 11419121 IC50 = 240 nM T23673 C0APW4 11422034 IC50 = 1200 nM T23673 CM3ZU2 11429946 IC50 = 320 nM T23673 CIQ9K8 11430708 IC50 = 550 nM T23673 CD2R4S 11430860 IC50 = 160 nM T23673 C8DA5W 11454055 IC50 = 250 nM T23673 CX7ZP1 11454895 IC50 = 450 nM T23673 CEKC20 11477628 IC50 = 230 nM T23673 CVT10K 11487778 IC50 = 810 nM T23673 CB6ME8 11503895 IC50 = 9 nM T23673 CRP2U5 11526671 Ki > 50000 nM T23673 CO9KP5 11583459 IC50 > 10000 nM T23673 C4U7HM 11621097 IC50 = 116 nM T23673 CU0E8O 11690457 Ki > 10000 nM T23673 C8JW5Z 11696578 IC50 = 38150 nM T23673 CB0AP2 11705863 Ki > 10000 nM T23673 CGI1D9 11717001 Ki = 0.54 nM T23673 CZY05V 11719421 IC50 = 68 nM T23673 C63CKJ 11750387 IC50 = 370 nM T23673 CH3JL9 11750681 IC50 = 190 nM T23673 CO09LN 11750815 IC50 = 260 nM T23673 C8L9ZM 11751978 IC50 = 200 nM T23673 CT8P5W 11775428 IC50 = 660 nM T23673 CIY7C5 12972078 IC50 = 18 nM T23673 C89WYZ 16038368 IC50 > 10000 nM T23673 CZK8V6 16043304 IC50 > 10000 nM T23673 C9TU1O 16046126 IC50 > 1000 nM T23673 C2FR4D 16049771 IC50 = 4 nM T23673 CKV4G1 16079040 IC50 = 1600 nM T23673 C2IF3P 16678352 IC50 = 180 nM T23673 C3IO1C 16679060 IC50 = 1700 nM T23673 C0H8UN 16730109 IC50 > 30000 nM T23673 C8G9AL 16756850 IC50 > 10000 nM T23673 C8M6LZ 17755310 IC50 = 19 nM T23673 CE14ZT 17941505 IC50 = 800 nM T23673 CAF63H 18322354 IC50 = 13000 nM T23673 C14YFA 21024387 IC50 = 170 nM T23673 C4AK5J 21037180 IC50 = 4 nM T23673 C9YR7W 21037208 IC50 = 18 nM T23673 C8ID6R 21037243 IC50 = 41 nM T23673 C2V1EQ 21037245 IC50 = 2 nM T23673 C9MTS8 21037247 IC50 = 9 nM T23673 C1TBC5 21037266 IC50 = 4 nM T23673 CZ23BW 21037364 IC50 = 9 nM T23673 C1CA7H 22040368 IC50 = 53 nM T23673 CG67FQ 22040397 IC50 = 12 nM T23673 CJ4E1M 22040403 IC50 = 780 nM T23673 CSJ67N 22040407 IC50 = 1 nM T23673 C8VJ3A 22040410 IC50 = 210 nM T23673 CHFO54 22040436 IC50 = 1 nM T23673 C19FQT 22040598 IC50 = 1 nM T23673 CJ3UH0 22040625 IC50 = 4 nM T23673 C02DQZ 22040627 IC50 = 20 nM T23673 CCA1D7 22040647 IC50 = 19 nM T23673 C4RP8N 22040656 IC50 = 15 nM T23673 CFK41E 22040722 IC50 = 120 nM T23673 C9A4LW 22040760 IC50 = 14 nM T23673 CSKZ32 22040783 IC50 = 150 nM T23673 CLX26F 22040796 IC50 = 110 nM T23673 CI3V6C 22040802 IC50 = 48 nM T23673 C9WU0J 22040805 IC50 = 490 nM T23673 CDN61H 22040847 IC50 = 10 nM T23673 C3SX8H 22040857 IC50 = 950 nM T23673 CJCL02 22040865 IC50 = 4 nM T23673 C6NM3T 22040925 IC50 = 28 nM T23673 CC84UT 22040937 IC50 = 150 nM T23673 CZM5W1 22040941 IC50 = 6 nM T23673 C30PJQ 22040960 IC50 = 7 nM T23673 CNI32B 22040966 IC50 = 2 nM T23673 C6FMB5 22040978 IC50 = 45 nM T23673 C9A1HQ 22041020 IC50 = 200 nM T23673 CKT6M2 22041042 IC50 = 7300 nM T23673 CM50PH 22041067 IC50 = 27 nM T23673 CRJ4H3 22041111 IC50 = 3500 nM T23673 CO37NP 22041112 IC50 = 1100 nM T23673 C4UMZ2 22041119 IC50 = 56 nM T23673 CI5KM3 22041171 IC50 = 9 nM T23673 C51FDU 22041175 IC50 = 8 nM T23673 CR3G0K 22041260 IC50 = 3 nM T23673 C69BSO 22041261 IC50 = 15 nM T23673 CU85MA 22041278 IC50 = 2 nM T23673 CGX61W 22041319 IC50 = 4 nM T23673 C7HUS0 23585267 IC50 = 28 nM T23673 CHQ23N 23585318 IC50 = 16 nM T23673 COSI68 23585320 IC50 = 11 nM T23673 CV9U8E 24745781 IC50 > 10000 nM T23673 C6JCE7 24753323 IC50 = 26 nM T23673 C50GZI 24753409 IC50 = 13 nM T23673 CC4RZ6 24753410 IC50 = 530 nM T23673 CB3D1Y 24753411 IC50 = 180 nM T23673 C6JF2R 24753412 IC50 = 5 nM T23673 CWX89I 24753603 IC50 = 220 nM T23673 C4CY3V 24753607 IC50 = 300 nM T23673 CQJ2D3 24753784 IC50 = 8 nM T23673 CP1E4R 24753786 IC50 = 32 nM T23673 CA3I4T 24753787 IC50 = 8 nM T23673 CW36DL 24753877 IC50 = 120 nM T23673 COAY09 24753878 IC50 = 23 nM T23673 C9H7EZ 24753971 IC50 = 1500 nM T23673 C6CT7I 24753973 IC50 = 63 nM T23673 CS98MR 24754053 IC50 = 6 nM T23673 C9Q3DE 24754054 IC50 = 4 nM T23673 CRJ9G6 24754132 IC50 = 4 nM T23673 CBD59Z 24754133 IC50 = 45 nM T23673 CKV76A 24754134 IC50 = 37 nM T23673 CM8HY9 24754207 IC50 = 3600 nM T23673 C7YG1N 24759534 IC50 = 630 nM T23673 CCS1U0 24862785 IC50 = 6 nM T23673 C6R4ZU 24863189 IC50 = 1520 nM T23673 CUIS63 24878671 IC50 = 6960 nM T23673 CBUG02 24879141 IC50 > 100000 nM T23673 C2F6KO 24879328 IC50 = 20260 nM T23673 C43HWQ 24883287 IC50 = 10000 nM T23673 C8DA5Q 24883334 IC50 = 10000 nM T23673 C13QYB 24884503 IC50 = 25 nM T23673 C5E1YD 24891645 IC50 = 5840 nM T23673 CY8L7E 24896769 IC50 > 10000 nM T23673 CJZE02 24963588 IC50 = 27 nM T23673 C3DI7Y 24995523 IC50 = 100 nM T23673 CS3Q8B 24995659 IC50 > 2000 nM T23673 CUJZ08 25059320 IC50 = 3200 nM T23673 C2ICS7 25065806 IC50 = 21 nM T23673 CA61PS 25066845 IC50 = 14 nM T23673 CR46MG 25066846 IC50 = 1 nM T23673 CF5AO8 25093353 IC50 > 10000 nM T23673 CAB5K2 25114576 IC50 = 870 nM T23673 C9PL5S 25137959 IC50 = 2000 nM T23673 CVJ0S5 25137960 IC50 = 10 nM T23673 C6FGQ1 25206346 IC50 = 23 nM T23673 CC71QJ 27666048 IC50 > 100000 nM T23673 CIJ56L 44142782 IC50 > 10000 nM T23673 CCFQ29 44187005 IC50 = 8.52 nM T23673 CR7K2T 44223999 Ki = 0.3 nM T23673 CJ75IB 44250343 IC50 = 120 nM T23673 CS2CK9 44250550 IC50 = 105 nM T23673 CLY1A3 44251218 IC50 = 200 nM T23673 C4O0CH 44272164 IC50 = 18000 nM T23673 CX28HG 44272165 IC50 = 18000 nM T23673 CNIJ29 44309757 IC50 > 10000 nM T23673 CH1TA5 44309758 IC50 = 570 nM T23673 C4P9ZA 44312235 IC50 = 29 nM T23673 CX57BA 44312236 IC50 = 40 nM T23673 C2D7RK 44312254 IC50 = 32 nM T23673 C8MF2U 44312272 IC50 = 65 nM T23673 C4XCW8 44312367 IC50 = 25 nM T23673 CGRP10 44312380 IC50 = 16 nM T23673 C2IC8R 44326529 IC50 = 15000 nM T23673 CT74PB 44326530 IC50 = 12000 nM T23673 C1W6BM 44326737 IC50 = 25000 nM T23673 CO0UF5 44326798 IC50 = 19000 nM T23673 C0E4TU 44326810 IC50 = 16000 nM T23673 C0GRN1 44326814 IC50 = 15000 nM T23673 CV37KZ 44326926 IC50 = 22000 nM T23673 C4ZD0E 44326936 IC50 = 20000 nM T23673 C0KD4U 44346053 IC50 = 8700 nM T23673 CO0FN8 44378490 IC50 = 130 nM T23673 CR1MV0 44378504 IC50 = 68 nM T23673 C4D5ZM 44378534 IC50 = 120 nM T23673 CI3W6L 44378535 IC50 = 38 nM T23673 C39PLZ 44378637 IC50 = 500 nM T23673 C9E7ID 44378798 IC50 = 270 nM T23673 C7HGZ5 44378800 IC50 = 460 nM T23673 CBGZ52 44378801 IC50 = 140 nM T23673 CIV90F 44378900 IC50 = 130 nM T23673 CI6T9Z 44378901 IC50 = 5800 nM T23673 C6CW1H 44378902 IC50 = 370 nM T23673 CJH86A 44385063 IC50 > 50000 nM T23673 CG46BQ 44386338 IC50 > 10000 nM T23673 CJTF35 44418481 IC50 = 100 nM T23673 CKV61A 44418488 IC50 = 630 nM T23673 CJ49OD 44418525 IC50 = 1000 nM T23673 C8LB9S 44418539 IC50 = 250 nM T23673 CO8X1V 44418540 IC50 = 158 nM T23673 C1IX6V 44418547 IC50 = 251 nM T23673 C4Q5UL 44418563 IC50 = 40 nM T23673 C8NZ9D 44418572 IC50 = 10 nM T23673 CJ3DL4 44418573 IC50 = 7 nM T23673 C10MKH 44448311 IC50 = 49 nM T23673 C1QN4V 44448333 IC50 = 41 nM T23673 CLQF97 44448334 IC50 = 26 nM T23673 C73THQ 44448354 IC50 = 5 nM T23673 C0DPU3 44448725 IC50 = 2 nM T23673 CFQN07 44448726 IC50 = 17 nM T23673 CR85LO 44448746 IC50 = 20 nM T23673 C5Y2JR 44448747 IC50 = 1 nM T23673 CA76JX 44448748 IC50 = 0.5 nM T23673 C9I0DU 44453753 IC50 = 6300 nM T23673 C2T7UV 44454440 IC50 = 8600 nM T23673 C0TN9Z 44454441 IC50 = 6300 nM T23673 C3P2TG 44454464 IC50 = 3500 nM T23673 CDN4M7 44565710 IC50 = 44 nM T23673 CB39SW 44565730 IC50 = 160 nM T23673 C13WTF 44565731 IC50 = 230 nM T23673 CEU40V 44565732 IC50 = 440 nM T23673 C6HEU1 44565743 IC50 = 2700 nM T23673 C5VL3A 44565744 IC50 = 4400 nM T23673 CI5M9V 44565745 IC50 = 500 nM T23673 CCD0E2 44565749 IC50 = 700 nM T23673 C4P7KM 44565750 IC50 = 820 nM T23673 CBZ1H2 44565751 IC50 = 1000 nM T23673 C39TYG 44565752 IC50 = 1100 nM T23673 C8QDY6 44565771 IC50 = 7500 nM T23673 CQAB41 44565772 IC50 = 10000 nM T23673 CUK3E8 44565773 IC50 = 650 nM T23673 CK24HZ 44565794 IC50 = 9500 nM T23673 CG0PL1 44565795 IC50 = 1400 nM T23673 C53FHZ 44565817 IC50 = 1500 nM T23673 C9VXN3 44578709 IC50 = 80 nM T23673 C3Y5AW 44589519 IC50 = 41 nM T23673 C09EWJ 44590206 IC50 = 17 nM T23673 CUA97D 46209401 IC50 = 1.4 nM T23673 C2P9QO 46228508 IC50 = 198 nM T23673 C6E5PY 46228822 IC50 = 126 nM T23673 C3T8AM 46228951 IC50 = 3 nM T23673 C4MKC5 46870033 IC50 = 11 nM T23673 C7LK1C 46945257 IC50 = 765 nM T23673 CHSF07 49806372 IC50 > 1000 nM T23673 C5ME3S 49806721 IC50 > 50000 nM T23673 CS7J8G 50937465 IC50 = 79 nM T23673 C2Q0GE 50990922 IC50 = 3000 nM T23673 C61DVY 50990961 IC50 = 2.2 nM T23673 CV3UP9 50992247 IC50 = 2.5 nM T23673 COVJ29 50994971 IC50 = 169 nM T23673 C5X9OM 51354603 IC50 = 10 nM T23673 C4DSG2 51354885 IC50 = 6.2 nM T23673 CQ85FC 51354886 IC50 = 110 nM T23673 C7MOQ0 51354887 IC50 = 70 nM T23673 C5KVT1 51355181 IC50 = 4.5 nM T23673 CS5F4Z 51355182 IC50 = 780 nM T23673 C4NFL7 51355183 IC50 = 3.3 nM T23673 C4W6PY 51355459 IC50 = 4.6 nM T23673 C95FWU 51355461 IC50 = 45 nM T23673 C4J3RE 51355733 IC50 = 6 nM T23673 CEQN27 52936621 Ki > 2000 nM T23673 CM24LF 52938983 IC50 = 2.87 nM T23673 CFR21J 52939107 IC50 = 22.41 nM T23673 CJQ31I 53239946 IC50 = 11 nM T23673 C7B3DE 53239955 IC50 = 13 nM T23673 C8UZE6 53239978 IC50 = 46 nM T23673 C1SKV3 53249125 IC50 = 1 nM T23673 C4CO1V 53317057 IC50 = 240.3 nM T23673 CE73CS 53323686 IC50 = 8319 nM T23673 CFP84X 53324920 IC50 = 1100 nM T23673 CD4H3S 53354074 Ki > 1000 nM T23673 CM7P3W 53357328 IC50 > 50000 nM T23673 CVG90B 53389651 IC50 > 10000 nM T23673 C89YCL 54580728 IC50 = 3 nM T23673 CA9I0J 54580729 IC50 = 4 nM T23673 C4X6DP 54581730 IC50 = 3 nM T23673 C2KHN1 54581731 IC50 = 1 nM T23673 CQ3U7M 54582720 IC50 = 140 nM T23673 C6ZR1A 54583026 IC50 = 530 nM T23673 CP7U4T 54584640 IC50 = 1 nM T23673 CC7T2A 56674921 IC50 = 170 nM T23673 CT4E8R 56832546 IC50 = 8500 nM T23673 CP58NG 56954518 IC50 = 930 nM T23673 CAK91L 56955954 IC50 = 206 nM T23673 C8LZ5B 56966054 IC50 = 10.6 nM T23673 CCE7J3 56966055 IC50 = 75.9 nM T23673 CP10UK 56966056 IC50 = 87.8 nM T23673 CMS50K 56966057 IC50 = 13.1 nM T23673 CRPT61 56966123 IC50 = 69.2 nM T23673 C6X0EZ 56966125 IC50 = 94.9 nM T23673 CLI12D 56966126 IC50 = 120.3 nM T23673 C9L4IJ 56966199 IC50 = 147.9 nM T23673 CTP30L 56966200 IC50 = 77.7 nM T23673 COA5X2 56966201 IC50 = 35.9 nM T23673 CIBO79 56966202 IC50 = 22.1 nM T23673 C2KDZ7 56966273 IC50 = 16.5 nM T23673 CGJ6F0 56966274 IC50 = 64.8 nM T23673 C48QKV 56966276 IC50 = 46.7 nM T23673 C4G7QD 57343225 IC50 = 73 nM T23673 CU4FW8 57397383 IC50 = 1600 nM T23673 C0BGR6 57399335 IC50 = 3 nM T23673 CZSM95 57412684 IC50 > 10000 nM T23673 CVK0G4 58056356 IC50 > 50000 nM T23673 CKB3A4 58102283 IC50 > 10000 nM T23673 CX1G3L 58102286 IC50 = 100 nM T23673 C1R8NM 59139106 IC50 = 78 nM T23673 CB34LP 59139113 IC50 = 120 nM T23673 CWK9I8 59139139 IC50 = 2500 nM T23673 CWN47R 59139154 IC50 = 70 nM T23673 CT0JG1 59139161 IC50 = 16 nM T23673 CP5GY6 59139172 IC50 = 81 nM T23673 CL4X3Z 59139185 IC50 = 70 nM T23673 C1PE3R 59139202 IC50 = 2400 nM T23673 CE82OV 59139228 IC50 = 1100 nM T23673 C3T5OF 59139235 IC50 = 56 nM T23673 CWO17Q 59139262 IC50 = 5 nM T23673 C5IYT0 59139264 IC50 = 25 nM T23673 C91SBH 59139388 IC50 = 830 nM T23673 C62EVK 59139472 IC50 > 50000 nM T23673 CT3EW2 59292007 IC50 > 1000 nM T23673 CXJ63M 59603829 IC50 = 560 nM T23673 CQEU96 59603842 IC50 = 48 nM T23673 C1MR8Q 60097495 IC50 > 10000 nM T23673 C9W0PE 60150671 IC50 = 75 nM T23673 C9NAL6 60152613 IC50 = 0.6 nM T23673 CSZA16 60155724 IC50 = 1814 nM T23673 CW3G6N 60196633 IC50 = 340 nM T23673 CUV14K 60196634 IC50 = 4300 nM T23673 CU32ED 60196737 IC50 = 175 nM T23673 CKB59I 60196738 IC50 > 10000 nM T23673 C40LVZ 60196740 IC50 > 10000 nM T23673 CV63UL 67240318 IC50 > 10000 nM T23673 CW17YX 68281294 IC50 = 1000 nM T23673 C5DGR9 69036886 IC50 = 4012 nM T23673 C4BT3M 69037249 IC50 = 2.9 nM T23673 CVBR46 70696651 IC50 = 81.5 nM T23673 CRX81Q 71575642 IC50 = 72 nM T23673 CT93OP 71682347 IC50 > 10000 nM T23673 C3NV9Q 71682348 IC50 > 10000 nM T23673 CN7M9G 71682349 IC50 = 293 nM T23673 C8KU4O 71682499 IC50 > 10000 nM T23673 C0XEQ1 71682500 IC50 = 30 nM T23673 CXSI14 71718330 IC50 > 100000 nM T23673 C1TM3P 71720141 IC50 > 100000 nM T23673 CU83YL 71730951 IC50 = 2.8 nM T23673 C7F3ZM 71736390 IC50 = 1.6 nM T23673 C9EM5X 71736552 IC50 = 6.7 nM T23673 CKYO24 71736864 IC50 = 5.6 nM T23673 CSVW76 72546488 IC50 = 570 nM T23673 C7HBR1 72546491 IC50 = 40 nM T23673 CXYT34 72546730 IC50 = 56 nM T23673 C1DAW5 72546731 IC50 = 50 nM T23673 C6R8DI 72943374 IC50 = 80 nM T23673 C80SEC 73504974 IC50 = 652 nM T23673 C3KVB2 73505180 IC50 = 92 nM T23673 CP4ZX2 76317169 IC50 = 120 nM T23673 C4DT2Z 76335375 IC50 = 55 nM T23673 CA5O6K 78325057 IC50 = 0.1 nM T23673 CCD78B 86295666 IC50 = 0.2 nM T23673 C2OGP3 86296699 IC50 = 0.2 nM T23673 C80LAH 86298305 EC50 = 200 nM T23673 CI2CG1 89670173 IC50 = 7 nM T23673 C1HW4B 89735655 IC50 = 950 nM T23673 C7TJR3 89814000 IC50 = 1.2 nM T23673 C4WP7D 89827799 IC50 = 7.2 nM T23673 CJE4A5 90407961 IC50 = 0.6 nM T23673 C9KN1H 90408121 EC50 = 52 nM T23673 CF45CE 90408582 IC50 = 0.4 nM T23673 C6RZ7J 90408826 EC50 = 20 nM T23673 CXZ6M2 90408889 EC50 = 76 nM T23673 C7QD9P 90409579 EC50 = 80 nM T23673 CU0GW5 90442604 IC50 = 0.8 nM T23673 CA2E5S 90456597 EC50 = 8 nM T23673 CW6S8P 90655795 IC50 > 50000 nM T23673 CNYK35 90655796 IC50 = 27000 nM T23673 CE4LR9 90655797 IC50 = 21 nM T23673 CWD4O3 90655989 IC50 > 50000 nM T23673 C26BSU 90666124 IC50 = 3200 nM T23673 CVQ1O6 90666126 IC50 = 286 nM T23673 C5AN9J 90666128 IC50 = 4300 nM T23673 CP76NE 90666130 IC50 > 50000 nM T23673 C85GHD 90666131 IC50 = 16500 nM T23673 CRP9I5 90666132 IC50 = 9200 nM T23673 CX1NV3 117609603 EC50 = 3960 nM T23673 CQ40CN 117609669 EC50 = 5 nM T23673 C5XEY9 117610044 EC50 = 64 nM T23673 C8E9JO 117610115 EC50 = 27 nM T23673 CG7QL4 118705925 IC50 = 8.79 nM T23673 C4AHL2 118711367 IC50 > 10000 nM T23673 CQCX41 118737057 IC50 = 27 nM T23673 C9KWP7 118870913 IC50 = 0.4 nM T23673 CSR81B 118887129 EC50 = 21 nM T23673 CV3MY8 118938835 IC50 = 0.1 nM T23673 CU52FB 118938855 IC50 = 0.1 nM T23673 C9NDH0 118938856 IC50 = 2 nM T23673 CTLH73 118938861 IC50 = 0.03 nM T23673 CL4MP3 118938866 IC50 = 6 nM T23673 C0UT7G 122177477 IC50 = 3.1 nM T23673 CSF49R 122177478 IC50 = 5.2 nM T23673 C5B6QT 122189918 IC50 = 44.8 nM T23673 C4X7SD 122192466 IC50 > 10000 nM T23673 CNX0Q2 122193763 IC50 > 10000 nM T23673 CWV0C3 122193764 IC50 = 4020 nM T23673 CSG98Y 122193765 IC50 > 10000 nM T23673 CCLQ75 122193769 IC50 = 6220 nM T23673 CXDR48 122193770 IC50 > 10000 nM T23673 CPA8C5 122193773 IC50 = 5840 nM T23673 CWM37L 123897305 IC50 = 71 nM T23673 CF5WH1 127039888 IC50 = 38600 nM T23673 CAG9K7 127046489 IC50 = 15 nM T23673 C6DP7Y 127047275 IC50 = 111 nM T23673 C3DVM9 127047276 IC50 = 566 nM T23673 CM81AR 127047922 IC50 = 695 nM T23673 CA2C3D 129010136 EC50 = 200 nM T23673 C0FM1R 130196825 IC50 = 27920 nM T23673 CR5P1D 132067922 IC50 = 0.6 nM T23673 CU1H0W 132497402 IC50 = 43.4 nM T23673 CZ81AL 134142029 IC50 = 0.024 nM T23673 C7PS8C 135271570 IC50 = 76 nM T23673 C8B5GZ 135513879 IC50 = 390 nM T23673 CGL3F1 135957036 IC50 = 50 nM T23673 C4REH9 135957052 IC50 = 76 nM T23673 C58FQY 135957053 IC50 = 156 nM T23673 CG9PJ7 135993841 IC50 = 960.9 nM T23673 CUA72Z 136042194 IC50 = 667.8 nM T23673 CL2D1A 136086817 IC50 = 146 nM T23673 CKG0N2 136086821 IC50 = 370 nM T23673 CH70WS 136086832 IC50 = 839 nM T23673 CG1R7B 136087060 IC50 = 6500 nM T23673 CRB3M4 136609929 IC50 = 2500 nM T23673 C0A9VE 136609930 IC50 = 1300 nM T23673 CW5YL0 136609931 IC50 > 50000 nM T23673 C3FC1W 137631894 IC50 = 7500 nM T23673 C7NFX9 137632089 IC50 = 8.5 nM T23673 C0Y1AW 137632207 IC50 = 150 nM T23673 C10BTW 137632556 IC50 > 10000 nM T23673 C2J9GO 137633617 IC50 > 10000 nM T23673 C7MD0H 137635615 IC50 = 28 nM T23673 CML76T 137635976 IC50 = 6200 nM T23673 CS9AW4 137636754 IC50 = 272 nM T23673 C08MHJ 137636777 IC50 = 0.7 nM T23673 CV3A5G 137637973 IC50 = 34.5 nM T23673 C7R0MS 137638615 IC50 = 2300 nM T23673 CE96AL 137639657 IC50 = 17300 nM T23673 CEPU59 137640849 IC50 = 220 nM T23673 CGR5B1 137642299 IC50 = 51 nM T23673 CA13KP 137642491 IC50 = 18.7 nM T23673 C26HIT 137643417 IC50 = 2100 nM T23673 CAT49C 137645403 IC50 = 374 nM T23673 CUES49 137646218 IC50 = 1800 nM T23673 CS6J8X 137646633 IC50 > 10000 nM T23673 C9Z6NB 137646838 IC50 = 770 nM T23673 CL8W4P 137647062 IC50 = 21.4 nM T23673 CGQ02E 137648059 IC50 = 6.3 nM T23673 C2HFR6 137648529 IC50 = 690 nM T23673 CL9HT1 137648599 IC50 = 21.9 nM T23673 CYR2I7 137649411 IC50 = 3050 nM T23673 C17GBS 137649678 IC50 = 1840 nM T23673 CEO70C 137650358 IC50 > 10000 nM T23673 CE7KF3 137650390 IC50 = 13.3 nM T23673 C4NM0R 137650776 IC50 = 1280 nM T23673 C3LAD6 137652990 IC50 > 100000 nM T23673 CL3P8Q 137653011 IC50 = 89 nM T23673 C5B9AM 137653362 IC50 = 860 nM T23673 C8K0OY 137655533 IC50 = 670 nM T23673 C3F8ZD 137656536 EC50 = 700 nM T23673 CMPJ36 137656808 IC50 = 14.4 nM T23673 C83XOY 137657177 IC50 = 53 nM T23673 CF7U5Y 137657487 IC50 > 10000 nM T23673 C3SD7B 137658277 IC50 = 4900 nM T23673 CVY3F0 137658568 IC50 = 1510 nM T23673 CJK81S 137659431 IC50 = 99 nM T23673 CNWY53 137659664 IC50 = 370 nM T23673 CUS48N 137659983 IC50 = 327 nM T23673 CA4V9R 137661906 IC50 = 100 nM T23673 COB9P2 141456067 IC50 = 7900 nM T23673 C6CN8H 142739455 IC50 = 61 nM T23673 CT25FH 145950796 IC50 = 8.5 nM T23673 C2I5WD 145979310 IC50 = 13.3 nM T23673 C6T4MU 145982183 IC50 = 40 nM T23673 CI1VH9 145985185 IC50 > 200000 nM T23673 CI7M2B 145988861 IC50 = 17.5 nM T23673 CNLH48 145988888 IC50 = 17600 nM T23673 CRT48W 145993502 IC50 = 3150 nM T23673 C2NKF8 155076930 IC50 = 182 nM T23673 CY1ZH2 155510358 IC50 = 336 nM T23673 CZ5S2M 155512875 IC50 = 2.7 nM T23673 C2MD1Q 155513187 IC50 > 10000 nM T23673 C0MZ9A 155513534 IC50 = 5160 nM T23673 CI54TD 155514548 IC50 = 1420 nM T23673 C2BA1L 155514841 IC50 = 1310 nM T23673 CX6SR0 155516442 IC50 = 420 nM T23673 CS31UH 155519078 IC50 = 1520 nM T23673 CU6Z5O 155520650 IC50 = 130 nM T23673 CP4JL5 155521754 IC50 = 4490 nM T23673 CVQ35F 155522102 IC50 = 3540 nM T23673 CM3DB7 155523430 IC50 = 480 nM T23673 CLY07C 155530863 IC50 = 450 nM T23673 CVQ24P 155532080 IC50 = 990 nM T23673 CS69CA 155532132 IC50 = 0.5 nM T23673 CJP67I 155535248 IC50 = 5320 nM T23673 C8ZF4H 155544511 IC50 = 3660 nM T23673 C8T0MQ 155544690 IC50 = 840 nM T23673 CJL37G 155544854 IC50 = 16400 nM T23673 CHE5F1 155553390 IC50 = 6260 nM T23673 CYC23K 155560669 IC50 = 110 nM T23673 C81JZW 155563388 IC50 = 410 nM T23673 C62CIM 155565320 IC50 = 420 nM T23673 CH3NO1 155566774 IC50 = 31.7 nM T23673 C0V2MU 135398506 Ki = 1.72 nM T23673 D00NWF 5730 IC50 = 70 nM T23673 D02XHC 448912 IC50 > 100000 nM T23673 D03MUZ 17759555 IC50 > 100000 nM T23673 D05UPS 44418518 IC50 = 398 nM T23673 D06WJA 9950176 IC50 = 1.4 nM T23673 D08LYB 5166 IC50 > 50 nM T23673 D0C0ZC 11676786 IC50 = 380 nM T23673 D0IR6U 5494425 IC50 > 10000 nM T23673 D0J4YA 9943465 IC50 > 12000 nM T23673 D0QN6U 9806182 IC50 = 810 nM T23673 D0V0QJ 389898 IC50 = 34500 nM T23673 D0Z5TQ 5924208 IC50 = 10.6 nM T48598 D05ROI 44462760 IC50 = 5880 nM T48598 D0Y9EW 42611257 IC50 = 16600 nM T48598 D04AHQ 71721540 IC50 = 150 nM T48598 CE2VX1 1381961 IC50 = 155000 nM T48598 C4K3AC 9870962 EC50 = 1065 nM T48598 C3MSB4 9954645 EC50 > 10000 nM T48598 C4BT3M 69037249 IC50 = 91 nM T48598 C3D6WC 71515468 IC50 = 200 nM T48598 CU83YL 71730951 IC50 = 48 nM T48598 C7F3ZM 71736390 IC50 = 46 nM T48598 C9EM5X 71736552 IC50 = 270 nM T48598 CKYO24 71736864 IC50 = 120 nM T48598 C2A4YP 86279165 Ki = 200000 nM T48598 C7TJR3 89814000 IC50 = 16 nM T48598 C4WP7D 89827799 IC50 = 160 nM T48598 CHJ6B8 90665836 IC50 = 1200 nM T48598 CFI02E 90665837 IC50 = 10000 nM T48598 CI6DB8 90665838 IC50 = 1800 nM T48598 C61RVL 90665839 IC50 = 10000 nM T48598 CW2UX9 90665840 IC50 = 10000 nM T48598 CDN49I 90665841 IC50 = 700 nM T48598 C0KI6U 90665842 IC50 = 1100 nM T48598 C0W7UI 90665843 IC50 = 2000 nM T48598 CYU7W2 90665844 IC50 = 2300 nM T48598 CEJ3D4 118019010 IC50 = 496 nM T48598 C0UT7G 122177477 IC50 = 57 nM T48598 CSF49R 122177478 IC50 = 120 nM T48598 CYP1B7 132145599 IC50 > 16000 nM T48598 CG7J5E 132162814 IC50 = 7600 nM T48598 CDWB35 132162815 IC50 > 16000 nM T48598 C1DW2E 132162816 IC50 > 16000 nM T48598 CJ1MY3 132162817 IC50 > 16000 nM T48598 C74FYN 132162819 IC50 > 16000 nM T48598 C2SIJ4 132162853 IC50 = 1900 nM T48598 CB80ZS 132163177 IC50 = 1500 nM T48598 C6CL4S 132163178 IC50 = 540 nM T48598 C3GPQ1 132163222 IC50 = 70 nM T48598 CULE35 135148667 IC50 = 8 nM T48598 C6DYW3 135148885 IC50 = 220 nM T48598 CU8T3N 136346978 Ki = 9 nM T48598 CC20EZ 136346980 Ki = 280 nM T48598 CY2L6T 136346989 Ki = 5000 nM T48598 CUG30Y 136347012 Ki > 25000 nM T48598 CS8YP7 137003167 IC50 = 939 nM T48598 CGS71A 137278705 IC50 = 51 nM T48598 CJ9N2K 137278711 IC50 = 68 nM T48598 C1HX7O 137278713 IC50 = 63 nM T48598 CK4MJ2 137278717 IC50 = 25 nM T48598 CA7GT6 137283289 Ki = 382 nM T48598 CS4W8U 137288869 IC50 = 69 nM T48598 C34DAC 137288870 IC50 = 36 nM T48598 CB42LP 137289789 Ki = 374 nM T48598 C0GNH8 137290307 Ki = 50000 nM T48598 CN2U1R 137290313 Ki = 8000 nM T48598 CX30GO 137290327 Ki = 2200 nM T48598 CW7Y3V 137292511 Ki = 15200 nM T48598 CXM3Y9 137297869 IC50 = 3330 nM T48598 C2XJN7 137297879 IC50 = 903 nM T48598 CRZH30 137297882 IC50 = 101 nM T48598 CBG13S 137297890 IC50 = 1800 nM T48598 C7BL0Z 137297899 IC50 = 7150 nM T48598 C1TWR9 137297909 IC50 = 20100 nM T48598 C85PEX 137297911 IC50 = 28 nM T48598 CS9D7J 137297914 IC50 = 3520 nM T48598 CTU65M 137297915 IC50 = 51 nM T48598 CJY69R 137297923 IC50 = 9150 nM T48598 CTO29V 137303087 Ki > 10000 nM T48598 C9SZ6B 137303128 Ki = 920 nM T48598 CVH3G7 137304434 Ki = 36000 nM T48598 C2LV5C 137304502 Ki = 5000 nM T48598 CV9Q5S 137314428 Ki = 380 nM T48598 CG7F2B 137314429 Ki > 20000 nM T48598 C8KFZ5 137316419 Ki = 2700 nM T48598 CQ7Z4X 137316471 Ki = 1600 nM T48598 C2M5GX 137317563 Ki = 3500 nM T48598 CJ07SA 137636907 IC50 = 50 nM T48598 CFA74W 137637303 IC50 = 64 nM T48598 C17EOK 137637743 IC50 = 1190 nM T48598 C7JU3W 137639238 IC50 = 35.8 nM T48598 CS93CA 137639750 IC50 = 1.6 nM T48598 CUS40W 137643713 IC50 = 59 nM T48598 CN4FM5 137645102 IC50 = 6.1 nM T48598 CK7S3H 137646089 IC50 = 1630 nM T48598 CFT25U 137647500 IC50 = 2.7 nM T48598 CM2XF3 137648559 IC50 = 426 nM T48598 C0UKF3 137648822 IC50 = 764 nM T48598 CP4V6Y 137650846 IC50 = 15400 nM T48598 CRF93P 137650861 IC50 = 19 nM T48598 CXO6C3 137652506 IC50 = 20600 nM T48598 CBIZ98 137653897 IC50 = 243 nM T48598 CLWD10 137660005 IC50 = 83 nM T48598 C78JQW 137661919 IC50 = 11 nM T48598 CKWQ13 138678754 IC50 < 5 nM T48598 CWM42J 138678756 IC50 = 18 nM T48598 C8S1AT 138678759 IC50 = 16 nM T48598 CA18QI 138678764 IC50 = 70 nM T48598 C9J3EN 138678770 IC50 = 132 nM T48598 C6SPK8 138678774 IC50 = 387 nM T48598 C7EV3T 138678780 IC50 = 610 nM T48598 CE7Q0H 138678786 IC50 = 97 nM T48598 C92HTX 138678788 IC50 = 81 nM T48598 C27KFX 138678799 IC50 = 150 nM T48598 C30MEF 138678890 IC50 = 211 nM T48598 C2DOL1 138679046 IC50 = 52 nM T48598 CR5A6H 139388519 IC50 = 780 nM T48598 CYRW58 139388529 IC50 = 4860 nM T48598 C5GLR3 139388566 IC50 = 169 nM T48598 CG1MO4 139388571 IC50 = 116 nM T48598 CNVK52 139388599 IC50 = 129 nM T48598 CXB0Y3 139388605 IC50 = 214 nM T48598 C8CRF6 139600305 IC50 = 115 nM T48598 CEL25S 140956840 IC50 = 11 nM T48598 C0NV4K 140956861 IC50 = 66 nM T48598 C1SJI0 142468965 IC50 = 18 nM T48598 CB29ZR 142468976 IC50 = 12 nM T48598 C9PC5N 142468998 IC50 = 12 nM T48598 C6S0VF 142469011 IC50 = 21 nM T48598 C3PD0Y 142469055 IC50 = 32 nM T48598 C7X6QM 142469058 IC50 = 97 nM T48598 CUW9Y5 146234885 IC50 = 128 nM T48598 CN08TQ 146234893 IC50 = 25 nM T48598 CB30HO 146235053 IC50 = 80 nM T48598 C2B5VH 146235304 IC50 = 47 nM T48598 CKM1C3 146235420 IC50 = 90 nM T48598 C5QBX0 146235429 IC50 = 53 nM T48598 C91ANQ 146235452 IC50 = 142 nM T48598 CAVJ61 146235508 IC50 = 34 nM T48598 CFKC35 146235592 IC50 = 164 nM T48598 C3HCA7 146235786 IC50 = 65 nM T48598 C89YKH 146235843 IC50 = 38 nM T48598 C5KX3F 146235857 IC50 = 306 nM T48598 C42CDB 146235944 IC50 = 53 nM T48598 CQW98L 146236007 IC50 = 146 nM T48598 C76QJC 146236012 IC50 = 56 nM T48598 C06VPI 146254335 IC50 = 109 nM T48598 C0U1KX 146254417 IC50 = 442 nM T48598 CZ7P4M 146254588 IC50 = 25 nM T48598 C3S5WI 146461338 IC50 = 29 nM T48598 CBI9U1 146585881 IC50 = 109 nM T48598 C1EFX9 146585884 IC50 = 683 nM T48598 C3H9BP 146585895 IC50 = 139 nM T48598 C1VJ4L 146630440 IC50 = 17900 nM T48598 C6S1IB 146630461 IC50 = 2120 nM T48598 C9I2WV 146630653 IC50 > 250000 nM T48598 C4IA5T 146630666 IC50 = 299 nM T48598 C51IYS 146630676 IC50 = 638 nM T48598 CW34ZK 146630683 IC50 = 1370 nM T48598 CVL6A5 146630701 IC50 = 4260 nM T48598 C4QH7U 146630731 IC50 = 6630 nM T48598 C0WAB5 146630732 IC50 = 14200 nM T48598 CYH28N 146630894 IC50 = 369 nM T48598 C5IV8H 146630905 IC50 = 1290 nM T48598 CIX1C8 146630907 IC50 = 174 nM T48598 CNK71Q 146631214 IC50 = 1270 nM T48598 C8H9TW 155523678 IC50 = 73 nM T48598 CBR9O0 155524545 IC50 = 4342 nM T48598 CVQ3H7 155528727 IC50 = 7653 nM T48598 C7Y3FZ 155549278 IC50 = 627 nM T48598 CMA86J 155564813 IC50 = 2780 nM T58093 D0S7BQ 52918384 IC50 = 12 nM T58093 D0T2IQ 443600 IC50 = 20 nM T58093 C8A6FD 9849925 IC50 = 30 nM T58093 C04KRJ 16034963 IC50 = 2.5 nM T58093 CJ42NE 16034968 IC50 = 0.52 nM T58093 CEYX96 16035081 IC50 = 0.93 nM T58093 CH97SC 16035085 IC50 = 2.1 nM T58093 CTC5O9 16035087 IC50 = 1.4 nM T58093 C4OQ3K 16035189 IC50 = 1.4 nM T58093 CG83UV 16035293 IC50 = 3.8 nM T58093 CGN4W5 16035295 IC50 = 3.2 nM T58093 CSFC45 16035507 IC50 = 2.2 nM T58093 CNTW74 16035824 IC50 = 12 nM T58093 CCDG98 16035825 IC50 = 5.2 nM T58093 CZC1T5 16035827 IC50 = 8 nM T58093 C48ARB 16036037 IC50 = 4.5 nM T58093 C1SMZ2 16036156 IC50 = 2.2 nM T58093 CP3H6M 16036157 IC50 = 4.4 nM T58093 C9YZ6I 16036158 IC50 = 1.4 nM T58093 C2I1YX 16036160 IC50 = 1.5 nM T58093 C3ZIH1 16036281 IC50 = 2.4 nM T58093 C5SOI2 16036282 IC50 = 3.4 nM T58093 C7JG1B 16036394 IC50 = 10 nM T58093 C3NWE9 16036395 IC50 = 2 nM T58093 CW16UL 16036656 IC50 = 5 nM T58093 C2VOZ5 16036657 IC50 = 4 nM T58093 C3IU1P 16036659 IC50 = 2 nM T58093 C9SHM6 16036661 IC50 = 3.7 nM T58093 CMOB46 16046174 IC50 = 7500 nM T58093 C7WH3R 25123230 IC50 = 30 nM T58093 CV15JQ 25123888 IC50 = 30 nM T58093 CFD1Z5 57345646 IC50 = 35800 nM T58093 C4GTE0 57345647 IC50 = 100100 nM T58093 CO8R3H 57878092 IC50 = 5 nM T58093 C0HY5X 57878097 IC50 = 2.3 nM T58093 C3W6PE 57878101 IC50 = 10 nM T58093 C2GJ1F 57878102 IC50 = 1.7 nM T58093 CX9UE4 57878122 IC50 = 1.6 nM T58093 C2F9SP 57878124 IC50 = 1.4 nM T58093 CH48QS 57878125 IC50 = 1.2 nM T58093 C5UJ7H 57878129 IC50 = 0.9 nM T58093 CU2KR4 57878131 IC50 = 1.7 nM T58093 C0WIY3 57878141 IC50 = 0.86 nM T58093 C1R5WU 57878145 IC50 = 1 nM T58093 C3XHZ9 70681653 IC50 = 1.3 nM T58093 C0C5BI 70685926 IC50 = 3.3 nM T58093 CMH5K3 70692221 IC50 = 2.3 nM T58093 C5SH2R 70694300 IC50 = 5.9 nM T58093 C5W1AK 138454269 IC50 = 2 nM T58093 CZUO38 155511087 IC50 = 2 nM T58093 C9F6LQ 155511457 IC50 = 5 nM T58093 C5DKE6 155511474 IC50 = 16 nM T58093 C45DSK 155512893 IC50 = 6 nM T58093 C6BQA2 155514815 IC50 = 11 nM T58093 CD58RH 155518934 IC50 = 5 nM T58093 C3WQH0 155520436 IC50 = 2 nM T58093 C0P4AY 155523706 IC50 = 10 nM T58093 CX3FD5 155526303 IC50 = 1 nM T58093 CEU4S5 155526689 IC50 = 0.63 nM T58093 CV3SG0 155529612 IC50 = 1 nM T58093 CJL2C8 155535353 IC50 = 18 nM T58093 CF5T2J 155536889 IC50 = 158 nM T58093 C7D4BJ 155541590 IC50 = 2 nM T58093 CL5AO7 155553287 IC50 = 20 nM T58093 CQF91W 155554205 IC50 = 3 nM T58093 CB1SN4 155557831 IC50 = 2 nM T58093 C94TBM 155560644 IC50 = 2 nM T58093 C4AD6J 155563341 IC50 = 1 nM T20600 D0J3SU 9847835 EC50 > 5000 nM T20600 C3T8NF 5288850 IC50 > 5000 nM T20600 C1KR5B 5327301 Ki = 22000 nM T20600 C37TKL 5327302 Ki = 1000 nM T20600 C64ZMN 5327304 Ki = 1400 nM T20600 C3IZ2W 5327307 Ki = 2300 nM T20600 C16DTL 5327308 Ki = 540 nM T20600 C4O3QY 5327309 Ki = 9700 nM T20600 C3GUM7 5327310 Ki = 2400 nM T20600 C3LZX9 8027611 IC50 > 20000 nM T20600 CFN2P6 9800285 Ki = 7500 nM T20600 CLTO67 9821317 IC50 = 18 nM T20600 C4XO3K 9821545 IC50 > 5000 nM T20600 CJI5T3 9823027 IC50 = 37 nM T20600 C74QTI 9823074 IC50 = 940 nM T20600 C6S3KT 9840223 Ki > 25000 nM T20600 CD05OL 9867192 IC50 = 1500 nM T20600 C2DMG1 9914167 IC50 > 5000 nM T20600 C9CV0Y 10001828 IC50 = 940 nM T20600 CX67SZ 10826725 Ki = 1000 nM T20600 CDX7A4 10963183 Ki = 190 nM T20600 CM8O6L 11257152 IC50 = 50 nM T20600 C4F8DC 11444079 IC50 > 500000 nM T20600 CDT9G3 11467504 IC50 = 3.44 nM T20600 CV4CP9 11496333 IC50 > 5000 nM T20600 CGE2J0 11497112 IC50 > 5000 nM T20600 C6IS9K 11509289 IC50 > 5000 nM T20600 C6L2MY 11509300 IC50 > 5000 nM T20600 CC31QO 11509301 IC50 > 5000 nM T20600 CS8OX7 11510566 IC50 > 500000 nM T20600 C7FY9B 11512139 IC50 > 5000 nM T20600 C15VFG 11515586 IC50 > 500000 nM T20600 CW6PC0 11519268 IC50 > 5000 nM T20600 CZC5D9 11525874 IC50 > 5000 nM T20600 C5BNE1 11533326 IC50 > 5000 nM T20600 CDK3Z5 11533935 IC50 = 3700 nM T20600 C4IC7E 11541867 IC50 > 500000 nM T20600 C3USR9 11543714 IC50 = 283 nM T20600 C3P2GZ 11548424 IC50 > 500000 nM T20600 CVX4M6 11548909 EC50 > 5000 nM T20600 C17OJS 11572844 IC50 = 201 nM T20600 CF0V3P 11576540 IC50 > 5000 nM T20600 C1T9DY 11576622 IC50 > 5000 nM T20600 C03KPR 11576852 EC50 > 5000 nM T20600 CN67DR 11583840 IC50 > 5000 nM T20600 CPD0M8 11584106 IC50 > 5000 nM T20600 CL16IM 11591540 IC50 > 5000 nM T20600 CE2TX6 11591919 IC50 > 500000 nM T20600 CG4Z9A 11598106 IC50 > 10000 nM T20600 CV6MF1 11614728 IC50 > 500000 nM T20600 CFP19E 11619968 IC50 > 5000 nM T20600 CA0LH6 11624920 IC50 > 5000 nM T20600 CEY39D 11628992 IC50 > 500000 nM T20600 C6UAV3 11632008 IC50 = 216 nM T20600 C6Y5MG 11634372 IC50 > 5000 nM T20600 CKJE92 11634649 IC50 > 5000 nM T20600 C91JNO 11639020 IC50 = 124 nM T20600 C4MCW2 11646889 IC50 = 137 nM T20600 C2KFU3 11647018 IC50 > 5000 nM T20600 CH20JE 11652994 IC50 = 2850 nM T20600 CN32TX 11664423 IC50 > 500000 nM T20600 CUD05C 11670894 IC50 > 5000 nM T20600 CX97NT 11684618 IC50 > 5000 nM T20600 C05YRV 11699954 IC50 > 500000 nM T20600 CKEX64 11700402 IC50 > 500000 nM T20600 C89COT 11705942 IC50 > 5000 nM T20600 C86PAH 11712912 IC50 > 5000 nM T20600 CXH9M5 16749067 IC50 = 407 nM T20600 C2DJ5W 16749068 IC50 = 9550 nM T20600 COM07G 16749069 IC50 = 698 nM T20600 CPG8Q0 16749161 IC50 = 744 nM T20600 CG84TK 16749162 IC50 = 823 nM T20600 CT3HD1 16749163 IC50 = 650 nM T20600 CZM4X2 16749164 IC50 = 610 nM T20600 CUZ8N4 16749267 IC50 = 8900 nM T20600 CMEK96 16749268 IC50 = 5025 nM T20600 C01HBN 16749269 IC50 = 918 nM T20600 CWG3C8 16749270 IC50 = 840 nM T20600 C8R3GD 16749271 IC50 = 515 nM T20600 CTI80F 25178948 EC50 > 5000 nM T20600 C2GI4J 25178949 EC50 > 5000 nM T20600 CQ2GM9 25178950 EC50 > 5000 nM T20600 C4GFV6 25179140 EC50 > 5000 nM T20600 CYL36B 25179141 IC50 = 4425 nM T20600 CGC69Q 25179143 EC50 > 5000 nM T20600 C27YJF 25179144 IC50 = 9967 nM T20600 C2YTB7 25179145 EC50 > 5000 nM T20600 C6GTV3 25179324 EC50 > 5000 nM T20600 CIC46T 25179513 EC50 > 5000 nM T20600 CK96WB 25179514 EC50 > 5000 nM T20600 CGX78D 25217029 IC50 = 450 nM T20600 CW2L9Q 25217030 IC50 = 770 nM T20600 C8UTC4 25217031 IC50 = 509 nM T20600 CZ43KQ 25217032 IC50 = 927 nM T20600 C2P9NI 25217145 IC50 = 4930 nM T20600 C8C9XU 42618276 IC50 > 15000 nM T20600 CFO93N 42618277 IC50 = 12833 nM T20600 CS1KQ0 42618278 IC50 = 325 nM T20600 CVI16X 42618279 IC50 = 545 nM T20600 C3MRA0 42618280 IC50 = 568 nM T20600 C8UO9S 42618281 IC50 = 425 nM T20600 C68NPR 42618282 IC50 = 453 nM T20600 CL41SD 42618283 IC50 = 591.7 nM T20600 CJ7U2E 42618284 IC50 = 151 nM T20600 CZL8C7 42618285 IC50 = 188 nM T20600 CNIQ28 42618286 IC50 = 230 nM T20600 C91OMB 42618287 IC50 = 9833 nM T20600 C5AC1L 42618288 IC50 = 156 nM T20600 CFU5T2 42618289 IC50 = 197 nM T20600 CK9H3M 42618290 IC50 = 280 nM T20600 CV4H2J 42618291 IC50 = 241 nM T20600 C7VPU3 42618292 IC50 = 358 nM T20600 C6R2FM 42618293 IC50 = 468 nM T20600 CT7VO2 44157085 IC50 > 500000 nM T20600 CWMU91 44157086 IC50 > 500000 nM T20600 C6LZ5Y 44157087 IC50 > 500000 nM T20600 CYSJ79 44157089 IC50 > 500000 nM T20600 CMX7W1 44157090 IC50 > 500000 nM T20600 C7B3VE 44158086 IC50 > 500000 nM T20600 C20WEJ 44158089 IC50 > 500000 nM T20600 C68KOD 44158154 IC50 > 500000 nM T20600 C4C1RU 44158155 IC50 > 500000 nM T20600 CN1YR9 44158157 IC50 > 500000 nM T20600 C80XPD 44158237 IC50 > 500000 nM T20600 CN09UV 44158238 IC50 > 500000 nM T20600 CT9DF4 44158240 IC50 > 500000 nM T20600 CHDF62 44158242 IC50 > 500000 nM T20600 CS6X1C 44158325 IC50 > 500000 nM T20600 C17TEZ 44158326 IC50 > 500000 nM T20600 CZ0VT3 44158328 IC50 > 500000 nM T20600 CD8WB9 44304162 Ki = 57000 nM T20600 CAB39E 44331552 IC50 = 32400 nM T20600 CE0FW4 44331565 IC50 = 21400 nM T20600 C8SZN9 44331566 IC50 = 12000 nM T20600 CMFW61 44331567 IC50 = 22600 nM T20600 CHYL38 44331577 IC50 = 1620 nM T20600 C1I9QH 44331578 IC50 = 18900 nM T20600 C4VGZ1 44331579 IC50 = 10100 nM T20600 CRZ01H 44331580 IC50 = 20500 nM T20600 CFOR90 44331674 IC50 = 14500 nM T20600 CK7VI8 44331675 IC50 = 717 nM T20600 CH7GS4 44331676 IC50 > 50000 nM T20600 C4FOD3 44331693 IC50 > 50000 nM T20600 CJY5L2 44331739 IC50 = 28600 nM T20600 C8N2GQ 44331740 IC50 = 11800 nM T20600 CW9K4Q 44331815 IC50 = 3370 nM T20600 CT76DG 44331816 IC50 = 33400 nM T20600 CC70GF 44331830 IC50 = 2530 nM T20600 CNJ19L 44331876 IC50 = 11110 nM T20600 C46IPA 44331879 IC50 > 10000 nM T20600 CP0Y8M 44331898 IC50 = 10 nM T20600 CF3R6W 44331908 IC50 > 10000 nM T20600 CTM5W1 44331914 IC50 = 3.5 nM T20600 C0YZ9O 44331915 IC50 = 15 nM T20600 C4NK1S 44331942 IC50 = 10 nM T20600 CXKY19 44331943 IC50 = 18560 nM T20600 C3FC8D 44331944 IC50 > 10000 nM T20600 CH1ZF2 44331953 IC50 = 589 nM T20600 C0QJ8V 44331957 IC50 = 4600 nM T20600 C1HBX6 44331963 IC50 = 14030 nM T20600 C7UXK5 44331964 IC50 = 10000 nM T20600 C42PGN 44331965 IC50 = 308 nM T20600 C5J7KX 44331966 IC50 > 50000 nM T20600 CG83FS 44331967 IC50 = 12500 nM T20600 CGAJ95 44331977 IC50 = 3610 nM T20600 CCYX84 44331980 IC50 > 10000 nM T20600 C5UIO2 44331987 IC50 = 32500 nM T20600 C0PM5C 44332004 IC50 = 4180 nM T20600 C4ENB1 44332005 IC50 = 1010 nM T20600 CFK4Z1 44332024 IC50 = 1280 nM T20600 CTM3G2 44332026 IC50 = 2720 nM T20600 C48ZEW 44332028 IC50 > 50000 nM T20600 C30MKG 44332029 IC50 > 50000 nM T20600 C7OS9X 44332050 IC50 = 9750 nM T20600 C9Y6NP 44332051 IC50 = 5050 nM T20600 C0VGF8 44332058 IC50 = 5860 nM T20600 CQU84D 44332068 IC50 = 21200 nM T20600 CBL91D 44332078 IC50 = 51200 nM T20600 C4VCM3 44332093 IC50 = 5900 nM T20600 C92QVT 44332108 IC50 = 1430 nM T20600 CQLZ09 44332109 IC50 = 13800 nM T20600 C4CUL6 44332112 IC50 = 3030 nM T20600 CN2YM6 44332113 IC50 = 1900 nM T20600 C4CY8K 44332118 IC50 = 7000 nM T20600 CXZ2N1 44332120 IC50 = 42700 nM T20600 CD56PK 44332121 IC50 > 50000 nM T20600 C5A6OJ 44332128 IC50 = 14500 nM T20600 C6IZ2R 44332129 IC50 = 3160 nM T20600 C5DY0G 44332136 IC50 = 1430 nM T20600 CQ1K9H 44332311 IC50 = 37 nM T20600 C9LOS2 44332330 IC50 = 305 nM T20600 C2U6GB 44332331 IC50 = 10300 nM T20600 CH01QW 44332332 IC50 = 11800 nM T20600 C8D5TB 44364680 Ki = 120 nM T20600 CJ6QG4 44417479 IC50 > 500000 nM T20600 C7RX9I 44418960 Ki = 550000 nM T20600 CXR1V5 44434249 IC50 = 61 nM T20600 C8Z4WO 44459967 IC50 = 5128.61 nM T20600 C86ORE 44459987 IC50 = 3548.13 nM T20600 CDY2W5 49796910 IC50 = 1.7 nM T20600 C3M2BW 52918163 IC50 = 8700 nM T20600 CF24IM 52918177 IC50 = 6900 nM T20600 CR9I7F 52918178 IC50 = 13450 nM T20600 C2VPU1 52918179 IC50 = 7750 nM T20600 C8Z2TQ 54580470 IC50 > 10000 nM T20600 CMU0B4 54581481 IC50 > 10000 nM T20600 CCS8Y3 54581987 IC50 = 1165 nM T20600 CJEP38 54582484 IC50 = 7666 nM T20600 C61NWL 54582924 IC50 = 9125 nM T20600 CO0AG3 54583923 IC50 = 747 nM T20600 CI2DL4 54583924 IC50 = 3475 nM T20600 CV2WU1 54583925 IC50 = 4700 nM T20600 CXA51D 54584867 IC50 = 6950 nM T20600 C8YSL0 54585834 IC50 = 1012 nM T20600 C9B5OF 54586343 IC50 = 2987 nM T20600 C7A8ER 54587376 IC50 = 9200 nM T20600 CGY3W2 71471109 IC50 > 100000 nM T20600 CKZ2H0 71582971 IC50 > 500000 nM T20600 C4WJ5F 71582972 IC50 > 500000 nM T20600 CXA62J 71582973 IC50 = 1030 nM T20600 CNZS31 71582974 IC50 > 500000 nM T20600 CE4L9D 71582975 IC50 > 500000 nM T20600 CXMS80 71583078 IC50 > 500000 nM T20600 C30UIL 71583079 IC50 > 500000 nM T20600 CJBC14 71583080 IC50 = 2610 nM T20600 C57MOP 71583081 IC50 > 500000 nM T20600 CS0YK9 71583082 IC50 > 500000 nM T20600 C3UTO9 71583083 IC50 > 500000 nM T20600 CW1R5Q 71583084 IC50 > 500000 nM T20600 CR57LS 71583192 IC50 > 500000 nM T20600 C8B3NZ 71583193 IC50 > 500000 nM T20600 CB6DY7 71583194 IC50 > 500000 nM T20600 CANH70 71716242 IC50 > 100000 nM T20600 C40WIR 71718085 IC50 = 100000 nM T20600 CU75VK 71719897 IC50 = 600 nM T20600 CBV6F1 71720507 IC50 > 100000 nM T20600 C4U5TO 76311196 IC50 > 10000 nM T20600 CSI53E 76311200 IC50 > 10000 nM T20600 CNOL37 76311201 IC50 = 3878 nM T20600 C8IS5Q 76314800 IC50 = 5082 nM T20600 CK41QI 76314804 IC50 > 10000 nM T20600 CHS61N 76314805 IC50 > 10000 nM T20600 CDY7K0 76318413 IC50 = 3790 nM T20600 CB2N6G 76322078 IC50 > 10000 nM T20600 C8SPW6 76322082 IC50 > 10000 nM T20600 CC2EP6 76325698 IC50 > 10000 nM T20600 CFY79U 76332916 IC50 > 10000 nM T20600 CD35SI 76332917 IC50 > 10000 nM T20600 C3FQX0 76336535 IC50 > 10000 nM T20600 CV4PE6 76336536 IC50 > 10000 nM T20600 CKCI60 90663142 IC50 = 310 nM T20600 C3GPO7 118723314 IC50 = 500000 nM T20600 C8H0EL 118723315 IC50 = 28500 nM T20600 CTE1O2 118723316 IC50 = 500000 nM T20600 CE8O9P 118723317 IC50 = 500000 nM T20600 C48DEF 118723325 IC50 = 500000 nM T20600 C67QMY 118723326 IC50 = 500000 nM T20600 CCJ27M 118723327 IC50 = 500000 nM T20600 COG92V 118723328 IC50 = 500000 nM T20600 CSX85P 118723329 IC50 = 500000 nM T20600 CICB42 118723330 IC50 = 78900 nM T20600 C13BRQ 118723331 IC50 = 12900 nM T20600 CWM2E8 133081971 IC50 > 9999 nM T20600 D08ORM 15487887 IC50 = 8 nM T20600 D0N5MU 4117381 Ki > 50000 nM T20600 D0Q9XX 515950 Ki = 1700 nM T20600 D0V6DX 10640 IC50 = 474 nM T20600 D0Y5IQ 44255320 IC50 = 5000 nM T28330 D04JEE 4946 EC50 > 5011.87 nM T28330 D0H7FW 9870520 Ki = 28.84 nM T28330 D0LI1C 44469321 IC50 > 30000 nM T28330 D01ZXW 122077 IC50 = 0.5623 nM T28330 D0C8ZD 121964 IC50 = 1900 nM T28330 D0EG1F 9914672 Ki = 79.43 nM T28330 D0F6CT 51353551 EC50 = 0.0024 nM T28330 D0W8TS 9898185 IC50 = 3162.28 nM T28330 D0W9ZY 52949124 EC50 = 0.5248 nM T28330 D0XJ0S 108187 IC50 = 1047.13 nM T28330 C7YKF2 1098327 Ki < 10000 nM T28330 CR7Y4G 1109919 Ki > 10000 nM T28330 CA0XN1 3081599 EC50 = 28 nM T28330 CF74HA 6918156 IC50 = 0.5 nM T28330 C6E0TB 9832467 Ki < 10000 nM T28330 C07OFK 9892971 IC50 > 10000 nM T28330 C57IBS 9913081 Ki < 10000 nM T28330 CRT68S 9960432 Ki = 125.89 nM T28330 CKTR60 10008654 IC50 = 5.2 nM T28330 CV56TJ 10031013 IC50 = 75.86 nM T28330 CD7XO3 10032955 EC50 = 3.162 nM T28330 C7SQA8 10032956 IC50 = 229.09 nM T28330 CDT69G 10051431 IC50 = 440 nM T28330 CFO8L6 10071178 Ki = 31.62 nM T28330 CL8M2B 10320262 Ki = 25.12 nM T28330 C16YAW 10343558 Ki = 25.12 nM T28330 CM1D3V 10350069 IC50 = 724.44 nM T28330 C4DIK2 10366068 Ki = 25.12 nM T28330 CD6B7H 10373077 EC50 = 3.981 nM T28330 CTE7N2 10388627 Ki = 25.12 nM T28330 CA5B8O 10391834 IC50 = 1584.89 nM T28330 CYU58T 10415786 IC50 = 39.81 nM T28330 C5Z8IP 10433726 Ki = 25.12 nM T28330 CM97BA 10460632 Ki = 3006 nM T28330 CB1X4K 10483574 IC50 = 79.43 nM T28330 CVE86S 10507071 IC50 = 6850 nM T28330 C91ZVY 10507109 Ki = 50.12 nM T28330 C36HIS 10507561 IC50 = 15.85 nM T28330 CKY68B 10509945 EC50 = 9.12 nM T28330 C1AE8J 10531224 IC50 = 1318.26 nM T28330 C9SUK0 10531430 IC50 = 1584.89 nM T28330 C4S2YR 10555164 IC50 = 138.04 nM T28330 CJZ47Q 10555363 IC50 = 36.31 nM T28330 CRI50M 10555571 IC50 = 42.66 nM T28330 CIN1C4 10555804 IC50 = 13.8 nM T28330 CM7LP6 10556460 IC50 = 309.03 nM T28330 C6LR2W 10580108 IC50 = 389.05 nM T28330 C0IT5X 10603713 IC50 = 17.38 nM T28330 CBRX06 10603714 IC50 = 20.89 nM T28330 C0AV6Q 10626596 IC50 = 524.81 nM T28330 CG02LF 10627173 IC50 = 10.81 nM T28330 CWF78P 10649606 EC50 = 0.014 nM T28330 C1QT8S 10674604 IC50 = 891.25 nM T28330 CXZ4C9 10675328 IC50 = 14.45 nM T28330 C84WOB 10698051 IC50 = 87.1 nM T28330 C89BME 10698109 IC50 = 154.88 nM T28330 CX8P5U 10698905 IC50 = 29.51 nM T28330 C90UHA 10699165 IC50 = 660.69 nM T28330 CG1KP5 10700916 EC50 = 1.549 nM T28330 CN53KG 10721792 IC50 = 120.23 nM T28330 C3R0HF 10722103 IC50 = 112.2 nM T28330 CA9O7Y 10722372 IC50 = 2511.89 nM T28330 CHD26N 10746778 IC50 = 1995.26 nM T28330 C7MS8F 10769675 IC50 = 478.63 nM T28330 C7KR4C 10769902 IC50 = 13.18 nM T28330 CU8KV7 10770092 IC50 = 17.78 nM T28330 CU59WT 10793168 IC50 = 107.15 nM T28330 CLMG75 10793883 IC50 = 38.9 nM T28330 C4G5HX 10794311 IC50 > 10000 nM T28330 CV2LI6 10817241 IC50 = 128.82 nM T28330 C8VBP1 10817395 IC50 = 8.318 nM T28330 CNL17K 10817407 IC50 = 354.81 nM T28330 CPER12 10819755 EC50 = 0.02512 nM T28330 C25UOS 10841112 IC50 = 89.13 nM T28330 C3Y6WE 10841358 IC50 = 42.66 nM T28330 C0ODR4 11027990 IC50 = 35.2 nM T28330 CT7HI5 11154873 Ki > 10000 nM T28330 CGR9A8 11178846 Ki > 10000 nM T28330 C2O3XT 11202178 Ki > 10000 nM T28330 C3NCV9 11212985 Ki > 10000 nM T28330 C8WK7R 11248998 Ki < 10000 nM T28330 C72OIE 11259485 Ki < 10000 nM T28330 CVL2X8 11281656 Ki > 10000 nM T28330 C2ZUE8 11292979 Ki < 10000 nM T28330 CL38VT 11293780 Ki < 10000 nM T28330 CD4I0A 11305046 Ki > 10000 nM T28330 CKL0X6 11316421 Ki < 10000 nM T28330 CBNS24 11316813 Ki < 10000 nM T28330 C9VA4Z 11352971 Ki > 10000 nM T28330 CU75AT 11353036 Ki < 10000 nM T28330 C3QE5S 11362975 Ki > 10000 nM T28330 COG3H2 11363465 Ki > 10000 nM T28330 C9DF4G 11363566 Ki < 10000 nM T28330 CXH69E 11385416 Ki > 10000 nM T28330 C9IX1T 11396307 Ki > 10000 nM T28330 CRA51C 11420366 Ki < 10000 nM T28330 COSZ16 11430523 Ki < 10000 nM T28330 CT0RI9 11431264 Ki < 10000 nM T28330 CXIN31 11442229 Ki > 10000 nM T28330 C9U8VO 11453391 Ki < 10000 nM T28330 C6AYO0 11454197 Ki < 10000 nM T28330 CE96SJ 11464858 Ki > 10000 nM T28330 C58JUC 11465671 Ki < 10000 nM T28330 CF9U1W 11511721 Ki = 1174.9 nM T28330 CV02EM 11512151 Ki = 50.12 nM T28330 C9TE6V 11527738 Ki = 10000 nM T28330 CYF52S 11534407 Ki = 79.43 nM T28330 C21ELY 11534594 Ki = 31.62 nM T28330 CA8WL2 11541048 Ki = 63.1 nM T28330 C7QYJ1 11555166 Ki = 724.44 nM T28330 C16KZS 11556194 Ki = 501.19 nM T28330 C8B2SH 11584582 Ki = 79.43 nM T28330 CK4H5O 11584903 Ki = 8709.64 nM T28330 C24OIW 11592162 Ki < 10000 nM T28330 CN6AR3 11605814 Ki < 10000 nM T28330 CT29GZ 11613982 Ki < 10000 nM T28330 CO3F1P 11627917 Ki = 79.43 nM T28330 C4EHB7 11635377 Ki = 12.59 nM T28330 COM97A 11656338 Ki = 5888.44 nM T28330 C51UDK 11667741 IC50 = 8100 nM T28330 CW79UI 11693225 Ki = 199.53 nM T28330 C42YZA 11700410 Ki = 158.49 nM T28330 CV9M3K 11712880 Ki = 1513.56 nM T28330 CK4SG5 11754311 Ki = 25.12 nM T28330 C65DTB 11765552 IC50 = 60.26 nM T28330 CSX23A 11786290 Ki < 10000 nM T28330 C8L2NZ 11801335 IC50 = 100 nM T28330 CSH7X6 11801911 IC50 = 16.98 nM T28330 C30NLE 15002730 Ki = 25.12 nM T28330 C2LBG8 15002734 Ki = 25.12 nM T28330 C5I4LT 15667001 IC50 = 16 nM T28330 CDJF92 15667003 IC50 = 4.2 nM T28330 CXH92N 15667011 IC50 = 0.99 nM T28330 C6QDI1 16090646 Ki < 10000 nM T28330 C3UCY1 16090647 Ki < 10000 nM T28330 C3HO2S 16090649 Ki < 10000 nM T28330 C4FKT8 16090650 Ki < 10000 nM T28330 CB19JY 16090651 Ki < 10000 nM T28330 CW7KL5 16090652 Ki > 10000 nM T28330 C9Q5YA 16090653 Ki > 10000 nM T28330 CA4PD3 16090658 Ki > 10000 nM T28330 CY9MB5 16090684 Ki > 10000 nM T28330 CY91OD 16090685 Ki > 10000 nM T28330 C4P8KS 16090686 Ki < 10000 nM T28330 C17IOA 16090687 Ki > 10000 nM T28330 C4ETX5 16090688 Ki > 10000 nM T28330 C37DEW 16090689 Ki > 10000 nM T28330 C7Q8LP 16090690 Ki > 10000 nM T28330 COJ46W 16090691 Ki < 10000 nM T28330 CNSU17 16090692 Ki > 10000 nM T28330 C49PFE 16090693 Ki > 10000 nM T28330 CI0XC5 16090694 Ki > 10000 nM T28330 C6QDP7 16090695 Ki > 10000 nM T28330 C3AVH8 16090699 Ki = 3162.28 nM T28330 C9R2PB 16090700 Ki = 199.53 nM T28330 C9K8RC 16090701 Ki = 7943.28 nM T28330 CH1UB0 16090702 Ki = 1995.26 nM T28330 CD7S4Q 16090703 Ki > 10000 nM T28330 CRS7B1 16090773 Ki > 10000 nM T28330 C2KCS0 16090774 Ki > 10000 nM T28330 C8IGT2 16090780 Ki > 10000 nM T28330 CM72TB 16090781 Ki > 10000 nM T28330 C8CI1X 16090782 Ki < 10000 nM T28330 C9QGU2 16090783 Ki > 10000 nM T28330 CF2IW8 16090784 Ki < 10000 nM T28330 CKCX80 16090785 Ki > 10000 nM T28330 C3D8HU 16090786 Ki < 10000 nM T28330 C8WSC9 16090788 Ki > 10000 nM T28330 CYQP41 16090789 Ki = 2511.89 nM T28330 C6MV4D 16090790 Ki > 10000 nM T28330 CJ94QO 16090791 Ki > 10000 nM T28330 C2G8TD 16090792 Ki < 10000 nM T28330 CRF40D 16090793 Ki < 10000 nM T28330 CX68OS 16090794 Ki > 10000 nM T28330 C0V8WI 16090795 Ki < 10000 nM T28330 C06QBM 16090796 Ki < 10000 nM T28330 C5NER1 16090797 Ki < 10000 nM T28330 C3T9MH 16100406 Ki = 130 nM T28330 CH6F0V 16100408 Ki = 8300 nM T28330 CY5F4S 16162108 EC50 = 269.15 nM T28330 C7YG3M 16731537 Ki < 10000 nM T28330 C7U3FA 16731711 Ki = 371.54 nM T28330 C3G0VB 16731712 Ki < 10000 nM T28330 CD9KY3 16731870 Ki < 10000 nM T28330 C6RS1M 16731872 Ki < 10000 nM T28330 CQ45MJ 16731874 Ki > 10000 nM T28330 C8FH9C 16732017 Ki = 6456.54 nM T28330 C9I7PZ 16732018 Ki = 4073.8 nM T28330 C8JR5Q 16732019 Ki = 1737.8 nM T28330 C2OQ0S 16732020 Ki = 6456.54 nM T28330 C5VUZ7 16732021 Ki = 389.05 nM T28330 CXN1C3 16732022 Ki < 10000 nM T28330 C34EYO 16732162 Ki = 457.09 nM T28330 C6CF0K 16732163 Ki < 10000 nM T28330 C4GZY1 16732164 Ki = 549.54 nM T28330 C8DU5M 16732165 Ki = 2511.89 nM T28330 CB7X3W 16732442 Ki < 10000 nM T28330 CY57CK 16732443 Ki = 5754.4 nM T28330 CO95FT 16732444 Ki = 2137.96 nM T28330 CE9M8H 16732592 Ki = 8128.31 nM T28330 C3J2CB 16732593 Ki = 6918.31 nM T28330 CU2FT3 16732598 Ki < 10000 nM T28330 CFT09X 16732750 Ki < 10000 nM T28330 CM4P7G 16732753 Ki < 10000 nM T28330 C9K4UR 16732755 Ki = 7943.28 nM T28330 CB2JR3 16732909 Ki > 10000 nM T28330 CZ14YT 16732911 Ki = 645.65 nM T28330 C35MZK 16732916 Ki = 1905.46 nM T28330 CR0A7J 16733051 Ki = 2951.21 nM T28330 C3LUI7 16733057 Ki < 10000 nM T28330 C9FU1Q 16733182 Ki < 10000 nM T28330 C93FYR 16733185 Ki = 549.54 nM T28330 CF3I5J 16733307 Ki = 660.69 nM T28330 CUF2R0 16733462 Ki = 8511.38 nM T28330 C0RH7Y 16733466 Ki = 2511.89 nM T28330 C1XWA0 16733469 Ki = 2089.3 nM T28330 CK04YG 16733644 Ki = 1698.24 nM T28330 C1RC2P 16733790 Ki < 10000 nM T28330 C76HVW 16755781 EC50 = 0.094 nM T28330 CO7F1T 16755782 EC50 = 1.1 nM T28330 CILG48 21842317 IC50 = 111 nM T28330 CLTI86 21842327 IC50 = 1200 nM T28330 C3NT8C 21842331 IC50 = 480 nM T28330 C53MSQ 21842340 IC50 = 293 nM T28330 CK8GY0 21842400 IC50 = 720 nM T28330 CPQ3K5 22171012 Ki = 25.12 nM T28330 C6VR4P 22171037 Ki = 25.12 nM T28330 C4Y3DN 22171039 Ki = 25.12 nM T28330 CH4V5J 22171089 Ki = 25.12 nM T28330 CKA98D 22171092 Ki = 25.12 nM T28330 CFL43N 23652473 IC50 > 1000000 nM T28330 CZ2PW8 24769543 EC50 = 0.033 nM T28330 CA7XZ6 24769546 IC50 = 0.018 nM T28330 C2YDQ3 24769604 IC50 = 0.01 nM T28330 CO46AU 24769605 EC50 = 0.065 nM T28330 CSCY65 24784940 IC50 = 2.5 nM T28330 C7HSF9 24784941 IC50 = 2.3 nM T28330 C14APO 24784942 IC50 = 22 nM T28330 C6X5AL 24785176 IC50 = 43 nM T28330 C4S1BJ 24785177 IC50 = 6.9 nM T28330 CE32FM 24785178 IC50 = 1.9 nM T28330 C6Y0AR 24785179 EC50 = 7.4 nM T28330 C0O2KU 24785180 EC50 = 5.5 nM T28330 C6ZNQ8 24785430 IC50 = 30 nM T28330 CXH90U 24785431 IC50 = 1.9 nM T28330 CC9TD5 24785432 EC50 = 175 nM T28330 C8A3XU 24785703 EC50 = 1.9 nM T28330 CZ14DY 24785705 IC50 = 0.42 nM T28330 CC8IW7 24861060 IC50 = 0.04 nM T28330 CZ9AS2 24861113 EC50 = 0.048 nM T28330 C6TM1P 24861114 EC50 = 0.053 nM T28330 C39NSA 24861174 EC50 = 0.4 nM T28330 CM0Q9T 24861391 IC50 = 0.03 nM T28330 CA5WE4 24861392 EC50 = 0.14 nM T28330 CCN34R 24861394 EC50 = 0.077 nM T28330 C5C4QR 24990933 IC50 < 50 nM T28330 C8HMZ0 25032312 Ki < 10000 nM T28330 C3NGL2 25032468 Ki < 10000 nM T28330 CK96SR 25033064 Ki < 10000 nM T28330 CM2Z9H 25033065 Ki < 10000 nM T28330 C1O7NJ 25033066 Ki < 10000 nM T28330 CITF86 25033148 Ki < 10000 nM T28330 C67SOQ 25033149 Ki < 10000 nM T28330 CJ10TY 25033150 Ki < 10000 nM T28330 C19WBD 44215880 Ki = 3.9 nM T28330 C6J7EK 44303510 IC50 > 10000 nM T28330 CWKM16 44303511 IC50 = 36.7 nM T28330 CY5Q8R 44303654 IC50 = 2175 nM T28330 CNH0W1 44303663 IC50 > 10000 nM T28330 CD80VI 44303664 IC50 = 2700 nM T28330 C0L8GD 44303722 IC50 = 364 nM T28330 CA8Z0J 44304324 IC50 = 190 nM T28330 C1VM8Q 44306360 IC50 = 31.62 nM T28330 C3ZDK0 44306744 IC50 = 19.95 nM T28330 CB5Q6O 44306823 IC50 = 5.012 nM T28330 CG9HF2 44306868 IC50 = 100 nM T28330 CP92WE 44306887 IC50 = 63.1 nM T28330 CN0SR5 44306888 IC50 = 100 nM T28330 C3MR8J 44328894 Ki = 10 nM T28330 C10ORA 44328951 Ki = 50.12 nM T28330 CZFL34 44329156 Ki = 79.43 nM T28330 CT7I5W 44330874 IC50 = 5.3 nM T28330 C4G1WN 44336539 EC50 = 0.02 nM T28330 C4HYP6 44355590 Ki = 3330 nM T28330 CVO2G3 44355745 Ki = 1080 nM T28330 CMS4H1 44355747 Ki = 3900 nM T28330 C8VW0Y 44355787 Ki = 10000 nM T28330 CHAZ51 44365304 IC50 = 3162.28 nM T28330 CMV8Q7 44365359 IC50 = 251.19 nM T28330 C1RNC2 44365788 IC50 = 10 nM T28330 CTD71M 44367000 IC50 = 2500 nM T28330 CN8SF3 44379428 Ki = 3 nM T28330 C9TZV6 44398261 IC50 = 3.8 nM T28330 CD69PS 44408411 Ki = 1000 nM T28330 C7QV6M 44408483 Ki = 560 nM T28330 C96ELC 44408632 Ki = 840 nM T28330 CI26KP 44417427 Ki > 10000 nM T28330 C0CV9L 44417429 Ki < 10000 nM T28330 CNZ3I4 44417439 Ki < 10000 nM T28330 C5OI3W 44418923 Ki > 10000 nM T28330 C4UPR1 44418924 Ki = 10000 nM T28330 CWT4D8 44425005 Ki = 7079.46 nM T28330 C2PEJ5 44425006 Ki = 3981.07 nM T28330 C7R2IK 44444763 Ki = 25.12 nM T28330 C0C1JA 44444767 Ki = 25.12 nM T28330 C91GMK 44444777 Ki = 25.12 nM T28330 CL94GA 44451519 Ki = 446.68 nM T28330 CXJ5N0 44451522 Ki = 616.6 nM T28330 CN8B5I 44451523 Ki < 10000 nM T28330 CMF6V5 44451547 Ki = 2089.3 nM T28330 C2MP5A 44451581 Ki = 281.84 nM T28330 C9SC7M 44451622 Ki = 2344.23 nM T28330 CH1K6S 44451830 Ki < 10000 nM T28330 CWEV38 44451843 Ki = 3890.45 nM T28330 CIS9D2 44451877 Ki = 1548.82 nM T28330 CVN2E4 44451920 Ki = 2344.23 nM T28330 C4DL5C 44469677 IC50 = 1 nM T28330 C9HFJ2 44562296 EC50 = 0.097 nM T28330 C1UA9S 44562297 EC50 = 0.04 nM T28330 CWT26N 44562298 EC50 = 0.095 nM T28330 C42LFU 44562299 IC50 = 0.08 nM T28330 CK78HN 44562300 EC50 = 0.082 nM T28330 C3QH7F 44562301 IC50 = 0.016 nM T28330 CSJ76G 44562302 EC50 = 0.034 nM T28330 CZ1MF9 44562303 IC50 = 0.067 nM T28330 CQ72YB 44562304 EC50 = 0.074 nM T28330 C9CDJ6 44562305 IC50 = 0.24 nM T28330 CM8A3V 44562306 EC50 = 0.097 nM T28330 CS3C0V 44562307 EC50 = 0.1 nM T28330 CR5Y4S 44562308 EC50 = 0.21 nM T28330 C9APN5 44562309 EC50 = 0.16 nM T28330 CF1BD0 44562310 EC50 = 0.18 nM T28330 C2JL9N 44562311 EC50 = 0.77 nM T28330 CT57RP 44562312 EC50 = 0.097 nM T28330 C2Y5XD 44562313 EC50 = 0.46 nM T28330 CJ72VF 44562314 EC50 = 0.14 nM T28330 C3IB9C 44578251 EC50 = 74 nM T28330 C3HFG1 44578305 IC50 = 8 nM T28330 CQ1DN3 44578398 IC50 = 630 nM T28330 C5FA0D 44578399 EC50 = 9.1 nM T28330 CG5PO8 44578422 IC50 = 16 nM T28330 C97ZLF 44578423 IC50 = 1.9 nM T28330 C5X3RK 44578424 EC50 = 1.1 nM T28330 CCS0G8 44578455 IC50 = 8.6 nM T28330 C45QLM 44578456 EC50 = 106 nM T28330 CW0F5K 44578457 EC50 = 0.078 nM T28330 CV5X3L 44578529 EC50 = 962 nM T28330 C4U0QS 44578530 IC50 = 130 nM T28330 CB31ZF 44578531 EC50 = 1349 nM T28330 CB9X2L 44578562 EC50 = 471 nM T28330 C8ES9Z 44578611 IC50 = 35 nM T28330 C65UYX 44578647 IC50 = 1.9 nM T28330 C94RSO 44578686 EC50 = 0.25 nM T28330 CLW1R5 44578727 EC50 = 0.53 nM T28330 CDIW83 44578728 EC50 = 0.13 nM T28330 CCP04Y 44578729 EC50 = 0.12 nM T28330 CJE1O8 44578764 EC50 = 0.26 nM T28330 C2A4JT 44578767 IC50 = 0.45 nM T28330 CPV6Q1 44578772 EC50 = 308 nM T28330 C6FE1M 45102806 Ki = 158.49 nM T28330 CM6BH7 45255234 Ki = 251.19 nM T28330 CYTL70 45486933 Ki = 100 nM T28330 CQH80S 45486935 Ki = 251.19 nM T28330 C7YUL8 45486936 Ki = 158.49 nM T28330 C1KLB2 45486940 Ki = 1995.26 nM T28330 COT6U7 45486941 Ki = 398.11 nM T28330 CAQ7Z9 45486947 Ki = 199.53 nM T28330 C6FGL0 45486949 Ki = 3981.07 nM T28330 CSR39Z 45486955 Ki = 199.53 nM T28330 CDZ82O 45486958 Ki = 3162.28 nM T28330 CMI20Q 45486964 Ki = 398.11 nM T28330 CD02XL 45486967 Ki = 158.49 nM T28330 C1X3BW 45486968 Ki = 316.23 nM T28330 CC8W1B 45486969 Ki = 199.53 nM T28330 CV17ZB 45486970 Ki = 3981.07 nM T28330 CZ04GO 45486971 Ki > 10000 nM T28330 C2WJI9 45486974 Ki = 25.12 nM T28330 C5HP4B 45486976 Ki = 251.19 nM T28330 CXR7T6 45486985 Ki = 316.23 nM T28330 CIX0G1 45486994 Ki = 1000 nM T28330 C1PZ8J 45486995 Ki = 1995.26 nM T28330 C06PMK 45486997 Ki = 3981.07 nM T28330 CQ31XM 45487002 Ki = 125.89 nM T28330 C3YB8W 45487003 Ki = 79.43 nM T28330 C6SQZ7 45487006 Ki = 100 nM T28330 CGH4V3 46234820 IC50 = 80.1 nM T28330 C5KH7S 46234969 IC50 = 4.24 nM T28330 CQAS17 46234970 IC50 = 44.7 nM T28330 CD0WG8 46235271 EC50 = 0.1202 nM T28330 CHD2N7 46235272 EC50 = 2.7 nM T28330 C94EJG 46869398 EC50 = 0.063 nM T28330 C8Y2QS 49798104 Ki > 10000 nM T28330 C6LEM8 49798106 IC50 = 125.89 nM T28330 C8EG6Y 49798111 Ki = 1400 nM T28330 C24DUW 49798112 Ki = 9 nM T28330 C2US0X 52940616 EC50 = 522 nM T28330 C5T0BN 52942901 EC50 = 91.3 nM T28330 CCOU43 52943046 EC50 = 628 nM T28330 CS2DM8 52944224 EC50 = 160 nM T28330 CL5G9A 52945789 EC50 = 1810 nM T28330 CW60FV 52946666 EC50 = 645 nM T28330 C4QWB8 52946667 IC50 = 246 nM T28330 CP0NO1 52950956 IC50 > 700 nM T28330 C7PC2V 52950958 IC50 > 700 nM T28330 CMYU60 52951093 IC50 > 700 nM T28330 C8ZL7M 52951227 IC50 > 700 nM T28330 C2VK4G 52951333 IC50 > 700 nM T28330 CG80QW 52951789 IC50 > 700 nM T28330 CXZL73 52952034 IC50 > 700 nM T28330 C6UQ3N 53233689 EC50 = 0.065 nM T28330 C2DIE0 53465843 Ki = 973 nM T28330 CB90RU 53465844 Ki = 0.32 nM T28330 C9J3NZ 54580263 EC50 = 38 nM T28330 CN56CG 54580264 IC50 = 2925 nM T28330 C74EHP 54580265 EC50 = 286 nM T28330 CV4Z2K 54580266 IC50 = 2.4 nM T28330 C6WDJ8 54580267 EC50 = 61 nM T28330 CF0V5K 54580295 EC50 = 0.71 nM T28330 CE98TJ 54580296 EC50 = 17 nM T28330 CGP10T 54581259 IC50 > 10000 nM T28330 CK85VP 54581260 IC50 = 35 nM T28330 C0XN2Z 54581261 EC50 = 34 nM T28330 C4SC7B 54581301 EC50 = 41 nM T28330 C8YT9J 54581302 EC50 = 9.6 nM T28330 CXP3W9 54582287 EC50 = 6.1 nM T28330 C5NZ0G 54582288 EC50 = 37 nM T28330 C7MT8A 54582313 EC50 = 5020 nM T28330 C10GBP 54583260 EC50 = 1.8 nM T28330 CSD2T3 54583296 EC50 = 0.24 nM T28330 CF12HS 54583297 EC50 = 59 nM T28330 CK01LS 54583298 EC50 = 0.2 nM T28330 C40TZF 54584222 IC50 > 10000 nM T28330 COGN42 54584255 EC50 = 7.5 nM T28330 CW6E2U 54586147 IC50 = 35 nM T28330 CB7AL6 54586148 IC50 = 0.18 nM T28330 CF1M5T 54586149 IC50 = 174 nM T28330 C5ME1Z 54586174 IC50 = 16.9 nM T28330 CE5SJ2 54586175 IC50 = 9.9 nM T28330 C9XP0E 54587149 IC50 = 33 nM T28330 CZ9S1K 54587150 EC50 = 1.3 nM T28330 CT14KG 54587151 EC50 = 256 nM T28330 C4HMO9 56663037 IC50 > 700 nM T28330 CZL6U4 56663263 IC50 > 700 nM T28330 CRL92U 56666696 IC50 > 700 nM T28330 CV38BZ 56683899 IC50 > 700 nM T28330 CSX93Z 70681224 EC50 = 31.9 nM T28330 CP73WX 70683295 IC50 = 68.6 nM T28330 C9V7QF 70683305 IC50 = 87.6 nM T28330 C15FHQ 70685411 IC50 = 248 nM T28330 CCQ5U4 70689603 EC50 = 52.5 nM T28330 C7BJ3X 70689619 EC50 = 2116.8 nM T28330 CQXZ61 70691750 EC50 = 12.9 nM T28330 C07BDF 70693814 IC50 = 340 nM T28330 CCN89Z 70695922 EC50 = 400 nM T28330 C0IJ1E 70695933 IC50 = 373 nM T28330 CR6KF1 70695934 IC50 = 38.1 nM T28330 CWH6T3 72548703 IC50 = 0.12 nM T28330 CNC3S0 73345637 IC50 = 15000 nM T28330 C5KT3R 73346888 IC50 < 100000 nM T28330 CG2PW4 73348650 IC50 = 32 nM T28330 CYL21W 73348651 IC50 = 6450 nM T28330 CO8BC0 73350236 IC50 = 26660 nM T28330 CIFQ07 73350237 IC50 = 7460 nM T28330 C5G8NK 73350238 IC50 = 7200 nM T28330 CE17QO 73351737 IC50 = 26340 nM T28330 CEVU91 73353218 IC50 = 6940 nM T28330 CGSW23 73354720 IC50 = 24750 nM T28330 CA8MQ1 73354785 Ki = 15 nM T28330 C6C0SX 90663256 IC50 = 7400 nM T28330 CZ61LK 127034966 EC50 > 5011.87 nM T28330 CA0SN5 127034967 EC50 > 5011.87 nM T28330 C1GY2T 135156251 EC50 > 10000 nM T28330 C3ZNX5 135423404 Ki = 467.74 nM T28330 CR79SC 135529065 Ki = 117.49 nM T28330 C0OK8I 135610887 Ki = 588.84 nM T28330 CEX49M 136000594 EC50 = 88 nM T28330 C8IP3M 136036821 Ki = 72.44 nM T28330 C6EOV2 136036823 Ki = 316.23 nM T28330 CB89KA 155514270 EC50 = 0.2512 nM T28330 C9MB4S 155514432 EC50 = 0.2138 nM T28330 CDK7N6 155515427 EC50 = 0.3631 nM T28330 C07LPH 155516677 EC50 = 0.1288 nM T28330 CBJH23 155517239 IC50 = 0.1096 nM T28330 CB1SI3 155517761 EC50 = 0.5012 nM T28330 CBG5S4 155517868 EC50 = 912.01 nM T28330 CTV3M6 155521287 IC50 = 5940 nM T28330 CKC61A 155524181 EC50 = 0.06761 nM T28330 CH5AU4 155524770 EC50 = 0.1585 nM T28330 CAE58M 155526914 EC50 = 0.1622 nM T28330 C9HIR7 155530671 EC50 = 0.06026 nM T28330 C30VKS 155531277 EC50 = 11.75 nM T28330 CKL8Y2 155532425 EC50 = 0.1096 nM T28330 CN0VP5 155532759 IC50 = 0.1072 nM T28330 C12IEY 155533399 EC50 = 0.166 nM T28330 CVBR79 155533520 EC50 = 8.511 nM T28330 CHV1D9 155535107 EC50 = 0.1072 nM T28330 C09DZK 155535249 EC50 = 0.166 nM T28330 CNB7M5 155535579 EC50 = 0.1698 nM T28330 CKI3E1 155536333 EC50 = 0.1349 nM T28330 CO07KD 155537344 EC50 = 0.1072 nM T28330 C8QIH3 155539345 IC50 = 0.06026 nM T28330 C2FBL5 155540394 EC50 = 1.122 nM T28330 CWP54F 155540415 EC50 = 602.56 nM T28330 CMV82T 155540739 EC50 = 0.2455 nM T28330 CB18RV 155542488 EC50 = 0.1905 nM T28330 CGN96I 155542545 EC50 = 3.311 nM T28330 CY6E8B 155543163 EC50 = 0.2951 nM T28330 CS5N7E 155543846 EC50 = 0.9772 nM T28330 C39DSM 155543995 EC50 = 0.3715 nM T28330 C7K4ZA 155544674 EC50 = 0.1288 nM T28330 CLB1R7 155546692 EC50 = 0.3236 nM T28330 C7Z8OY 155547906 IC50 = 0.07943 nM T28330 C1PV3I 155548381 EC50 = 0.389 nM T28330 C1GEA7 155550911 EC50 = 1.622 nM T28330 CQ9S8X 155551968 EC50 = 0.2138 nM T28330 C1DG3Q 155552556 EC50 = 0.182 nM T28330 C4QSR2 155553269 IC50 = 40.74 nM T28330 C3K4NQ 155553502 EC50 = 11.75 nM T28330 C51ZHW 155555065 IC50 = 0.09772 nM T28330 C8V6RX 155555346 IC50 = 0.0871 nM T28330 CDF1E8 155557064 EC50 = 0.1148 nM T28330 CN68GS 155557285 EC50 = 229.09 nM T28330 CO1N8R 155558199 EC50 > 1000 nM T28330 C0GE9L 155559320 IC50 = 0.07586 nM T28330 C2DFE4 155560670 IC50 = 0.07943 nM T28330 CLI24D 155562281 IC50 = 0.04266 nM T28330 CFZ19O 155564367 EC50 = 117.49 nM T28330 CFYB81 155564421 EC50 = 0.1549 nM T28330 CQ8G9E 155566319 IC50 = 0.07413 nM T28330 CK98TD 155568312 EC50 = 0.5012 nM T28330 CP23WI 44572148 Ki = 173.78 nM T28330 D00OFV 3035433 IC50 = 1400 nM T28330 D01ADK 11693641 Ki > 10000 nM T28330 D01AQC 9811733 Ki = 3600 nM T28330 D02ZML 5311148 IC50 = 22.91 nM T28330 D03EPA 11051303 IC50 = 97.72 nM T28330 D05QBF 443375 Ki = 0.02344 nM T28330 D05RRZ 10348659 IC50 = 63.1 nM T28330 D05YZC 59751 Ki = 10.4 nM T28330 D06BRA 11520765 IC50 = 6456.54 nM T28330 D06CIH 11200806 IC50 = 4000 nM T28330 D06KWA 11442807 IC50 = 12700 nM T28330 D07ICW 11556976 Ki = 32 nM T28330 D07LQQ 11564210 Ki = 9.6 nM T28330 D09EMR 11136782 IC50 = 1949.84 nM T28330 D0E2OG 11614928 Ki = 910 nM T28330 D0F1VP 44409521 IC50 = 2800 nM T28330 D0F1XY 44408590 Ki > 10000 nM T28330 D0FF6S 16038374 IC50 > 2000 nM T28330 D0I8AF 9833444 EC50 = 0.04365 nM T28330 D0I9PH 16100409 Ki = 1900 nM T28330 D0J7GJ 44408484 Ki = 10000 nM T28330 D0N6DN 44408524 IC50 = 4073.8 nM T28330 D0O7PT 60182 IC50 = 195 nM T28330 D0QP2S 44408526 Ki = 1900 nM T28330 D0R4GI 11040230 Ki = 5100 nM T28330 D0S7SO 16100407 Ki > 10000 nM T28330 D0TR0U 10942040 IC50 = 1096.48 nM T28330 D0U6OA 10909103 Ki = 5700 nM T28330 D0V9DY 16100410 Ki = 7000 nM T28330 D0X7LC 11061906 Ki = 870 nM T28330 D0Z4SS 44572147 Ki = 3.715 nM T18143 D03VOJ 8768 IC50 = 239000 nM T18143 C54JUR 25043 IC50 = 141000 nM T18143 C70HVL 77888 IC50 = 137000 nM T18143 CPI2E4 80447 IC50 = 71600 nM T18143 C07AKH 786691 IC50 = 20000 nM T18143 CY4MC6 3505109 IC50 = 145000 nM T18143 CGN9J7 44267478 IC50 = 25000 nM T18143 CH4Q6A 145964401 IC50 = 6100 nM T18143 CHU61S 145964420 IC50 = 600 nM T18143 C6YCA8 145964710 IC50 = 700 nM T18143 CV6F7L 145966788 IC50 = 600 nM T18143 CBWX17 145967285 IC50 = 900 nM T18143 COR9X3 145972736 IC50 = 700 nM T18143 CQ0M2X 145972809 IC50 = 7500 nM T18143 CF95RZ 145972878 IC50 = 600 nM T18143 CXI0D1 145975081 IC50 = 700 nM T18143 CG84ZR 145975487 IC50 = 400 nM T18143 C91FOT 145976006 IC50 = 800 nM T18143 C3F4UH 145978039 IC50 = 500 nM T79062 D00TLN 2913 Ki = 50.12 nM T79062 D00XWD 135409453 Ki < 100 nM T79062 D01AZG 5073 Ki = 0.4 nM T79062 D01ZII 2726 Ki = 10.72 nM T79062 D02HED 4748 Ki = 23 nM T79062 D03ELL 2159 Ki = 25.12 nM T79062 D03WEX 9966051 Ki = 19 nM T79062 D04JEE 4946 EC50 > 5011.87 nM T79062 D05MBZ 129211 Ki = 84 nM T79062 D05XGO 11154555 Ki = 111 nM T79062 D05ZIK 4205 Ki = 265 nM T79062 D06XZR 27400 Ki = 25 nM T79062 D08VRO 3822 Ki = 1258.93 nM T79062 D09IOI 2170 Ki = 500 nM T79062 D09TPF 23897 Ki = 265 nM T79062 D0CQ0Z 33630 Ki = 280 nM T79062 D0D1AL 3559 Ki = 316.23 nM T79062 D0G8NN 119570 Ki = 1188 nM T79062 D0H3HM 60795 Ki = 10.3 nM T79062 D0H7KF 5002 Ki = 63.1 nM T79062 D0P0OU 11978813 Ki = 3.7 nM T79062 D0R1JV 60854 Ki = 5 nM T79062 D0R6RO 4184 Ki = 56 nM T79062 D0U1OE 5452 Ki = 70 nM T79062 D0UA0I 28693 Ki = 6.31 nM T79062 D0V4QS 135398745 Ki = 79.43 nM T79062 D0W5HK 216239 Ki = 7071 nM T79062 D0X6BV 6918314 Ki = 3900 nM T79062 D0Z1RV 135398737 Ki = 5.5 nM T79062 D0Z6UC 5358 Ki = 1000 nM T79062 D04GMY 11842633 Ki < 100 nM T79062 D08CJK 1150 Ki = 158.49 nM T79062 D09IRN 21071390 Ki = 8635 nM T79062 D0N1HW 5311200 Ki = 226.3 nM T79062 D0R9HI 11256720 Ki = 14230 nM T79062 D00OWF 5280953 Ki = 5500 nM T79062 D02JMI 9888211 Ki = 100 nM T79062 D03ZZH 9887537 Ki = 63.1 nM T79062 D06DZI 107780 Ki > 10000 nM T79062 D06ZVC 10150497 Ki = 679 nM T79062 D07BCO 5684 Ki = 10000 nM T79062 D08AWI 11430856 Ki = 700 nM T79062 D08PUW 64982 IC50 > 200000 nM T79062 D0B7SP 11292933 Ki = 158.49 nM T79062 D0K8NW 5074 Ki = 15.85 nM T79062 D0L9SN 4431 Ki = 0.6 nM T79062 D0M7LV 5761 Ki = 6.31 nM T79062 D0Q2JS 10436045 Ki = 63.1 nM T79062 D0U7VZ 11225102 Ki < 100 nM T79062 D0YP7L 6604889 Ki = 0.3388 nM T79062 CZUI83 2769 Ki = 1000 nM T79062 C5H9CN 9287 Ki = 102.33 nM T79062 CFGH18 27620 Ki = 364 nM T79062 C8Y6DE 37461 Ki = 63.1 nM T79062 C6WDL7 49756 Ki = 145 nM T79062 CIOE06 69729 Ki = 140 nM T79062 CN9GK1 104911 Ki > 10000 nM T79062 CBH8L0 156308 Ki = 5000 nM T79062 CGT8R0 160510 Ki = 280 nM T79062 CLK7P3 169713 IC50 = 143 nM T79062 C4J5ZF 185617 IC50 = 63400 nM T79062 C9XWA6 198914 Ki = 1100 nM T79062 CP2DY7 198967 Ki = 97000 nM T79062 CVI6X5 213046 Ki = 0.5 nM T79062 C2V5FA 398712 Ki = 30 nM T79062 CYV1R3 417052 Ki = 2960 nM T79062 CD8Z9H 424430 Ki = 26 nM T79062 C4O6RK 435595 Ki = 84 nM T79062 CFJ3R2 452533 Ki = 27 nM T79062 CGF6W2 642376 IC50 = 126600 nM T79062 CTN56Q 647533 Ki > 4000 nM T79062 CXQ6U0 735755 IC50 > 10000 nM T79062 C2VLP8 752521 Ki = 2083 nM T79062 C9FI5L 1296368 Ki = 25390 nM T79062 C6VZT7 1984087 Ki = 8000 nM T79062 CGS9R7 2133793 Ki = 4718 nM T79062 CG9N3A 2136365 Ki = 6371 nM T79062 CT8KN9 2232766 Ki = 2307 nM T79062 CA2OY6 2737389 Ki = 1.4 nM T79062 CE50LO 2756712 Ki = 25 nM T79062 C1C4LH 2843443 Ki = 12250 nM T79062 CRA6F5 2853434 Ki = 1473 nM T79062 C3QRD6 2867758 Ki = 6100 nM T79062 CL2G3H 2870750 Ki = 13020 nM T79062 CC74QS 2872937 Ki = 20090 nM T79062 CRF65H 2880253 Ki = 10100 nM T79062 CET7C8 2921525 Ki = 14100 nM T79062 C2DE6R 2927683 Ki = 3800 nM T79062 CF01YE 2928642 Ki = 8400 nM T79062 CY8R6Q 2948971 Ki = 18080 nM T79062 CLXQ01 2950739 Ki = 10400 nM T79062 CO0C7J 2962174 Ki = 84500 nM T79062 CAM8H3 3066250 IC50 = 9800 nM T79062 CT9L0D 3084440 Ki = 80 nM T79062 C6SA2G 3132842 Ki = 37200 nM T79062 CNX8I1 3245407 IC50 > 1000 nM T79062 CX8W7I 3377940 Ki = 1700 nM T79062 CS8KE2 3649661 Ki = 472 nM T79062 C6SHA4 4713248 Ki = 950 nM T79062 CRUB15 4723431 Ki = 1281 nM T79062 C7PX9E 4790508 Ki = 197 nM T79062 C9NKP1 5216959 Ki = 265 nM T79062 C4BKS2 5242341 Ki = 502 nM T79062 C4J3HP 5640104 Ki = 3490 nM T79062 CGM63Y 6540428 Ki = 12.59 nM T79062 C0QCK1 6918455 Ki = 3981.07 nM T79062 CW0ZE5 6918542 Ki = 600 nM T79062 CC5PQ0 6918601 Ki > 5800 nM T79062 C1WXY3 6918603 Ki < 7943.28 nM T79062 CD0Z4I 6918648 Ki = 3162.28 nM T79062 C8AL9V 6918689 Ki < 100000 nM T79062 CI0X2F 7059581 Ki = 1 nM T79062 C2F3BY 7125890 Ki = 9566 nM T79062 CUD06Z 9796627 Ki = 1600 nM T79062 CFC9Y5 9799318 Ki = 6.457 nM T79062 CG0UK3 9803482 Ki = 16.98 nM T79062 CE0DI5 9804612 Ki = 79.43 nM T79062 CNX4F0 9805456 Ki < 5011.87 nM T79062 CWOS30 9817810 Ki = 29 nM T79062 CFBH76 9820952 Ki = 31.62 nM T79062 CBN06W 9839050 Ki = 13 nM T79062 CE3W4V 9845006 Ki = 2.138 nM T79062 CM13ZV 9856041 Ki = 24000 nM T79062 C0ZR3E 9861687 IC50 > 1000 nM T79062 CNCK78 9862256 Ki = 460 nM T79062 C4H7DK 9864569 IC50 < 50 nM T79062 CB1F0C 9867475 Ki = 1300 nM T79062 C7AB8O 9870053 Ki < 5011.87 nM T79062 CQ4LC2 9872676 Ki = 1750 nM T79062 CCLN49 9878197 Ki = 49 nM T79062 C9NF3D 9881600 Ki = 0.6 nM T79062 C08DBF 9885982 Ki = 3 nM T79062 CL1W0B 9887186 Ki = 5.754 nM T79062 CJW1P5 9888494 Ki = 2.239 nM T79062 C6N8UE 9889681 Ki < 10000 nM T79062 CM52WU 9890119 Ki = 2511.89 nM T79062 CEG1K5 9891002 Ki = 1584.89 nM T79062 C7QMK5 9891617 Ki < 5011.87 nM T79062 CEL29O 9891618 Ki = 1995.26 nM T79062 C3J8GU 9892409 Ki < 7943.28 nM T79062 CAM25C 9894665 Ki = 10 nM T79062 CUN81Q 9905249 Ki > 10000 nM T79062 CYWQ50 9906447 Ki > 10000 nM T79062 C9B3EA 9911844 Ki = 7.24 nM T79062 C78MDV 9913554 Ki = 1000 nM T79062 CR9KM0 9921064 Ki = 290 nM T79062 C4UYZ7 9927441 Ki = 3700 nM T79062 CYVZ47 9934284 Ki = 39.81 nM T79062 CO2RS8 9934709 Ki = 0.6761 nM T79062 CWO45F 9935387 Ki = 630.96 nM T79062 CX6E8C 9945703 Ki = 6 nM T79062 CQ04ZS 9950396 Ki = 400 nM T79062 CK8NR2 9954121 Ki < 10000 nM T79062 CHOJ30 9956365 Ki = 3.548 nM T79062 CFR41N 9957068 Ki < 3981.07 nM T79062 CFN50J 9978683 Ki = 579 nM T79062 CS40QN 10015688 Ki = 0.7 nM T79062 CV7R9F 10020040 Ki = 335.9 nM T79062 CK18LT 10020895 Ki > 5000 nM T79062 C2EUY0 10035109 Ki > 10000 nM T79062 C57TZR 10042333 Ki = 1345 nM T79062 C0KWB6 10062885 Ki = 1.1 nM T79062 CR68SH 10064053 Ki = 9.78 nM T79062 C8Z6MA 10067306 IC50 = 1217 nM T79062 CKA5F4 10084076 Ki = 18 nM T79062 C93RNG 10090247 Ki = 7 nM T79062 CA5H7K 10106205 Ki = 16 nM T79062 C4Q3UL 10154897 Ki = 3 nM T79062 C7F1ED 10183148 IC50 = 135000 nM T79062 CW09SL 10202089 Ki = 6 nM T79062 C4Q2SH 10249573 Ki = 10 nM T79062 CMRA02 10257042 Ki < 794.33 nM T79062 CH31DX 10267394 Ki = 412.3 nM T79062 CTWJ70 10274894 Ki = 2.042 nM T79062 CU89JD 10314060 Ki = 102.8 nM T79062 C9IAV3 10346043 Ki = 1.023 nM T79062 CA7IM5 10379532 Ki = 1.096 nM T79062 CR3KU9 10380133 IC50 > 5000 nM T79062 CMZA83 10383646 Ki = 753 nM T79062 C4L5PQ 10404657 Ki = 8.511 nM T79062 C04WGF 10407367 IC50 = 511 nM T79062 C4TPN1 10413595 Ki = 0.3162 nM T79062 C2B0IU 10421236 IC50 > 10000 nM T79062 CR4LS0 10430623 Ki = 1563 nM T79062 CD7U5I 10433930 Ki = 1.995 nM T79062 CO7IV6 10450593 Ki = 0.1995 nM T79062 COV85C 10472143 Ki = 14 nM T79062 C5LBS7 10472158 IC50 = 1362 nM T79062 C26KCR 10475231 Ki = 2 nM T79062 CEF2O6 10478367 Ki = 1412 nM T79062 CL70NJ 10499156 Ki = 10 nM T79062 CN29IF 10500557 Ki = 2.138 nM T79062 CWH7R8 10521887 Ki = 26.33 nM T79062 C9B7LR 10552788 Ki = 19.95 nM T79062 CHE80N 10573876 Ki = 1.995 nM T79062 CAVR62 10596321 Ki = 10 nM T79062 CO23YX 10597140 Ki = 15.85 nM T79062 CZ6WS8 10619437 Ki = 125.89 nM T79062 CAPO49 10638372 Ki = 105 nM T79062 CK08CW 10643153 Ki = 10000 nM T79062 CN40TJ 10668422 Ki < 1000 nM T79062 CBE87R 10706626 Ki = 13.4 nM T79062 CU32PG 10714877 Ki = 10.35 nM T79062 C1PG3A 10715573 Ki = 31.62 nM T79062 CJ4HC8 10715998 Ki = 15.85 nM T79062 CZ3A0O 10737314 Ki = 100 nM T79062 CIVN21 10767321 Ki = 15.85 nM T79062 C2AFT6 10785644 Ki = 1584.89 nM T79062 C3SWV9 10785714 Ki = 5 nM T79062 C75SKC 10811746 Ki = 3.802 nM T79062 CG4X1R 10834268 Ki = 1.862 nM T79062 C8MHZ9 10835110 Ki = 3.981 nM T79062 C5Q4IJ 10862697 Ki = 2.344 nM T79062 CFY4V1 10862787 Ki = 12 nM T79062 CVT7J1 10873805 Ki = 7.32 nM T79062 CNEP25 10884517 Ki = 7.943 nM T79062 C67UIY 10884717 Ki = 6.457 nM T79062 CRI50E 10885636 IC50 = 1440 nM T79062 C9C2FI 10895284 Ki = 72.44 nM T79062 CD4YL2 10896196 Ki = 19.05 nM T79062 CX65PW 10907460 IC50 = 2040 nM T79062 CEGJ41 10917174 Ki = 6.026 nM T79062 CU09AV 10937901 IC50 = 762 nM T79062 C7PWT9 10938620 Ki = 109.65 nM T79062 CA42MT 10939416 Ki = 8.71 nM T79062 CNB39C 10947658 Ki = 12 nM T79062 CSLT97 10949380 IC50 = 663 nM T79062 C2MBP7 10949445 Ki = 8.128 nM T79062 C74SOA 10950559 Ki = 74 nM T79062 C47MYE 10960943 Ki = 97.72 nM T79062 CJD58C 10971401 Ki = 4.786 nM T79062 C51NOQ 10982183 Ki < 10000 nM T79062 CK6VF7 10991109 Ki = 63 nM T79062 C4O7MD 10994400 Ki = 101 nM T79062 CJC9K4 11005810 IC50 = 998 nM T79062 C3FIP5 11016205 Ki = 3.68 nM T79062 CS0Z2D 11024311 Ki < 10000 nM T79062 CRS62E 11025847 Ki = 3.548 nM T79062 C0HA7O 11047374 Ki = 1.995 nM T79062 C23JHR 11047568 IC50 = 1430 nM T79062 C80UIZ 11048252 Ki = 416.87 nM T79062 CONV96 11058267 Ki = 45.71 nM T79062 CD4BW6 11058564 Ki = 43.65 nM T79062 CZN25U 11059148 Ki = 23.99 nM T79062 CG41BK 11071079 IC50 = 726 nM T79062 C15USQ 11101733 Ki = 19.05 nM T79062 C7OFQ4 11102049 Ki = 29.51 nM T79062 CCJ1U3 11112531 Ki = 147 nM T79062 C7DE0U 11113605 IC50 = 1170 nM T79062 CVE8T3 11121216 Ki = 31 nM T79062 C5I0XL 11133795 Ki = 223.87 nM T79062 C0VZK2 11143387 Ki = 9.7 nM T79062 CS90QD 11145126 Ki = 7.079 nM T79062 CYJ79P 11153905 Ki = 2.55 nM T79062 C8ZN3B 11166042 Ki = 37 nM T79062 CEHV65 11173572 Ki = 13.4 nM T79062 C6CL1Y 11178830 Ki = 125.89 nM T79062 C0W4SM 11186523 Ki = 6.5 nM T79062 CXQ3K0 11186985 Ki = 2.91 nM T79062 C5J4NR 11199511 Ki = 8 nM T79062 C9N5QU 11200511 Ki = 74 nM T79062 C90WSG 11248705 Ki = 125.89 nM T79062 CM08DU 11259115 Ki = 200 nM T79062 C4S2VF 11277147 Ki = 17.6 nM T79062 CY6MX5 11282296 EC50 = 2460 nM T79062 CW40XM 11294248 Ki = 251 nM T79062 C9BLC7 11304596 Ki = 501.19 nM T79062 CJS9C0 11304851 IC50 = 25000 nM T79062 CI79LV 11307899 Ki = 6.31 nM T79062 C1VSE5 11327643 Ki = 1000 nM T79062 CGD42N 11361090 Ki > 5000 nM T79062 CXW6B5 11373831 Ki = 19 nM T79062 CBV52J 11384146 Ki = 24 nM T79062 C1BP0U 11385380 Ki > 1000 nM T79062 CF4OX6 11397149 Ki = 79.43 nM T79062 C30ZMW 11397459 Ki = 200 nM T79062 C7GXP9 11397799 Ki = 9 nM T79062 C85LYP 11430418 IC50 = 1000 nM T79062 CNF28A 11432177 EC50 = 6320 nM T79062 CJK2S4 11453751 Ki = 221 nM T79062 CMFC18 11453756 Ki = 200 nM T79062 C9K8UW 11515799 Ki = 7.65 nM T79062 CVAC51 11524003 Ki = 1.19 nM T79062 C7YRP3 11524413 Ki = 0.38 nM T79062 CFW50Y 11525867 Ki = 9.5 nM T79062 C2M0JG 11532105 Ki = 40 nM T79062 C5VHK0 11536843 Ki = 5.1 nM T79062 C0YZ7L 11536844 Ki = 3.3 nM T79062 C1V5CH 11559090 Ki > 10000 nM T79062 C14HEP 11560285 Ki = 296 nM T79062 C1HP5K 11566558 Ki = 4.31 nM T79062 CNH1K4 11568826 Ki = 520 nM T79062 C8NMI4 11575479 Ki = 600 nM T79062 C1I4DF 11582132 Ki = 25 nM T79062 C6D1MA 11584660 Ki > 1995.26 nM T79062 C1M2CP 11589069 Ki = 0.38 nM T79062 CU45DK 11595209 Ki > 10000 nM T79062 CE9W6J 11595790 Ki = 16.8 nM T79062 CGX8F6 11596869 Ki > 3980000 nM T79062 CX5ZM0 11603891 Ki = 5.38 nM T79062 C8EPV2 11610908 Ki = 64 nM T79062 CUA05E 11617668 Ki = 5.4 nM T79062 CD4HR8 11633354 Ki = 2.1 nM T79062 C2OU7Y 11638332 Ki > 10000 nM T79062 C9OLN0 11646336 Ki = 5 nM T79062 CJBV31 11652871 IC50 = 118100 nM T79062 CCX0S1 11653869 Ki = 0.49 nM T79062 CO1L8J 11661471 Ki = 1.02 nM T79062 C4L7TV 11662592 Ki = 4.48 nM T79062 CD91CP 11666595 Ki = 33 nM T79062 CXRC27 11667458 Ki = 10.9 nM T79062 C42RHW 11674602 Ki = 94 nM T79062 CL31JB 11683077 Ki = 11.1 nM T79062 CEQ6W7 11694810 Ki = 4.3 nM T79062 C2QCF5 11697434 Ki = 18 nM T79062 CHR8U4 11697659 Ki = 2.81 nM T79062 C3IML2 11709509 Ki = 0.3 nM T79062 C1N7MO 11725453 Ki = 1 nM T79062 CV82QX 11729084 Ki = 25.12 nM T79062 CLYJ75 11729823 Ki = 8.76 nM T79062 C7PVL8 11730467 IC50 = 2130 nM T79062 CG72CS 11732538 Ki = 20 nM T79062 CMO0I9 11739679 Ki = 1555 nM T79062 C57IKL 11740526 Ki = 9.772 nM T79062 CPG15O 11743399 IC50 > 1000 nM T79062 CYV02C 11747350 Ki = 510 nM T79062 C3F5DX 11761059 IC50 = 4420 nM T79062 C9LUA7 11773414 Ki = 800 nM T79062 C37LEP 11785183 EC50 = 1820 nM T79062 C7A2QD 11793826 Ki = 630.96 nM T79062 C3PY7W 11811833 Ki = 21.88 nM T79062 CQV92N 11825614 Ki = 10.47 nM T79062 CW4BC2 11826723 Ki = 12.3 nM T79062 CXLW54 11948707 Ki = 328 nM T79062 C8JQL7 11957735 IC50 = 1713 nM T79062 C1QY2P 12005903 Ki = 15770 nM T79062 C8EDN0 12088080 Ki = 3 nM T79062 C8RB6W 12088082 Ki = 9 nM T79062 CLC82F 12374770 Ki = 176 nM T79062 CCG14E 13091356 Ki = 420 nM T79062 CYN95Z 13091359 Ki = 97 nM T79062 C4V6AS 14135325 IC50 = 179000 nM T79062 CAO70J 14748689 IC50 = 949 nM T79062 C7VAI1 15011772 IC50 > 10000 nM T79062 C30CHU 15512229 Ki < 316.23 nM T79062 CKBD37 15542627 Ki = 17.38 nM T79062 C65SCN 15599151 Ki = 1240 nM T79062 CTPX97 15803947 Ki = 1.3 nM T79062 C1LWZ6 16006605 Ki = 2.4 nM T79062 CK36NS 16006607 Ki = 1 nM T79062 C3M8GJ 16026344 Ki = 5232 nM T79062 C1SR0O 16071847 Ki > 5000 nM T79062 CD3E8L 16093484 Ki = 8.7 nM T79062 CEW91O 16093485 Ki = 2.5 nM T79062 CZ1WJ4 16117151 Ki = 3970 nM T79062 CM32ZX 16117153 Ki > 5000 nM T79062 CXTB90 16117279 Ki = 3216 nM T79062 C1F2LS 16118795 Ki > 5000 nM T79062 C69VDS 16118923 Ki > 5000 nM T79062 CZ2IS9 16660294 Ki > 10000 nM T79062 CT9GP4 16763549 Ki = 13100 nM T79062 CR63LE 17055181 Ki = 3700 nM T79062 C0QX5J 17374371 Ki = 12590 nM T79062 CB2J3R 17747575 IC50 > 100 nM T79062 C42YEX 18133517 Ki = 3187 nM T79062 CI90UP 18133518 Ki = 2544 nM T79062 C7R1IG 18137015 Ki = 1029 nM T79062 C4I1FW 18137017 Ki = 1342 nM T79062 C07EOI 18137020 Ki = 1417 nM T79062 C9PV8A 18180076 IC50 = 1582 nM T79062 CI6TS8 18377342 Ki = 562.34 nM T79062 CHFJ09 18377388 Ki = 173.78 nM T79062 C5KB2J 18377409 Ki = 15.85 nM T79062 CI91VX 18377415 Ki = 812.83 nM T79062 CXR67I 18663036 Ki = 18.4 nM T79062 C6AOE8 19426635 IC50 = 18.62 nM T79062 CUI3R1 19605739 Ki = 1 nM T79062 C7T8JC 19958494 Ki = 318.2 nM T79062 C6LI5E 19958507 Ki = 411 nM T79062 CBY03N 20846175 Ki < 10000 nM T79062 CISE25 21091965 Ki = 80 nM T79062 C6H9WC 21092408 Ki = 88 nM T79062 C3T5HF 21509921 Ki = 100 nM T79062 CFN81Q 21527771 Ki = 656 nM T79062 CH59WN 21533446 Ki = 1044 nM T79062 C4B0TN 21557475 Ki = 1200 nM T79062 CT7XG9 21830793 Ki = 12.9 nM T79062 C9X8PI 22001618 Ki = 2.6 nM T79062 CBN84K 22065997 Ki = 212.9 nM T79062 C1QBE0 22273749 Ki = 11.22 nM T79062 C6UXL4 22330705 Ki = 21400 nM T79062 CZG9S2 22425072 Ki = 12710 nM T79062 CW0V5M 22449331 Ki = 4.467 nM T79062 CPD8Q7 22549784 Ki = 26650 nM T79062 CZ7J4B 22857296 Ki = 6.4 nM T79062 C0L5QK 23111951 Ki = 270 nM T79062 CY10BQ 23133427 Ki = 2.7 nM T79062 C5BUL7 23151712 Ki = 43 nM T79062 C3IF7P 23151734 Ki = 185 nM T79062 C0NI3J 23290944 Ki = 198 nM T79062 C57MVP 23369416 Ki = 3.4 nM T79062 C6HE8J 23369421 Ki = 26 nM T79062 CAE7K1 23369450 Ki = 1838 nM T79062 CWQ2X3 23369455 Ki = 48 nM T79062 C7EPU0 23369457 Ki = 1029 nM T79062 CRT2Z3 23661667 Ki = 54 nM T79062 CHGE36 23661734 Ki = 46 nM T79062 C5ZSR7 23661735 Ki = 1200 nM T79062 CQE1N7 23906630 Ki = 16020 nM T79062 CD7CV6 24771120 Ki = 6900 nM T79062 CCEH06 24781896 IC50 > 100 nM T79062 CD86PT 24781897 IC50 > 100 nM T79062 CP7TJ3 24781898 IC50 > 100 nM T79062 CF17PW 24781899 IC50 > 100 nM T79062 C1JSY8 24781900 IC50 > 100 nM T79062 CJI2O1 24782049 IC50 > 100 nM T79062 CK9T1F 24782050 IC50 > 100 nM T79062 C2O7MV 24782051 IC50 > 100 nM T79062 C0G3RV 24782052 IC50 > 100 nM T79062 CR8DV4 24782058 IC50 > 100 nM T79062 C58AMS 24829343 Ki = 0.79 nM T79062 CDC91N 24839550 Ki < 10000 nM T79062 CY21RE 24841480 Ki = 330 nM T79062 CT2YG6 24853955 Ki = 0.6 nM T79062 C2KD1T 24854037 Ki = 0.66 nM T79062 C1BPD9 24854039 Ki = 5.3 nM T79062 CGPC24 24854040 Ki = 8.27 nM T79062 CM01LB 24854041 Ki = 0.67 nM T79062 CI7G6M 24854043 Ki = 4.75 nM T79062 C4WUP5 24854044 Ki = 1.1 nM T79062 CY1XA8 24854103 Ki = 6.99 nM T79062 C42KBQ 24854105 Ki = 1.96 nM T79062 CUW23K 24854106 Ki = 44 nM T79062 CX7MK6 24854108 Ki = 33.38 nM T79062 CS90OD 24854109 Ki = 21 nM T79062 CFHM49 24854111 Ki = 1.45 nM T79062 C80ANM 24854181 Ki = 1.24 nM T79062 CSL8E3 24854183 Ki = 1.5 nM T79062 CFR74S 24854185 Ki = 1.8 nM T79062 CW2Z5A 24854186 Ki = 25.4 nM T79062 C9GYO8 24854187 Ki = 0.43 nM T79062 CB9M0N 24854266 Ki = 9.07 nM T79062 C0LQ1R 24854267 Ki = 3.4 nM T79062 CP23KC 24854269 Ki = 6.57 nM T79062 CI5LC8 24854270 Ki = 9.46 nM T79062 CCUS10 24854272 Ki = 5.97 nM T79062 CFX96I 24854273 Ki = 0.4 nM T79062 C6Y3AG 24854368 Ki = 2.07 nM T79062 CTS4E5 24854369 Ki = 2.55 nM T79062 COZ84H 24854370 Ki = 5.11 nM T79062 C3X9MD 24854371 Ki = 0.6 nM T79062 C7ZEF0 24856058 IC50 > 10000 nM T79062 C3HK0J 24865725 Ki = 19.95 nM T79062 C0O6FX 24865727 Ki = 15.85 nM T79062 C98ZIV 24882509 IC50 = 11.99 nM T79062 C6L7KS 24887518 Ki < 3162.28 nM T79062 CAOF91 24894071 IC50 > 10000 nM T79062 CMN75S 24901425 Ki = 1659.59 nM T79062 CF7IV1 24963856 Ki = 6.2 nM T79062 C8DJG7 24963860 Ki = 8.6 nM T79062 C35XOJ 24964217 Ki = 8.4 nM T79062 CP6K8J 25024727 IC50 > 10000 nM T79062 CI95EF 25192947 Ki = 0.47 nM T79062 CKAS93 25256850 Ki = 6 nM T79062 CW07GN 25256855 Ki = 7 nM T79062 CM2T9Y 25263297 Ki = 5100 nM T79062 CFJM71 25263302 Ki = 5800 nM T79062 CHJ35A 32354149 Ki = 885 nM T79062 CS5QG1 35391328 Ki = 773 nM T79062 C8G7EY 36418162 IC50 = 476 nM T79062 CDV36I 37219401 Ki = 855 nM T79062 CG56DF 42388639 IC50 = 20 nM T79062 C6VL8I 42388965 IC50 = 140 nM T79062 CS2G3E 42388975 IC50 = 289 nM T79062 CJ8FH4 42389129 IC50 = 681 nM T79062 CO51RQ 42389139 IC50 > 10000 nM T79062 CBV62E 42389293 IC50 = 3241 nM T79062 CNV94Z 42389303 IC50 = 9314 nM T79062 CSRX20 42389457 IC50 = 53 nM T79062 CH5QX6 42389467 IC50 = 47 nM T79062 CV9C4D 42428409 Ki = 78 nM T79062 C1SD3E 42618253 Ki = 1230 nM T79062 C0BWG1 42618254 Ki = 902 nM T79062 CAG71H 42618255 Ki = 864 nM T79062 CQ96KL 42618256 Ki = 566 nM T79062 CC1Z7P 42618257 Ki = 1867 nM T79062 CFB70T 42618258 Ki = 17960 nM T79062 CJV5N3 42618259 Ki = 2500 nM T79062 CHA26S 42618260 Ki = 296 nM T79062 CX1KC4 42618261 Ki = 168 nM T79062 C2VWK7 42618262 Ki = 267 nM T79062 CV0CD8 42618263 Ki = 243 nM T79062 CS5TJ8 42618264 Ki = 38 nM T79062 CKOJ59 42618265 Ki = 20 nM T79062 C4J9RQ 42618266 Ki = 78 nM T79062 C16TUL 42618267 Ki = 11 nM T79062 CH3NO7 42618269 Ki = 21 nM T79062 CMGJ03 42618270 Ki = 134 nM T79062 CR6OX0 42618271 Ki > 5000 nM T79062 C7SN5E 42618272 Ki = 31 nM T79062 C3VR7E 42618273 Ki = 335 nM T79062 CA0B9F 42625181 Ki = 68 nM T79062 C3L0TN 42625183 Ki = 69 nM T79062 CW0OU4 42625185 Ki > 1000 nM T79062 CHY12B 42625186 Ki > 1000 nM T79062 CP5X3K 42625188 Ki > 1000 nM T79062 C8QSX3 42625267 Ki = 193 nM T79062 CTM69J 42625269 Ki = 350 nM T79062 CPDG98 42625353 Ki = 63 nM T79062 CK3QD2 42625354 Ki > 1000 nM T79062 CJ64FG 42625356 Ki = 250 nM T79062 C27KEF 42625359 Ki = 160 nM T79062 CN81SE 42625440 Ki = 7 nM T79062 CF7DM0 42625445 Ki = 22 nM T79062 CJI51X 42625446 Ki = 69 nM T79062 CLH7Y0 42626289 Ki = 158 nM T79062 C75QPL 42626291 Ki = 203 nM T79062 C5VTZ6 42626293 Ki = 74 nM T79062 C70SWL 42626361 Ki = 63 nM T79062 CY7W2J 42631003 Ki = 0.153 nM T79062 CV2X5B 42635027 IC50 = 89 nM T79062 CBSD79 42635028 IC50 = 384 nM T79062 CR1S3J 42635029 IC50 = 339 nM T79062 CS9Q3H 42635204 IC50 = 12 nM T79062 C5XBV7 42635205 IC50 = 567 nM T79062 CQ2M5S 42635387 IC50 = 124 nM T79062 CR3KM7 42635388 IC50 = 107 nM T79062 C8TFQ9 42635389 IC50 = 580 nM T79062 CFO4Y1 42635570 IC50 = 223 nM T79062 CWU54L 42635571 IC50 = 373 nM T79062 CV27CE 42635572 IC50 = 377 nM T79062 CJ3NP5 42636941 IC50 > 1000 nM T79062 C0AI7N 43229249 Ki = 354.81 nM T79062 C2RSL9 43840296 Ki = 226 nM T79062 CJ41QV 44126269 Ki = 0.389 nM T79062 CVG6X1 44209472 Ki = 208 nM T79062 CD5AB7 44209480 Ki = 90 nM T79062 C2FDB1 44250364 IC50 > 10000 nM T79062 C8MC0Q 44251387 IC50 > 10000 nM T79062 C5YEA8 44251388 IC50 > 10000 nM T79062 C0BSF6 44251389 IC50 > 10000 nM T79062 CP8S2J 44266156 Ki = 4.467 nM T79062 CM0CW8 44266160 Ki = 6.918 nM T79062 C0P8IF 44266163 Ki = 0.4074 nM T79062 CU67NF 44266164 Ki = 9.333 nM T79062 C14ACY 44266178 Ki = 37.15 nM T79062 CN3ES2 44266182 Ki = 2.042 nM T79062 CKLS45 44266203 Ki = 14.13 nM T79062 CARU58 44266221 Ki = 0.5623 nM T79062 CA1WJ4 44266222 Ki = 2.754 nM T79062 CS2MU8 44266229 Ki = 20.42 nM T79062 CZ84XC 44266244 Ki = 9.12 nM T79062 CR16DY 44266245 Ki = 11.75 nM T79062 CVHM20 44266253 Ki = 27.54 nM T79062 CK7AF0 44266267 Ki = 25.12 nM T79062 C1FTY0 44266268 Ki = 1.66 nM T79062 CU61ZS 44266284 Ki = 11.22 nM T79062 C0C6RL 44266289 Ki = 10.23 nM T79062 C5NS9O 44266315 Ki = 2.512 nM T79062 CO5H2Q 44266317 Ki = 18.62 nM T79062 C6OW2N 44268087 Ki = 32 nM T79062 CNHE76 44276598 Ki = 2.138 nM T79062 CC2OD4 44278111 Ki > 10000 nM T79062 CRMA84 44278114 Ki = 713 nM T79062 CF0Y4M 44278115 Ki > 10000 nM T79062 CA93MC 44319240 Ki = 12.59 nM T79062 C34FTE 44319435 Ki = 8.318 nM T79062 CW16JD 44324737 Ki > 1000 nM T79062 CA84SN 44324765 Ki > 1000 nM T79062 COA3H4 44324800 Ki > 1000 nM T79062 CY04JW 44324972 Ki > 1000 nM T79062 C5VLY2 44326733 Ki = 9 nM T79062 CT7DN4 44327688 Ki = 2.399 nM T79062 CER86D 44327952 Ki = 83 nM T79062 CP9B2K 44340834 Ki = 1.82 nM T79062 CB23YQ 44340835 Ki = 0.7943 nM T79062 CC25ZK 44340836 Ki = 0.5012 nM T79062 CZBQ72 44340850 Ki = 0.8318 nM T79062 CTM65V 44340854 Ki = 0.7079 nM T79062 C6F9XL 44340882 Ki = 57.54 nM T79062 C2S1ZT 44340883 Ki = 6.457 nM T79062 CG6PD8 44340897 Ki = 22.91 nM T79062 CQ3WH6 44341114 Ki = 6.31 nM T79062 C9BDG2 44341126 Ki = 6.457 nM T79062 CK37NE 44341130 Ki = 25.7 nM T79062 CO0ZY5 44341131 Ki = 165.96 nM T79062 CD9ZS8 44342270 IC50 = 849 nM T79062 CPWJ26 44343212 Ki = 39.81 nM T79062 CMX45U 44348383 IC50 = 2.2 nM T79062 CUXH48 44352308 Ki = 1460 nM T79062 C3LKN1 44364048 Ki = 3.162 nM T79062 CND4W7 44368304 Ki = 19.95 nM T79062 C6CUM2 44368306 Ki = 31.62 nM T79062 CH3G4F 44368358 Ki = 31.62 nM T79062 C2S8AQ 44368373 Ki = 100000 nM T79062 C1EO8C 44368383 Ki = 1584.89 nM T79062 CAEZ93 44368384 Ki = 630.96 nM T79062 CK9OQ3 44368683 Ki = 125.89 nM T79062 CB0E1J 44368705 Ki = 10 nM T79062 CS21UK 44368731 Ki = 1.995 nM T79062 CRF67K 44368732 Ki = 3.981 nM T79062 C61PEQ 44368754 Ki = 15.85 nM T79062 CT2BR5 44372581 Ki = 5.012 nM T79062 C08EKS 44374206 Ki = 1200 nM T79062 CVL3U2 44374207 Ki = 7.2 nM T79062 CV8CP3 44374225 Ki = 22 nM T79062 C7FE5A 44374226 Ki = 6800 nM T79062 CX9S1K 44374227 Ki = 3200 nM T79062 C04WKH 44374233 Ki = 4.1 nM T79062 CB2S7T 44374234 Ki = 100 nM T79062 CV62ZP 44374298 Ki = 170 nM T79062 CJ4A2U 44374299 Ki = 12 nM T79062 C4VXQ1 44388858 Ki = 4.3 nM T79062 CTPG47 44388956 Ki > 2000 nM T79062 C1UMV6 44393001 Ki = 60 nM T79062 C64IKJ 44393004 Ki = 4 nM T79062 CT8Y5A 44393007 Ki = 4 nM T79062 C1F5IX 44393021 Ki = 13 nM T79062 C9VH1B 44393022 Ki = 16 nM T79062 CG9S1O 44393045 Ki = 2 nM T79062 CGRD59 44393052 Ki = 23 nM T79062 CBJ84O 44393053 Ki = 54 nM T79062 CPS9T7 44393056 Ki > 1000 nM T79062 C4HVE3 44393057 Ki > 1000 nM T79062 CKV3Z0 44393069 Ki = 3 nM T79062 C7HIJ9 44393072 Ki = 10 nM T79062 C20PMS 44393073 Ki = 0.4 nM T79062 C1E0QH 44393074 Ki = 36 nM T79062 C3H6ML 44393075 Ki = 8 nM T79062 C53UVJ 44393088 Ki = 2 nM T79062 C89NKB 44393089 Ki > 1000 nM T79062 C2QX0I 44393090 Ki > 1000 nM T79062 C0F9MP 44393091 Ki = 0.3 nM T79062 CCS5Q4 44393092 Ki = 0.4 nM T79062 C1KBZ7 44393093 Ki > 1000 nM T79062 CO6EY0 44393113 Ki = 2 nM T79062 C9GEU3 44393114 Ki = 33 nM T79062 CX4C9P 44393133 Ki = 6 nM T79062 CE03ZW 44393134 Ki = 1 nM T79062 C69CFB 44393154 Ki > 41000 nM T79062 CP9K0J 44393161 Ki = 2 nM T79062 CY60BQ 44393162 Ki > 1000 nM T79062 CG5UE1 44393169 Ki = 0.3 nM T79062 CG18AU 44393170 Ki = 5 nM T79062 CZ18RL 44393171 Ki = 5 nM T79062 CHV6D3 44393180 Ki = 0.6 nM T79062 CZB65R 44393192 Ki = 0.4 nM T79062 CK85EB 44393193 Ki = 0.4 nM T79062 CVC86L 44393228 Ki = 3 nM T79062 C7AR1C 44393229 Ki = 4 nM T79062 C4B0OI 44397588 Ki = 1000 nM T79062 C5FP0R 44397589 Ki = 1258.93 nM T79062 CE3G8U 44397670 Ki = 3981.07 nM T79062 CX7O9S 44401041 Ki = 80 nM T79062 C5XC2B 44401042 Ki = 92 nM T79062 CD56EA 44401105 Ki = 35 nM T79062 CW3PC2 44401106 Ki = 34 nM T79062 C9WH7P 44401164 Ki = 6.2 nM T79062 C9CWX1 44401194 Ki = 57 nM T79062 CXT84G 44401243 Ki = 251 nM T79062 C1B4QL 44403095 Ki > 10000 nM T79062 C1YL7Z 44403098 Ki > 10000 nM T79062 CFV98A 44403101 Ki > 10000 nM T79062 C6OY9S 44403102 Ki > 10000 nM T79062 CH4SX6 44403105 Ki > 10000 nM T79062 C4LKC1 44404394 Ki = 342 nM T79062 C3EJ4G 44404396 Ki > 10000 nM T79062 CG87PW 44409290 Ki > 1000 nM T79062 CXO64D 44437860 Ki = 107 nM T79062 CWO35N 44437861 Ki > 5000 nM T79062 CKZF16 44439165 Ki = 39.81 nM T79062 CA4HZ3 44439167 Ki = 79.43 nM T79062 CRC2Y5 44439387 Ki = 800 nM T79062 C3ZT7I 44439388 Ki = 3500 nM T79062 CKU9N8 44439389 Ki = 7800 nM T79062 C20VDP 44439390 Ki = 45 nM T79062 C6RKA9 44439391 Ki = 36 nM T79062 CI9D7G 44439392 Ki = 20 nM T79062 CDE27X 44439393 Ki = 35 nM T79062 CIQW67 44439394 Ki = 170 nM T79062 CV93LJ 44439395 Ki = 46 nM T79062 CPX5Q2 44439396 Ki = 200 nM T79062 C2R0SX 44439397 Ki = 2200 nM T79062 C4CMV7 44439398 Ki = 400 nM T79062 C8YQ4P 44439399 Ki = 500 nM T79062 C6YA9O 44439400 Ki = 5300 nM T79062 C89ZPX 44439401 Ki = 25000 nM T79062 CE60JL 44439402 Ki = 2700 nM T79062 C65GSE 44439403 Ki = 1000 nM T79062 CKUG90 44439404 Ki = 100 nM T79062 CTYP87 44439405 Ki = 300 nM T79062 C3UBA6 44439406 Ki > 300000 nM T79062 C7HV8X 44439407 Ki = 36000 nM T79062 CD4T3S 44439408 Ki = 200 nM T79062 C07XPE 44439409 Ki = 100 nM T79062 CMU43Q 44439410 Ki = 3600 nM T79062 C2S6HQ 44448054 Ki = 55 nM T79062 C3Z7FI 44451927 IC50 = 119.95 nM T79062 CSD7R5 44451929 IC50 = 2197.86 nM T79062 C3MCY7 44451930 IC50 = 1300 nM T79062 C3R7BH 44451931 IC50 = 369.83 nM T79062 CRFN53 44451952 IC50 = 260.02 nM T79062 CZE3T1 44451953 IC50 = 199.99 nM T79062 CJTX92 44451954 IC50 = 190 nM T79062 CINR86 44451957 IC50 = 2500 nM T79062 CK4GN8 44451959 IC50 = 500 nM T79062 CL29TJ 44451979 IC50 = 620 nM T79062 C57SBC 44451980 IC50 = 16 nM T79062 CEST18 44451982 IC50 = 54.95 nM T79062 CV7EY2 44451984 IC50 = 500 nM T79062 C7L9DK 44451985 IC50 = 939.72 nM T79062 C15JOU 44451986 IC50 = 510 nM T79062 CM34IO 44452005 IC50 = 190 nM T79062 C39KGW 44452006 IC50 = 269.77 nM T79062 CRN4F8 44452007 IC50 = 49 nM T79062 CY43VF 44452008 IC50 = 42 nM T79062 CW80FP 44452010 IC50 = 680 nM T79062 C3L6IQ 44452037 IC50 = 28.97 nM T79062 CR4N5K 44452038 IC50 = 1199.5 nM T79062 CN6PT7 44452039 IC50 = 130.02 nM T79062 CB0CK5 44452040 IC50 = 769.13 nM T79062 C74KEA 44452041 IC50 = 769.13 nM T79062 CL2EH4 44452042 IC50 = 8994.98 nM T79062 CO1W6H 44452078 IC50 = 97 nM T79062 CT2VN0 44452080 IC50 = 199.99 nM T79062 CA91RH 44452081 IC50 = 419.76 nM T79062 C6U4YS 44452082 IC50 = 928.97 nM T79062 C7DAM2 44452084 IC50 > 10000 nM T79062 CP1E6V 44452114 IC50 = 1000 nM T79062 COR7N6 44452115 IC50 = 16 nM T79062 C65HFP 44452117 IC50 = 470 nM T79062 C8F7IQ 44452118 IC50 = 349.95 nM T79062 CN4YL1 44452139 IC50 = 230 nM T79062 CMP20V 44452141 IC50 = 680 nM T79062 CG1C6X 44452142 IC50 = 92 nM T79062 C7A9JI 44452143 IC50 = 26 nM T79062 C78UTQ 44452144 IC50 = 1999.86 nM T79062 CQR12V 44452145 IC50 > 10000 nM T79062 CF3H6V 44452166 IC50 = 19 nM T79062 C6SC1Q 44452167 IC50 = 91 nM T79062 C56JMP 44452169 IC50 > 10000 nM T79062 CQ5U1I 44452170 IC50 = 20.99 nM T79062 CX8OK7 44452171 IC50 = 45 nM T79062 CS72NU 44452193 IC50 = 54.95 nM T79062 C5ZF1H 44452195 IC50 = 97.95 nM T79062 CTAP34 44452196 IC50 = 199.99 nM T79062 CUG1W4 44452197 IC50 = 420 nM T79062 C5DNK1 44452199 IC50 = 710 nM T79062 CA3Y7E 44452217 IC50 = 48 nM T79062 CFUM27 44452219 IC50 = 1100 nM T79062 CAI2D5 44452221 IC50 = 690 nM T79062 CVAU93 44452222 IC50 = 460.26 nM T79062 CD0CQ5 44452223 IC50 = 1400 nM T79062 C6TN5J 44452224 IC50 = 79.98 nM T79062 CD8AJ3 44452243 IC50 = 79 nM T79062 C69RGK 44452244 IC50 > 10000 nM T79062 C1HEZ2 44452245 IC50 = 110 nM T79062 CJD35V 44452246 IC50 = 84.92 nM T79062 C23DZP 44452247 IC50 = 159.96 nM T79062 CLPR24 44452249 IC50 = 449.78 nM T79062 CJY18I 44452251 IC50 = 1099.01 nM T79062 C0G6ZC 44452273 IC50 = 28.97 nM T79062 CD5IY1 44452274 IC50 = 210 nM T79062 CX4DR9 44452275 IC50 = 590 nM T79062 CDLB90 44452276 IC50 = 1500 nM T79062 C6CT8L 44452277 IC50 = 109.9 nM T79062 CF5G0O 44452278 IC50 = 130 nM T79062 CKU52M 44452279 IC50 = 639.73 nM T79062 CP4M7B 44452298 IC50 = 590.2 nM T79062 CMBT16 44452301 IC50 = 939.72 nM T79062 CFH72P 44452302 IC50 = 2398.83 nM T79062 CRE1X3 44452305 IC50 = 95 nM T79062 C4B8JL 44452324 IC50 = 74 nM T79062 C0B3LC 44452327 IC50 = 75 nM T79062 C6SF7C 44452328 IC50 = 449.78 nM T79062 C6V1WM 44452329 IC50 = 400 nM T79062 CQX6I3 44452331 IC50 = 650 nM T79062 C8HI7Q 44452332 IC50 = 730 nM T79062 CCHJ25 44452357 IC50 = 349.95 nM T79062 C5U3VQ 44452359 IC50 = 920 nM T79062 C2QBM9 44452362 IC50 = 7294.58 nM T79062 CZL97F 44455426 Ki = 116 nM T79062 CYS7T4 44455943 Ki = 73 nM T79062 C6BFI0 44456033 Ki = 6 nM T79062 CG91RD 44456395 Ki = 12.4 nM T79062 C12XGE 44456400 Ki = 1148.15 nM T79062 C13YGE 44460471 Ki = 31 nM T79062 CHA10N 44460639 Ki = 166 nM T79062 C7KP0I 44460641 Ki = 125 nM T79062 C7HNZ8 44460642 Ki = 140 nM T79062 CVF5C3 44460669 Ki = 109 nM T79062 CQ2ID1 44460701 Ki = 139 nM T79062 C9DUW7 44460708 Ki = 10 nM T79062 C4YB7R 44460724 Ki = 109 nM T79062 CN6K9F 44460725 Ki = 23 nM T79062 CF6A9J 44460738 Ki = 34 nM T79062 C46ZGA 44460739 Ki = 158 nM T79062 CV0PU6 44460744 Ki = 182 nM T79062 C8P1MO 44460759 Ki = 288 nM T79062 CCL32X 44460808 Ki = 88 nM T79062 C9UW7I 44460917 Ki = 70 nM T79062 C3PK8D 44460918 Ki = 145 nM T79062 CSI97R 44460980 Ki = 70 nM T79062 CCX4G5 44461045 Ki = 17 nM T79062 C0RE6D 44461048 Ki = 9 nM T79062 CR6J9L 44461052 Ki = 163 nM T79062 C05GVU 44461064 Ki = 1573 nM T79062 C7G4MW 44461065 Ki = 10 nM T79062 CKE9C5 44461066 Ki = 16 nM T79062 C62CSN 44461069 Ki = 37 nM T79062 CK5SR9 44461070 Ki = 14 nM T79062 C4DL5C 44469677 IC50 > 10000 nM T79062 CEX18U 44517732 Ki = 195 nM T79062 C3I9NZ 44517733 Ki = 339 nM T79062 C3D4HR 44537940 Ki > 5000 nM T79062 CJ7U3K 44554227 Ki > 5000 nM T79062 CM0I1P 44554393 Ki > 5000 nM T79062 CNHA47 44554395 Ki > 5000 nM T79062 C0NGQ3 44575261 IC50 > 150000 nM T79062 CEGL62 44576914 IC50 > 10000 nM T79062 CW8OI7 44576978 IC50 = 103 nM T79062 C1S9PB 44576979 IC50 > 10000 nM T79062 C0TN9C 44576980 IC50 > 10000 nM T79062 C3R0YE 44577013 IC50 > 10000 nM T79062 CRCH48 44582675 Ki = 59 nM T79062 CEJ4R8 44582676 Ki = 210 nM T79062 CZGP86 44582677 Ki = 5170 nM T79062 C5QB4K 44582678 Ki = 498 nM T79062 C01RCI 44582705 Ki = 731 nM T79062 CXL25V 44582706 Ki > 10000 nM T79062 C8MR1X 44582707 Ki = 6241 nM T79062 C4IT1N 44582708 Ki = 2862 nM T79062 CB0S4Z 44592109 IC50 > 1000 nM T79062 C6KTM4 45028192 Ki = 9549.93 nM T79062 C0DLU3 45109862 IC50 = 456 nM T79062 CGB2Z0 45113400 Ki = 42 nM T79062 CV1F6P 45268647 Ki = 276 nM T79062 CGZ08S 45269494 Ki = 198 nM T79062 CR2QP3 45272864 Ki = 177 nM T79062 CX15SL 45272891 Ki = 140 nM T79062 CTD71C 45273807 Ki = 161 nM T79062 C13MCR 45273816 Ki = 150 nM T79062 CZ71RN 45278805 IC50 = 333 nM T79062 CZN6M7 45278882 IC50 = 408 nM T79062 C6NT3Q 45278883 IC50 = 493 nM T79062 CS5BA4 45278886 IC50 = 524 nM T79062 C0CHF4 45482789 IC50 > 10000 nM T79062 CH90CZ 45488126 Ki > 500 nM T79062 CG9U2R 45488130 Ki > 500 nM T79062 C7N4GP 45488138 Ki > 500 nM T79062 CH29KP 45488139 Ki > 500 nM T79062 CDAJ27 45488143 Ki > 500 nM T79062 CZYC01 45488151 Ki > 500 nM T79062 C8PH0Y 45488152 Ki > 500 nM T79062 CC2OU0 45488156 Ki > 500 nM T79062 CL4G8T 45488165 Ki > 500 nM T79062 C5NDO6 45488166 Ki > 500 nM T79062 C0GMN4 45488171 Ki > 500 nM T79062 C3ZAL4 45488172 Ki > 500 nM T79062 C3PYL9 45488174 Ki > 500 nM T79062 CFT7C5 45488175 Ki > 500 nM T79062 CX1A2N 45488179 Ki > 500 nM T79062 CA8I7U 45488180 Ki > 500 nM T79062 C01QBM 45488181 Ki > 500 nM T79062 COX47A 45488183 Ki > 500 nM T79062 C8ETO2 45488184 Ki > 500 nM T79062 C5FQ4S 46224879 Ki = 0.2089 nM T79062 CXUL12 46232559 IC50 = 195 nM T79062 CU2RG8 46232560 IC50 = 456 nM T79062 C9RQ8U 46232586 IC50 = 110 nM T79062 C2B3ZP 46232587 IC50 = 87 nM T79062 C3I8TO 46232588 IC50 = 567 nM T79062 COW9V6 46232589 IC50 = 172 nM T79062 CGV2J5 46232620 IC50 = 678 nM T79062 CWHG97 46232621 IC50 = 980 nM T79062 CUQW08 46232622 IC50 = 1236 nM T79062 C5REP7 46232623 IC50 = 500 nM T79062 C2QOW0 46232652 IC50 = 888 nM T79062 C9I7XS 46232653 IC50 = 1508 nM T79062 C5D0BH 46232654 IC50 = 419 nM T79062 C5PAL9 46232689 IC50 = 24 nM T79062 CT5C0M 46232690 IC50 = 160 nM T79062 CF53BL 46232691 IC50 = 442 nM T79062 CE1ID7 46232729 IC50 = 2296 nM T79062 CN0CO9 46232730 IC50 = 152 nM T79062 C0VXA5 46232731 IC50 = 334 nM T79062 C1C4OF 46232732 IC50 = 147 nM T79062 CMR8O9 46232770 IC50 = 500 nM T79062 CTY9H7 46232771 IC50 = 121 nM T79062 C5TBE8 46232772 IC50 = 316 nM T79062 COH03R 46232773 IC50 = 124 nM T79062 CZ2W7X 46232817 IC50 = 93 nM T79062 C0N4YP 46232818 IC50 = 117 nM T79062 CTJ89I 46232819 IC50 = 188 nM T79062 CS98DM 46232820 IC50 = 342 nM T79062 C8P3HD 46232858 IC50 = 49.6 nM T79062 CP04TS 46232859 IC50 = 749 nM T79062 C8W0IJ 46232860 IC50 = 12.3 nM T79062 CF5M2T 46232861 IC50 = 6.3 nM T79062 C21CHG 46232975 IC50 = 35.3 nM T79062 CO41KX 46232976 IC50 = 657 nM T79062 CIK94R 46232977 IC50 = 316 nM T79062 CB67ST 46232978 IC50 = 363 nM T79062 CRU0F7 46233014 IC50 = 526 nM T79062 C7W5TE 46233349 Ki = 2240 nM T79062 C10LFM 46233350 Ki = 128 nM T79062 C5NT9Y 46233351 Ki = 1614 nM T79062 C4T3HL 46233352 Ki = 26 nM T79062 C75PCA 46233382 Ki = 669 nM T79062 CV2FO0 46233383 Ki = 1429 nM T79062 C0QBP6 46233384 Ki > 10000 nM T79062 CL54OR 46233385 Ki > 10000 nM T79062 C3RH1V 46233448 Ki > 10000 nM T79062 C8USF7 46233449 Ki = 1485 nM T79062 C69MQR 46233450 Ki = 0.3 nM T79062 CNGP15 46233483 Ki > 10000 nM T79062 C42SVX 46700866 IC50 > 10000 nM T79062 CD0K6E 46700867 IC50 = 5600 nM T79062 C5TC2S 46830335 IC50 > 10000 nM T79062 C1K7FL 46830336 IC50 > 10000 nM T79062 C1N4KX 46842383 IC50 > 10000 nM T79062 CC62SX 46866711 IC50 = 2874 nM T79062 C03LTM 46869265 Ki = 220000 nM T79062 CB8GE1 46884818 IC50 > 10000 nM T79062 C4MQ0A 46884856 IC50 > 10000 nM T79062 CCNT25 46884898 IC50 > 10000 nM T79062 C3MSG2 46885027 IC50 > 10000 nM T79062 CB7XI0 46885213 IC50 > 10000 nM T79062 CY28OS 47556338 Ki = 888 nM T79062 C2LZJ0 49783209 Ki = 5702 nM T79062 C57SMG 49783415 Ki > 10000 nM T79062 C0TG6I 49783419 Ki > 10000 nM T79062 CR40BA 49836386 IC50 > 1000 nM T79062 C4R2YS 49850567 Ki = 199.53 nM T79062 C07JTU 49850570 Ki = 39.81 nM T79062 CK68QR 49850672 Ki = 25.12 nM T79062 CN5XR1 49850772 Ki = 125.89 nM T79062 CR4EZ0 49850870 Ki = 100 nM T79062 C5K4EC 49850872 Ki = 63.1 nM T79062 C8AW0R 49850874 Ki = 79.43 nM T79062 C6OQV2 49862237 Ki = 15 nM T79062 C9KIU1 49864289 IC50 = 3038 nM T79062 CHO9C0 49864292 IC50 = 2044 nM T79062 C90MTG 49864602 IC50 = 1006 nM T79062 C5BCS4 49864722 IC50 = 4425 nM T79062 CKZO79 49864723 IC50 = 3865 nM T79062 C74LZS 49864724 IC50 = 2059 nM T79062 C2RY0J 50878551 Ki = 16.98 nM T79062 C1W6TV 50898777 Ki > 10000 nM T79062 CXMZ73 50898778 Ki > 10000 nM T79062 CX48AD 51002362 Ki = 1956 nM T79062 C8TA1J 51003550 IC50 > 10000 nM T79062 CQ1UJ7 51003551 IC50 = 2007 nM T79062 CGMI37 51003586 IC50 > 10000 nM T79062 CE4KP1 51050257 Ki > 10000 nM T79062 CT3HG0 52952098 Ki > 100000 nM T79062 CDM75V 52952099 Ki = 14125.38 nM T79062 CR0ES9 52952100 Ki > 100000 nM T79062 CI9BF4 52952200 Ki = 91201.08 nM T79062 C31KMJ 52952201 Ki > 100000 nM T79062 CG4AW2 52952202 Ki = 15135.61 nM T79062 C3KZA4 52952203 Ki > 100000 nM T79062 C0MC9X 52952204 Ki > 100000 nM T79062 CT7A6Q 52952304 Ki > 100000 nM T79062 CR96JZ 52952305 Ki > 100000 nM T79062 CN70EP 52952306 Ki > 100000 nM T79062 CUI85Q 52952307 Ki = 9120.11 nM T79062 CJ94KO 52952308 Ki = 7244.36 nM T79062 C39XRU 52952309 Ki = 4786.3 nM T79062 C53DTC 52952419 Ki = 53703.18 nM T79062 COZ2U3 52952420 Ki = 12589.25 nM T79062 CG0L5I 52952421 Ki = 8709.64 nM T79062 CHC1S3 52952422 Ki = 263.03 nM T79062 CP37CU 52952423 Ki > 100000 nM T79062 C6LRO4 52952424 Ki = 27542.29 nM T79062 CMJ62D 53245590 Ki = 930 nM T79062 CGY45S 53248361 Ki = 161 nM T79062 CE9L8G 53248365 Ki = 50 nM T79062 C61DNP 53320009 IC50 = 143 nM T79062 C9ZDR5 53320010 IC50 = 620 nM T79062 CQLK01 53322638 IC50 > 10000 nM T79062 C32YWL 53324045 Ki = 326 nM T79062 CY28UP 53324535 Ki = 14 nM T79062 CRQF15 53325242 Ki = 969 nM T79062 C70WHV 53361627 Ki = 404 nM T79062 CU4B6N 53370045 Ki = 125 nM T79062 CKQ6A3 53376040 Ki = 739 nM T79062 C65CWD 53377240 Ki > 10000 nM T79062 CSGU70 53377324 Ki = 418 nM T79062 CG24AT 53381002 Ki = 1985 nM T79062 CMOZ61 53475319 Ki = 770 nM T79062 C0J8XZ 54598062 Ki = 26 nM T79062 C8SJ1Z 54758201 Ki = 107 nM T79062 C6G2AC 54758202 Ki = 72 nM T79062 CU6HI4 54758203 Ki = 96 nM T79062 C5KGQ3 54758204 Ki = 11 nM T79062 CS6PX1 54758293 Ki = 5.1 nM T79062 C6X3OI 54758294 Ki = 139 nM T79062 CS9L0P 54758295 Ki = 4 nM T79062 CUD7N0 54758296 Ki = 52 nM T79062 C1H2GP 54758297 Ki = 16 nM T79062 CG3UJ4 54758298 Ki = 6.7 nM T79062 C89NYL 54758391 Ki = 40 nM T79062 CTH56O 54758392 Ki = 13 nM T79062 CAZ5T6 54764323 Ki = 13 nM T79062 COZ82F 55479093 Ki = 155 nM T79062 CW89BT 56595402 Ki > 1000 nM T79062 C4C3XQ 56595529 Ki > 1000 nM T79062 C6W1RA 56649648 Ki = 132 nM T79062 C2SW7J 56649649 Ki = 77 nM T79062 CQTR49 56649650 Ki = 97 nM T79062 CH37LU 56663451 IC50 > 10000 nM T79062 CJKO58 56852956 Ki = 338.84 nM T79062 C1ZG7A 56933434 Ki = 0.6 nM T79062 CO0N2W 56943599 Ki = 6.7 nM T79062 C3DF5Z 56943600 Ki = 3.2 nM T79062 C19BDH 56943695 Ki = 10 nM T79062 CS7K3T 56943891 Ki = 6.9 nM T79062 CZ4L3S 56944082 Ki = 0.1 nM T79062 C5NI3K 56944086 Ki = 67 nM T79062 C37BYO 56944186 Ki = 5.1 nM T79062 C9UOZ6 56944189 Ki = 5.9 nM T79062 CH7V9J 56944190 Ki = 5.1 nM T79062 CE49MC 56944191 Ki = 4.4 nM T79062 CX2RP5 56944287 Ki = 15 nM T79062 CB0P9N 56944383 Ki = 1.6 nM T79062 CEQ7I3 56944384 Ki = 1.3 nM T79062 CHWI01 56944473 Ki = 13 nM T79062 C6Y4ZQ 56944564 Ki = 1.8 nM T79062 C3B0MZ 56944565 Ki = 1.6 nM T79062 CI4KW0 56944664 Ki = 1.1 nM T79062 C39YHD 56944665 Ki = 0.8 nM T79062 C1W3GL 56944666 Ki = 1.4 nM T79062 C7J4UT 56944667 Ki = 1.5 nM T79062 CZT80U 56944668 Ki = 0.8 nM T79062 CTW2F5 56944763 Ki = 0.4 nM T79062 C50WEX 56944764 Ki = 1.1 nM T79062 CX0ZW2 56944859 Ki = 1.3 nM T79062 C1ST9U 56944860 Ki = 140 nM T79062 CQKL90 56944861 Ki = 110 nM T79062 CS5J6Y 56944862 Ki = 90 nM T79062 CFLB40 56944863 Ki = 65 nM T79062 C53OTR 56944864 Ki = 70 nM T79062 C5T3RI 56944951 Ki = 18 nM T79062 CR6H7U 56944952 Ki = 10 nM T79062 C1Y2RP 56944953 Ki = 6 nM T79062 C1BH7I 56944954 Ki = 2 nM T79062 CTK9I8 56944955 Ki = 29 nM T79062 CCF1A5 56944956 Ki = 2 nM T79062 C2YVT8 56945042 Ki = 51 nM T79062 CNI2G3 56945043 Ki = 17 nM T79062 CF9V3Q 56945045 Ki = 33 nM T79062 CE4S5M 56945046 Ki = 38 nM T79062 C1TC7Q 56963799 Ki > 10000 nM T79062 C3ZG6J 57325520 Ki = 56 nM T79062 CDK7B0 57325521 Ki = 47 nM T79062 CR9MZ4 57384073 Ki = 16 nM T79062 CO7BG0 57390335 Ki = 335 nM T79062 CP05DB 57390336 Ki = 235 nM T79062 C1TH4R 57390337 Ki = 41 nM T79062 CATM39 57390694 Ki = 2060 nM T79062 C6S0IE 57390695 Ki = 2810 nM T79062 C83GWU 57391158 Ki = 604 nM T79062 CPE8N4 57391622 Ki = 68 nM T79062 CHG51U 57391624 Ki = 36 nM T79062 CIHJ73 57392107 Ki = 55 nM T79062 CY02VL 57392108 Ki = 38 nM T79062 C93QRW 57393876 Ki = 267 nM T79062 CUF40C 57393877 Ki = 334 nM T79062 CR7FB5 57393878 Ki = 1255 nM T79062 C7VFQ3 57394663 Ki = 50 nM T79062 CEW0O4 57395084 Ki = 88 nM T79062 CL96RC 57395086 Ki = 25 nM T79062 CSI7X2 57395597 Ki = 360 nM T79062 CJ15YT 57395598 Ki = 228 nM T79062 CK53EW 57395599 Ki = 37 nM T79062 C51GCK 57396417 Ki = 207 nM T79062 CZ2SJ8 57396419 Ki = 40 nM T79062 CZ8KA2 57396855 Ki = 381 nM T79062 CN7QE4 57396857 Ki = 334 nM T79062 C2Q6CJ 57397410 Ki = 132 nM T79062 CFQA13 57397411 Ki = 995 nM T79062 C7W5XA 57398619 Ki = 113 nM T79062 CFT56H 57399088 Ki = 3010 nM T79062 CGX5Q1 57399089 Ki = 79 nM T79062 CTF76G 57399090 Ki = 156 nM T79062 C0XFB2 57399091 Ki = 90 nM T79062 CI6ET3 57399092 Ki = 29 nM T79062 CMX4K5 57399093 Ki = 33 nM T79062 CJ41PW 57399432 Ki = 413 nM T79062 CAN0W7 57399866 Ki = 145 nM T79062 C9BG7C 57399868 Ki = 126 nM T79062 C5HGO2 57400281 Ki = 69 nM T79062 CT7Q3E 57400828 Ki = 506829 nM T79062 CFBP89 57400829 Ki = 1420 nM T79062 C3D1UP 57400830 Ki = 187 nM T79062 C5GPJ0 57401515 Ki = 210 nM T79062 CG8MF3 57401516 Ki = 353 nM T79062 CZX05B 57401706 Ki = 291 nM T79062 CN9J5I 57402588 Ki = 224 nM T79062 C92HON 57402951 Ki = 356 nM T79062 CX0B5M 57403525 Ki = 1042 nM T79062 C3A1YW 57403839 Ki = 310 nM T79062 CA10YX 57403841 Ki = 335 nM T79062 CYSV60 60165411 Ki = 337 nM T79062 CB9GC6 60165412 Ki = 62.6 nM T79062 CI5PM3 60165413 Ki = 107 nM T79062 C2Q5VD 60165416 Ki = 329 nM T79062 C9JL3F 60165418 Ki = 228.9 nM T79062 C31PEN 60165535 Ki = 35.6 nM T79062 CP60YF 60165537 Ki = 211 nM T79062 C85OTH 60165541 Ki = 425.8 nM T79062 CJO91V 60165543 Ki = 2467 nM T79062 CJDC53 60165545 Ki = 242 nM T79062 C3K5JN 60165681 Ki = 2917 nM T79062 C5RUP6 60167166 Ki = 790 nM T79062 CRH49P 60167309 Ki = 983 nM T79062 COHK72 60167451 Ki = 125.89 nM T79062 C30SVG 60167452 Ki = 512.86 nM T79062 CB4HT7 60195992 Ki = 109 nM T79062 C4Q6LO 60195993 Ki = 1.9 nM T79062 C04CRJ 60195994 Ki = 93 nM T79062 C4BG3H 60195995 Ki > 5000 nM T79062 C87FDE 60195996 Ki = 7 nM T79062 C6VWY1 60196073 Ki = 13 nM T79062 CM92UX 60196074 Ki = 23 nM T79062 C18AVJ 60196075 Ki = 80 nM T79062 CZN64D 60196076 Ki = 96 nM T79062 CIN29U 60196077 Ki = 7.1 nM T79062 C3LTC1 60196078 Ki = 8.2 nM T79062 C7WLN1 60196079 Ki = 6.9 nM T79062 C5N3SG 60196080 Ki = 1.4 nM T79062 C6AUO2 66800823 Ki = 25 nM T79062 C34ACQ 66800909 Ki = 2 nM T79062 CGT9E6 66800910 Ki = 6.3 nM T79062 C0QY7D 66800916 Ki = 4.6 nM T79062 CM58FG 66800926 Ki = 200 nM T79062 CQ43WD 66800934 Ki = 19 nM T79062 CK0I5J 66800939 Ki = 1.5 nM T79062 C0X2SF 66800942 Ki = 3.8 nM T79062 CN30YT 66800947 Ki = 9 nM T79062 CZ3MR6 66800959 Ki = 180 nM T79062 C92CMO 66800965 Ki = 91 nM T79062 CFPK92 66800991 Ki = 6.3 nM T79062 C13GMO 66801000 Ki = 13 nM T79062 CZ1TF9 66801018 Ki = 2.6 nM T79062 CBO9U3 66801028 Ki = 8.8 nM T79062 C3K8DC 66801052 Ki = 80 nM T79062 CA4DM3 66801062 Ki = 4.1 nM T79062 C2OUX9 66801107 Ki = 1.7 nM T79062 C4J5RZ 66801115 Ki = 54 nM T79062 C1H8BS 66801116 Ki = 41 nM T79062 C4JGC6 66801120 Ki = 18 nM T79062 CX2GN1 66801139 Ki = 0.9 nM T79062 C1NG8S 66801140 Ki = 5.3 nM T79062 CR7OW6 66801158 Ki = 0.8 nM T79062 CJU53X 66801160 Ki = 9.5 nM T79062 CH3BJ8 66801167 Ki = 0.5 nM T79062 C0AV5M 66801173 Ki = 9.9 nM T79062 C0V9EF 66801186 Ki = 3.2 nM T79062 CTHY41 66801210 Ki = 0.7 nM T79062 CSD67P 66801225 Ki = 4.3 nM T79062 C8J3YU 66801226 Ki = 9.9 nM T79062 CX45OZ 66801229 Ki = 1.5 nM T79062 C1S0EV 66801230 Ki = 3.2 nM T79062 C7S1KY 66801234 Ki = 0.9 nM T79062 CB53AV 66801246 Ki = 14 nM T79062 C3F1TZ 66801251 Ki = 34 nM T79062 CF8O9U 66801259 Ki = 57 nM T79062 C2Q9FS 66801263 Ki = 0.7 nM T79062 C7Y9VP 66801267 Ki = 2500 nM T79062 CED17M 66801271 Ki = 0.9 nM T79062 C41VYW 66801295 Ki = 14 nM T79062 C2FYL1 66801333 Ki = 180 nM T79062 CS75LK 66801335 Ki = 29 nM T79062 CR2N0J 66801344 Ki = 15 nM T79062 CDH7S9 66801346 Ki = 1.2 nM T79062 CGC4U6 66801354 Ki = 120 nM T79062 CY4FM5 66801379 Ki = 3.4 nM T79062 C3RX4C 66801425 Ki = 120 nM T79062 C7JD0I 66801429 Ki = 24 nM T79062 CN8OU1 66801430 Ki = 150 nM T79062 C93EGP 66801455 Ki = 4.1 nM T79062 COR1H8 66801528 Ki = 80 nM T79062 C1F3YV 66801537 Ki = 69 nM T79062 CIRW86 66801551 Ki = 0.2 nM T79062 C75WXP 66801561 Ki = 240 nM T79062 C8H5PD 66801565 Ki = 1.3 nM T79062 CT5SP8 66801605 Ki = 9 nM T79062 C8MH0I 66801613 Ki = 20 nM T79062 CC8JV6 66801624 Ki = 520 nM T79062 C3EI2F 66801625 Ki = 150 nM T79062 C49XBJ 66801673 Ki = 34 nM T79062 C0XG6B 66801701 Ki = 380 nM T79062 C42EBQ 66801837 Ki = 610 nM T79062 CW3AI2 66803474 Ki = 0.6 nM T79062 CPKH06 66803497 Ki = 12 nM T79062 CNJE57 66803500 Ki = 61 nM T79062 CN6FZ1 66803595 Ki = 1 nM T79062 C1LEH8 67268994 Ki = 30 nM T79062 CLA7F3 68281136 Ki = 23 nM T79062 C84MZH 68281137 Ki = 270 nM T79062 CR5KY1 71061607 Ki = 18 nM T79062 C72XPZ 71061659 Ki = 23.8 nM T79062 CKE2Y4 71061750 Ki = 26.1 nM T79062 CD1ET2 71061756 Ki = 23.5 nM T79062 C5KM2W 71061887 Ki = 11.2 nM T79062 C0D5SC 71062035 Ki = 15.2 nM T79062 CNQ65S 71062123 Ki = 12.7 nM T79062 CC43QK 71151588 Ki = 180 nM T79062 C3PUX5 71449549 Ki = 27 nM T79062 CN82LY 71449550 Ki = 311 nM T79062 C40DOC 71449627 Ki = 276 nM T79062 C8U6NR 71449628 Ki = 709 nM T79062 C7Y6LC 71449629 Ki = 7 nM T79062 C91SZN 71449641 Ki = 13 nM T79062 C2GCN7 71449642 Ki = 121 nM T79062 CQN93U 71449643 Ki = 7 nM T79062 CEJ3B4 71449644 Ki = 16 nM T79062 C5SAJ1 71449645 Ki = 28 nM T79062 C3XNC2 71450247 Ki = 1914 nM T79062 C9VZ8J 71450550 Ki = 3505 nM T79062 C2IXB6 71451344 Ki = 409 nM T79062 C7DCR4 71451345 Ki = 1672 nM T79062 CC6QP7 71451441 Ki = 161 nM T79062 CHT21G 71451454 Ki = 2222 nM T79062 C2QZL4 71451455 Ki = 78 nM T79062 CXI5Q2 71451456 Ki = 2375 nM T79062 CKJZ57 71451457 Ki = 29 nM T79062 C0F1HU 71451458 Ki = 15 nM T79062 CTZ24N 71451459 Ki = 6 nM T79062 C70JUP 71451460 Ki = 4 nM T79062 C4NDR3 71452382 Ki = 6259 nM T79062 C6ZWV2 71452383 Ki = 6873 nM T79062 CGO4M1 71453156 Ki = 815 nM T79062 C6EFP9 71453157 Ki = 391 nM T79062 CUK2P5 71453252 Ki = 12 nM T79062 CKI58Z 71453278 Ki = 21 nM T79062 C1QM8D 71453279 Ki = 58 nM T79062 C6O4KT 71453280 Ki = 9 nM T79062 CL49VI 71453281 Ki = 4 nM T79062 CGXT64 71453282 Ki = 12 nM T79062 CQ3XC8 71454898 Ki = 865 nM T79062 CWY38Z 71454899 Ki = 1188 nM T79062 CGO13Q 71454997 Ki = 20 nM T79062 C0K1JV 71454998 Ki = 46 nM T79062 C3JF1D 71454999 Ki = 0.3 nM T79062 C2QZ1N 71455000 Ki = 7 nM T79062 C6FE5D 71455001 Ki = 293 nM T79062 C4L0JN 71455002 Ki = 2 nM T79062 C8YH0J 71455083 Ki = 60 nM T79062 CAQF34 71455625 Ki = 1945 nM T79062 C6G2HC 71455894 Ki = 3647 nM T79062 C5O6LT 71456677 Ki = 1500 nM T79062 CLX0G4 71456770 Ki = 85 nM T79062 CE19SD 71456779 Ki = 97 nM T79062 CWR40I 71456780 Ki = 2195 nM T79062 CZUX67 71456781 Ki = 10 nM T79062 CZ17FC 71456782 Ki = 9 nM T79062 CKF09U 71456783 Ki = 16 nM T79062 CJKV72 71456784 Ki = 10 nM T79062 C7MNB5 71457264 Ki = 6371 nM T79062 CMJ1O9 71457409 Ki = 1018 nM T79062 CVI7S2 71457690 Ki = 2447 nM T79062 CG83QI 71458516 Ki = 334 nM T79062 CE6OC0 71458622 Ki = 1144 nM T79062 CZ8L0D 71458623 Ki = 17 nM T79062 CW79AY 71458624 Ki = 59 nM T79062 C2XV5L 71458625 Ki = 5 nM T79062 CUAC42 71458626 Ki = 5 nM T79062 C37EBC 71458647 Ki = 60 nM T79062 CM6OP1 71458648 Ki = 1362 nM T79062 CRGE05 71458649 Ki = 1438 nM T79062 CJN4S1 71458650 Ki = 14 nM T79062 CNT5J9 71458651 Ki = 10 nM T79062 C3NAM7 71458652 Ki = 11 nM T79062 CS83IF 71459269 Ki = 150 nM T79062 CK5T4P 71459604 Ki = 3601 nM T79062 CG0WO9 71459954 Ki = 329 nM T79062 CMW0T6 71460453 Ki = 93 nM T79062 C9W7CF 71460454 Ki = 3372 nM T79062 C09VSE 71460455 Ki = 1104 nM T79062 CBU8J7 71460456 Ki = 2224 nM T79062 CT17XB 71460468 Ki = 178 nM T79062 C63YLA 71461049 Ki = 3473 nM T79062 CJD96I 71461050 Ki = 384 nM T79062 CZ6G8V 71462064 Ki = 2674 nM T79062 CI0K3L 71462065 Ki = 415 nM T79062 CD0G8Q 71462066 Ki = 407 nM T79062 CK5JC7 71462067 Ki = 329 nM T79062 C42IZX 71462068 Ki = 873 nM T79062 CB30LT 71462154 Ki = 204 nM T79062 C7Y1XU 71462155 Ki = 427 nM T79062 CLS2A6 71462156 Ki = 1108 nM T79062 C7AX1Q 71462178 Ki = 41 nM T79062 C1CS0Z 71462179 Ki = 27 nM T79062 C4P3JU 71462776 Ki = 153 nM T79062 C3GUQ2 71462777 Ki > 10000 nM T79062 CT2ME3 71574204 Ki = 21 nM T79062 C3SXR5 71574206 Ki = 46 nM T79062 C2YRI9 71574208 Ki = 31 nM T79062 C62RWV 71574210 Ki = 12 nM T79062 CKC53S 71574212 Ki = 30 nM T79062 CNV42M 71574298 Ki = 41 nM T79062 C9PGQ1 71574300 Ki = 124 nM T79062 C2LXH5 71574302 Ki = 31 nM T79062 C2YPB8 71574304 Ki = 27 nM T79062 CK7GM0 71574306 Ki = 56 nM T79062 C7EQ2F 71602523 Ki = 537 nM T79062 C29INM 71602524 Ki > 10000 nM T79062 CK2C5Q 71602525 Ki > 10000 nM T79062 C1T0VP 71602526 Ki > 10000 nM T79062 C4BFZ0 71602581 Ki > 10000 nM T79062 C82MIC 71602582 Ki > 10000 nM T79062 C69MFB 71602583 Ki = 432 nM T79062 CG21CD 71602584 Ki > 10000 nM T79062 CQZ2O3 71602585 Ki > 10000 nM T79062 C9UE3T 71602586 Ki = 1850 nM T79062 C6B4VK 71602587 Ki = 1737.8 nM T79062 C9XWR8 71602639 Ki = 1200 nM T79062 CH91JF 71602640 Ki = 2754.23 nM T79062 C2KRC8 71602641 Ki > 10000 nM T79062 C1I9AS 71602642 Ki > 10000 nM T79062 CW3Z9S 71602643 Ki > 10000 nM T79062 C6MH1U 71602644 Ki > 10000 nM T79062 CKR10Z 71602687 Ki = 658 nM T79062 C3ZQ5D 71602688 Ki = 295.12 nM T79062 CJ89YE 71602689 Ki = 218.78 nM T79062 C6L3DJ 71602690 Ki = 199.53 nM T79062 C2ABS7 71602691 Ki = 309.03 nM T79062 CI86QM 71602692 Ki = 42.66 nM T79062 CC45VZ 71602739 Ki = 77 nM T79062 CXP3V8 71602740 Ki = 45.71 nM T79062 CVL36N 71678345 Ki = 1659.59 nM T79062 C0PF3I 71678857 Ki = 15 nM T79062 C0W2YA 71727193 Ki = 195 nM T79062 C79TLS 71727194 Ki = 16950 nM T79062 CFB10W 71727195 Ki = 13500 nM T79062 C6CIB5 71727196 Ki = 1145 nM T79062 C7Z3JS 71727308 Ki = 426 nM T79062 C3ATN5 72197484 IC50 = 1564 nM T79062 C20HSN 72197485 IC50 = 1059 nM T79062 CN8A5R 72197486 IC50 = 1003 nM T79062 CL3BF7 72197668 IC50 = 497 nM T79062 CUVJ59 72197845 Ki = 196 nM T79062 CIKU20 72198011 Ki = 345 nM T79062 COH95V 72198014 Ki = 589 nM T79062 C0WY2V 72198191 Ki = 1165 nM T79062 C7AOY4 72198754 IC50 = 62 nM T79062 C4M7KP 72198756 IC50 > 100 nM T79062 CWHF29 72547876 Ki = 43.7 nM T79062 CF47JC 72547878 Ki = 32.4 nM T79062 C12CIH 72548115 Ki = 26.1 nM T79062 C1UX8Q 72548117 Ki = 47.6 nM T79062 C4K1WO 72548349 Ki = 66.1 nM T79062 CWH6T3 72548703 IC50 = 0.39 nM T79062 C4T0SK 72549767 Ki = 186.5 nM T79062 CE4U6J 72549768 Ki = 64.5 nM T79062 C1QZ4F 72549986 Ki = 37.9 nM T79062 C17XNV 72549988 Ki = 43.7 nM T79062 CD7V6P 72550196 Ki = 36.5 nM T79062 C1SZ3K 72550200 Ki = 34.7 nM T79062 C62EFS 72550423 Ki = 34.7 nM T79062 CK0F1L 72550641 Ki = 46.6 nM T79062 C8Z0NM 72550642 Ki = 8.69 nM T79062 CL6W2Q 72550645 Ki = 15.9 nM T79062 CUH4Z3 72550864 Ki = 405.3 nM T79062 C9J4QU 72550865 Ki = 25.9 nM T79062 C8A3DU 72551082 Ki = 31.4 nM T79062 C78LYM 72698087 Ki > 10000 nM T79062 C63HPK 72698088 Ki > 10000 nM T79062 C7W4RH 72734860 Ki = 12.4 nM T79062 C8UCZ5 72734861 Ki > 100 nM T79062 CZ6SQ7 72734863 Ki = 42 nM T79062 C8JT6B 72734864 Ki = 144 nM T79062 CW4IB9 72734866 Ki > 1000 nM T79062 CY0AE3 72735038 Ki = 239 nM T79062 CAZ84Y 72735039 Ki > 1000 nM T79062 C0MT4E 72735040 Ki > 1000 nM T79062 C0CK8H 72735041 Ki > 100 nM T79062 CC6Q5R 72771081 Ki < 100 nM T79062 CC65OA 73213195 Ki = 199.53 nM T79062 CW83DK 73213196 Ki = 194.98 nM T79062 CCV91B 73346042 Ki = 17.2 nM T79062 CXM8O2 73347306 IC50 = 3100 nM T79062 C9X8GY 73347307 IC50 > 1000 nM T79062 C4ZM8R 73347582 Ki = 9.7 nM T79062 C6BS5L 73349361 Ki = 4423 nM T79062 CL38VQ 73351112 Ki > 1000 nM T79062 CC8I7X 73351903 IC50 = 1800 nM T79062 CG4M8P 73351905 IC50 = 3700 nM T79062 CAR7Z5 73354882 IC50 = 480 nM T79062 CET52A 73356443 IC50 = 690 nM T79062 CUB97Z 74538690 Ki = 35 nM T79062 C2E7QW 75201901 Ki = 7800 nM T79062 C8IDL3 75306277 Ki = 79.43 nM T79062 CX17RZ 76280896 Ki = 71 nM T79062 C45OSP 76284193 Ki = 53 nM T79062 C0CRJ1 76284452 Ki = 34.5 nM T79062 CS17IJ 76284453 Ki = 12.8 nM T79062 CH82JU 76284455 Ki = 45.2 nM T79062 CRO7Q9 76284721 Ki = 15.9 nM T79062 C4BIC2 76284724 Ki = 3.82 nM T79062 C0EKY7 76284725 Ki = 66.7 nM T79062 C3GXV8 76310809 Ki = 1200 nM T79062 C19EPD 76310810 Ki = 48 nM T79062 CK2X7A 76310812 Ki = 92 nM T79062 CXJG08 76314094 Ki > 1000 nM T79062 CN7GD5 76314435 Ki = 317 nM T79062 CLO9M1 76314437 Ki = 1920 nM T79062 CD8A5H 76318011 Ki = 6.9 nM T79062 C1Y9SX 76318012 Ki = 20 nM T79062 CEHK31 76321734 Ki = 4.5 nM T79062 C5F1XU 76321735 Ki = 4.5 nM T79062 CC8TR0 76321736 Ki = 70 nM T79062 C94VNF 76324975 Ki = 64.2 nM T79062 C18OSZ 76325346 Ki = 17 nM T79062 C62CZO 76325348 Ki = 27 nM T79062 COGC62 76325350 Ki = 18 nM T79062 C1Q5NC 76325352 Ki = 8.7 nM T79062 CZ6P1E 76328545 Ki > 1000 nM T79062 C0OI2M 76328889 Ki = 283 nM T79062 C51CME 76328891 Ki = 41 nM T79062 CBFE85 76328893 Ki = 62 nM T79062 C5WG9E 76328895 Ki = 60 nM T79062 C6OV4J 76328897 Ki = 65 nM T79062 CL83OY 76332574 Ki = 649 nM T79062 CN3QO1 76332576 Ki = 15 nM T79062 CDBS57 76332578 Ki = 34 nM T79062 C97OVP 76332580 Ki = 4440 nM T79062 C1LT6C 76332582 Ki = 3907 nM T79062 CP0D6T 76332584 Ki = 94 nM T79062 CW3AK0 76335863 Ki = 33.4 nM T79062 CYT34W 76336176 Ki = 33 nM T79062 C9XFL1 76336178 Ki = 18 nM T79062 C0GD2B 76336180 Ki = 20 nM T79062 CV90GC 76336182 Ki = 189 nM T79062 C51CXD 76336183 Ki = 54 nM T79062 CMG58X 76336185 Ki = 10.8 nM T79062 C28RIZ 76518514 Ki = 472 nM T79062 C9S0XK 86288947 Ki = 3 nM T79062 CEPC94 86288948 Ki = 3 nM T79062 CHE2U4 90178632 Ki = 16 nM T79062 CFDW68 90644074 Ki = 10 nM T79062 C0T8RE 90644075 Ki = 380 nM T79062 C2KE9G 90644076 Ki = 94 nM T79062 C1SOF5 90644077 Ki = 150 nM T79062 CIE9Z2 90644078 Ki = 900 nM T79062 C37CYS 90654670 Ki = 101 nM T79062 C0IQ5R 90654671 Ki = 51 nM T79062 CVG2C1 90654672 Ki = 78 nM T79062 CU0ON1 90654673 Ki = 111 nM T79062 CJR3Y9 90654674 Ki = 148 nM T79062 CO1H4U 90654675 Ki = 551 nM T79062 CAY64Z 90654676 Ki = 302 nM T79062 CH0R8B 90654677 Ki = 579 nM T79062 CRFB56 90654678 Ki = 476 nM T79062 CPR21O 90654679 Ki = 393 nM T79062 C6YLV3 90654680 Ki = 725 nM T79062 CGUY51 90654681 Ki = 223 nM T79062 CK8X4O 90654682 Ki = 295 nM T79062 CH8UQ9 90654683 Ki = 107 nM T79062 CTQ23Z 90654684 Ki = 95 nM T79062 C9Q2JW 90654685 Ki = 1196 nM T79062 C98TJR 90654686 Ki = 18 nM T79062 CG3OI7 90654687 Ki = 22 nM T79062 CKTV83 90654688 Ki = 28 nM T79062 CVK85U 90654689 Ki = 163 nM T79062 CLG75D 90654690 Ki = 153 nM T79062 C7T9HW 90654691 Ki = 495 nM T79062 C92BZL 90654692 Ki = 567 nM T79062 C6CD9R 90654693 Ki = 634 nM T79062 C6H9NV 90654694 Ki = 1199 nM T79062 CR74SD 90654695 Ki = 4151 nM T79062 C7VM4O 90654696 Ki = 1865 nM T79062 CGFU53 90654697 Ki = 1312 nM T79062 C7BEZ8 90654698 Ki = 3134 nM T79062 CZ3IM2 90654699 Ki = 478 nM T79062 C8TMK5 90654700 Ki = 1188 nM T79062 C7GK3C 90654701 Ki = 113 nM T79062 CN8BO1 90654702 Ki = 179 nM T79062 CHIW63 90654703 Ki = 108 nM T79062 C1SAW2 90654704 Ki = 50 nM T79062 CJG31T 90654831 Ki = 95 nM T79062 CMU45O 90654832 Ki = 77 nM T79062 C3C4BW 90654834 Ki = 157 nM T79062 C8QWR3 90654835 Ki = 34 nM T79062 C6ZR9L 90654837 Ki = 70 nM T79062 C0AC7R 90654839 Ki = 72 nM T79062 CKLG40 90654841 Ki = 122 nM T79062 C5JS8D 90654843 Ki = 135 nM T79062 C4VHZ6 90654845 Ki = 45 nM T79062 CG78PS 90654847 Ki = 172 nM T79062 CL39WP 90654849 Ki = 123 nM T79062 C0TVQ9 90654851 Ki = 46 nM T79062 C4I1CU 90654853 Ki = 31 nM T79062 CZ28YC 90654855 Ki = 78 nM T79062 CRO83N 90654857 Ki = 456 nM T79062 C72RKV 90656669 Ki = 20.8 nM T79062 CJ8H1R 90656670 Ki = 92.5 nM T79062 CSF25H 90656671 Ki = 90.1 nM T79062 CGD60Y 90656672 Ki = 12.1 nM T79062 C4H1SB 90656673 Ki = 81.4 nM T79062 CID83U 90656674 Ki = 161.4 nM T79062 C0VDH3 90656675 Ki = 252.1 nM T79062 CC1L7T 90656676 Ki = 57 nM T79062 CCQU80 90656678 Ki = 84.8 nM T79062 CNSW31 90656679 Ki = 161.2 nM T79062 CITS52 90656680 Ki = 179.2 nM T79062 C3GA5B 90656681 Ki = 111.7 nM T79062 C9SX5R 90656682 Ki = 10.1 nM T79062 CGEF35 90656683 Ki = 2.9 nM T79062 C76OIR 90656684 Ki = 434.2 nM T79062 CH9F4Q 90656685 Ki = 20 nM T79062 C8NB7D 90656686 Ki = 161.1 nM T79062 C13YLN 90656687 Ki = 39.6 nM T79062 CU82QN 90656688 Ki = 63.3 nM T79062 CNB76X 90656689 Ki = 77.9 nM T79062 CPQ46T 90656690 Ki = 108.8 nM T79062 C6QO1P 90656691 Ki = 13.2 nM T79062 C6TF2G 90656692 Ki = 8.1 nM T79062 CGP76X 90656694 Ki = 30 nM T79062 C3O2KS 90656695 Ki = 16.7 nM T79062 CYLZ26 90656696 Ki = 12 nM T79062 C9RH6O 90656697 Ki = 226 nM T79062 C5MP1J 90656699 Ki = 39.4 nM T79062 C5L9IQ 90656701 Ki = 95.6 nM T79062 C6NG4Q 90656703 Ki = 191 nM T79062 C63JKH 90656705 Ki = 137.5 nM T79062 C7NV3E 90656707 Ki = 242.1 nM T79062 CK6UO3 90656708 Ki = 310 nM T79062 C6N5CS 90656709 Ki = 40 nM T79062 CX49HI 90656710 Ki = 3.1 nM T79062 CRX47O 90656711 Ki = 11.6 nM T79062 CTHD25 90656712 Ki = 6.6 nM T79062 CID86Z 90656713 Ki = 12.8 nM T79062 C5Q8PH 90656714 Ki = 63.1 nM T79062 CS9E1R 90656715 Ki = 332 nM T79062 CCOV98 90664359 Ki = 10490 nM T79062 CA8B0H 90664441 Ki = 328 nM T79062 CP48OR 90664581 Ki = 612 nM T79062 C4MUI2 90664601 IC50 = 11 nM T79062 CXD5Q9 90664621 Ki = 17420 nM T79062 CP2MK1 90664692 Ki = 5800 nM T79062 CO9H3P 90664694 Ki = 153 nM T79062 CE6D5M 90664808 Ki = 296 nM T79062 CT7Z1V 90664944 Ki = 184 nM T79062 CHT7D5 90664962 IC50 = 6.8 nM T79062 CQCE48 90665063 Ki = 276 nM T79062 C4EQ5K 90665189 Ki = 484 nM T79062 C0J5YH 91864602 Ki = 3.548 nM T79062 CDWS84 91937906 Ki = 157 nM T79062 CEN10X 92042876 Ki = 5.2 nM T79062 CW6XB3 92042877 Ki = 15 nM T79062 CUQ6V0 92042918 Ki < 1000 nM T79062 CS62HU 101747513 Ki = 5.6 nM T79062 C4DG3V 102364516 Ki = 0.7 nM T79062 C4WDR8 109018769 Ki = 4.34 nM T79062 CD76TH 109026949 Ki = 52 nM T79062 C3DMI5 109026956 Ki = 29.5 nM T79062 C2G0WH 109026957 Ki = 23.5 nM T79062 CYB18Z 109027017 Ki = 26.2 nM T79062 C0M3CD 118051679 Ki = 42 nM T79062 CEMZ15 118464420 Ki = 401 nM T79062 CV2L6O 118464425 Ki = 516 nM T79062 CFNG86 118464427 Ki = 427 nM T79062 CMSN80 118626035 Ki = 19 nM T79062 CT3AI0 118626042 Ki = 75 nM T79062 CKNJ72 118626045 Ki = 23 nM T79062 CGB42Y 118626088 Ki = 66 nM T79062 C0XJT5 118626089 Ki = 19 nM T79062 CIE4C7 118626101 Ki = 4 nM T79062 C1NYS5 118626120 Ki = 142 nM T79062 CPG04R 118626121 Ki = 3 nM T79062 C3S5LJ 118626129 Ki = 1 nM T79062 CY3F0N 118626140 Ki = 97 nM T79062 CE07IQ 118626142 Ki = 4 nM T79062 C72OZY 118626161 Ki = 1 nM T79062 CY3E7S 118626169 Ki = 52 nM T79062 CHRB75 118626208 Ki = 349 nM T79062 CSN13R 118706278 Ki = 41 nM T79062 CIG56H 118706280 Ki > 1000 nM T79062 CF5ZR8 118706282 Ki = 14 nM T79062 CD1XJ5 118706284 Ki = 29 nM T79062 CL4Y6K 118706285 Ki = 4.1 nM T79062 C32KAS 118706287 Ki = 160 nM T79062 C1K5NC 118706290 Ki = 87 nM T79062 CGA0O1 118706292 Ki = 41 nM T79062 CA0V9U 118706294 Ki = 50 nM T79062 C0NSU5 118706296 Ki = 180 nM T79062 CFOE72 118706299 Ki = 57 nM T79062 C1DI6Y 118706301 Ki = 4.1 nM T79062 CH3Z8R 118706732 Ki = 4 nM T79062 CN4I3G 118706734 Ki = 2.3 nM T79062 C2Q4OP 118709739 Ki = 28 nM T79062 CZ68PL 118709740 Ki = 24 nM T79062 CSB25E 118709750 Ki = 917 nM T79062 CD4S9R 118709751 Ki = 882 nM T79062 CBP52O 118709752 Ki = 36 nM T79062 CO72SF 118709753 Ki = 29 nM T79062 CJQR81 118709754 Ki = 41 nM T79062 CPW1D5 118709755 Ki = 62 nM T79062 C1TMO7 118709756 Ki = 2.7 nM T79062 CZ9H5G 118711997 Ki = 22 nM T79062 CH9W0A 118713587 Ki = 36.48 nM T79062 CK43CN 118713588 Ki = 7.77 nM T79062 CL0TS7 118713589 Ki = 0.99 nM T79062 C4RD6F 118713590 Ki = 41.93 nM T79062 CIG13W 118713591 Ki = 46.83 nM T79062 CX5L1H 118713592 Ki = 1.72 nM T79062 CDWY84 118713593 Ki = 2.84 nM T79062 CO5S1I 118713594 Ki = 57.39 nM T79062 CI91US 118713595 Ki = 20 nM T79062 CW92LT 118713679 Ki = 5.9 nM T79062 C8P9YT 118713680 Ki = 5.16 nM T79062 CZ1K5R 118713681 Ki = 14.1 nM T79062 CH7ZE8 118713682 Ki = 2.96 nM T79062 CKX78H 118713683 Ki = 11.68 nM T79062 C5LSA7 118713684 Ki = 2.9 nM T79062 CPAI54 118713685 Ki = 45.57 nM T79062 C6U2LR 118713686 Ki = 7.58 nM T79062 CYA6E4 118713687 Ki = 7.73 nM T79062 CZ9UL2 118713688 Ki = 8.49 nM T79062 CI5XK3 118717210 Ki = 1.2 nM T79062 CYJQ09 118717212 Ki > 100 nM T79062 C1TSR8 118717214 Ki = 1.4 nM T79062 C7YX3Q 118717215 Ki = 0.6 nM T79062 CEZ4M6 118717216 Ki = 0.76 nM T79062 C1E4GL 118717218 Ki = 4.9 nM T79062 CSJ6N3 118717219 Ki = 1.8 nM T79062 C5LFW4 118717221 Ki = 1.7 nM T79062 CZ65GI 118717222 Ki = 1.3 nM T79062 C1F9ZM 118724639 Ki = 346 nM T79062 CGA86P 118728506 Ki = 168 nM T79062 C9PGE7 118728507 Ki = 357 nM T79062 CR4GE1 118728510 Ki = 30.1 nM T79062 C14LZH 118728511 Ki = 147 nM T79062 C14RAC 118728513 Ki = 68.4 nM T79062 CQK04P 118728514 Ki = 1464 nM T79062 CK9CG4 118728521 Ki = 307 nM T79062 C1N9JU 118728522 Ki = 1082 nM T79062 C1UZ8G 118728523 Ki = 35.8 nM T79062 CPCE84 118728524 Ki = 12.9 nM T79062 CBN06J 118728525 Ki = 6.88 nM T79062 CF3QE0 118728526 Ki = 143 nM T79062 CJG4Q1 118728527 Ki = 1650 nM T79062 C4NFW1 118728528 Ki = 88.5 nM T79062 CO8LF9 118728529 Ki = 213 nM T79062 CCN7R8 118728530 Ki = 2.99 nM T79062 C5O2NU 118729733 Ki = 17890 nM T79062 CB3Y2W 118731347 Ki = 116 nM T79062 CWZF06 118731348 Ki = 18 nM T79062 CA3O1H 118731349 Ki = 30 nM T79062 CU8P4W 118731350 Ki = 43 nM T79062 C8GKX6 118731351 Ki = 6 nM T79062 C2J4VC 118731352 Ki = 10 nM T79062 CF7NH5 118731353 Ki = 11 nM T79062 CQ8F6C 118731354 Ki = 77 nM T79062 CR9J0O 118731355 Ki = 135 nM T79062 CU12XM 118731356 Ki = 5 nM T79062 C4CEV7 118731357 Ki = 16 nM T79062 CU6T2D 118731358 Ki = 15 nM T79062 C95WKJ 118731359 Ki = 30 nM T79062 C20QAO 118731360 Ki = 40 nM T79062 CT6J8V 118731361 Ki = 22 nM T79062 C7QVJ4 118731362 Ki = 10 nM T79062 CA2X3O 118731363 Ki = 9 nM T79062 C4DV8I 118731364 Ki = 9 nM T79062 CHVY82 118731365 Ki = 12 nM T79062 CM5FG1 118731366 Ki = 9 nM T79062 C75OXS 118736395 Ki = 473 nM T79062 C74FCM 118736396 Ki = 61 nM T79062 C3F8PA 118736397 Ki > 1000 nM T79062 CHI8V7 121209051 Ki = 322 nM T79062 C7W3EY 122178698 Ki = 69 nM T79062 CF8P1H 122178699 Ki = 15 nM T79062 C48MFR 122178700 Ki = 24 nM T79062 CZ72QS 122178701 Ki = 58 nM T79062 C4VY8A 122178702 Ki = 52 nM T79062 C2KF4Z 122178703 Ki = 28 nM T79062 CX6MJ2 122178704 Ki = 34 nM T79062 CA53KF 122178705 Ki = 24 nM T79062 C8XD3F 122178706 Ki = 38 nM T79062 CTRC59 122178707 Ki = 22 nM T79062 C5QV8D 122178708 Ki = 50 nM T79062 C84UED 122178709 Ki = 20 nM T79062 CV96JK 122178710 Ki = 23 nM T79062 CM89KS 122178711 Ki = 54 nM T79062 C7ODW3 122195524 Ki > 900 nM T79062 CBHT01 122377930 Ki = 9 nM T79062 CG63UZ 122483217 Ki = 281.84 nM T79062 C3RX0B 122483224 Ki = 2336 nM T79062 C57RDF 122483225 Ki = 1071.52 nM T79062 C7PL6Q 122483228 Ki = 588.84 nM T79062 CW32JF 122483234 Ki = 251.19 nM T79062 C7K4ZC 122483237 Ki = 1307 nM T79062 C4JFD9 122483243 Ki = 549.54 nM T79062 CZ27HR 122483245 Ki = 151.36 nM T79062 C89LZM 122483248 Ki = 794.33 nM T79062 CM8HO9 122483250 Ki = 616 nM T79062 CB9U5S 122483253 Ki = 1398 nM T79062 CL4J6V 122483257 Ki = 831.76 nM T79062 C86NGA 122483259 Ki = 309.03 nM T79062 C24ZNM 122483261 Ki = 512.86 nM T79062 C2SWA8 122483263 Ki = 1047.13 nM T79062 C1G4YN 122483273 Ki = 676.08 nM T79062 CLW53P 122483274 Ki = 86 nM T79062 C8IZ9U 122483279 Ki = 949 nM T79062 CO63ET 122483280 Ki = 30 nM T79062 CJ84WM 122483287 Ki = 125.89 nM T79062 C5IV3P 122483288 Ki = 1281 nM T79062 C0Y7NI 122483295 Ki = 1905.46 nM T79062 CKSQ23 122483303 Ki = 2137.96 nM T79062 C4QM2E 124247485 Ki = 104 nM T79062 CLWM12 126720394 Ki = 8748 nM T79062 C8Q1JB 126720403 Ki = 11920 nM T79062 C1U3SZ 126720425 Ki = 7139 nM T79062 C5G8FD 126720440 Ki = 12340 nM T79062 CD50YM 127024949 Ki = 20 nM T79062 C4GF2D 127024950 Ki = 40 nM T79062 CJ76IB 127024951 Ki = 4 nM T79062 CKB42V 127025036 Ki = 157 nM T79062 CIHZ54 127025242 Ki = 2 nM T79062 CCY7P3 127025243 Ki = 1 nM T79062 CNJ4Z1 127025244 Ki = 9 nM T79062 CTBN56 127026052 Ki = 398.11 nM T79062 C26NMB 127026071 Ki = 74 nM T79062 C1YD7M 127026119 Ki = 344 nM T79062 CUO7Y8 127026120 Ki = 27 nM T79062 CDU21O 127026131 Ki = 4 nM T79062 C9HDP8 127026132 Ki = 70 nM T79062 CTYP30 127026133 Ki = 14 nM T79062 C19BOM 127026141 Ki = 50 nM T79062 CZFB49 127026142 Ki = 285 nM T79062 C2FT3B 127026143 Ki = 197 nM T79062 CP4J5H 127026144 Ki = 264 nM T79062 C6BIU4 127026145 Ki = 201 nM T79062 C1FA2U 127026146 Ki = 198 nM T79062 CE43NR 127026147 Ki = 39 nM T79062 CDAP16 127026434 Ki = 1918 nM T79062 C2XO3L 127026443 Ki = 54 nM T79062 C80QHX 127026444 Ki = 17 nM T79062 CBF64M 127026450 Ki = 12 nM T79062 CO1FB4 127026451 Ki = 14 nM T79062 CC13RA 127026452 Ki = 20 nM T79062 CBE56W 127026514 Ki = 74 nM T79062 C0SZI4 127026515 Ki = 38 nM T79062 CX6EI2 127026750 Ki = 19 nM T79062 CEG15O 127026751 Ki = 16 nM T79062 C1J4QY 127026752 Ki = 14 nM T79062 C0WB2U 127026753 Ki = 7 nM T79062 C62UMZ 127027143 Ki = 602.56 nM T79062 C4L0KU 127027144 Ki = 363.08 nM T79062 C0UOJ6 127027386 Ki = 72 nM T79062 C9IH1A 127027387 Ki = 26 nM T79062 C0TC7E 127027388 Ki = 53 nM T79062 CZ4W6I 127027389 Ki = 168 nM T79062 C4YR7A 127027390 Ki = 162 nM T79062 C3FA0I 127027391 Ki = 319 nM T79062 CC71UE 127027715 Ki = 292 nM T79062 CY2TW9 127028152 Ki = 223 nM T79062 CAZJ04 127028153 Ki = 89 nM T79062 CR48GO 127028154 Ki = 234 nM T79062 C8MC1I 127028408 Ki = 1023.29 nM T79062 CD8H7W 127028471 Ki = 47 nM T79062 C4EAY5 127028472 Ki = 10 nM T79062 CUS8R9 127028473 Ki = 14 nM T79062 CA10BY 127028634 Ki = 163 nM T79062 CZ26YR 127028797 Ki = 17 nM T79062 CI2R1N 127028798 Ki = 56 nM T79062 CS8GJ5 127028799 Ki = 837 nM T79062 CU0WQ3 127029375 Ki = 908 nM T79062 CS1GX5 127029649 Ki = 1190 nM T79062 C9N3BE 127029650 Ki = 141 nM T79062 CQFS48 127029651 Ki = 177 nM T79062 C7F3YE 127029652 Ki = 79 nM T79062 CZ61LK 127034966 EC50 > 5011.87 nM T79062 CA0SN5 127034967 EC50 > 5011.87 nM T79062 CQ0ZT9 127035062 Ki = 700 nM T79062 CU49VE 127036186 Ki = 154.88 nM T79062 CG06BD 127036932 Ki = 74.13 nM T79062 CVW71O 127036953 Ki = 48.98 nM T79062 C7N5DF 127037679 Ki = 8 nM T79062 CD13VY 127037680 Ki = 24 nM T79062 CTE43C 127037681 Ki = 19 nM T79062 C0LGK6 127037682 Ki = 21 nM T79062 C2XBE8 127037921 Ki = 49 nM T79062 CX0CN4 127037922 Ki = 18 nM T79062 CDAE15 127038033 Ki = 7 nM T79062 CFA6Q8 127038034 Ki = 44 nM T79062 CERL85 127038035 Ki = 49 nM T79062 C8TC9G 127038281 Ki = 10 nM T79062 CPK2Z7 127038282 Ki = 84 nM T79062 CYJ2D5 127039593 Ki = 56 nM T79062 CQED51 127039753 Ki = 7 nM T79062 CL4E2K 127039754 Ki = 36 nM T79062 CES26L 127039755 Ki = 6 nM T79062 CQ36LP 127039756 Ki = 7 nM T79062 C7KA2C 127040443 Ki = 200 nM T79062 CKBZ01 127040444 Ki = 42 nM T79062 CFAB12 127040760 Ki = 8 nM T79062 CWQ47G 127040761 Ki = 28 nM T79062 C8D4AV 127040908 Ki = 13 nM T79062 CE12AY 127041106 Ki = 19 nM T79062 C71LGS 127041107 Ki = 9 nM T79062 C6RI9V 127041108 Ki = 8 nM T79062 C15BGV 127041244 Ki = 9 nM T79062 CU0J4S 127041258 Ki = 18 nM T79062 C20MZH 127041259 Ki = 10 nM T79062 CP16CZ 127041260 Ki = 70 nM T79062 CZT53S 127041261 Ki = 68 nM T79062 C0FJP2 127041563 Ki = 58 nM T79062 CUC3F9 127041564 Ki = 58 nM T79062 COG9D2 127041874 Ki = 100 nM T79062 CS4WH1 127042184 Ki = 5 nM T79062 C13AIN 127042185 Ki = 7 nM T79062 CR59TP 127042539 Ki = 56 nM T79062 C54IZC 127042540 Ki = 28 nM T79062 C8G1HF 127042841 Ki = 53 nM T79062 CC7BU0 127049059 Ki = 1511 nM T79062 C42FHY 127049060 Ki > 10000 nM T79062 CF2QY9 127049061 Ki = 286 nM T79062 CX53AC 127050632 Ki = 1584.89 nM T79062 CTL0S1 127051516 Ki = 626 nM T79062 CTL8J1 127051843 Ki = 755 nM T79062 CF6V9Q 127051844 Ki = 12 nM T79062 C8TNB1 127051845 Ki = 16.98 nM T79062 C5ONG1 127051864 Ki = 1000 nM T79062 CVQW26 127051865 Ki = 79.43 nM T79062 CRF85X 127052458 Ki = 10 nM T79062 CCY71I 127052465 Ki = 330 nM T79062 C2E9VX 127052467 Ki = 51.29 nM T79062 CPO4C3 127052468 Ki = 86 nM T79062 CSQ2N8 127052486 Ki = 313 nM T79062 C4YJ8H 127052487 Ki = 111 nM T79062 CT9RS4 127052488 Ki = 778 nM T79062 CLU7C1 127052757 Ki = 26.92 nM T79062 C95KYT 127052758 Ki = 100 nM T79062 CYNR02 127052759 Ki = 48.98 nM T79062 C14YJU 127052778 Ki = 501.19 nM T79062 C1JAS7 127052779 Ki = 189 nM T79062 C7MQK8 127053042 Ki = 22.5 nM T79062 C50GOC 130442480 Ki = 8100 nM T79062 CM04RF 130442572 Ki = 4100 nM T79062 C4LJ2Y 132503215 Ki = 55 nM T79062 CM8B1L 132525569 Ki = 7.1 nM T79062 CU5L0K 132525570 Ki = 1.6 nM T79062 CA10SQ 132547275 Ki = 44.8 nM T79062 C6E1GN 132547276 Ki = 23.5 nM T79062 C6VTW3 132547277 Ki = 35.1 nM T79062 CI70OP 132547278 Ki = 45.1 nM T79062 C3Q1LA 132547279 Ki = 8.42 nM T79062 CAVB41 132584404 Ki > 10000 nM T79062 CS0MB3 132938109 Ki = 33 nM T79062 C8O2EP 134130246 Ki = 37 nM T79062 C8M9FH 134130379 Ki = 613 nM T79062 CA4GX3 134130447 Ki = 143 nM T79062 C7ZDA2 134130462 Ki = 53.7 nM T79062 CWL50Q 134130594 Ki = 1310 nM T79062 C8TG2O 134130846 Ki = 327 nM T79062 CHP3J4 134131015 Ki = 1377 nM T79062 CQ4IF8 134131147 Ki = 94.7 nM T79062 C6N5FS 134131151 Ki = 1328 nM T79062 CH4XB2 134131159 Ki = 990 nM T79062 CR32SP 134131265 Ki = 181 nM T79062 C0JKL5 134131283 Ki = 276 nM T79062 C0RQC6 134131976 Ki = 27 nM T79062 CQX4U3 134133064 Ki = 6.31 nM T79062 CTS3J4 134133483 Ki = 18.5 nM T79062 C0J2ML 134133604 Ki = 0.4677 nM T79062 CP0E5M 134133632 Ki = 497 nM T79062 CM0TS6 134133967 Ki = 44.67 nM T79062 CNV91Q 134134210 Ki = 23 nM T79062 C0ZLJ3 134134279 Ki = 648 nM T79062 CC1DO8 134134456 Ki = 25.5 nM T79062 CMS79H 134135372 Ki = 1038 nM T79062 C2Q3JY 134135516 Ki = 76 nM T79062 CJG3U0 134136134 Ki = 9.5 nM T79062 CGX03A 134136246 Ki = 131.83 nM T79062 C4VR6O 134137104 Ki = 18 nM T79062 C08ZBY 134137332 Ki = 32 nM T79062 CXF52V 134137560 Ki = 15.5 nM T79062 CN4LI8 134137732 Ki = 11.5 nM T79062 CWO5R6 134138168 Ki = 18 nM T79062 CRC2V0 134139826 Ki = 54 nM T79062 CG30KH 134140472 Ki = 126 nM T79062 CHK39T 134141166 Ki = 8 nM T79062 CLW86T 134141354 Ki = 257 nM T79062 C2NOX7 134141985 Ki = 34 nM T79062 CK54QW 134142259 Ki = 259 nM T79062 C6PSI9 134142907 Ki = 87 nM T79062 CR5L4K 134144303 Ki = 138 nM T79062 CYF16Z 134144798 Ki = 3063 nM T79062 C80TGJ 134144864 Ki = 25 nM T79062 CGW1D0 134145143 Ki = 1476 nM T79062 CK5RU9 134145903 Ki = 10 nM T79062 C2E0ID 134146185 Ki = 44 nM T79062 CC9P2T 134146194 Ki = 43.65 nM T79062 CV0QZ5 134147124 Ki = 52 nM T79062 C41XSD 134147935 Ki = 108 nM T79062 CFD13P 134147951 Ki = 1019 nM T79062 C8NBO0 134148917 Ki = 772 nM T79062 CBU81N 134149168 Ki > 10000 nM T79062 C0J8HT 134150597 Ki = 691 nM T79062 CE6LN3 134151118 Ki = 21 nM T79062 CLU34D 134151427 Ki = 265 nM T79062 C2JN8Y 134151729 Ki = 36.5 nM T79062 C76BZW 134151980 Ki = 16 nM T79062 CIV4H5 134152583 Ki = 254 nM T79062 CB6M5Y 134153538 Ki = 144 nM T79062 CX4W7F 134153716 Ki = 12 nM T79062 C79TEI 134154068 Ki = 25 nM T79062 C5B4GR 134154108 Ki = 1123 nM T79062 CMJ1U3 134154387 Ki = 65 nM T79062 C4M0FW 134154531 Ki = 79 nM T79062 C4VGJ5 134154679 Ki = 67 nM T79062 C6QAY2 134155116 Ki = 1.585 nM T79062 C79QLN 134155460 Ki = 91 nM T79062 CIUZ94 134155476 Ki = 10.5 nM T79062 C90QNV 134155645 Ki = 14 nM T79062 C97EWM 134155651 Ki = 389 nM T79062 CVR87Q 134156222 Ki = 125.89 nM T79062 CAB4K6 134156305 Ki = 19 nM T79062 C50XNE 134156520 Ki = 4.5 nM T79062 CUHE07 134157171 Ki = 6.5 nM T79062 CV8JU6 134157289 Ki = 73 nM T79062 CL6DN0 134157769 Ki = 14.5 nM T79062 C5IM7X 135367399 Ki = 363.08 nM T79062 C41JQV 135367400 Ki = 501.19 nM T79062 C2RN9U 135367403 Ki = 1407 nM T79062 C74JIA 135367404 Ki = 881 nM T79062 C6N8GM 135367405 Ki = 46.77 nM T79062 C6LU0C 135367816 Ki = 70 nM T79062 CTX68N 135367817 Ki = 883 nM T79062 CD2TH9 135367820 Ki = 52.48 nM T79062 CM7SA8 135367821 Ki = 369 nM T79062 CP21LA 135367855 Ki = 425 nM T79062 C5AMD9 135367857 Ki = 16 nM T79062 C6SKM3 135367858 Ki = 707.95 nM T79062 C5URG0 135367869 Ki = 1230.27 nM T79062 CBA7P6 135367917 Ki = 1436 nM T79062 C9DVI7 135367936 Ki = 386 nM T79062 CR0U6A 135367959 Ki = 316.23 nM T79062 CVE08Y 135458392 Ki = 15.3 nM T79062 CP7HN4 135458393 Ki = 33.3 nM T79062 CS8XJ6 135458394 Ki = 13.2 nM T79062 C9B7XA 135458410 Ki = 23.3 nM T79062 CFV9A3 135458427 Ki = 4.2 nM T79062 CKX4N8 135458428 Ki = 38.9 nM T79062 C9ZCL5 135458672 Ki = 4194 nM T79062 CTE23K 135464118 Ki = 512 nM T79062 CD6L8Q 135895192 Ki = 13.6 nM T79062 CA1M8B 135966709 Ki = 2.4 nM T79062 CUKO20 136020617 Ki > 10000 nM T79062 COF0U5 136020618 Ki > 10 nM T79062 CF89JI 136030596 Ki > 10000 nM T79062 CE8GB9 136030693 Ki > 10000 nM T79062 C65VFI 136030744 Ki > 10000 nM T79062 COIX80 136054961 Ki > 10000 nM T79062 C19GLK 136116062 Ki = 366.3 nM T79062 CQ2GP6 136118614 Ki = 1223 nM T79062 C8RH6M 136118617 Ki = 4114 nM T79062 CG5TX8 136118653 Ki = 3350 nM T79062 C40LYH 136118659 Ki = 5367 nM T79062 CY5GU4 136118730 Ki = 799 nM T79062 CB12QP 136152964 Ki = 24.8 nM T79062 CFX06E 136152966 Ki = 17.6 nM T79062 C37YXA 136152971 Ki = 7.7 nM T79062 CY0C1X 136152972 Ki = 1704 nM T79062 CX53NC 136180316 Ki = 145 nM T79062 CZ7WT9 136180317 Ki = 21.2 nM T79062 CQP2Y6 136180318 Ki = 1135 nM T79062 CQT9H5 136180319 Ki = 228 nM T79062 CLPU18 136180320 Ki = 11.9 nM T79062 C0LO6Q 136180321 Ki = 101 nM T79062 CAE39V 136188797 Ki > 10000 nM T79062 CWP0V5 136216703 Ki = 1600 nM T79062 CLAP52 136259032 Ki > 10000 nM T79062 CHM36P 137631892 Ki = 52 nM T79062 CU01TV 137633827 Ki > 10000 nM T79062 CC51JN 137635185 Ki > 10000 nM T79062 C94VXJ 137635884 Ki = 95 nM T79062 CFM92C 137636384 Ki = 3692 nM T79062 CDX39B 137637994 Ki = 142 nM T79062 C3LYX9 137641832 Ki > 10000 nM T79062 C5WS6Q 137642134 Ki = 14 nM T79062 CWUM83 137644521 Ki > 10000 nM T79062 CDA80E 137644790 Ki = 36 nM T79062 CZ8CU6 137645501 Ki = 56 nM T79062 CCP38D 137645926 Ki = 37 nM T79062 CVX74E 137646045 Ki = 438 nM T79062 CPI68E 137646281 Ki = 128 nM T79062 CMXI62 137649997 Ki = 209 nM T79062 C52IRM 137650705 Ki = 37 nM T79062 CKG08R 137650961 Ki = 165 nM T79062 CU4S1W 137651887 Ki = 5 nM T79062 CVK26R 137652044 Ki = 174 nM T79062 CHFK13 137652210 Ki > 10000 nM T79062 C51CGJ 137652310 Ki = 29 nM T79062 C2E3FV 137653850 Ki = 18 nM T79062 CX82HS 137654666 Ki = 32 nM T79062 C0SKV1 137654850 Ki > 10000 nM T79062 C4VG0U 137655411 Ki = 39 nM T79062 CO3L7F 137656918 Ki > 10000 nM T79062 CX4D7Y 137660741 Ki = 52 nM T79062 C0R6XM 138691314 Ki = 6 nM T79062 CU3Y7W 138691316 Ki = 20 nM T79062 CH2W4P 138691317 Ki = 531 nM T79062 CHSC40 138691321 Ki = 36 nM T79062 C18UZA 138691329 Ki = 42 nM T79062 C1XWV0 138691338 Ki = 30 nM T79062 C6LE1A 138691362 Ki = 44 nM T79062 CN9R4A 138691364 Ki = 5 nM T79062 C8H2KR 138691366 Ki = 302 nM T79062 C2Z9CD 139488518 Ki = 386 nM T79062 CJK95T 139488527 Ki = 22 nM T79062 CZ6H9M 139488539 Ki = 16 nM T79062 CAF2H8 139488606 Ki = 4 nM T79062 C54CIL 139488740 Ki = 18 nM T79062 CN3G0A 140936451 Ki > 10000 nM T79062 C4EU2S 141745651 Ki = 0.99 nM T79062 CCO6R0 141745657 Ki = 2.2 nM T79062 CO5DR9 145949220 Ki = 23 nM T79062 CWAF96 145949371 Ki = 10 nM T79062 CHG2W6 145950605 Ki = 9 nM T79062 COU57L 145950881 Ki = 7 nM T79062 CD4M6B 145951915 Ki = 85 nM T79062 C78AUI 145952711 Ki = 8 nM T79062 CA2J5S 145954503 Ki = 71200 nM T79062 C0JO8B 145954831 Ki = 10 nM T79062 CHI1V8 145956064 Ki = 566 nM T79062 CSER68 145956892 Ki = 20 nM T79062 CLVI07 145957637 Ki = 213 nM T79062 C91IDE 145958490 Ki = 1205 nM T79062 C8VS7K 145959257 Ki = 94 nM T79062 CSIZ31 145959706 Ki = 12 nM T79062 C67GQI 145961372 Ki = 2797 nM T79062 C4Y1PK 145963314 Ki = 6 nM T79062 C7KC3T 145963830 Ki > 10000 nM T79062 C5VWM7 145963860 Ki = 74 nM T79062 CCK5G1 145963863 Ki = 902 nM T79062 C4Y2AL 145964000 Ki = 3142 nM T79062 CV7YW9 145964086 Ki = 170 nM T79062 CHDN35 145964150 Ki > 10000 nM T79062 CR2B9G 145964154 Ki = 290 nM T79062 C1KH2E 145964159 Ki = 3600 nM T79062 C7YKQ4 145964390 Ki = 93 nM T79062 C95NZO 145964427 Ki = 89 nM T79062 C2P5NK 145964621 Ki = 67 nM T79062 CK0T1M 145964694 Ki = 213 nM T79062 C6T4RY 145964846 Ki = 90 nM T79062 CE9K3L 145964944 Ki = 12 nM T79062 C12OVL 145965034 Ki > 10000 nM T79062 CBS74V 145965054 Ki = 4 nM T79062 C9D8IB 145965203 Ki = 15 nM T79062 C1MIR9 145965401 Ki = 258 nM T79062 CLP94W 145965668 Ki = 245 nM T79062 C8TF9G 145965840 Ki = 121 nM T79062 C5W4LM 145965940 Ki > 10000 nM T79062 C53EFW 145966154 Ki = 547 nM T79062 CB05QA 145966199 Ki = 59 nM T79062 C1T4DN 145966418 Ki = 55 nM T79062 CV03XA 145967457 Ki = 1580 nM T79062 C81VUO 145967771 Ki > 10 nM T79062 CJS56K 145967795 Ki > 10000 nM T79062 CQ8EM6 145969402 Ki = 29 nM T79062 CA82FL 145970078 Ki = 2 nM T79062 CF74MR 145971390 Ki = 1671 nM T79062 C1T7GL 145971527 Ki = 12500 nM T79062 C8A2XG 145971561 Ki = 38 nM T79062 CN64ZR 145971588 Ki = 1154 nM T79062 CQJ5O8 145971635 Ki > 10000 nM T79062 C56RAO 145972025 Ki = 284 nM T79062 C79TNE 145972796 Ki > 10000 nM T79062 CJHI43 145972875 Ki = 52 nM T79062 CS7WG8 145973438 Ki = 1154 nM T79062 C8KYV6 145973487 Ki = 313 nM T79062 CEOY46 145973577 Ki = 388 nM T79062 CL74IP 145973853 Ki = 6 nM T79062 CR0CX6 145974087 Ki = 50 nM T79062 C6XIN0 145974114 Ki > 10000 nM T79062 C8KZ5T 145974165 Ki = 0.75 nM T79062 C05IVJ 145974184 Ki = 172 nM T79062 CW6EX3 145974189 Ki = 32 nM T79062 CD8ZL6 145974750 Ki > 10 nM T79062 C3WG0J 145975106 Ki = 52 nM T79062 C6PH4F 145975226 Ki > 10000 nM T79062 CN8U3P 145975289 Ki = 86 nM T79062 CSVR94 145975713 Ki = 408 nM T79062 COY2P3 145975720 Ki = 21 nM T79062 CL7EX5 145975776 Ki = 1050 nM T79062 C1BI8E 145975778 Ki = 534 nM T79062 C7R2MD 145975905 Ki = 100 nM T79062 C71CYU 145975946 Ki > 10000 nM T79062 C0V4AL 145975992 Ki = 275 nM T79062 C2TN8W 145976085 IC50 > 10000 nM T79062 C8XFM7 145976120 Ki = 3027 nM T79062 CF5B0W 145976158 Ki = 41 nM T79062 C8BJI2 145976292 Ki = 58 nM T79062 CZ5XK2 145976408 Ki = 67 nM T79062 C14OJW 145976618 Ki = 34 nM T79062 C0LRB2 145976686 Ki = 110 nM T79062 C34XME 145976696 Ki = 70 nM T79062 CTCM92 145976698 Ki = 415 nM T79062 CIZ69S 145976722 Ki = 228 nM T79062 CT7WO5 145976787 Ki = 213 nM T79062 CI8AN3 145976890 Ki = 32 nM T79062 C81CSM 145976946 Ki = 931 nM T79062 CXDR94 145977222 Ki = 3160 nM T79062 C8NW7Y 145977256 Ki = 43 nM T79062 CHS96B 145977297 Ki = 3.2 nM T79062 C6BFY7 145977338 Ki = 7400 nM T79062 C4L8EZ 145977467 Ki = 64 nM T79062 CC1DZ5 145977555 Ki = 204 nM T79062 C0Y6QO 145977799 Ki = 3300 nM T79062 C3BI1R 145978113 Ki > 10000 nM T79062 CP8C6M 145978146 Ki = 104 nM T79062 C6HQI0 145978420 Ki = 203 nM T79062 C8VL3Y 145978472 Ki = 529 nM T79062 C82NXP 145978482 Ki = 602 nM T79062 CQU8R0 145978665 Ki > 10000 nM T79062 C6AV9G 145978819 Ki > 10000 nM T79062 C20XQJ 145979626 Ki = 3609 nM T79062 C87MSW 145980271 Ki = 812 nM T79062 CW2CO4 145980458 Ki = 11 nM T79062 C8I7QL 145980875 Ki = 1120 nM T79062 CPK34X 145981875 Ki = 1.1 nM T79062 COY79P 145982165 Ki = 5 nM T79062 CEK60A 145982506 Ki = 165 nM T79062 CI59TX 145983018 Ki = 1119 nM T79062 CYC58R 145983059 Ki = 45 nM T79062 C4F5OT 145983128 Ki = 14 nM T79062 C5ZG9M 145983139 Ki = 7 nM T79062 CV2GU9 145983144 Ki = 65 nM T79062 C4PKM2 145983390 Ki = 19 nM T79062 C9LR8C 145983405 Ki = 0.55 nM T79062 CIAF74 145983468 Ki = 57 nM T79062 CE7MF4 145983751 Ki = 69 nM T79062 CDQ4U7 145983760 Ki = 19 nM T79062 CYW9B2 145983794 Ki = 32 nM T79062 C8I1WG 145983961 Ki = 3 nM T79062 CP5H4D 145984065 Ki = 8 nM T79062 CJ35DM 145984299 Ki = 9 nM T79062 CU7E4M 145984511 Ki = 51 nM T79062 C6JUY0 145984737 Ki = 12 nM T79062 CID02G 145984807 Ki = 672 nM T79062 CM5X3V 145985050 Ki = 0.4 nM T79062 CG10LK 145985224 Ki = 17 nM T79062 CFJ9B3 145985233 Ki = 12 nM T79062 C5AOI6 145985289 Ki = 24 nM T79062 CW30NA 145985505 Ki = 10 nM T79062 C7ZRP1 145985527 Ki = 12 nM T79062 C2XY8Q 145985533 Ki = 7 nM T79062 C7NI4X 145985585 Ki = 6 nM T79062 C9LJ5T 145985692 Ki = 1 nM T79062 C7QIX0 145985718 Ki = 52 nM T79062 C6V5QS 145985823 Ki = 12 nM T79062 C07GKD 145985958 Ki = 1340 nM T79062 CCM18E 145986031 Ki = 22 nM T79062 CR0XQ3 145986138 Ki = 31 nM T79062 CT37DW 145986720 Ki = 824 nM T79062 CNJH37 145986752 Ki = 949 nM T79062 C3VN5O 145987559 Ki = 165 nM T79062 CI0PA9 145987771 Ki = 3.3 nM T79062 CIS9P2 145988193 Ki = 12 nM T79062 CUGO10 145988693 Ki = 1574 nM T79062 C9D2OG 145988738 Ki = 3 nM T79062 C4C0YP 145988913 Ki = 172 nM T79062 CDY48U 145989143 Ki = 0.26 nM T79062 C3GPR9 145990093 Ki = 2085 nM T79062 C2Q5UK 145990353 Ki = 3 nM T79062 CT7AB8 145990459 Ki = 2172 nM T79062 C4GV8Q 145990586 Ki = 120 nM T79062 CVBR36 145991084 Ki = 0.79 nM T79062 C9TK6G 145991864 Ki = 2.6 nM T79062 CB8CM6 145992305 Ki = 209 nM T79062 CCP2U1 145992489 Ki = 10000 nM T79062 CLPU06 145992567 Ki = 224 nM T79062 CBI94R 145992877 Ki = 1.1 nM T79062 CI19KS 145993474 Ki = 2.3 nM T79062 C0TL8E 145993714 Ki = 19 nM T79062 CC2G1V 146025727 Ki = 3800 nM T79062 C5ZOJ3 146680920 Ki = 7832 nM T79062 CG97ER 146709966 Ki = 1000 nM T79062 CF5B2L 147653864 Ki = 398.11 nM T79062 C9T0PS 153061504 Ki = 691.83 nM T79062 CAF36V 153287539 Ki = 1000 nM T79062 C1FA0K 153287541 Ki = 19.95 nM T79062 CEQ69Z 153287542 Ki = 23.44 nM T79062 C6P3SR 153287553 Ki = 6.3 nM T79062 C3G5CJ 153287557 Ki = 199.53 nM T79062 CW31CT 153287566 Ki = 2.692 nM T79062 CYP86E 153287567 Ki = 199.53 nM T79062 CS73ZC 153287568 Ki = 1258.93 nM T79062 CV9G7Z 153287572 Ki > 10000 nM T79062 CO85KL 153287574 Ki = 1000 nM T79062 CZ1K4D 155510674 Ki = 21 nM T79062 CLX3D8 155510732 IC50 = 650 nM T79062 CC3KP7 155510927 Ki = 1148 nM T79062 CM4RB0 155511262 Ki = 3147 nM T79062 C9KX6O 155511928 Ki = 280 nM T79062 CZ7HP4 155512406 Ki = 40.1 nM T79062 C4OL0A 155512409 Ki = 3.43 nM T79062 CXF90M 155512487 Ki = 895 nM T79062 CO68LC 155512944 Ki = 49 nM T79062 C90FST 155513438 Ki = 51 nM T79062 C95QOT 155514378 Ki = 2352 nM T79062 C3SQI7 155514459 Ki > 10000 nM T79062 CI4DT8 155514575 Ki = 2455 nM T79062 CJUI87 155514774 Ki = 45 nM T79062 CQ84DA 155514889 Ki = 298 nM T79062 C3NB0D 155515324 Ki = 98430 nM T79062 C0Q8PR 155515407 Ki = 1833 nM T79062 CWO56B 155515415 Ki > 10000 nM T79062 CU0PY6 155515687 Ki = 9.42 nM T79062 C2TN5D 155515890 Ki = 184 nM T79062 C7KT0D 155515919 Ki = 1096 nM T79062 C13LOV 155515942 Ki = 6660 nM T79062 C7OF4C 155516118 Ki = 13750 nM T79062 CJ1Z0D 155516162 Ki > 10000 nM T79062 CG5M1O 155516282 Ki = 3743 nM T79062 CG53LH 155516399 Ki = 0.85 nM T79062 CU8TC0 155517162 Ki = 25 nM T79062 CW0B5K 155518159 Ki > 10000 nM T79062 CYB12O 155518974 Ki = 116500 nM T79062 CHVF41 155519045 Ki = 401 nM T79062 CCEZ93 155519102 Ki = 38730 nM T79062 CQD2J7 155519393 Ki = 9855 nM T79062 C2SXT1 155519515 Ki = 167 nM T79062 C0KLD8 155519559 Ki = 6248 nM T79062 C07BTO 155519598 Ki = 291 nM T79062 CUSA24 155519891 Ki = 1258.93 nM T79062 C5FL7R 155520499 Ki = 822 nM T79062 C8OC3W 155520552 Ki = 140 nM T79062 CTV2F6 155521010 Ki = 380 nM T79062 CQ76MP 155521503 Ki = 3715 nM T79062 C1OS6D 155522116 Ki > 10000 nM T79062 C98RDQ 155522218 Ki = 1115 nM T79062 C2TV4Y 155522487 Ki > 10000 nM T79062 CP6H1D 155522562 Ki = 432 nM T79062 CUQ61M 155522867 Ki = 7.54 nM T79062 CUG8L3 155522920 Ki > 10000 nM T79062 CD9QU6 155523519 Ki = 20 nM T79062 C5KYB4 155524228 Ki = 458 nM T79062 C6APG2 155524374 Ki = 36.6 nM T79062 CK4B0R 155524491 Ki = 1361 nM T79062 CUO93F 155524808 Ki = 305 nM T79062 CQB0M8 155524884 Ki > 10000 nM T79062 C65UZD 155524956 Ki = 286 nM T79062 C6MZJ9 155525703 Ki = 74 nM T79062 C81OCJ 155526014 Ki = 80.3 nM T79062 CZ81JA 155526026 Ki = 120 nM T79062 C1U2XO 155526651 Ki = 119 nM T79062 CXH79K 155526720 Ki = 11 nM T79062 CW68KC 155528355 Ki > 10000 nM T79062 C7C1EF 155528967 Ki = 1444 nM T79062 C5J7AU 155529153 Ki = 4247 nM T79062 C9KS5C 155529450 Ki = 58 nM T79062 CKZ25Y 155529679 Ki = 195 nM T79062 C3X4IA 155530328 Ki = 233 nM T79062 C9PC3D 155530350 Ki = 5996 nM T79062 CVLC03 155530779 Ki = 871 nM T79062 C98YQF 155531012 Ki = 258 nM T79062 C4W6VC 155531065 Ki = 1622 nM T79062 C5HWP4 155531362 Ki > 10000 nM T79062 CKDE38 155531753 Ki = 1 nM T79062 CCT8V9 155531846 Ki = 9531 nM T79062 C05KFL 155532137 Ki = 56.2 nM T79062 CMPU81 155532470 Ki > 10000 nM T79062 CX35QS 155532545 Ki > 10000 nM T79062 CX6DV4 155533028 Ki = 696 nM T79062 C23GDV 155533534 Ki = 1712 nM T79062 C3OEH2 155533648 Ki = 710 nM T79062 C15RYP 155533660 Ki > 10000 nM T79062 CY01GZ 155533850 Ki = 1384 nM T79062 CP3J8B 155534152 Ki = 3467 nM T79062 C3L0CP 155534184 Ki = 2431 nM T79062 CG85SB 155534301 Ki = 475 nM T79062 CG8Y7W 155534312 Ki = 366 nM T79062 C3VGT0 155534362 Ki = 1922 nM T79062 CW7SV9 155534575 Ki = 35 nM T79062 C75FSY 155534794 Ki = 2512 nM T79062 CTO4S9 155534839 Ki = 2 nM T79062 C6KF4E 155535154 Ki = 546 nM T79062 C8G7AW 155535428 Ki > 10000 nM T79062 C8O4IQ 155535827 Ki = 35 nM T79062 C14JEX 155535878 Ki = 776 nM T79062 CB79ZW 155536080 Ki > 10000 nM T79062 C5I1JA 155536087 Ki = 322 nM T79062 C72FLG 155536152 Ki = 3804 nM T79062 CW2SC8 155536533 Ki = 106 nM T79062 CTB93R 155536809 Ki = 462 nM T79062 C7FVE8 155537034 Ki = 6 nM T79062 C36FRH 155537074 Ki = 2095 nM T79062 CD75GP 155537227 Ki > 10000 nM T79062 CVS04L 155537788 Ki = 23 nM T79062 CB8IC7 155538144 Ki = 273 nM T79062 C5F2GI 155538236 Ki = 1092 nM T79062 COYG20 155538350 Ki = 933 nM T79062 C9TIU2 155538367 Ki = 53 nM T79062 CYC1P3 155538451 Ki = 73 nM T79062 CM08NT 155538716 Ki > 10000 nM T79062 CQ69UA 155538814 Ki = 5818 nM T79062 C0Q5NT 155538877 Ki = 133 nM T79062 CAT98F 155539483 Ki = 1158 nM T79062 C6S8BA 155539600 Ki = 4570 nM T79062 C9S2IA 155539605 Ki = 2765 nM T79062 C42GUK 155540147 Ki > 10000 nM T79062 C1X0IO 155540198 Ki = 197 nM T79062 C9J3BQ 155540635 Ki = 65.1 nM T79062 C1KA8C 155540755 Ki = 43.8 nM T79062 CR2K1T 155540795 Ki > 10000 nM T79062 CNU92V 155540807 Ki = 25 nM T79062 CUY87S 155540823 Ki = 119 nM T79062 COS2E7 155541072 Ki = 6417 nM T79062 CP7UG2 155541866 Ki = 3298 nM T79062 COZ46W 155541871 Ki = 53 nM T79062 CB62ZS 155542237 Ki = 2455 nM T79062 CXCW81 155542321 Ki = 11950 nM T79062 C9FS3Y 155542461 Ki > 10000 nM T79062 C9RV7W 155542678 Ki = 1.99 nM T79062 CT6HY4 155543250 Ki = 29 nM T79062 C68MSK 155543653 Ki = 8361 nM T79062 CZ7O0A 155544139 Ki = 5840 nM T79062 CD84VK 155544810 Ki = 336 nM T79062 C2XZD8 155545087 Ki = 404 nM T79062 CCX6T2 155545402 Ki = 3.3 nM T79062 CO9X1Z 155545526 Ki > 10000 nM T79062 CI0YL8 155545625 Ki = 70 nM T79062 C74GFO 155546189 Ki = 203 nM T79062 CH3W9N 155546350 Ki = 1445 nM T79062 C4UT5Z 155546595 Ki = 125 nM T79062 C98AIL 155546781 Ki = 3.54 nM T79062 CD02EN 155547436 Ki = 371 nM T79062 COJ27N 155547693 Ki = 10660 nM T79062 CAT9X4 155548275 Ki = 8511 nM T79062 C5LYE8 155548677 Ki = 5316 nM T79062 C0KZB5 155549018 Ki = 50.2 nM T79062 C87JGN 155549153 Ki > 10000 nM T79062 CGP8O5 155549315 Ki = 291 nM T79062 C52FRY 155549978 Ki = 192 nM T79062 C8HPN7 155551113 Ki = 420 nM T79062 C61IVC 155551353 Ki = 8 nM T79062 CHS71N 155551685 Ki = 119 nM T79062 CM26AV 155551704 Ki > 1000 nM T79062 C6E9LK 155552054 Ki = 366 nM T79062 CQ48CS 155552188 Ki = 0.9 nM T79062 CA1WS9 155552212 Ki = 5095 nM T79062 C38YJB 155552311 Ki = 2761 nM T79062 C87PTM 155552707 Ki = 11 nM T79062 CDQ7C2 155552798 Ki = 48960 nM T79062 CPV35U 155552826 Ki = 161 nM T79062 CDV6B9 155554036 Ki = 9247 nM T79062 CKF75H 155554324 Ki = 124 nM T79062 C6ZSU3 155554462 Ki = 2871 nM T79062 C8JKT1 155555378 Ki = 19.3 nM T79062 C2E5TR 155555506 Ki = 525 nM T79062 CUNK28 155555525 Ki > 10000 nM T79062 CO52HW 155556527 Ki = 5888 nM T79062 C1N5VF 155556756 Ki > 10000 nM T79062 CJCL47 155556806 Ki = 75.8 nM T79062 CJBX01 155557042 Ki = 199.53 nM T79062 C5QYS0 155557134 Ki = 34 nM T79062 CD2L3K 155557443 Ki = 21 nM T79062 CER48T 155557500 Ki > 10000 nM T79062 C2L0PC 155557720 Ki = 16 nM T79062 CF6H3V 155558408 Ki = 15180 nM T79062 C4I2OY 155558563 Ki = 27.8 nM T79062 C9TB5D 155559092 Ki = 2366 nM T79062 CP4JO7 155559794 Ki > 10000 nM T79062 COG70U 155560942 Ki = 7079 nM T79062 C2HF6P 155561581 Ki = 2329 nM T79062 COL7N8 155561901 Ki = 46 nM T79062 CL45NV 155561914 Ki = 17780 nM T79062 CJ57BI 155561978 Ki = 22 nM T79062 C0SDZ8 155561990 IC50 = 12 nM T79062 CW7M1D 155561995 Ki = 1112 nM T79062 C93KWN 155562202 Ki = 266 nM T79062 CO3C6L 155562423 Ki > 10000 nM T79062 C5AI0S 155562519 Ki = 641 nM T79062 C5BQ8U 155562652 Ki = 958 nM T79062 CF6B4W 155562834 Ki = 344 nM T79062 CZ6IA2 155562918 Ki = 514 nM T79062 CRCW25 155562997 Ki = 50 nM T79062 CBH14K 155563164 Ki > 10000 nM T79062 CG1L8E 155563286 Ki > 10000 nM T79062 C38WXS 155563374 Ki = 7322 nM T79062 C0INS4 155563826 Ki > 10000 nM T79062 CK0IW3 155563911 Ki = 6 nM T79062 C5TS7Q 155564824 Ki = 710 nM T79062 CQK8E3 155565209 Ki = 54.7 nM T79062 CE2YG1 155565215 Ki = 12.2 nM T79062 C2MIU5 155565813 Ki = 2730 nM T79062 C7P5VG 155566191 Ki = 206 nM T79062 C7O6YP 155566439 Ki = 16050 nM T79062 CG35LB 155566508 Ki = 24.2 nM T79062 CU46EB 155566665 Ki > 10000 nM T79062 C67LAG 155566854 Ki = 9120 nM T79062 CW1TN7 155566925 Ki = 14 nM T79062 C41UWT 155567307 Ki = 84 nM T79062 CA8OE0 155567476 Ki = 9.08 nM T79062 CC06FO 155567938 Ki = 1.86 nM T79062 CA68TK 155568224 Ki = 614 nM T79062 C4EX7C 155568246 Ki = 320 nM T79062 C4POS3 155568373 Ki = 32.7 nM T79062 C67MIN 155568606 Ki = 0.8 nM T79062 CXP3E4 155568794 Ki = 1501 nM T79062 CB5IP9 155569021 Ki = 166 nM T79062 C0CZK6 155569337 Ki > 10000 nM T79062 CP9V7M 155569396 Ki = 138 nM T79062 C3ZNX6 155569414 Ki = 552 nM T79062 CZ8RV4 155569568 Ki = 2170 nM T79062 C3N9VU 10251906 Ki > 500 nM T79062 CP9TR0 10324985 Ki = 9.1 nM T79062 D00CRA 1574 Ki = 1258 nM T79062 D00GSD 25107716 Ki = 0.58 nM T79062 D00MXS 5281703 IC50 > 350000 nM T79062 D00OBS 44559159 Ki > 10000 nM T79062 D00VRV 10171 Ki = 10 nM T79062 D00YEV 5281605 IC50 > 350000 nM T79062 D01KAX 135453290 EC50 = 5600 nM T79062 D01KVG 9843179 Ki = 1.995 nM T79062 D01WWC 16573 Ki = 20 nM T79062 D02HZG 888311 Ki = 2663 nM T79062 D02RAY 16754 Ki = 43 nM T79062 D02UWB 1809 Ki = 0.3981 nM T79062 D02YSX 197033 Ki = 7.943 nM T79062 D03DET 10287730 Ki = 501.19 nM T79062 D03NBX 637308 IC50 = 47600 nM T79062 D03TDN 1342 Ki = 83 nM T79062 D03TSY 24825775 Ki = 2.5 nM T79062 D03ZHB 44455973 Ki = 97.4 nM T79062 D04AQE 1833 Ki = 2 nM T79062 D04TPO 16006492 Ki = 15.85 nM T79062 D05EQG 5265 Ki = 19.95 nM T79062 D05GDP 599482 Ki = 1400 nM T79062 D05LKO 44414722 Ki = 840 nM T79062 D05XGR 6918647 Ki = 2511.89 nM T79062 D05ZUX 44207909 Ki >= 1000 nM T79062 D06VDN 443391 IC50 > 1000 nM T79062 D07JRV 46233381 Ki = 553 nM T79062 D07JTZ 9843889 Ki = 89 nM T79062 D07LRJ 5312149 Ki = 260 nM T79062 D08BCF 5011 Ki = 3033 nM T79062 D08CKM 9863250 Ki = 3 nM T79062 D08DOG 25130235 Ki = 5900 nM T79062 D08OFG 11177588 Ki > 10000 nM T79062 D08UOX 5281148 IC50 = 117500 nM T79062 D08VGJ 9904281 Ki = 294 nM T79062 D09BNS 439280 Ki = 2.12 nM T79062 D09RPR 16737207 Ki > 10000 nM T79062 D09RXU 45488131 Ki > 500 nM T79062 D09WIL 10028436 Ki = 1.995 nM T79062 D0B9TN 46233353 Ki = 4110 nM T79062 D0BG5H 11957684 Ki = 1.259 nM T79062 D0C5GF 6918515 Ki = 155 nM T79062 D0C5XQ 1832 Ki = 30 nM T79062 D0CA9H 25107518 Ki = 16.6 nM T79062 D0CK9K 6918513 Ki = 300 nM T79062 D0F0IA 11301655 Ki > 2000 nM T79062 D0F6CD 5202 Ki = 0.11 nM T79062 D0FF6S 16038374 IC50 > 10000 nM T79062 D0FU5E 10220053 Ki > 1000 nM T79062 D0G7QT 10131112 IC50 = 3000 nM T79062 D0G8CV 9954003 Ki = 7.943 nM T79062 D0H3KU 172267 Ki = 466 nM T79062 D0H7PC 6918553 Ki > 10000 nM T79062 D0H9QG 5312148 Ki = 31.6 nM T79062 D0HE4S 68788 Ki = 18 nM T79062 D0I0ML 35985234 Ki = 7.5 nM T79062 D0J6JT 1355 Ki = 304 nM T79062 D0K0HU 16747715 Ki = 7.6 nM T79062 D0K5NZ 68848 Ki = 7.943 nM T79062 D0KS0I 24894910 EC50 > 10000 nM T79062 D0L5MW 181743 Ki = 67 nM T79062 D0LT5D 11267988 Ki = 3.38 nM T79062 D0LV7U 10667433 Ki = 32 nM T79062 D0O3GF 1220 Ki = 388 nM T79062 D0OG0R 10337743 IC50 = 4764 nM T79062 D0R3GW 10296414 Ki = 199.53 nM T79062 D0T2RY 9948320 Ki >= 1000 nM T79062 D0X4PH 11224758 Ki = 0.22 nM T79062 D0X6MT 4106 EC50 = 0.6 nM T79062 D0X7SD 888197 Ki = 156 nM T79062 D0X9YS 23642275 Ki = 0.6 nM T79062 D0XX2U 16006606 Ki = 8.2 nM T79062 D0Y0SA 135399666 EC50 > 10000 nM T79062 D0Y9TL 13702393 Ki = 793 nM T68251 D00HNB 25419 IC50 = 145000 nM T68251 D00MDP 466151 Ki = 0.05 nM T68251 D01UBX 451415 IC50 = 9900 nM T68251 D01XWG 30323 IC50 = 1900 nM T68251 D04AIT 5280445 IC50 = 3610 nM T68251 D07VLY 31703 IC50 = 1100 nM T68251 D0K8KX 5280343 IC50 = 6680 nM T68251 D0Q8CS 60937 IC50 = 7200 nM T68251 D0R9BG 1990 IC50 = 15000000 nM T68251 D0RA5Q 72172 IC50 = 3400 nM T68251 D0S0LZ 54671203 IC50 = 24000 nM T68251 D0V4GY 9552079 IC50 = 7630 nM T68251 D0VM2L 68740 IC50 = 7000 nM T68251 D04LTF 9868980 IC50 = 0.46 ug.mL-1 T68251 D05VZE 119031 IC50 = 0.43 nM T68251 D0F2JS 15547703 IC50 = 190 nM T68251 D0MW3H 9824350 Ki = 154 nM T68251 D0N4IV 10718956 IC50 = 1.7 nM T68251 D0U2BH 65064 IC50 = 9600 nM T68251 D09EFW 46861776 IC50 = 3.42 nM T68251 D0G1LL 74221072 IC50 = 35000 nM T68251 D0LO1Z 5281858 IC50 = 6300 nM T68251 D0N6ZA 74221131 IC50 > 100000 nM T68251 D0UM5R 74221070 IC50 = 4700 nM T68251 D00UCC 9827497 IC50 = 0.78 nM T68251 D01DVX 9847838 IC50 = 482 nM T68251 D03BOZ 3342298 Ki = 0.22 nM T68251 D05VNG 9908389 IC50 = 1.8 nM T68251 D08CEE 10478364 Ki = 200 nM T68251 D0E5GY 9904965 IC50 = 7.4 nM T68251 D0P8YC 5362422 IC50 = 0.73 nM T68251 D0Q1CD 6918336 Ki = 11 nM T68251 D0T2IQ 443600 IC50 = 3000 nM T68251 D0T9HG 132519 IC50 = 0.104 nM T68251 D0Y1XT 128564 Ki < 1 nM T68251 CNA81R 1836 Ki = 80 nM T68251 CQS47H 2299 IC50 = 0.5 nM T68251 CZ45IU 4219 IC50 = 3.6 nM T68251 C24IRS 4222 Ki = 2000 nM T68251 CW1H7U 4323 IC50 = 5.998 nM T68251 CS8X0P 16124 IC50 = 49000 nM T68251 CL2W6Q 38422 IC50 = 7100 nM T68251 CA3M5F 68443 IC50 = 389000 nM T68251 CYEU83 69033 Ki = 70000 nM T68251 C0PY5N 77754 Ki > 100 nM T68251 C5Z1QA 96028 IC50 > 200000 nM T68251 CP4O2C 121255 Ki = 65000 nM T68251 CCY6L8 169853 IC50 = 31400 nM T68251 C7ROG5 177347 IC50 = 91.3 nM T68251 CP7Q8T 240910 Ki = 15000 nM T68251 CX3DK6 283995 Ki = 9000 nM T68251 CBN39D 285263 IC50 = 86.74 nM T68251 COFX01 352863 Ki = 70000 nM T68251 CNM0P3 391527 IC50 = 7 nM T68251 C4U7SY 401129 IC50 = 18700 nM T68251 CV60YH 445010 IC50 = 5 nM T68251 CK9M3P 445018 IC50 = 1 nM T68251 C4D7TS 448002 IC50 = 9.1 nM T68251 CR51PG 448593 Ki = 210 nM T68251 CC54LQ 450256 IC50 > 100000 nM T68251 CG1I8P 467296 IC50 = 88000 nM T68251 CTPW02 467297 IC50 = 34000 nM T68251 C9I8WB 478379 Ki = 0.2 nM T68251 C45JSH 639942 IC50 = 5.28 nM T68251 CP91NX 677915 IC50 = 1649.92 nM T68251 CS4O7K 685005 IC50 > 500000 nM T68251 CDE9V2 689424 IC50 = 1945.82 nM T68251 C5O0TJ 690158 IC50 = 8.95 nM T68251 C7TPR6 690965 IC50 = 5.37 nM T68251 CP1Q6R 703233 IC50 = 61000 nM T68251 C9FL2X 721434 IC50 = 1785.67 nM T68251 CTO15S 727131 IC50 = 9.17 nM T68251 CTV50K 727184 IC50 = 1859.32 nM T68251 C2CL6X 732134 IC50 = 6.32 nM T68251 CPKI76 765318 IC50 = 9.99 nM T68251 CXME85 766168 IC50 = 9.72 nM T68251 CWQG91 770865 IC50 > 1000 nM T68251 CQB03J 780790 IC50 = 6.41 nM T68251 C7EHR1 787183 IC50 = 5.46 nM T68251 C5MF2E 795596 IC50 = 1853.73 nM T68251 C1K0NF 795855 IC50 = 9.13 nM T68251 CW56XG 875024 IC50 = 9.66 nM T68251 C17IXT 910211 IC50 = 9.02 nM T68251 C9IFC6 1348435 IC50 = 2700 nM T68251 C8A5CX 1800786 IC50 = 500 nM T68251 CN9C8D 2140735 IC50 = 350000 nM T68251 C36DGS 2211098 IC50 = 53 nM T68251 CN6E3U 2366268 IC50 = 3600 nM T68251 C1ND5S 2734394 IC50 = 121000 nM T68251 CN62WX 2800809 IC50 > 10000 nM T68251 CEHZ37 3042462 IC50 = 383000 nM T68251 CY3TD6 3348132 Ki = 20 nM T68251 CME24U 3649035 IC50 = 26000 nM T68251 C3EI6T 4085085 IC50 = 67000 nM T68251 CBN96T 4358655 IC50 = 50118.72 nM T68251 CC5O4E 4369384 IC50 = 2000 nM T68251 CP8D7Y 4478236 IC50 = 20 nM T68251 CQ4Y5M 4626827 IC50 = 4.6 nM T68251 CZBY34 5220706 Ki = 72000 nM T68251 C20HRJ 5273475 IC50 = 6.24 nM T68251 CZS0G5 5276565 IC50 > 100000 nM T68251 C3JN0F 5277465 IC50 > 100000 nM T68251 CRJK67 5277481 IC50 = 37400 nM T68251 CYF7S5 5277490 IC50 = 15500 nM T68251 CQ4VL5 5287415 IC50 = 0.8 nM T68251 CW5SE3 5288615 IC50 = 4.7 nM T68251 CJ3QI1 5288814 IC50 = 2905 nM T68251 C5IDT0 5289314 Ki = 115 nM T68251 CVLS16 5319161 IC50 = 3880 nM T68251 CZC3I7 5326979 IC50 = 58000 nM T68251 CL89FO 5496920 Ki = 33 nM T68251 CDI23X 5941957 IC50 > 100000 nM T68251 C1K8FQ 6439677 IC50 = 800 nM T68251 CJG2B7 6476333 IC50 = 8960 nM T68251 CL5DH0 6479915 IC50 = 3580 nM T68251 CQEF36 6539670 IC50 = 1 nM T68251 C1LQD2 6540261 IC50 = 1100 nM T68251 CP7BG0 6852146 IC50 = 5 nM T68251 CN5L2B 6852147 IC50 = 1.5 nM T68251 CP2XK7 6882342 IC50 = 120000 nM T68251 CPFV65 6916013 Ki = 81.28 nM T68251 C7AZE5 6930803 IC50 = 100 nM T68251 C7Y1BX 9543420 IC50 = 13.3 nM T68251 CIJ25V 9794947 IC50 = 20000 nM T68251 CLK61C 9797144 Ki = 73 nM T68251 C7NP9Z 9798247 IC50 = 28 nM T68251 CET56A 9801414 Ki = 10 nM T68251 C76RCQ 9801569 IC50 = 341 nM T68251 C68HMJ 9801786 IC50 = 380 nM T68251 CJY12B 9802219 Ki > 3000 nM T68251 CIXD67 9802768 IC50 = 0.33 nM T68251 CUSD58 9803469 IC50 = 19 nM T68251 C4A0XM 9804305 IC50 = 457 nM T68251 CQ46XD 9804842 IC50 = 8700 nM T68251 CP65QD 9805079 Ki = 482 nM T68251 C1HP7E 9805710 IC50 = 25 nM T68251 CASW18 9806452 Ki = 17 nM T68251 C76CKA 9807105 Ki = 805 nM T68251 CTK6J8 9808181 IC50 = 34200 nM T68251 C9RQM7 9808674 IC50 = 0.3 nM T68251 CTO36D 9817594 IC50 = 30000 nM T68251 C5OE1B 9821883 Ki = 11 nM T68251 CJC20A 9822095 IC50 = 17 nM T68251 C6KJ9W 9822461 IC50 = 8.7 nM T68251 C6IX7G 9822926 IC50 < 0.1 nM T68251 C1MPW9 9823182 IC50 = 19 nM T68251 CTF8V4 9823391 Ki > 3000 nM T68251 CVN5Z3 9823395 IC50 = 12 nM T68251 C1PW5U 9824010 IC50 = 998 nM T68251 CDJB86 9825720 IC50 = 0.1 nM T68251 CXL65P 9825920 Ki > 3300 nM T68251 CL0G8K 9825927 IC50 = 602.56 nM T68251 C65ZHY 9826199 IC50 = 0.61 nM T68251 C1I6KQ 9826286 Ki = 500 nM T68251 C1A7NJ 9827355 Ki = 0.71 nM T68251 C3SZ8Y 9827469 Ki = 1244 nM T68251 C7I2FO 9828039 Ki = 324 nM T68251 C1GR4N 9828276 IC50 > 25000 nM T68251 CC1NG5 9829581 IC50 = 20 nM T68251 C7SRM4 9837496 IC50 = 3000 nM T68251 C9PW7L 9841168 Ki = 28.5 nM T68251 C5XL7R 9841323 IC50 = 0.6 nM T68251 CA7DJ9 9842114 IC50 = 3.199 nM T68251 C32JRZ 9843079 IC50 = 140 nM T68251 C6YT5W 9843479 IC50 = 40 nM T68251 CWY1J9 9846501 Ki > 3000 nM T68251 CE9AL3 9847113 IC50 < 0.1 nM T68251 CA1IP0 9847191 Ki > 3000 nM T68251 C8IMT2 9847787 IC50 = 1.1 nM T68251 C7VXJ5 9848025 IC50 = 3.9 nM T68251 C4IEK0 9850035 IC50 = 0.2 nM T68251 CD1KW6 9851858 Ki = 0.01 nM T68251 C5DGI9 9851911 IC50 = 6.6 nM T68251 C2FYO3 9852206 Ki = 0.01 nM T68251 C5TUJ7 9862317 IC50 = 39 nM T68251 C8GE7U 9862764 IC50 = 59 nM T68251 CS5JT6 9864502 IC50 = 59 nM T68251 CQ0J1G 9865191 IC50 = 17 nM T68251 CI8Z0R 9866250 IC50 = 1.6 nM T68251 CQ9SG1 9866486 IC50 = 1208 nM T68251 CR10NL 9866770 Ki > 3000 nM T68251 C0YN1X 9867935 IC50 = 20 nM T68251 CK3F1T 9868079 IC50 = 1.3 nM T68251 CX57RB 9868249 Ki > 3000 nM T68251 CJS23I 9868333 Ki > 3333 nM T68251 CJ8DP1 9868672 IC50 > 6000 nM T68251 C24JSB 9868858 IC50 = 2 nM T68251 CLQ29X 9869597 IC50 = 262 nM T68251 CG17NZ 9869811 IC50 = 4 nM T68251 CMEA71 9869947 IC50 = 0.5 nM T68251 C38BVX 9870100 IC50 = 19 nM T68251 CZO2I0 9870133 IC50 = 3 nM T68251 CA48SX 9870269 IC50 = 743 nM T68251 CD1XQ2 9871305 IC50 = 1.9 nM T68251 CSM16R 9871355 IC50 = 158 nM T68251 CHU9I8 9871883 IC50 < 1 nM T68251 C5NM6P 9872886 Ki = 91 nM T68251 C0TCJ2 9880675 Ki = 667 nM T68251 CW8IC4 9882151 IC50 > 100000 nM T68251 C0ZT7A 9883002 Ki = 13.9 nM T68251 C75DAZ 9885136 IC50 = 0.65 nM T68251 CG35XZ 9885916 IC50 = 148 nM T68251 CZBK85 9886177 IC50 = 21 nM T68251 C2M4EC 9887473 Ki > 3333 nM T68251 C4PB5Z 9887544 IC50 = 2.6 nM T68251 C3ZG6O 9887870 IC50 = 4 nM T68251 C8AJB7 9888429 Ki > 3000 nM T68251 CVP45O 9888530 IC50 = 175 nM T68251 CDW1O4 9888922 IC50 = 196 nM T68251 CD1U5P 9889190 IC50 = 12 nM T68251 C27HMG 9889517 IC50 = 1.6 nM T68251 C26SZX 9890226 IC50 = 0.4 nM T68251 CWN19T 9890526 IC50 = 3.3 nM T68251 CD79UJ 9890632 IC50 = 92000 nM T68251 CU65HY 9891358 IC50 = 0.06 nM T68251 C3QSE6 9891814 IC50 = 18 nM T68251 CF1X0W 9892321 IC50 = 534 nM T68251 CH69LT 9892815 IC50 < 0.1 nM T68251 CZU7Y4 9892876 IC50 = 73 nM T68251 CK1F3O 9892889 Ki > 305 nM T68251 C1NCU4 9894184 IC50 = 300 nM T68251 CX5G0F 9894469 IC50 = 1300 nM T68251 CZK6O9 9895099 IC50 = 300 nM T68251 CSIB97 9896504 IC50 > 30000 nM T68251 C5DW9S 9902427 IC50 > 30000 nM T68251 C97GSC 9903557 Ki = 1915 nM T68251 CD78ZQ 9907286 IC50 = 0.7 nM T68251 CN6WJ1 9909994 IC50 = 230 nM T68251 CJ3K1I 9910075 IC50 = 1480 nM T68251 CPO8V1 9910282 IC50 = 430 nM T68251 CM2F7R 9910302 IC50 = 1.1 nM T68251 C6NUE9 9910550 IC50 = 0.5 nM T68251 CP4LS8 9910727 IC50 = 87 nM T68251 CT50EC 9912183 Ki = 194 nM T68251 C62VZI 9912382 IC50 = 0.7 nM T68251 C3AZP0 9913479 IC50 = 0.3999 nM T68251 CR98KH 9913488 IC50 = 853 nM T68251 CSZV76 9913881 IC50 = 41 nM T68251 C7ZY1L 9914029 IC50 = 62 nM T68251 CA3FW0 9918908 IC50 = 0.004 nM T68251 CG1A6B 9924640 IC50 > 100000 nM T68251 C4YGT6 9928325 IC50 = 7.5 nM T68251 CK5OV9 9930210 IC50 = 33 nM T68251 C03GVA 9932290 Ki = 210 nM T68251 C1I2FW 9932632 Ki > 3000 nM T68251 CCHZ97 9932731 IC50 = 58000 nM T68251 CDXR37 9933197 IC50 = 0.1 nM T68251 CX17KQ 9933408 IC50 = 29 nM T68251 CF26MY 9934052 Ki > 3000 nM T68251 CA5V8M 9934053 Ki = 433 nM T68251 C57WSD 9934240 IC50 = 7 nM T68251 C65ION 9935032 IC50 = 0.1 nM T68251 CGFD83 9936194 IC50 = 188 nM T68251 C1HRU9 9936228 IC50 = 4.1 nM T68251 C68MQN 9936625 Ki = 435 nM T68251 C9OUC8 9936681 IC50 = 196 nM T68251 CG38KL 9936728 Ki = 1.1 nM T68251 CE59TP 9936926 IC50 = 547 nM T68251 CX7VQ9 9937188 IC50 = 10.96 nM T68251 CLM2R8 9941370 Ki = 3.5 nM T68251 C0IBF2 9941371 Ki = 0.03 nM T68251 CA30JY 9946988 IC50 = 70 nM T68251 CWZC93 9947332 IC50 > 100000 nM T68251 CSN61C 9948296 Ki = 1497 nM T68251 C16HTN 9948666 Ki = 27 nM T68251 CF1DO9 9950475 Ki > 567 nM T68251 CQY54S 9952396 IC50 = 2.1 nM T68251 C8C3DL 9953278 IC50 = 539.51 nM T68251 C16GIN 9953861 Ki > 1267 nM T68251 CR6EX3 9953909 Ki = 446 nM T68251 C8RXN6 9954304 IC50 = 297 nM T68251 C9X0YR 9954867 Ki = 6300 nM T68251 CK9HX0 9955125 IC50 = 0.4 nM T68251 C05HGV 9955795 IC50 = 1.1 nM T68251 C8M2RB 9956613 IC50 > 10000 nM T68251 C3Q2UJ 9956686 IC50 = 0.4 nM T68251 CS73TB 9956692 Ki = 2800 nM T68251 CI5TW9 9956699 IC50 = 529 nM T68251 CN76XI 9957653 IC50 = 1 nM T68251 CVG0O2 9959014 IC50 = 0.9 nM T68251 CN8TK0 9959428 IC50 = 661 nM T68251 CV40RB 9960075 Ki = 391 nM T68251 C9DRB7 9966028 IC50 = 110 nM T68251 C8K5VD 9969928 IC50 > 30000 nM T68251 CFQ15E 9976696 IC50 = 22 nM T68251 C0HL2X 9976697 IC50 = 2.7 nM T68251 C09LSY 9979489 Ki > 3333 nM T68251 CUA65C 9982414 IC50 = 12 nM T68251 CJGR30 9983604 IC50 = 0.5 nM T68251 CILK24 9983687 Ki = 1 nM T68251 CO0TX7 9993891 Ki > 600000 nM T68251 C3KX1B 9998685 Ki = 1 nM T68251 CB2J3S 9999667 IC50 = 10 nM T68251 C8W5UK 9999879 IC50 = 120 nM T68251 C6TO0A 10001582 Ki = 1.5 nM T68251 C59WEK 10001843 IC50 < 0.1 nM T68251 C5HN3L 10001964 IC50 = 222 nM T68251 CP5N4E 10005114 Ki = 43 nM T68251 C6U3CK 10006134 IC50 = 0.5 nM T68251 CA8C6U 10008733 Ki = 0.01 nM T68251 CR7T3J 10009978 Ki = 700 nM T68251 C71YGT 10025307 Ki = 4.7 nM T68251 C6O0MN 10026682 Ki = 5300 nM T68251 C6DGR7 10027203 Ki = 1.5 nM T68251 C4VJX9 10027747 IC50 = 32000 nM T68251 CM52RO 10030422 IC50 = 10 nM T68251 CJR59P 10031295 Ki > 3333 nM T68251 CX2W9O 10037048 IC50 = 200 nM T68251 C7J9ZF 10039403 IC50 = 32 nM T68251 C1X0SA 10041385 Ki = 8 nM T68251 CO39PK 10042482 Ki = 39.81 nM T68251 CW2MK1 10043732 Ki = 46 nM T68251 C7CT4E 10045150 IC50 = 0.34 nM T68251 CHF92V 10047100 Ki = 0.23 nM T68251 CCF5Z4 10047585 IC50 = 0.3 nM T68251 CAN59F 10047708 IC50 = 2.2 nM T68251 CV59KC 10049292 Ki = 340 nM T68251 CLZ87W 10051236 Ki = 1598 nM T68251 CSHD67 10054852 IC50 = 0.4 nM T68251 C42YWK 10055393 IC50 = 229.09 nM T68251 CSW7B3 10067146 Ki = 2.8 nM T68251 C69DPZ 10068042 IC50 = 15800 nM T68251 CD3RL7 10070821 Ki > 10000 nM T68251 CB28NP 10073353 IC50 = 30 nM T68251 CJK0R1 10074190 IC50 = 1 nM T68251 CU7DJ1 10081163 Ki = 77000 nM T68251 C8AEK4 10093420 IC50 = 0.38 nM T68251 C5W4ZA 10094362 IC50 = 300 nM T68251 CA6X2Z 10095338 IC50 = 0.6 nM T68251 CMY3X2 10098158 IC50 = 6.1 nM T68251 C2XV5J 10098250 IC50 = 0.4 nM T68251 C3V2HW 10099112 IC50 = 2 nM T68251 CXV2Y3 10109170 Ki = 433 nM T68251 CY6HZ7 10111132 IC50 = 74900 nM T68251 C0G7IY 10114318 Ki = 1870 nM T68251 C4P1LB 10116618 IC50 = 0.44 nM T68251 CU0D4S 10117481 Ki > 3333 nM T68251 CP5L0W 10117663 Ki > 3300 nM T68251 C7OPQ8 10118047 IC50 = 35 nM T68251 C7A8MI 10120093 IC50 < 0.1 nM T68251 CT4V0P 10120622 IC50 = 0.39 nM T68251 CY2N3D 10127629 Ki > 3330 nM T68251 C1N4MJ 10127670 Ki > 3330 nM T68251 CIL09Z 10127889 Ki > 3330 nM T68251 CYU19P 10127901 Ki > 3330 nM T68251 C07KFI 10128313 Ki > 3330 nM T68251 CB3I6K 10128659 Ki > 3330 nM T68251 C6ZK3A 10128916 Ki > 3330 nM T68251 CH0UW2 10129190 Ki > 3330 nM T68251 CZM7F4 10132758 IC50 = 80000 nM T68251 CDR73P 10135184 Ki > 2128 nM T68251 C7KR3Y 10136680 Ki = 440 nM T68251 CNU93J 10136924 Ki = 450 nM T68251 C1CDF2 10136925 Ki = 340 nM T68251 CJ9EX4 10138303 Ki = 550 nM T68251 CFXC89 10139040 Ki > 3333 nM T68251 CGC6S5 10139402 Ki > 3333 nM T68251 CP8QV4 10140363 Ki = 1920 nM T68251 CU6Y9T 10140438 Ki > 3333 nM T68251 CE75BY 10140776 Ki = 1400 nM T68251 CIH36M 10141214 IC50 = 18 nM T68251 C6MSI0 10141443 IC50 = 33000 nM T68251 CLXF15 10141613 Ki > 3300 nM T68251 C7VF1K 10141614 Ki > 3300 nM T68251 CWB5O4 10142326 Ki > 3300 nM T68251 CL7P6G 10143019 IC50 = 0.098 nM T68251 CPXB21 10143028 Ki > 3333 nM T68251 C23WZR 10143587 Ki > 3300 nM T68251 CZW98O 10156375 Ki = 3.8 nM T68251 CYO8D2 10159633 Ki > 3333 nM T68251 CQ4SJ5 10160197 Ki > 3333 nM T68251 CQ41YI 10161391 Ki > 3333 nM T68251 C7SXD4 10162245 Ki > 3300 nM T68251 CO6PS3 10162900 Ki = 150 nM T68251 CR5H6E 10163627 Ki > 2128 nM T68251 CI9VJ5 10163857 Ki > 3333 nM T68251 CR17PV 10164205 Ki > 3333 nM T68251 CZO5V4 10164317 IC50 < 0.4 nM T68251 CCM0Y8 10165180 Ki = 2167 nM T68251 C5ZO9J 10166232 IC50 = 0.53 nM T68251 C6IW4O 10173876 Ki > 3330 nM T68251 CGB27E 10174981 Ki > 3330 nM T68251 CL47AR 10175070 Ki > 3330 nM T68251 C4ULO6 10175077 Ki > 3330 nM T68251 C4QY3V 10175210 Ki = 3100 nM T68251 C84ZQD 10175219 Ki > 3330 nM T68251 CIT0H4 10175323 Ki > 3330 nM T68251 C95IGP 10175331 Ki = 2170 nM T68251 C4PDJ5 10175366 Ki = 110 nM T68251 CT7U0M 10175426 Ki > 3330 nM T68251 CD4AO0 10180362 IC50 = 2300 nM T68251 CEWF13 10180993 IC50 = 81800 nM T68251 CCX3T6 10183064 Ki > 15000 nM T68251 CDM94B 10183693 Ki > 3300 nM T68251 CHB2D3 10184071 Ki > 3333 nM T68251 C3E9NF 10184537 Ki > 3300 nM T68251 CTDP62 10184579 Ki > 3300 nM T68251 CXQ8N0 10185100 Ki > 3333 nM T68251 CK0P3F 10186536 Ki > 2128 nM T68251 CV7YI1 10186544 Ki > 3300 nM T68251 C51RPY 10195069 Ki > 3330 nM T68251 CCHX74 10195307 Ki = 200 nM T68251 C94KHT 10195527 Ki = 930 nM T68251 CDG35O 10196192 Ki = 370 nM T68251 CY36NO 10196425 Ki > 3330 nM T68251 C1JG5W 10196775 Ki > 3330 nM T68251 CVRZ27 10198038 IC50 = 80 nM T68251 C5CUM9 10202769 Ki > 3333 nM T68251 CX8BS3 10203685 Ki > 3333 nM T68251 CE1LI3 10204303 Ki = 90 nM T68251 C32RAQ 10204620 Ki > 3300 nM T68251 CQFP69 10206106 Ki = 270 nM T68251 CS1CA5 10207780 Ki = 1333 nM T68251 C4K1MJ 10208262 Ki > 2128 nM T68251 CYE02Q 10209301 IC50 = 2.6 nM T68251 CD76KE 10209382 Ki > 3333 nM T68251 CG8FA4 10218128 Ki > 3330 nM T68251 C7Y2US 10218353 Ki > 3330 nM T68251 C1C7AH 10223757 Ki > 3333 nM T68251 CYG10Z 10223774 Ki > 3333 nM T68251 CV5X8A 10224181 IC50 > 30000 nM T68251 CGKU70 10224396 Ki = 240 nM T68251 C7K1OR 10224602 IC50 = 1800 nM T68251 CLH71C 10225319 Ki > 3333 nM T68251 C2X1KF 10226116 Ki = 2566 nM T68251 C9CSG3 10226996 IC50 = 650 nM T68251 CUE63Q 10227853 Ki > 3300 nM T68251 C19DFP 10227854 Ki > 3300 nM T68251 CM7B5T 10228228 Ki > 3333 nM T68251 C7T0WH 10229644 IC50 = 1.1 nM T68251 CD2HP3 10230012 Ki = 1333 nM T68251 CCRM18 10231253 IC50 = 1.2 nM T68251 CCTY95 10237492 Ki > 3330 nM T68251 CQH2U3 10238391 IC50 = 200 nM T68251 CO8M7Q 10239526 Ki > 3330 nM T68251 CCQ9V5 10239716 Ki > 3330 nM T68251 CEO4X5 10239762 Ki > 3330 nM T68251 CU7TQ3 10239803 Ki > 3330 nM T68251 CLAX20 10250594 IC50 = 4.2 nM T68251 C0J3TC 10250722 Ki = 60 nM T68251 CL67DT 10252311 Ki < 2.8 nM T68251 CQJ0R3 10252900 Ki = 0.66 nM T68251 CK9DF5 10253223 IC50 = 12000 nM T68251 CQF3V9 10253673 IC50 = 9 nM T68251 CD8QY2 10253933 IC50 > 10000 nM T68251 CB6SE4 10256227 IC50 = 91 nM T68251 C7HZ1M 10270281 IC50 = 21700 nM T68251 C3XD1E 10271240 IC50 > 100000 nM T68251 C2MES9 10271604 Ki > 100000 nM T68251 CWJ02G 10273315 IC50 > 30000 nM T68251 C0K2ES 10273642 Ki > 3333 nM T68251 CJZP24 10273657 Ki > 3333 nM T68251 CK18DB 10273985 Ki > 2128 nM T68251 CGP97S 10274748 Ki = 140 nM T68251 C13NKU 10275545 Ki > 3333 nM T68251 C1NGV9 10276473 Ki > 3333 nM T68251 CES6A5 10276821 Ki = 1566 nM T68251 C1W7SN 10277073 Ki > 3333 nM T68251 CO18TA 10277120 Ki > 3333 nM T68251 CY6K1G 10277706 Ki > 3300 nM T68251 C2XU3O 10278147 IC50 = 0.67 nM T68251 C3IG0K 10280852 IC50 = 0.2 nM T68251 C80WUO 10282084 IC50 = 0.33 nM T68251 C7TWG0 10289551 Ki > 3330 nM T68251 CJ63ER 10289607 Ki > 3330 nM T68251 CR48SA 10289842 Ki > 3330 nM T68251 CO60CU 10290029 Ki = 2700 nM T68251 CJTV12 10293283 IC50 > 30000 nM T68251 CS69YG 10293394 IC50 = 3500 nM T68251 C89YGA 10295733 Ki > 2128 nM T68251 CDU36Y 10296475 Ki = 520 nM T68251 CTL3Y8 10296608 Ki > 3333 nM T68251 C48IRP 10296785 Ki = 500 nM T68251 CQ1Z0G 10298111 IC50 = 35 nM T68251 CN14MI 10298369 Ki > 3333 nM T68251 CU5E9Z 10299198 Ki = 1357 nM T68251 C25EKM 10299665 Ki > 3300 nM T68251 CQ5BE8 10299709 IC50 = 0.35 nM T68251 C1BR6A 10300063 Ki > 3333 nM T68251 C80VEU 10300077 Ki > 3333 nM T68251 C8U3KW 10301524 IC50 = 0.57 nM T68251 CFAU84 10301584 Ki > 3333 nM T68251 CP5AU1 10302088 Ki > 3333 nM T68251 C63BRA 10303333 IC50 = 34 nM T68251 CE1KM9 10311498 Ki > 3330 nM T68251 CJ15OB 10311501 Ki > 3330 nM T68251 C5F0EV 10311947 Ki > 3330 nM T68251 C4R9ZK 10311997 Ki = 83 nM T68251 CE6MB0 10312141 Ki = 116 nM T68251 C7G6QW 10312268 Ki > 3330 nM T68251 CQ5IT9 10312372 Ki > 3330 nM T68251 CP1GW0 10318094 Ki = 0.57 nM T68251 CIDW49 10319098 Ki > 3333 nM T68251 CF4KT9 10320002 Ki > 3333 nM T68251 CG23FV 10320328 IC50 = 4 nM T68251 CJWH74 10321975 Ki > 3333 nM T68251 CVKT01 10322744 IC50 = 50 nM T68251 CY08WJ 10322755 Ki > 3000 nM T68251 CQH5D4 10324032 IC50 = 0.1 nM T68251 CPI8R0 10324532 Ki = 3 nM T68251 CSFZ76 10325592 Ki = 1376 nM T68251 C1C4VZ 10326004 Ki = 0.9 nM T68251 C7UZA4 10340758 IC50 = 3.2 nM T68251 CCK1A4 10342176 IC50 = 8 nM T68251 CFO74N 10343375 Ki = 430 nM T68251 CJIW74 10343996 IC50 = 0.31 nM T68251 C94ANQ 10347529 IC50 = 0.6 nM T68251 C9FU5G 10362663 IC50 = 1 nM T68251 CWIM61 10364088 IC50 = 756 nM T68251 CL4B2U 10364155 IC50 = 567 nM T68251 CBA5I4 10365560 Ki = 1.1 nM T68251 CH89GT 10365752 IC50 = 3.4 nM T68251 CI0T8K 10366352 Ki > 3333 nM T68251 C6WZ4F 10367355 IC50 = 16 nM T68251 CT81YN 10370089 IC50 = 30 nM T68251 CBTO07 10370226 Ki > 3333 nM T68251 C0IUQ7 10387351 Ki > 3333 nM T68251 CZNT94 10389113 IC50 = 4 nM T68251 CY2G0R 10391428 Ki > 3333 nM T68251 C16BSA 10394828 IC50 = 50 nM T68251 CFKA79 10395015 Ki > 2000 nM T68251 C9HM1A 10402302 IC50 = 76000 nM T68251 CLP05D 10407603 IC50 = 5.2 nM T68251 C98HMP 10413940 Ki = 249 nM T68251 C7K0HG 10414437 Ki = 31 nM T68251 CH1S2G 10414974 Ki = 2.5 nM T68251 C4J7IP 10416507 Ki = 86 nM T68251 C0V9FN 10433382 IC50 = 0.1995 nM T68251 CS32HR 10435935 IC50 = 5.1 nM T68251 C7XE1L 10437629 IC50 = 5000 nM T68251 C5WV1N 10439082 Ki = 1867 nM T68251 C54UDR 10453826 IC50 = 891.25 nM T68251 CQUR30 10454592 Ki = 0.21 nM T68251 C6T8VC 10456675 Ki = 0.6918 nM T68251 C8M9FE 10462640 Ki = 30000 nM T68251 CA7DM9 10474389 IC50 = 0.7 nM T68251 CNQZ36 10483139 Ki = 410 nM T68251 COT6G1 10492779 Ki > 200000 nM T68251 C9KHT4 10495552 Ki = 30 nM T68251 CA7HT2 10498521 Ki = 15 nM T68251 C6KD0A 10498747 IC50 = 1.4 nM T68251 CL8O6I 10500340 Ki = 69 nM T68251 CGK80V 10500816 Ki = 35 nM T68251 CVID65 10500886 Ki = 17.78 nM T68251 CP37WK 10501527 Ki = 17 nM T68251 CK6YN5 10501862 Ki = 6 nM T68251 CZ2UY0 10502046 IC50 = 1 nM T68251 C36OMW 10502172 IC50 = 1 nM T68251 C9QE1B 10502327 Ki = 8 nM T68251 CHOX65 10502351 IC50 = 6.7 nM T68251 C5V8HJ 10502382 IC50 < 0.4 nM T68251 CJZ5T8 10502487 IC50 = 2770 nM T68251 CZ1R5Q 10502869 Ki = 8100 nM T68251 CBNM82 10503128 IC50 < 0.4 nM T68251 CO9S5H 10503708 Ki = 12 nM T68251 C5Y4IA 10504081 IC50 = 104 nM T68251 CD80YF 10504445 IC50 = 0.38 nM T68251 C2C7TE 10504472 IC50 = 2 nM T68251 CT2NM3 10505241 Ki = 19 nM T68251 CK2AB5 10505370 Ki = 2400 nM T68251 CH6S8Y 10505729 IC50 > 10000 nM T68251 C65KOE 10506125 IC50 = 33 nM T68251 C6D7JF 10506147 IC50 = 7 nM T68251 C7S0DB 10506158 IC50 = 16 nM T68251 CNH3L8 10506415 IC50 = 280 nM T68251 CS8V1G 10507004 Ki = 30 nM T68251 CV2T7C 10507137 Ki = 1800 nM T68251 C03MRW 10507152 Ki = 1.2 nM T68251 CDSO53 10507214 IC50 = 8.3 nM T68251 CFJ96A 10507282 Ki = 84 nM T68251 CC6H8T 10507755 Ki = 0.8 nM T68251 C9C5EL 10521197 IC50 = 8.4 nM T68251 CBT12Q 10522080 IC50 = 0.8 nM T68251 CXD8I5 10523292 Ki = 75 nM T68251 CZ36JW 10523383 IC50 = 530 nM T68251 C90HBF 10523728 Ki = 13 nM T68251 CQEH42 10524134 IC50 = 0.7 nM T68251 CYU87N 10524260 IC50 = 0.5 nM T68251 CX6EB7 10524337 Ki = 1800 nM T68251 CQTF46 10524338 Ki = 300 nM T68251 CYB53K 10525912 Ki = 33 nM T68251 CJK6G1 10526509 IC50 < 0.4 nM T68251 CSLO13 10526877 IC50 = 1000 nM T68251 CEK90M 10527263 IC50 = 50 nM T68251 CA83ON 10527749 IC50 = 18 nM T68251 CYGU41 10529315 IC50 = 1475 nM T68251 CBV6X5 10529587 IC50 = 4.4 nM T68251 CGK37L 10529602 Ki = 1.5 nM T68251 CIOJ69 10529720 Ki = 3000 nM T68251 C6PGE1 10530040 Ki = 380 nM T68251 C30UCT 10530499 Ki = 13 nM T68251 CQ82VY 10530944 Ki = 24 nM T68251 CEV6I5 10531005 Ki = 50 nM T68251 CJ2TZ3 10531167 Ki = 19 nM T68251 CS0AD8 10532048 Ki 17 nM T68251 C0WHA9 10546565 Ki = 9 nM T68251 C06NQR 10547080 IC50 = 66 nM T68251 C40ZXE 10547784 Ki = 7 nM T68251 CS10ZB 10549106 Ki = 19 nM T68251 C4PK0U 10549114 IC50 = 2.4 nM T68251 C4TA1K 10549256 IC50 < 0.4 nM T68251 C5JS8L 10549329 Ki = 10 nM T68251 CG27UI 10549756 Ki = 39 nM T68251 C82HQE 10550145 Ki = 6 nM T68251 C7WQ5Z 10550399 IC50 = 1 nM T68251 C1FA6T 10551440 IC50 = 50 nM T68251 CC2FM6 10551489 IC50 = 2391 nM T68251 C5UD0A 10551910 IC50 = 19 nM T68251 C4K3UD 10552661 Ki = 11 nM T68251 CU8QP7 10552732 Ki = 10 nM T68251 COYU34 10553872 Ki = 1900 nM T68251 C0S6GT 10554037 Ki = 16 nM T68251 CSQC42 10554611 Ki = 80 nM T68251 C7P5AW 10554727 Ki = 34 nM T68251 CI8XG0 10554869 IC50 = 8 nM T68251 CYJ41F 10554927 Ki = 3600 nM T68251 CZ41HP 10554978 Ki = 16 nM T68251 CD3R8V 10562830 IC50 = 8.32 nM T68251 CT7O9M 10569678 IC50 = 2 nM T68251 C8RWE4 10569743 IC50 = 36 nM T68251 C0M4VN 10570699 IC50 < 100 nM T68251 CE14GM 10570702 IC50 = 3 nM T68251 CUQ29Z 10571396 Ki = 170 nM T68251 CBXZ79 10572150 IC50 = 6 nM T68251 CPF0R5 10572544 Ki = 20 nM T68251 C21VZS 10573362 IC50 = 1.6 nM T68251 C42IAF 10573603 Ki = 15 nM T68251 CG39CF 10574279 Ki = 13 nM T68251 C8LYR6 10574340 IC50 < 1000 nM T68251 C42BTA 10576058 IC50 < 40 nM T68251 CH7Z2V 10576110 IC50 = 81 nM T68251 CK3JV9 10576740 IC50 = 3.3 nM T68251 CJ7KH8 10578213 Ki = 49 nM T68251 C1KH7E 10578728 IC50 = 9 nM T68251 CK05ZH 10579086 Ki = 0.7 nM T68251 C3R2SO 10580533 Ki = 20 nM T68251 C8J6HS 10591505 Ki = 83.18 nM T68251 CIUO27 10593253 IC50 = 2 nM T68251 CB20LM 10594000 Ki = 18 nM T68251 CUTS47 10594564 IC50 = 33 nM T68251 CN4Y6H 10594565 IC50 = 7 nM T68251 CD65OG 10594830 IC50 = 10.96 nM T68251 CJQY74 10595685 IC50 = 50 nM T68251 CI71CK 10595804 Ki = 10 nM T68251 CYNC76 10596158 IC50 = 12 nM T68251 CD65NF 10597516 Ki = 25 nM T68251 CP2H8O 10597673 Ki = 9 nM T68251 CL7EX4 10598952 IC50 > 1000 nM T68251 CUZ73T 10599048 IC50 = 50 nM T68251 CQCW86 10599579 IC50 < 0.4 nM T68251 CW18QK 10599594 IC50 = 1.2 nM T68251 CR1JI4 10600645 IC50 = 7 nM T68251 CN3E8J 10600844 Ki = 1.3 nM T68251 CJ86TP 10601066 IC50 > 1000 nM T68251 C5WUG1 10601082 Ki = 810 nM T68251 CEJ1U0 10603377 Ki = 18 nM T68251 C5G9MI 10610114 Ki = 120 nM T68251 C84URB 10610500 Ki > 100000 nM T68251 CPW6A4 10617505 IC50 > 1000 nM T68251 CL02BO 10618584 IC50 = 12 nM T68251 C06CAN 10619639 Ki = 12 nM T68251 CV14UH 10619971 Ki = 15 nM T68251 CR69NK 10621302 IC50 = 20 nM T68251 CSQ96T 10621933 Ki = 0.44 nM T68251 CVZ32G 10622447 Ki = 20 nM T68251 CL62YC 10622822 IC50 = 24 nM T68251 CL67UQ 10623250 IC50 = 8 nM T68251 C4FYL1 10623748 IC50 = 34 nM T68251 C6R4EG 10624005 Ki = 2 nM T68251 CR8X1Q 10624346 IC50 = 0.65 nM T68251 CKF6D7 10625329 Ki = 7.3 nM T68251 CGB29T 10625771 IC50 = 0.6 nM T68251 C6H9CT 10626366 Ki = 6900 nM T68251 C70MFZ 10626445 Ki = 18 nM T68251 C5VGB1 10626732 Ki = 21 nM T68251 C3NKC0 10626927 Ki = 17 nM T68251 CA63VQ 10640307 Ki = 36 nM T68251 C7KGM3 10642071 IC50 = 0.3 nM T68251 CI2QB9 10642965 IC50 < 0.4 nM T68251 CM1OZ6 10643325 IC50 = 5.9 nM T68251 C41RKE 10643401 Ki = 10 nM T68251 CUAI71 10643973 Ki = 2 nM T68251 CPYV83 10647658 Ki = 71000 nM T68251 CVX7Q2 10648390 Ki = 11 nM T68251 C4TXZ1 10648776 Ki = 100 nM T68251 C6S1KA 10649216 IC50 > 10000 nM T68251 C07FPQ 10649518 Ki = 55 nM T68251 COT6B8 10650624 Ki = 15 nM T68251 C69SPO 10650906 Ki = 0.6 nM T68251 CT23XW 10650907 Ki = 1.8 nM T68251 C13GKL 10658560 IC50 = 315000 nM T68251 C97KZU 10665624 IC50 = 39 nM T68251 CW1E7L 10667540 IC50 = 310 nM T68251 CF0E6H 10668745 IC50 = 13 nM T68251 CSCL07 10668823 Ki = 6.3 nM T68251 C4HJS1 10669027 Ki = 50 nM T68251 CFYC35 10669215 Ki = 3 nM T68251 C6TC0Z 10669216 Ki = 2.5 nM T68251 C78GYJ 10670529 IC50 = 1.3 nM T68251 C5FWS1 10670820 IC50 = 10 nM T68251 C4QVL0 10670896 Ki = 3 nM T68251 CB1F4G 10671203 IC50 = 110 nM T68251 C3DXN5 10671411 Ki = 0.92 nM T68251 CWB19K 10671441 Ki = 1.4 nM T68251 CXDM24 10671863 Ki = 0.54 nM T68251 C17LYV 10672346 IC50 = 26 nM T68251 CMU74I 10672857 IC50 = 6 nM T68251 CU6Y4O 10674458 Ki = 1600 nM T68251 CXTP56 10688727 IC50 < 1 nM T68251 CU5M1J 10691797 Ki = 42 nM T68251 CSA80H 10692194 IC50 < 1 nM T68251 CS5CL7 10692307 IC50 < 0.4 nM T68251 CR5KF8 10692994 IC50 = 535 nM T68251 CDI12G 10693559 IC50 = 6.8 nM T68251 C8JX1G 10693698 Ki = 3 nM T68251 CVML68 10693881 IC50 = 0.7 nM T68251 CM1T7K 10694510 Ki = 2.6 nM T68251 C7SM1E 10694604 Ki = 3.5 nM T68251 C3E1DX 10695165 IC50 = 4.4 nM T68251 C7ZQM4 10695491 Ki = 0.6 nM T68251 CZGC63 10695865 IC50 = 24 nM T68251 CVQF97 10695971 IC50 = 0.3 nM T68251 CW6CF7 10696226 IC50 = 2 nM T68251 C1YFC3 10696977 IC50 = 9 nM T68251 C4BME8 10697140 IC50 = 23 nM T68251 CBN9K8 10697378 Ki = 22 nM T68251 C1O5CQ 10697393 Ki = 210 nM T68251 CM4AI6 10698165 Ki = 100 nM T68251 C4THQ9 10698311 Ki = 280 nM T68251 C6Y1OU 10698367 Ki = 150 nM T68251 CG5JM9 10698412 Ki = 2.8 nM T68251 C56VSE 10698786 Ki = 1.5 nM T68251 C5E8QF 10707457 Ki = 87 nM T68251 C2GL3A 10714610 Ki = 44 nM T68251 C4IWF2 10714988 IC50 = 6 nM T68251 CO9KV7 10715115 IC50 < 1 nM T68251 C78CKH 10715629 IC50 > 20000 nM T68251 CE1D6G 10716217 IC50 = 3.5 nM T68251 C0ZX6T 10717308 IC50 = 9 nM T68251 C3TGW8 10717400 Ki = 61.66 nM T68251 CZ1M3L 10718058 Ki = 19 nM T68251 CQZ7M8 10718133 Ki = 13 nM T68251 CB96HF 10718916 IC50 > 1000 nM T68251 CN8AK6 10718996 Ki = 0.52 nM T68251 C2IS9D 10719476 Ki = 0.73 nM T68251 CVW81M 10719595 IC50 = 28 nM T68251 CI96XV 10720740 Ki = 14 nM T68251 CIV3P5 10720775 Ki = 760 nM T68251 C65IGZ 10720864 Ki = 21 nM T68251 CTGL64 10721152 Ki = 580 nM T68251 CF46SQ 10721337 Ki = 19 nM T68251 C4J1WN 10721454 IC50 = 0.2 nM T68251 CC1FB8 10721904 Ki = 2.5 nM T68251 CB2QD0 10723468 Ki = 0.9 nM T68251 CO7VP4 10737552 Ki = 18 nM T68251 C51DZG 10737732 IC50 = 11 nM T68251 C1LS5U 10738104 IC50 = 1 nM T68251 CL74TG 10738165 IC50 = 0.4 nM T68251 CB8G2D 10739728 Ki = 15 nM T68251 C4FWC9 10740485 Ki = 66 nM T68251 CKJD45 10741133 IC50 = 450 nM T68251 C0WKL7 10741470 Ki = 10 nM T68251 CPDX27 10741484 IC50 > 1000 nM T68251 C0QT2F 10741956 Ki = 7 nM T68251 CLI7B3 10742101 IC50 > 1000 nM T68251 CKX5R3 10742142 IC50 = 33 nM T68251 C39DPG 10742191 IC50 = 4.8 nM T68251 CHW23E 10742387 IC50 = 20 nM T68251 CY2BZ0 10742536 Ki = 41 nM T68251 C1LF0S 10744337 Ki = 48 nM T68251 CEV8X0 10744751 Ki = 25 nM T68251 CSM9H7 10745124 Ki = 800 nM T68251 C5BZ0J 10745489 Ki = 25 nM T68251 C9ILP3 10745718 IC50 = 31 nM T68251 C4IF2L 10745725 Ki = 25 nM T68251 CK30AE 10745748 Ki = 1.6 nM T68251 CWF50D 10745851 Ki = 21 nM T68251 CE09PI 10757715 IC50 = 6 nM T68251 CA3F1N 10758013 Ki = 43.65 nM T68251 CTKR07 10758266 Ki > 200000 nM T68251 CY9W4M 10760229 IC50 > 1000 nM T68251 CLEG16 10761206 Ki = 30 nM T68251 CDX13Z 10761730 Ki = 13 nM T68251 CA4U7D 10762262 Ki = 18 nM T68251 CP2G0N 10763745 Ki = 0.89 nM T68251 C68THN 10763851 IC50 = 0.3 nM T68251 CM54WS 10764477 Ki = 2400 nM T68251 CAG53Y 10764489 IC50 = 11.4 nM T68251 C7X6EC 10764497 Ki = 1500 nM T68251 CY8LV5 10765345 IC50 = 4.7 nM T68251 C3P2TS 10766036 IC50 = 17 nM T68251 CA6C0Z 10766622 Ki = 0.7943 nM T68251 CN6P1J 10766950 IC50 = 2.2 nM T68251 C0R1ZA 10767025 Ki = 0.64 nM T68251 CWR5Z3 10767105 IC50 = 29 nM T68251 CR4I1E 10767157 IC50 = 6 nM T68251 C7Q2EM 10767236 IC50 = 3 nM T68251 CNT4D0 10767387 Ki = 19 nM T68251 C18QVD 10768090 Ki = 61 nM T68251 C01YKA 10768236 IC50 = 13 nM T68251 CQ7J4I 10769007 IC50 = 12 nM T68251 C6VKJ9 10769394 Ki = 16 nM T68251 CQ6U2Y 10780743 Ki = 19 nM T68251 CIN4A9 10783989 Ki = 20 nM T68251 C15PVT 10785952 Ki = 20 nM T68251 CLAP90 10785969 IC50 = 23 nM T68251 C8AF9L 10787938 Ki = 0.88 nM T68251 C0DFB9 10788617 IC50 = 1 nM T68251 CNAE08 10788733 IC50 = 5 nM T68251 CXQD12 10789326 IC50 = 100 nM T68251 CM74LH 10789594 IC50 = 13 nM T68251 C8EOY6 10790150 Ki = 47 nM T68251 CHWG02 10790787 IC50 = 33 nM T68251 C0NP2Z 10790811 IC50 > 1000 nM T68251 C31EHR 10791372 IC50 = 84 nM T68251 C3P7LZ 10792025 Ki = 1.9 nM T68251 C8D1EN 10792133 IC50 = 3.9 nM T68251 C9VML0 10807861 Ki = 226000 nM T68251 CN8I3Z 10808172 IC50 = 9 nM T68251 CP72JG 10810483 IC50 = 4.8 nM T68251 CT1AI4 10810573 IC50 = 2 nM T68251 CU9F7V 10810684 Ki = 15 nM T68251 CS0O7M 10811110 Ki = 17 nM T68251 C49HCM 10812120 IC50 < 40 nM T68251 CEM1J0 10812918 IC50 < 40 nM T68251 CZB7L2 10812929 IC50 = 1.3 nM T68251 C4TF0K 10813874 IC50 < 0.4 nM T68251 CIUN51 10814028 IC50 = 46 nM T68251 CS7BY4 10816934 IC50 = 4 nM T68251 C3AI5Z 10831752 IC50 = 49 nM T68251 CMX2J7 10832371 IC50 > 1000 nM T68251 CF50HD 10832925 IC50 = 4 nM T68251 COE82D 10833334 Ki = 38.9 nM T68251 C5OG4U 10833497 IC50 = 61 nM T68251 C2A0IX 10833840 IC50 = 46.3 nM T68251 CH90ZB 10834348 IC50 = 14 nM T68251 C9M1JI 10834357 Ki = 10.96 nM T68251 CND0X1 10834889 IC50 = 130 nM T68251 CT3MN0 10837022 Ki = 4.6 nM T68251 CGR16B 10837261 IC50 = 1000 nM T68251 CR0E9Q 10837740 Ki = 3.89 nM T68251 C9H4CP 10838922 Ki = 0.52 nM T68251 CB32OK 10838949 IC50 > 1000 nM T68251 CR50UM 10839419 Ki = 5 nM T68251 CHWQ34 10839761 Ki = 1300 nM T68251 CA76MU 10840059 IC50 = 1160 nM T68251 CPD3L7 10840455 Ki = 32 nM T68251 CR2UX3 10840602 Ki = 94 nM T68251 CL1KG7 10840630 Ki = 24 nM T68251 CI0HR4 10840639 Ki = 39 nM T68251 C6ZSP8 10862104 Ki < 2.8 nM T68251 CQ1L7C 10863755 Ki = 690 nM T68251 C0AQL8 10873958 Ki < 2.8 nM T68251 CBQ70P 10874312 IC50 = 6.3 nM T68251 CLG40T 10874819 IC50 = 260 nM T68251 CXY47P 10875332 IC50 = 383 nM T68251 CJ0LE4 10876254 Ki = 50 nM T68251 CIB8Y1 10884337 Ki = 8 nM T68251 C3AY8O 10885569 IC50 = 20 nM T68251 CAU0I3 10885834 IC50 = 0.9 nM T68251 CDZ04P 10887027 Ki = 11 nM T68251 C7AMS4 10895808 Ki = 49 nM T68251 CPJ0I8 10896934 IC50 = 76 nM T68251 CU7YE0 10896986 IC50 = 0.7 nM T68251 C3FQT7 10903871 Ki = 82 nM T68251 CAF1N8 10906013 IC50 = 2500 nM T68251 CX93MR 10907320 IC50 = 9 nM T68251 CM9G8A 10907701 IC50 = 0.42 nM T68251 C13CJH 10907740 IC50 = 62 nM T68251 C69ZTR 10913644 Ki = 312 nM T68251 C2QR0W 10914151 Ki = 701 nM T68251 C7XE3L 10917417 Ki < 2.8 nM T68251 CGI2T1 10928606 IC50 = 176 nM T68251 CXHA75 10928874 IC50 = 1 nM T68251 CXY4L6 10929354 IC50 = 829 nM T68251 CDSQ41 10929404 IC50 = 106 nM T68251 C1QVT6 10939850 IC50 = 0.93 nM T68251 CWO29J 10940364 IC50 = 13 nM T68251 C89IYC 10948209 Ki < 2.8 nM T68251 CC46WL 10950008 Ki > 3000 nM T68251 C9YOU4 10951375 IC50 = 16 nM T68251 CJI1G0 10951750 IC50 = 1 nM T68251 CNBR78 10952384 IC50 = 8.82 nM T68251 C0A2IR 10958121 Ki = 14 nM T68251 C5HS4F 10961382 Ki = 491 nM T68251 CMY8S6 10961569 IC50 = 1.3 nM T68251 CPA1Q2 10961828 IC50 = 2.8 nM T68251 C30FBA 10970628 Ki = 19 nM T68251 CU2Q8S 10971085 IC50 = 320 nM T68251 CQ68IE 10972732 IC50 = 0.34 nM T68251 CJHO94 10972891 IC50 = 1.7 nM T68251 CTP6I0 10973485 IC50 = 3.6 nM T68251 C9DM0P 10980832 Ki = 11 nM T68251 CL7K8S 10983560 Ki < 3 nM T68251 C3UH2B 10983665 Ki = 647 nM T68251 CR9J5B 10983887 IC50 = 1.7 nM T68251 C68LPK 10983913 IC50 = 1.4 nM T68251 CS7D0Z 10984030 IC50 = 0.72 nM T68251 CV4J2F 10984597 IC50 = 0.3 nM T68251 C0G8TE 10993343 Ki = 11 nM T68251 CW8Z6R 10993677 Ki = 2518 nM T68251 CCX0L6 10994350 IC50 = 3.2 nM T68251 CW0Y6I 10994897 IC50 = 2.4 nM T68251 C3QX0T 11005761 IC50 = 0.45 nM T68251 CJM41O 11006091 IC50 = 1.3 nM T68251 C4PNK3 11006191 IC50 = 1810 nM T68251 C95NXQ 11006894 Ki = 0.64 nM T68251 C7WEZ4 11009332 Ki = 21000 nM T68251 C9WPH7 11016072 Ki = 880 nM T68251 CBE68H 11016073 Ki = 850 nM T68251 CG2DK0 11016448 IC50 < 0.4 nM T68251 C3IYK8 11016511 IC50 = 0.32 nM T68251 CF30UR 11016519 IC50 = 3.78 nM T68251 CODQ51 11016616 IC50 < 0.4 nM T68251 C6IHF5 11026991 IC50 > 8 nM T68251 C3LF1Y 11027584 Ki = 3001 nM T68251 CF5KU1 11027718 IC50 = 1.5 nM T68251 CA49QF 11027968 IC50 = 0.91 nM T68251 CLXZ15 11037377 Ki = 4.3 nM T68251 CT2S0G 11038175 IC50 = 7.4 nM T68251 C3W9IT 11046880 Ki = 408 nM T68251 C5R7JX 11049650 Ki = 1595 nM T68251 CW42KO 11049937 IC50 = 1.9 nM T68251 CQ08SN 11049982 IC50 = 1.8 nM T68251 C23KPN 11050468 IC50 = 2.3 nM T68251 C9RU4I 11059620 IC50 = 2.8 nM T68251 CH8O1E 11060081 Ki = 154 nM T68251 CM6X1E 11061555 Ki > 2000 nM T68251 C1N5PT 11070986 IC50 = 3.2 nM T68251 C18EIZ 11071831 IC50 = 0.6 nM T68251 C43JOG 11080156 Ki = 38 nM T68251 CT3VX4 11080936 Ki = 361 nM T68251 CG0A4C 11081333 IC50 = 25 nM T68251 C05MUK 11081992 IC50 = 1.6 nM T68251 CUNM68 11083152 Ki = 231 nM T68251 CS29GX 11091928 IC50 = 2.8 nM T68251 CE8V9B 11092295 IC50 = 4.22 nM T68251 CR8ZA7 11092551 IC50 = 14 nM T68251 CT2CH7 11092701 IC50 = 9.5 nM T68251 C6R7XB 11092861 Ki = 960 nM T68251 CX69YN 11093502 IC50 = 1.2 nM T68251 CR4V2D 11101785 Ki = 410 nM T68251 C8CK3E 11102531 IC50 = 24 nM T68251 C6G2DI 11111616 Ki = 23 nM T68251 CUK03P 11112062 Ki = 5812 nM T68251 CWV45Z 11112302 Ki < 2.8 nM T68251 CY1SR9 11113744 IC50 = 58.1 nM T68251 CNGP50 11122963 IC50 = 0.35 nM T68251 C8YVE5 11123989 IC50 = 5 nM T68251 CNBG53 11124956 IC50 = 1.6 nM T68251 CX2B6C 11125147 Ki = 450 nM T68251 C9GJ7C 11133809 Ki = 94 nM T68251 C2YBQ7 11134935 IC50 = 7.2 nM T68251 C8DMW5 11135133 IC50 = 83 nM T68251 CD3N8B 11135304 IC50 = 16 nM T68251 CF52TX 11143173 Ki = 1507 nM T68251 CH61QF 11144824 IC50 = 2.4 nM T68251 C8HM2R 11145437 Ki = 75 nM T68251 CHF19X 11146467 Ki = 32 nM T68251 C5WS3E 11147931 IC50 = 1000 nM T68251 CM0QK6 11156328 IC50 = 10 nM T68251 C9H1CW 11156691 IC50 = 16 nM T68251 CD1Q0L 11157488 IC50 = 1590 nM T68251 CZ8KI2 11157757 IC50 = 1500 nM T68251 CM04FR 11168103 IC50 = 10 nM T68251 CVR01T 11168326 IC50 = 7.21 nM T68251 CMKT17 11168614 IC50 = 886 nM T68251 C63CLD 11169065 IC50 = 1200 nM T68251 CD3WL8 11179683 IC50 = 8.4 nM T68251 C2LZ7F 11191803 IC50 = 85 nM T68251 CPA84O 11192618 IC50 = 1630 nM T68251 CCQ6N8 11194666 IC50 = 150 nM T68251 C43ONW 11202395 Ki > 3333 nM T68251 CO76XI 11205873 IC50 = 5000 nM T68251 C9R7OM 11207122 IC50 = 50000 nM T68251 CO87YZ 11215538 IC50 = 5000 nM T68251 CIZW31 11226189 IC50 = 323 nM T68251 C3LEA2 11226622 IC50 = 7 nM T68251 CEL1F0 11248884 IC50 = 19 nM T68251 CUOH67 11252195 IC50 = 500 nM T68251 CJZ3P6 11257884 Ki = 0.4 nM T68251 CO7T3M 11261246 IC50 = 0.41 nM T68251 CWG8Y6 11271094 IC50 = 236 nM T68251 C2OJ8Q 11272747 IC50 = 15000 nM T68251 CJX60I 11284255 IC50 = 5110 nM T68251 C6LJM4 11284404 IC50 = 522 nM T68251 CP17ID 11284983 IC50 = 1700 nM T68251 CF9O2R 11286824 IC50 = 3000 nM T68251 C1IW7N 11292680 IC50 = 0.09 nM T68251 C8C5AV 11294179 Ki > 3333 nM T68251 C7H9JG 11295013 IC50 = 26 nM T68251 C0ZI3J 11298263 IC50 > 200000 nM T68251 C78QSH 11307739 IC50 = 16 nM T68251 CRP08M 11310883 IC50 = 1000 nM T68251 CJ09XO 11317090 IC50 = 5 nM T68251 CK91YW 11317404 IC50 = 68 nM T68251 CLH50U 11318841 IC50 = 1760 nM T68251 C1SN8I 11319030 IC50 = 63 nM T68251 CN2P4G 11328571 IC50 = 321 nM T68251 C9FW7I 11330706 IC50 = 3650 nM T68251 C0XR3B 11330861 IC50 = 3010 nM T68251 CQH57S 11342435 IC50 = 135 nM T68251 CZ8B0D 11349945 Ki < 3.3 nM T68251 CYAK73 11353754 IC50 = 81 nM T68251 CA5P8H 11355488 IC50 = 76000 nM T68251 C7QNX8 11363138 IC50 = 1662 nM T68251 CHG6W0 11365417 IC50 = 62 nM T68251 CM8Y1J 11367571 IC50 = 3000 nM T68251 CTQK48 11373358 Ki > 3333 nM T68251 CLE30X 11374591 IC50 = 2.14 nM T68251 C5KU3Z 11376005 IC50 = 595 nM T68251 CEM0A7 11387990 IC50 = 6200 nM T68251 COZN84 11388372 IC50 = 15 nM T68251 CUJ4V0 11391937 IC50 = 8.2 nM T68251 C9ABX8 11397130 Ki > 3333 nM T68251 CF78WB 11398934 IC50 = 1410 nM T68251 C13NCF 11400989 IC50 = 300 nM T68251 CZM5E8 11410471 IC50 = 30 nM T68251 CU04HF 11419551 IC50 = 47 nM T68251 C4K9DO 11421151 IC50 = 3.2 nM T68251 C30PFC 11421763 IC50 = 2060 nM T68251 CK95HW 11429232 Ki = 0.4 nM T68251 C01FLQ 11441438 Ki = 3.2 nM T68251 CFE6A0 11443957 IC50 = 37 nM T68251 CZY3W9 11444262 IC50 = 12 nM T68251 CI0V6L 11447356 IC50 = 4000 nM T68251 COS67B 11456566 IC50 = 1370 nM T68251 CCMT46 11457732 IC50 = 20 nM T68251 C96DRO 11466734 IC50 = 581 nM T68251 C7QF0G 11467517 IC50 = 2150 nM T68251 CQ1D6E 11470070 IC50 = 200 nM T68251 C1KP2Q 11473879 Ki > 3333 nM T68251 CZBF91 11476645 IC50 = 156 nM T68251 C5Z4UP 11504653 IC50 > 2000 nM T68251 CWS35C 11510523 IC50 = 1270 nM T68251 C5G8PM 11511807 IC50 > 2000 nM T68251 C5VUM2 11517085 Ki = 300 nM T68251 C43OXZ 11519233 IC50 = 9 nM T68251 C5MO0U 11526826 IC50 = 5.3 nM T68251 CI8R5J 11529867 IC50 = 23100 nM T68251 C9Y6LH 11533683 IC50 = 3270 nM T68251 CE01PG 11543178 IC50 = 15370 nM T68251 C2OA3K 11547967 IC50 = 546 nM T68251 C1NZB9 11548265 IC50 = 0.3 nM T68251 CIWP38 11555036 IC50 = 18 nM T68251 C47VIT 11562805 IC50 = 4000 nM T68251 C61BQP 11562817 IC50 = 1563 nM T68251 CO9BC3 11562986 IC50 = 1272 nM T68251 CW5A4S 11569716 IC50 = 6.3 nM T68251 CHV2G1 11575995 Ki > 10000000 nM T68251 C3H2DG 11577137 IC50 = 135 nM T68251 CM6GO2 11577517 IC50 > 2000 nM T68251 CXT05D 11581283 IC50 = 1120 nM T68251 CX2PQ5 11588332 IC50 = 5740 nM T68251 C0Q5FU 11592023 IC50 > 2000 nM T68251 CSQ5M8 11598899 IC50 = 264 nM T68251 CTQ87G 11599024 IC50 = 1440 nM T68251 COT65V 11599397 IC50 > 2000 nM T68251 CUL5H2 11605631 IC50 = 4 nM T68251 CQ7G5D 11613116 IC50 = 1999 nM T68251 C0VCJ8 11613810 IC50 = 3.6 nM T68251 CXKU59 11620780 IC50 > 5000 nM T68251 CCBS59 11634234 IC50 = 280 nM T68251 CZO71U 11639846 IC50 = 550 nM T68251 CNY92D 11640694 Ki > 30000 nM T68251 CFV49P 11641262 IC50 < 1.5 nM T68251 CH3V8F 11663480 IC50 > 2000 nM T68251 CR2UN0 11669859 IC50 = 7.4 nM T68251 CK9F4P 11673778 IC50 = 9000 nM T68251 C90GCV 11675055 IC50 = 2110 nM T68251 C0WV8R 11678029 IC50 > 2000 nM T68251 CFC74O 11678245 IC50 = 574 nM T68251 C28WNK 11682752 Ki = 16 nM T68251 CY0T4D 11685065 IC50 > 2000 nM T68251 CRF7V9 11691964 IC50 = 1.3 nM T68251 CKGR97 11692294 IC50 = 1999 nM T68251 C6ORK5 11692747 IC50 = 655 nM T68251 C3U6ZR 11697504 Ki = 33000 nM T68251 C4BGI2 11698938 IC50 = 6958 nM T68251 C6PM1J 11713686 IC50 = 1380 nM T68251 C1MJ3P 11713694 IC50 = 126 nM T68251 C2BJ3X 11716217 Ki = 4599 nM T68251 C4FU2H 11717997 IC50 = 3430 nM T68251 C4ECU2 11720597 IC50 = 315 nM T68251 CCD93H 11730086 Ki = 80 nM T68251 C68KBY 11732585 Ki = 85 nM T68251 C7CED0 11733417 IC50 = 549 nM T68251 CI0KL2 11733573 IC50 = 13 nM T68251 C64LQC 11733862 Ki > 3000 nM T68251 CIU03K 11734219 Ki = 332 nM T68251 CJOE40 11748355 Ki = 4.8 nM T68251 C4HD9K 11751106 IC50 = 271 nM T68251 CG8U3H 11753351 IC50 = 3810 nM T68251 CO8QT0 11753905 Ki = 1100 nM T68251 C3P0TZ 11754739 Ki = 238 nM T68251 CJ4G5D 11754907 IC50 = 16.2 nM T68251 CD6S0B 11757331 IC50 > 100000 nM T68251 C5E7KU 11757592 Ki = 0.6 nM T68251 CUC9R5 11758082 IC50 = 0.7 nM T68251 CF2J8V 11758099 IC50 = 1000 nM T68251 CQ3Y4E 11761293 IC50 = 110 nM T68251 C6K8HR 11761578 Ki = 136 nM T68251 C04DFH 11783486 Ki = 4.8 nM T68251 CQP12F 11787159 IC50 = 86 nM T68251 C7BV5P 11792968 Ki = 40.74 nM T68251 CV16JZ 11793588 IC50 > 1000 nM T68251 CCSD72 11795621 IC50 = 7.8 nM T68251 CY8N1U 11795715 Ki = 5 nM T68251 CY7H2T 11795824 Ki = 12 nM T68251 C3DE6J 11796352 IC50 = 5.4 nM T68251 CK24XT 11796481 Ki = 8 nM T68251 C46KHU 11796490 IC50 = 5.2 nM T68251 C47OIA 11797154 IC50 = 0.8 nM T68251 CJ4VL3 11797382 IC50 = 10 nM T68251 C7VLP9 11798303 IC50 < 200 nM T68251 CHQR96 11798386 IC50 < 0.4 nM T68251 CZ3C9P 11798873 IC50 = 1.5 nM T68251 CXFP23 11798966 IC50 = 3.311 nM T68251 C19RCP 11799753 Ki = 3.7 nM T68251 CHS4I2 11800528 Ki = 38 nM T68251 CZ5LP1 11800650 IC50 = 10 nM T68251 CQ9HE2 11811551 IC50 = 53 nM T68251 CK03NI 11811717 Ki = 35 nM T68251 CLW3F1 11812791 IC50 = 24.2 nM T68251 C20PYA 11813392 IC50 = 12 nM T68251 CH3SV6 11813493 IC50 = 76 nM T68251 C8DY3Z 11817193 IC50 = 1000 nM T68251 CEN02U 11822212 Ki = 75 nM T68251 CDU9S2 11824087 Ki = 52 nM T68251 C3VO5H 11824148 Ki = 0.3 nM T68251 CKEM29 11827006 IC50 = 46 nM T68251 CV2MX4 11832221 Ki = 108 nM T68251 C48QEH 11833533 Ki < 2.8 nM T68251 CI2OP1 11942810 IC50 = 2700 nM T68251 C4XR5G 11963536 IC50 = 664 nM T68251 C02BWA 11967143 Ki > 2000 nM T68251 CB80OT 12000718 IC50 > 20000 nM T68251 C43PJZ 12000720 IC50 > 20000 nM T68251 CN72PQ 12037467 IC50 = 82.17 nM T68251 CKI97Z 12344252 IC50 > 200000 nM T68251 C0K8ZX 12404978 IC50 > 500000 nM T68251 C0JID3 12447203 Ki > 100000 nM T68251 CKSL53 12507616 IC50 > 200000 nM T68251 CTHQ39 12635073 Ki = 14000 nM T68251 CIQX87 12635074 Ki = 72000 nM T68251 C0XKJ1 12671872 IC50 = 1000 nM T68251 COF8W3 13008156 IC50 > 200000 nM T68251 CC9DK6 13384604 IC50 = 300 nM T68251 CSR94V 13559594 IC50 = 3.28 nM T68251 C71ASU 13644537 IC50 = 8.22 nM T68251 CQTX49 13738810 IC50 > 100000 nM T68251 CVH7N1 13746652 IC50 = 9800 nM T68251 C1AJO7 13968141 IC50 > 300000 nM T68251 CP8L5J 14104451 IC50 = 2000 nM T68251 CLS53V 14151811 IC50 = 9500 nM T68251 CQ3D9C 14151815 IC50 = 18000 nM T68251 C8TH1O 14177156 IC50 > 500000 nM T68251 CM9PD5 14237653 IC50 = 12400 nM T68251 CA2H8V 14303060 IC50 = 170 nM T68251 C7KDL3 14616290 IC50 = 98020 nM T68251 CY4XO2 14616291 IC50 > 500000 nM T68251 C1Q5JU 14616298 IC50 = 67010 nM T68251 C9TF7I 14616299 IC50 = 246260 nM T68251 CHU6J5 14616300 IC50 = 81010 nM T68251 C86DNV 14616301 IC50 = 64300 nM T68251 C47DQP 14732854 IC50 = 19000 nM T68251 C1IZ7D 15296597 Ki = 15 nM T68251 CGH19T 15296844 IC50 > 300000 nM T68251 CSU04W 15406874 IC50 = 5.8 nM T68251 C63MFQ 15435266 IC50 = 3 nM T68251 CH80JI 15435267 Ki = 25 nM T68251 CZ0NL1 15484680 IC50 = 6 nM T68251 CT68FI 15487434 Ki = 120 nM T68251 CJR3Z8 15487435 Ki = 110 nM T68251 C46XNB 15487436 Ki = 560 nM T68251 CP2C4Z 15524387 Ki = 31600 nM T68251 CAF7R5 15524388 Ki = 52 nM T68251 C17HGN 15524389 Ki = 6600 nM T68251 CFH8Y6 15524390 Ki = 35000 nM T68251 C3N1KV 15629940 IC50 > 100000 nM T68251 CVUY27 15631189 IC50 = 8490 nM T68251 C5TLB4 15765753 IC50 = 3.97 nM T68251 C5FA3L 15871222 IC50 = 0.7 nM T68251 CB3A4Z 15941413 Ki = 78 nM T68251 CA40FE 15941550 Ki = 6 nM T68251 CM3D1L 15941553 Ki = 110 nM T68251 CQ0ZL7 15941677 Ki = 23 nM T68251 C6F9WV 15941679 Ki = 70 nM T68251 C7C1HI 15941680 Ki = 34 nM T68251 CU2C1R 15987326 IC50 = 1040 nM T68251 CL7KX3 16040152 IC50 = 3 ug.mL-1 T68251 CTZ3R1 16040153 IC50 = 12.4 ug.mL-1 T68251 C4VW5F 16058482 IC50 = 35 nM T68251 C4WX2I 16108938 IC50 > 1000 nM T68251 CD51GI 16108939 IC50 = 5 nM T68251 C5YVB0 16108940 IC50 = 446 nM T68251 CB4DU9 16108941 IC50 > 5000 nM T68251 CBW71J 16108942 IC50 > 5000 nM T68251 CG6R9L 16108943 IC50 = 960 nM T68251 CN62KM 16108944 IC50 = 150 nM T68251 C7YS5Q 16108947 IC50 = 200 nM T68251 CLD2Y4 16108948 IC50 > 5000 nM T68251 CJR95O 16108949 IC50 > 1000 nM T68251 CRQ26L 16108950 IC50 = 350 nM T68251 CH80AG 16108951 IC50 = 13 nM T68251 CWB0G9 16108952 IC50 = 64 nM T68251 CS46XU 16126723 IC50 = 1.2 nM T68251 CC6OH2 16129741 IC50 = 43200 nM T68251 CH7D2Q 16420684 IC50 = 21200 nM T68251 C91EXN 16655061 IC50 = 555 nM T68251 CQS0F5 16719301 IC50 = 180 nM T68251 C0OUC6 16726064 IC50 = 23000 nM T68251 C75XDI 16730519 IC50 > 2000 nM T68251 C2W1VA 16739287 Ki = 5000 nM T68251 C6F9LM 16748789 IC50 > 30000 nM T68251 CXB10H 16748901 IC50 > 100000 nM T68251 C7YJZ5 17748252 IC50 = 2200 nM T68251 C3S2TQ 17754305 IC50 = 431 nM T68251 CQG89Z 17853548 IC50 = 64190 nM T68251 C2ZAX1 18002715 Ki > 3300 nM T68251 C12UGK 18002722 Ki > 3300 nM T68251 C0IYW8 18002726 Ki > 3300 nM T68251 C8N1DM 18002729 Ki > 3300 nM T68251 CCG96A 18002736 Ki > 3300 nM T68251 C5MLG1 18002745 Ki > 3300 nM T68251 CXT4H2 18002752 Ki > 3300 nM T68251 C26WHK 18002758 Ki > 3300 nM T68251 CV90XS 18002764 Ki > 3300 nM T68251 C8KPM7 18002765 Ki > 3300 nM T68251 CMJ0K3 18002771 Ki > 3300 nM T68251 C2CO9Z 18002775 Ki > 3300 nM T68251 CK8FS7 18173159 IC50 = 6 nM T68251 CX10BM 18173179 IC50 = 24 nM T68251 CQO70Y 18173222 IC50 = 82 nM T68251 C6F8WH 18319167 IC50 = 6 nM T68251 C57FQG 18319202 IC50 = 1790 nM T68251 CJ8G9A 18319234 IC50 = 334.97 nM T68251 CE4J1B 18319263 IC50 = 1300 nM T68251 CXG1K2 18363133 IC50 > 10000 nM T68251 C37BNA 18363136 IC50 > 10000 nM T68251 C0KOW7 18363142 IC50 > 10000 nM T68251 CP04KS 18363146 IC50 > 10000 nM T68251 CLZD96 18363152 IC50 > 10000 nM T68251 CW3KB9 18363153 IC50 > 10000 nM T68251 CK30ZO 18363159 IC50 > 10000 nM T68251 CZU27R 18363164 IC50 > 10000 nM T68251 CC0UV8 18363169 IC50 > 10000 nM T68251 CR3CQ4 18363187 IC50 > 10000 nM T68251 CH5IU9 18363209 IC50 > 10000 nM T68251 CJGZ27 18363210 IC50 > 10000 nM T68251 CWI2A9 18363212 IC50 > 10000 nM T68251 C31LQZ 18363213 IC50 > 10000 nM T68251 CE60WD 18363216 IC50 > 10000 nM T68251 C3L6DU 18363223 IC50 > 10000 nM T68251 CI53DY 18379040 Ki > 3333 nM T68251 CB1U5T 18379077 Ki > 3333 nM T68251 CSX97G 18379115 Ki > 3333 nM T68251 CJHL25 18379123 Ki > 3333 nM T68251 CR0B8G 18379149 Ki > 3333 nM T68251 CS4V5K 18379187 Ki > 3333 nM T68251 CCTY94 18379210 Ki > 3333 nM T68251 CA6K5S 18379235 Ki > 3333 nM T68251 CCSK49 18379254 Ki > 3333 nM T68251 CP4T7S 18379435 Ki > 3333 nM T68251 C9Y5GX 18379443 Ki > 3333 nM T68251 CXL6T9 18379569 IC50 = 173 nM T68251 CKY98M 18379668 IC50 = 9 nM T68251 CSY0N8 18394511 IC50 > 300000 nM T68251 C9J8IN 18445902 IC50 = 800 nM T68251 C5B9WG 18533077 IC50 = 800 nM T68251 C50AEZ 18616892 IC50 = 23.5 nM T68251 CYA3H7 18790040 IC50 > 10000 nM T68251 CBN28Y 18790155 Ki = 270 nM T68251 C03CET 18914685 Ki = 2000 nM T68251 CIEH93 19382975 IC50 = 6400 nM T68251 C60WKH 20196702 IC50 = 5.09 nM T68251 CK8MP3 20620240 Ki = 230 nM T68251 CPC4G6 20620273 Ki = 410 nM T68251 C26UJT 20620561 IC50 = 16 nM T68251 C2E3CY 20620614 IC50 = 48 nM T68251 CVEX54 20620688 IC50 = 6.6 nM T68251 CV1SD8 20620714 IC50 = 11 nM T68251 C3GAC4 20620715 IC50 = 270 nM T68251 C7QV8K 20620757 IC50 = 1100 nM T68251 CVO73Y 20620827 IC50 = 450 nM T68251 CQ14NY 20620831 IC50 = 940 nM T68251 C5RQ8A 20620860 IC50 = 10 nM T68251 CPK09X 20651316 IC50 = 1.4 nM T68251 CG1BD4 20689551 IC50 = 180 nM T68251 C48TWB 20728102 IC50 > 2000 nM T68251 C18RXS 20735191 IC50 < 0.1 nM T68251 C4I1OM 20735209 IC50 = 400 nM T68251 CF1CK9 20735364 IC50 = 0.5 nM T68251 CW3D7O 20760308 Ki = 1002 nM T68251 C09JTR 21130554 IC50 = 0.2 nM T68251 C6VP1T 21130556 IC50 = 0.2 nM T68251 C15UGO 21130558 IC50 = 5 nM T68251 C9H3IG 21130559 IC50 = 1.3 nM T68251 C8Q2OD 21130561 IC50 = 1.3 nM T68251 C25FAD 21130562 IC50 = 0.2 nM T68251 CW2Q5A 21130590 IC50 = 79.98 nM T68251 C9HMC0 21130591 IC50 = 184 nM T68251 CT87YK 21699971 IC50 = 5200 nM T68251 CH4G5T 21699977 IC50 = 400 nM T68251 CQ1GI3 21699983 IC50 = 650000 nM T68251 CJZ58F 21699985 IC50 = 37000 nM T68251 CA3WG1 21699989 IC50 = 4 nM T68251 CE72FU 21700004 IC50 = 950000 nM T68251 CRG8J9 21700008 IC50 = 20 nM T68251 C5JC6W 21700038 IC50 = 160000 nM T68251 CY18IE 21700054 IC50 = 89 nM T68251 CW1YS9 21700072 IC50 = 20 nM T68251 C3QAP8 21700080 IC50 = 45000 nM T68251 CG0RI5 21700124 IC50 = 5900 nM T68251 CR81NU 21700137 IC50 = 1300 nM T68251 CJ4C3K 21700144 IC50 = 85 nM T68251 C94FZS 21700146 IC50 = 26 nM T68251 CXME27 21700151 IC50 = 3400 nM T68251 CFK4Y7 21700160 IC50 = 6900 nM T68251 CIJ93L 21700163 IC50 = 25000 nM T68251 CN80JR 21700178 IC50 = 4 nM T68251 CB1QH3 21700191 IC50 = 480000 nM T68251 CUVE24 21700204 IC50 = 260000 nM T68251 CM42ZR 21700258 IC50 = 4 nM T68251 CMW12T 21700264 IC50 = 1 nM T68251 CKAJ52 21867770 IC50 = 0.7 nM T68251 C45UGA 21996090 IC50 = 16 nM T68251 CIC4S9 22004232 IC50 = 3.4 nM T68251 C36WFA 22096205 IC50 > 100000 nM T68251 CO91AD 22341241 Ki > 3333 nM T68251 CE5DH1 22484408 IC50 = 1.8 nM T68251 CZT05X 22484417 Ki = 550 nM T68251 CZT64B 22484431 Ki = 410 nM T68251 C1O7RC 22485248 IC50 = 400 nM T68251 CAM10T 22485252 IC50 = 0.8 nM T68251 CBJS34 22485260 IC50 < 0.1 nM T68251 C9MU7N 22485263 IC50 = 4.4 nM T68251 CEGJ03 22485276 IC50 = 3.3 nM T68251 C7VB8G 22485289 IC50 = 0.5 nM T68251 CNB02I 22485291 IC50 < 0.1 nM T68251 CAY3N6 22485292 IC50 = 1 nM T68251 C94OCJ 22485302 IC50 = 0.1 nM T68251 C3YL5X 22485311 IC50 = 0.1 nM T68251 C80RSQ 22485314 IC50 = 0.1 nM T68251 CWA03L 22485327 IC50 = 0.2 nM T68251 C6JRW5 22485340 IC50 = 0.1 nM T68251 C5JZF1 22485344 IC50 = 0.35 nM T68251 CI7MY5 22485346 IC50 = 0.1 nM T68251 CI1YL7 22485347 IC50 = 0.25 nM T68251 C25OBD 22485356 IC50 = 0.3 nM T68251 C7I0EW 22485367 IC50 = 0.2 nM T68251 CL64TJ 22485368 IC50 = 0.2 nM T68251 CT4GF9 22485381 IC50 = 6350 nM T68251 C27NDB 22485386 IC50 = 1.7 nM T68251 CTJ9I3 22485392 IC50 = 0.3 nM T68251 C3MG9P 22485396 IC50 = 0.4 nM T68251 CZY10U 22485408 IC50 = 0.3 nM T68251 C89AGT 22485413 IC50 = 0.2 nM T68251 C03NLM 22485417 IC50 = 0.1 nM T68251 C8GHU9 22485432 IC50 = 0.2 nM T68251 C9BT5F 22626996 IC50 = 77 nM T68251 C2Q4XK 22707806 IC50 = 0.1 nM T68251 CD4Z6P 22707833 IC50 = 3500 nM T68251 CMYK90 22707860 IC50 < 0.1 nM T68251 CVF9M4 22922043 IC50 = 23320 nM T68251 CX2JO7 22950015 IC50 = 335 nM T68251 COCN69 22956916 Ki = 1111 nM T68251 C85PXN 22956934 Ki = 771 nM T68251 CIYA45 22985930 IC50 < 0.1 nM T68251 CF75MS 23017979 IC50 = 60000 nM T68251 CQJ3S4 23018008 IC50 = 30000 nM T68251 CM5H2P 23061661 IC50 > 10000 nM T68251 C97LAR 23061665 IC50 > 10000 nM T68251 C2DG6O 23288322 Ki = 2000 nM T68251 C5XW9M 23310222 IC50 = 9 ug.mL-1 T68251 C9IW3E 23433373 IC50 = 1000 nM T68251 CX32YK 23513795 IC50 = 19 nM T68251 C6IZ1S 23513821 IC50 = 113 nM T68251 CPNM93 23513825 IC50 = 62 nM T68251 CML90Q 23513831 IC50 = 54 nM T68251 C87RTM 23513845 IC50 = 249 nM T68251 C4R2AJ 23625454 IC50 = 513 nM T68251 CD3U8A 23627203 Ki = 1300 nM T68251 C8UIC6 23644662 Ki > 100000 nM T68251 CCLA40 23644663 Ki > 100000 nM T68251 CSZ6J4 23645528 Ki = 3.2 nM T68251 C6UH9Q 23645529 Ki = 0.8913 nM T68251 CD0JP3 23645530 Ki = 0.7943 nM T68251 CM37EC 23645531 Ki = 2.399 nM T68251 C9PD5F 23645532 Ki = 2.884 nM T68251 C1OE7R 23645533 Ki = 0.7943 nM T68251 CCSN04 23645534 Ki = 1.4 nM T68251 CU08WI 23645535 Ki = 0.6918 nM T68251 CY41UC 23645536 Ki = 15 nM T68251 CX15EH 23645537 Ki = 3.7 nM T68251 CD3Q6G 23645538 Ki = 12 nM T68251 CE6NQ2 23645539 Ki = 19000 nM T68251 C4VK3U 23645540 Ki = 14000 nM T68251 C8VM1C 23645541 Ki = 73000 nM T68251 C0MUT6 23645542 Ki = 21000 nM T68251 CNI07H 23645543 Ki = 23000 nM T68251 CHK2X1 23645544 Ki = 38000 nM T68251 CW1V2Z 23645545 Ki = 14000 nM T68251 C6SP7T 23645546 Ki = 11000 nM T68251 CD9QO2 23645547 Ki = 900 nM T68251 C25YLZ 23645548 Ki = 90 nM T68251 CL1KC0 23652834 IC50 = 8.37 nM T68251 CL24JR 23655078 IC50 = 940 nM T68251 COIZ43 23655713 IC50 = 4350 nM T68251 CURM98 23655714 IC50 > 100000 nM T68251 CO90JC 23655717 IC50 = 5590 nM T68251 C3M2NQ 23655718 IC50 = 207 nM T68251 C56NMQ 23655910 IC50 = 9110 nM T68251 C9QZX5 23655911 IC50 = 6120 nM T68251 CA8W3K 23656106 IC50 = 239 nM T68251 CU4R7T 23656291 IC50 = 4 nM T68251 CVZ2M1 23656293 IC50 = 22 nM T68251 CL5C1I 23656295 IC50 = 30 nM T68251 CZP12E 23656450 IC50 = 2 nM T68251 CA2PY5 23657418 IC50 = 335 nM T68251 CN9TY1 23657419 IC50 = 992 nM T68251 C9FHZ1 23657421 IC50 = 19 nM T68251 CY9LF1 23657422 IC50 = 8 nM T68251 C28SPW 23657691 IC50 = 41000 nM T68251 CVJ1T7 23657695 IC50 = 20000 nM T68251 CAL05Q 23657697 IC50 = 35000 nM T68251 C6AW7U 23692637 IC50 = 2000 nM T68251 C7KF1N 23729138 IC50 = 6.8 nM T68251 C35QME 24742028 IC50 = 3 nM T68251 CY6KA0 24755074 IC50 = 5000 nM T68251 CG3J2L 24768528 IC50 = 120 nM T68251 CQCJ17 24768595 IC50 = 0.53 nM T68251 C5M3YW 24799779 Ki = 1000000 nM T68251 CWLT01 24806172 IC50 = 61 nM T68251 CN59KZ 24806173 IC50 = 1233 nM T68251 CH4X8K 24806175 IC50 = 13 nM T68251 C9RW0A 24806176 IC50 = 5.2 nM T68251 C18FRG 24807817 IC50 > 100000 nM T68251 CW3X0F 24852010 IC50 = 5.6 nM T68251 C2U0NS 24852011 IC50 = 8.3 nM T68251 C6YPS8 24852048 IC50 = 5 nM T68251 CUK6F1 24852487 IC50 = 95.9 nM T68251 C0MPV5 24852489 IC50 = 59.4 nM T68251 CK0CI6 24860421 IC50 = 334 nM T68251 CZI59C 24860423 IC50 = 97 nM T68251 CE29HI 24860424 IC50 = 1530 nM T68251 CT10JE 24860425 IC50 = 216 nM T68251 CRC98J 24860426 IC50 = 46 nM T68251 C8MKR0 24860427 IC50 = 1312 nM T68251 C3S6DX 24860428 IC50 = 56 nM T68251 C2LNE4 24860429 IC50 = 4181 nM T68251 CF4D0X 24860430 IC50 > 1666 nM T68251 CNR3U7 24866945 IC50 > 100000 nM T68251 CRZ7Y6 24868315 IC50 = 1.8 nM T68251 CFL04M 24881245 IC50 > 300000 nM T68251 CLIC14 24881246 IC50 = 60000 nM T68251 C3U8ZQ 24882385 IC50 = 230 nM T68251 C02WIB 24882535 IC50 = 20 nM T68251 C4FI5C 24901479 IC50 = 40 nM T68251 C6F0ZP 24901485 IC50 = 4.6 nM T68251 C4SP3O 24936157 IC50 = 0.67 nM T68251 CBUA83 24936183 IC50 = 12.6 nM T68251 CQ2K9H 24936215 IC50 = 488 nM T68251 C0EA5F 24936382 IC50 = 0.04 nM T68251 C78OAU 24944977 IC50 = 114 nM T68251 CO6CJ5 24945161 IC50 = 3600 nM T68251 C1C0NX 24945244 IC50 = 5300 nM T68251 CLTQ28 24945246 IC50 = 250 nM T68251 C7ZA6S 24945247 IC50 = 380 nM T68251 CH3O0V 24951588 IC50 = 83 nM T68251 C8I4PT 24951589 IC50 = 17 nM T68251 C2Q1BK 24951590 IC50 = 11 nM T68251 COMJ45 24951950 IC50 = 333 nM T68251 C3JGU2 24951952 IC50 = 24 nM T68251 CC7U2T 24951953 IC50 = 12 nM T68251 CV86KA 24952316 IC50 = 27 nM T68251 CYJ2E9 24952318 IC50 = 2535 nM T68251 CYKM71 24952674 IC50 = 139 nM T68251 C7MC8J 24952678 IC50 = 9.2 nM T68251 C0ZB8O 24953024 IC50 = 5.7 nM T68251 C5Z8XR 24953380 IC50 = 47 nM T68251 C2LN5E 24953381 IC50 = 119 nM T68251 CT2N3H 24953730 IC50 = 9.9 nM T68251 C1KH2Q 24953731 IC50 = 8.6 nM T68251 C0Q5BT 24954067 IC50 = 5.5 nM T68251 C6FI8O 24954068 IC50 = 5.6 nM T68251 CN29BR 24954070 IC50 = 5.5 nM T68251 CL1YO0 24954431 IC50 = 2.5 nM T68251 C3H9EO 24954432 IC50 = 7.6 nM T68251 CB60LR 24954795 IC50 = 24 nM T68251 C7P5YH 24954798 IC50 = 2.8 nM T68251 C5BG6I 24955154 IC50 = 32 nM T68251 CCE45B 24955155 IC50 = 56 nM T68251 CH53AG 24955156 IC50 = 47 nM T68251 CZC1P7 24955511 IC50 = 35 nM T68251 CL2G8J 24955513 IC50 = 281 nM T68251 CXG36M 24955514 IC50 = 4.8 nM T68251 CXO9Y4 24955857 IC50 = 36 nM T68251 CKY2F6 24955858 IC50 = 9.3 nM T68251 C4LJ8N 24955859 IC50 = 70 nM T68251 CX4MY3 24955861 IC50 = 67 nM T68251 CR29SO 24956227 IC50 = 509 nM T68251 CSM26P 24956228 IC50 = 102 nM T68251 C13JHO 24956229 IC50 = 4 nM T68251 C01QMC 24956580 IC50 = 1057 nM T68251 C8M5PJ 24956581 IC50 = 142 nM T68251 CC90AR 24956582 IC50 = 2382 nM T68251 CQH6I4 24956585 IC50 = 178 nM T68251 CHJ50Q 24956943 IC50 = 202 nM T68251 CN2AS5 24956945 IC50 = 670 nM T68251 C2HN8M 24956948 IC50 = 9.5 nM T68251 C2VEZ0 24957161 IC50 = 1318 nM T68251 CNCA57 25004194 Ki = 1.6 nM T68251 CIO26D 25022463 IC50 = 3 nM T68251 CWO3E0 25022465 IC50 = 170000 nM T68251 CAQ9Z1 25022681 Ki > 3333 nM T68251 CU6M9K 25060725 IC50 = 5400 nM T68251 CF7X2P 25060975 IC50 = 19000 nM T68251 CVR52U 25066764 IC50 = 60 nM T68251 CD2KA4 25102047 IC50 = 1.5 nM T68251 CRW96X 25102048 IC50 = 1 nM T68251 CQ3O9P 25102050 IC50 = 0.33 nM T68251 CSHA26 25102051 IC50 = 1.4 nM T68251 C7ADO2 25102197 IC50 = 0.37 nM T68251 CUR58H 25116339 IC50 = 297300 nM T68251 CA5DJ4 25138228 Ki = 2267000 nM T68251 CX6D9J 25138245 Ki > 3000 nM T68251 C7A6JQ 25138250 Ki = 5700 nM T68251 C6N7EQ 25138258 Ki > 3333 nM T68251 C7AD1J 25138259 Ki = 2933 nM T68251 CJ9TQ2 25138260 Ki > 3333 nM T68251 CUT8I7 25138261 Ki = 3300 nM T68251 CBD9X6 25138262 Ki > 3333 nM T68251 C8LX1S 25138263 Ki = 1367 nM T68251 C3OV1L 25138264 Ki > 3333 nM T68251 C92WVM 25138265 Ki > 3333 nM T68251 CMCS41 25138266 Ki > 3333 nM T68251 C1FJV5 25138267 Ki > 3333 nM T68251 C9N6WT 25138268 Ki > 3333 nM T68251 CF4QI1 25138269 Ki > 3333 nM T68251 C6P5UL 25138270 Ki > 3333 nM T68251 CQE0L7 25138271 Ki > 3333 nM T68251 C59XWU 25138272 Ki > 3333 nM T68251 C1TNQ3 25141117 Ki = 8.5 nM T68251 CYZ2J7 25141282 IC50 = 2 nM T68251 CR35QP 25144971 IC50 > 2500 nM T68251 C0Y5BC 25145683 IC50 > 2500 nM T68251 CGW49I 25146686 IC50 > 200000 nM T68251 CP0YF8 25146956 IC50 = 2900 nM T68251 C12AVL 25146957 IC50 = 3400 nM T68251 C10MBE 25146958 IC50 = 1500 nM T68251 CIUY75 25146959 IC50 = 2100 nM T68251 C5MG9N 25146960 IC50 = 6100 nM T68251 C83IOD 25147056 IC50 = 2200 nM T68251 C1IA0W 25147057 IC50 = 100 nM T68251 CB3W1I 25147058 IC50 = 800 nM T68251 CC35MZ 25147059 IC50 = 2200 nM T68251 CO5H9V 25147060 IC50 = 1600 nM T68251 CM20ZC 25147061 IC50 = 5 nM T68251 C2KZ0T 25147062 IC50 = 12 nM T68251 C5RMI2 25147153 IC50 = 100 nM T68251 C43YCQ 25147154 IC50 = 16 nM T68251 CPQW89 25147155 IC50 = 109 nM T68251 CQ3I6B 25147156 IC50 = 1100 nM T68251 CA34UT 25147158 IC50 = 4200 nM T68251 C3R0DB 25147159 IC50 = 5200 nM T68251 CV4ZE9 25147248 IC50 = 2100 nM T68251 C73HYI 25147249 IC50 = 3000 nM T68251 CV14TY 25147250 IC50 = 1 nM T68251 CUW8X2 25147251 IC50 = 4 nM T68251 C0Z7NX 25147252 IC50 = 11 nM T68251 CU1KO6 25147352 IC50 = 1000 nM T68251 CB1DY9 25147768 IC50 = 182900 nM T68251 CB7V8Y 25147773 IC50 = 0.35 nM T68251 C3KF1V 25178145 IC50 = 1.57 nM T68251 C8PMK7 25178356 IC50 > 100000 nM T68251 CG5Y2R 25178357 IC50 = 24.7 nM T68251 C4PZY6 25180866 IC50 = 145 nM T68251 CEP9Q2 25180867 IC50 = 0.5 nM T68251 C9HZG2 25181078 IC50 = 5120 nM T68251 CMYP34 25181079 IC50 = 2230 nM T68251 C7U1YC 25181080 IC50 = 25.3 nM T68251 C85HLG 25181081 IC50 = 16.2 nM T68251 CHR2P1 25183768 Ki > 25000 nM T68251 CZ8CR1 25190501 Ki > 3333 nM T68251 CO8CD1 25190502 Ki > 3333 nM T68251 C0R6MU 25212135 IC50 > 100000 nM T68251 C76PIF 26183540 IC50 = 33260 nM T68251 C9GCO4 28602444 IC50 = 48000 nM T68251 CW17CN 40516924 IC50 > 500000 nM T68251 C89YBJ 40582645 IC50 > 500000 nM T68251 C6AR8O 42623563 IC50 = 22000 nM T68251 CX0VP7 42623564 IC50 = 28000 nM T68251 C0H3RD 42627769 IC50 = 270 nM T68251 CB0QL3 42630085 IC50 = 37800 nM T68251 C7OX3C 42630086 IC50 = 47600 nM T68251 CAR56O 42645280 IC50 = 170200 nM T68251 CA6PS7 42645281 IC50 = 23500 nM T68251 C7R4JW 42645285 IC50 = 11200 nM T68251 CS29ZL 42645288 IC50 = 99700 nM T68251 C9JE0F 42645511 IC50 = 112100 nM T68251 CMK8T4 42645513 IC50 = 99700 nM T68251 CUF1L4 42645514 IC50 = 201900 nM T68251 C9WL3F 42645516 IC50 = 219400 nM T68251 C8OK0L 42645753 IC50 = 100700 nM T68251 C6K7LG 42645755 IC50 = 328500 nM T68251 CWS5M7 42645986 IC50 = 221000 nM T68251 CQBN65 42645987 IC50 = 632400 nM T68251 C6PI2X 42645989 IC50 = 211300 nM T68251 C8KM4E 43366432 IC50 = 8000 nM T68251 CPO1Z3 44123600 IC50 = 0.2 nM T68251 CWS64Q 44143474 IC50 > 15000 nM T68251 C7HV5Q 44143475 IC50 = 1590 nM T68251 C06IJY 44143476 IC50 = 1401 nM T68251 CVM82U 44143477 IC50 = 1241 nM T68251 C5XEB8 44143478 IC50 = 516 nM T68251 C0ZW7S 44143480 IC50 = 1093 nM T68251 C7K0YS 44143481 IC50 = 2674 nM T68251 CWU1K0 44143482 IC50 = 3614 nM T68251 CA29EQ 44143483 IC50 = 96 nM T68251 CA5P3E 44143484 IC50 = 15099 nM T68251 C7ER1N 44143485 IC50 = 855 nM T68251 C8YNO3 44143486 IC50 = 145 nM T68251 CLJG93 44143487 IC50 = 1743 nM T68251 CJB54F 44143488 IC50 = 2140 nM T68251 CH1IR0 44144307 IC50 = 14110 nM T68251 CT96JB 44199512 IC50 = 142900 nM T68251 C85BFQ 44199516 IC50 = 331100 nM T68251 CT80ED 44219901 Ki = 25 nM T68251 C94JVY 44219902 IC50 = 74 nM T68251 C7J6GH 44219903 IC50 = 26 nM T68251 C9J7WL 44219904 IC50 = 360 nM T68251 CRQ71E 44219905 IC50 = 310 nM T68251 C4Z0ID 44219906 IC50 = 56 nM T68251 CRNA25 44220092 IC50 = 17 nM T68251 C9T5ZF 44220093 IC50 = 9.6 nM T68251 CV38TE 44222825 IC50 = 5.5 nM T68251 CJI73R 44222826 IC50 = 1.5 nM T68251 CGQ30N 44222827 Ki = 3.8 nM T68251 CCI64J 44224245 IC50 = 66 nM T68251 CLRT69 44247751 IC50 = 3.5 nM T68251 CAR34Y 44263877 IC50 = 8.8 nM T68251 CEV08N 44263913 IC50 = 1.6 nM T68251 C5ZI0X 44263926 IC50 = 0.68 nM T68251 CO3C1E 44263994 IC50 = 2.7 nM T68251 C9XJ7U 44264020 IC50 = 3.4 nM T68251 C6L0MJ 44264021 IC50 = 2.4 nM T68251 CJ1WE7 44264036 IC50 = 0.7 nM T68251 C50QFR 44264375 IC50 = 5.3 nM T68251 CDL25C 44265349 Ki < 2.8 nM T68251 C3W4QO 44265401 Ki = 48 nM T68251 C2Q3JV 44265407 Ki = 2033 nM T68251 CN59QT 44265437 Ki = 500 nM T68251 CZA61K 44265475 Ki = 4.5 nM T68251 CD4A7F 44265476 Ki = 1133 nM T68251 CT6FK0 44265480 Ki < 2.8 nM T68251 C67HUL 44265485 Ki < 1 nM T68251 CH0O3I 44265492 Ki = 39 nM T68251 C4C7DY 44265493 Ki = 21 nM T68251 C0DFG7 44265501 Ki = 27 nM T68251 CXSD62 44265506 Ki = 310 nM T68251 CCM8K0 44265512 Ki = 2.8 nM T68251 CB3E6O 44265527 Ki < 2.8 nM T68251 COU3Y8 44266817 IC50 = 31 nM T68251 CUA5E0 44266818 IC50 = 8 nM T68251 CG23BI 44266830 IC50 = 8 nM T68251 C3YK0O 44268937 IC50 = 1000 nM T68251 C5DG8Z 44268941 IC50 = 200 nM T68251 C3SGT4 44268967 IC50 = 400 nM T68251 C1Z0GQ 44269012 IC50 = 1000 nM T68251 C18VGL 44269017 IC50 = 10000 nM T68251 CRF2Z5 44271421 IC50 = 8.05 nM T68251 CG7X5F 44272675 IC50 = 42.5 nM T68251 C2MWR0 44275913 Ki = 6.1 nM T68251 CKV1E7 44275972 Ki = 20 nM T68251 C6YT3K 44280285 Ki = 300 nM T68251 CC2O3U 44280323 Ki = 14 nM T68251 CIE09F 44280336 Ki = 0.3 nM T68251 CA1V6Y 44280345 Ki = 2 nM T68251 CI9L2E 44280411 Ki = 472 nM T68251 C8KZ2F 44281541 IC50 = 50 nM T68251 CRK8H6 44281557 IC50 = 66 nM T68251 CTJ7Q2 44281563 IC50 = 2.5 nM T68251 COU71D 44281564 IC50 = 64 nM T68251 CJ2PG9 44281705 IC50 = 23 nM T68251 C1M3JR 44281777 IC50 = 6.2 nM T68251 CL18QW 44281786 IC50 = 52 nM T68251 C3ES4Z 44281796 IC50 = 1.3 nM T68251 C60HIN 44281797 IC50 = 2.3 nM T68251 C8U5GR 44281941 IC50 = 110 nM T68251 CN23FC 44282968 IC50 = 1700 nM T68251 C2TV5I 44282969 IC50 = 50 nM T68251 CG3LF0 44282970 IC50 = 200 nM T68251 CC5XL3 44286083 IC50 = 48 nM T68251 CXT37W 44286406 IC50 = 35000 nM T68251 CB1R9G 44286414 IC50 > 10000 nM T68251 C7CU3J 44286466 IC50 = 19000 nM T68251 CZ2AL1 44286483 IC50 > 100000 nM T68251 C8I2EF 44286485 IC50 > 10000 nM T68251 C48FEB 44286518 IC50 = 130 nM T68251 CKM8V6 44286563 IC50 = 61 nM T68251 CJ1HT6 44288855 IC50 > 10000 nM T68251 CT38HI 44289140 IC50 > 10000 nM T68251 CAH30U 44289181 IC50 > 10000 nM T68251 CH1TS5 44289182 IC50 > 10000 nM T68251 CMZ2O6 44289200 IC50 > 10000 nM T68251 CBLC60 44289352 Ki = 31 nM T68251 CZO75J 44289369 Ki = 0.8 nM T68251 CRT7O2 44289382 Ki = 8 nM T68251 C7WUJ2 44289459 IC50 > 10000 nM T68251 CJ73FW 44289479 IC50 > 10000 nM T68251 CWMI67 44289482 IC50 > 10000 nM T68251 C1L4ZU 44289489 IC50 > 10000 nM T68251 C19EJM 44289515 IC50 > 10000 nM T68251 C6TI3X 44289520 Ki > 10000 nM T68251 CA52ED 44289521 Ki > 10000 nM T68251 C30KSP 44289579 Ki = 38 nM T68251 CHC08W 44289601 Ki = 36 nM T68251 CZ4EI7 44289602 Ki = 8 nM T68251 CEML82 44289603 Ki = 88 nM T68251 CM26JT 44289604 Ki = 27 nM T68251 CLY4K5 44289640 Ki = 4 nM T68251 C7GY8M 44289643 Ki > 10000 nM T68251 CV9B2F 44289867 Ki > 10000 nM T68251 CJ7VW3 44291166 IC50 = 0.7 nM T68251 C75IEN 44291420 IC50 = 30 nM T68251 CF21CS 44291532 IC50 = 0.7 nM T68251 CU75TB 44291559 IC50 = 53 nM T68251 C06JAO 44291626 IC50 = 49 nM T68251 C5XS0I 44294322 Ki = 1533 nM T68251 CC4V8S 44295180 IC50 = 50 nM T68251 CRW07Z 44295181 IC50 = 20 nM T68251 CL5QG6 44295202 IC50 = 540 nM T68251 CF0T8W 44295423 IC50 = 180 nM T68251 CVS7I1 44295425 IC50 = 550 nM T68251 CAFB18 44296974 Ki = 75 nM T68251 C5RSX9 44300181 IC50 = 19000 nM T68251 CKN3P7 44302022 IC50 = 100 nM T68251 C2Y0PK 44302023 IC50 = 9 nM T68251 C5S3UO 44302024 IC50 = 8 nM T68251 C8ERW6 44302042 IC50 = 10 nM T68251 C6JXH0 44302043 IC50 = 90 nM T68251 CI56DL 44302044 IC50 = 50 nM T68251 CWB83G 44302076 IC50 = 3 nM T68251 CY1J9U 44302096 IC50 = 5 nM T68251 CW94ZQ 44302164 IC50 = 47 nM T68251 C2FSR6 44302165 IC50 < 0.15 nM T68251 CQ54PZ 44302166 IC50 = 0.5 nM T68251 C9U3XT 44302167 IC50 = 0.6 nM T68251 C5X1WY 44302183 IC50 = 7 nM T68251 CQS19O 44302187 IC50 = 39810.72 nM T68251 C7G3BN 44302200 IC50 = 7 nM T68251 CMB4Q8 44302221 IC50 = 200 nM T68251 C70QWV 44302327 IC50 = 900 nM T68251 CZP20C 44302339 IC50 = 14 nM T68251 CO73BW 44302357 IC50 = 9 nM T68251 C6R0VK 44302358 IC50 = 500 nM T68251 CXUZ19 44302359 IC50 = 1 nM T68251 CNL4E2 44302361 IC50 = 19.95 nM T68251 C6YB0Q 44302364 IC50 = 10000 nM T68251 CCW65Y 44302378 IC50 = 1.995 nM T68251 CDK9W1 44302383 IC50 = 30.2 nM T68251 CYG80V 44302385 IC50 = 15 nM T68251 C7ZBR4 44302396 IC50 = 0.6 nM T68251 C8S5WT 44302397 IC50 = 1 nM T68251 CPC25G 44302409 IC50 = 13 nM T68251 C4QL0I 44302411 IC50 = 1 nM T68251 C4NDA2 44302416 IC50 = 12 nM T68251 C24ZWF 44302429 IC50 = 17 nM T68251 C4I6WO 44302430 IC50 = 0.8 nM T68251 CYL71W 44302432 IC50 = 3 nM T68251 C2X3QG 44302433 IC50 = 1000 nM T68251 C1J2AN 44302479 IC50 = 794.33 nM T68251 CE3BX0 44302505 IC50 = 200 nM T68251 C5H6OV 44302627 IC50 = 8 nM T68251 C6QR7C 44302634 IC50 = 15 nM T68251 CG8KJ0 44302661 IC50 = 5 nM T68251 CUZS20 44302663 IC50 = 600 nM T68251 CX1M3Q 44302666 IC50 = 6 nM T68251 C36CQP 44302952 IC50 = 12 nM T68251 CALD50 44304020 Ki > 3000 nM T68251 CTU4S6 44304048 Ki > 3000 nM T68251 CSVK45 44304230 Ki > 3000 nM T68251 CLH14M 44305978 IC50 = 5.9 nM T68251 CZ49UN 44305988 IC50 = 2.3 nM T68251 C6I8JA 44306058 IC50 = 1.9 nM T68251 CB5EY3 44306200 IC50 = 6.5 nM T68251 C0YOH1 44306202 IC50 = 3.8 nM T68251 CMA39E 44306203 IC50 = 2.1 nM T68251 CL58OS 44306208 IC50 = 14000 nM T68251 CAY2S4 44306209 IC50 = 1400 nM T68251 C27NJX 44306277 IC50 = 0.3 nM T68251 C6O1AN 44306279 IC50 = 0.8 nM T68251 C5AM6P 44308844 IC50 = 1587.17 nM T68251 CZUY51 44310789 Ki = 8.1 nM T68251 CH92OI 44310813 Ki = 3 nM T68251 CI4Y5N 44310825 Ki = 13 nM T68251 C5W8QH 44310847 Ki = 6.9 nM T68251 CLQV12 44310863 Ki = 0.44 nM T68251 CN9P5A 44310921 Ki = 0.42 nM T68251 CXB76U 44310932 Ki = 0.7 nM T68251 CMW5G3 44310933 Ki = 8.1 nM T68251 CBY0T1 44310973 Ki = 25 nM T68251 C5D9FS 44311011 Ki = 0.59 nM T68251 C2GC9W 44311172 Ki = 18 nM T68251 C0K1IL 44311187 Ki = 1.3 nM T68251 CL3CS0 44311254 Ki = 43 nM T68251 CV63JP 44311265 Ki = 1.9 nM T68251 CS56ER 44311267 Ki = 46 nM T68251 C5MBT7 44311268 Ki = 7.5 nM T68251 CM64HK 44311313 Ki = 1.9 nM T68251 CLQ48B 44311332 Ki = 6.7 nM T68251 C5AO7Z 44311335 Ki = 0.7 nM T68251 C78TEU 44311349 Ki = 0.96 nM T68251 CJEM64 44311491 Ki = 1.1 nM T68251 C2W5NQ 44311510 Ki = 0.47 nM T68251 C2MIT8 44311525 Ki = 1 nM T68251 CP7L6Q 44311566 Ki = 4 nM T68251 C0B4HZ 44312333 Ki = 12.88 nM T68251 CK9XB7 44314087 IC50 = 20 nM T68251 C8MRB1 44314322 IC50 = 0.36 nM T68251 CB6UL7 44314349 IC50 = 1.5 nM T68251 C3R0DL 44314366 IC50 = 1.9 nM T68251 C5ZTU6 44314442 Ki = 3.82 nM T68251 C2JUX9 44314443 Ki = 1.17 nM T68251 C92MGV 44314566 IC50 = 0.86 nM T68251 CLT6E0 44314618 IC50 = 3.7 nM T68251 CC95EZ 44314744 Ki = 0.33 nM T68251 CY63DG 44314754 Ki = 0.01 nM T68251 C8ZD7F 44314755 Ki = 10 nM T68251 COF0B1 44314762 Ki = 0.08 nM T68251 C59CBZ 44314763 Ki = 0.06 nM T68251 C9L1NY 44314788 Ki = 0.01 nM T68251 CM04TG 44314789 Ki = 0.03 nM T68251 C7LCN0 44314824 Ki = 10.3 nM T68251 CNM6W8 44314841 Ki = 0.01 nM T68251 C9K8JZ 44314900 Ki = 0.254 nM T68251 CXRE70 44314901 Ki = 0.06 nM T68251 CK3H1Y 44314929 Ki = 2.24 nM T68251 CS5A6Z 44314930 Ki = 0.06 nM T68251 CNB72W 44314931 Ki = 0.05 nM T68251 CBXI30 44314932 Ki = 0.02 nM T68251 CCF80X 44314958 Ki = 812 nM T68251 C3N8RQ 44314969 Ki = 1.83 nM T68251 C9SRT4 44314970 Ki = 1.03 nM T68251 C61DST 44314974 Ki = 0.03 nM T68251 CE2J4M 44314975 Ki = 0.01 nM T68251 CQE0D3 44314976 Ki = 0.59 nM T68251 CI2V1Y 44314995 Ki = 123 nM T68251 C48NVD 44314999 Ki = 0.01 nM T68251 CB7F0J 44315000 Ki = 0.3 nM T68251 CSY78M 44315028 Ki = 1300 nM T68251 CDZ5O3 44315029 Ki = 550 nM T68251 C6HW5G 44315084 Ki = 0.01 nM T68251 CV6KW1 44315085 Ki = 0.02 nM T68251 CH48TD 44315155 IC50 = 110 nM T68251 CAUQ47 44315167 Ki = 6 nM T68251 COA01P 44315179 Ki = 3000 nM T68251 CQ1R9E 44315204 Ki = 3.06 nM T68251 CL32FZ 44315221 Ki = 620 nM T68251 CDN4Y5 44315222 Ki = 860 nM T68251 C62FXJ 44315244 IC50 = 2.6 nM T68251 CP9M6W 44315277 Ki = 0.1 nM T68251 C3SZO4 44315279 Ki = 18.9 nM T68251 CSG05N 44315321 Ki = 0.02 nM T68251 COD08C 44315324 Ki = 46.5 nM T68251 C50IQE 44315333 IC50 = 6.6 nM T68251 C37JMW 44315348 Ki = 6.4 nM T68251 C89IQW 44318090 IC50 = 1 nM T68251 CJU31O 44321285 Ki = 17 nM T68251 C41VFA 44321286 Ki = 8 nM T68251 C5S2ZU 44321484 Ki = 85 nM T68251 CLQ23M 44321485 Ki = 202 nM T68251 CHF76Q 44321540 Ki = 9 nM T68251 CVOL49 44321593 Ki = 30 nM T68251 CB97GK 44321601 Ki = 26 nM T68251 CT0O7Y 44321602 Ki = 260 nM T68251 CU62BP 44321746 Ki = 11 nM T68251 CQU2K9 44321782 Ki = 100 nM T68251 CV8T3N 44321783 Ki = 19 nM T68251 CIBO50 44321801 Ki = 6 nM T68251 C4E8GU 44321802 Ki = 30 nM T68251 CYDN18 44321803 Ki = 40 nM T68251 C7Z4DQ 44321887 Ki = 24 nM T68251 CFJ20T 44321932 Ki = 10 nM T68251 C2E3RF 44321966 Ki = 75 nM T68251 CW9S1N 44321967 Ki = 330 nM T68251 C1FI3O 44321975 Ki = 14 nM T68251 CLB8J6 44321976 Ki = 80 nM T68251 CR0KN1 44322209 Ki = 250 nM T68251 C5LE1P 44322210 Ki = 31 nM T68251 CQ7AW8 44322211 Ki = 250 nM T68251 CJY2O7 44322214 Ki = 275 nM T68251 CR9GI0 44322215 Ki = 145 nM T68251 CYR6E5 44323170 Ki = 2000 nM T68251 C29OCD 44325165 Ki = 90 nM T68251 C20UGO 44325517 Ki = 157 nM T68251 C1SRC9 44325555 Ki = 6.9 nM T68251 CHMC02 44325564 Ki = 210 nM T68251 C8P6UA 44325625 Ki = 0.02 nM T68251 CBY75J 44325686 Ki = 1900 nM T68251 C6A1JX 44325696 Ki = 0.05 nM T68251 CJU3R8 44325730 Ki = 0.01 nM T68251 CBV73K 44325744 Ki = 0.03 nM T68251 C06ZAH 44325745 Ki = 0.01 nM T68251 C70UFH 44325749 Ki = 0.02 nM T68251 C8EWP2 44325750 Ki = 0.02 nM T68251 C2QL0B 44325810 Ki = 0.03 nM T68251 CS4EV5 44325831 IC50 = 3000 nM T68251 CU9B2Q 44325832 IC50 = 220 nM T68251 CP1NU9 44325834 Ki = 0.59 nM T68251 C7VRX2 44325907 Ki = 0.01 nM T68251 C80RKL 44326171 IC50 > 100000 nM T68251 C64XEI 44326172 IC50 = 670 nM T68251 C08MOK 44326187 IC50 > 100000 nM T68251 C3UB9D 44326260 IC50 = 17000 nM T68251 C1D8RA 44326261 IC50 = 2000 nM T68251 CK6P3C 44326668 IC50 = 370 nM T68251 C63XAO 44327476 IC50 = 90000 nM T68251 C7S4GH 44327780 IC50 = 200000 nM T68251 CXO1S8 44327801 IC50 = 100000 nM T68251 CW1QN6 44327818 IC50 > 500000 nM T68251 CTH2Y7 44327914 IC50 = 120000 nM T68251 CWYJ75 44327915 IC50 = 150000 nM T68251 C27ZST 44327916 IC50 = 60000 nM T68251 COAF26 44327936 IC50 > 500000 nM T68251 C9O8LM 44327939 IC50 = 160000 nM T68251 CB5L2U 44327940 IC50 = 72000 nM T68251 CI29FZ 44327960 IC50 = 155000 nM T68251 CV2U6R 44327961 IC50 = 54000 nM T68251 C8HUF1 44328149 IC50 > 500000 nM T68251 C85QTP 44328155 IC50 = 1000 nM T68251 CLK87J 44328168 IC50 = 150000 nM T68251 CMHZ13 44328169 IC50 > 500000 nM T68251 CZQ6N7 44328189 IC50 > 100000 nM T68251 C1IG0A 44328244 IC50 = 230000 nM T68251 CEI1V4 44328245 IC50 = 40000 nM T68251 CPI3A5 44328246 IC50 = 100000 nM T68251 CPU60Z 44328254 IC50 = 150000 nM T68251 CW3RX8 44328256 IC50 = 370000 nM T68251 CN81EA 44328258 IC50 = 43000 nM T68251 CR8XQ3 44328259 IC50 = 114000 nM T68251 CCD48V 44328263 IC50 = 2000 nM T68251 C31OKH 44328271 IC50 > 500000 nM T68251 CUA04P 44328279 IC50 = 125000 nM T68251 CHB05O 44328283 IC50 = 52000 nM T68251 CLC39W 44328295 IC50 = 110000 nM T68251 C36FCK 44328296 IC50 = 51000 nM T68251 CI46AP 44328297 IC50 > 500000 nM T68251 CR9YN5 44328312 IC50 > 500000 nM T68251 C8W9KN 44328316 IC50 = 50000 nM T68251 CPT80U 44328317 IC50 = 60000 nM T68251 CBD0Z2 44329014 IC50 = 5.97 nM T68251 CMLA39 44329018 IC50 = 1.3 nM T68251 C84MVU 44329019 IC50 = 5.73 nM T68251 C90CHA 44329405 IC50 = 7079.46 nM T68251 C2PB4Z 44329622 IC50 = 500 nM T68251 CI3Z4K 44329623 IC50 = 80 nM T68251 C6OL8M 44329636 IC50 = 10000 nM T68251 CB0G1H 44329644 IC50 = 1995.26 nM T68251 CA65RO 44329672 IC50 = 1995.26 nM T68251 CK9HO7 44329673 IC50 = 2000 nM T68251 C07GRS 44329693 IC50 = 60 nM T68251 CBH16R 44329694 IC50 = 600 nM T68251 CG3E7A 44329712 IC50 = 19.95 nM T68251 C9SN6I 44329713 IC50 = 3000 nM T68251 CZ2FW6 44329725 IC50 = 1995.26 nM T68251 CDKI48 44329741 IC50 = 500 nM T68251 CK3M2H 44329742 IC50 = 3000 nM T68251 C39RDS 44329886 IC50 = 50 nM T68251 C3YAF6 44329898 IC50 = 7000 nM T68251 C63RHP 44329909 IC50 = 95.5 nM T68251 CVQA75 44329910 IC50 = 398.11 nM T68251 C84SLI 44329926 IC50 = 100 nM T68251 CJS6B1 44329927 IC50 = 398.11 nM T68251 C2K6OU 44329943 IC50 = 95.5 nM T68251 C5BYR4 44329998 IC50 = 3400 nM T68251 C0SMC9 44330092 IC50 = 21 nM T68251 C35SIO 44330094 IC50 = 12.88 nM T68251 C3NM2G 44330095 IC50 = 0.7943 nM T68251 C6SCU5 44330119 IC50 = 0.26 nM T68251 C69KPL 44330130 IC50 = 109.65 nM T68251 C9P6ZF 44330131 IC50 = 10 nM T68251 C9R1ZE 44330132 IC50 = 55000 nM T68251 CKS01F 44330133 IC50 = 2187.76 nM T68251 CLU8I7 44330135 IC50 = 7000 nM T68251 C1IE0S 44330147 IC50 > 100000 nM T68251 CPG7N2 44330149 IC50 = 15000 nM T68251 CYP6S4 44330152 IC50 = 6000 nM T68251 CMGA28 44330163 IC50 = 41000 nM T68251 CXI49L 44330197 IC50 = 4000 nM T68251 CDQM84 44330198 IC50 = 0.048 nM T68251 CH6EN4 44330225 IC50 = 3388.44 nM T68251 C3GA9Q 44330226 IC50 = 0.23 nM T68251 CG2Q8W 44332306 IC50 = 36 nM T68251 C5NG0R 44334948 IC50 = 30 nM T68251 CFP3X8 44334949 IC50 = 53 nM T68251 CV5RF0 44334963 IC50 = 441 nM T68251 C4AOZ7 44334981 IC50 = 143 nM T68251 CXW59C 44334982 IC50 = 4.6 nM T68251 CCH1W8 44334983 IC50 = 2.5 nM T68251 CQ0UI1 44335017 IC50 = 32 nM T68251 CX58SB 44335240 IC50 = 1.64 nM T68251 CA96JG 44335285 IC50 = 15.4 nM T68251 CI5X0G 44339523 IC50 = 7.2 nM T68251 CB9K8T 44339536 IC50 = 9.5 nM T68251 C2R3XN 44339554 IC50 = 6.5 nM T68251 C2CRY1 44339556 IC50 = 8.6 nM T68251 CTBU53 44339564 IC50 = 23 nM T68251 C58OSK 44339567 IC50 = 7.2 nM T68251 CX2KJ3 44339574 IC50 = 110 nM T68251 CEK3G0 44339588 IC50 = 8.5 nM T68251 C7ZR6H 44339589 IC50 = 1100 nM T68251 C0WP9C 44339590 IC50 = 2.7 nM T68251 C5C2LI 44339654 IC50 = 1 nM T68251 CLD2P9 44339900 Ki = 4400 nM T68251 C2D6VN 44339918 Ki = 2.1 nM T68251 CRQJ09 44339936 Ki = 1300 nM T68251 C4JLG8 44340091 Ki = 6.1 nM T68251 CXW34P 44340094 Ki = 19 nM T68251 CGV94P 44340160 Ki = 7.3 nM T68251 C3IS1O 44340161 Ki = 130 nM T68251 CPK5W0 44340172 Ki = 26 nM T68251 CJ4Z9W 44340207 Ki = 570 nM T68251 CZ31VY 44340208 Ki = 12 nM T68251 C4B9QZ 44340327 Ki = 20 nM T68251 C2XY8H 44340328 Ki = 2.1 nM T68251 CAT48Z 44340657 Ki = 20 nM T68251 C3CYZ8 44340673 Ki = 1100 nM T68251 CRI8Q4 44340696 Ki = 1100 nM T68251 CF1QZ3 44340718 Ki = 70 nM T68251 C09ILT 44340727 Ki = 120 nM T68251 C6AS8J 44340740 Ki = 570 nM T68251 CL0U9T 44340810 Ki = 60 nM T68251 CV6W7Z 44340812 Ki = 770 nM T68251 C3WZM0 44340828 Ki = 2300 nM T68251 CW53EF 44340868 Ki = 350 nM T68251 C6ZDV3 44340869 Ki = 120 nM T68251 CR1ID4 44340923 Ki = 110 nM T68251 CL9I4M 44341538 Ki = 1533 nM T68251 CE3MT4 44341611 Ki = 4650 nM T68251 CJTZ45 44341652 Ki = 200000 nM T68251 C2XP4N 44342352 Ki = 3000 nM T68251 C2SZB1 44342614 IC50 = 6 nM T68251 CTQ6P4 44344631 IC50 = 34200 nM T68251 CBH9I5 44344658 IC50 = 750 nM T68251 CCF94Z 44349787 IC50 = 572 nM T68251 C1L2GF 44350073 IC50 = 20 nM T68251 CQ5RN6 44350101 IC50 = 130 nM T68251 CE2X3Q 44350116 IC50 > 100 nM T68251 CO9R4W 44356376 Ki > 3333 nM T68251 C3MZA1 44356386 Ki > 3333 nM T68251 CH1E2S 44356406 Ki > 3333 nM T68251 C84LUM 44356631 Ki > 3333 nM T68251 CG6T9A 44356632 Ki > 3333 nM T68251 C3WFH7 44356634 Ki > 3333 nM T68251 CB8KY4 44356635 Ki > 3333 nM T68251 COIA82 44356636 Ki > 3333 nM T68251 C4BU6T 44356644 Ki > 3333 nM T68251 CH9YT4 44356659 Ki > 3333 nM T68251 C68LMR 44356675 Ki > 3333 nM T68251 C69YIP 44356686 Ki > 3333 nM T68251 CT05XN 44356687 Ki 1079 nM T68251 CML03W 44356689 Ki > 3333 nM T68251 CQ4NP5 44356690 Ki > 3333 nM T68251 CE8U2Y 44356714 Ki > 3333 nM T68251 CCY5U3 44356804 Ki = 200 nM T68251 C27LMU 44356852 Ki > 3333 nM T68251 CTU64D 44356889 Ki > 3333 nM T68251 C4TM1I 44356890 Ki > 3333 nM T68251 C1WA4B 44356906 Ki > 3333 nM T68251 C50ELY 44356907 Ki 675 nM T68251 CVU8L2 44356924 Ki > 3333 nM T68251 CD1GW2 44356953 Ki > 1011 nM T68251 CR41QN 44356969 Ki > 2454 nM T68251 C3BT0N 44356971 Ki = 642 nM T68251 C81OIZ 44356983 Ki > 3333 nM T68251 CHNC03 44356993 Ki > 3333 nM T68251 C9Z3RT 44356998 Ki > 3333 nM T68251 CR4A7G 44356999 Ki = 476 nM T68251 C2VS6P 44357000 Ki = 1537 nM T68251 CES1G8 44357007 Ki > 3333 nM T68251 C6NQ7K 44357012 Ki = 656 nM T68251 C2HIN3 44357023 Ki > 3333 nM T68251 CI4JO7 44357024 Ki 585 nM T68251 CW4VQ3 44357029 Ki > 3333 nM T68251 C2AIT6 44357209 Ki > 3333 nM T68251 CJK2P7 44357220 Ki > 3333 nM T68251 CIX6G5 44357225 Ki > 3333 nM T68251 CT4C6P 44360260 IC50 = 4.2 nM T68251 CY5I3O 44360286 IC50 = 35 nM T68251 C40OCB 44360287 IC50 = 1.8 nM T68251 C3IW9L 44360784 IC50 = 1.4 nM T68251 CGQ92A 44364037 IC50 = 33 nM T68251 C36YLM 44364111 IC50 = 150 nM T68251 CN4T7Q 44364119 IC50 = 76 nM T68251 CH4TE7 44364121 IC50 = 24 nM T68251 CPE91Y 44364122 IC50 = 18 nM T68251 CG2X0C 44364224 IC50 = 430 nM T68251 C1F8XN 44364249 IC50 = 26 nM T68251 CWM47H 44364250 IC50 = 27 nM T68251 C0W5TL 44364251 IC50 = 1099 nM T68251 C3TPO7 44364266 IC50 = 853 nM T68251 CJ2B8F 44364280 IC50 = 724 nM T68251 C90CYD 44367175 IC50 = 4 nM T68251 C2DV0R 44367276 IC50 = 0.5 nM T68251 C5BAW2 44367284 IC50 < 0.4 nM T68251 C2YG5E 44367285 IC50 = 11 nM T68251 CUDF82 44367309 IC50 = 1 nM T68251 CA0CJ1 44368580 IC50 = 25.7 nM T68251 CW0Y3K 44368632 IC50 = 30 nM T68251 CU8FD2 44368650 IC50 = 109.65 nM T68251 CLE71V 44368654 IC50 = 15.14 nM T68251 CQ27XL 44368655 IC50 = 3.388 nM T68251 CH9G3O 44368849 IC50 = 1 nM T68251 CV6ZG4 44368850 IC50 = 1.288 nM T68251 CB2U9G 44368858 IC50 = 270 nM T68251 CN78UB 44368864 IC50 = 5.754 nM T68251 CV8ZA4 44368865 IC50 = 1.585 nM T68251 CW8O3S 44368924 IC50 = 50.12 nM T68251 C6CD9A 44368928 IC50 = 280 nM T68251 C5HF6P 44368940 IC50 = 330 nM T68251 CE30XV 44368941 IC50 = 50 nM T68251 CG2P9T 44368942 IC50 = 83.18 nM T68251 C7HT1U 44368944 IC50 = 3467.37 nM T68251 C1CW5A 44368946 IC50 = 6165.95 nM T68251 CV86QS 44368963 IC50 = 331.13 nM T68251 C4C7UJ 44368968 IC50 = 38 nM T68251 C3EW6B 44368969 IC50 = 416.87 nM T68251 C4I6ME 44368970 IC50 = 61 nM T68251 C8IZC4 44369030 IC50 = 2430 nM T68251 CDW8V9 44369031 IC50 = 6.4 nM T68251 C82BOI 44369038 IC50 = 776.25 nM T68251 C65FBJ 44369041 IC50 = 53.7 nM T68251 CI0S2R 44369094 IC50 = 310 nM T68251 CFI10T 44369095 IC50 = 34 nM T68251 CQGM80 44369096 IC50 = 210 nM T68251 CIR84S 44369104 IC50 = 920 nM T68251 C6SBW5 44369107 IC50 = 100 nM T68251 CAF5P0 44369163 IC50 = 52000 nM T68251 CHC71X 44369164 IC50 = 1700 nM T68251 CY5L0D 44369186 IC50 = 1 nM T68251 C1JZK6 44369209 IC50 = 86 nM T68251 C9BAO2 44369213 IC50 = 6800 nM T68251 CCJ63B 44369214 IC50 = 11 nM T68251 C4E7DM 44369266 IC50 = 41 nM T68251 CI0ZD9 44371783 IC50 = 20 nM T68251 C4VR5M 44371799 IC50 = 251 nM T68251 C4FHG7 44371800 IC50 = 38 nM T68251 CQ5UR4 44372530 IC50 = 240 nM T68251 CCZ6J3 44379232 Ki = 470 nM T68251 CW20ML 44379249 Ki = 110 nM T68251 CXM06G 44379250 Ki = 5.7 nM T68251 CK0B1D 44379273 Ki = 220 nM T68251 COD6P1 44379499 Ki = 2.6 nM T68251 C84YPO 44379547 Ki > 1000 nM T68251 C3EV2A 44384940 IC50 = 530 nM T68251 C0XE8K 44384941 IC50 = 13000 nM T68251 C3IJO9 44384994 IC50 > 50000 nM T68251 CZ6PU7 44389401 Ki = 1.8 nM T68251 CO4W0Y 44389552 Ki = 0.4 nM T68251 CWQ19I 44389560 IC50 = 10.3 nM T68251 C5R4EW 44389591 IC50 = 935 nM T68251 CC7QW9 44391352 IC50 = 21 nM T68251 C89FTQ 44393434 Ki > 3300 nM T68251 CCO3S9 44393444 Ki > 3300 nM T68251 CNO4P6 44393516 Ki > 3300 nM T68251 C5OIK4 44393520 Ki > 3300 nM T68251 C80NZE 44394179 Ki > 3300 nM T68251 CXD05N 44394645 Ki > 100000 nM T68251 CGQ98X 44394681 Ki = 153000 nM T68251 C8MY4S 44394703 Ki = 88000 nM T68251 CCEI41 44394814 Ki > 2000000 nM T68251 CCZ09V 44394886 Ki > 100000 nM T68251 CZB81D 44395506 IC50 = 5 nM T68251 CAU5R4 44397021 IC50 = 23.3 nM T68251 CQR73V 44397047 IC50 = 27.8 nM T68251 CSO92L 44397377 IC50 = 1.9 nM T68251 CMWU78 44397457 IC50 = 19 nM T68251 CU1E2Z 44397536 IC50 = 14 nM T68251 CQ1Y4E 44397568 IC50 = 4 nM T68251 C12MNT 44397632 IC50 = 2 nM T68251 CZ45GV 44397680 IC50 = 12.1 nM T68251 C7Y1VK 44397699 IC50 = 3.9 nM T68251 CHL9S2 44399294 Ki = 2530 nM T68251 CD49UI 44399312 Ki = 600 nM T68251 C3LS8N 44399509 Ki = 3330 nM T68251 CIA8T3 44399555 Ki > 3330 nM T68251 C8PR7S 44400182 IC50 = 9 nM T68251 CQ9F0K 44400232 IC50 = 9 nM T68251 C91POV 44402021 IC50 = 197 nM T68251 CYCJ78 44402280 IC50 = 9.8 nM T68251 CWG3M4 44402281 IC50 > 10000 nM T68251 C9KGL0 44404474 IC50 = 0.91 nM T68251 C92KDG 44404475 IC50 = 7.1 nM T68251 C07CGB 44404477 IC50 = 1050 nM T68251 C7VH3G 44404484 IC50 = 259 nM T68251 CC29XL 44404490 IC50 = 1770 nM T68251 CCN16G 44404500 IC50 = 164 nM T68251 C69GZU 44404501 IC50 = 688 nM T68251 CY6WL5 44404502 IC50 = 1490 nM T68251 CWGQ46 44404503 IC50 = 1610 nM T68251 CLXM58 44404504 IC50 = 2500 nM T68251 C1F9HO 44404506 IC50 = 4340 nM T68251 CLU41O 44404507 IC50 = 7000 nM T68251 C30DKN 44404553 IC50 = 0.04 nM T68251 C0G4MR 44405997 IC50 > 380000 nM T68251 CZ0XC1 44405998 IC50 = 685000 nM T68251 CIC60V 44406452 IC50 = 28 nM T68251 CHM26J 44406652 Ki = 8100 nM T68251 C1K3QM 44406655 IC50 = 20 nM T68251 C6YG5S 44406678 IC50 = 2.6 nM T68251 CB5ZS0 44411587 IC50 = 52 nM T68251 C4Z0BX 44411591 IC50 = 3060 nM T68251 CHV64P 44411592 IC50 = 0.84 nM T68251 CL6IG9 44411599 IC50 = 6.8 nM T68251 C6IKL1 44411602 IC50 = 0.7 nM T68251 CM2UL0 44411603 IC50 = 1.5 nM T68251 CBT4E7 44411614 IC50 = 4 nM T68251 CH8B4W 44411639 IC50 = 1.1 nM T68251 CS74LI 44411640 IC50 = 54 nM T68251 C43HTC 44411693 IC50 = 3 nM T68251 C8HSN2 44411697 IC50 = 1.2 nM T68251 CKQ8P6 44411698 IC50 = 0.74 nM T68251 CVQ82B 44411701 IC50 = 33 nM T68251 C87VNZ 44411702 IC50 = 1.3 nM T68251 C83MTG 44411776 IC50 = 0.98 nM T68251 CT1A8Q 44411815 IC50 = 295 nM T68251 CQLV08 44411816 IC50 = 556 nM T68251 CP16XL 44411819 IC50 = 1.8 nM T68251 C9COT4 44411820 IC50 = 6.5 nM T68251 C3Q8PM 44411822 IC50 = 4.4 nM T68251 CEB0S4 44411823 IC50 = 0.7 nM T68251 CRB85W 44411826 IC50 = 2.3 nM T68251 CV1NO8 44411829 IC50 = 1.7 nM T68251 CPH6V5 44411830 IC50 = 0.62 nM T68251 CRKL06 44411835 IC50 = 145 nM T68251 C0FDM1 44411836 IC50 = 8.6 nM T68251 CUV27I 44411839 IC50 = 19 nM T68251 CD5KV9 44411846 IC50 = 12 nM T68251 C7CU1F 44411852 IC50 = 1.3 nM T68251 CA9OS4 44411865 IC50 = 1.9 nM T68251 CVM7Y3 44413975 IC50 = 49 nM T68251 C4X0GA 44413977 IC50 = 15 nM T68251 CH01EO 44413978 IC50 = 24 nM T68251 CQ8HK9 44413979 IC50 = 553 nM T68251 CBT0P2 44413982 IC50 = 46 nM T68251 CIJ39D 44413983 IC50 = 16 nM T68251 C9BA0V 44413987 IC50 = 111 nM T68251 CE3WP0 44413991 IC50 = 518 nM T68251 CDUI73 44413992 IC50 = 3.1 nM T68251 CH2X6W 44413997 IC50 = 44 nM T68251 CHN85S 44414002 IC50 = 345 nM T68251 C2OJ4B 44414029 IC50 = 302 nM T68251 CT5PC9 44422672 IC50 = 2.3 nM T68251 CS9D5U 44422720 IC50 = 0.39 nM T68251 CNWM05 44422723 IC50 = 1.8 nM T68251 C58LAY 44422724 IC50 = 20 nM T68251 CDQU41 44422736 IC50 = 53 nM T68251 CVUB56 44422737 IC50 = 30 nM T68251 CB8G2W 44422743 IC50 = 24 nM T68251 CFX42T 44422744 IC50 = 980 nM T68251 C9EL7F 44422749 IC50 = 790 nM T68251 CY49HT 44423674 IC50 = 9600 nM T68251 CHI5G1 44423675 IC50 = 1060 nM T68251 CFC3M6 44423676 IC50 = 1500 nM T68251 CO24JF 44423677 IC50 = 5000 nM T68251 C7F9DB 44423678 IC50 = 30000 nM T68251 CJ6GW5 44423679 IC50 = 1980 nM T68251 CUKM29 44423680 IC50 = 2100 nM T68251 C3R0FS 44423681 IC50 = 660 nM T68251 C14DBJ 44423682 IC50 = 730 nM T68251 CU5QV9 44425142 IC50 > 100000 nM T68251 CW8RY1 44425150 IC50 = 5900 nM T68251 C45WZX 44426073 IC50 = 10 ug.mL-1 T68251 CK5H7O 44429877 IC50 = 5000 nM T68251 CQL1X9 44429878 IC50 = 73 nM T68251 C1CYV2 44429879 IC50 = 82 nM T68251 C7AXP9 44429880 IC50 = 58 nM T68251 CXOS97 44429881 IC50 = 11 nM T68251 C2MQ0I 44429882 IC50 = 37 nM T68251 CQ5PT8 44429883 IC50 = 37 nM T68251 CQRO36 44429884 IC50 = 161 nM T68251 CM27YB 44429885 IC50 = 54 nM T68251 C9JH0T 44429886 IC50 = 4 nM T68251 CD2B3T 44429887 IC50 = 62.6 nM T68251 C6V1CO 44429888 IC50 = 2058 nM T68251 CBC6W4 44429889 IC50 = 40 nM T68251 C7A0LF 44429890 IC50 = 176 nM T68251 CS0M3L 44429891 IC50 = 99.5 nM T68251 CX93QY 44429892 IC50 = 19 nM T68251 C7SWV1 44429893 IC50 = 33 nM T68251 C8QKS0 44429894 IC50 = 22 nM T68251 CBS47K 44429896 IC50 = 32 nM T68251 CI7TG1 44429897 IC50 = 61.3 nM T68251 CLJ48T 44429898 IC50 = 51 nM T68251 C3F9CK 44429899 IC50 = 51 nM T68251 C8PVF7 44429900 IC50 = 31 nM T68251 C6U0TK 44429901 IC50 = 20 nM T68251 CBK9M5 44429902 IC50 = 58 nM T68251 C72YFT 44429903 IC50 = 172 nM T68251 CMO9Q3 44429905 IC50 = 183 nM T68251 C8BHL5 44431844 IC50 > 2000 nM T68251 CR1DN9 44431845 IC50 > 2000 nM T68251 CHFB16 44431846 IC50 > 2000 nM T68251 C0C3ZT 44431847 IC50 > 2000 nM T68251 CS49GV 44431848 IC50 > 2000 nM T68251 C4AVK5 44431849 IC50 > 2000 nM T68251 C5DH4Q 44431850 IC50 > 2000 nM T68251 CLHE45 44431851 IC50 > 2000 nM T68251 CYG29L 44431852 IC50 > 2000 nM T68251 C4OF5L 44431853 IC50 > 2000 nM T68251 CWU7G8 44434565 IC50 = 123 nM T68251 CF9HU5 44434566 IC50 = 280 nM T68251 CV3M6F 44434578 IC50 = 120 nM T68251 CJN1K9 44439853 Ki = 20 nM T68251 C71IPQ 44439982 IC50 = 4000 nM T68251 C2WJP3 44439983 IC50 = 4400 nM T68251 CU9Z1H 44439984 IC50 = 1000 nM T68251 C0G4AS 44439985 IC50 = 3800 nM T68251 CV8D9L 44439986 IC50 = 4300 nM T68251 CKP8T1 44439987 IC50 = 2200 nM T68251 CUT86C 44439988 IC50 = 1200 nM T68251 CKC81R 44439990 IC50 = 1200 nM T68251 CPNM45 44439991 IC50 = 600 nM T68251 CROG92 44439992 IC50 = 300 nM T68251 C30RNZ 44439993 IC50 = 1200 nM T68251 C19MPB 44439994 IC50 = 13000 nM T68251 C2N1UC 44439995 IC50 = 1400 nM T68251 C4T0AW 44439996 IC50 = 1800 nM T68251 CJT4H2 44439997 IC50 = 1300 nM T68251 CYM08I 44439998 IC50 = 1700 nM T68251 C83KQO 44439999 IC50 = 15600 nM T68251 C4Y9JD 44440000 IC50 = 500 nM T68251 C5PWG9 44440001 IC50 = 10600 nM T68251 C70MGQ 44440455 Ki > 3333 nM T68251 CDY53F 44440460 Ki > 3333 nM T68251 CTB9P6 44440461 Ki = 307 nM T68251 C63RLK 44440462 Ki > 3333 nM T68251 C23JBO 44440463 Ki > 3333 nM T68251 CT9P3Y 44440464 Ki > 3333 nM T68251 CX32AM 44440465 Ki > 3333 nM T68251 C6FOC7 44440466 Ki > 3333 nM T68251 CMPX37 44440467 Ki > 3333 nM T68251 CV4F6Z 44440468 Ki > 3333 nM T68251 C6K8VB 44440469 Ki > 3333 nM T68251 C4Y0UM 44440470 Ki > 3333 nM T68251 CHU49A 44440471 Ki > 3333 nM T68251 C8OI4L 44440472 Ki > 3333 nM T68251 CV58YW 44441018 Ki > 3333 nM T68251 CV85PN 44441019 Ki > 3333 nM T68251 C5O2WK 44441020 Ki > 3333 nM T68251 CU67WS 44441021 Ki > 3333 nM T68251 CXZ53B 44441022 Ki > 3333 nM T68251 C8S7UT 44441023 Ki > 3333 nM T68251 CT4PZ9 44441024 Ki > 3333 nM T68251 CU9GE6 44441025 Ki > 3333 nM T68251 CB2IT4 44441026 Ki > 3333 nM T68251 CN4X2F 44441027 Ki > 3333 nM T68251 CPF45Y 44441028 Ki > 3333 nM T68251 CAM23N 44441029 Ki > 3333 nM T68251 C23BPG 44441030 Ki > 3333 nM T68251 C5YMT6 44441031 Ki > 3333 nM T68251 C9A6GJ 44441032 Ki > 3333 nM T68251 CYSU19 44441033 Ki > 3333 nM T68251 CB9P0C 44442303 IC50 = 870 nM T68251 C7HO0Y 44442304 IC50 = 1630 nM T68251 CAR3S2 44442305 IC50 = 960 nM T68251 CZK0A9 44442306 IC50 = 2230 nM T68251 C71MCV 44442307 IC50 = 840 nM T68251 CN70HO 44442308 IC50 = 520 nM T68251 CVE5P0 44442309 IC50 = 1110 nM T68251 C3PT7N 44442310 IC50 = 840 nM T68251 CGS18B 44442311 IC50 = 1620 nM T68251 CIZL27 44442312 IC50 = 760 nM T68251 CCFV76 44442313 IC50 = 700 nM T68251 C4HYM6 44442314 IC50 = 260 nM T68251 CZ2PE6 44442315 IC50 = 1030 nM T68251 C3I7RG 44442317 IC50 = 2570 nM T68251 CGR6E7 44442318 IC50 = 1230 nM T68251 C97ZHM 44442319 IC50 = 1450 nM T68251 C3DIB8 44442320 IC50 = 1000 nM T68251 C0HX1L 44445199 IC50 = 67000 nM T68251 CPQT35 44445200 IC50 = 66000 nM T68251 C2X6IP 44445201 IC50 = 72000 nM T68251 CSRB79 44445202 IC50 = 70000 nM T68251 C2O6KZ 44445203 IC50 = 101000 nM T68251 CASF34 44445204 IC50 = 65000 nM T68251 CQZ6M0 44445205 IC50 = 69000 nM T68251 CH7Z5M 44445206 IC50 = 73000 nM T68251 C71CPO 44445207 IC50 > 150 nM T68251 CO9QA4 44445209 IC50 = 70000 nM T68251 CH3UQ5 44445210 IC50 = 110000 nM T68251 C6B4LG 44445211 IC50 > 150 nM T68251 C1WA5N 44445212 IC50 = 90000 nM T68251 CM2CD0 44445213 IC50 = 71000 nM T68251 C6ZX2P 44445214 IC50 = 70000 nM T68251 C9KE8P 44445215 IC50 = 71000 nM T68251 C68QEF 44445216 IC50 = 66000 nM T68251 CCK7W2 44445217 IC50 = 70000 nM T68251 C58BQA 44445218 IC50 = 69000 nM T68251 C4CGN2 44445219 IC50 = 39000 nM T68251 C1IVR6 44445220 IC50 = 86000 nM T68251 CG2U7H 44445221 IC50 = 64000 nM T68251 CVW48J 44445222 IC50 = 69000 nM T68251 CL3HZ8 44445223 IC50 = 69000 nM T68251 CPY73U 44445224 IC50 = 57000 nM T68251 C9MA2F 44445225 IC50 = 68000 nM T68251 C9SJM3 44445226 IC50 = 107000 nM T68251 CH91WG 44445228 IC50 = 90000 nM T68251 CO59HI 44445229 IC50 = 109000 nM T68251 C62WPE 44445230 IC50 = 125000 nM T68251 COIR35 44445231 IC50 = 107000 nM T68251 CBH0M7 44445233 IC50 = 33000 nM T68251 CIS7M5 44445234 IC50 > 150 nM T68251 CKN60A 44445235 IC50 = 73000 nM T68251 CP4XL8 44445237 IC50 = 65000 nM T68251 CJA79R 44445239 IC50 = 111000 nM T68251 CA72BI 44445240 IC50 = 103000 nM T68251 CZJB48 44445241 IC50 > 150000 nM T68251 C85EVH 44445242 IC50 > 150000 nM T68251 C9DI7F 44445243 IC50 = 73000 nM T68251 CVLH67 44445244 IC50 = 85000 nM T68251 CIP3X8 44445245 IC50 = 119000 nM T68251 CL1MK6 44445246 IC50 = 100000 nM T68251 C0CX7T 44445247 IC50 = 7000 nM T68251 CEZ2P7 44445248 IC50 = 98000 nM T68251 CL0K9Q 44445249 IC50 = 110000 nM T68251 C9T2SH 44445250 IC50 = 125000 nM T68251 C5EFP9 44445251 IC50 = 90000 nM T68251 CLJ71G 44445252 IC50 = 91000 nM T68251 C8TF3E 44445253 IC50 = 63000 nM T68251 C4CAY7 44445254 IC50 = 124000 nM T68251 CH1LE5 44445255 IC50 = 108000 nM T68251 CLP96W 44445256 IC50 = 66000 nM T68251 CK8S4Z 44445257 IC50 = 79000 nM T68251 C03EJW 44445258 IC50 = 90000 nM T68251 CO9SM5 44445261 IC50 = 96000 nM T68251 C3FX8B 44445262 IC50 = 108000 nM T68251 CZS8N5 44445263 IC50 = 98000 nM T68251 CMW2U6 44445264 IC50 = 100000 nM T68251 CB47AH 44445265 IC50 = 110000 nM T68251 CA43LS 44445266 IC50 = 42000 nM T68251 C23MDF 44445267 IC50 = 46000 nM T68251 C9K3DI 44445268 IC50 = 93000 nM T68251 C2ZAK4 44445269 IC50 = 77000 nM T68251 CIVC64 44445270 IC50 = 85000 nM T68251 C8W1HX 44445271 IC50 > 150000 nM T68251 CTFR27 44445272 IC50 > 150000 nM T68251 C20DNO 44445273 IC50 > 150000 nM T68251 CWLC15 44445274 IC50 > 150000 nM T68251 CZD5M3 44445275 IC50 > 150000 nM T68251 CJET46 44445276 IC50 > 150000 nM T68251 CI58AM 44445277 IC50 = 149000 nM T68251 CDN37V 44445278 IC50 > 150000 nM T68251 CE36AB 44445279 IC50 > 150000 nM T68251 CV9KX5 44445280 IC50 > 150000 nM T68251 C4S2WX 44445281 IC50 > 150000 nM T68251 C0HXS4 44445391 IC50 = 620 nM T68251 CT1CP7 44445392 IC50 = 4380 nM T68251 CRNK10 44445393 IC50 = 3080 nM T68251 CF0LR3 44445394 IC50 = 776 nM T68251 C9WQ8E 44445790 IC50 = 3.388 nM T68251 CEGL68 44445796 IC50 = 3981.07 nM T68251 CH2Y7W 44445813 Ki = 2.1 nM T68251 C4J2QM 44445814 Ki = 6.1 nM T68251 CP5H1Q 44446267 IC50 = 6 nM T68251 C30TQK 44446273 IC50 = 1470 nM T68251 CB76CO 44446275 IC50 = 860 nM T68251 C20HIJ 44446753 IC50 = 13 nM T68251 C9CS8E 44446754 IC50 = 21 nM T68251 C4Z7IQ 44446755 IC50 = 50 nM T68251 C4K5QT 44446756 IC50 = 1100 nM T68251 CZEH45 44446757 IC50 = 24 nM T68251 C47SRV 44446758 IC50 = 433 nM T68251 C8CVO1 44446759 IC50 = 2500 nM T68251 C8HM5N 44446763 IC50 = 159 nM T68251 CU5Z4V 44446765 IC50 = 14 nM T68251 C9USL8 44446766 IC50 = 4999 nM T68251 CYO65B 44446797 IC50 = 63 nM T68251 CPI3T0 44446799 IC50 < 5 nM T68251 CGH0A2 44446805 IC50 = 32 nM T68251 CH72RW 44446806 IC50 > 5000 nM T68251 CTKX08 44446807 IC50 = 391 nM T68251 CJ1MP7 44446808 IC50 = 1387 nM T68251 CJN1L7 44446821 IC50 = 39 nM T68251 C4LF6Y 44446822 Ki = 302 nM T68251 C9FG5A 44446823 IC50 = 35 nM T68251 C1P0BV 44446824 IC50 = 37 nM T68251 C5AW3N 44446825 IC50 = 50 nM T68251 C17YSI 44446827 IC50 = 53 nM T68251 C3O8AX 44446835 IC50 = 472 nM T68251 CE2OM1 44446839 IC50 = 106 nM T68251 C49VJF 44446842 IC50 = 86 nM T68251 CF4DL2 44446843 IC50 = 960 nM T68251 C8OS4K 44446845 IC50 > 5000 nM T68251 CIP23G 44447330 IC50 = 10 nM T68251 CPS5M4 44447343 IC50 = 64 nM T68251 CB3F0E 44447344 IC50 = 53 nM T68251 C6WSC7 44447346 IC50 = 52 nM T68251 C6MOB0 44447348 IC50 = 549 nM T68251 CM7JV0 44447353 IC50 = 13 nM T68251 CY2XR5 44447363 IC50 = 1400 nM T68251 CU2BC6 44447364 IC50 > 10000 nM T68251 CXS34M 44447371 IC50 = 262 nM T68251 CD8RX4 44447437 IC50 > 2000 nM T68251 CLNK98 44447442 IC50 > 2000 nM T68251 CA5J9Q 44454525 IC50 > 10000 nM T68251 C6L1OH 44454554 IC50 = 283 nM T68251 CHTY64 44454555 IC50 = 297 nM T68251 CLNM62 44454612 IC50 = 247 nM T68251 CZ2QY4 44454641 IC50 = 344 nM T68251 C7DIB0 44454661 IC50 = 401 nM T68251 CTR91D 44454664 IC50 = 582 nM T68251 CR3PO9 44454741 IC50 = 1262 nM T68251 C1ZSK0 44454742 IC50 = 286 nM T68251 CM8AG1 44454790 IC50 = 2917 nM T68251 CCH42M 44454856 IC50 = 893 nM T68251 CQG09B 44454861 IC50 = 61 nM T68251 CQ5YK3 44454864 IC50 = 73 nM T68251 CLG57Z 44454888 IC50 = 2317 nM T68251 CMEJ96 44454891 IC50 = 147 nM T68251 CV07DO 44455123 IC50 = 4591 nM T68251 C9MHD2 44455124 IC50 = 108.4 nM T68251 C2L1VK 44455161 IC50 = 5.7 nM T68251 C4CZ7N 44455196 IC50 = 4.9 nM T68251 CZ15QG 44455197 IC50 = 104.5 nM T68251 CJ6L1K 44455200 IC50 = 1.7 nM T68251 CLK5O7 44455240 IC50 = 6.1 nM T68251 CSKN69 44455242 IC50 = 5 nM T68251 C3U9VM 44455265 IC50 = 22.4 nM T68251 CG65TZ 44455266 IC50 = 6.5 nM T68251 C14QTI 44455267 IC50 = 41 nM T68251 CSX4F2 44455294 IC50 = 6.1 nM T68251 CJ29BT 44455298 IC50 = 66.4 nM T68251 CCK15P 44455331 IC50 = 66.2 nM T68251 CW8IB7 44455332 IC50 = 662 nM T68251 C9ZXF4 44455360 IC50 = 242 nM T68251 CFB78A 44455363 IC50 > 1000 nM T68251 CW46RV 44455498 Ki = 1500 nM T68251 CXNP45 44455499 Ki = 2733 nM T68251 C6CED5 44455528 Ki > 3333 nM T68251 CUQH30 44455553 Ki = 1700 nM T68251 C83KYJ 44455582 Ki > 3333 nM T68251 CK5N1S 44455612 Ki > 3333 nM T68251 CU2E7V 44455613 Ki > 3333 nM T68251 CH1DI4 44455614 Ki > 3333 nM T68251 CFQ79A 44455647 Ki > 3333 nM T68251 C3J1SV 44455676 IC50 = 36.8 nM T68251 CS6HL1 44455704 IC50 > 1000 nM T68251 CR4EX3 44455706 IC50 > 1000 nM T68251 CC01WS 44455737 IC50 = 377 nM T68251 C0R9SH 44455760 IC50 = 167.5 nM T68251 C6FV2Z 44455783 Ki > 3333 nM T68251 C7W6XV 44455786 IC50 = 72 nM T68251 CO58GJ 44455787 IC50 = 184 nM T68251 CPYV60 44455807 Ki = 2633 nM T68251 CLAT19 44455811 IC50 > 1000 nM T68251 C3TS1X 44455813 IC50 = 10.6 nM T68251 C92AFN 44455816 IC50 = 84.5 nM T68251 CGA0T4 44455829 Ki > 3333 nM T68251 CIR06N 44455835 IC50 = 16.7 nM T68251 C38VBL 44455836 IC50 = 17.2 nM T68251 CKB6E7 44455837 IC50 = 468 nM T68251 CV2B4N 44455858 Ki > 3333 nM T68251 CL6UY9 44455865 IC50 > 1000 nM T68251 CVR58Q 44455879 Ki > 3333 nM T68251 CWZ8K6 44455880 Ki > 3333 nM T68251 CEN93Y 44460382 Ki > 10000 nM T68251 CL30OP 44460588 Ki = 220 nM T68251 C0A1KH 44460605 Ki = 77 nM T68251 CDN1V6 44460606 Ki = 110 nM T68251 CJ6PN3 44460646 Ki = 11 nM T68251 CU8A1O 44460672 Ki = 6100 nM T68251 CIQ87B 44460676 Ki = 4840 nM T68251 C5B8NZ 44460690 Ki = 12 nM T68251 CK4WU2 44460737 Ki = 130 nM T68251 CG0Z7I 44478924 IC50 = 1300 nM T68251 CFO27Y 44478926 IC50 = 230 nM T68251 CBZJ29 44478927 IC50 = 9.7 nM T68251 CRJ24K 44479197 IC50 = 7 nM T68251 CGOH82 44479198 IC50 = 710 nM T68251 CLV56M 44479199 IC50 = 47 nM T68251 CY92OQ 44479458 IC50 = 9900 nM T68251 CH1QG9 44479459 IC50 = 100 nM T68251 CB1NT7 44479460 IC50 = 38 nM T68251 C0JQ9L 44479699 IC50 = 73 nM T68251 C0DN1Q 44479700 IC50 = 58000 nM T68251 CTG24W 44479702 IC50 = 2400 nM T68251 CGZ49M 44479703 IC50 = 190 nM T68251 CAK94X 44563337 IC50 = 193 nM T68251 CSH4K3 44563364 IC50 = 10000 nM T68251 CAF95R 44563365 IC50 = 10000 nM T68251 CO4FQ1 44563366 IC50 = 10000 nM T68251 C6WA3X 44563401 IC50 = 10000 nM T68251 CX5L7N 44563402 IC50 = 24 nM T68251 CJ8V4U 44563403 IC50 = 18 nM T68251 CN2BM4 44563404 IC50 = 100 nM T68251 C3KCV6 44563405 IC50 = 740 nM T68251 CI0R5M 44563465 IC50 = 310 nM T68251 C5IQ9Z 44563466 IC50 = 320 nM T68251 C6ZEW9 44563467 IC50 = 1400 nM T68251 CZ2EL1 44563468 IC50 = 300 nM T68251 CDV6R7 44563469 IC50 = 92 nM T68251 CJ2BU5 44563487 IC50 = 37 nM T68251 CP54WT 44563489 IC50 = 1813 nM T68251 C1UXP6 44563490 IC50 = 310 nM T68251 CZ0W1A 44563491 IC50 = 1273 nM T68251 C37UAM 44563492 IC50 = 65 nM T68251 C4BD0N 44563493 IC50 = 247 nM T68251 CNP6M7 44563494 IC50 = 45 nM T68251 C0J6LB 44563970 IC50 = 2600 nM T68251 CR6NO2 44564180 IC50 = 6 nM T68251 C3US0I 44569010 IC50 = 3200 nM T68251 C3TAN1 44569011 IC50 = 2200 nM T68251 CF0L2W 44569012 IC50 = 50 nM T68251 CGI35S 44569013 IC50 = 200 nM T68251 C8PO5Q 44569024 IC50 = 40 nM T68251 C52JXP 44569036 IC50 = 3500 nM T68251 CU1NI6 44569037 IC50 = 2700 nM T68251 CS9CH4 44569038 IC50 = 40 nM T68251 C63ZQK 44569039 IC50 = 10 nM T68251 C2WE7H 44569040 IC50 = 1300 nM T68251 CO8FB4 44569058 IC50 = 90 nM T68251 C3K4ED 44569059 IC50 = 5200 nM T68251 CPWR76 44569060 IC50 = 1500 nM T68251 CU39FK 44569061 IC50 = 200 nM T68251 CR6H0X 44569062 IC50 = 700 nM T68251 CTWR37 44569063 IC50 = 8900 nM T68251 C6M9SH 44569081 IC50 = 500 nM T68251 C5RN7U 44569082 IC50 = 4 nM T68251 CQ9OA7 44569083 IC50 = 20 nM T68251 C70UVG 44571513 IC50 = 50500 nM T68251 CCV74H 44576563 IC50 = 400 nM T68251 C59TCG 44576564 IC50 = 2000 nM T68251 CMI9S4 44576565 IC50 = 9500 nM T68251 CD8ZI4 44576587 IC50 = 100 nM T68251 CQ87CS 44576614 IC50 = 200 nM T68251 CJY2W3 44576615 IC50 = 300 nM T68251 CL92CH 44576616 IC50 = 200 nM T68251 CIU84E 44576617 IC50 = 1100 nM T68251 C9ODS1 44576618 IC50 = 1500 nM T68251 C35DWL 44576631 IC50 = 6 nM T68251 C6ZL1U 44576632 IC50 = 8 nM T68251 CK09LV 44576633 IC50 = 8 nM T68251 CFL76T 44576634 IC50 = 11 nM T68251 CC58GQ 44576635 IC50 = 12 nM T68251 CPT42K 44580109 IC50 > 5000 nM T68251 CQ7W5I 44580110 Ki > 3000 nM T68251 CWD32S 44580184 IC50 = 664 nM T68251 CQ4ZR1 44580422 IC50 = 750 nM T68251 C0XJ5C 44580496 Ki > 3333 nM T68251 CK68GT 44580539 Ki = 1.37 nM T68251 CXIY57 44580801 Ki > 10000000 nM T68251 C0OA8Y 44580802 Ki > 10000000 nM T68251 CNC4D7 44581071 Ki = 7000000 nM T68251 CDF48U 44581111 Ki > 10000000 nM T68251 C06BRD 44582547 IC50 = 107200 nM T68251 C51VNE 44582548 IC50 = 287300 nM T68251 CLK3R4 44582549 IC50 = 76800 nM T68251 CZTW24 44582550 IC50 = 52800 nM T68251 CP0AJ7 44582568 IC50 = 59900 nM T68251 CCZ07T 44582586 IC50 = 76100 nM T68251 CN58BM 44582588 IC50 = 71200 nM T68251 C3UJ2Q 44582621 IC50 = 659600 nM T68251 C35BEJ 44582622 IC50 = 501500 nM T68251 C3UE5R 44582644 IC50 = 116300 nM T68251 CX1GV0 44582645 IC50 = 71400 nM T68251 C3IU2S 44582646 IC50 = 64300 nM T68251 C63ODU 44582647 IC50 = 120800 nM T68251 C7EAZ1 44582685 IC50 = 235800 nM T68251 CZW4O6 44582686 IC50 = 159100 nM T68251 C3AX6W 44582687 IC50 = 211400 nM T68251 CC0LO7 44582688 IC50 = 283600 nM T68251 CX63IA 44582689 IC50 = 256100 nM T68251 CL73BH 44582717 IC50 = 79600 nM T68251 CY2PM8 44582718 IC50 = 83200 nM T68251 C9EPQ6 44582719 IC50 = 76800 nM T68251 CF1G7I 44582720 IC50 = 101500 nM T68251 C15RUQ 44582746 IC50 = 76500 nM T68251 C3CJD0 44582747 IC50 = 397600 nM T68251 C16RAH 44582748 IC50 = 368100 nM T68251 CQ9XG5 44582769 IC50 = 470600 nM T68251 C7UTR1 44582771 IC50 = 470700 nM T68251 CE2D6Z 44582793 IC50 = 340800 nM T68251 CUR8M1 44582868 IC50 = 55300 nM T68251 CNK9C7 44582869 IC50 = 628000 nM T68251 CX49HN 44582873 IC50 = 369400 nM T68251 C56WPA 44582874 IC50 = 169400 nM T68251 C8TGB1 44582875 IC50 = 114900 nM T68251 CYV0N5 44582876 IC50 = 26100 nM T68251 CR4SF2 44582887 IC50 = 52300 nM T68251 C50OTD 44582888 IC50 = 54400 nM T68251 CDX63O 44582890 IC50 = 33600 nM T68251 C6X0FM 44582904 IC50 = 71200 nM T68251 CY3N7I 44582905 IC50 = 86300 nM T68251 CY4A6F 44582906 IC50 = 108700 nM T68251 CD0J5R 44582907 IC50 = 122400 nM T68251 C2Z4HB 44583600 IC50 = 1277 nM T68251 CD4Q8C 44583601 IC50 = 8 nM T68251 CD2AQ7 44583620 IC50 = 92 nM T68251 CLZ6X5 44583621 IC50 = 81 nM T68251 C5HA4P 44583622 IC50 = 180 nM T68251 C7PR8I 44583623 IC50 = 106 nM T68251 CDRC42 44583654 IC50 = 100 nM T68251 C5HEX6 44583655 IC50 = 1090 nM T68251 CM79HD 44583656 IC50 > 5000 nM T68251 C20FCM 44583672 IC50 > 5000 nM T68251 CLAU98 44586492 IC50 = 8760 nM T68251 CY8X7P 44586493 IC50 = 2930 nM T68251 CDS86C 44586529 IC50 = 3140 nM T68251 COD20L 44586530 IC50 = 12700 nM T68251 C1W2SV 44586531 IC50 = 17800 nM T68251 C5S0OJ 44586532 IC50 = 50500 nM T68251 CB2P7I 44586533 IC50 = 7480 nM T68251 CKRT49 44586578 IC50 = 19200 nM T68251 C8XY1Z 44586579 IC50 = 13100 nM T68251 CE9BZ5 44586580 IC50 = 25500 nM T68251 CXDF71 44586581 IC50 = 14300 nM T68251 COFY06 44586582 IC50 = 8080 nM T68251 CI2PT3 44586626 IC50 = 8000 nM T68251 C4GQ6Y 44586627 IC50 = 12600 nM T68251 CTO94B 44586628 IC50 = 3540 nM T68251 C9Y0CR 44586662 IC50 = 11700 nM T68251 CBV5P8 44586663 IC50 = 32000 nM T68251 C2U0CY 44586664 IC50 = 9940 nM T68251 C1IBA2 44588219 IC50 = 151400 nM T68251 C6XE5V 44588251 IC50 = 771900 nM T68251 C1UW6M 44588252 IC50 = 802300 nM T68251 CXF40R 44588253 IC50 = 78800 nM T68251 CQF2I5 44588254 IC50 = 546800 nM T68251 CBA1Y8 44588279 IC50 > 1000000 nM T68251 C8RI4Q 44591819 IC50 = 30000 nM T68251 C6BXS2 44591880 IC50 = 37700 nM T68251 CM9IN6 44592481 IC50 = 14400 nM T68251 CZNQ90 44593458 IC50 = 9 nM T68251 CR3Q4N 44593532 IC50 = 7100 nM T68251 CH8QS0 44596287 IC50 = 128 nM T68251 CTW7F2 44601281 IC50 = 1.6 nM T68251 CW5A2D 44608129 IC50 = 86 nM T68251 CT7KX5 44608938 IC50 = 96 nM T68251 CJRP30 44608939 IC50 = 458 nM T68251 COI5K3 44608942 IC50 = 706 nM T68251 CS4C5T 44609098 IC50 = 200 nM T68251 CMLV87 44609099 IC50 = 706 nM T68251 C3T9SV 44609100 IC50 = 54 nM T68251 C19LWR 44634267 IC50 = 0.13 nM T68251 CM0I4J 45101511 IC50 = 1475 nM T68251 CZP79X 45268488 IC50 = 379 nM T68251 CK50JB 45268522 IC50 = 8990 nM T68251 C2B0GI 45268787 Ki = 1 nM T68251 CVG5I2 45269378 IC50 = 4000 nM T68251 CQC5Y4 45269386 IC50 = 2840 nM T68251 CACH13 45269631 IC50 = 12 nM T68251 CTOH60 45270200 IC50 = 4410 nM T68251 C2H5IY 45271017 IC50 = 3590 nM T68251 C0YT8W 45271893 IC50 = 1150 nM T68251 CVNO86 45271894 IC50 = 1410 nM T68251 C7OQB3 45271912 IC50 = 2470 nM T68251 C3SWC7 45272759 IC50 = 7500 nM T68251 CH4NL1 45376336 IC50 = 1937.23 nM T68251 C36HRP 45377138 IC50 > 22000 nM T68251 C6B7ZY 45377564 IC50 > 500000 nM T68251 C5HAR6 45377565 IC50 > 20000 nM T68251 CKR0Q8 45377703 IC50 > 24000 nM T68251 C3SQL2 45378250 IC50 = 190 nM T68251 CQE49A 45378251 IC50 = 1.5 nM T68251 CO4AC6 45378252 IC50 = 17 nM T68251 C42FPG 45378253 IC50 = 4.2 nM T68251 CI82BN 45378254 IC50 = 21 nM T68251 C6MY2W 45380188 IC50 = 190 nM T68251 C9P0DG 45380189 IC50 = 29 nM T68251 CRY0E8 45380190 IC50 = 0.7 nM T68251 C0MPH3 45380191 IC50 = 390 nM T68251 CMPE63 45482676 IC50 = 1500 nM T68251 CZS39O 45487302 IC50 = 210 nM T68251 C4ZWY7 45487310 IC50 = 432 nM T68251 C9SV0H 45487311 IC50 = 581 nM T68251 C6GCM7 45487332 IC50 < 5 nM T68251 CCF05Q 45487333 IC50 = 102 nM T68251 C23NRD 45487334 IC50 > 2000 nM T68251 CY09ZU 45487335 IC50 = 344 nM T68251 CQHJ85 45487342 IC50 = 11 nM T68251 C3ZLN1 45487343 IC50 = 12 nM T68251 CI6DW2 45487357 IC50 < 5 nM T68251 COX40Y 45487358 IC50 = 102 nM T68251 CF1T7M 45487359 IC50 = 843 nM T68251 CRXI29 45487373 IC50 > 2000 nM T68251 CYL32E 45487376 IC50 = 235 nM T68251 CO5P9I 45487386 IC50 = 506 nM T68251 CS9Y8G 45487387 IC50 > 2000 nM T68251 CAN4J2 45487388 IC50 = 1662 nM T68251 CWLC18 45487393 IC50 = 471 nM T68251 CO9NJ2 45487398 IC50 = 365 nM T68251 CDN5Q6 45487399 IC50 = 502 nM T68251 CI4KJ5 45487400 IC50 = 613 nM T68251 C49HOI 45487401 IC50 = 730 nM T68251 CBK43U 45487402 IC50 < 5 nM T68251 C56WVI 46184724 Ki > 50000 nM T68251 CMB53L 46212112 IC50 = 159390 nM T68251 CX58KQ 46212114 IC50 = 58220 nM T68251 C9PXD0 46212116 IC50 = 17170 nM T68251 C6KHO2 46212117 IC50 = 36040 nM T68251 C9XGD0 46212861 IC50 = 187410 nM T68251 CLWA85 46228171 IC50 > 1000000 nM T68251 CFQ67J 46228182 IC50 > 1000000 nM T68251 CCV7T2 46228183 IC50 > 1000000 nM T68251 CU2WI8 46228191 IC50 > 1000000 nM T68251 CT6JZ9 46228192 IC50 = 594300 nM T68251 C6H7AB 46228205 IC50 = 999000 nM T68251 CJ9SD0 46228215 IC50 = 447200 nM T68251 C7WS9P 46228222 IC50 > 1000000 nM T68251 C71RSJ 46228223 IC50 > 1000000 nM T68251 CKCE97 46228233 IC50 > 1000000 nM T68251 CWUG47 46228234 IC50 = 324400 nM T68251 CM3YZ1 46228235 IC50 > 1000000 nM T68251 CYUM78 46228241 IC50 > 1000000 nM T68251 C6HCD2 46228242 IC50 > 1000000 nM T68251 C0GX8M 46228245 IC50 > 1000000 nM T68251 C9FM5N 46228246 IC50 = 176500 nM T68251 C4KA1Y 46228247 IC50 > 1000000 nM T68251 C7HIE4 46228248 IC50 = 131000 nM T68251 CQVZ58 46228249 IC50 > 1000000 nM T68251 C5WV8N 46228250 IC50 > 1000000 nM T68251 CR0BP8 46228264 IC50 > 1000000 nM T68251 CGW3Q4 46228265 IC50 > 1000000 nM T68251 CVN7J0 46228266 IC50 = 166600 nM T68251 C51LDC 46228283 IC50 > 1000000 nM T68251 C2JVF4 46228308 IC50 = 196600 nM T68251 C7Z6XB 46228317 IC50 > 1000000 nM T68251 C0S8FV 46231953 IC50 = 400 nM T68251 CN3OS2 46232362 IC50 = 6460800 nM T68251 CF9D2G 46232363 IC50 = 124320 nM T68251 C5GT8X 46232364 IC50 = 624480 nM T68251 C9A8BO 46232365 IC50 = 2000000 nM T68251 CP49KE 46232415 IC50 = 24180 nM T68251 CFZX82 46232416 IC50 = 26170 nM T68251 C3L7VK 46232417 IC50 = 1362800 nM T68251 C4XOU1 46232418 IC50 = 56600 nM T68251 C1S8BQ 46232490 IC50 = 106000 nM T68251 CAV06U 46232491 IC50 = 105300 nM T68251 CVF9D5 46232492 IC50 = 9426500 nM T68251 C18JTQ 46232493 IC50 = 1750000 nM T68251 CFA58J 46232533 IC50 = 2757800 nM T68251 C9C7IE 46232534 IC50 = 11520000 nM T68251 CFU05P 46232535 IC50 = 1920500 nM T68251 CSU81E 46233057 IC50 = 58140 nM T68251 C8SM5H 46233058 IC50 = 30050 nM T68251 C8W7RP 46233059 IC50 = 10490 nM T68251 C3IA9P 46233060 IC50 = 37290 nM T68251 CZ6C8P 46703060 IC50 = 5.97 nM T68251 C0DHL4 46703061 IC50 = 1721.82 nM T68251 CYA45K 46703062 IC50 = 3.55 nM T68251 CY72WL 46703063 IC50 = 5.27 nM T68251 C1YHS2 46703064 IC50 = 1679.56 nM T68251 C8HX7K 46840956 IC50 = 45820 nM T68251 CH0Z1E 46844314 Ki = 1208 nM T68251 C8MR0H 46847340 IC50 = 4000 nM T68251 C20BTY 46856241 Ki = 43600 nM T68251 C0ECU2 46861775 IC50 = 8.95 nM T68251 C0Y9NZ 46861793 IC50 = 8.31 nM T68251 C2S4YC 46866644 IC50 = 15000 nM T68251 C7QR8Y 46866645 IC50 = 10000 nM T68251 CUH07J 46866646 IC50 = 7000 nM T68251 C8GK4C 46866647 IC50 = 4000 nM T68251 C5L8GF 46871738 IC50 = 12.1 nM T68251 CR1KF7 46871739 IC50 = 3.7 nM T68251 C8Q6YR 46871740 IC50 = 5.3 nM T68251 C58YSM 46871741 IC50 = 6000 nM T68251 C3X5EN 46873064 IC50 = 53670 nM T68251 CR96AK 46890762 IC50 > 10000 nM T68251 C5G9FX 46890763 IC50 = 1400 nM T68251 COP78K 46890764 IC50 = 4500 nM T68251 C60QSB 46890765 IC50 = 1600 nM T68251 CQ5P9V 46890766 IC50 = 700 nM T68251 CB90YN 46890767 IC50 = 5600 nM T68251 CUA7L6 46890821 IC50 = 3600 nM T68251 C9BNQ7 46890822 IC50 = 1600 nM T68251 CTF20Y 46890823 IC50 = 1750 nM T68251 CR3QW7 46891107 IC50 = 21.1 nM T68251 C5MK3A 46891108 IC50 = 88 nM T68251 CQ5E1H 46891109 IC50 = 40 nM T68251 C0NW9D 46891110 IC50 = 370 nM T68251 C91LGI 46891170 IC50 = 48.5 nM T68251 CGI5B4 46891171 IC50 = 330 nM T68251 CZPM12 46891172 IC50 = 18.4 nM T68251 C2V6MW 46891173 IC50 = 35 nM T68251 CZWT45 46891207 IC50 = 1400 nM T68251 CFE58Q 46891208 IC50 = 5.4 nM T68251 C8S7QX 46891209 IC50 = 32.6 nM T68251 C5Y0MN 46891255 IC50 = 3700 nM T68251 CJ16SE 46891256 IC50 = 2 nM T68251 C7Y9TE 46891257 IC50 = 82 nM T68251 C7DT6W 46891258 IC50 = 700 nM T68251 CLF7Y4 46891311 IC50 = 900 nM T68251 C2IN7Y 46891312 IC50 = 3100 nM T68251 CNXU57 46891313 IC50 = 70 nM T68251 CJB5D0 46891314 IC50 = 5400 nM T68251 CVK0E5 46891356 IC50 = 500 nM T68251 C89RPO 46891357 IC50 = 505 nM T68251 CVB6K4 46891358 IC50 = 1750 nM T68251 C67WEK 46891359 IC50 = 800 nM T68251 CPQ37V 46891414 IC50 > 10000 nM T68251 C5LTI6 46891459 IC50 = 2900 nM T68251 C92FBL 46891460 IC50 = 2100 nM T68251 C1A0OE 46891522 IC50 = 2100 nM T68251 C2I6FV 46891523 IC50 = 2400 nM T68251 CAZ9Q5 46891524 IC50 = 7300 nM T68251 CG02KB 46891525 IC50 = 1700 nM T68251 C7ZG8J 46891526 IC50 > 10000 nM T68251 CRQ13J 46891580 IC50 = 2500 nM T68251 CERM39 46891581 IC50 = 5500 nM T68251 CN8WF9 46891582 IC50 = 7000 nM T68251 C86RLM 46891583 IC50 = 900 nM T68251 CM7S5T 46891584 IC50 = 6000 nM T68251 CRY18A 46891617 IC50 = 900 nM T68251 C0F7SU 46905989 IC50 = 112000 nM T68251 C49PYF 46907509 IC50 = 8.92 nM T68251 C2U1GW 46907510 IC50 = 9.11 nM T68251 C7MUS8 46907512 IC50 = 1820.53 nM T68251 C71YRF 46907513 IC50 = 1873.02 nM T68251 CVH58U 46907580 IC50 = 8.3 nM T68251 C0S9WB 46919610 Ki = 1900 nM T68251 CXDL74 46927871 IC50 = 8270 nM T68251 CE3H7I 46938726 IC50 < 0.1 nM T68251 C9T0HR 46938727 IC50 < 0.1 nM T68251 C0YR7M 46938728 IC50 < 0.1 nM T68251 C2TE8J 47162079 IC50 = 60000 nM T68251 CC42DK 49863560 IC50 = 129000 nM T68251 C4UWB6 49863561 IC50 = 18500 nM T68251 CMR3B0 49863562 IC50 = 121000 nM T68251 CBE6H5 49863563 IC50 = 127000 nM T68251 CR0I9V 49863564 IC50 = 12000 nM T68251 CD17YP 49863589 IC50 = 272000 nM T68251 CXW4C6 49863590 IC50 = 107000 nM T68251 C1B6ZU 49863591 IC50 = 155000 nM T68251 C0S2OT 49863592 IC50 > 1000000 nM T68251 CT3W2H 49863593 IC50 > 1000000 nM T68251 CG96WY 49863619 IC50 = 22700 nM T68251 CG40UX 49863620 IC50 = 315650 nM T68251 C0IX5P 49863621 IC50 > 1000000 nM T68251 CSC7K2 49863622 IC50 = 141000 nM T68251 C1FLD5 49863915 IC50 = 122000 nM T68251 CL90XE 49863932 IC50 > 1000000 nM T68251 CXZ8Y3 49863933 IC50 = 60400 nM T68251 CKXZ37 49863934 IC50 = 62700 nM T68251 CFD6O0 49863953 IC50 = 71600 nM T68251 C1L6TV 49863954 IC50 = 131000 nM T68251 CEL71O 49863955 IC50 = 46900 nM T68251 CJB0T7 49863956 IC50 = 454000 nM T68251 C7S9QA 50913428 IC50 > 500000 nM T68251 CO4XE9 50913573 IC50 > 500000 nM T68251 C2T1AZ 50925490 IC50 = 3000 nM T68251 CJG7H2 50941564 IC50 = 8800 nM T68251 C5B6SP 50941565 IC50 = 7200 nM T68251 CV4BM3 50941566 IC50 = 10800 nM T68251 C29WVD 50941567 IC50 = 8400 nM T68251 CKN8Z0 50941568 IC50 = 5600 nM T68251 CQ64FL 50941569 IC50 = 3900 nM T68251 CC4V0N 50941747 IC50 = 4300 nM T68251 C7AU4S 50943150 IC50 > 100000 nM T68251 CXF4V3 50990921 IC50 > 6300 nM T68251 CAS94N 51346773 Ki = 390 nM T68251 CP65WT 51346774 Ki = 90 nM T68251 C5OIA2 51346775 Ki = 280 nM T68251 CU2SX3 51355576 Ki > 10000 nM T68251 CQM4E7 52936345 IC50 = 19 ug.mL-1 T68251 CLA96C 53232689 Ki = 400 nM T68251 C3BGW0 53233015 Ki = 20500 nM T68251 CZ06OY 53233469 IC50 = 360 nM T68251 CMQZ70 53242178 IC50 > 23000 nM T68251 CC9HK5 53245646 IC50 = 6309.57 nM T68251 CRI92N 53311230 IC50 > 10000 nM T68251 C74CKF 53318123 Ki = 61 nM T68251 C47DIU 53318911 IC50 = 120 nM T68251 CC6DR2 53318912 IC50 = 4200 nM T68251 C7V1NC 53320225 IC50 = 350 nM T68251 CVH2B7 53320226 IC50 = 2800 nM T68251 CO8QK2 53320227 IC50 = 180 nM T68251 CNS3F2 53321542 IC50 = 1900 nM T68251 C4UE6R 53322469 IC50 = 30000 nM T68251 C1N2BX 53322876 IC50 = 1700 nM T68251 CSYW40 53322877 IC50 = 35000 nM T68251 CGUC59 53322878 IC50 = 2400 nM T68251 C3QHA6 53322879 IC50 = 2200 nM T68251 CI3WL5 53323418 Ki = 240 nM T68251 C0H7FQ 53324260 IC50 = 26000 nM T68251 CU7YG9 53325497 IC50 = 170 nM T68251 C4G1HK 53325498 IC50 > 9100 nM T68251 CO5L1I 53325499 IC50 = 12000 nM T68251 CZA03W 53326760 IC50 = 530 nM T68251 CM53CG 53326761 IC50 = 2500 nM T68251 CWR6T4 53326860 IC50 = 500 nM T68251 CPY02U 53327890 IC50 = 2.3 nM T68251 CPGE80 53327891 IC50 = 6 nM T68251 CLJ4G2 53328858 IC50 = 1.5 nM T68251 C4G3QL 53328859 IC50 = 2.5 nM T68251 CX1TW0 53328860 IC50 = 1.3 nM T68251 C0ZX5G 53329215 IC50 = 4 nM T68251 CSU52A 53329216 IC50 = 17 nM T68251 CHF62Q 53361485 IC50 = 140 nM T68251 CJ3F4R 53361486 IC50 = 37 nM T68251 C6Y2EV 53374826 IC50 > 100000 nM T68251 CNY03Z 53378637 Ki = 440 nM T68251 CX3DU4 53378973 Ki = 390 nM T68251 CTD1H9 53378974 Ki = 240 nM T68251 CQ04KO 53389286 IC50 = 384 nM T68251 C1IFJ8 53957122 IC50 = 210000 nM T68251 CTJ48R 54185618 IC50 = 17800 nM T68251 C24SIM 54334252 IC50 = 39 nM T68251 CSUW40 54352406 IC50 = 10 nM T68251 C7RC3A 54371779 IC50 = 10 nM T68251 C3M8GZ 54580051 IC50 = 61000 nM T68251 CL0WM9 54580052 IC50 > 10000 nM T68251 CK26XF 54580053 IC50 > 10000 nM T68251 C3LF0P 54580544 Ki = 9200 nM T68251 CA8U9V 54580837 IC50 = 4000 nM T68251 CVO09J 54581546 Ki = 110 nM T68251 CWB2Q6 54581896 IC50 = 170 nM T68251 CVK72M 54582073 IC50 = 1300 nM T68251 CBK18O 54582074 IC50 > 10000 nM T68251 CP2F1B 54582075 IC50 > 10000 nM T68251 CZNU23 54582076 IC50 > 10000 nM T68251 C0U5HZ 54582077 IC50 > 10000 nM T68251 C8SG9Y 54582079 IC50 > 10000 nM T68251 CZI6S3 54582080 IC50 = 3500 nM T68251 CD09BZ 54582543 IC50 = 1300 nM T68251 CH6Q2Z 54583016 IC50 > 10000 nM T68251 C3V9LQ 54583017 IC50 = 150 nM T68251 CT80KQ 54583018 IC50 = 620 nM T68251 CPT4L5 54583019 IC50 > 10000 nM T68251 CK52YD 54583511 Ki = 530 nM T68251 CF0SK8 54583712 IC50 = 2.5 nM T68251 CBEV27 54584024 IC50 = 3300 nM T68251 CM87DP 54584025 IC50 = 1100 nM T68251 C28GKQ 54585927 IC50 > 10000 nM T68251 CAZ76E 54586892 IC50 > 10000 nM T68251 CM0OQ3 54586893 IC50 > 10000 nM T68251 CK1NS7 54586894 IC50 > 10000 nM T68251 CMC4Y1 54586895 IC50 > 10000 nM T68251 C2MKX5 54586896 IC50 = 3800 nM T68251 CU91QP 54586897 IC50 > 10000 nM T68251 CI08RQ 54586898 IC50 = 1400 nM T68251 C6PRI4 54586899 IC50 = 7600 nM T68251 CG37UX 54587429 Ki = 430 nM T68251 CL9SC3 54587769 Ki > 40000 nM T68251 C13FSJ 54669762 Ki = 24 nM T68251 CHS01Z 54669766 Ki = 520 nM T68251 C8YLA4 54669829 IC50 = 7.5 nM T68251 C1KA8X 54669830 IC50 = 2.55 nM T68251 CZA6Q9 54669831 IC50 = 24 nM T68251 CF23NJ 54669841 IC50 = 23 nM T68251 C71KLJ 54679182 IC50 = 1260 nM T68251 CC67RV 54681831 IC50 = 610 nM T68251 C83NUI 54687474 IC50 = 9300 nM T68251 CZ6V0U 54724681 IC50 > 50000 nM T68251 CJ6HT4 54726662 IC50 = 19000 nM T68251 C9P5ES 54752445 IC50 = 0.39 nM T68251 C0HKC9 54752446 IC50 = 0.57 nM T68251 C6D9IE 54753443 IC50 = 1729.19 nM T68251 CLP2C1 54753981 IC50 = 393140 nM T68251 CQD2Z6 54757100 IC50 = 63.6 nM T68251 C7E9SG 54757202 Ki = 78000 nM T68251 CMJ90D 54757404 Ki = 62 nM T68251 CD1A3F 54757406 Ki = 69 nM T68251 C4EFI5 54757409 Ki = 420 nM T68251 C5D1TI 56649332 IC50 = 1.8 nM T68251 CGTV56 56658262 IC50 = 151600 nM T68251 C9Z4TW 56658263 IC50 = 110100 nM T68251 CAV9S4 56658410 IC50 = 42200 nM T68251 CLKA98 56659256 IC50 = 73 nM T68251 CAFN81 56659257 IC50 = 269 nM T68251 C5ATG7 56659258 IC50 = 95 nM T68251 CR0HX7 56659259 IC50 = 25 nM T68251 CI8RY0 56659946 IC50 = 249240 nM T68251 C0NK1P 56659952 IC50 = 307270 nM T68251 CL6GF3 56659954 IC50 = 166110 nM T68251 CP5K7G 56661758 IC50 = 100100 nM T68251 C1EW4P 56661759 IC50 = 105600 nM T68251 C5FR4E 56661895 IC50 = 119500 nM T68251 CG7E1O 56662736 IC50 = 13 nM T68251 CZF86Q 56662737 IC50 = 264 nM T68251 CT2G8L 56662738 IC50 = 24 nM T68251 C3LQY5 56662739 IC50 = 31 nM T68251 CQY15M 56663413 IC50 = 463380 nM T68251 CWM2L3 56663417 IC50 = 836490 nM T68251 C48JHP 56663421 IC50 = 267730 nM T68251 CIG9J2 56663694 IC50 = 1021 nM T68251 C8YPU6 56665194 IC50 = 84300 nM T68251 CV46HL 56665195 IC50 = 173100 nM T68251 C3L5SO 56665196 IC50 = 108900 nM T68251 CH4M6V 56665197 IC50 = 40600 nM T68251 C20IZG 56665371 IC50 > 1000000 nM T68251 C8ZD7Q 56666204 IC50 = 45 nM T68251 CKB12J 56666205 IC50 = 54 nM T68251 CR21IL 56666206 IC50 = 100 nM T68251 CT65HD 56666207 IC50 = 311 nM T68251 C2IVE9 56666208 IC50 = 706 nM T68251 CPM8U1 56666842 IC50 = 540030 nM T68251 CC8HS0 56669604 IC50 = 9.8 nM T68251 CLO80F 56669605 IC50 = 60 nM T68251 CPS48C 56669606 IC50 = 329 nM T68251 CGMF96 56669607 IC50 = 47 nM T68251 CG0N1D 56670269 IC50 = 251910 nM T68251 CD1UX2 56670273 IC50 = 276440 nM T68251 C6O4TD 56672133 IC50 > 1000000 nM T68251 CRZF93 56672134 IC50 = 157400 nM T68251 C5C3OA 56672135 IC50 = 149200 nM T68251 CSU81T 56672275 IC50 = 133800 nM T68251 CBX8M4 56673120 IC50 = 15 nM T68251 C6Z7VA 56673121 IC50 = 86 nM T68251 C2YJZ8 56673122 IC50 = 2.9 nM T68251 C3BD9S 56673123 IC50 = 264 nM T68251 CG10FP 56673124 IC50 = 681 nM T68251 CMNQ68 56673125 IC50 = 20 nM T68251 CY80GQ 56673788 IC50 = 656770 nM T68251 C8C3QL 56675664 IC50 = 111300 nM T68251 CWI28X 56676443 IC50 = 16 nM T68251 CSPX53 56676444 IC50 = 22 nM T68251 CJU1M7 56676445 IC50 = 16 nM T68251 CGD90C 56676446 IC50 = 268 nM T68251 CCA39I 56676447 IC50 = 83 nM T68251 CL67JD 56677116 IC50 = 516830 nM T68251 CWH5R6 56677118 IC50 = 939570 nM T68251 CX80RM 56677120 IC50 = 157420 nM T68251 CKLQ67 56678865 IC50 = 67400 nM T68251 C3ZAX6 56678866 IC50 = 44100 nM T68251 C2M1TR 56678867 IC50 = 119300 nM T68251 CNE08Y 56678974 IC50 = 40400 nM T68251 C7G9AH 56678975 IC50 = 94000 nM T68251 C02GOU 56679764 IC50 = 9.4 nM T68251 CFDR70 56679765 IC50 = 13 nM T68251 CLPF34 56679766 IC50 = 29 nM T68251 C0XP1D 56679767 IC50 = 50 nM T68251 CTE68Z 56679768 IC50 = 30 nM T68251 CES0V3 56679769 IC50 = 411 nM T68251 C0L2JS 56682178 IC50 = 61300 nM T68251 C8UB9G 56682179 IC50 = 83900 nM T68251 C4XL3Y 56682293 IC50 = 86600 nM T68251 CK70XW 56682294 IC50 = 107100 nM T68251 C67VUX 56682295 IC50 = 52700 nM T68251 CIB34L 56683087 IC50 = 10 nM T68251 CM79IH 56683088 IC50 = 1.1 nM T68251 CSL1X7 56683089 IC50 = 104 nM T68251 CSR32E 56683090 IC50 = 86 nM T68251 CWJ65H 56683091 IC50 = 308 nM T68251 CEO93F 56683092 IC50 = 106 nM T68251 CO8FP7 56683093 IC50 = 80 nM T68251 C6KT1Z 56683094 IC50 = 25 nM T68251 CJCI10 56683095 IC50 = 54 nM T68251 C5F7WT 56683096 IC50 = 142 nM T68251 C62FZC 56835063 IC50 = 501 nM T68251 CKJ9S1 56835167 IC50 = 30 nM T68251 C21CLZ 56835168 IC50 = 240 nM T68251 C0L2TS 56835169 IC50 = 1200 nM T68251 CKEV19 56850269 IC50 > 500000 nM T68251 C13DBR 56850270 IC50 > 500000 nM T68251 C05CTJ 56850271 IC50 = 30000 nM T68251 CX8QD5 56850272 IC50 = 310000 nM T68251 C1I9RE 56850407 IC50 > 500000 nM T68251 CVJ90W 56850408 IC50 = 24000 nM T68251 CPI5G0 56850409 IC50 = 83000 nM T68251 C8TH2F 56945850 IC50 = 203 nM T68251 CD72TG 56945851 IC50 = 5 nM T68251 C8J4SC 56945854 IC50 = 64 nM T68251 C1AIZ6 56945963 IC50 = 29 nM T68251 CXQC91 56945964 IC50 = 58 nM T68251 CM4H9D 56945965 IC50 = 44 nM T68251 CUT4S2 56946063 IC50 = 202 nM T68251 C2CQR8 56946064 IC50 = 22 nM T68251 C2H8PG 56946065 IC50 = 13 nM T68251 CW2P6A 56946167 IC50 = 12 nM T68251 CT8S3G 56946168 IC50 = 52 nM T68251 C6LR7O 56964014 IC50 = 328 nM T68251 CE12KU 56964015 IC50 = 158 nM T68251 CL42CX 56964110 IC50 = 219 nM T68251 C0KPD8 57384084 IC50 = 9 nM T68251 CV67JB 57384091 IC50 = 53 nM T68251 C5WFN6 57391082 IC50 = 1 nM T68251 C9BN4F 57391101 IC50 = 7 nM T68251 CI0X9S 57391136 IC50 = 10 nM T68251 CD9J1C 57391201 IC50 > 10000 nM T68251 CN2H9K 57391204 IC50 = 5011.87 nM T68251 CR8MW2 57391205 IC50 = 5011.87 nM T68251 CA25DM 57391224 IC50 = 200 nM T68251 C6P9XK 57391225 IC50 = 144 nM T68251 COT76D 57391411 IC50 > 500000 nM T68251 CJZ0U8 57391412 IC50 > 500000 nM T68251 CAQB32 57391413 IC50 = 4000 nM T68251 CCB9H2 57391414 IC50 = 9 nM T68251 CC57MO 57392866 IC50 = 3.7 nM T68251 C4IWN7 57392867 IC50 = 85 nM T68251 C1ZG3T 57392880 IC50 = 2 nM T68251 CH1I4N 57392901 IC50 = 102 nM T68251 C7CV1B 57392902 IC50 = 6913 nM T68251 C25FAK 57392903 IC50 = 16 nM T68251 C4CK0Q 57392968 IC50 = 7943.28 nM T68251 CNQ9B2 57392969 IC50 = 19952.62 nM T68251 CTYP14 57392972 IC50 = 7943.28 nM T68251 C5VB0U 57392973 IC50 = 6309.57 nM T68251 CMQL31 57392974 IC50 > 10000 nM T68251 C39OHF 57392975 IC50 = 7943.28 nM T68251 CX89EL 57392993 IC50 = 607 nM T68251 C0F3ZD 57393177 IC50 > 500000 nM T68251 CUJD65 57393178 IC50 = 400000 nM T68251 CMB13S 57393179 IC50 = 9000 nM T68251 CJ30LT 57393180 IC50 = 340000 nM T68251 CT2E8Z 57393181 IC50 = 31000 nM T68251 C2O9QP 57394596 IC50 = 2 nM T68251 CN9X5F 57394606 IC50 = 2 nM T68251 CP5BX6 57394607 IC50 = 3.9 nM T68251 CA09RY 57394649 IC50 = 197 nM T68251 CDCW73 57394678 IC50 > 500000 nM T68251 CH6BA3 57394709 IC50 > 10000 nM T68251 CNOH63 57394711 IC50 = 7300 nM T68251 C1CYK9 57394729 IC50 = 25 nM T68251 C9JC3H 57394730 IC50 = 200 nM T68251 C80FML 57394731 IC50 = 111 nM T68251 CYFJ06 57394732 IC50 = 3286 nM T68251 CE5X3D 57394850 IC50 = 10 nM T68251 C82ATC 57394900 IC50 = 3000 nM T68251 C2X8UO 57394901 IC50 > 500000 nM T68251 CN8A6U 57394902 IC50 = 330000 nM T68251 CG43ME 57394903 IC50 = 13 nM T68251 C18PVK 57396348 IC50 > 1000 nM T68251 CM8K2T 57396360 IC50 > 1000 nM T68251 COXA03 57396390 IC50 = 308 nM T68251 CO17CH 57396398 IC50 = 306 nM T68251 CDES09 57396473 IC50 = 1995.26 nM T68251 CONH52 57396474 IC50 = 7943.28 nM T68251 CV51ME 57396475 IC50 = 6309.57 nM T68251 CJB27Z 57396489 IC50 = 81 nM T68251 C34RZI 57396490 IC50 = 178 nM T68251 CD5G3V 57396665 IC50 > 500000 nM T68251 CEB81P 57396666 IC50 > 500000 nM T68251 CMNU14 57396667 IC50 > 500000 nM T68251 CN0LI1 57396668 IC50 = 710 nM T68251 C2MI0H 57398136 IC50 = 1599 nM T68251 C98EXD 57398159 IC50 = 3 nM T68251 C1BIM8 57398160 IC50 = 11 nM T68251 C0KPT7 57398161 IC50 = 2.4 nM T68251 CD6Q9F 57398187 IC50 = 163 nM T68251 CSX81J 57398194 IC50 = 1610 nM T68251 CBH82N 57398195 IC50 = 45 nM T68251 C0YHM7 57398273 IC50 = 83 nM T68251 C5R1PU 57398274 IC50 = 3670 nM T68251 C0ZL1D 57399843 IC50 = 2050 nM T68251 CI6WB3 57399844 IC50 = 30083 nM T68251 C5SVE2 57399911 IC50 > 10000 nM T68251 CZ4GX2 57399912 IC50 = 7943.28 nM T68251 C4J5LE 57399913 IC50 = 7943.28 nM T68251 CH1J9Q 57399914 IC50 > 10000 nM T68251 CD50CO 57399918 IC50 = 3981.07 nM T68251 C82HGR 57399936 IC50 = 4370 nM T68251 CAX15U 57399937 IC50 = 9200 nM T68251 C1CN3U 57401566 IC50 = 2319 nM T68251 C3EKY4 57401585 IC50 = 4 nM T68251 CBZ36R 57401604 IC50 = 3 nM T68251 CM9D3A 57401688 IC50 > 10000 nM T68251 CF02UP 57401689 IC50 = 3981.07 nM T68251 CVO56U 57401690 IC50 = 7943.28 nM T68251 CN27EP 57401691 IC50 = 6309.57 nM T68251 CJLZ14 57401692 IC50 > 10000 nM T68251 C2AI8P 57401693 IC50 > 10000 nM T68251 CLNT30 57401717 IC50 = 798 nM T68251 CKL68A 57401718 IC50 = 307 nM T68251 C5IYO8 57401900 IC50 > 500000 nM T68251 CI1ML6 57401901 IC50 > 500000 nM T68251 C2IE0C 57401902 IC50 = 6800 nM T68251 C39ELP 57403329 IC50 = 15 nM T68251 CWP09F 57403330 IC50 > 1000 nM T68251 CIB91W 57403331 IC50 = 0.55 nM T68251 C63WPS 57403332 IC50 = 0.49 nM T68251 CXF62Z 57403333 IC50 = 16 nM T68251 CT26AL 57403355 IC50 = 931 nM T68251 C6OQH8 57403420 IC50 = 1258.93 nM T68251 C2Z6EC 57403421 IC50 = 5011.87 nM T68251 CA5Z2V 57403422 IC50 = 6309.57 nM T68251 CK68EY 57403424 IC50 = 7943.28 nM T68251 CQN8L6 57403445 IC50 = 232 nM T68251 C2L1SE 57403446 IC50 = 180 nM T68251 C0G2VY 57403564 IC50 = 0.8 nM T68251 CK4CJ0 57403617 IC50 = 290000 nM T68251 C5D0WE 57403618 IC50 > 500000 nM T68251 C7K2AP 57403619 IC50 > 500000 nM T68251 CE9B2P 57403620 IC50 = 1700 nM T68251 C1DRY0 57403621 IC50 = 200 nM T68251 C2MH8O 57523473 IC50 = 0.35 nM T68251 C57CEM 57523505 IC50 = 4 nM T68251 CS8W4L 57523538 IC50 = 5 nM T68251 CIT7B9 57523539 IC50 = 2 nM T68251 C56QXU 57523540 IC50 = 4 nM T68251 CX8IU3 57523541 IC50 = 30 nM T68251 CE8CL9 57523575 IC50 = 107 nM T68251 CWUP89 57523576 IC50 = 0.13 nM T68251 CT2QS3 57523577 IC50 = 0.07 nM T68251 CK6M0Y 57523578 IC50 = 0.1 nM T68251 C0HVU7 57523611 IC50 = 3 nM T68251 C5Q0ND 57523641 IC50 = 1.2 nM T68251 CWH7V8 57561293 IC50 = 533 nM T68251 C1PHI6 57708731 IC50 = 510 nM T68251 CF2Z7W 57708783 IC50 = 62 nM T68251 C9KV2W 57708792 IC50 = 660 nM T68251 CE36GP 57708799 IC50 = 670 nM T68251 C23QGY 57708843 IC50 > 1000 nM T68251 C2J5CW 57708880 IC50 = 230 nM T68251 C1K6AP 57708886 IC50 = 14 nM T68251 CY1N3J 57792153 IC50 = 1167 nM T68251 C6BKQ0 57874709 IC50 = 46000 nM T68251 CCKD80 58307579 Ki = 2.3 nM T68251 CX73PT 59033102 IC50 > 25000 nM T68251 CAT67H 59910477 IC50 = 79 nM T68251 CTZJ24 59910497 IC50 = 885 nM T68251 C1T2QI 60144811 IC50 = 545000 nM T68251 CZ18UT 67684770 IC50 = 10700 nM T68251 CLOE02 70682288 Ki = 600 nM T68251 CH2Q3V 70682301 IC50 = 53 nM T68251 C4NG7I 70682302 IC50 = 24 nM T68251 C6YOW4 70682303 IC50 = 10 nM T68251 CH76IU 70684364 Ki = 450 nM T68251 CZ63AG 70684365 Ki = 300 nM T68251 C6YH8C 70684382 IC50 = 3.8 nM T68251 CQ50YR 70684390 IC50 = 66 nM T68251 CTR64D 70686538 IC50 = 149 nM T68251 C0Q6JA 70686539 IC50 = 179 nM T68251 C8B6WD 70688393 IC50 = 11650 nM T68251 CGR3J2 70688394 IC50 = 23280 nM T68251 CTUN76 70688632 Ki = 61 nM T68251 C3LCG0 70688633 Ki = 180 nM T68251 CV9Y7S 70688643 IC50 = 7.3 nM T68251 CB4ZL3 70690154 IC50 > 500000 nM T68251 CJY19I 70690714 IC50 = 15 nM T68251 CFM0Q5 70690777 IC50 = 0.2 nM T68251 CWVI71 70691250 IC50 = 144 nM T68251 CJ3OY4 70692312 IC50 > 500000 nM T68251 C1A0VU 70692840 Ki = 110 nM T68251 CY4E9Z 70692916 IC50 > 100000 nM T68251 C0HFX4 70694371 IC50 > 500000 nM T68251 C0HE2P 70694634 IC50 = 15470 nM T68251 CLE79H 70696450 IC50 > 500000 nM T68251 CENQ98 70697478 IC50 = 450 nM T68251 C1XNI9 70941086 IC50 > 100000 nM T68251 C7BHO9 70941091 IC50 = 34700 nM T68251 C37VPQ 70941121 IC50 = 10300 nM T68251 CF7PC5 70941155 IC50 > 100000 nM T68251 CL7JF9 71304794 IC50 = 63 nM T68251 CSY30R 71304795 IC50 = 10 nM T68251 CNPG78 71304796 IC50 = 170 nM T68251 CA92XR 71449332 IC50 = 85500 nM T68251 COM1B0 71449369 IC50 = 143 nM T68251 CA6IB0 71450469 IC50 > 1000000 nM T68251 CK2AT8 71451145 IC50 = 12500 nM T68251 C5NYF7 71451146 IC50 = 1400 nM T68251 CW06TJ 71451147 IC50 = 67 nM T68251 CA7M9F 71451166 IC50 = 39000 nM T68251 CD4CP2 71451167 IC50 = 60000 nM T68251 C6M9VL 71451168 IC50 = 8100 nM T68251 C7HUF5 71451169 IC50 = 120 nM T68251 CMW3O0 71451330 Ki > 200000 nM T68251 CT5J7F 71452300 IC50 > 1000000 nM T68251 C23NVO 71452301 IC50 > 1000000 nM T68251 C7UIS9 71452970 IC50 = 67500 nM T68251 CC1B0Z 71452971 IC50 = 83700 nM T68251 CNMP23 71452972 IC50 = 27600 nM T68251 CIP9J5 71452973 IC50 = 8100 nM T68251 CUZ9S0 71452974 IC50 = 120 nM T68251 C71TWC 71452975 IC50 = 3900 nM T68251 CE98YL 71452999 IC50 = 184 nM T68251 C8VC6N 71453000 IC50 = 30 nM T68251 C4VKI1 71453001 IC50 = 87 nM T68251 C4E6PS 71453593 IC50 = 20000 nM T68251 C5K8WS 71454094 IC50 = 573000 nM T68251 CP2D3C 71454095 IC50 > 1000000 nM T68251 CGE27K 71454723 IC50 = 3000 nM T68251 C3VQW4 71455829 IC50 > 1000000 nM T68251 C4EJX2 71456472 IC50 = 37 nM T68251 C9QS6E 71456659 Ki = 20 nM T68251 C1JI6W 71458326 IC50 = 74600 nM T68251 C8ZR2I 71458327 IC50 = 1700 nM T68251 CV2J5Y 71458328 IC50 = 460 nM T68251 C29YHS 71458330 IC50 = 900 nM T68251 CXC1U7 71458350 IC50 = 121 nM T68251 C4IZ5V 71458351 IC50 = 181 nM T68251 CKR4D0 71459517 IC50 > 1000000 nM T68251 CKV4Q6 71460169 IC50 = 4500 nM T68251 CYF62U 71460170 IC50 = 750 nM T68251 C3LFX2 71460171 IC50 = 270 nM T68251 CDRO30 71460172 IC50 = 25 nM T68251 C6WN3A 71460173 IC50 = 13 nM T68251 CZO86D 71460193 IC50 = 278 nM T68251 C6UQW4 71461261 IC50 > 1000000 nM T68251 CKW27N 71461578 IC50 = 19.6 nM T68251 CX7W4A 71461879 IC50 = 2400 nM T68251 CKXO81 71461880 IC50 = 6300 nM T68251 CI4M8V 71461881 IC50 = 7600 nM T68251 CHD70Q 71461882 IC50 = 29 nM T68251 C7MLC8 71461883 IC50 = 17 nM T68251 CWL97M 71461905 IC50 = 301 nM T68251 CUT3H5 71461906 IC50 = 148 nM T68251 C06AXC 71461907 IC50 = 58 nM T68251 CSW59Y 71461908 IC50 = 1340 nM T68251 C9QE5X 71462985 IC50 > 1000000 nM T68251 CATP87 71465323 IC50 = 32.8 nM T68251 C0H3BX 71465324 IC50 = 6.4 nM T68251 CTM24Y 71465370 IC50 = 7.2 nM T68251 C6ZV0X 71465371 IC50 = 9.3 nM T68251 C7NYO8 71465420 IC50 = 6.3 nM T68251 C0E3FD 71465421 IC50 = 3.9 nM T68251 CW1K8M 71465466 IC50 > 100000 nM T68251 C28OYX 71465467 IC50 = 35700 nM T68251 C12BUO 71465468 IC50 > 100000 nM T68251 CP37ZB 71465510 IC50 = 2100 nM T68251 CR2T8F 71503450 IC50 = 2.8 nM T68251 C56YRV 71516803 IC50 < 1 nM T68251 C52QIK 71516804 IC50 = 5.1 nM T68251 C79ZRK 71516805 IC50 = 1.6 nM T68251 C3L7SD 71533484 IC50 = 227 nM T68251 CZH5S9 71533485 IC50 = 52 nM T68251 C4YRC7 71533486 IC50 = 21 nM T68251 CGM72Q 71540498 IC50 = 57 nM T68251 CXA1I5 71540599 IC50 = 54 nM T68251 C7CV9E 71540600 IC50 = 149 nM T68251 CA4BP6 71540601 IC50 = 82 nM T68251 CMZ3T2 71540715 IC50 = 67 nM T68251 CXY83G 71540716 IC50 = 56 nM T68251 C1ZH2G 71540717 IC50 = 69 nM T68251 CT4UD5 71540831 IC50 = 145 nM T68251 CP7SX8 71540832 IC50 = 71 nM T68251 C9IW7R 71540833 IC50 = 54 nM T68251 C6MA8T 71540949 IC50 = 598 nM T68251 C52FXB 71547352 IC50 = 1.7 nM T68251 C9RE0A 71559535 IC50 = 8.44 nM T68251 C47TMN 71559652 IC50 = 8.46 nM T68251 CN2XB4 71559653 IC50 = 5.57 nM T68251 CZHQ79 71559654 IC50 = 1524.69 nM T68251 CO59LK 71559762 IC50 = 4.18 nM T68251 CGL35Z 71559763 IC50 = 5.62 nM T68251 C7U5LE 71559764 IC50 = 1674.81 nM T68251 CD6L1J 71559765 IC50 = 4.32 nM T68251 CXKO04 71559766 IC50 = 5.73 nM T68251 CA14SK 71559767 IC50 = 1724.94 nM T68251 COZ56A 71559768 IC50 = 9.09 nM T68251 CZ9X1J 71559769 IC50 = 1867.71 nM T68251 C5NHI1 71559770 IC50 = 8.59 nM T68251 CF9JE8 71559897 IC50 = 9.11 nM T68251 CGT96R 71559898 IC50 = 5.47 nM T68251 C01PTX 71559899 IC50 = 1674.23 nM T68251 C96OCB 71559900 IC50 = 5.53 nM T68251 CJB0D9 71559901 IC50 = 1764.37 nM T68251 C6Y1IE 71559902 IC50 = 4.09 nM T68251 C24ZYC 71559903 IC50 = 5.62 nM T68251 CC3MY7 71559904 IC50 = 1754.54 nM T68251 C7WMU5 71560026 IC50 = 9.01 nM T68251 C60VEX 71560027 IC50 = 1578.64 nM T68251 CN1VF7 71560028 IC50 = 8.39 nM T68251 CSY3D5 71560029 IC50 = 9.04 nM T68251 CH5J4A 71602247 IC50 = 16 nM T68251 CH53IU 71602248 IC50 = 230 nM T68251 C97EWQ 71602249 IC50 = 61 nM T68251 CNX9B1 71652215 IC50 = 1.4 nM T68251 C7RZN9 71652216 IC50 = 3.8 nM T68251 C0NTU7 71652382 IC50 = 0.43 nM T68251 CA5XS1 71652383 IC50 = 46 nM T68251 CYS46I 71652677 IC50 = 3200 nM T68251 CX67VE 71654516 IC50 = 3000 nM T68251 C6KEH0 71680708 Ki = 27 nM T68251 C7DMX5 71680709 Ki = 3.9 nM T68251 CFPM82 71680710 Ki = 35 nM T68251 C9ZOM7 71680866 Ki = 3.1 nM T68251 CQ68LT 71680868 Ki = 7000 nM T68251 CFH2V0 71681183 Ki = 49 nM T68251 CV3X1T 71682766 Ki = 810 nM T68251 C5EAO8 71682767 Ki = 430 nM T68251 C80EYX 71682913 Ki = 7200 nM T68251 CIBD03 71682914 Ki = 240 nM T68251 C41BYG 71682915 Ki = 4.6 nM T68251 C93XEI 71682916 Ki = 67 nM T68251 CQ29PJ 71682917 Ki = 50000 nM T68251 CFWN65 71683062 Ki = 5700 nM T68251 CM4E5A 71716445 IC50 = 4.19 nM T68251 C45PSZ 71717046 IC50 = 9.26 nM T68251 C9Z4PI 71718276 IC50 = 8.41 nM T68251 C2XW5I 71718291 IC50 = 9.41 nM T68251 C3L4XU 71718301 IC50 = 3.3 nM T68251 C18RDB 71719502 IC50 = 4.43 nM T68251 C6FVE5 71734008 IC50 < 1 nM T68251 CN95PL 71734104 IC50 < 1 nM T68251 CV37BJ 71734105 IC50 = 4.8 nM T68251 C7H8VM 71734106 IC50 < 1 nM T68251 CHBV73 71734107 IC50 < 1 nM T68251 C6C1JF 71734108 IC50 = 14 nM T68251 CR28AW 71734195 IC50 = 7 nM T68251 C2YJR3 71734196 IC50 = 141 nM T68251 CJC6N5 71734197 IC50 = 5.2 nM T68251 CEF50T 71734198 IC50 = 3.6 nM T68251 CLWC38 72193198 IC50 < 1 nM T68251 CX4G0R 72204928 IC50 = 28200 nM T68251 CG9C6U 72204929 IC50 = 6000 nM T68251 C5A6XZ 72204930 IC50 = 20000 nM T68251 C0XZK4 72204931 IC50 = 15000 nM T68251 CM8Y7X 72204932 IC50 = 36000 nM T68251 C6RY4X 72204933 IC50 = 6600 nM T68251 C4N5AB 72204934 IC50 = 20800 nM T68251 C3H2FZ 72205111 IC50 = 42000 nM T68251 CQ0VX7 72205112 IC50 = 25000 nM T68251 CQ7TI1 72205113 IC50 = 2800 nM T68251 CPAW52 72205114 IC50 = 2100 nM T68251 C2LD3J 72205115 IC50 = 2800 nM T68251 CE4J8F 72711063 Ki = 290 nM T68251 CW2RF1 72711064 Ki = 490 nM T68251 CC5T1Q 72711065 Ki = 680 nM T68251 C7YFC8 72711513 IC50 = 1045 nM T68251 CTM4P2 72713638 IC50 = 1.2 nM T68251 C0N2JX 72713639 IC50 = 3 nM T68251 CF4K8Y 72713862 IC50 = 7.5 nM T68251 C3R6JO 72713863 IC50 = 48 nM T68251 CW9D3V 72713864 IC50 = 15 nM T68251 CQ6FH3 72713865 IC50 = 7.8 nM T68251 C4FYB0 72713866 IC50 = 20 nM T68251 CH6SI1 72713867 IC50 = 41 nM T68251 CS21QM 72713868 IC50 = 670 nM T68251 CB56AP 72714081 IC50 = 18 nM T68251 C1CK0E 72714082 IC50 = 1750 nM T68251 CP5Q8W 72714083 IC50 = 1870 nM T68251 CA03NU 72714084 IC50 = 125000 nM T68251 CRUH64 72714085 IC50 = 3800 nM T68251 COQZ24 72714091 Ki = 160 nM T68251 CC0ZX4 72714092 Ki = 230 nM T68251 CW8I1S 72714093 Ki = 310 nM T68251 C3Q9LV 72714094 Ki = 480 nM T68251 CZFY06 72714322 IC50 = 4100 nM T68251 CDY70J 72714323 IC50 = 1440 nM T68251 CD56BA 72714324 IC50 = 240 nM T68251 CE51LQ 72714333 Ki = 550 nM T68251 CK6D5F 72714334 Ki = 760 nM T68251 C1R2UZ 72714335 Ki = 690 nM T68251 CH4VF7 72714336 Ki = 440 nM T68251 C4VSK6 72714337 Ki = 560 nM T68251 CG4KW2 72714338 Ki = 420 nM T68251 C9FL7V 72714339 Ki = 50 nM T68251 CT5U1W 72734852 IC50 = 428990 nM T68251 C4OEI9 72734853 IC50 = 20620 nM T68251 C4AT5M 72734854 IC50 = 6559 nM T68251 CA7I9Q 72734855 IC50 = 10800 nM T68251 CJ5N2K 72734856 IC50 = 679 nM T68251 CCQ27I 72734857 IC50 = 1802 nM T68251 CCP65R 72735032 IC50 = 5438 nM T68251 C5XL1A 72735033 IC50 = 386 nM T68251 CYT1H0 72735034 IC50 = 530 nM T68251 CW6IE4 72735035 IC50 = 325 nM T68251 C58RHN 72735036 IC50 = 678.1 nM T68251 CFB5U1 72735037 IC50 = 325 nM T68251 CXY79G 72737387 IC50 = 2776 nM T68251 C6M1OD 72737388 IC50 = 834.9 nM T68251 CY4M3X 72737389 IC50 = 28190 nM T68251 CQM2E0 72737390 IC50 = 9480 nM T68251 CFQX60 72737391 IC50 = 878 nM T68251 C4BAJ5 72737560 IC50 = 77930 nM T68251 CRP56E 72737561 IC50 = 3093 nM T68251 C3J8GN 72737562 IC50 = 7480 nM T68251 CS2JM8 72737563 IC50 = 678 nM T68251 CZ0G7Y 72737564 IC50 = 786 nM T68251 COHR84 72737565 IC50 = 877 nM T68251 CLV1F5 72737566 IC50 = 516 nM T68251 CDX2F9 72984326 IC50 = 9.25 nM T68251 C6SR0A 73106454 IC50 = 61.94 nM T68251 CUKG79 73292708 IC50 = 0.9 nM T68251 C5D3CJ 73292709 IC50 = 4 nM T68251 CL69NM 73292710 IC50 = 4 nM T68251 CQ4RO1 73292711 IC50 = 0.7 nM T68251 C7CT2E 73292869 IC50 = 4 nM T68251 CA0LS6 73292870 IC50 = 0.9 nM T68251 CJU3V6 73292871 IC50 = 5 nM T68251 C3PGF2 73292872 IC50 = 3 nM T68251 C0O8VM 73292873 IC50 = 2 nM T68251 CBR9I5 73293034 IC50 = 3 nM T68251 C9FD2C 73293035 IC50 = 3 nM T68251 C7LP5J 73293036 IC50 = 2 nM T68251 C9PQG1 73293037 IC50 = 5 nM T68251 C4PF1H 73293038 IC50 = 0.4 nM T68251 CE39WF 73293196 IC50 = 4 nM T68251 CU96XE 73293197 IC50 = 9 nM T68251 CGC51Z 73293198 IC50 = 2 nM T68251 CC83FW 73293199 IC50 = 2 nM T68251 CS6T8M 73293200 IC50 = 0.5 nM T68251 C38IDL 73345835 Ki = 1.7 nM T68251 CR1LT3 73346934 IC50 = 200630 nM T68251 C25SOB 73349251 IC50 = 0.8 nM T68251 CW01EA 73349535 IC50 > 10000 nM T68251 C8ROG3 73350414 Ki = 14 nM T68251 CF7AB2 73350415 Ki = 17 nM T68251 C2PFM4 73351930 Ki = 200 nM T68251 COC60V 73352986 IC50 = 671560 nM T68251 CI09CY 73354906 Ki = 8.5 nM T68251 CA5T7P 73603957 IC50 = 3000 nM T68251 C8VN1R 74221194 IC50 = 1800 nM T68251 C7M4FT 74430862 IC50 = 35670 nM T68251 CD28XO 74966628 IC50 = 109.9 nM T68251 CG1AU5 74991907 IC50 = 2.6 nM T68251 C65RFS 74991938 IC50 = 6.6 nM T68251 CX89MG 75002237 IC50 = 34197.94 nM T68251 CD7P3T 75002250 IC50 = 750 nM T68251 CU73SM 75018048 IC50 = 26 nM T68251 C1BTU7 75018058 IC50 = 29.99 nM T68251 CX9VB7 75018063 IC50 = 15 nM T68251 CLHO50 75018065 IC50 = 3.396 nM T68251 CQL0E1 75018100 IC50 = 1 nM T68251 CC9UA2 75018101 IC50 = 1.3 nM T68251 CYB42V 75018103 IC50 = 269.77 nM T68251 C1FTQ8 75018104 IC50 = 5.8 nM T68251 C5M2FT 75018105 IC50 = 1.6 nM T68251 CF5ZC7 75018120 IC50 = 50 nM T68251 CFW35X 75018121 IC50 = 280 nM T68251 C4GK3X 75018123 IC50 = 5105.05 nM T68251 C6FPO0 75018124 IC50 = 84 nM T68251 CMS1L6 75018126 IC50 = 3500 nM T68251 CW78YB 75018133 IC50 = 38.02 nM T68251 CZP6X1 75018134 IC50 = 414 nM T68251 CS1D6P 75018135 IC50 = 0.4 nM T68251 CHAP32 75018146 IC50 = 2430 nM T68251 CEF3L5 75018147 IC50 = 6.397 nM T68251 CPMC39 75018148 IC50 = 779.83 nM T68251 CBNW85 75018149 IC50 = 53.95 nM T68251 C57SNU 75018158 IC50 = 309.74 nM T68251 CCL95X 75018159 IC50 = 33.96 nM T68251 CXC24A 75018160 IC50 = 210 nM T68251 C9F8BU 75018162 IC50 = 920 nM T68251 C4OP3D 75018163 IC50 = 100 nM T68251 C7YPR3 75018171 IC50 = 51999.6 nM T68251 CT8Y6H 75018172 IC50 = 1698.24 nM T68251 C5Z1CN 75018180 IC50 = 1 nM T68251 CW7OX3 75018184 IC50 = 6800 nM T68251 C68QBF 75018185 IC50 = 10.99 nM T68251 CSBO46 75018194 IC50 = 41 nM T68251 CUB7V9 76329513 IC50 = 0.26 nM T68251 C5LB0U 78426619 IC50 > 100000 nM T68251 CET6N8 78426757 IC50 > 100000 nM T68251 CKD41G 81689861 IC50 = 1000 nM T68251 CBL02O 85040463 IC50 = 27.99 nM T68251 CHAG58 85052312 IC50 = 6.6 nM T68251 CJ67RP 85055259 IC50 = 59 nM T68251 CVHM18 85082338 IC50 = 11.99 nM T68251 CRC43U 85102289 IC50 = 0.4 nM T68251 C3Z0PJ 85141621 IC50 = 0.2 nM T68251 C28SQI 85198610 IC50 = 11 nM T68251 CUE7G4 86287514 IC50 = 24000 nM T68251 CGQ8F3 86287515 IC50 = 1800 nM T68251 CJ37XE 86287516 IC50 = 3200 nM T68251 COV8I9 86291010 IC50 = 1088 nM T68251 C76RBA 86298624 IC50 = 230 nM T68251 C93FKI 86298625 IC50 = 110 nM T68251 CVLU48 86298626 IC50 = 192 nM T68251 CAB2F5 87349434 Ki = 13000 nM T68251 CY74HT 89136066 IC50 = 2 nM T68251 C1MDQ8 89136114 IC50 = 1400 nM T68251 CO2FL5 90137145 IC50 = 310 nM T68251 CIJ96H 90644155 IC50 = 4800 nM T68251 CX7EW1 90644156 IC50 = 30000 nM T68251 CK5GZ4 90644157 IC50 = 52000 nM T68251 C7O1YN 90644158 IC50 = 19000 nM T68251 CEN6C1 90644159 IC50 = 4900 nM T68251 C8X9UZ 90644160 IC50 = 16000 nM T68251 C3H6SG 90656558 IC50 = 980 nM T68251 CFE10C 90656560 IC50 = 1030 nM T68251 CD4L8R 90656562 IC50 = 4190 nM T68251 CEST81 90656564 IC50 = 2710 nM T68251 C7J0CO 90656566 IC50 = 520 nM T68251 CE9Y4D 90656568 IC50 = 1940 nM T68251 CZVG63 90656570 IC50 = 720 nM T68251 CT0QG6 90656572 IC50 = 760 nM T68251 CFPR48 90656574 IC50 = 3360 nM T68251 CDF06N 90656576 IC50 = 1810 nM T68251 CQ3R1A 90656578 IC50 = 270 nM T68251 CWV0Z9 90656580 IC50 = 1280 nM T68251 CGX01J 90656582 IC50 = 430 nM T68251 C6M1VH 90656584 IC50 = 26180 nM T68251 C1GUD2 90656586 IC50 = 38320 nM T68251 C5KWT1 90656588 IC50 = 7430 nM T68251 CS7PZ6 90656590 IC50 = 5760 nM T68251 CGF9P3 90656592 IC50 = 1520 nM T68251 CM46JO 90656594 IC50 = 5210 nM T68251 CXL84V 90656596 IC50 = 2070 nM T68251 C7EIO6 90656598 IC50 = 2320 nM T68251 CRH7F2 90656600 IC50 = 4360 nM T68251 CKW64G 90656602 IC50 = 2950 nM T68251 C4CU3D 90656604 IC50 = 2050 nM T68251 CVPH63 90663059 Ki = 18000 nM T68251 C6AK3O 90663060 Ki = 15000 nM T68251 CUZD67 90663061 Ki = 8000 nM T68251 CTQ17J 90663062 Ki = 33000 nM T68251 CQGJ90 90663063 Ki = 6000 nM T68251 C0ZH1K 90663064 Ki = 17000 nM T68251 CD53CF 90663065 Ki = 5000 nM T68251 C1A4QT 90663067 Ki = 8000 nM T68251 CLW7Q8 90663069 Ki = 24000 nM T68251 C6JY4Q 90663070 Ki = 36000 nM T68251 C7YU1I 90663071 Ki = 10000 nM T68251 C07RTW 90663072 Ki = 11000 nM T68251 CZ68QM 90663073 Ki = 18000 nM T68251 CVTJ63 90663074 Ki = 7000 nM T68251 C9J8HB 90663075 Ki = 4000 nM T68251 C06GRV 90663076 Ki = 2000 nM T68251 CF2L9A 90663077 Ki = 40000 nM T68251 CGL0N7 90663078 Ki = 12000 nM T68251 COP05M 90663079 Ki = 13000 nM T68251 C1E5CB 90663080 Ki = 35000 nM T68251 C6IXP4 90663081 Ki = 41000 nM T68251 C0S7NT 90663082 Ki = 12000 nM T68251 C8MOY6 90663083 Ki = 20000 nM T68251 C4NP9W 90663084 Ki = 16000 nM T68251 CD3C8E 90663085 Ki = 16000 nM T68251 C63NOF 90663086 Ki = 15000 nM T68251 CU3LC2 90663087 Ki = 17000 nM T68251 CQ9C5I 90667651 IC50 = 0.53 nM T68251 CGXO89 90667652 IC50 = 0.61 nM T68251 CRT54C 101910871 IC50 = 11000 nM T68251 C1J3CK 117094707 IC50 = 5400 nM T68251 CDO15M 118721026 IC50 = 12.5 nM T68251 CHO72Q 118721027 IC50 = 1449 nM T68251 C5ZS4E 118722686 IC50 = 2100 nM T68251 CIZB24 118722687 IC50 = 6100 nM T68251 C5C0ZX 118722688 IC50 = 7100 nM T68251 C4V3FD 118723755 IC50 = 3 nM T68251 CH6OW5 122179777 IC50 = 85350 nM T68251 CLCW15 122181996 IC50 > 100000 nM T68251 CZO32N 122181998 IC50 > 100000 nM T68251 C40DWG 122181999 IC50 > 100000 nM T68251 CJFS09 122190237 IC50 = 590 nM T68251 CRN56G 122191012 IC50 = 235.2 nM T68251 CGC3E2 122191014 IC50 = 144.6 nM T68251 CS61WU 122191016 IC50 = 256.2 nM T68251 CV3SP6 122191017 IC50 = 299.2 nM T68251 C8ZOT4 122191645 IC50 = 7920 nM T68251 CU6LT0 122191646 IC50 = 2884.03 nM T68251 CER90U 122191647 IC50 = 8511.38 nM T68251 C8X2BN 122191648 IC50 = 3235.94 nM T68251 CQ3US9 122191649 IC50 = 4830 nM T68251 C86DWE 122191650 IC50 = 11220.18 nM T68251 CQ14HT 122191651 IC50 = 9430 nM T68251 C8B1HC 122191652 IC50 = 6760.83 nM T68251 CN6WP3 122191653 IC50 = 208.93 nM T68251 CJ5R2S 122192039 IC50 = 4168.69 nM T68251 CK45AP 122192040 IC50 = 794.33 nM T68251 C2W4VX 122192041 IC50 = 2700 nM T68251 C3R5YP 122192042 IC50 = 12589.25 nM T68251 C8EB9C 122192043 IC50 = 11440 nM T68251 CF2K9Z 122192044 IC50 = 14791.08 nM T68251 C68DRB 122192045 IC50 = 2089.3 nM T68251 C2L7ZO 122192046 IC50 = 2150 nM T68251 C1BH0V 122192047 IC50 = 23820 nM T68251 C9MX4H 122192048 IC50 = 17782.79 nM T68251 CE4MD1 122192049 IC50 = 15488.17 nM T68251 CU13GZ 122192050 IC50 = 2818.38 nM T68251 CN1OP2 122192051 IC50 = 9900 nM T68251 C2WV6G 122192052 IC50 = 14791.08 nM T68251 CD2I6H 122192053 IC50 = 16840 nM T68251 CQ7RZ6 122192054 IC50 = 3630.78 nM T68251 COIP89 122195564 IC50 = 360 nM T68251 C8Z1BF 124196387 IC50 = 17000 nM T68251 CF9C4N 127025165 IC50 = 6.5 nM T68251 CH59PY 127025166 IC50 = 791 nM T68251 CT03QA 127026888 IC50 = 370 nM T68251 CO1DJ9 127027301 IC50 = 11.66 nM T68251 CM7B5S 127029507 IC50 = 628 nM T68251 C6HA8I 127029508 IC50 > 100000 nM T68251 CPM3N2 127029509 IC50 = 56.3 nM T68251 C3B9EY 127029510 IC50 > 100000 nM T68251 C9NLI6 127030239 IC50 = 112260 nM T68251 CW3C0H 127030240 IC50 = 38650 nM T68251 CHC1V8 127031459 IC50 = 34790 nM T68251 C5GJB1 127031460 IC50 = 9390 nM T68251 C3R8PS 127031461 IC50 = 13220 nM T68251 C07FRX 127031462 IC50 = 90810 nM T68251 C9QC5M 127031784 IC50 = 1050 nM T68251 CX25ZP 127031785 IC50 = 210410 nM T68251 CIP36Q 127032630 IC50 = 1890 nM T68251 CA5I7G 127032946 IC50 = 410 nM T68251 CEO26U 127032998 IC50 = 28520 nM T68251 CL16WE 127033305 IC50 = 5520 nM T68251 C9RZO5 127033306 IC50 = 640 nM T68251 C20GLU 127033307 IC50 = 240 nM T68251 C2XUV8 127033875 IC50 = 74910 nM T68251 COM48Q 127033876 IC50 = 28760 nM T68251 C30DFR 127033877 IC50 = 223370 nM T68251 CA8HJ9 127033878 IC50 = 36790 nM T68251 CQ3HV1 127034380 IC50 = 566890 nM T68251 CV1YR6 127036461 IC50 = 2000 nM T68251 CDIC57 127037442 IC50 = 3 nM T68251 CV3NQ6 127037443 IC50 = 2400 nM T68251 CWI7K3 127037444 IC50 > 10000 nM T68251 C9QLI2 127037445 IC50 = 9000 nM T68251 CCA0R8 127037446 IC50 = 1100 nM T68251 C89QOM 127043503 IC50 = 51 nM T68251 CK3I0F 127043504 IC50 = 263 nM T68251 C9E5YJ 127043505 IC50 = 31 nM T68251 CW1Q3D 127043506 IC50 = 76 nM T68251 CFDC75 127043682 IC50 = 193 nM T68251 C1C7WB 127044036 IC50 = 123 nM T68251 C16UNQ 127044037 IC50 = 472 nM T68251 CN58BX 127044038 IC50 = 672 nM T68251 C5DMP0 127044039 IC50 = 419 nM T68251 CPF6U7 127044139 IC50 = 177 nM T68251 C5FPE1 127044169 IC50 > 500 nM T68251 C7YE9B 127044170 IC50 > 500 nM T68251 CT9B0Q 127044462 IC50 = 44.65 nM T68251 CL3X1A 127044649 IC50 = 98 nM T68251 C7X1YO 127044650 IC50 = 186 nM T68251 C8RZ7T 127044651 IC50 = 41 nM T68251 C3I4PT 127044652 IC50 = 103 nM T68251 CBR1V9 127044680 IC50 = 85.9 nM T68251 CDX86T 127044818 IC50 = 30 nM T68251 C56OJV 127044819 IC50 = 24 nM T68251 CF7A5N 127044986 IC50 = 843 nM T68251 CGLJ92 127045131 IC50 = 203 nM T68251 C4HY6K 127045132 IC50 = 208 nM T68251 CWO1X0 127045258 IC50 = 806 nM T68251 C43ORS 127045609 IC50 = 291 nM T68251 C21LIW 127053364 IC50 = 0.19 nM T68251 CR5VQ8 127053365 IC50 = 2.2 nM T68251 C19QXS 127053368 IC50 > 10000 nM T68251 CJ0G9N 127053369 IC50 > 10000 nM T68251 C2Q6UH 127053370 IC50 > 10000 nM T68251 CWM7U2 127053371 IC50 = 21.8 nM T68251 C1VRM8 127053372 IC50 > 10000 nM T68251 CT76DR 127053375 IC50 = 2.05 nM T68251 CYA92R 130282633 IC50 = 890 nM T68251 CO3QE2 130282636 IC50 = 1000 nM T68251 C4MB7N 132285189 Ki = 85 nM T68251 CTN42D 132941363 IC50 = 11000 nM T68251 C83FAY 134130294 Ki = 15.9 nM T68251 CT3G2U 134133460 IC50 = 0.16 nM T68251 C8VLY0 134144890 IC50 = 110 nM T68251 C93ZLI 134145328 IC50 = 107 nM T68251 CN9D7G 134155756 IC50 = 2600 nM T68251 CU24IK 134694685 IC50 = 190 nM T68251 CHV2U1 135438561 IC50 = 5300 nM T68251 C4FVJ1 135487604 IC50 = 79600 nM T68251 C6GR3K 135567051 IC50 = 83 nM T68251 C1MOD4 135567320 IC50 = 730 nM T68251 CYH23I 136054468 IC50 = 32 nM T68251 CZ8DW1 136054472 IC50 = 86 nM T68251 C9H0DL 136054473 IC50 = 120 nM T68251 CX7MI0 136054475 IC50 = 65 nM T68251 CA5JR6 136054481 IC50 = 14 nM T68251 CO2VU9 136054484 IC50 < 10 nM T68251 CV47JN 136054485 IC50 = 10 nM T68251 CZ48WO 136054487 IC50 = 23 nM T68251 CR9CY5 136054490 IC50 < 10 nM T68251 C8FGT0 136054495 IC50 = 110 nM T68251 CGH39U 136054498 IC50 < 10 nM T68251 C2TO7Y 136054508 IC50 = 160 nM T68251 CG70BZ 136054516 IC50 = 3 nM T68251 CSM57W 136054520 IC50 = 0.57 nM T68251 CXNG40 136118011 Ki = 2472 nM T68251 C1IOH9 136118012 Ki > 3333 nM T68251 CTY79S 136118013 Ki > 3333 nM T68251 CTE87J 136118014 Ki > 3333 nM T68251 CJG54U 136219136 IC50 > 30000 nM T68251 C3CAV5 136219141 IC50 > 30000 nM T68251 CPB07Z 136241630 IC50 = 800 nM T68251 CIEW62 136380958 IC50 = 8.3 nM T68251 CSEY19 137175240 IC50 = 7170 nM T68251 C9HS7J 137287436 IC50 = 1.9 nM T68251 C4UMY5 137636781 IC50 > 5000 nM T68251 CR8H9Z 137644167 IC50 > 5000 nM T68251 CB8M6U 137646865 IC50 > 5000 nM T68251 CK4LE6 137647628 IC50 = 2700 nM T68251 C9CIY6 137651719 IC50 = 2 nM T68251 CS80YI 137652598 IC50 = 280 nM T68251 CZB75K 137657128 IC50 > 10000 nM T68251 CC3I9B 137660260 IC50 > 5000 nM T68251 C4H0EM 137661370 IC50 = 3100 nM T68251 CZ8H6N 137661550 IC50 = 5800 nM T68251 C37HMX 137701229 Ki = 37 nM T68251 C5FWA2 145949488 IC50 = 584 nM T68251 CZS1N7 145949693 IC50 = 936 nM T68251 C6IPV3 145949783 IC50 = 4800 nM T68251 C72LGN 145950074 IC50 = 2850 nM T68251 CU53BP 145950331 IC50 > 5000 nM T68251 CY8C4A 145950332 IC50 = 189 nM T68251 CAJ25P 145951291 IC50 > 5000 nM T68251 C3EF7N 145952515 IC50 = 114 nM T68251 CW1GS2 145952760 IC50 > 5000 nM T68251 CFN1R7 145952843 IC50 = 187 nM T68251 CV80WQ 145954107 IC50 > 5000 nM T68251 C16VNH 145954604 IC50 = 500 nM T68251 CQF50V 145954863 IC50 = 128 nM T68251 C2HAG8 145955226 IC50 = 8520 nM T68251 CH0ZO5 145955778 IC50 = 362 nM T68251 CVZ5U7 145955868 IC50 = 232 nM T68251 C8TPR1 145956198 IC50 > 5000 nM T68251 COR96H 145956298 IC50 = 2120 nM T68251 CR8U7Y 145956318 IC50 > 5000 nM T68251 C7R3FE 145956426 IC50 = 1650 nM T68251 CUS0Y9 145957234 IC50 > 5000 nM T68251 C6MHN7 145957508 IC50 > 5000 nM T68251 CQ15DP 145957734 IC50 = 4070 nM T68251 C5K7PV 145958060 IC50 > 5000 nM T68251 CBE02W 145958354 IC50 > 5000 nM T68251 CQL4O0 145959327 IC50 > 5000 nM T68251 CG03OE 145959777 IC50 = 210 nM T68251 CIQ9J2 145960035 IC50 = 5340 nM T68251 CRY63E 145963538 IC50 > 5000 nM T68251 CX7PL8 145963779 IC50 = 75.25 nM T68251 CPRZ56 145963828 IC50 = 72.02 nM T68251 C5JTM2 145963892 IC50 = 38.68 nM T68251 CFLU54 145964255 IC50 = 57.24 nM T68251 C3MDU9 145965508 IC50 = 81210 nM T68251 C8ZI7P 145965593 IC50 = 53.14 nM T68251 C6ASH4 145965758 IC50 = 58.02 nM T68251 CABQ48 145965824 IC50 = 54.74 nM T68251 C8M7FR 145966330 IC50 = 660 nM T68251 CCO03H 145966492 IC50 = 32.71 nM T68251 CZG2P7 145966498 IC50 = 33.47 nM T68251 C4P0GM 145966951 IC50 = 53.82 nM T68251 C5ICD0 145967022 IC50 = 1350 nM T68251 CI80WY 145967366 IC50 = 19.57 nM T68251 CFE1A5 145971595 Ki = 127 nM T68251 CWY5X0 145971805 IC50 = 414 nM T68251 C1FPG2 145972660 IC50 = 219 nM T68251 CYFI60 145973042 IC50 = 2500 nM T68251 CZHR42 145973116 IC50 = 203400 nM T68251 CQF05Z 145973471 IC50 = 50.55 nM T68251 CJF73O 145973630 IC50 = 172 nM T68251 CC1BF5 145973750 IC50 = 58.08 nM T68251 COA47B 145973991 IC50 = 54.68 nM T68251 C1VO8L 145974965 IC50 = 73.82 nM T68251 CQ0DP4 145975098 IC50 = 55.13 nM T68251 CV9D1F 145975682 IC50 > 100000 nM T68251 CI9VB4 145975902 IC50 > 10000 nM T68251 CX7M9L 145976456 IC50 > 5000 nM T68251 C5C6VJ 145976464 IC50 = 54180 nM T68251 C1KPL5 145976497 IC50 = 670 nM T68251 C7RG1J 145976981 IC50 = 62.87 nM T68251 C18OCA 145976989 IC50 = 230000 nM T68251 C5HW7O 145977208 IC50 = 36.83 nM T68251 CPD1B0 145977213 IC50 > 5000 nM T68251 C79VAX 145977588 IC50 = 49.69 nM T68251 CG9KD3 145977825 IC50 > 1000 nM T68251 C60INE 145977843 IC50 = 83.04 nM T68251 CN6JB8 145978296 IC50 > 1000 nM T68251 C5Z7XW 145983264 IC50 = 182 nM T68251 C0EMZ9 145984335 IC50 = 345 nM T68251 CBNO84 145985441 IC50 = 414 nM T68251 CDW7K5 145986213 IC50 = 102 nM T68251 CM7YB8 145998092 IC50 = 1300 nM T68251 C2C8QR 153033791 IC50 = 58430 nM T68251 C2CZ9B 155511425 IC50 = 5700 nM T68251 CZ25LW 155512044 IC50 = 11000 nM T68251 CV10AF 155512426 IC50 = 151 nM T68251 C1V4CS 155512637 IC50 > 10000 nM T68251 CMQ8W6 155512861 IC50 = 7500 nM T68251 CFHU79 155514943 IC50 = 55 nM T68251 C13OQY 155515143 IC50 = 8800 nM T68251 CND4L8 155515645 IC50 = 9549.93 nM T68251 CC15YH 155515706 IC50 > 10000 nM T68251 C98HMU 155515777 IC50 = 1.2 nM T68251 C0OSL9 155516668 IC50 = 21379.62 nM T68251 C6N3DB 155517141 IC50 = 0.28 nM T68251 C3I5AL 155519394 IC50 = 6500 nM T68251 CS6ZT7 155519964 IC50 = 21 nM T68251 CG2RF3 155520398 IC50 = 2100 nM T68251 CL16UE 155520835 IC50 > 10000 nM T68251 C5C1SL 155521791 IC50 > 10000 nM T68251 C59YHT 155522902 IC50 = 503 nM T68251 C4AH9W 155525335 IC50 > 10000 nM T68251 CM9AP3 155526116 IC50 > 10000 nM T68251 C6RBG9 155527660 IC50 = 2800 nM T68251 C83IXL 155528558 IC50 = 0.16 nM T68251 CT4PA7 155528661 IC50 > 10000 nM T68251 CWB4X1 155529076 IC50 > 10000 nM T68251 CSG54J 155529234 IC50 > 10000 nM T68251 C2G0BE 155529579 IC50 > 10000 nM T68251 CC5FA9 155529859 IC50 > 10000 nM T68251 CQUA53 155531128 IC50 = 3000 nM T68251 C7TP3R 155531151 IC50 > 10000 nM T68251 CZSY48 155533962 IC50 = 3600 nM T68251 C5WTE3 155534754 IC50 = 6700 nM T68251 CG47PB 155534833 IC50 = 3000 nM T68251 C4VCN3 155535749 IC50 = 12860 nM T68251 C2WCU5 155536887 IC50 = 10715.19 nM T68251 C4DSL8 155536899 IC50 > 10000 nM T68251 C12LFZ 155540134 IC50 = 620 nM T68251 CNH2K4 155540729 IC50 = 3300 nM T68251 CO90SD 155541304 IC50 = 11748.98 nM T68251 CRY3D4 155541376 IC50 = 13 nM T68251 CV0ZI3 155542003 IC50 = 12302.69 nM T68251 CJN8X5 155542058 Ki = 0.5 nM T68251 CO8ZY9 155542845 IC50 = 0.048 nM T68251 CH9E0W 155543836 IC50 = 34673.69 nM T68251 C1VL8X 155544079 IC50 > 10000 nM T68251 CYK18P 155544623 IC50 > 10000 nM T68251 CBSJ86 155544856 IC50 = 11220.18 nM T68251 CWEG57 155545190 IC50 = 3 nM T68251 CP6W3Q 155545205 IC50 > 10000 nM T68251 CLWS20 155545852 IC50 = 47863.01 nM T68251 COH0W2 155546374 IC50 = 492 nM T68251 CLT8Z2 155546617 IC50 = 2.38 nM T68251 C3FRY8 155547834 IC50 = 0.096 nM T68251 C1FP0M 155548067 IC50 = 32 nM T68251 C9AOK6 155550135 IC50 = 3000 nM T68251 C9ZUH8 155553520 IC50 = 6200 nM T68251 CPQ84I 155553728 IC50 > 10000 nM T68251 CM7C1P 155555245 IC50 = 16240 nM T68251 CS62RN 155556052 IC50 = 13803.84 nM T68251 C94NQE 155556307 IC50 > 10000 nM T68251 C9FC1W 155557598 IC50 = 3200 nM T68251 CJHM29 155557941 IC50 = 8310 nM T68251 CD3M6P 155558654 IC50 = 16870 nM T68251 CPDF57 155558916 IC50 = 57543.99 nM T68251 CG2DI6 155560100 IC50 = 8800 nM T68251 CQJ07L 155561559 IC50 = 8800 nM T68251 C3BA9L 155561798 IC50 = 5 nM T68251 CH40UO 155562232 IC50 = 4.1 nM T68251 C6SAE0 155562336 IC50 = 8.9 nM T68251 CD18KU 155563750 IC50 = 7600 nM T68251 CM0LN1 155563771 IC50 = 810 nM T68251 CQ4WE0 155563852 IC50 = 28183.83 nM T68251 C29SMF 155565303 IC50 > 10000 nM T68251 C51ZMC 155565586 IC50 = 700 nM T68251 CZ0WK1 155566979 IC50 = 3800 nM T68251 CP9YX2 155567218 IC50 = 2400 nM T68251 C8D5VK 155567855 IC50 = 3500 nM T68251 CHL0F3 155567858 IC50 > 10000 nM T68251 C5U9LI 155569346 IC50 = 570 nM T68251 CLT4Y6 10138589 Ki = 300 nM T68251 C5U3AO 57394286 IC50 = 23 nM T68251 C0YL9R 9975488 IC50 = 1900 nM T68251 D00RNA 44446270 IC50 = 200 nM T68251 D00TRF 44423683 IC50 = 94000 nM T68251 D01UNE 44580457 Ki = 30 nM T68251 D02ECA 448942 IC50 > 100000 nM T68251 D02EFQ 10549609 IC50 = 5 nM T68251 D02UYR 9907830 Ki = 0.3 nM T68251 D03AMR 9849669 Ki = 7 nM T68251 D04GOO 10111838 IC50 > 100000 nM T68251 D04PAW 16216218 IC50 = 60000 nM T68251 D04VPH 45376872 IC50 = 18000 nM T68251 D04WWO 9889867 Ki > 3333 nM T68251 D05BMD 44423684 IC50 = 137000 nM T68251 D05JPV 44406790 IC50 = 3070 nM T68251 D05THD 44478925 IC50 = 1300 nM T68251 D06EHW 11625778 IC50 = 35 nM T68251 D06HSC 136117931 IC50 = 65000 nM T68251 D06NDR 44423687 IC50 = 81800 nM T68251 D06ZRX 5281717 IC50 = 27600 nM T68251 D07DRT 46175162 Ki = 3.8 nM T68251 D07GEL 10344307 Ki = 1.1 nM T68251 D07MJD 44479701 IC50 = 510 nM T68251 D07VXX 16721024 IC50 = 151000 nM T68251 D08ICI 44446277 IC50 = 590 nM T68251 D08NSS 5288596 IC50 < 0.1 nM T68251 D09GIL 66160 IC50 = 50000 nM T68251 D09USO 5277466 IC50 > 100000 nM T68251 D09ZOA 25049753 IC50 = 2 nM T68251 D0A0FY 44479457 IC50 = 35000 nM T68251 D0A4TC 446504 IC50 = 3 nM T68251 D0A5MV 11581319 IC50 = 1660 nM T68251 D0B3UN 44580458 Ki = 192 nM T68251 D0D7GL 10789 IC50 = 146000 nM T68251 D0E5MB 44411812 IC50 = 792 nM T68251 D0F2HJ 45257111 IC50 = 196500 nM T68251 D0F7BE 4369084 Ki = 3000 nM T68251 D0FO2B 1923 IC50 = 130000 nM T68251 D0G0OP 44423685 IC50 = 68000 nM T68251 D0G3YZ 11391583 IC50 = 4520 nM T68251 D0H2PA 9886977 Ki = 0.5 nM T68251 D0H6CK 10160968 Ki > 3333 nM T68251 D0J0WJ 45257110 IC50 = 232500 nM T68251 D0K4TI 49292 IC50 = 1300 nM T68251 D0L4EO 11609208 IC50 = 440 nM T68251 D0L6ND 10089677 IC50 = 1.7 ug.mL-1 T68251 D0N8YA 159596 IC50 = 15000 nM T68251 D0NP8A 10370504 IC50 = 1790 nM T68251 D0NV9C 22004198 IC50 = 40 nM T68251 D0P2TS 9818682 IC50 > 60000 nM T68251 D0Q4TA 10044321 IC50 = 12 nM T68251 D0Q9LC 44385624 IC50 = 868 nM T68251 D0R2BO 194777 IC50 = 0.7 nM T68251 D0S9OL 10155934 IC50 = 1200 nM T68251 D0T1FR 44457233 IC50 = 4000 nM T68251 D0UI1P 46228278 IC50 = 178600 nM T68251 D0V9EN 689043 IC50 = 24.26 nM T68251 D0VI2A 44447430 IC50 = 537 nM T68251 D0W2UK 6914621 Ki = 2050 nM T68251 D0W3ME 4369080 Ki = 3000 nM T68251 D0XK7G 10445302 IC50 = 32 nM T68251 D0Y1XM 44423686 IC50 = 33700 nM T68251 D0Y5IQ 44255320 IC50 = 5000 nM T68251 D0Y7NV 2220392 IC50 = 898 nM T68251 D0Z4LO 9832179 IC50 = 23 nM T68251 D0Z4NU 46228282 IC50 = 285900 nM T72319 CV39DH 1072048 Ki = 33100 nM T72319 C64ZSL 43430547 IC50 > 30000 nM T72319 CQ4P5B 44755448 IC50 > 30000 nM T72319 C3NE8O 46931242 IC50 > 30000 nM T72319 C6O8RT 55872720 IC50 > 30000 nM T72319 C2P7SD 56577044 IC50 > 10000 nM T72319 CXY3E4 57720618 IC50 > 30000 nM T72319 CY9Z8F 60735522 IC50 > 30000 nM T72319 CB0SA4 61041645 IC50 > 30000 nM T72319 CT9M2C 61041646 IC50 > 30000 nM T72319 C3I5DM 61041804 IC50 > 30000 nM T72319 C84MGB 61242835 IC50 > 30000 nM T72319 C0Y6KO 62947261 IC50 > 30000 nM T72319 C8XEI4 63259457 IC50 > 30000 nM T72319 C0WX5O 70679311 IC50 > 30000 nM T72319 CEW3R6 71598546 IC50 > 30000 nM T72319 CUD65X 73333125 IC50 > 10000 nM T72319 CHQ18I 73333126 IC50 > 10000 nM T72319 C9UDN1 73333127 IC50 > 10000 nM T72319 C9K1NV 73333128 IC50 > 10000 nM T72319 C4UE6G 73333129 IC50 > 10000 nM T72319 CV2SJ4 73333225 IC50 > 10000 nM T72319 CF8HO3 73333226 IC50 > 10000 nM T72319 CVH9F0 73333227 IC50 > 10000 nM T72319 C4PYG2 73333229 IC50 > 10000 nM T72319 CBJC52 73333322 IC50 > 10000 nM T72319 CVEN67 73334066 IC50 > 10000 nM T72319 CYL3M7 73334067 IC50 > 10000 nM T72319 C6T7YX 73334068 IC50 > 10000 nM T72319 C70XCT 73334069 IC50 > 10000 nM T72319 C8QWP1 73334070 IC50 > 10000 nM T72319 CR98DL 73334157 IC50 > 10000 nM T72319 CJD9C1 73334158 IC50 > 10000 nM T72319 CLRM71 73334159 IC50 > 10000 nM T72319 C43NER 73334160 IC50 > 10000 nM T72319 CD2HX4 73334161 IC50 > 10000 nM T72319 CC89FN 73334162 IC50 > 10000 nM T72319 COV3R1 73334262 IC50 > 10000 nM T72319 CZD0N1 73334263 IC50 > 10000 nM T72319 CU3KG0 73334264 IC50 > 10000 nM T72319 CMLV27 73334265 IC50 > 10000 nM T72319 CD0VK7 73334266 IC50 > 10000 nM T72319 C1SGJ3 73334267 IC50 > 10000 nM T72319 C3PYF5 73334361 IC50 > 10000 nM T72319 C8H9JF 73334363 IC50 > 10000 nM T72319 C8XE1J 73334364 IC50 > 10000 nM T72319 CN40ZI 73334365 IC50 > 10000 nM T72319 CF9GA5 73334366 IC50 > 10000 nM T72319 C69WLM 73334479 IC50 > 10000 nM T72319 CG32QB 73334480 IC50 > 10000 nM T72319 CVE0S2 73334481 IC50 > 10000 nM T72319 C2S8XN 73334482 IC50 > 10000 nM T72319 CXJP87 73334483 IC50 > 10000 nM T72319 C57KSE 73334484 IC50 > 10000 nM T72319 CAQ18T 73334592 IC50 > 10000 nM T72319 CA67YG 73334593 IC50 > 10000 nM T72319 CNS84D 73334594 IC50 > 10000 nM T72319 C93HWE 73334595 IC50 > 10000 nM T72319 C87UBE 73334596 IC50 > 10000 nM T72319 CKSY83 73334696 IC50 > 10000 nM T72319 C36QHM 73334697 IC50 > 10000 nM T72319 CF63HU 73334698 IC50 > 10000 nM T72319 CQBX27 73334699 IC50 > 10000 nM T72319 C0OW1V 73334700 IC50 > 10000 nM T72319 C2VFJ9 73349256 IC50 > 30000 nM T72319 CG80NF 73349257 IC50 > 10000 nM T72319 COY1J2 73349259 IC50 > 10000 nM T72319 CNO9Z5 73350843 IC50 > 10000 nM T72319 C8U0ZX 73352326 IC50 > 10000 nM T72319 CRZ62F 73355036 IC50 = 8100 nM T72319 CD26ZM 73386663 IC50 = 73000 nM T72319 C2OXQ5 76314887 IC50 > 30000 nM T72319 C3X7EW 76314888 IC50 > 30000 nM T72319 C1YKN5 76314889 IC50 > 30000 nM T72319 C4E1BN 76318504 IC50 > 30000 nM T72319 CF76CT 76318505 IC50 > 30000 nM T72319 CLVA91 76318506 IC50 > 30000 nM T72319 C9LNK4 76318507 IC50 > 30000 nM T72319 CL87KC 76318508 IC50 > 30000 nM T72319 CET23F 76318509 IC50 > 30000 nM T72319 C01JLF 76322168 IC50 > 30000 nM T72319 C2SEM0 76322169 IC50 > 30000 nM T72319 CRH48X 76322170 IC50 > 30000 nM T72319 C5CZV2 76325789 IC50 > 30000 nM T72319 CS6GL0 76333019 IC50 > 30000 nM T72319 C7IUX5 76333020 IC50 > 30000 nM T72319 CZC8W2 76336632 IC50 > 30000 nM T72319 CYQ0B9 76336633 IC50 > 30000 nM T72319 CK2N0L 76336634 IC50 > 30000 nM T72319 CS4W5I 76336635 IC50 > 30000 nM T72319 CM6H9O 76336636 IC50 > 30000 nM T72319 CL8E1A 83748040 IC50 > 30000 nM T72319 CK5MX8 90655573 IC50 = 11000 nM T72319 C0S3XK 90655574 IC50 = 6800 nM T72319 CC50PO 90655575 IC50 = 5700 nM T72319 CA07UL 90655576 IC50 = 67000 nM T72319 CSUT18 90655577 IC50 = 23000 nM T72319 CD43OR 90655578 IC50 = 62000 nM T72319 C2A3RQ 90655579 IC50 = 35000 nM T72319 CEOP54 90655580 IC50 = 10100 nM T72319 CAM67V 90655581 IC50 = 10300 nM T72319 CLR17Q 90655582 IC50 = 13000 nM T72319 C28HZW 90655583 IC50 = 11000 nM T72319 CA1Y5I 90655584 IC50 = 21000 nM T72319 CQY83C 90655585 IC50 = 11200 nM T72319 CQTF13 90655586 IC50 = 6000 nM T72319 C83EFC 90655587 IC50 = 8800 nM T72319 C25ZNR 90655588 IC50 = 39000 nM T72319 C0GIC4 90655589 IC50 = 120000 nM T72319 CR6VS0 90655590 IC50 = 53000 nM T72319 C6KU2N 90655591 IC50 > 500000 nM T72319 C65HLO 90655592 IC50 = 9000 nM T72319 C4ACU9 90655593 IC50 = 79000 nM T72319 C74MKT 90655594 IC50 = 560000 nM T72319 CM21PY 90655595 IC50 > 250000 nM T72319 C78GYV 90655596 IC50 > 500000 nM T72319 C86DBC 90655597 IC50 > 250000 nM T72319 C9QU1T 90655598 IC50 > 250000 nM T72319 CWXY79 90655599 IC50 = 35000 nM T72319 C8M3HN 90655600 IC50 = 102000 nM T72319 C1MDL6 90655601 IC50 = 26000 nM T72319 C1MDK2 90655602 IC50 = 23000 nM T72319 CCD42S 90655603 IC50 = 22000 nM T72319 C7C9MF 90655604 IC50 = 105000 nM T72319 C27CIT 90655605 IC50 = 8600 nM T72319 C9PUC5 90655606 IC50 = 7800 nM T72319 CK2F6S 90655607 IC50 = 26000 nM T72319 C5T9WY 90655608 IC50 = 57000 nM T72319 C2EUX8 90655609 IC50 = 91000 nM T72319 C2A3CS 90655610 IC50 = 23000 nM T72319 C45VLK 90655611 IC50 = 89000 nM T72319 CN54XB 90655612 IC50 = 26000 nM T72319 C14LVC 90655613 IC50 = 67000 nM T72319 C64DAW 90655614 IC50 = 58000 nM T72319 C5H9VJ 90655615 IC50 = 100000 nM T72319 C9Z6BP 90655616 IC50 = 58000 nM T72319 C31VJO 90655617 IC50 > 250000 nM T72319 CAFW32 90655618 IC50 > 250000 nM T72319 CNZ4D8 90655619 IC50 = 34000 nM T72319 CY1PL8 90655620 IC50 = 53000 nM T72319 C5F6MO 90655621 IC50 > 2000000 nM T72319 C54UJD 90655622 IC50 > 2000000 nM T72319 C3OB0Z 90655623 IC50 = 4600 nM T72319 CW2ND5 90655624 IC50 = 6200 nM T72319 C87RLM 90655625 IC50 = 6300 nM T72319 C05HED 90655626 IC50 = 6700 nM T72319 C2BM7J 90655627 IC50 > 250000 nM T72319 CM51GQ 90655628 IC50 = 8800 nM T72319 CSL98F 90655629 IC50 = 57000 nM T72319 CLT0P1 90655635 IC50 = 27000 nM T72319 CW25YP 90666882 IC50 > 30000 nM T72319 CQI7D0 90666883 IC50 > 30000 nM T72319 C72IZG 90666884 IC50 > 30000 nM T72319 CCDK35 90666885 IC50 > 30000 nM T72319 C2DCW6 90666886 IC50 > 30000 nM T72319 CXN36J 90666887 IC50 > 30000 nM T72319 CG2S0B 90666888 IC50 > 30000 nM T72319 C19VSG 90666889 IC50 > 30000 nM T72319 CBG12J 90666890 IC50 > 30000 nM T72319 C90LPT 90666891 IC50 > 30000 nM T72319 C0IOH4 90666892 IC50 > 30000 nM T72319 C1CU2X 101043861 IC50 = 37 nM T72319 C0YL6Q 102602632 IC50 = 16000 nM T72319 C4Z1BN 102602634 IC50 = 130 nM T72319 C30MVB 127034580 IC50 = 1700 nM T72319 CR72CK 127044991 Ki = 25000 nM T72319 CVT1R7 127044992 Ki = 10000 nM T72319 CFJ30Y 127044993 Ki = 16900 nM T72319 CWA1V6 127044994 Ki = 10000 nM T72319 CMY6T7 127045145 Ki = 4800 nM T72319 CW6BT0 127045602 Ki = 39300 nM T72319 C6NBV2 134130627 IC50 = 35 nM T72319 COEW21 134131637 IC50 > 60000 nM T72319 C9XOG1 134131644 IC50 > 60000 nM T72319 CUW67R 134133875 IC50 = 240 nM T72319 CA1LH4 134133965 IC50 > 60000 nM T72319 C7PCM8 134134706 IC50 > 60000 nM T72319 C3PR2V 134134858 IC50 = 3100 nM T72319 CZB51D 134137731 IC50 = 51000 nM T72319 CKI23U 134139941 IC50 > 60000 nM T72319 C1OEI2 134140369 IC50 > 60000 nM T72319 C62JBE 134141602 IC50 = 220 nM T72319 CB20QF 134142297 IC50 > 60000 nM T72319 C29JUC 134142686 IC50 = 56 nM T72319 CS69VL 134143576 IC50 = 25000 nM T72319 C3XG2N 134144118 IC50 = 81 nM T72319 CZ83CB 134144237 IC50 = 51000 nM T72319 C48DSU 134145156 IC50 > 60000 nM T72319 C5C0HU 134145218 IC50 = 32000 nM T72319 CX1QB4 134145347 IC50 = 53000 nM T72319 C5IMF8 134145736 IC50 > 60000 nM T72319 CQX43Z 134145760 IC50 = 570 nM T72319 CX71GT 134146508 IC50 = 47 nM T72319 CE0C7P 134146658 IC50 = 740 nM T72319 CJY6D2 134146764 IC50 > 60000 nM T72319 C7NBT1 134148174 IC50 = 1700 nM T72319 C02JMB 134148668 IC50 = 61 nM T72319 CTL0D2 134149263 IC50 = 1200 nM T72319 C3BD1U 134149299 IC50 = 250 nM T72319 CS73OF 134149994 IC50 = 41000 nM T72319 C1MLU3 134151077 IC50 > 60000 nM T72319 C21YGK 134151685 IC50 > 60000 nM T72319 CES73F 134152016 IC50 = 1100 nM T72319 CIZV46 134152824 IC50 > 60000 nM T72319 C38AYE 134153154 IC50 = 230 nM T72319 CD5VJ0 134153698 IC50 = 18000 nM T72319 C4C7VM 134154055 IC50 = 75 nM T72319 CPAK59 134154083 IC50 = 4400 nM T72319 C9SAU3 134154301 IC50 = 32 nM T72319 CVK52O 134155339 IC50 = 35 nM T72319 CUH81S 134156240 IC50 = 26000 nM T72319 CB3YE8 134156251 IC50 = 63 nM T72319 CQ35RF 134157076 IC50 > 60000 nM T72319 CU0Z1S 134157587 IC50 = 28000 nM T72319 CFHK68 134157612 IC50 = 2600 nM T72319 D0W9RR 57339144 IC50 > 10000 nM T97353 D01TJY 53340771 IC50 > 10 nM T97353 CS24BW 11973730 IC50 = 15 nM T97353 CG3FV0 16727128 IC50 = 214 nM T97353 CAVY89 23636144 IC50 = 102 nM T97353 C1VUH4 23636254 IC50 = 17 nM T97353 C6LR7V 23636255 IC50 = 50 nM T97353 C5MSF6 23636502 IC50 = 29 nM T97353 C8B7QE 72949858 IC50 > 5000 nM T97353 C5ALQ2 76285468 IC50 = 4 nM T97353 CQ8BX7 76310576 IC50 = 163 nM T97353 C0JKX6 76310577 IC50 = 588 nM T97353 CUAH40 76310578 IC50 = 978 nM T97353 C4EK9U 76310579 IC50 > 4000 nM T97353 COZ54T 76310580 IC50 > 1000 nM T97353 CHI2U7 76310581 IC50 > 1000 nM T97353 COI21T 76310597 IC50 = 34 nM T97353 CL3EO0 76310599 IC50 = 470 nM T97353 CA9X2E 76310600 IC50 > 4000 nM T97353 CT1AJ4 76314216 IC50 = 114 nM T97353 C90ZKU 76314217 IC50 = 233 nM T97353 CA42YR 76314218 IC50 = 731 nM T97353 CXQ41E 76314219 IC50 > 10000 nM T97353 CUHZ51 76314232 IC50 = 667 nM T97353 COQ48X 76314233 IC50 = 1297 nM T97353 C1M7ZG 76317786 IC50 = 178 nM T97353 CIQ0T7 76317787 IC50 = 745 nM T97353 C1I6HO 76317788 IC50 = 1050 nM T97353 CSA72F 76317789 IC50 > 1000 nM T97353 CC3U8I 76317804 IC50 > 1000 nM T97353 C5UPA9 76317805 IC50 = 366 nM T97353 CBR9F0 76317806 IC50 = 36 nM T97353 CV23LI 76317807 IC50 > 5000 nM T97353 C0O4QY 76321498 IC50 = 101 nM T97353 CG7H4W 76321513 IC50 = 792 nM T97353 C1BQF4 76321514 IC50 = 38 nM T97353 C2ZH7K 76321515 IC50 = 497 nM T97353 CS9W7I 76321516 IC50 = 909 nM T97353 C7HC0P 76321517 IC50 > 4000 nM T97353 C8QH1P 76321518 IC50 = 731 nM T97353 CI9T5J 76325099 IC50 = 142 nM T97353 C2C6EW 76325100 IC50 > 4000 nM T97353 CSVC17 76325118 IC50 > 4000 nM T97353 CMH79B 76325119 IC50 = 12 nM T97353 C1HJO0 76325120 IC50 = 869 nM T97353 CCN7M6 76328682 IC50 = 1900 nM T97353 CP7AC0 76328683 IC50 > 5000 nM T97353 CX3Y7N 76328684 IC50 = 270 nM T97353 CZM19H 76332361 IC50 = 134 nM T97353 C18OJH 76332362 IC50 = 176 nM T97353 CA1LM2 76335971 IC50 = 106 nM T97353 C4I5DV 76335989 IC50 > 1000 nM T97353 CVI67F 90665342 EC50 = 2000 nM T19567 C3MA9U 342139 Ki = 3200 nM T19567 CDUE24 778225 IC50 < 200 nM T19567 CL16MS 822778 IC50 = 1000 nM T19567 CDX3Q5 5289024 Ki = 10 nM T19567 C7W8IX 5486943 Ki = 46 nM T19567 C3X1UJ 11507040 Ki = 600 nM T19567 C8N6MC 24808481 Ki = 420 nM T19567 C75WCL 52949691 Ki = 700 nM T19567 C54CBK 54585170 Ki = 5900 nM T19567 CTL94E 57520838 Ki = 9.4 nM T19567 CJQ9O0 57520839 Ki = 11 nM T19567 C8S9PM 57520840 Ki > 3000 nM T19567 C9G2HN 57520841 Ki = 50 nM T19567 C3N4MF 57520842 Ki = 29 nM T19567 CU4NZ2 57520938 Ki = 41 nM T19567 CD0M8V 57520940 Ki = 14 nM T19567 CCS1L3 57520941 Ki = 0.53 nM T19567 CEL56T 57520942 Ki = 20 nM T19567 CM6RX9 57520943 Ki = 9 nM T19567 C9Q4XE 57520944 Ki = 180 nM T19567 C1Z0LC 57520945 Ki = 1200 nM T19567 CE09OR 57520946 Ki = 200 nM T19567 C3Z6AE 57521037 Ki = 14 nM T19567 C6XB7H 57521039 Ki = 2.4 nM T19567 CXN9G4 57521040 Ki = 74 nM T19567 C9RU7B 57521041 Ki = 760 nM T19567 CC6UT9 57521043 Ki = 26 nM T19567 C78HYG 57521133 Ki = 0.36 nM T19567 C42KWH 57521134 Ki = 5.3 nM T19567 C9DFB0 57521135 Ki > 3000 nM T19567 C6SZ1P 57521138 Ki = 50 nM T19567 CR23AT 57521139 Ki = 58 nM T19567 CCQM76 59153288 Ki = 5.5 nM T19567 C4K2LU 59153299 Ki = 5.6 nM T19567 CK76DI 60202405 Ki = 2.8 nM T19567 C2LBW7 66551925 Ki = 190 nM T19567 C9CZS3 67205978 Ki = 70 nM T19567 C10MDK 69082696 Ki = 13 nM T19567 C39VMJ 69082892 Ki = 3.3 nM T19567 CYH83A 69083992 Ki = 1800 nM T19567 CT1PN0 69084444 Ki = 1700 nM T19567 CPV2D7 69085518 Ki = 960 nM T19567 CBZ82I 69085541 Ki = 72 nM T19567 CY2W3Z 69085646 Ki > 3000 nM T19567 C6BE5X 71271461 Ki = 270 nM T19567 C74PAB 86223063 Ki = 2200 nM T19567 CL0ZX5 86223064 Ki > 100000 nM T19567 CPT0J9 86275056 IC50 < 200 nM T19567 CIOU35 86275306 IC50 = 1000 nM T19567 CT4E5W 102436701 Ki = 4.1 nM T19567 C53VJW 135301646 IC50 = 3.715 nM T19567 C26OPR 135301656 IC50 = 147.91 nM T19567 CZVS32 135301671 IC50 = 3.89 nM T19567 CZJV94 135301685 IC50 = 18.2 nM T19567 CS4UK6 135301687 IC50 = 181.97 nM T19567 C9LA1K 135301762 IC50 = 20.42 nM T19567 CVW5G9 135301817 IC50 = 77.62 nM T19567 CG93EF 135301914 IC50 = 6.026 nM T19567 CGL0U2 135301919 IC50 = 13.18 nM T19567 C94GAU 135301927 IC50 = 2630.27 nM T19567 CY4MV6 135566354 Ki = 0.41 nM T19567 C4OVP2 136416802 Ki = 44 nM T19567 C7ZCT8 136416815 Ki = 69 nM T19567 C1OA7D 136416820 Ki = 0.55 nM T19567 C50OXS 136416829 Ki = 23 nM T19567 CX54DV 136416830 Ki = 28 nM T19567 CH94UL 136416849 Ki = 7.9 nM T19567 C9L0UB 136416923 Ki = 3 nM T19567 C0QWG9 142408858 IC50 = 10.23 nM T19567 CLZ91U 145971636 Ki > 200000 nM T19567 C4YPL9 145972068 Ki = 3460 nM T19567 CZVU97 155511644 Ki = 800 nM T19567 CMI8N3 155513321 Ki = 1600 nM T19567 C2CI4A 155514380 Ki = 600 nM T19567 CJ45PR 155520478 Ki = 2000 nM T19567 C95LZD 155522194 Ki = 700 nM T19567 CA35VB 155524076 Ki = 2100 nM T19567 C2QA1Z 155525301 Ki = 3200 nM T19567 C1E0UF 155535661 Ki = 3800 nM T19567 C2DI7E 155536657 IC50 = 3700 nM T19567 C3K1BZ 155537205 Ki = 15900 nM T19567 C9F2JN 155538608 Ki = 35 nM T19567 C5T9KE 155542416 Ki > 3000 nM T19567 C08TBV 155543421 IC50 = 223.87 nM T19567 C9S4MT 155549437 Ki = 1200 nM T19567 CAM36F 155550472 Ki = 3500 nM T19567 C3XE9Y 155554199 Ki = 900 nM T19567 C3WT2Q 155556441 Ki > 3000 nM T19567 C3PHB1 155557026 Ki = 2200 nM T19567 C3FA0E 155558092 Ki = 6700 nM T19567 C2I8VX 155559220 Ki = 8300 nM T19567 CUH07S 155560032 IC50 = 25000 nM T19567 CC5FE7 155564581 Ki > 3000 nM T19567 CB1V8A 155564612 Ki > 3000 nM T84621 D02STN 132971 IC50 = 1608 nM T84621 D02YPG 667484 IC50 = 0.5 nM T84621 D07ABV 468595 IC50 = 310 nM T84621 D09LNI 3365 IC50 = 30000 nM T84621 D0C1WH 3902 IC50 = 2620 nM T84621 D0Q9JT 4174 IC50 = 14.6 nM T84621 D0ZX1P 59693 IC50 = 6.3 nM T84621 D03AJU 44139752 IC50 = 2.5 nM T84621 D0D3PF 6918191 IC50 = 95000 nM T84621 D0SX7F 60876 Ki = 35 nM T84621 C9LCD8 3823 IC50 = 127 nM T84621 CFO8Y3 83332 IC50 = 24800 nM T84621 C78IXN 563347 IC50 = 246 nM T84621 CNG05O 571156 IC50 = 779 nM T84621 C5NT4U 583968 IC50 = 24 nM T84621 C1Y5HM 603115 IC50 = 16700 nM T84621 C8HZL4 618231 IC50 = 3 nM T84621 C7XD4N 706178 IC50 = 10200 nM T84621 CJ4FE1 853038 IC50 = 635 nM T84621 CI16RF 867617 IC50 = 500 nM T84621 CC29WP 886929 IC50 = 194 nM T84621 C6S1WJ 955210 IC50 > 1000 nM T84621 CB5KN2 1118253 IC50 = 14300 nM T84621 C83OBD 3021561 IC50 = 763 nM T84621 CBY4W2 3102914 IC50 > 1000 nM T84621 C1JAT6 6539761 IC50 = 715 nM T84621 CTE57C 6539762 IC50 = 1424 nM T84621 CF17BE 6539771 IC50 = 903 nM T84621 CJ7RS8 6539772 IC50 = 206 nM T84621 CQD13Z 6539787 IC50 = 143 nM T84621 CQ0HD5 6539812 IC50 = 58 nM T84621 CQ9XM0 6539813 IC50 = 26 nM T84621 CP51TH 6539814 IC50 = 96 nM T84621 CP4VI2 6540030 IC50 = 31.4 nM T84621 CR6LS8 6540031 IC50 = 3.3 nM T84621 CU3C1Y 6540034 IC50 = 6.9 nM T84621 CXEW82 6540035 IC50 = 15 nM T84621 CBKX32 6540037 IC50 = 18.7 nM T84621 C8MRI7 6540038 IC50 = 20.6 nM T84621 C8JXY1 6540039 IC50 = 11.17 nM T84621 CZK3T4 6540040 IC50 = 28.7 nM T84621 CDS26H 6540041 IC50 = 19.5 nM T84621 CX38PV 9927427 IC50 = 2 nM T84621 C64PHS 10083522 IC50 = 75000 nM T84621 CTH96I 10584844 IC50 = 5 nM T84621 CA13SW 10711620 IC50 = 79 nM T84621 CZW6V4 10828130 IC50 = 13.4 nM T84621 C6G3JV 11032034 IC50 = 47.86 nM T84621 C1TP7W 11232831 IC50 = 72 nM T84621 CN4T0K 11544009 IC50 = 4898 nM T84621 C9IJ3T 11594132 IC50 = 10505 nM T84621 CW2B3A 11738647 IC50 = 933 nM T84621 C27WEU 12229396 IC50 = 32 nM T84621 CCU19N 13045366 IC50 = 61 nM T84621 C4ELY3 13276694 IC50 = 2848 nM T84621 C1F5IT 13688212 IC50 = 40 nM T84621 C8WU6R 14424120 IC50 = 663 nM T84621 C8LSJ6 15182477 IC50 = 76000 nM T84621 CQ03PZ 16654684 IC50 = 816 nM T84621 CY0RV3 18668566 IC50 = 15 nM T84621 CRDM03 18679298 IC50 = 48 nM T84621 CN8IQ3 18785133 IC50 = 30.9 nM T84621 C1R2FU 22406650 IC50 = 253 nM T84621 C6D2NZ 24692916 IC50 = 1000 nM T84621 C07XJP 24696760 IC50 = 7500 nM T84621 CW3C5U 24896569 IC50 = 4329 nM T84621 C29WQM 25033651 IC50 = 291 nM T84621 C1VPF8 25033652 IC50 = 3109 nM T84621 C9Q8ZK 25033657 IC50 > 20000 nM T84621 CWIC10 25033659 IC50 > 10000 nM T84621 CAI47X 25033725 IC50 > 5000 nM T84621 C1XW6O 25033727 IC50 = 2135 nM T84621 CW5A1U 25033730 IC50 = 1159 nM T84621 CV49HP 25033731 IC50 = 686 nM T84621 C86AIT 25033734 IC50 > 10000 nM T84621 CEJ89P 25033804 IC50 = 2748 nM T84621 C3UF1V 25033806 IC50 = 1076 nM T84621 CF46OB 25033808 IC50 > 20000 nM T84621 CBI59C 25033810 IC50 = 1370 nM T84621 CV19DG 25034278 IC50 = 461 nM T84621 CEP93C 25034345 IC50 = 100 nM T84621 CSX16E 25034347 IC50 = 15 nM T84621 CXDF80 25034348 IC50 = 255 nM T84621 C56WJS 25034349 IC50 = 199 nM T84621 CGD93B 25034350 IC50 = 614 nM T84621 CK3L1J 25034351 IC50 = 1760 nM T84621 C9MF8O 25034425 IC50 = 99 nM T84621 CW7V9I 25034428 IC50 = 64 nM T84621 CH6U1E 25034429 IC50 = 248 nM T84621 CLP17I 25034432 IC50 = 875 nM T84621 CTB95M 25034489 IC50 = 41557 nM T84621 CBLS47 25034490 IC50 = 37796 nM T84621 CW82MN 25034491 IC50 = 31 nM T84621 CJ8M0E 25034492 IC50 = 435 nM T84621 COSJ63 25034493 IC50 = 10 nM T84621 C7KAR1 25034657 IC50 > 10000 nM T84621 C0MEI5 25129119 IC50 = 1956 nM T84621 C2QU1N 25129120 IC50 = 3559 nM T84621 C2FE6G 25129122 IC50 = 2452 nM T84621 CJ48LA 25129123 IC50 = 785 nM T84621 CX4GM7 25129462 IC50 = 24003 nM T84621 C9IFV2 25129463 IC50 = 19816 nM T84621 C6D8UQ 25129464 IC50 = 11307 nM T84621 CJCE15 25130854 IC50 = 1811 nM T84621 C9AS7H 25131165 IC50 = 2936 nM T84621 C9G8MJ 25131494 IC50 = 735 nM T84621 CA7OP2 25131495 IC50 = 9639 nM T84621 CZX08M 25142015 Ki = 15 nM T84621 C1WM2B 25147691 IC50 = 6.9 nM T84621 CYT15G 25180102 IC50 = 5970 nM T84621 CGX76Y 25180105 IC50 = 4371 nM T84621 CMU54R 25180107 IC50 = 290 nM T84621 C0XHA2 25180109 IC50 = 742 nM T84621 C9LQJ6 25180110 IC50 = 5177 nM T84621 CHJ2S3 25180298 IC50 = 339 nM T84621 C1HGB6 25180299 IC50 = 1671 nM T84621 C90UKD 25180304 IC50 = 1145 nM T84621 CPQ6A9 25180305 IC50 = 745 nM T84621 C6ZE9H 25180500 IC50 = 191 nM T84621 C6FN2Z 25180502 IC50 = 5402 nM T84621 C9DB1G 25180503 IC50 = 87 nM T84621 CIZ82U 25180504 IC50 = 769 nM T84621 CJS97E 30507078 IC50 = 5920 nM T84621 C70VMZ 44203017 IC50 = 1987 nM T84621 CT3XM4 44206480 IC50 = 116 nM T84621 C9UWB5 44206481 IC50 = 57 nM T84621 CDTS58 44387709 IC50 = 12.3 nM T84621 CT4L0R 44455927 IC50 = 19 nM T84621 C69QUY 44456068 IC50 > 1000 nM T84621 CM8BT1 44456104 IC50 = 110 nM T84621 C68FJH 44456188 IC50 = 167 nM T84621 CP50NM 44456189 IC50 = 329 nM T84621 CVR70K 44456190 IC50 = 782 nM T84621 C9JCL1 44456223 IC50 = 213 nM T84621 C6BE0T 44456226 IC50 = 107 nM T84621 CO4PI7 44479388 IC50 = 715 nM T84621 C1K6QY 44479389 IC50 = 2296 nM T84621 CLPH49 44479390 IC50 = 247 nM T84621 C2EM5N 44479391 IC50 = 13 nM T84621 CNTI30 44479392 IC50 = 545 nM T84621 C40IPE 44479393 IC50 = 34 nM T84621 C8JHS9 44479641 IC50 = 333 nM T84621 C2P4XT 44479643 IC50 = 158 nM T84621 CWP4Y8 44479644 IC50 = 141 nM T84621 C81QJE 44479645 IC50 = 1288 nM T84621 CO8T3N 44479646 IC50 = 2077 nM T84621 C4YN0S 44479648 IC50 = 28546 nM T84621 CF12OV 44479882 IC50 = 58 nM T84621 CCN58W 44479883 IC50 = 103 nM T84621 C7GV6X 44479884 IC50 = 17 nM T84621 CH8RO1 44479885 IC50 = 40 nM T84621 CES96D 44479886 IC50 = 490 nM T84621 CH02ZN 44480128 IC50 = 21 nM T84621 C1LSH2 44480129 IC50 = 1374 nM T84621 C3UQS0 44480130 IC50 = 43 nM T84621 C4KG5O 44480131 IC50 = 4646 nM T84621 COI7E8 44480132 IC50 = 496 nM T84621 C9KS5O 44480133 IC50 = 2058 nM T84621 CLMI41 44480134 IC50 = 128 nM T84621 CYH9A6 44480385 IC50 = 1312 nM T84621 C9V8CH 44480386 IC50 = 28 nM T84621 CL8KQ3 44480387 IC50 = 54 nM T84621 CT50NZ 44480388 IC50 = 796 nM T84621 CKO4N3 44480389 IC50 = 1692 nM T84621 CT3MO9 44480390 IC50 = 15 nM T84621 CN7LT2 44482245 IC50 = 776 nM T84621 CO63LK 44569291 IC50 = 152 nM T84621 CW06BV 45103704 IC50 = 104 nM T84621 C9Z4YB 45103705 IC50 = 123 nM T84621 CB2FC9 45103804 IC50 = 112.2 nM T84621 C4Q2FU 45103806 IC50 = 43.65 nM T84621 CQF56Z 45103807 IC50 = 12.02 nM T84621 C0RY2G 46233602 IC50 = 213 nM T84621 CUV83E 46854605 IC50 = 3100 nM T84621 CIA08B 46854608 IC50 = 37470 nM T84621 CWJ3F1 46854758 IC50 = 7300 nM T84621 CKRQ67 46854759 IC50 = 7180 nM T84621 CZ1YJ0 46854760 IC50 = 5060 nM T84621 CIC9S5 49799473 IC50 = 2000 nM T84621 C3Q6AS 49862488 IC50 = 26.1 nM T84621 CM43HV 49862547 IC50 = 50.2 nM T84621 CFDH59 49862548 IC50 = 103 nM T84621 CNIA98 49862549 IC50 = 544 nM T84621 CKY2J9 49862550 IC50 = 566 nM T84621 C0N4RT 49862551 IC50 = 930 nM T84621 CLI23H 49862552 IC50 = 122 nM T84621 CGU86D 49862599 IC50 = 55.7 nM T84621 CY8WD5 49862600 IC50 = 119 nM T84621 CS4IP9 49862601 IC50 = 76 nM T84621 C63XUS 49862602 IC50 = 204 nM T84621 C6O7JQ 49862603 IC50 = 471 nM T84621 C8G7FR 49862604 IC50 = 340 nM T84621 CP5D8Q 49862650 IC50 = 20.6 nM T84621 C6X0JA 49862651 IC50 = 222 nM T84621 C7BTK9 49862652 IC50 = 245 nM T84621 C79MQZ 49862653 IC50 = 234 nM T84621 CL8DR6 49862654 IC50 = 182 nM T84621 CMXR96 51355428 IC50 = 45 nM T84621 C5KTL3 51355429 IC50 = 40 nM T84621 C4UTM8 51355430 IC50 = 31 nM T84621 CH5C9K 51355431 IC50 = 20 nM T84621 CRK2Q9 51355432 IC50 = 5 nM T84621 CF7RG5 51355433 IC50 = 20 nM T84621 C41SUK 51355703 IC50 = 100 nM T84621 CM6T7H 51355704 IC50 = 80 nM T84621 CZDA87 51355705 IC50 = 25 nM T84621 CO1V0Y 51355706 IC50 = 45 nM T84621 C2OCG3 51355707 IC50 = 50 nM T84621 CIR0L7 51356252 IC50 = 933 nM T84621 CY69GL 52450897 IC50 = 188 nM T84621 CMTX50 52936939 IC50 = 2045 nM T84621 CC7Q8A 52936940 IC50 = 183 nM T84621 CTD3M1 52936941 IC50 = 1748 nM T84621 C98MZS 52937039 IC50 = 44 nM T84621 CZ72GJ 53316510 IC50 = 46 nM T84621 CR7L6V 53317838 IC50 = 80 nM T84621 CD9JL4 53319024 IC50 = 16100 nM T84621 CJBC94 53319146 IC50 > 1000 nM T84621 CYN7S9 53319147 IC50 = 43 nM T84621 C6WXT3 53320325 IC50 = 369 nM T84621 C20LRW 53320468 IC50 = 32 nM T84621 CU80BY 53320469 IC50 > 1000 nM T84621 C1SH0Q 53321768 IC50 > 1000 nM T84621 CEA3Y9 53321769 IC50 > 1000 nM T84621 C90DZC 53322953 IC50 = 5 nM T84621 CU1V2C 53323093 IC50 = 128 nM T84621 CYU1S5 53323094 IC50 > 1000 nM T84621 CS4A9O 53324450 IC50 = 46 nM T84621 C0B7TL 53325759 IC50 = 197 nM T84621 CVG4U6 53325760 IC50 = 4 nM T84621 CO68YD 53326854 IC50 = 75 nM T84621 C4NU2F 53475401 IC50 = 42 nM T84621 CAE25J 53763992 IC50 = 500 nM T84621 C51RVD 56645155 IC50 = 2857 nM T84621 CG06MB 56645361 IC50 = 401 nM T84621 CUS9L4 56645362 IC50 = 3984 nM T84621 C4N0WL 56645363 IC50 = 100 nM T84621 CTO1X9 56645364 IC50 = 370 nM T84621 C57NSZ 56645568 IC50 = 42 nM T84621 C6PUX9 56645570 IC50 = 435 nM T84621 CTW6K2 56645571 IC50 = 258 nM T84621 CX05HC 56645572 IC50 = 723 nM T84621 CPCW12 56645777 IC50 = 374 nM T84621 C32FWC 56645967 IC50 = 251 nM T84621 CXYW61 56645969 IC50 = 334 nM T84621 C2AP7F 56646158 IC50 = 435 nM T84621 CKWB83 56646160 IC50 = 477 nM T84621 CA3VO0 56949328 IC50 > 7500 nM T84621 CH8CP7 57329709 IC50 = 246 nM T84621 CQD5B4 57329785 IC50 = 76 nM T84621 C8GUF0 57329786 IC50 = 29 nM T84621 CE4YX9 57329787 IC50 = 40 nM T84621 CRAD59 57329788 IC50 = 72 nM T84621 CH8FQ9 57329789 IC50 = 101 nM T84621 C4USR5 57329791 IC50 = 62 nM T84621 C2C5PD 57329792 IC50 = 75 nM T84621 C3D8CZ 57329793 IC50 = 16 nM T84621 CKH02M 57329866 IC50 = 61 nM T84621 C30NOK 57329940 IC50 = 33 nM T84621 C37KZO 57329941 IC50 = 28 nM T84621 CZH28K 57329942 IC50 = 12 nM T84621 CR6EH0 57329943 IC50 = 151 nM T84621 CWN9V2 57329944 IC50 = 60 nM T84621 CFLA57 57330005 IC50 = 21 nM T84621 C2JR3S 57330006 IC50 = 11 nM T84621 C1EZM8 57330007 IC50 = 124 nM T84621 C5H2LE 57330008 IC50 = 69 nM T84621 C05XKT 57330009 IC50 = 98 nM T84621 C26GFC 57330010 IC50 = 32 nM T84621 CS38WC 57330011 IC50 = 6 nM T84621 C54EUF 57330012 IC50 = 1122 nM T84621 C4MN9B 57330078 IC50 = 1711 nM T84621 C5K3VT 57330079 IC50 = 240 nM T84621 C3LVG9 57330084 IC50 = 610 nM T84621 CMNH08 57330085 IC50 = 8 nM T84621 CY58ZD 57330086 IC50 = 2 nM T84621 C7OK1X 57775654 IC50 = 149 nM T84621 CB6RN7 58255346 IC50 = 50 nM T84621 CFXY47 58255349 IC50 = 29 nM T84621 C34JIZ 58255359 IC50 = 224 nM T84621 C7ZH6D 58255361 IC50 = 3.4 nM T84621 C2TUJ7 58255382 IC50 = 2.2 nM T84621 CMBV34 58255389 IC50 = 40 nM T84621 C3DPC0 58255407 IC50 = 40 nM T84621 C9DK1X 58255415 IC50 = 3737 nM T84621 CQEW75 58255430 IC50 = 144 nM T84621 CTI0D7 58255435 IC50 = 5399 nM T84621 C7L1NK 58255436 IC50 = 27 nM T84621 CRQ70M 58255438 IC50 = 1.4 nM T84621 C72VNQ 58255447 IC50 = 6.5 nM T84621 CLQ65O 58255479 IC50 = 347 nM T84621 CP6RA9 58255482 IC50 = 11940 nM T84621 C6DHG3 58255496 IC50 = 70 nM T84621 CAJ17Z 58255506 IC50 = 13 nM T84621 C7AX1R 58255531 IC50 = 110 nM T84621 CJX70M 58255566 IC50 = 745 nM T84621 C64JZC 58255572 IC50 = 438 nM T84621 CW71EO 58255581 IC50 = 2487 nM T84621 CYD9N5 58255637 IC50 = 20 nM T84621 CB7N8A 60195126 IC50 = 19 nM T84621 CX4N0I 62707515 IC50 = 790 nM T84621 CH3QU4 62918897 IC50 = 971 nM T84621 CE6L7O 65040275 IC50 > 10000 nM T84621 C0G3LA 66559847 IC50 = 1098 nM T84621 C4RSI6 66559935 IC50 = 1077 nM T84621 CDX7I8 66559936 IC50 = 1167 nM T84621 CF9EQ5 66559939 IC50 = 1422 nM T84621 CQN6D3 66559940 IC50 = 16170 nM T84621 CN4H8G 66559941 IC50 = 4087 nM T84621 CTP6Q4 66559942 IC50 = 4589 nM T84621 C9EGW2 66575742 IC50 = 3570 nM T84621 CMXA10 66575743 IC50 = 1770 nM T84621 CKWB91 66575744 IC50 = 110 nM T84621 C7I3MW 66575745 IC50 = 16990 nM T84621 CPN17S 66575746 IC50 = 12620 nM T84621 CG0ZA7 66575747 IC50 = 16100 nM T84621 C6HF0U 66575748 IC50 = 7900 nM T84621 CEW4O6 66575816 IC50 = 17296 nM T84621 CDI93T 66575817 IC50 = 428 nM T84621 C6B7PN 66576767 IC50 = 407 nM T84621 CYHS25 66576769 IC50 = 1501 nM T84621 CBP6I7 66576773 IC50 = 2198 nM T84621 CM6U5S 66576848 IC50 > 30000 nM T84621 CNB21T 66576849 IC50 > 10000 nM T84621 C2PFB6 66576850 IC50 > 10000 nM T84621 CDU8R7 66576852 IC50 = 6930 nM T84621 C4NYB0 66576930 IC50 = 1810 nM T84621 C3LP5H 66576931 IC50 = 3910 nM T84621 CE03WG 66576932 IC50 = 6970 nM T84621 CVZ4E0 66692998 IC50 > 10000 nM T84621 C1RLT0 67199421 IC50 = 3451 nM T84621 CC34QF 67509960 IC50 = 21 nM T84621 CQL7H6 67510362 IC50 = 167 nM T84621 CN9VU2 67510431 IC50 = 320 nM T84621 C40FEA 67511528 IC50 = 362 nM T84621 C2MH1G 67515607 IC50 = 126 nM T84621 CC4A7Z 67515696 IC50 = 106 nM T84621 CE27NZ 67515801 IC50 = 782 nM T84621 CZCW84 67515869 IC50 = 362 nM T84621 CKJN74 67515874 IC50 = 409 nM T84621 CW20PM 67516106 IC50 = 502 nM T84621 C14VNF 67516160 IC50 = 1000 nM T84621 CL0XQ7 67516179 IC50 = 971 nM T84621 CM7Z1T 67516370 IC50 = 95 nM T84621 CK1LB2 67516475 IC50 = 542 nM T84621 C5VM6T 67516855 IC50 = 139 nM T84621 CQ0NP7 68053462 IC50 > 10000 nM T84621 CV72CY 68053552 IC50 = 1980 nM T84621 CVF40X 68053622 IC50 = 1831 nM T84621 CG0T8B 68053623 IC50 = 2101 nM T84621 CU76KO 68053624 IC50 > 8333 nM T84621 CYZK18 68053631 IC50 > 8333 nM T84621 CSI12Z 68053632 IC50 > 10000 nM T84621 C0N3IK 68053729 IC50 = 17.7 nM T84621 C19JSA 68053730 IC50 = 250 nM T84621 C5N2MQ 68053837 IC50 = 677 nM T84621 CCJT39 68053838 IC50 = 3923 nM T84621 CF32HJ 70680985 IC50 = 500 nM T84621 CPB63L 70680997 IC50 = 73 nM T84621 CE78SM 70683110 IC50 = 168 nM T84621 CM6LN8 70683111 IC50 = 246 nM T84621 CK0DY6 70683112 IC50 = 611 nM T84621 C9E4ZQ 70685192 IC50 = 269 nM T84621 CW5F3G 70691516 IC50 = 500 nM T84621 C1VMF2 70977969 IC50 = 29540 nM T84621 C70TUP 71455138 IC50 = 139 nM T84621 CFG4L5 71456934 IC50 = 44 nM T84621 CI16NC 71520311 IC50 = 1336 nM T84621 CE9A6B 71520312 IC50 > 5000 nM T84621 C03VKJ 71520313 IC50 = 750 nM T84621 C5J7DI 71520314 IC50 = 16 nM T84621 CE0N5C 71520315 IC50 = 41 nM T84621 C4Z6YP 71520316 IC50 = 1230 nM T84621 CC8Z6L 71520431 IC50 = 4 nM T84621 C1DK9P 71520432 IC50 = 140 nM T84621 C9NOQ1 71521632 IC50 = 68 nM T84621 C0OTA2 71521716 IC50 = 2270 nM T84621 CVLE07 71521717 IC50 = 1220 nM T84621 CJKX84 71521718 IC50 = 36 nM T84621 CZ5P9U 71521719 IC50 = 78 nM T84621 C1YCB0 71521720 IC50 = 1420 nM T84621 CE57PM 71521721 IC50 > 5000 nM T84621 C0O2SA 71521798 IC50 = 276 nM T84621 CMEC10 71521799 IC50 = 2539 nM T84621 CR9O5T 71521800 IC50 = 1688 nM T84621 C0JBI3 71521801 IC50 = 532 nM T84621 CE7Z4I 71521802 IC50 = 88 nM T84621 CW2AG4 71521803 IC50 = 646 nM T84621 C6ID7K 71521804 IC50 = 92 nM T84621 CO5BE7 71535395 IC50 = 280 nM T84621 CCF8Z7 71535398 IC50 = 530 nM T84621 CC16AO 71535399 IC50 = 590 nM T84621 CPZ5S8 71535400 IC50 = 100 nM T84621 CI4W5N 71535682 IC50 = 490 nM T84621 CCRS95 71535683 IC50 = 1800 nM T84621 C58SMB 71574941 IC50 = 0.5 nM T84621 CC09FQ 71574942 IC50 = 19.2 nM T84621 CA2T5L 71574943 IC50 = 156.3 nM T84621 C9MFZ7 71574944 IC50 = 80.1 nM T84621 CW73OE 71574945 IC50 = 25.4 nM T84621 C70NHJ 71574946 IC50 = 92.5 nM T84621 CLH83S 71574947 IC50 = 24.4 nM T84621 CF71AB 71575030 IC50 = 13.1 nM T84621 CCG1S5 71575031 IC50 = 5.5 nM T84621 CH9WE7 71575032 IC50 = 268.4 nM T84621 CO4ZQ7 71575033 IC50 = 415.8 nM T84621 CT86GV 71575034 IC50 = 785.3 nM T84621 CKPV51 71621803 IC50 > 100000 nM T84621 CG09JH 71716351 IC50 = 72 nM T84621 C56LUJ 71716957 IC50 = 219 nM T84621 CJE01S 71745100 IC50 = 4520 nM T84621 CX0WV5 71817943 IC50 = 235 nM T84621 CN1LU6 71817944 IC50 = 1609 nM T84621 CGV4U3 71817945 IC50 = 1159 nM T84621 CJ4L5G 71818086 IC50 = 2935 nM T84621 COXA51 71818087 IC50 = 224 nM T84621 CP1A3M 71818088 IC50 = 1415 nM T84621 CPJ42T 71818089 IC50 = 450 nM T84621 CAP03I 71818090 IC50 = 447 nM T84621 CO23PK 71818091 IC50 = 245 nM T84621 CL4X6A 71818092 IC50 = 7099 nM T84621 CL8GK5 71818093 IC50 = 2824 nM T84621 C4ZVG0 71818094 IC50 = 362 nM T84621 CH2GR0 71818232 IC50 = 238 nM T84621 C0VGQ9 71818233 IC50 = 12286 nM T84621 C5QRF2 71818234 IC50 = 2426 nM T84621 CCG7R3 72703685 IC50 = 250 nM T84621 CAU4Z0 72703889 IC50 = 1010 nM T84621 C56KEC 72703890 IC50 = 1480 nM T84621 C4AEX3 73347616 IC50 = 38 nM T84621 CFD46C 73347617 IC50 = 5 nM T84621 C26LJW 73347618 IC50 = 1015 nM T84621 CIHF35 73350707 IC50 = 51 nM T84621 CT26EZ 73355186 IC50 > 5000 nM T84621 C0NXU4 73355187 IC50 = 87 nM T84621 CML29U 73355188 IC50 = 427 nM T84621 CC5TO4 73356735 IC50 = 125 nM T84621 CWZ3A1 73356736 IC50 = 1.3 nM T84621 C9CY3K 73442767 IC50 = 34 nM T84621 CU6IQ9 73603293 IC50 = 4737 nM T84621 C6MQ8L 73603294 IC50 > 5000 nM T84621 CR81XZ 73603295 IC50 = 1423 nM T84621 CJS6Y2 73603296 IC50 > 5000 nM T84621 C1GR7W 73603297 IC50 > 5000 nM T84621 CM4L6N 73603298 IC50 = 1523 nM T84621 CAIB62 73603299 IC50 > 5000 nM T84621 C7G6KZ 73603343 IC50 = 52 nM T84621 CDX9R1 73603344 IC50 = 516 nM T84621 C7KV2S 73603345 IC50 = 6093 nM T84621 CM10ZX 73603346 IC50 = 3723 nM T84621 CJSY07 73603348 IC50 = 1379 nM T84621 CS03UP 73603349 IC50 = 6812 nM T84621 C56LYP 73603350 IC50 = 6642 nM T84621 C9RKH0 73603387 IC50 = 803 nM T84621 CG86BD 73603388 IC50 = 3125 nM T84621 C2R3ZB 73603389 IC50 = 3756 nM T84621 C5ARE7 73603390 IC50 = 160 nM T84621 CTMF86 73603391 IC50 = 366 nM T84621 C5RG4C 75593332 IC50 = 10.74 nM T84621 CMN51L 76286753 IC50 > 8300 nM T84621 C06HYT 76286902 IC50 = 1299 nM T84621 CPU3T6 76317295 IC50 = 7.2 nM T84621 CZ2U9K 76321000 IC50 = 1.5 nM T84621 C4UO5H 76331904 IC50 < 0.1 nM T84621 CP10SN 76335488 IC50 = 0.3 nM T84621 C1YJW0 77846787 IC50 = 32 nM T84621 CV73PD 77846790 IC50 = 82 nM T84621 C0DIH7 77846872 IC50 = 17 nM T84621 COI25M 77846873 IC50 = 67 nM T84621 CJI8R0 77846875 IC50 = 29 nM T84621 CZK4J1 77846962 IC50 = 70 nM T84621 CEK89G 77846963 IC50 = 110 nM T84621 C5BA8Z 77846964 IC50 = 187 nM T84621 C4D6XJ 77847803 IC50 = 63 nM T84621 CF7O4Q 77847804 IC50 = 40 nM T84621 C2ASY0 86730379 IC50 = 880 nM T84621 CA4QV9 86730380 IC50 = 33 nM T84621 C24ZMT 86730381 IC50 = 37 nM T84621 C9W6RO 86730382 IC50 = 600 nM T84621 C3UMP9 89471867 IC50 = 640 nM T84621 CW8TF6 89471869 IC50 = 300 nM T84621 CL30TR 89471870 IC50 = 760 nM T84621 CJ0H5V 89471872 IC50 = 1100 nM T84621 C3BUS8 89471889 IC50 = 930 nM T84621 CI7HY8 89471890 IC50 = 800 nM T84621 CF2AY7 89471891 IC50 > 8700 nM T84621 CQF07X 89471892 IC50 = 830 nM T84621 C62KFZ 89961587 IC50 > 10000 nM T84621 C8XS2I 89961629 IC50 = 317 nM T84621 C75PMO 89961672 IC50 > 8333 nM T84621 CX0M7B 89961716 IC50 = 1357 nM T84621 C3JN5I 89961721 IC50 > 10000 nM T84621 CSJT14 89961765 IC50 = 1473 nM T84621 CR5D6Y 89961785 IC50 > 10000 nM T84621 C7TI3V 89961787 IC50 > 8333 nM T84621 C2QP7I 89961848 IC50 > 10000 nM T84621 C81FEN 89961879 IC50 > 10000 nM T84621 CI6P0R 89961978 IC50 > 8333 nM T84621 C89TEU 89968659 IC50 = 5705 nM T84621 C7BC5N 89968688 IC50 > 10000 nM T84621 C3XIF5 90252771 IC50 = 1.1 nM T84621 CGZ2S1 90252806 IC50 = 470 nM T84621 C4F9VB 90252809 IC50 = 1400 nM T84621 CE2TM0 90252810 IC50 > 8300 nM T84621 CGVL78 90252811 IC50 > 8300 nM T84621 C0S3HV 90252812 IC50 = 916 nM T84621 C4M8TO 90252814 IC50 = 1200 nM T84621 CM0T2X 90252815 IC50 > 8300 nM T84621 CY5IC7 90252834 IC50 = 98 nM T84621 CF05JI 90252835 IC50 = 1000 nM T84621 C72ICB 90252839 IC50 > 8300 nM T84621 C84NVA 90252850 IC50 = 338 nM T84621 CBY46O 90252851 IC50 = 856 nM T84621 CNVA50 90252852 IC50 = 386 nM T84621 C0Z2TI 90252864 IC50 = 47 nM T84621 CV30CD 90252953 IC50 = 535 nM T84621 C3MV7S 90252954 IC50 = 1690 nM T84621 CD5ST8 90252956 IC50 > 8300 nM T84621 C3JH4P 90252957 IC50 > 8300 nM T84621 CCU4F7 90252958 IC50 = 1987 nM T84621 C89BFG 90333640 IC50 = 58 nM T84621 C82YUB 90644545 IC50 = 302 nM T84621 CVFA18 90644546 IC50 = 736 nM T84621 CR50EN 90644547 IC50 = 61 nM T84621 C46ZNM 90644548 IC50 = 435 nM T84621 CS6N1P 90644549 IC50 = 4100 nM T84621 CB5HI4 90644550 IC50 = 2300 nM T84621 CHD21I 90666137 IC50 = 21.2 nM T84621 CLB2E7 91827654 IC50 = 4402 nM T84621 C5GV1L 101882447 IC50 = 5 nM T84621 CMH51N 118496543 IC50 = 779 nM T84621 C3ZPQ1 118496545 IC50 = 149 nM T84621 CJ9Z0S 118496546 IC50 = 22 nM T84621 C7UN3R 118496547 IC50 = 197 nM T84621 CJ54UQ 118618017 IC50 = 872 nM T84621 CLS25A 118714825 IC50 = 111 nM T84621 CT0FH7 118714826 IC50 = 327 nM T84621 CD8T1P 118714827 IC50 = 1674 nM T84621 C85BVO 118714828 IC50 = 690 nM T84621 CYFP62 118714829 IC50 = 499 nM T84621 CE3ZF1 118714830 IC50 = 2003 nM T84621 C5HKE1 118714831 IC50 = 1750 nM T84621 C7BD3X 118714832 IC50 = 587 nM T84621 C9BM7X 118714833 IC50 = 188 nM T84621 CML4K7 118714834 IC50 = 68 nM T84621 CE5L8U 118714835 IC50 = 2001 nM T84621 CD8YA9 118714836 IC50 > 5000 nM T84621 CRNL64 118714837 IC50 = 28 nM T84621 C4F6AY 118714838 IC50 = 65 nM T84621 CZ9L5S 118714839 IC50 = 334 nM T84621 CU3XP2 118714840 IC50 = 26 nM T84621 C0BRP1 118714841 IC50 = 278 nM T84621 C6M5VU 118714842 IC50 = 382 nM T84621 CQ5KI0 118714843 IC50 = 929 nM T84621 C32MDK 118714844 IC50 = 71 nM T84621 C15PAW 118714845 IC50 = 49 nM T84621 CPH51S 118714846 IC50 = 62 nM T84621 C1L4YZ 118714847 IC50 = 137 nM T84621 CLM64U 118714848 IC50 = 309 nM T84621 C5UD3K 118714849 IC50 = 1224 nM T84621 CNW8E3 118714850 IC50 = 65 nM T84621 CMXG03 118714851 IC50 = 114 nM T84621 CTWO23 118714852 IC50 = 60 nM T84621 CAW36P 118714853 IC50 = 663 nM T84621 C4Y2UF 118714854 IC50 = 1167 nM T84621 CJK08Q 118714855 IC50 = 6 nM T84621 CP4O0C 118720463 IC50 = 6712 nM T84621 CV4IC9 118720464 IC50 = 4196 nM T84621 CKG28R 118720465 IC50 = 7315 nM T84621 CGXD81 118720466 IC50 = 1096 nM T84621 CF1W7I 118720467 IC50 = 8947 nM T84621 COZU39 118720468 IC50 = 4797 nM T84621 CWG6L8 118720469 IC50 = 4487 nM T84621 C2HV3Y 118720470 IC50 = 5549 nM T84621 CX56BZ 118720471 IC50 = 6548 nM T84621 CO8H3J 118720472 IC50 = 7427 nM T84621 C7WEQ3 118720473 IC50 = 5812 nM T84621 CG8PB5 118720474 IC50 = 4710 nM T84621 CN2U6B 118720475 IC50 = 6189 nM T84621 CU7FW1 118720476 IC50 = 6674 nM T84621 CCJ17Z 118720477 IC50 = 5076 nM T84621 CB4DS9 118720479 IC50 = 8550 nM T84621 CC9V6K 118720480 IC50 = 8333 nM T84621 CP7X1B 118720481 IC50 = 9346 nM T84621 CPT58L 118720482 IC50 = 4717 nM T84621 C3E7TA 118720483 IC50 = 6534 nM T84621 CS01NU 118720484 IC50 = 6164 nM T84621 CAW5K3 118723935 IC50 = 48 nM T84621 CK8UL1 118723936 IC50 = 111 nM T84621 CIW7O0 118723937 IC50 = 63 nM T84621 C42CEZ 118723938 IC50 = 48 nM T84621 CJQ63E 118723939 IC50 = 258 nM T84621 CCXN71 118723940 IC50 = 57 nM T84621 CS78BD 118723941 IC50 = 50 nM T84621 C9W3QX 118723942 IC50 > 500 nM T84621 COJ2K8 118723943 IC50 = 15 nM T84621 CZ23UL 118723944 IC50 = 24 nM T84621 CIWU64 118723945 IC50 = 30 nM T84621 CZI6A0 118723946 IC50 = 109 nM T84621 COB46M 118723947 IC50 = 518 nM T84621 CYM08W 118726850 IC50 = 120 nM T84621 CR32JU 118726851 IC50 = 4.5 nM T84621 C2OAI6 118726852 IC50 = 7483 nM T84621 CDHI10 118733086 IC50 > 10000 nM T84621 C18PWB 118733087 IC50 > 10000 nM T84621 C8WJ2Y 118733088 IC50 > 10000 nM T84621 C31ZXP 118733089 IC50 > 10000 nM T84621 CHR84E 118733090 IC50 > 10000 nM T84621 CAQ72M 118733091 IC50 > 10000 nM T84621 CIV1Z5 118733092 IC50 > 10000 nM T84621 CU3Y9W 118733093 IC50 > 10000 nM T84621 CF49NU 118733094 IC50 > 10000 nM T84621 CK73VU 118733095 IC50 > 10000 nM T84621 CR1WU5 118733096 IC50 > 10000 nM T84621 C1V7WI 118735163 IC50 = 279 nM T84621 C6YG9R 118735164 IC50 = 1207 nM T84621 C5C4FZ 118735165 IC50 = 540 nM T84621 C1ZLM6 118735166 IC50 = 23 nM T84621 CQXM57 118735167 IC50 = 13 nM T84621 C0RYM4 118735168 IC50 = 6 nM T84621 C0DCB9 118735169 IC50 = 50 nM T84621 CG4QF3 118735170 IC50 = 2 nM T84621 CD3IY5 118735171 IC50 = 8 nM T84621 C0JZ2Y 118735172 IC50 = 508 nM T84621 C2WS7A 118735173 IC50 = 1201 nM T84621 CYEA24 118735174 IC50 = 51 nM T84621 CZ9X4J 118735175 IC50 = 60 nM T84621 CG14RD 118735176 IC50 = 183 nM T84621 CQ3KR4 118735177 IC50 = 46 nM T84621 C1Z9FX 118735178 IC50 = 812 nM T84621 C2VJU4 118735179 IC50 = 26 nM T84621 CXWH51 118735180 IC50 = 38 nM T84621 C3YUS9 118735181 IC50 = 12 nM T84621 CEH97S 118735182 IC50 = 594 nM T84621 C03HKR 118735183 IC50 = 1150 nM T84621 CC38HG 118735184 IC50 = 1665 nM T84621 C8QIC4 118735185 IC50 = 2665 nM T84621 CZET62 118735186 IC50 = 182 nM T84621 CZ8U2C 118735187 IC50 = 6 nM T84621 CUAE09 121004872 IC50 > 8333 nM T84621 C1OT4E 121458684 IC50 = 1552 nM T84621 C9ETN3 121458685 IC50 = 795 nM T84621 C4V2HU 121458987 IC50 = 225 nM T84621 CPGD72 121458994 IC50 = 117 nM T84621 CXW13O 122179553 IC50 > 10000 nM T84621 C3E0VM 122179554 IC50 > 10000 nM T84621 CJVX13 122179555 IC50 > 8333 nM T84621 CWN9K7 122179556 IC50 > 10000 nM T84621 CV2PQ1 122191831 IC50 > 8333 nM T84621 C2AHB5 122191832 IC50 > 8333 nM T84621 CFZH01 122191833 IC50 > 8333 nM T84621 C1XKA8 122191834 IC50 > 8333 nM T84621 CG4S8F 122191835 IC50 = 887 nM T84621 C37NLK 122191836 IC50 > 8333 nM T84621 CVT7A2 127027254 IC50 = 86.9 nM T84621 C5QNG6 127027265 IC50 > 10000 nM T84621 CIZO64 127027266 IC50 > 10000 nM T84621 C9RXH3 127027267 IC50 > 10000 nM T84621 CEM84R 127027569 IC50 = 1600.8 nM T84621 CT83ZE 127027570 IC50 = 326.9 nM T84621 CHZ54G 127027571 IC50 = 29.5 nM T84621 C2ZFR8 127027572 IC50 = 108.9 nM T84621 CV1BD6 127027573 IC50 = 9.7 nM T84621 C0E6DW 127027574 IC50 > 10000 nM T84621 C2MFJ8 127027575 IC50 > 10000 nM T84621 CM8T9G 127028498 IC50 = 612.3 nM T84621 CQO36B 127028499 IC50 = 58.1 nM T84621 C1M7GD 127028500 IC50 = 222.5 nM T84621 CN42BR 127028817 IC50 = 82.7 nM T84621 C3IMJ8 127028818 IC50 = 179.6 nM T84621 CPEM69 127028819 IC50 = 372.1 nM T84621 C70XOB 127030295 IC50 = 3598.4 nM T84621 CZ7L4J 127031191 IC50 > 10000 nM T84621 C49IME 127031799 IC50 = 88.2 nM T84621 CHS8L7 131982520 IC50 = 1900 nM T84621 C95PYQ 131982530 IC50 = 350 nM T84621 C5IWD9 131982539 IC50 = 2400 nM T84621 CSIP72 131982576 IC50 < 100 nM T84621 CS8C7T 131982729 IC50 = 1100 nM T84621 CHDP80 131982862 IC50 = 410 nM T84621 C1BNU6 131982871 IC50 > 10000 nM T84621 C6CB0I 132585204 IC50 = 2 nM T84621 C7SM9W 134129925 IC50 = 387 nM T84621 CB3EL1 134134056 IC50 = 1595 nM T84621 CB79AO 134134186 IC50 = 1308 nM T84621 CPZX32 134135994 IC50 = 10000 nM T84621 CS2P0E 134136577 IC50 = 2192 nM T84621 CH3V9Q 134139925 IC50 = 460 nM T84621 CFUE13 134141128 IC50 = 1573 nM T84621 COUK40 134141967 IC50 = 1996 nM T84621 CX3Y9D 134142597 IC50 = 1674 nM T84621 CQF59S 134143092 IC50 = 787 nM T84621 C1HG8V 134144349 IC50 = 1739 nM T84621 CFC8O6 134145376 IC50 = 220 nM T84621 C31WNO 134145695 IC50 > 8000 nM T84621 C7JEU2 134148873 IC50 = 250 nM T84621 C2JOB5 134152002 IC50 = 1544 nM T84621 CTXL17 134153274 IC50 = 1000 nM T84621 C3OLF2 134153424 IC50 > 8000 nM T84621 C12LPH 134153935 IC50 = 355 nM T84621 C8ROI0 134153997 IC50 = 630 nM T84621 CDV8M5 134155385 IC50 = 4600 nM T84621 C74ONC 134156861 IC50 = 4460 nM T84621 CKL9N7 135185757 IC50 = 4629 nM T84621 C8HTS7 135185761 IC50 > 10000 nM T84621 C1D4CS 135185764 IC50 = 5380 nM T84621 CMQC50 135185766 IC50 = 378 nM T84621 CIS5H8 135185771 IC50 = 4157 nM T84621 CF0EC1 135185786 IC50 = 4325 nM T84621 C8GB5V 135185787 IC50 = 2035 nM T84621 CH30EN 135185789 IC50 = 3330 nM T84621 CMR5C9 135185792 IC50 = 3926 nM T84621 CX97YM 135185793 IC50 = 1907 nM T84621 CS5FX2 135185796 IC50 = 2267 nM T84621 CV9RM5 135185801 IC50 = 4987 nM T84621 C8MF2Z 135185815 IC50 = 390 nM T84621 CX57GP 135185833 IC50 = 4809 nM T84621 CSZA19 135185836 IC50 = 5723 nM T84621 C6G1CH 135185858 IC50 = 4771 nM T84621 C9LU0C 135185886 IC50 = 4171 nM T84621 CZ1JS3 135186252 IC50 > 10000 nM T84621 CWU63C 136008115 IC50 = 17 nM T84621 CAV9U3 136219390 IC50 = 230 nM T84621 CC7LY3 136239517 IC50 = 960 nM T84621 C2V0IM 136244612 IC50 = 75 nM T84621 CYIF59 136245971 IC50 > 5000 nM T84621 CM97FH 137631528 IC50 = 48 nM T84621 C9LY0O 137631806 IC50 = 1 nM T84621 CH05YR 137633095 IC50 = 20 nM T84621 COG72W 137633343 IC50 = 93 nM T84621 C3QE1V 137633417 IC50 = 3 nM T84621 CVM54L 137634483 IC50 = 4 nM T84621 CV2S5Q 137637282 IC50 = 110 nM T84621 CUIX95 137637496 IC50 = 210 nM T84621 C14LXC 137638585 IC50 = 13 nM T84621 C1D0WG 137638612 IC50 = 9 nM T84621 CF1D5C 137639549 IC50 = 11 nM T84621 C8V7CD 137639692 IC50 = 6 nM T84621 C1SH2M 137639834 IC50 = 1.8 nM T84621 CZA2S8 137639890 IC50 = 14 nM T84621 C0N4PJ 137640302 IC50 = 124 nM T84621 COEV02 137642385 IC50 = 16 nM T84621 CH35RE 137642529 IC50 = 0.6 nM T84621 CP1EJ0 137642735 IC50 = 22 nM T84621 C29FMO 137642787 IC50 = 137 nM T84621 COGQ01 137644314 IC50 = 16 nM T84621 CA73KP 137644560 IC50 = 150 nM T84621 C4UP3J 137647900 IC50 = 2 nM T84621 CI31EQ 137649226 IC50 = 516 nM T84621 CS5BW7 137650545 IC50 = 4 nM T84621 CF71RE 137650772 IC50 = 104 nM T84621 CQ54YG 137651298 IC50 = 5 nM T84621 C4CL2W 137651728 IC50 = 42 nM T84621 CK7QJ4 137651744 IC50 = 2 nM T84621 CI5D2P 137652926 IC50 = 5 nM T84621 CIH34U 137653629 IC50 = 520 nM T84621 CV9I5G 137653991 IC50 = 13 nM T84621 C28VRO 137654883 IC50 = 19 nM T84621 CEV94S 137655303 IC50 = 148 nM T84621 CY5IK7 137655531 IC50 = 2 nM T84621 CUL37V 137655879 IC50 = 1 nM T84621 CN2CQ1 137656473 IC50 = 62 nM T84621 C53NVI 137657989 IC50 = 3 nM T84621 CNI0C1 137658011 IC50 = 42 nM T84621 C32WHO 137658276 IC50 = 181 nM T84621 C0G2UI 137658690 IC50 = 58 nM T84621 CLNU74 137659288 IC50 = 57 nM T84621 CA5LI1 137659926 IC50 = 14 nM T84621 C7YI9N 137660712 IC50 = 10 nM T84621 CFU1Z3 145960404 IC50 = 130 nM T84621 C1IU5W 145960520 IC50 = 1200 nM T84621 CQFH90 145960862 IC50 = 590 nM T84621 CNIB73 145960902 IC50 = 480 nM T84621 C0KNY4 145961099 IC50 < 100 nM T84621 CGI39P 145961215 IC50 = 2100 nM T84621 CW84OQ 145961259 IC50 > 10000 nM T84621 C92JOV 145961758 IC50 > 10000 nM T84621 CR6JH8 145961916 IC50 = 2200 nM T84621 CS4EO5 145962296 IC50 = 180 nM T84621 C1O0NQ 145962517 IC50 = 5700 nM T84621 C6VO0A 145962577 IC50 < 100 nM T84621 CY20CQ 145962664 IC50 > 10000 nM T84621 C6F7UE 145962949 IC50 = 58 nM T84621 C5O4RQ 145963242 IC50 > 10000 nM T84621 CGA01F 145963470 IC50 = 470 nM T84621 CH0TM7 145963574 IC50 > 10000 nM T84621 C0TZR1 145964456 IC50 = 19.2 nM T84621 CRJM82 145965429 IC50 = 6.6 nM T84621 CN7B1I 145968025 IC50 = 12.3 nM T84621 C82JTH 145971322 IC50 = 11.4 nM T84621 C5R6SH 145973507 IC50 = 5.8 nM T84621 C41LQE 145976039 IC50 = 4.7 nM T84621 C01TYI 145976345 IC50 = 15.4 nM T84621 CG23BW 145977901 IC50 = 6.5 nM T84621 C65ZFY 145978611 IC50 = 4.1 nM T84621 CI48QV 145979205 IC50 = 77 nM T84621 C9IQK7 145980859 IC50 = 17 nM T84621 CCKL25 145981178 IC50 = 120 nM T84621 CY4G3E 145981780 IC50 = 0.8 nM T84621 CYI3V5 145988023 IC50 = 29 nM T84621 CH6DJ3 155527950 IC50 = 4523 nM T84621 C80XNT 155530085 IC50 = 1668 nM T84621 C5XB1F 155530577 IC50 > 10000 nM T84621 C6DXN8 155559405 IC50 > 10000 nM T84621 C4UQS2 155564575 IC50 > 10000 nM T84621 CXM62E 155566406 IC50 = 9072 nM T84621 D00BVP 11847320 IC50 = 7 nM T84621 D00DSE 49864196 IC50 = 928 nM T84621 D00DUJ 11687499 IC50 = 7553 nM T84621 D00PXF 44206698 IC50 = 32.36 nM T84621 D01JZO 2779191 IC50 = 1000 nM T84621 D01REI 46901610 IC50 = 1400 nM T84621 D01SUE 6539759 IC50 = 888 nM T84621 D01SZX 46867545 IC50 = 99.1 nM T84621 D02ALK 11514074 IC50 = 2671 nM T84621 D02BXS 46901445 IC50 = 902 nM T84621 D02CSU 6539786 IC50 = 931 nM T84621 D02GFK 25034431 IC50 = 1521 nM T84621 D02JUJ 25034344 IC50 = 8925 nM T84621 D02LWB 6540046 IC50 = 2391 nM T84621 D02NAG 6539765 IC50 = 1472 nM T84621 D02PSL 45103913 IC50 = 6.166 nM T84621 D02UZI 6540056 IC50 = 288 nM T84621 D02XHH 6540043 IC50 = 23.5 nM T84621 D02ZQM 25180104 IC50 = 4921 nM T84621 D03CWL 14535954 IC50 = 323.59 nM T84621 D03EXD 49864181 IC50 = 251 nM T84621 D03KLN 11413434 IC50 = 81 nM T84621 D03MKT 6539788 IC50 = 1098 nM T84621 D03TRM 6540032 IC50 = 25.9 nM T84621 D03VRC 2989557 IC50 = 211 nM T84621 D03YHZ 25147692 IC50 = 33 nM T84621 D04CFP 46901927 IC50 = 469 nM T84621 D04CLL 6539775 IC50 = 763 nM T84621 D04ELJ 6539766 IC50 = 270 nM T84621 D04IBH 11616637 IC50 = 4481 nM T84621 D04ISG 11680597 IC50 = 2724 nM T84621 D04PKP 23644953 IC50 = 2896 nM T84621 D04QPK 6539783 IC50 = 774 nM T84621 D04WJN 10588478 IC50 = 70.8 nM T84621 D05FFY 14231155 IC50 = 141 nM T84621 D05IXU 25130517 IC50 = 953 nM T84621 D05MQE 6539785 IC50 = 657 nM T84621 D05QPR 12229388 IC50 = 489.78 nM T84621 D06CWR 24754344 IC50 = 67 nM T84621 D06HFV 6539805 IC50 = 27 nM T84621 D06JYY 25130848 IC50 = 2804 nM T84621 D06NFC 45103808 IC50 = 16 nM T84621 D06RSD 45103911 IC50 = 307 nM T84621 D07CTI 10853186 IC50 = 22.3 nM T84621 D07DQJ 45103810 IC50 = 7 nM T84621 D07EJK 10632289 IC50 = 478 nM T84621 D07IQG 10473365 IC50 = 6.7 nM T84621 D07JCO 12354256 IC50 = 6338 nM T84621 D07JMO 10220337 IC50 = 143 nM T84621 D07NAH 21772021 IC50 = 207 nM T84621 D07PYC 6539760 IC50 = 87 nM T84621 D07SOM 11847316 IC50 = 12 nM T84621 D07VGT 46901929 IC50 = 627 nM T84621 D07WLT 25180108 IC50 = 3964 nM T84621 D08AZK 6539767 IC50 = 1937 nM T84621 D08EZA 11847317 IC50 = 187 nM T84621 D08FAB 11845485 IC50 = 5826 nM T84621 D08HHA 19902087 IC50 = 204.17 nM T84621 D08HPU 6540052 IC50 = 503 nM T84621 D08IDC 24827305 IC50 = 238 nM T84621 D08ORG 10198247 IC50 = 281.84 nM T84621 D08PNF 6539770 IC50 = 790 nM T84621 D08WHC 10397593 IC50 = 206 nM T84621 D08YGW 10444038 IC50 = 4.786 nM T84621 D08ZTZ 11529133 IC50 = 2517 nM T84621 D09CPC 13728862 IC50 = 6746 nM T84621 D09HEA 1236449 IC50 = 368 nM T84621 D09HOE 6539789 IC50 = 34 nM T84621 D09QDY 6540033 IC50 = 6.1 nM T84621 D09VPA 6539794 IC50 = 2640 nM T84621 D09VQZ 46901616 IC50 = 4742 nM T84621 D09YXV 6539769 IC50 = 1448 nM T84621 D09ZHX 11847318 IC50 = 27 nM T84621 D0AK9S 22466877 IC50 = 18 nM T84621 D0AW7Q 46867544 IC50 = 463 nM T84621 D0B2UM 25034430 IC50 = 114 nM T84621 D0C6US 6540055 IC50 = 2529 nM T84621 D0C7YL 6481821 IC50 = 390 nM T84621 D0D7YL 11586681 IC50 = 2452 nM T84621 D0D8KN 45103805 IC50 = 181 nM T84621 D0D8YE 6540048 IC50 = 5684 nM T84621 D0D9FR 6539795 IC50 = 484 nM T84621 D0E0ZS 46901613 IC50 = 307 nM T84621 D0E8DX 25180300 IC50 = 580 nM T84621 D0E9WX 6540042 IC50 = 26.2 nM T84621 D0F5AC 46867542 IC50 = 15.1 nM T84621 D0F5YU 6539793 IC50 = 301 nM T84621 D0G6QL 23644748 IC50 = 1317 nM T84621 D0G9WP 18407230 IC50 = 819 nM T84621 D0HL9S 1265319 IC50 = 234.42 nM T84621 D0I1YH 46901446 IC50 = 342 nM T84621 D0I2UH 44187006 IC50 = 5.754 nM T84621 D0I5NW 6540047 IC50 = 1729 nM T84621 D0I9PA 25180306 IC50 = 13378 nM T84621 D0JE1I 9815923 IC50 = 9.5 nM T84621 D0K2DR 12050204 IC50 = 5952 nM T84621 D0K5KG 6540050 IC50 = 1268 nM T84621 D0L2QD 45103910 IC50 = 72.44 nM T84621 D0L4NG 6540054 IC50 = 1615 nM T84621 D0L8KL 11275595 IC50 = 805 nM T84621 D0LJ9D 46901783 IC50 = 415 nM T84621 D0M7FS 6539764 IC50 = 125 nM T84621 D0M9VK 11514098 IC50 = 849 nM T84621 D0MA9G 6540051 IC50 = 2117 nM T84621 D0N1GH 11601068 IC50 = 691 nM T84621 D0N1PQ 11506923 IC50 = 1577 nM T84621 D0N4VI 3021558 IC50 = 639 nM T84621 D0N5GZ 12229395 IC50 = 258 nM T84621 D0N8QD 15594569 IC50 = 691.83 nM T84621 D0N9PY 6539773 IC50 = 2368 nM T84621 D0NV7W 45103912 IC50 = 19.95 nM T84621 D0NX0M 6540049 IC50 = 578 nM T84621 D0O7TC 25180103 IC50 = 525 nM T84621 D0P1UO 45103914 IC50 = 26.92 nM T84621 D0PH1G 13688208 IC50 = 47.86 nM T84621 D0Q0BK 46901611 IC50 = 850 nM T84621 D0Q3CX 25034343 IC50 = 52 nM T84621 D0Q3JZ 6539774 IC50 = 2697 nM T84621 D0Q5ZZ 25129117 IC50 = 640 nM T84621 D0Q6BJ 25034426 IC50 = 151 nM T84621 D0Q8KM 44206482 IC50 = 28 nM T84621 D0R0TE 11557864 IC50 = 5419 nM T84621 D0RJ6S 11558270 IC50 = 2939 nM T84621 D0S4KP 25034427 IC50 = 843 nM T84621 D0S4WQ 12229386 IC50 = 151.36 nM T84621 D0S8FV 44586852 IC50 = 1047 nM T84621 D0T8JU 45103811 IC50 = 10.96 nM T84621 D0U7RR 6539768 IC50 = 320 nM T84621 D0V3YH 6539784 IC50 = 304 nM T84621 D0V6QN 45103915 IC50 = 128.82 nM T84621 D0V8CR 6539763 IC50 = 311 nM T84621 D0VL3R 25180303 IC50 = 1977 nM T84621 D0W8IZ 45103809 IC50 = 25.12 nM T84621 D0WN9P 46901444 IC50 = 287 nM T84621 D0X0IH 77918 IC50 = 135 nM T84621 D0X1QS 6540053 IC50 = 1291 nM T84621 D0Y3AV 25034346 IC50 = 373 nM T84621 D0Y5KX 46901443 IC50 = 522 nM T84621 D0YD9J 6539792 IC50 = 1515 nM T84621 D0YS2F 6539776 IC50 = 955 nM T84621 D0Z3GX 46901784 IC50 = 422 nM T35173 D03MXK 25022340 Ki = 5.1 nM T35173 D07CLV 46940575 IC50 = 12.9 nM T35173 D09MIN 24737642 IC50 = 11 nM T35173 D08XOV 50913339 IC50 = 1.3 nM T35173 D0YN1X 71661892 Ki = 5.4 nM T35173 CO1ZE4 9927170 IC50 = 690 nM T35173 CY3RV2 17756618 Ki = 2 nM T35173 CBM94F 23646361 Ki = 328 nM T35173 C8XJG1 24754961 Ki > 10000 nM T35173 C3EN8I 24857831 IC50 = 1860 nM T35173 C7XTN2 25138055 Ki = 5.9 nM T35173 CJ2VZ4 25138056 Ki = 4.2 nM T35173 C29PBM 25138057 Ki = 370 nM T35173 CLO6Y8 25138058 Ki = 20 nM T35173 CPN8E5 25138069 Ki = 1 nM T35173 CWH17B 25138070 Ki = 132 nM T35173 C0BJQ6 25173661 Ki = 20800 nM T35173 CW4U0R 25180313 Ki = 3 nM T35173 CAL8M3 25209021 Ki = 0.25 nM T35173 CD29TU 25209022 Ki = 2.09 nM T35173 C2KPJ0 44576646 IC50 = 1890 nM T35173 C96OTK 46830178 Ki = 24 nM T35173 CECL56 46830179 Ki = 393 nM T35173 C8RDC3 46888403 Ki = 292 nM T35173 CP40QG 46929436 Ki = 4.2 nM T35173 CQ0A5I 46929438 Ki = 47 nM T35173 C5FK8W 46929440 IC50 = 5.3 nM T35173 C1TIK8 46930628 Ki = 22.5 nM T35173 CVC3T5 46930723 Ki = 24.8 nM T35173 CNQO70 52951104 Ki = 1.7 nM T35173 C30GIF 53237922 Ki = 6 nM T35173 CW7AF2 53238154 Ki = 2 nM T35173 C5JPH2 53238155 Ki = 1.2 nM T35173 CW71DY 53238387 Ki = 2 nM T35173 C16JNG 53238388 Ki = 3 nM T35173 C3IPJ4 53238615 Ki = 2 nM T35173 CH0L8C 53238616 Ki = 2 nM T35173 CF83PC 53238842 Ki = 2.5 nM T35173 C2HB0C 53238843 Ki = 3 nM T35173 C7SR2W 53239063 Ki = 2.5 nM T35173 CM46PV 53239064 Ki = 4 nM T35173 CNFD80 53239285 Ki = 7 nM T35173 CCL6I5 53239286 Ki = 11 nM T35173 C61NHL 56945169 Ki = 3.3 nM T35173 C2WXP5 56945170 Ki = 6.4 nM T35173 C7YW1J 56945269 Ki = 6.9 nM T35173 CR7TD9 56945270 Ki = 14 nM T35173 CAD3P5 56945392 Ki = 4 nM T35173 CDYL09 56945393 Ki = 11 nM T35173 C7X1ZF 56946798 Ki = 1.7 nM T35173 C05JAE 56946799 Ki = 1.3 nM T35173 CE6SU4 57689264 Ki = 2 nM T35173 C62ZCQ 57689338 Ki = 25.3 nM T35173 C3KDR0 58609608 IC50 = 209 nM T35173 CTYP01 66972671 IC50 = 2.6 nM T35173 CZI6S5 66972777 IC50 = 4 nM T35173 CK0FP7 66972990 IC50 = 2.7 nM T35173 CQ9Y8K 66972994 IC50 = 3.2 nM T35173 CTKN28 66973039 IC50 = 2.5 nM T35173 CR9CO4 66973072 IC50 = 3.4 nM T35173 CKQ68O 66973165 IC50 = 4.9 nM T35173 CAD24O 66973224 IC50 = 7.6 nM T35173 C0R9TP 66973397 IC50 = 14 nM T35173 CQ1O6Z 66973400 IC50 = 2.1 nM T35173 C1NV7Q 71528757 EC50 = 36 nM T35173 C5RD4E 71570901 IC50 = 214 nM T35173 C9IT5Y 71570902 IC50 = 235 nM T35173 CY83OB 71571046 EC50 = 20 nM T35173 CAR8J2 71578011 IC50 = 1320 nM T35173 CVPJ20 71581702 IC50 = 47 nM T35173 CP9G3R 71581703 IC50 = 11 nM T35173 C3F4OT 71581838 IC50 = 40 nM T35173 CLIU93 71582189 IC50 = 16 nM T35173 C1VME6 71582339 IC50 = 10 nM T35173 CZ8DF4 71661893 Ki = 12.6 nM T35173 CB0O2T 71662077 Ki = 7.7 nM T35173 COCI81 71662078 Ki = 9.9 nM T35173 CNU16X 71662256 Ki = 2.1 nM T35173 CJRL34 71662257 Ki = 10 nM T35173 C2UM5A 71662420 Ki = 11 nM T35173 CVZK59 71662421 Ki = 7.4 nM T35173 CW4G0O 71662584 Ki = 13.3 nM T35173 C8AY6G 71662585 Ki = 7.9 nM T35173 C2UVF7 76335647 IC50 = 21 nM T35173 CZQO17 86650974 IC50 = 1.7 nM T35173 C9PHL5 89569624 IC50 = 24 nM T35173 CO0IY8 89570499 IC50 = 232 nM T35173 CD57CO 89570570 IC50 = 1490 nM T35173 C2ARB5 89570664 IC50 = 900 nM T35173 CIH2F9 90657109 IC50 = 366 nM T35173 CIH5V8 90664859 IC50 = 1300 nM T35173 C7APL4 118732792 IC50 = 1360 nM T35173 CDZ6M0 118732793 IC50 = 2880 nM T35173 C64NWU 118732794 IC50 = 180 nM T35173 CI69WD 118732795 IC50 = 17 nM T35173 C14FGL 122187534 IC50 = 3 nM T35173 C6NFD0 134419123 IC50 = 330 nM T35173 C87BOG 138377561 IC50 = 5.7 nM T35173 C0B8GK 138377594 IC50 = 140 nM T35173 CA43ML 142585287 IC50 > 1000 nM T35173 CGF6R2 142585309 IC50 > 1000 nM T35173 C0HC8R 142585337 IC50 > 9000 nM T35173 C0RHF1 142585361 IC50 > 10000 nM T35173 C5AI8Z 142585365 IC50 > 10000 nM T35173 CM7IG2 142585375 IC50 > 1500 nM T35173 CG46IU 145954838 IC50 > 1000 nM T35173 CKEJ30 145979040 IC50 = 353.3 nM T35173 C7XM4Q 145979112 IC50 = 53.5 nM T35173 CLRM52 145979809 IC50 = 304 nM T35173 CL4F9B 145981512 IC50 = 1103 nM T35173 C1K6AY 145982930 IC50 > 1000 nM T35173 C3L1ZW 145985393 IC50 = 56.6 nM T35173 CY8JR0 145986444 IC50 = 364.3 nM T35173 C1HWA3 145988725 IC50 = 212.1 nM T35173 CX7AV2 145991404 IC50 = 30.6 nM T35173 C79EXP 145992527 IC50 = 15 nM T35173 CK8JB2 155512591 IC50 = 40 nM T35173 CEH0W4 155523271 IC50 = 353 nM T35173 C23UZA 155554597 IC50 = 12.5 nM T35173 CR3UQ4 155561157 IC50 = 9 nM T35173 D03KZH 25172871 Ki = 6.3 nM T35173 D0BW7P 44589292 Ki = 4.8 nM T35173 D0Q7TL 24754886 Ki = 1.84 nM T35173 D0VK7M 49847690 IC50 = 21 nM T91442 D05RQB 457964 IC50 = 600 nM T91442 CZP5J2 3415 IC50 < 280 nM T91442 CQ87XE 72187 IC50 = 5800 nM T91442 CU3P0Y 484047 IC50 = 70 nM T91442 C61SXL 492406 IC50 = 370 nM T91442 CZ1A8T 503580 IC50 = 770 nM T91442 C8F1DN 6482394 IC50 = 460 nM T36445 CJ73BT 45486346 Ki = 53 nM T36445 C9ETC4 45486354 Ki = 70 nM T36445 CVPG40 45486356 Ki = 3.65 nM T36445 CSQ2K4 45486357 Ki = 1.7 nM T36445 C0ET8W 137630787 Ki = 2 nM T36445 D0Y9PH 45486355 Ki = 0.75 nM T82467 CL80QG 11820 IC50 > 100000 nM T82467 C2IJU0 440987 IC50 > 1000000 nM T82467 CV56WH 1637655 IC50 = 23000 nM T82467 CM1AE9 3370466 IC50 = 7943.28 nM T82467 CGE54P 3573716 IC50 = 10000 nM T82467 CS9M8A 3577407 IC50 = 5011.87 nM T82467 CJ4U6Y 3589423 IC50 = 10000 nM T82467 C2U9DI 3657707 IC50 = 31622.78 nM T82467 CPN2V4 3673391 IC50 = 10000 nM T82467 C28EBX 4790771 IC50 > 100000 nM T82467 CXBG75 5125956 IC50 = 50118.72 nM T82467 CL91JP 9452375 IC50 = 79432.82 nM T82467 C1W7TE 16258532 IC50 = 1258.93 nM T82467 C25EUG 16272810 IC50 = 1258.93 nM T82467 CK2ES3 16313990 IC50 > 100000 nM T82467 CZ59FR 16316459 IC50 > 100000 nM T82467 CEN83U 16323492 IC50 = 12589.25 nM T82467 CM1R8O 16344932 IC50 > 100000 nM T82467 CO8M7K 17405877 IC50 = 31622.78 nM T82467 C9IP3Q 17446910 IC50 > 100000 nM T82467 CLP9S1 24687782 IC50 = 12589.25 nM T82467 CEL5F7 26851836 IC50 > 1000000 nM T82467 CG3PR6 52912222 IC50 > 31622.78 nM T82467 CF8B4E 60498769 IC50 > 100000 nM T82467 CHOS65 91820723 IC50 = 100000 nM T82467 C0TNJ7 91820724 IC50 = 12589.25 nM T82467 CAZ9M0 91826677 IC50 = 2511.89 nM T82467 CEN52P 91826678 IC50 = 1000 nM T82467 C3BR8O 118021718 IC50 > 80000 nM T82467 CC14FI 118933132 IC50 > 100000 nM T82467 CWC98G 121499171 IC50 = 2700 nM T82467 CO9J5W 122179607 IC50 = 15848.93 nM T82467 C3WOE8 122179608 IC50 = 50118.72 nM T82467 CW03JY 122179609 IC50 = 3981.07 nM T82467 CHNS18 122179610 IC50 = 1258.93 nM T82467 C2Q0OY 122179611 IC50 = 5011.87 nM T82467 C9GPL4 122179612 IC50 = 1995.26 nM T82467 CZX41C 122179613 IC50 = 1258.93 nM T82467 CJDK15 122179614 IC50 = 1584.89 nM T82467 CSF76G 122179615 IC50 = 794.33 nM T82467 CY7U0Z 122179616 IC50 = 1258.93 nM T82467 C1MV9L 122179617 IC50 = 1584.89 nM T82467 CJ81BV 122179618 IC50 = 3981.07 nM T82467 CZ69QO 122180530 IC50 > 100000 nM T82467 C7D5VP 122180531 IC50 > 100000 nM T82467 CRY84E 122180532 IC50 > 100000 nM T82467 C0J1AY 122180533 IC50 > 100000 nM T82467 CPIV02 122180534 IC50 > 100000 nM T82467 CC9XH7 122180535 IC50 > 100000 nM T82467 C0IWE1 122180536 IC50 = 501187.23 nM T82467 CEF19P 122180537 IC50 = 25118.86 nM T82467 C20LOD 122180538 IC50 = 63095.73 nM T82467 C73OMU 122180539 IC50 = 19952.62 nM T82467 CZSB51 122180540 IC50 = 31622.78 nM T82467 CJ4LO2 122180541 IC50 = 79432.82 nM T82467 C4TB0F 122180542 IC50 = 12589.25 nM T82467 CTXL15 122180543 IC50 = 15848.93 nM T82467 CUDY80 122180544 IC50 > 100000 nM T82467 C0SC2Y 122180545 IC50 > 100000 nM T82467 CR6T4G 122180546 IC50 = 50118.72 nM T82467 CHJG86 122180547 IC50 > 100000 nM T82467 CYZV97 122180548 IC50 > 100000 nM T82467 C0AIU8 122180549 IC50 = 50118.72 nM T82467 CPUS31 122180550 IC50 = 31622.78 nM T82467 CD62RB 122180551 IC50 = 39810.72 nM T82467 C8UCV9 122180552 IC50 = 7943.28 nM T82467 C72NLB 122180553 IC50 = 5011.87 nM T82467 CR0K5P 122180554 IC50 = 15848.93 nM T82467 CZ6L2N 122180555 IC50 = 6309.57 nM T82467 CKH49I 122180556 IC50 = 25118.86 nM T82467 CS4PD6 122180557 IC50 = 10000 nM T82467 CWC9I4 122180558 IC50 = 3162.28 nM T82467 CE7SL5 122180559 IC50 = 2511.89 nM T82467 CR6YD4 122180560 IC50 = 1258.93 nM T82467 C8HCK6 122180561 IC50 = 1258.93 nM T82467 CX9C6Y 122180562 IC50 = 3162.28 nM T82467 CPZ67Y 122180563 IC50 = 19952.62 nM T82467 CN1LE0 122180564 IC50 = 39810.72 nM T82467 CGLF82 122181547 IC50 = 199.53 nM T82467 CZGK74 122181548 IC50 = 125.89 nM T82467 C9P3GX 122181549 IC50 = 316.23 nM T82467 C3QJ5L 122181550 IC50 = 31.62 nM T82467 C3NC4V 122181552 IC50 = 125.89 nM T82467 C41ZXJ 122181555 IC50 = 199.53 nM T82467 C6I3VJ 122181557 IC50 = 39.81 nM T82467 C7CJR2 122181559 IC50 = 5011.87 nM T82467 CP5Z1C 122181560 IC50 = 1584.89 nM T82467 C61RTG 122181561 IC50 = 63095.73 nM T82467 CT62FG 122181571 IC50 = 79.43 nM T82467 C8F9VG 129196931 IC50 = 166 nM T82467 CO3A0E 134817551 IC50 = 251.19 nM T82467 CP4X5W 134817552 IC50 = 100 nM T82467 CA40QW 135535536 IC50 = 10000 nM T82467 CQT3A9 137636309 IC50 > 100000 nM T82467 CQ6XB7 139030526 IC50 = 316.23 nM T82467 CJ3FL8 145982835 IC50 = 251.19 nM T82467 CA2W8M 145984295 IC50 = 199.53 nM T82467 CE05ZV 145984432 IC50 = 25118.86 nM T82467 CV4GH7 145984467 IC50 = 251.19 nM T82467 CT6V0I 145985751 IC50 = 39.81 nM T82467 C0GHY5 145986052 IC50 = 125.89 nM T82467 CK98QJ 146035912 IC50 = 100 nM T82467 C2D1SB 155512075 IC50 = 1995.26 nM T82467 CD3LA9 155512613 IC50 = 1995.26 nM T82467 CE13CA 155515130 IC50 = 3981.07 nM T82467 CPM43N 155516232 IC50 > 100000 nM T82467 C23BXS 155517049 IC50 = 3162.28 nM T82467 C6Q3JK 155517968 IC50 = 1000 nM T82467 CFP24B 155518498 IC50 = 1995.26 nM T82467 CB49NL 155521254 IC50 = 63.1 nM T82467 CC30UG 155521851 IC50 = 1258.93 nM T82467 CL1P4M 155523233 IC50 = 1258.93 nM T82467 C1W8JL 155523577 IC50 = 50118.72 nM T82467 C2K9NI 155523694 IC50 = 2511.89 nM T82467 C0VS8H 155523850 IC50 = 1258.93 nM T82467 C3NYK0 155523937 IC50 = 1000 nM T82467 CW8O7G 155525483 IC50 = 794.33 nM T82467 CKR6V3 155528325 IC50 = 1584.89 nM T82467 COX8K5 155529510 IC50 = 1995.26 nM T82467 CVMC06 155529991 IC50 = 630.96 nM T82467 CL93CM 155530154 IC50 = 1000 nM T82467 CEI09V 155530332 IC50 = 251.19 nM T82467 CY7ST9 155530616 IC50 = 1000 nM T82467 CJ93LE 155531635 IC50 = 1995.26 nM T82467 C82UPM 155532741 IC50 = 3162.28 nM T82467 CAEQ29 155534550 IC50 = 1000 nM T82467 CY08SU 155535485 IC50 = 2511.89 nM T82467 CAL2G4 155538392 IC50 > 1000000 nM T82467 C9ISB5 155538742 IC50 = 2511.89 nM T82467 C1MQP2 155539283 IC50 = 1995.26 nM T82467 C45FSO 155539489 IC50 = 15848.93 nM T82467 CXTO91 155541586 IC50 = 2511.89 nM T82467 CSVH67 155541704 IC50 > 1000000 nM T82467 CNSP97 155542781 IC50 = 501.19 nM T82467 C6FHM8 155543582 IC50 = 630.96 nM T82467 CEA1C5 155545659 IC50 = 30 nM T82467 CM51BF 155546089 IC50 = 12589.25 nM T82467 CFTR89 155546746 IC50 = 1584.89 nM T82467 CRBT87 155547095 IC50 > 1000000 nM T82467 CQNO46 155548910 IC50 = 2511.89 nM T82467 C4VKR0 155551851 IC50 = 1258.93 nM T82467 C2FWB9 155551946 IC50 = 25.12 nM T82467 CT35SU 155553650 IC50 = 6309.57 nM T82467 C0SYN6 155554629 IC50 = 3162.28 nM T82467 CDO08V 155555578 IC50 = 3981.07 nM T82467 C12QHG 155555950 IC50 = 1584.89 nM T82467 C7S8GF 155556284 IC50 > 100000 nM T82467 C6N1CG 155557122 IC50 = 1000 nM T82467 CYM3K9 155557522 IC50 = 2511.89 nM T82467 CSGH17 155559412 IC50 = 1995.26 nM T82467 C1YWF9 155559659 IC50 > 1000000 nM T82467 C3IDR8 155559983 IC50 > 1000000 nM T82467 C5X6EL 155560182 IC50 = 251.19 nM T82467 CS1C5W 155560567 IC50 = 3162.28 nM T82467 C3UC7H 155560671 IC50 = 10000 nM T82467 C7EDG4 155564694 IC50 = 3162.28 nM T82467 C6MX5G 155564795 IC50 > 1000000 nM T82467 CXRJ70 155566441 IC50 = 1258.93 nM T82467 C2PIK0 155567275 IC50 = 1000 nM T82467 CM5FL1 155567534 IC50 = 2511.89 nM T82467 C7C9DH 155568184 IC50 = 6309.57 nM T82467 CZ2VN0 155569163 IC50 = 1258.93 nM T82467 D00XRH 91820725 IC50 = 1258.93 nM T82467 D0F5TZ 91827383 IC50 = 1258.93 nM T82467 D0O6XT 91827373 IC50 > 100000 nM T13260 D00AXJ 4189 IC50 = 600 nM T13260 D00ZFP 5870 Ki = 2500 nM T13260 D02STN 132971 IC50 > 5000 nM T13260 D04DJN 10635 Ki = 220 nM T13260 D06XMU 6013 Ki = 600 nM T13260 D07ABV 468595 IC50 = 8400 nM T13260 D09GOS 2812 IC50 = 1.8 nM T13260 D09LNI 3365 IC50 = 22000 nM T13260 D0B4IF 456201 IC50 = 951.48 nM T13260 D0C1WH 3902 Ki = 0.02 nM T13260 D0C7JF 13769 Ki = 35000 nM T13260 D0D2VS 60198 Ki = 10.2 nM T13260 D0G2MW 446284 IC50 = 53200 nM T13260 D0K8KX 5280343 IC50 = 12 nM T13260 D0M6DO 2145 IC50 = 5.2 nM T13260 D0Q5XX 445580 IC50 = 33200 nM T13260 D0W0BF 2187 Ki = 0.13 nM T13260 D0ZX1P 59693 Ki = 0.05 nM T13260 D03AJU 44139752 IC50 = 856 nM T13260 D05NJI 5287541 IC50 = 300 nM T13260 D08UGX 60652 IC50 = 44.67 nM T13260 D09NST 449459 IC50 = 530000 nM T13260 D0B4VE 10251 IC50 = 8000 nM T13260 D0G5CS 68071 IC50 = 900 nM T13260 D0L4FS 5280961 Ki = 100000 nM T13260 D0U3EP 445154 IC50 > 40 ug.mL-1 T13260 D0W4EB 10090750 IC50 = 6000 nM T13260 D0DK4I 4534 IC50 = 11 nM T13260 D03YPJ 5163 IC50 > 100000 nM T13260 D06JUR 56487 Ki = 1100 nM T13260 D09BKE 4553 IC50 = 680 nM T13260 D0C0JT 4495 IC50 = 27000 nM T13260 D0D3PF 6918191 IC50 = 1.38 nM T13260 D0SX7F 60876 Ki = 7.6 nM T13260 D0Y2OG 177865 IC50 = 0.5 nM T13260 C9LCD8 3823 IC50 = 60 nM T13260 C9NZY3 12452 Ki = 17 nM T13260 C2L1YD 22458 IC50 = 4110 nM T13260 CPY1G9 59694 Ki = 1.5 nM T13260 C87SRA 60796 IC50 = 1.4 nM T13260 CQ0IC4 63062 IC50 = 530000 nM T13260 CLJB07 65544 IC50 = 840 nM T13260 CHI68V 66425 Ki = 100 nM T13260 CG5ZC1 66842 Ki = 100 nM T13260 CMV4R6 67343 Ki = 100 nM T13260 C5JLH9 69088 IC50 > 125700 nM T13260 CRGU58 86488 IC50 = 19000 nM T13260 CR0XY7 88598 IC50 > 10000 nM T13260 CKN0O5 92267 IC50 > 16200 nM T13260 C2Q3LF 92775 IC50 = 9600 nM T13260 CEOP93 100332 IC50 > 40 ug.mL-1 T13260 C1D3WF 101928 IC50 = 1733 nM T13260 C56OAF 104880 Ki = 2.5 nM T13260 C1U3VY 124075 IC50 = 3920 nM T13260 CX30LQ 124600 IC50 = 4000 nM T13260 C64SKJ 125502 Ki = 60.9 nM T13260 CC1ES3 125503 Ki = 172 nM T13260 CPU8L1 125637 Ki = 18 nM T13260 CHWM72 125921 IC50 = 230 nM T13260 CV7MN1 126221 Ki = 17.6 nM T13260 CW45IU 126253 IC50 = 4600 nM T13260 C5E0PO 126735 IC50 = 61.66 nM T13260 CZW26T 128011 Ki = 5 nM T13260 C7CRO3 128300 Ki = 90 nM T13260 CV2KS6 129500 Ki = 5.8 nM T13260 C4UV3D 130636 Ki = 9.9 nM T13260 C7MK6N 131078 IC50 = 310 nM T13260 C9KN0L 131099 Ki = 170 nM T13260 C0JR2M 131426 Ki = 2220 nM T13260 CL0T6W 131798 IC50 = 5.754 nM T13260 C7N1EF 132907 Ki = 5 nM T13260 CL9ZS8 138203 IC50 = 11880 nM T13260 CF83MK 146141 Ki = 34 nM T13260 CPVI09 146142 Ki = 1 nM T13260 C1RTX5 146485 IC50 = 2700 nM T13260 C9H4TV 147045 Ki = 120 nM T13260 CWJ40O 151432 Ki = 120 nM T13260 C5AS9H 155976 IC50 > 40 ug.mL-1 T13260 C3Y7WX 158280 IC50 > 40 ug.mL-1 T13260 C9DTE4 160767 IC50 = 29000 nM T13260 CT5E1S 165184 IC50 > 50000 nM T13260 CYWS98 185848 IC50 > 40 ug.mL-1 T13260 CL5U9T 190972 Ki = 9.8 nM T13260 C0EOM6 193441 Ki = 1000 nM T13260 C1S9AI 196342 Ki = 15 nM T13260 CE4U0D 198531 IC50 > 50000 nM T13260 C36VAO 199390 IC50 > 50000 nM T13260 CU9BQ6 219377 IC50 = 46700 nM T13260 CAD54R 239595 IC50 = 250 nM T13260 C5WUK4 256446 IC50 = 4810 nM T13260 CQ6A8P 266151 IC50 = 800 nM T13260 COA9C7 280309 IC50 = 9000 nM T13260 C1C5TO 281901 Ki = 180 nM T13260 CS86KD 283391 IC50 = 20 nM T13260 CD8E9U 313177 IC50 = 37600 nM T13260 CE9R4U 316687 IC50 = 130 nM T13260 CNP1J9 334704 IC50 > 40 ug.mL-1 T13260 CU7L1E 343584 IC50 = 126000 nM T13260 CHL4T1 387487 IC50 = 95300 nM T13260 CA9B4J 390805 IC50 = 176000 nM T13260 C3AJN7 396930 IC50 = 100 nM T13260 CD2UN0 432882 IC50 = 11000 nM T13260 C7HME8 439246 IC50 = 2.9 nM T13260 CK2EB0 461948 IC50 = 6 nM T13260 CDM69B 484455 IC50 = 2160 nM T13260 CQ59RG 484458 IC50 = 580 nM T13260 CZO45T 484460 IC50 = 9230 nM T13260 CB2DY7 484461 IC50 = 1520 nM T13260 CS2RK5 484470 IC50 = 4000 nM T13260 CRED51 484475 IC50 = 3650 nM T13260 CLR9O8 492641 IC50 = 4590 nM T13260 CL21UY 508444 IC50 = 350 nM T13260 CQSN41 508446 IC50 = 300 nM T13260 CUWG73 508447 IC50 = 460 nM T13260 CQ4KL6 508448 IC50 = 2960 nM T13260 CS7DT2 508449 IC50 = 1510 nM T13260 C3GNC0 508450 IC50 = 1180 nM T13260 C7TVD8 508451 IC50 = 190 nM T13260 CW8JE3 508452 IC50 = 2200 nM T13260 CLAW60 508453 IC50 = 1530 nM T13260 C8L5OZ 510041 IC50 = 1240 nM T13260 CNB76G 510042 IC50 = 260 nM T13260 CH95MB 510043 IC50 = 1090 nM T13260 C9NGK0 510044 IC50 = 1370 nM T13260 CEZW17 510045 IC50 = 1040 nM T13260 CTLY25 510046 IC50 = 510 nM T13260 C7X6RO 510048 IC50 = 110 nM T13260 CX65UW 510049 IC50 = 1320 nM T13260 CXC2M7 510050 IC50 = 1680 nM T13260 CM23DG 510051 IC50 = 1000 nM T13260 C7TYH9 585624 IC50 = 3200 nM T13260 C5LJK2 591809 IC50 = 260 nM T13260 CI5FK2 591810 IC50 = 41000 nM T13260 C2QEF8 596715 IC50 > 50000 nM T13260 C3P1FA 606677 IC50 = 3050 nM T13260 CG72HV 622979 Ki = 58 nM T13260 CQ90BJ 623313 Ki = 140 nM T13260 CU4V9W 623696 Ki = 3000 nM T13260 CZ0AH3 638278 IC50 = 3800 nM T13260 CHV1X7 638701 IC50 = 3980 nM T13260 CM9IU5 641375 IC50 = 31100 nM T13260 CO28QU 641376 IC50 = 31100 nM T13260 CZ14PX 641378 IC50 > 40 ug.mL-1 T13260 CS2IQ3 715186 IC50 = 10600 nM T13260 CE4JQ8 782123 IC50 > 105800 nM T13260 C8EDM5 838923 IC50 = 39710 nM T13260 CFZ7C3 882273 IC50 = 5030 nM T13260 CP25US 1009065 IC50 = 50 nM T13260 CJQK73 1027647 IC50 = 529663443.9 nM T13260 CE9SH3 1291064 IC50 = 11600 nM T13260 C48SKB 1292107 IC50 = 2190 nM T13260 CEOM25 1294577 IC50 = 780 nM T13260 C6B9RE 1481465 IC50 = 22810 nM T13260 C1SH3T 1548910 IC50 > 50000 nM T13260 C7VE1Z 1548995 IC50 = 370000 nM T13260 CB93KS 1550302 IC50 = 9200 nM T13260 C3T8GZ 1831259 IC50 > 10000 nM T13260 CF18YS 2313447 IC50 = 1100 nM T13260 COYU39 2475352 IC50 = 200 nM T13260 CB4N3X 2725996 Ki = 234.3 nM T13260 C8SYF6 2725997 IC50 = 4 nM T13260 C68PUH 2725998 Ki = 63.38 nM T13260 CO84NG 2827372 IC50 = 16.5 nM T13260 CPXD41 2843385 IC50 = 1000 nM T13260 C3M7VX 2939932 IC50 = 10600 nM T13260 C8XJ1B 2992689 IC50 = 172 nM T13260 C3H1DE 2998104 IC50 = 1500 nM T13260 CUVM41 3035832 IC50 = 190 nM T13260 CZ1LD9 3298129 IC50 > 25000 nM T13260 C2SE4A 3346379 IC50 = 4300 nM T13260 C2OS4U 3361302 IC50 = 1100 nM T13260 CCD73S 3399276 IC50 = 3880 nM T13260 CBKQ75 3418244 IC50 = 370 nM T13260 C7O2MH 3943788 IC50 = 80 nM T13260 C40QVD 3964390 IC50 > 40 ug.mL-1 T13260 C7LX0V 4083407 IC50 = 59979107.63 nM T13260 C0WA7C 4103051 Ki = 830 nM T13260 CJ1U7P 4369413 IC50 = 100 nM T13260 CK17YZ 4369414 IC50 = 0.82 nM T13260 C1WIR4 4499193 IC50 > 31622.78 nM T13260 CXNH97 4993111 IC50 = 3670 nM T13260 C5OAR6 5121919 IC50 > 50000 nM T13260 CG0C4J 5281255 IC50 > 40 ug.mL-1 T13260 CM9Z0B 5312198 IC50 = 761 nM T13260 CF67ON 5314722 IC50 > 25000 nM T13260 CEW6B3 5315503 IC50 > 40 ug.mL-1 T13260 C3KDP7 5325467 IC50 = 16310 nM T13260 CW1UM5 5357488 IC50 > 351700 nM T13260 CBF75X 5376779 IC50 > 250000 nM T13260 CUV49J 5472143 IC50 = 5200 nM T13260 CR6N4L 5481966 IC50 > 40 ug.mL-1 T13260 C7VSM2 5702471 IC50 = 9332.54 nM T13260 CST49O 5702960 IC50 > 250000 nM T13260 C84XUK 6035693 IC50 = 5495.41 nM T13260 C3F7JB 6159604 IC50 = 12022.64 nM T13260 C1HZJ2 6438825 IC50 > 40 ug.mL-1 T13260 C2B1RH 6450879 IC50 > 40 ug.mL-1 T13260 CR8IB1 6457965 IC50 = 21700 nM T13260 C26KXD 6458748 IC50 = 2500 nM T13260 C39IEC 6461420 IC50 = 119 nM T13260 CP3O0B 6463551 IC50 = 61.6 nM T13260 CE93VI 6473542 IC50 = 100 nM T13260 C73LCV 6475119 IC50 = 42.7 ug.mL-1 T13260 C21BZK 6493479 IC50 = 63.7 nM T13260 CCO4Q3 6493484 IC50 = 440 nM T13260 CI13SQ 6523638 IC50 = 25000 nM T13260 C1JAT6 6539761 IC50 = 6580 nM T13260 CTE57C 6539762 IC50 = 3790 nM T13260 CF17BE 6539771 IC50 = 1130 nM T13260 CJ7RS8 6539772 IC50 = 4000 nM T13260 CP02JW 6539778 IC50 = 979489.99 nM T13260 CW1U8J 6539779 IC50 > 36000 nM T13260 CQD13Z 6539787 IC50 = 650 nM T13260 CQB1U5 6539798 IC50 = 800 nM T13260 C79FTC 6539799 IC50 = 1010 nM T13260 C5Z9KY 6539802 IC50 = 90 nM T13260 C7CAB8 6539809 IC50 > 36000 nM T13260 COU5D2 6539810 IC50 > 36000 nM T13260 CQ0HD5 6539812 IC50 = 720 nM T13260 CQ9XM0 6539813 IC50 = 1940 nM T13260 CF1R9J 6539815 IC50 > 36000 nM T13260 CMA37K 6539816 IC50 > 36000 nM T13260 CP4VI2 6540030 IC50 = 226 nM T13260 CR6LS8 6540031 IC50 = 190 nM T13260 CU3C1Y 6540034 IC50 = 125 nM T13260 CXEW82 6540035 IC50 = 119 nM T13260 CBKX32 6540037 IC50 = 120 nM T13260 C8MRI7 6540038 IC50 = 218 nM T13260 C8JXY1 6540039 IC50 = 20 nM T13260 CZK3T4 6540040 IC50 = 330 nM T13260 CDS26H 6540041 IC50 = 39 nM T13260 C2FRW5 6540044 IC50 = 970 nM T13260 C2JBQ1 6540045 IC50 = 810 nM T13260 CV0FA1 7330517 IC50 = 40950 nM T13260 CG9RF6 7515053 IC50 > 250000 nM T13260 C1DZ2H 7537616 IC50 = 150 nM T13260 C8VJ4X 8963350 IC50 > 50000 nM T13260 C0J1AS 9794431 IC50 = 10000 nM T13260 CS23XK 9797346 Ki = 10 nM T13260 C9QVL1 9816909 IC50 = 8900 nM T13260 CJ37SX 9818699 IC50 = 1.38 nM T13260 C2YB9F 9819524 IC50 = 12 nM T13260 CF7Z3J 9837392 IC50 = 2.9 nM T13260 C56CLB 9838063 IC50 = 680 nM T13260 CKJ1I6 9838340 IC50 = 580 nM T13260 CF3Z5V 9839853 Ki = 1.4 nM T13260 C35UMF 9890209 IC50 > 500000 nM T13260 CZ15MX 9908653 Ki = 36 nM T13260 CWL3O1 9926844 IC50 = 40000 nM T13260 C9Y3CA 9928113 IC50 = 12 nM T13260 CF24CV 9947889 Ki = 100 nM T13260 C0PHJ6 9948207 Ki = 70 nM T13260 C9BIH0 9948368 IC50 = 95.5 nM T13260 CZFV57 9949484 Ki = 1 nM T13260 CXH81D 9951467 IC50 = 0.12 nM T13260 CO1Z0A 9971194 IC50 = 5600 nM T13260 CBLP75 9972072 IC50 = 42.66 nM T13260 CDT6N2 9972577 IC50 = 8.8 nM T13260 C46LXP 9973019 Ki = 3.4 nM T13260 CB9DF4 9973046 IC50 = 20 nM T13260 C9JPT7 9974683 Ki = 1.4 nM T13260 CW1KO5 9976841 Ki = 36 nM T13260 C6W9NM 9978572 Ki = 16.5 nM T13260 C6Z0WQ 9991753 IC50 = 5000 nM T13260 CR16JI 9991838 IC50 = 530 nM T13260 CZV57I 9992344 IC50 = 6300 nM T13260 CQH4B7 9992433 IC50 = 14000 nM T13260 C2B4RF 9992450 IC50 = 4300 nM T13260 CVU3L0 9993026 IC50 = 3019.95 nM T13260 C85AUN 9998048 IC50 = 38.02 nM T13260 C0J8VR 10000064 IC50 = 78.5 nM T13260 C49HDL 10013868 IC50 = 170 nM T13260 C1FX2N 10014477 IC50 = 9300 nM T13260 C1KAV4 10015136 IC50 = 230 nM T13260 CPG39R 10018603 Ki = 3.4 nM T13260 C58EOH 10019839 IC50 = 130 nM T13260 CX7H2S 10020109 IC50 = 44 nM T13260 C0RP1F 10020714 IC50 = 44 nM T13260 CU12IF 10022210 IC50 = 130 nM T13260 CI7V2F 10023315 Ki = 36 nM T13260 C5PUD9 10026826 IC50 = 210 nM T13260 C5NAU2 10036028 IC50 = 600 nM T13260 C5Y0MK 10036693 IC50 = 380 nM T13260 CU7CI9 10042609 IC50 = 55 nM T13260 CV1K0G 10046399 IC50 = 51.8 nM T13260 C8MC0P 10051115 IC50 = 1650 nM T13260 C6W9NL 10060155 IC50 = 4200 nM T13260 C30LGM 10060824 IC50 = 3400 nM T13260 C64YSN 10064550 IC50 = 62 nM T13260 C9UMW8 10064832 IC50 = 600 nM T13260 C6Y1OT 10067777 Ki = 2.8 nM T13260 CI3S7F 10069029 IC50 = 220 nM T13260 CR13PX 10069113 Ki = 36 nM T13260 CX3FH6 10069477 Ki = 2.8 nM T13260 CR1V5S 10082665 IC50 = 93000 nM T13260 C64PHS 10083522 IC50 = 30 nM T13260 CR13LC 10084738 IC50 = 8700 nM T13260 CB65ED 10086187 Ki = 1.4 nM T13260 CL9X0W 10087126 Ki = 5000 nM T13260 C9YRP5 10087312 IC50 = 57 nM T13260 CPH49E 10087422 IC50 = 61.5 nM T13260 CD0MQ9 10088785 Ki = 1.4 nM T13260 CZB62D 10089657 Ki = 2.8 nM T13260 CNI2R6 10091150 IC50 = 102 nM T13260 C4JM1P 10104524 IC50 = 2400 nM T13260 C92KBY 10105573 IC50 > 19000 nM T13260 C7W5GI 10171354 IC50 = 14000 nM T13260 CD6JG2 10228895 IC50 = 500 nM T13260 CG2U1S 10242773 IC50 = 1000 nM T13260 CC08OX 10243987 IC50 = 590 nM T13260 CG24IZ 10247264 IC50 > 20000 nM T13260 CTK8F5 10248614 Ki = 9.3 nM T13260 C3YC9I 10263082 IC50 = 1900 nM T13260 C4CDG7 10264163 IC50 = 23000 nM T13260 CO2LT5 10286610 IC50 = 860 nM T13260 CD39LQ 10291777 IC50 = 100 nM T13260 CL6WE9 10295791 IC50 = 24000 nM T13260 C5LRW4 10298511 IC50 = 25100 nM T13260 CE2Z5S 10313881 IC50 = 41 nM T13260 C3PYH4 10317448 IC50 = 280 nM T13260 C6AOP4 10317522 IC50 = 530 nM T13260 CMO02D 10317756 Ki = 67000 nM T13260 C65BFK 10317931 IC50 = 400 nM T13260 C64YEQ 10318379 Ki = 9.8 nM T13260 CTUL01 10331100 IC50 = 185 nM T13260 CM81OX 10332392 IC50 = 3715.35 nM T13260 CZ4W0C 10332529 IC50 = 41 nM T13260 CQGS52 10334324 Ki = 1000 nM T13260 CQX4C8 10335739 Ki = 3.4 nM T13260 CT69PQ 10336071 IC50 = 100 nM T13260 C9RX2D 10338362 Ki = 9.3 nM T13260 CUDL75 10340374 Ki = 13.1 nM T13260 C0EO5N 10340839 Ki = 9.3 nM T13260 C07JGF 10355617 IC50 = 3300 nM T13260 CH5DS4 10358509 Ki = 5000 nM T13260 CWY9D0 10360147 Ki = 40 nM T13260 CELR79 10360875 IC50 = 63 nM T13260 CO69BI 10361506 IC50 = 49 nM T13260 CN7JK2 10368162 IC50 = 1650 nM T13260 CYNM04 10376335 IC50 = 260 nM T13260 CWY1X4 10379617 IC50 = 190 nM T13260 C5IZ0X 10380012 IC50 = 35000 nM T13260 CTX86G 10381606 IC50 = 233 nM T13260 COK7N8 10382166 IC50 = 1230 nM T13260 C06BMI 10384926 Ki = 13.1 nM T13260 C8CW6Y 10385742 Ki = 9.8 nM T13260 CP8G9A 10398594 IC50 = 13000 nM T13260 CXY9P7 10398686 IC50 = 1200 nM T13260 C1HZC5 10399349 IC50 = 240 nM T13260 CIJ01W 10400011 IC50 = 170 nM T13260 C3UN8Z 10400778 IC50 = 7900 nM T13260 CJ31WC 10403482 Ki = 42 nM T13260 C9LW2Z 10403903 IC50 = 49 nM T13260 CC5YT4 10404407 IC50 = 3000 nM T13260 CG7P5I 10404636 IC50 = 130 nM T13260 C9Q7CT 10407320 Ki = 36 nM T13260 C8KUR2 10421663 IC50 = 22000 nM T13260 C59NEQ 10426743 IC50 = 4300 nM T13260 CRV19P 10444266 IC50 = 1300 nM T13260 CR0O6C 10447478 IC50 = 20000 nM T13260 CTYP51 10448246 Ki = 5.1 nM T13260 CPAE70 10449017 IC50 = 1460 nM T13260 CUM3X2 10449331 IC50 = 2400 nM T13260 CQWX01 10450499 IC50 > 20000 nM T13260 C4L6ED 10450517 IC50 = 600 nM T13260 CM1IU9 10466775 IC50 = 6400 nM T13260 CT0H4G 10466776 IC50 = 750 nM T13260 C7TL6U 10467336 IC50 = 4786.3 nM T13260 C3YI0N 10467502 IC50 = 17000 nM T13260 C5DP9Z 10471817 IC50 = 10 nM T13260 CSM4H0 10472175 IC50 = 60 nM T13260 CIG25U 10474687 Ki = 10 nM T13260 C9W6YH 10488782 IC50 = 160 nM T13260 CYR2O4 10489655 IC50 = 680 nM T13260 CH7IA3 10489983 IC50 = 38000 nM T13260 CTW6A7 10494334 Ki = 17 nM T13260 CP8F4R 10495337 Ki = 4.7 nM T13260 CG0A6X 10513321 IC50 = 18000 nM T13260 CH2R0N 10513661 IC50 = 3900 nM T13260 C5RHY3 10538018 IC50 = 200 nM T13260 C7I6JP 10562688 IC50 = 239.88 nM T13260 CH8FS5 10565166 Ki = 3.1 nM T13260 C4L8OX 10566080 IC50 = 51000 nM T13260 C9PMK8 10566304 Ki = 12 nM T13260 C43DIK 10571994 Ki = 17 nM T13260 CN2RF5 10585362 IC50 > 250000 nM T13260 C7S5RV 10586086 IC50 = 220 nM T13260 CTI0R2 10587179 IC50 > 250000 nM T13260 CU5GI9 10594307 Ki = 5 nM T13260 C3RM0Y 10595083 Ki = 2.5 nM T13260 C3DH9W 10608774 IC50 = 920 nM T13260 CZ2H3N 10610950 IC50 > 250000 nM T13260 C02GMY 10617003 Ki = 2.5 nM T13260 CNR3V1 10618506 IC50 > 10000 nM T13260 C1F9IE 10636984 Ki = 5.3 nM T13260 C5TVC0 10637984 Ki = 12 nM T13260 CC39RI 10644237 Ki = 7 nM T13260 C04DNA 10656613 IC50 > 250000 nM T13260 C5ION6 10660701 IC50 = 3100 nM T13260 C9QN4J 10660816 IC50 = 36000 nM T13260 CJYQ87 10661641 Ki = 2.5 nM T13260 C8MOG9 10662151 Ki = 12 nM T13260 C8D0PV 10662758 Ki = 2.5 nM T13260 CUA2P0 10663766 Ki = 2.5 nM T13260 C8OUR1 10663913 Ki = 17 nM T13260 CPKA25 10665849 Ki = 17 nM T13260 CAYD96 10667894 Ki = 8.5 nM T13260 CP98RW 10680142 IC50 = 6000 nM T13260 CE12OS 10682353 IC50 = 24000 nM T13260 C0N2BV 10684551 IC50 = 9100 nM T13260 C01ZPW 10684552 IC50 = 10800 nM T13260 C1CGU5 10686589 Ki = 17 nM T13260 COB2W4 10690043 IC50 = 50 nM T13260 C0SIE5 10691220 Ki = 2.5 nM T13260 CMN02T 10708503 Ki = 1100 nM T13260 C1OME3 10710388 IC50 = 5200 nM T13260 CA13SW 10711620 IC50 = 549.54 nM T13260 CUQN16 10714213 IC50 > 10000 nM T13260 CO3JR0 10727176 IC50 = 51000 nM T13260 CBG72H 10729611 IC50 > 250000 nM T13260 CFE87L 10729612 IC50 = 27000 nM T13260 CYW4V9 10731755 IC50 > 10000 nM T13260 CKD29U 10738189 Ki = 9 nM T13260 CHL74J 10752290 IC50 = 103000 nM T13260 CU5W7P 10752634 IC50 = 350 nM T13260 CM3GX1 10753431 IC50 > 250000 nM T13260 C7U3ZR 10755577 IC50 = 4600 nM T13260 C4EXR1 10761806 IC50 = 1100 nM T13260 CZSA79 10774377 IC50 = 111000 nM T13260 CCD9R4 10774996 IC50 = 2400 nM T13260 C9GC0A 10775929 IC50 = 2600 nM T13260 CG27MD 10776192 IC50 > 250000 nM T13260 CNGQ30 10800145 IC50 = 1100 nM T13260 CJ5LW6 10806186 IC50 = 18100 nM T13260 CR25UM 10806331 Ki = 1100 nM T13260 C7P8IX 10810323 Ki = 10 nM T13260 CO53EU 10811011 Ki = 7 nM T13260 C0EAP2 10823139 IC50 = 700 nM T13260 C94PCN 10826001 IC50 = 8000 nM T13260 CN7I8H 10827014 IC50 = 16000 nM T13260 CZW6V4 10828130 IC50 = 2290.87 nM T13260 CM8WH3 10846478 IC50 = 3340 nM T13260 CU3I7B 10847200 IC50 = 440 nM T13260 CLZ5Q7 10853458 Ki = 37 nM T13260 C6RWM5 10854674 Ki = 17 nM T13260 C3UJ7E 10859502 Ki = 68 nM T13260 C26ARU 10859572 Ki = 22 nM T13260 CM5B1D 10883602 IC50 = 12 nM T13260 CVD0E9 10895435 IC50 > 40 ug.mL-1 T13260 CW9Z8X 10900865 IC50 > 40 ug.mL-1 T13260 CP85BH 10902291 Ki = 100 nM T13260 CWZC05 10903498 IC50 = 6.9 nM T13260 C59BGC 10904721 IC50 = 1.1 nM T13260 CXD1M3 10913975 IC50 > 40 ug.mL-1 T13260 C9UJN5 10914511 Ki = 60 nM T13260 CHX8K0 10927303 Ki = 70 nM T13260 CR6CX8 10957235 Ki = 170 nM T13260 C7QXL8 10958364 IC50 > 40 ug.mL-1 T13260 CX9N0T 10990534 IC50 > 40 ug.mL-1 T13260 C0VSL5 11001084 IC50 = 4500 nM T13260 CE3YX7 11015855 IC50 > 40 ug.mL-1 T13260 C04SCF 11023115 Ki = 110 nM T13260 CU5B1T 11033539 Ki = 58 nM T13260 CUQP81 11034900 Ki = 60 nM T13260 CZR21O 11066682 Ki = 250 nM T13260 CRE6W0 11078050 Ki = 90 nM T13260 CWR14N 11079165 IC50 = 39 nM T13260 C9IE5F 11085889 IC50 = 1600 nM T13260 CC2NG5 11109070 IC50 = 23 nM T13260 C52NIS 11140706 IC50 = 1800 nM T13260 CMB40V 11140772 IC50 = 2400 nM T13260 CDI1L7 11141249 Ki = 800 nM T13260 CZ31ND 11141567 IC50 = 5500 nM T13260 C5LS1V 11153057 Ki = 900 nM T13260 C63APE 11164320 IC50 = 610 nM T13260 C7TKN9 11164739 IC50 = 9200 nM T13260 CM59ZA 11176755 Ki = 1160 nM T13260 C1A9IY 11179136 IC50 = 530 nM T13260 C2KJ6H 11196148 IC50 = 168 nM T13260 CTA9B3 11197738 IC50 = 50 nM T13260 CFQ8X5 11213800 IC50 > 100000 nM T13260 C0IC8T 11218132 IC50 = 13900 nM T13260 CQ0IG4 11219074 IC50 = 3600 nM T13260 C1TP7W 11232831 IC50 = 150 nM T13260 CQGN76 11241635 IC50 = 31622.78 nM T13260 CR9UT3 11243132 IC50 = 100000 nM T13260 CC9X2S 11244229 IC50 > 100000 nM T13260 CD15BO 11244509 IC50 = 32 nM T13260 CFYD58 11246736 Ki = 1690 nM T13260 C8PJ7G 11265329 IC50 = 31622.78 nM T13260 C2A0GX 11276968 IC50 = 3380 nM T13260 C0V4IO 11288325 IC50 = 280 nM T13260 CR1JS5 11310894 IC50 = 9770 nM T13260 CRW74G 11322098 IC50 = 144 nM T13260 CI9H7S 11347268 Ki = 3.4 nM T13260 C8SK0O 11356920 IC50 = 1122.02 nM T13260 C9AO5H 11381850 IC50 > 50000 nM T13260 CXDT28 11392371 IC50 = 250 nM T13260 C5X7KI 11402766 IC50 = 26915.35 nM T13260 CH4VM5 11413971 IC50 = 2818.38 nM T13260 CX63YZ 11417114 IC50 = 3600 nM T13260 CF7J8A 11426612 IC50 = 5128.61 nM T13260 CAU8M0 11448232 IC50 = 2820 nM T13260 CO7U8R 11485667 IC50 > 100000 nM T13260 CA90VB 11493223 Ki = 100 nM T13260 CXP5I7 11493374 IC50 = 440 nM T13260 C8P4VL 11493892 IC50 = 960 nM T13260 CEFC74 11495013 IC50 = 12 nM T13260 CV02WR 11515409 IC50 = 1210 nM T13260 C3XAL1 11522408 IC50 = 15.3 nM T13260 CV58AY 11522728 IC50 = 470 nM T13260 CV3U7F 11530377 Ki = 100 nM T13260 CN4T0K 11544009 IC50 = 970 nM T13260 CDG7N4 11544414 IC50 = 110 nM T13260 CSW1P3 11551000 IC50 = 2810 nM T13260 CL5E7M 11558482 IC50 = 870 nM T13260 CAEQ30 11565696 IC50 = 300 nM T13260 CHJB42 11567631 IC50 = 0.92 nM T13260 CF51ZE 11568594 IC50 = 3.9 nM T13260 CX6OV1 11572776 Ki = 100 nM T13260 CVK75E 11572824 IC50 = 760 nM T13260 C5KNY1 11573432 IC50 = 630.96 nM T13260 COX19Z 11581191 IC50 = 176 nM T13260 C9IJ3T 11594132 IC50 = 1252 nM T13260 CBV48A 11595426 IC50 = 95.5 nM T13260 CKTA53 11603462 IC50 = 0.77 nM T13260 C3VHL8 11611589 IC50 = 99 nM T13260 CAM20K 11624089 Ki = 75 nM T13260 CB2L9J 11624690 IC50 = 160 nM T13260 C5Y6MN 11633212 IC50 = 25.5 nM T13260 C2UBZ0 11639518 IC50 = 290 nM T13260 C7SYX1 11644772 IC50 = 5870 nM T13260 C0ZD2V 11645369 IC50 = 230 nM T13260 C2WF8E 11653632 IC50 = 3960 nM T13260 C9QOK8 11654142 IC50 = 17.5 nM T13260 C1OU0F 11667385 IC50 = 2.291 nM T13260 CP6TI4 11681050 Ki = 147 nM T13260 CZA7U6 11687547 IC50 > 25000 nM T13260 CWH82Z 11696602 IC50 = 49 nM T13260 CZ50DQ 11708478 IC50 > 2000 nM T13260 C7WN6I 11716932 IC50 = 4490 nM T13260 CTHL93 11722357 Ki = 1.4 nM T13260 C59DIH 11723061 Ki = 4.9 nM T13260 CS4AR9 11723111 Ki = 3.4 nM T13260 CZH43C 11725276 IC50 = 1800 nM T13260 C0MD6A 11732219 IC50 = 2.3 nM T13260 CFB08O 11737365 IC50 = 0.06 nM T13260 CW2B3A 11738647 IC50 = 51 nM T13260 CD0KR5 11739060 IC50 = 107.15 nM T13260 CUTV09 11758702 IC50 > 16100 nM T13260 CLND03 11758964 IC50 = 150000 nM T13260 CG79IH 11760852 IC50 = 1800 nM T13260 CM2LK4 11774754 IC50 > 100000 nM T13260 CA7S0C 11779699 Ki = 5000 nM T13260 CIJQ20 11784241 IC50 > 50000 nM T13260 C83WAR 11792329 Ki = 2.5 nM T13260 C0LM8Q 11793414 Ki = 17 nM T13260 CIU5X2 11807837 Ki = 50 nM T13260 CZC18Q 11824496 IC50 = 1500 nM T13260 C3V9LP 11833981 IC50 = 420 nM T13260 C7W4TJ 11842924 IC50 = 910 nM T13260 CTCY19 11843079 IC50 = 2500 nM T13260 C81VMW 11843080 IC50 = 10000 nM T13260 C9YK3J 12137521 IC50 > 100000 nM T13260 CY0A2H 12846880 IC50 > 50000 nM T13260 CW7EC6 12854713 IC50 = 38300 nM T13260 CP94EZ 13257279 IC50 = 170000 nM T13260 CNKO41 13288738 IC50 = 54 nM T13260 C70ESC 13437151 IC50 > 50000 nM T13260 CW02LQ 13537950 IC50 = 245000 nM T13260 C90PFA 13537951 IC50 = 6000 nM T13260 CJ05FQ 13537952 IC50 = 2500 nM T13260 C6OQT1 13537953 IC50 = 3600 nM T13260 CAQK75 13537954 IC50 = 3200 nM T13260 CK6AZ4 13537955 IC50 = 330 nM T13260 C6RM8P 13537956 IC50 = 2400 nM T13260 C9XFJ0 13596071 Ki = 1750 nM T13260 C29SJW 13633181 Ki = 41 nM T13260 CY8V7Z 13633182 Ki = 36 nM T13260 C9LM0A 13633183 Ki = 73 nM T13260 CZP9U6 13633184 Ki = 36 nM T13260 CUX8Y6 13660214 IC50 > 300000 nM T13260 CJ41AQ 13660215 IC50 = 135000 nM T13260 CT0A6S 13660217 IC50 = 16000 nM T13260 CMR8V5 13660219 IC50 = 3000 nM T13260 C7YMZ1 13660220 IC50 = 3000 nM T13260 C9ZAK2 13660222 IC50 = 400 nM T13260 C6CVT0 13660223 IC50 = 1100 nM T13260 CL0B9C 13660224 IC50 = 600 nM T13260 CM26OE 13686727 IC50 = 1150 nM T13260 CB1XD6 13688211 IC50 = 3.2 nM T13260 C1F5IT 13688212 IC50 = 3.2 nM T13260 CA6Z5U 13688213 IC50 = 21 nM T13260 C0D4XQ 13688215 IC50 > 1000 nM T13260 CG0KB9 13688216 IC50 = 17.6 nM T13260 C3D8YA 13688218 IC50 = 14.3 nM T13260 CNF97R 13833941 IC50 = 880 nM T13260 C8LRB9 13900578 IC50 = 385000 nM T13260 CT1EY3 13900579 IC50 = 31000 nM T13260 C7IM0K 13900580 IC50 = 40000 nM T13260 CNC7F2 13900581 IC50 = 21000 nM T13260 CXLQ60 13900582 IC50 = 6600 nM T13260 C3HEP2 13900583 IC50 = 1500 nM T13260 C3DM0W 13900584 IC50 = 3000 nM T13260 C3TLJ9 13900585 IC50 = 10000 nM T13260 CS5G4U 13900586 IC50 = 30000 nM T13260 CG7O6E 13964844 Ki = 10000 nM T13260 C28GTK 13990942 Ki = 55 nM T13260 CS82TI 13990943 Ki = 53 nM T13260 CAY1C9 13991369 Ki = 100 nM T13260 C7LKS8 14055913 Ki = 690 nM T13260 CE6L1R 14055915 Ki = 260 nM T13260 CVU6D4 14068934 Ki = 1200 nM T13260 C27JCM 14068935 IC50 = 2500 nM T13260 C9X6BY 14068936 Ki = 50 nM T13260 CQO06Z 14068937 Ki = 1.5 nM T13260 CEK04X 14068938 Ki = 20 nM T13260 CY8M0H 14068939 IC50 = 4000 nM T13260 C7G8AL 14068940 IC50 = 200 nM T13260 C4WV0N 14068941 IC50 = 200 nM T13260 CYM3T7 14068942 IC50 = 2000 nM T13260 C8PIS0 14068943 IC50 = 7000 nM T13260 CNG31F 14068944 IC50 = 700 nM T13260 CDIY35 14077737 Ki = 45 nM T13260 C8GXN7 14097196 IC50 = 7.6 nM T13260 CLZ6B8 14097212 IC50 = 2 nM T13260 CN48CH 14097214 IC50 = 14.1 nM T13260 C0G6FZ 14131679 IC50 > 10000 nM T13260 CG3QI0 14166614 IC50 = 1180 nM T13260 C98EGQ 14196997 IC50 = 100 nM T13260 CL74NV 14213544 IC50 > 40 ug.mL-1 T13260 CI3FX8 14231148 IC50 = 47.86 nM T13260 CC8A0Q 14231150 IC50 = 10.96 nM T13260 CVG0J5 14231162 IC50 = 37.15 nM T13260 C67SBC 14231174 IC50 = 58.88 nM T13260 C58ATZ 14236566 IC50 > 40 ug.mL-1 T13260 CX17LO 14311671 Ki = 670 nM T13260 CDT9L8 14442755 Ki = 260 nM T13260 CJ2CW1 14442756 Ki = 103000 nM T13260 CJX8L5 14442758 Ki = 1198000 nM T13260 CL23QM 14442760 Ki = 130000 nM T13260 CY1G3T 14442762 Ki = 893000 nM T13260 CBI6E0 14442764 Ki = 13000 nM T13260 CI93VX 14442766 Ki = 8560 nM T13260 CKI1V2 14442768 Ki = 3980 nM T13260 C1LZV9 14442770 Ki = 45000 nM T13260 C2TWN4 14442772 Ki = 97000 nM T13260 CQ47RM 14542252 IC50 > 40 ug.mL-1 T13260 C91JNH 14607641 Ki = 100 nM T13260 CM4J5C 14670839 IC50 > 20000 nM T13260 C6CX1G 14732022 Ki = 46 nM T13260 C9OIP8 14777454 Ki = 12 nM T13260 CM52ZO 14777455 Ki = 12 nM T13260 CGE64N 14777478 Ki = 610 nM T13260 CB78FM 14852902 IC50 = 95.5 nM T13260 C3L8RM 14860771 Ki = 170 nM T13260 CYJU57 14860774 Ki = 289 nM T13260 CD6GC9 14860775 Ki = 170 nM T13260 C5EL2K 14860776 IC50 = 38000 nM T13260 CJ47KS 14860787 IC50 = 44000 nM T13260 C86IZO 14860791 IC50 = 100000 nM T13260 CUK4V7 14860794 Ki = 228 nM T13260 CUC7R6 14860795 Ki = 455 nM T13260 CT8X3G 14860799 Ki = 443 nM T13260 CQ2KA6 14860801 IC50 = 26000 nM T13260 CG41LP 14860811 Ki = 7750 nM T13260 C3TC1N 14872622 IC50 = 111 nM T13260 CIX71V 14872623 IC50 = 225 nM T13260 CLSM38 14872624 IC50 = 13 nM T13260 CN3O6Y 14872625 IC50 = 97 nM T13260 CY9G4S 14872626 IC50 = 240 nM T13260 CKW32M 14872634 IC50 = 2000 nM T13260 CK94GY 14872635 IC50 = 62 nM T13260 CD30OJ 14872636 IC50 = 31 nM T13260 C2OL5D 14872637 IC50 = 49 nM T13260 CLAX71 14890692 IC50 = 150 nM T13260 C62CXN 14890719 IC50 = 2100 nM T13260 C71PWS 14890720 IC50 = 13000 nM T13260 C92AQW 14927492 Ki = 1410 nM T13260 C92OWZ 14929519 IC50 > 98400 nM T13260 CP9F8I 14939800 IC50 = 17000 nM T13260 CS26UK 15068090 Ki = 926 nM T13260 C19BZH 15068091 Ki = 870 nM T13260 C3WMI4 15072946 IC50 = 6300 nM T13260 CRHI64 15072947 IC50 = 8912.51 nM T13260 CVU3M9 15072948 IC50 = 691.83 nM T13260 CD06BM 15072949 IC50 = 8600 nM T13260 CFM3T0 15072950 IC50 = 3000 nM T13260 C39GNY 15072951 IC50 = 2200 nM T13260 CBC15T 15072952 IC50 = 6200 nM T13260 CI2QF0 15072953 IC50 = 4900 nM T13260 CAM0B5 15079867 IC50 = 7.2 nM T13260 C69EXT 15079869 IC50 = 43.65 nM T13260 CB0HE6 15079883 IC50 = 95.5 nM T13260 C8KQE9 15180664 IC50 = 290 nM T13260 C3RQS5 15182462 IC50 = 3350 nM T13260 CJ09IM 15182464 IC50 = 69 nM T13260 C9KTC2 15182466 IC50 = 10000 nM T13260 C0H2MI 15182467 IC50 = 30.2 nM T13260 CQM9J1 15182468 IC50 = 370 nM T13260 C7D1CO 15182471 IC50 = 2800 nM T13260 CL7C3M 15182472 IC50 = 2818.38 nM T13260 C5YCE7 15182473 IC50 = 933.25 nM T13260 CB0K4F 15182475 IC50 = 330 nM T13260 C8LSJ6 15182477 IC50 = 66 nM T13260 C07YXF 15192231 IC50 = 96 nM T13260 CSR6T4 15250744 IC50 = 650 nM T13260 CL4E7S 15250885 Ki = 38 nM T13260 CRBA42 15250961 Ki = 100 nM T13260 CX03MI 15250962 Ki = 100 nM T13260 CG28BA 15341075 Ki = 6 nM T13260 CV05SR 15341076 Ki = 12 nM T13260 C30CFK 15383327 Ki = 58 nM T13260 CY5D3M 15485639 IC50 > 50000 nM T13260 C4E5CF 15516845 IC50 > 242400 nM T13260 C6W1EU 15541561 IC50 = 1700 nM T13260 C6FW0G 15658944 IC50 = 2700 nM T13260 CCEG42 15658945 IC50 = 800 nM T13260 C5FH9P 15658946 IC50 = 940 nM T13260 CS97IP 15658947 Ki = 36 nM T13260 CMZ08Y 15658949 Ki = 169 nM T13260 CXQG31 15680919 IC50 = 23000 nM T13260 C1OD2W 15680920 IC50 > 200000 nM T13260 CJ80RP 15680922 IC50 = 4100 nM T13260 C0NHV8 15680923 IC50 = 26000 nM T13260 CMD4C5 15703577 IC50 = 1200 nM T13260 C2CZB1 15710342 IC50 = 10000 nM T13260 CN4H6E 15754992 Ki = 2200 nM T13260 C2TB7G 15765776 IC50 = 42300 nM T13260 CZ32OY 15801213 Ki = 8.8 nM T13260 CV3N8J 15819093 Ki = 143 nM T13260 CTQK31 15926847 Ki = 1424 nM T13260 C7ZF5H 15926848 Ki = 1424 nM T13260 CK90YW 15926849 Ki = 61 nM T13260 CT7KD6 15926850 Ki = 60.9 nM T13260 C1T5KN 15926851 Ki = 174 nM T13260 CX7EL3 15926852 Ki = 60.9 nM T13260 CATK37 15926853 Ki = 94 nM T13260 C6FX8Y 15926855 Ki = 95 nM T13260 CYKA87 15926857 Ki = 88 nM T13260 CIN54V 15926859 Ki = 88 nM T13260 C31YEX 15949288 IC50 = 3000 nM T13260 CWIH26 16004744 IC50 = 180 nM T13260 CDO2P0 16051602 IC50 = 180 nM T13260 CA2MG0 16051603 IC50 = 700 nM T13260 CR0V1J 16051604 IC50 = 1100 nM T13260 CN05YL 16051605 IC50 = 1340 nM T13260 CBR91V 16051709 IC50 = 550 nM T13260 CI7AB0 16059386 IC50 = 20000 nM T13260 C4IX5G 16063410 IC50 = 12630 nM T13260 CAJ31C 16078976 IC50 = 3680 nM T13260 CU32JA 16114920 IC50 = 28300 nM T13260 C1WMH9 16124988 IC50 = 2170 nM T13260 C43QWJ 16124989 IC50 = 330 nM T13260 C0CA7G 16125055 IC50 = 2330 nM T13260 C9PM6N 16125056 IC50 = 7820 nM T13260 CG8R9J 16125059 IC50 = 580 nM T13260 CAT4J7 16125061 IC50 = 330 nM T13260 C30WQC 16125062 IC50 = 850 nM T13260 CY6T7B 16125116 IC50 = 230 nM T13260 CQI2W7 16125118 IC50 = 1170 nM T13260 C0A1WJ 16125119 IC50 = 370 nM T13260 CVG37K 16125176 IC50 = 810 nM T13260 CF93LW 16125180 IC50 = 400 nM T13260 C9JBA6 16125181 IC50 = 260 nM T13260 CDG07Z 16125182 IC50 = 490 nM T13260 CR9SW1 16125242 IC50 = 2680 nM T13260 C42SBM 16125249 IC50 = 1750 nM T13260 C4H7BV 16125314 IC50 = 7450 nM T13260 C9FQU1 16125315 IC50 = 5850 nM T13260 CXD90Z 16125316 IC50 = 5740 nM T13260 C8OYB6 16125317 IC50 = 470 nM T13260 CK1YQ5 16125318 IC50 = 1780 nM T13260 C3M9OJ 16125319 IC50 = 2400 nM T13260 C38VAJ 16125320 IC50 = 650 nM T13260 CU3X2I 16125321 IC50 = 520 nM T13260 CBL30A 16126879 IC50 = 70 nM T13260 C9BC0L 16732000 IC50 > 100000 nM T13260 C6G0AI 16737077 IC50 > 261500 nM T13260 C03XMV 16737078 IC50 > 261500 nM T13260 CI6AJ9 16737167 IC50 > 271400 nM T13260 CUB9P7 16737277 IC50 = 3670 nM T13260 C3IJ8X 16737837 IC50 = 13950 nM T13260 C6ITS8 16738014 IC50 = 4670 nM T13260 CZ7PO3 16738015 IC50 = 28650 nM T13260 C4VB7R 16738021 IC50 = 4080 nM T13260 C5B7NL 16738022 IC50 = 4750 nM T13260 CX5QL0 16738023 IC50 = 12100 nM T13260 CC9XH1 16738210 IC50 = 54670 nM T13260 CJNP76 16738212 IC50 = 82940 nM T13260 CEIO82 16738409 IC50 > 283750 nM T13260 CB79UM 16738411 IC50 = 7670 nM T13260 CCE5G1 16738412 IC50 = 25140 nM T13260 C8QEL7 16738421 IC50 > 295500 nM T13260 CF9ZR8 16738422 IC50 > 310200 nM T13260 CG3F9E 16747839 IC50 = 0.6 nM T13260 CUX1Q4 16747937 IC50 = 560 nM T13260 CN43EH 16747938 IC50 = 7.3 nM T13260 C19REJ 16747939 IC50 = 260 nM T13260 CFI2P7 16747940 IC50 = 5.3 nM T13260 CBZE53 16747941 IC50 = 31 nM T13260 C6RB8S 16747942 IC50 = 25.9 nM T13260 CC5OW7 16748063 IC50 = 17.7 nM T13260 C6H2YB 16748064 IC50 = 400 nM T13260 CVHS73 16748915 IC50 = 0.33 nM T13260 CFX0I7 16749017 IC50 = 1.5 nM T13260 C23CUO 16749018 IC50 = 2.8 nM T13260 CEB09A 16749022 IC50 = 27 nM T13260 C03MDH 16749112 IC50 = 0.88 nM T13260 C6L3DF 16749115 IC50 = 0.51 nM T13260 CS7G6V 16749118 IC50 = 7.6 nM T13260 C0C8HL 16749219 IC50 = 159 nM T13260 CZV59A 16749224 IC50 = 0.18 nM T13260 CNG1F9 16749332 IC50 = 0.5 nM T13260 CQNA43 16749333 IC50 = 1.2 nM T13260 CNHX39 16749336 IC50 = 0.4 nM T13260 CBU08D 16749337 IC50 = 42 nM T13260 C6U7AF 16749441 IC50 = 2.9 nM T13260 CG5KQ0 16749446 IC50 = 24 nM T13260 CC2YU9 17255947 IC50 = 28.7 nM T13260 CHUA83 17966236 Ki = 2400 nM T13260 CKQJ89 18599501 Ki = 8.2 nM T13260 C6WT3S 18628989 IC50 = 913 nM T13260 CZ7PK3 18632820 IC50 = 1000 nM T13260 CT85EY 18731901 IC50 > 50000 nM T13260 CK3SA5 19043020 IC50 = 288.4 nM T13260 C4YOJ7 19043038 IC50 = 147.91 nM T13260 CKX53Q 19043046 IC50 = 870.96 nM T13260 CNS3K1 20757276 IC50 = 750 nM T13260 CK87YW 20841680 Ki = 106 nM T13260 CSKO15 21044501 IC50 = 0.51 nM T13260 CVA07N 21044507 IC50 = 0.73 nM T13260 CA7ZH9 21121774 Ki = 610 nM T13260 C16NDX 21142052 IC50 > 12500 nM T13260 CWPF92 21278956 IC50 = 2300 nM T13260 C3K1MC 21682806 IC50 = 300 nM T13260 C9WKT3 21976841 IC50 = 2.8 nM T13260 CK2ZS8 21976856 IC50 = 43 nM T13260 CE7PI2 21976872 IC50 = 2.5 nM T13260 CN5FM4 21976888 IC50 = 15 nM T13260 C9CG8L 21976892 IC50 = 10 nM T13260 C6WC7P 21976903 IC50 = 2.9 nM T13260 C75VCH 21976905 IC50 = 178 nM T13260 CR9C7D 21976908 IC50 = 0.28 nM T13260 C1KU7Z 22278552 Ki = 150 nM T13260 CR73VN 22809920 Ki = 100 nM T13260 C25LBI 23220724 IC50 = 4580 nM T13260 CLV8H7 23365315 IC50 = 18.2 nM T13260 C9ALK0 23383196 IC50 = 270 nM T13260 CHL65N 23585513 IC50 = 14.4 nM T13260 CHW5O3 23585518 IC50 = 275 nM T13260 CMN52Q 23585571 IC50 = 0.2 nM T13260 CN3CK2 23585671 IC50 = 0.5 nM T13260 CWR42I 23585720 IC50 = 0.15 nM T13260 C43IUA 23585722 IC50 = 0.2 nM T13260 CVFG27 23585723 IC50 = 0.1 nM T13260 CVJ95M 23585770 IC50 = 6 nM T13260 C30WOI 23585773 IC50 = 74 nM T13260 C5VWK3 23644932 Ki = 1820 nM T13260 CT8BJ4 23644933 Ki = 250 nM T13260 C6D9MC 23644934 Ki = 4400 nM T13260 COB81D 23644935 IC50 = 18000 nM T13260 C91ZAQ 23644936 IC50 > 50000 nM T13260 CWX70I 23644937 IC50 > 50000 nM T13260 C2I1BV 23644938 IC50 > 50000 nM T13260 C13NZL 23644951 IC50 = 85 nM T13260 CKBT84 23644968 Ki = 54 nM T13260 CC7FB8 23644969 Ki = 19 nM T13260 CJ3FX4 23644970 Ki = 22 nM T13260 C40DSL 23644971 Ki = 16 nM T13260 C8LJ4B 23644972 Ki = 11 nM T13260 C38VLD 23644973 Ki = 25 nM T13260 CNQ12D 23644974 Ki = 20 nM T13260 CR8VS6 23644975 Ki = 43 nM T13260 CF47DK 23644976 Ki = 4.7 nM T13260 CH5L6T 23644977 Ki = 7 nM T13260 CY1EL0 23644978 Ki = 14 nM T13260 C20LOE 23644979 Ki = 5 nM T13260 CDZN28 23644980 Ki = 8 nM T13260 CBVS04 23644981 Ki = 7.8 nM T13260 CO26RY 23644982 IC50 = 0.037 nM T13260 C4BPW5 23644983 IC50 = 0.11 nM T13260 CYV81F 23644984 IC50 = 0.23 nM T13260 CGF0J4 23644985 IC50 = 9 nM T13260 CVX82D 23644986 IC50 > 50 nM T13260 CG98LY 23644987 IC50 = 0.049 nM T13260 C9JD7L 23644988 IC50 = 0.32 nM T13260 C9JHP1 23644989 IC50 = 0.44 nM T13260 C7ZTD4 23644990 IC50 = 12 nM T13260 COF70P 23644991 IC50 > 50 nM T13260 CYG5P8 23644992 IC50 = 0.19 nM T13260 C74ILW 23644993 IC50 = 0.16 nM T13260 C5T6NR 23644994 IC50 = 0.12 nM T13260 C6FK7A 23644995 IC50 = 0.05 nM T13260 CIN07U 23644996 IC50 = 0.26 nM T13260 C8NY5J 23644997 IC50 = 0.13 nM T13260 C6EZ5V 23644998 Ki = 0.38 nM T13260 C0KZA5 23644999 Ki = 0.18 nM T13260 CKH5D2 23645000 Ki = 2.9 nM T13260 C27FSX 23645001 Ki = 44 nM T13260 CIQ42N 23645002 IC50 > 50 nM T13260 CX8Q9F 23645003 Ki = 0.14 nM T13260 C50OAY 23645004 Ki = 0.34 nM T13260 C5I6RZ 23645005 Ki = 5.5 nM T13260 C6PFS4 23645006 IC50 > 50 nM T13260 CIKQ38 23645007 IC50 > 50 nM T13260 C2DK6T 23645008 Ki = 0.045 nM T13260 CM2JR9 23645024 IC50 = 7400 nM T13260 C0HD7V 23645025 IC50 = 22 nM T13260 C73XCN 23645026 IC50 = 870 nM T13260 CTU28I 23645027 IC50 > 10000 nM T13260 CTUW15 23645028 IC50 > 10000 nM T13260 CL35CQ 23645029 IC50 = 10000 nM T13260 C2P7DG 23645030 IC50 > 10000 nM T13260 C89VHK 23645031 IC50 > 10000 nM T13260 CGKW86 23645032 IC50 > 1000 nM T13260 C2I9XH 23645033 IC50 = 400 nM T13260 C3J6KZ 23645034 IC50 > 10000 nM T13260 CEM21C 23645035 IC50 > 1000 nM T13260 CQ1KF8 23645036 IC50 > 1000 nM T13260 C1IT7Q 23645037 IC50 > 1000 nM T13260 CM81SC 23645038 IC50 > 1000 nM T13260 CA7DX4 23645039 IC50 > 1000 nM T13260 C1CQ4N 23645040 IC50 = 1000 nM T13260 CJV60Q 23645041 IC50 = 570 nM T13260 CQH8D4 23645042 IC50 = 270 nM T13260 C9L5EJ 23645043 IC50 = 50 nM T13260 C1X5NC 23645044 IC50 > 1000 nM T13260 CA76DP 23645045 IC50 > 1000 nM T13260 CLK43G 23645046 IC50 > 1000 nM T13260 C74MFK 23645047 IC50 = 330 nM T13260 CF48RD 23645048 IC50 = 50 nM T13260 C3A5VO 23645049 IC50 > 1000 nM T13260 CS2T8L 23645050 IC50 > 1000 nM T13260 CB24PD 23645051 IC50 > 1000 nM T13260 CLCA31 24204030 IC50 = 3100 nM T13260 CQ41JU 24204037 IC50 = 2400 nM T13260 CPJ8Z9 24205803 IC50 = 4400 nM T13260 CRH52Y 24205804 IC50 = 9100 nM T13260 C2PYN1 24420563 IC50 = 160 nM T13260 CP1YO7 24424201 IC50 = 800 nM T13260 CGVM50 24431784 IC50 > 50000 nM T13260 C6D2NZ 24692916 IC50 = 3715.35 nM T13260 CBU73T 24806841 IC50 > 25000 nM T13260 CA0YQ2 24806842 IC50 > 25000 nM T13260 CC92RE 24806843 IC50 > 25000 nM T13260 C17MET 24807041 IC50 > 25000 nM T13260 C9CMI7 24807042 IC50 > 25000 nM T13260 CZ6I0R 24807043 IC50 > 25000 nM T13260 CMY75P 24807044 IC50 > 25000 nM T13260 CJO96W 24807045 IC50 > 25000 nM T13260 CS8GB3 24807046 IC50 = 2170 nM T13260 C2B4HN 24807239 IC50 = 17370 nM T13260 C39TNQ 24807240 IC50 = 1100 nM T13260 C3PRI8 24807241 IC50 = 16670 nM T13260 CM4P0V 24807242 IC50 = 1770 nM T13260 CS01MP 24807243 IC50 = 250 nM T13260 C3BSZ8 24807244 IC50 = 690 nM T13260 CNTI27 24807245 IC50 = 690 nM T13260 C18DIO 24807434 IC50 = 440 nM T13260 C6CA8F 24807435 IC50 = 1070 nM T13260 C8NR1Y 24807436 IC50 = 120 nM T13260 CC73NY 24873506 IC50 = 1370 nM T13260 CAX9V3 24873507 IC50 = 1540 nM T13260 CS2IG5 24873508 IC50 = 610 nM T13260 C5TA7V 24873509 IC50 = 630 nM T13260 CW3C5U 24896569 IC50 = 38 nM T13260 CS5H2A 24896701 IC50 > 15300 nM T13260 CBZ10U 24901645 IC50 = 13 nM T13260 CY27CS 24901646 IC50 = 12 nM T13260 CD9IV7 24901647 IC50 = 3 nM T13260 CMFU23 24901648 IC50 = 3.2 nM T13260 CTJ76G 24901649 IC50 = 14.3 nM T13260 CJ7R6C 24901650 IC50 = 2457 nM T13260 CVS08H 24901651 IC50 = 169 nM T13260 C2H8EA 24901652 IC50 = 215 nM T13260 CUF1O4 24901653 IC50 = 5.5 nM T13260 C9C0AB 24901654 IC50 = 1.8 nM T13260 CEB6G1 24901655 IC50 = 0.6 nM T13260 CE5QO1 24901656 IC50 = 3.4 nM T13260 C23PCS 25022806 IC50 = 13.7 nM T13260 CF02OB 25071641 IC50 = 11.5 nM T13260 CMXL59 25111668 Ki = 2100 nM T13260 C35FYQ 25111796 IC50 > 500000 nM T13260 C8J2AP 25111799 IC50 > 500000 nM T13260 C06ECA 25111909 Ki = 1530 nM T13260 CON29S 25141424 IC50 = 0.45 nM T13260 CZX08M 25142015 Ki = 13 nM T13260 CV2DP9 25180002 IC50 = 6500 nM T13260 C0XHA2 25180109 IC50 = 426 nM T13260 CS8YW6 25227426 IC50 = 33000 nM T13260 CC1S3T 25256841 IC50 = 24400 nM T13260 CA4G8Y 42597583 IC50 = 13 nM T13260 C5N9MC 42611455 IC50 = 5300 nM T13260 C93BZJ 42618027 IC50 = 1250 nM T13260 C4YXR5 42618028 IC50 = 31500 nM T13260 CVLR83 42618034 IC50 = 5680 nM T13260 CUWO14 42618035 IC50 = 760 nM T13260 CZW8L2 43137984 IC50 = 289 nM T13260 CCZY29 44266320 IC50 = 620 nM T13260 C1BGQ4 44266331 IC50 = 1600 nM T13260 CEHD28 44266353 IC50 = 800 nM T13260 C79VFZ 44275189 Ki = 12 nM T13260 CQ31TG 44275201 Ki = 22 nM T13260 C83QEP 44275202 Ki = 6.7 nM T13260 CDK2T1 44275250 Ki = 5.1 nM T13260 CJ48ZL 44275251 Ki = 63 nM T13260 C78OQW 44275252 Ki = 31 nM T13260 CG4FB5 44275253 Ki = 10 nM T13260 C0OE3W 44275268 Ki = 21 nM T13260 CZ9K6I 44275269 Ki = 11 nM T13260 CP29RM 44275270 Ki = 37 nM T13260 CP2QV1 44275283 Ki = 5.6 nM T13260 C1A6OS 44275328 Ki = 4.7 nM T13260 CLN69H 44275329 Ki = 62 nM T13260 C1LQC6 44275331 Ki = 1.4 nM T13260 CZWI57 44275351 Ki = 8.8 nM T13260 C9R1OJ 44275355 Ki = 4.6 nM T13260 CC30JG 44276238 IC50 = 777000 nM T13260 CN9W6A 44276773 Ki = 75 nM T13260 C7GMW1 44277065 Ki = 1 nM T13260 C76XWA 44277083 Ki = 7 nM T13260 C3SU7M 44286352 IC50 = 170 nM T13260 CH4TJ0 44286353 IC50 = 2900 nM T13260 C74AKY 44286427 IC50 = 200 nM T13260 C0KVR6 44286475 IC50 = 70 nM T13260 C4WE8P 44286839 IC50 = 110 nM T13260 C2T1CJ 44286840 IC50 = 90 nM T13260 CZO6F2 44287464 Ki = 30 nM T13260 C8D9XI 44287465 Ki = 27 nM T13260 CK76RT 44287659 IC50 = 4400 nM T13260 C08POV 44287660 IC50 = 10000 nM T13260 CMA78S 44287741 IC50 = 4400 nM T13260 CGUX54 44287754 IC50 = 1200 nM T13260 CNF17L 44287801 Ki = 30 nM T13260 C5F6MV 44294033 Ki = 63 nM T13260 CHNJ98 44294100 Ki = 27 nM T13260 C7T9RN 44294311 Ki = 926 nM T13260 C5U1JS 44294312 Ki = 870 nM T13260 CMW32B 44294314 Ki = 11 nM T13260 C5JHW7 44294332 Ki = 190 nM T13260 C4TY5K 44306234 IC50 = 200 nM T13260 CCE7A4 44306491 IC50 = 52020 nM T13260 CUQ6L9 44306493 IC50 = 2170 nM T13260 CGU34E 44306494 IC50 = 3000 nM T13260 C9GRJ2 44306526 IC50 = 590 nM T13260 CN34EP 44306915 IC50 = 190 nM T13260 C8RQ5W 44306929 IC50 = 880 nM T13260 C80ZJS 44307719 Ki = 47 nM T13260 C76BWU 44307720 Ki = 28 nM T13260 CM52NG 44307837 Ki = 100 nM T13260 CF1K2N 44310044 Ki = 3000 nM T13260 CB30FN 44310045 Ki = 1800 nM T13260 C0QZ5L 44310046 Ki = 7000 nM T13260 C3QWV2 44310077 Ki = 13000 nM T13260 C32AUZ 44310078 Ki = 2000 nM T13260 CLJ45R 44310148 Ki = 1400 nM T13260 CEOU45 44310393 Ki = 5500 nM T13260 CZMQ71 44310410 Ki = 11000 nM T13260 CKNF03 44310411 Ki = 45000 nM T13260 C6X7WP 44310412 Ki = 9800 nM T13260 C90SJZ 44310767 Ki = 5300 nM T13260 C8W3VA 44310768 Ki = 11000 nM T13260 CO2SE0 44323417 IC50 = 3200 nM T13260 CRW0C1 44323482 IC50 = 2400 nM T13260 C0FAY8 44323523 IC50 = 2500 nM T13260 CRG1T9 44323592 IC50 = 31000 nM T13260 CQM56K 44323610 IC50 = 10000 nM T13260 C63FUL 44323664 IC50 = 3000 nM T13260 CVF86M 44323741 IC50 = 245000 nM T13260 CZIS73 44323756 IC50 = 21000 nM T13260 C0J6ZI 44323759 IC50 = 3600 nM T13260 CQC0G4 44323760 IC50 = 30000 nM T13260 CADY94 44323768 IC50 = 800 nM T13260 CGK6B2 44323782 IC50 = 1500 nM T13260 CQT35R 44323783 IC50 = 6600 nM T13260 CR5S8Z 44323807 IC50 = 40000 nM T13260 C87RGX 44323808 IC50 = 385000 nM T13260 CY1OB4 44323813 IC50 = 4000 nM T13260 CI0H9D 44323814 IC50 = 6000 nM T13260 CLE87R 44328597 Ki = 18.9 nM T13260 CX8DV2 44328668 Ki = 13.1 nM T13260 CXS8N4 44330891 Ki = 25000 nM T13260 C38YFI 44330892 Ki = 1100 nM T13260 C09VTC 44330997 Ki = 12 nM T13260 CFW8Q5 44330998 Ki = 3000 nM T13260 C5CF2O 44331012 Ki = 4.7 nM T13260 CQ85VL 44331071 Ki = 1 nM T13260 CL1YN0 44331102 Ki = 35000 nM T13260 CJIW38 44331119 Ki = 56 nM T13260 CHY39A 44331123 Ki = 1.3 nM T13260 C2MZO4 44331205 Ki = 2.3 nM T13260 CZHI57 44331221 Ki = 3 nM T13260 CXY2W3 44331222 Ki = 9 nM T13260 C28YNW 44331250 Ki = 33000 nM T13260 CR1YC8 44331322 IC50 = 30 nM T13260 CQR2U5 44333942 IC50 = 340 nM T13260 CL4Q0F 44333943 IC50 = 97 nM T13260 CX6Q1N 44334361 IC50 = 89 nM T13260 CB2D4V 44334394 IC50 = 9700 nM T13260 CSO4C8 44334411 IC50 = 11800 nM T13260 CCZ60G 44334579 IC50 = 310 nM T13260 CBZV02 44334580 IC50 = 120 nM T13260 CSR90W 44334594 IC50 = 2000 nM T13260 C8GAF6 44334595 IC50 = 3200 nM T13260 CIB4F8 44339828 Ki = 37 nM T13260 CS2F5B 44340058 Ki = 10 nM T13260 C7PT2A 44340059 Ki = 47.6 nM T13260 C9YAC2 44340330 Ki = 65.8 nM T13260 C0SC3B 44341451 IC50 = 5400 nM T13260 CAD1S9 44341468 IC50 = 238 nM T13260 CKE5L8 44353429 IC50 = 236 nM T13260 CYO3B6 44353430 IC50 = 245 nM T13260 C0UDL7 44353435 IC50 = 342 nM T13260 C3XP8T 44353437 IC50 = 950 nM T13260 C0KIV8 44353626 IC50 = 800 nM T13260 CME45Q 44353627 IC50 = 658 nM T13260 CX43HZ 44353643 IC50 = 490 nM T13260 CQ5UK0 44354378 IC50 = 530 nM T13260 CO8XJ3 44354706 IC50 = 120 nM T13260 C7YDP6 44354757 IC50 = 1320 nM T13260 C1W6IR 44354758 IC50 = 3960 nM T13260 C4AXM5 44354773 IC50 = 440 nM T13260 CZN1X8 44354907 IC50 = 30000 nM T13260 CN8M5U 44354930 IC50 = 5600 nM T13260 CCA28Y 44354942 IC50 = 55000 nM T13260 CNRO38 44354943 IC50 = 3850 nM T13260 CQIP34 44354944 IC50 = 80500 nM T13260 CO1W4F 44355172 IC50 = 8900 nM T13260 CX2R3P 44355187 IC50 > 20000 nM T13260 CCF7G1 44355188 IC50 = 1700 nM T13260 C64IWU 44358640 IC50 = 7100 nM T13260 CR5M1D 44369877 Ki = 18 nM T13260 C3BDK1 44369898 Ki = 65 nM T13260 CKNO08 44369927 Ki = 59 nM T13260 CL19DY 44376315 IC50 = 92.9 nM T13260 CZE46J 44378054 IC50 = 42 nM T13260 C1I0NW 44381001 IC50 > 250000 nM T13260 CDTS58 44387709 IC50 = 15 nM T13260 CUNZ83 44394828 IC50 = 1400 nM T13260 C8I1AE 44394829 IC50 = 31600 nM T13260 C2TLS9 44404116 Ki = 50 nM T13260 CLV8R2 44408288 IC50 = 29.7 nM T13260 C9DS0J 44408292 IC50 = 26.3 nM T13260 CTD91Q 44408293 IC50 = 23.7 nM T13260 C5X7TN 44408294 IC50 = 19.3 nM T13260 CIBP08 44421541 IC50 = 57.54 nM T13260 C0WU4A 44421546 IC50 = 93.33 nM T13260 CCIE32 44421551 IC50 = 3715.35 nM T13260 C9A6IF 44421559 IC50 = 47.86 nM T13260 C5FO6U 44424773 IC50 > 310170 nM T13260 C6BE0T 44456226 IC50 > 5000 nM T13260 CY7OD4 44461241 IC50 > 50000 nM T13260 C4BAS8 44462074 Ki = 228 nM T13260 C9BE8F 44462253 Ki = 455 nM T13260 C92QWL 44521066 IC50 = 0.12 nM T13260 CG16BM 44554135 IC50 = 11500 nM T13260 C47OVI 44562528 IC50 > 500000 nM T13260 CY42QT 44562549 IC50 > 500000 nM T13260 CP3T7B 44567161 IC50 > 40 ug.mL-1 T13260 C90PBX 44567164 IC50 > 40 ug.mL-1 T13260 C49DYC 44567218 IC50 = 7500 nM T13260 CO63LK 44569291 IC50 = 2.3 nM T13260 CNZV98 44577912 IC50 = 93.8 nM T13260 CRP8A7 44577913 IC50 = 18.7 nM T13260 CW8XY2 44577949 IC50 = 1620 nM T13260 C5CSL8 44578878 IC50 = 17300 nM T13260 C2ZWD9 44578879 IC50 = 5060 nM T13260 C4F2AM 44578880 IC50 = 1040 nM T13260 C1AT7Y 44578921 IC50 = 1060 nM T13260 C60AKC 44579025 IC50 = 320 nM T13260 C50KAN 44579026 IC50 = 9960 nM T13260 CJQ67H 44579027 IC50 = 2490 nM T13260 CS4JR7 44579028 IC50 = 1070 nM T13260 CHWK61 44579029 IC50 = 870 nM T13260 C8QW4K 44579570 IC50 = 13040 nM T13260 CP53WC 44580785 IC50 = 17000 nM T13260 CGBT61 45028483 IC50 > 10000 nM T13260 CVO41F 45140953 IC50 = 2 nM T13260 CRZ6N5 45140954 IC50 = 0.5 nM T13260 C01WQZ 45141152 IC50 = 2.4 nM T13260 CT5CR6 45141153 IC50 = 0.22 nM T13260 CC3FT1 45141154 IC50 = 0.35 nM T13260 C8PB0I 45141156 IC50 = 146 nM T13260 CL2Y7U 45141157 IC50 = 29.3 nM T13260 CH1LB7 45141158 IC50 = 19 nM T13260 CDE83B 45141365 IC50 = 52 nM T13260 CGA6Y4 45141366 IC50 = 112 nM T13260 CCIP58 45141367 IC50 = 280 nM T13260 C2S5QX 45141368 IC50 = 24 nM T13260 C2YJ8N 45141369 IC50 = 80 nM T13260 CO4UA1 45141370 IC50 = 920 nM T13260 C5CB0P 45141371 IC50 = 284 nM T13260 CTN65F 45141372 IC50 = 380 nM T13260 CGK5O7 45141601 IC50 = 571 nM T13260 C68SZB 45141602 IC50 = 0.8 nM T13260 C0C3AW 45141603 IC50 = 1.9 nM T13260 C0U7CG 45141604 IC50 = 0.3 nM T13260 CQ4JE3 45378299 IC50 = 97000 nM T13260 CUR6C8 45378303 IC50 = 5100 nM T13260 CY2SV8 45379302 IC50 = 44000 nM T13260 CSE09V 46177290 IC50 = 12100 nM T13260 C4XCR3 46177291 IC50 = 12100 nM T13260 C4S2AI 46198256 Ki = 16.1 nM T13260 CT07FB 46204132 IC50 = 6400 nM T13260 CN47GA 46228644 IC50 = 4.6 nM T13260 C6AMH8 46228668 IC50 = 1.7 nM T13260 CLD4Z5 46228698 IC50 = 0.22 nM T13260 CZH36E 46834487 IC50 > 50000 nM T13260 CUV83E 46854605 IC50 = 12000 nM T13260 CIA08B 46854608 IC50 = 9500 nM T13260 CWJ3F1 46854758 IC50 = 5060 nM T13260 CKRQ67 46854759 IC50 = 49500 nM T13260 CZ1YJ0 46854760 IC50 = 48700 nM T13260 CINV65 46867541 IC50 = 101 nM T13260 CL06TP 46887017 IC50 = 17.2 nM T13260 C0KFI6 46887054 IC50 = 17.2 nM T13260 C6R1HA 46887055 IC50 = 6 nM T13260 CD65CW 46887468 IC50 = 71.8 nM T13260 CM0EK7 46887507 IC50 = 200 nM T13260 CGBE96 46887549 IC50 = 210 nM T13260 C74CER 46887577 IC50 = 3.5 nM T13260 C2OMW7 46895138 IC50 = 12000 nM T13260 CYEA34 46913124 IC50 = 70 nM T13260 C5JR7T 46913125 IC50 = 36 nM T13260 CN1CV7 46939057 Ki = 97 nM T13260 CP8HY2 46939058 Ki = 27 nM T13260 CD67MH 46939156 Ki = 23 nM T13260 C1MFE9 46939157 Ki = 75 nM T13260 C0K8YL 46939158 Ki = 39 nM T13260 CX7B9G 46939159 Ki = 30 nM T13260 CL37EV 46939160 Ki = 56 nM T13260 C9CQU0 46953209 IC50 = 59.2 nM T13260 CUQ0Z7 46957695 IC50 = 13200 nM T13260 CU0KW6 46958302 IC50 = 991 nM T13260 CHN2P9 46960541 IC50 = 34.5 nM T13260 CR3OI4 46960542 IC50 = 46.7 nM T13260 CW3V2P 46962897 IC50 = 499 nM T13260 CQ0XE9 46964149 IC50 = 10600 nM T13260 CL0F1J 46964152 IC50 > 25000 nM T13260 CV3UT0 46967737 IC50 = 3100 nM T13260 CBAE65 46968168 IC50 = 248 nM T13260 CKJ9S6 46968847 IC50 = 3100 nM T13260 CO2XL1 46970377 IC50 = 9 nM T13260 C0GZ4Q 46980515 IC50 = 498 nM T13260 C8QCH2 49779539 IC50 = 2.1 nM T13260 C7V2XL 49779540 IC50 = 0.25 nM T13260 CIC9S5 49799473 IC50 = 5750 nM T13260 C5ZNK0 49799653 IC50 = 21860 nM T13260 CZG04F 49799654 IC50 = 8490 nM T13260 CX5LZ9 50915159 IC50 = 0.018 nM T13260 C8N5OK 50991893 IC50 = 0.21 nM T13260 C0RUX1 50994677 IC50 > 10000 nM T13260 CL2O0Y 50994839 IC50 > 16200 nM T13260 CTG6R4 51041013 IC50 = 4400 nM T13260 CGX85M 51042201 IC50 = 30700 nM T13260 CWG69M 51042401 IC50 = 32300 nM T13260 C1AT4L 51042402 IC50 = 26800 nM T13260 C1VF4Z 51346982 IC50 = 0.015 nM T13260 C6Y3EL 51346989 IC50 = 0.015 nM T13260 C8GQS7 51351108 IC50 > 50000 nM T13260 CB8ND9 51354813 IC50 > 16900 nM T13260 CMXR96 51355428 IC50 = 114 nM T13260 C5KTL3 51355429 IC50 = 113 nM T13260 C4UTM8 51355430 IC50 = 130 nM T13260 CH5C9K 51355431 IC50 = 235 nM T13260 CRK2Q9 51355432 IC50 = 207 nM T13260 CF7RG5 51355433 IC50 = 141 nM T13260 C8XHD9 51355434 IC50 = 267 nM T13260 C41SUK 51355703 IC50 = 178 nM T13260 CM6T7H 51355704 IC50 = 127 nM T13260 CZDA87 51355705 IC50 = 481 nM T13260 CO1V0Y 51355706 IC50 = 169 nM T13260 C2OCG3 51355707 IC50 = 165 nM T13260 CGLU79 51355708 IC50 = 72 nM T13260 CL6XD4 51355709 IC50 = 72 nM T13260 C57MWS 51355970 IC50 = 292 nM T13260 CYC86A 51355971 IC50 = 690 nM T13260 CP7V3Q 51355972 IC50 = 112 nM T13260 CR6NH8 51355973 IC50 = 164 nM T13260 C6SD4P 51355974 IC50 = 296 nM T13260 C97MZT 51355975 IC50 = 81 nM T13260 CJU1O7 51355976 IC50 = 70 nM T13260 CIR0L7 51356252 IC50 = 47 nM T13260 C0BW7G 51356253 IC50 = 105 nM T13260 C39RVA 51356254 IC50 = 3750 nM T13260 C3P5LI 51356255 IC50 = 455 nM T13260 CKXR01 51356256 IC50 = 67 nM T13260 CF21EH 51356258 IC50 = 317 nM T13260 C4M5ZT 51356554 IC50 = 532 nM T13260 CS7X3R 51356555 IC50 = 4010 nM T13260 CR7UG9 51356556 IC50 = 313 nM T13260 C87FEB 51520434 IC50 = 600 nM T13260 C42JIQ 52912619 IC50 = 5040 nM T13260 CY0TF7 53237486 IC50 = 510 nM T13260 C5WQX4 53237725 IC50 = 1000 nM T13260 CD7HC1 53305315 IC50 = 91 nM T13260 C5SN8I 53317948 IC50 = 11000 nM T13260 CQZV41 53318733 IC50 = 30000 nM T13260 C9OPT6 53320278 IC50 = 0.75 nM T13260 CDM50Q 53320823 IC50 = 660 nM T13260 CRLJ68 53321508 IC50 = 700 nM T13260 CCNP36 53321604 IC50 = 0.47 nM T13260 CDV3X5 53323228 IC50 = 3600 nM T13260 C4WY6N 53323229 IC50 = 1000 nM T13260 CFC42O 53323677 IC50 > 16800 nM T13260 CFMK70 53324579 IC50 = 280 nM T13260 C48XBG 53325332 IC50 = 860 nM T13260 CA32FG 53325544 IC50 = 0.05 nM T13260 CN0SW9 53326827 IC50 = 0.1 nM T13260 CSQ45A 53326828 IC50 = 0.15 nM T13260 C0AL2O 53482563 IC50 = 11.8 nM T13260 C0P3VM 53637746 Ki = 58 nM T13260 CAE25J 53763992 IC50 = 970 nM T13260 CUXV34 54026593 Ki = 120 nM T13260 C53FSN 54165563 Ki = 7 nM T13260 C8FA6I 54348149 Ki = 58 nM T13260 CA19BF 54513089 Ki = 25 nM T13260 CE0PC5 54576531 IC50 = 4640 nM T13260 CS0NM1 54576532 IC50 = 1360 nM T13260 CA3YL8 54580402 IC50 = 5790 nM T13260 CB5QY9 54583302 IC50 = 34 nM T13260 CB02LJ 54584262 IC50 = 32 nM T13260 C34FYG 54584352 IC50 = 66.5 nM T13260 CLPG92 54586184 IC50 = 36 nM T13260 C91LBU 54597383 IC50 = 3300 nM T13260 C6G8HK 54597384 IC50 = 1800 nM T13260 CV2NS6 54729584 IC50 = 220 nM T13260 C70EIF 54756790 IC50 > 50000 nM T13260 CZU5L8 54768666 IC50 = 17340 nM T13260 C4C1ZY 54768667 IC50 = 10700 nM T13260 C5AVO9 54770656 IC50 = 12200 nM T13260 C2RW0G 54770885 IC50 = 12010 nM T13260 CW6EK4 54770886 IC50 = 4700 nM T13260 CTP0G9 54770887 IC50 = 5070 nM T13260 CHY71M 54770888 IC50 = 10600 nM T13260 CS42BX 54770889 IC50 = 16020 nM T13260 CU07HL 54770890 IC50 = 19320 nM T13260 CD2JA7 54770891 IC50 = 10330 nM T13260 CD1V8X 54771121 IC50 = 79980 nM T13260 CMX14D 54771122 IC50 = 10970 nM T13260 CVED14 54771123 IC50 = 16110 nM T13260 CPJW41 54771124 IC50 = 7730 nM T13260 C8JEH4 54771125 IC50 = 10950 nM T13260 CA4JF1 54771126 IC50 = 12160 nM T13260 C6Y8ND 54771341 IC50 = 10960 nM T13260 C7E3KS 54771342 IC50 = 14830 nM T13260 C6NRM1 54771343 IC50 = 19360 nM T13260 C3MR9N 54771344 IC50 = 13540 nM T13260 CI5QD9 54771345 IC50 = 13720 nM T13260 C7KBU3 54771346 IC50 = 12940 nM T13260 C7LOA4 54771347 IC50 = 31260 nM T13260 C8OI5N 54771563 IC50 = 13350 nM T13260 CUF4O0 54771564 IC50 = 13370 nM T13260 CP1UM5 54771565 IC50 = 16410 nM T13260 C3ZKB4 54771566 IC50 = 11610 nM T13260 C3YD8A 54771567 IC50 = 26770 nM T13260 C3URW8 54771568 IC50 = 15210 nM T13260 C2BYD3 54771787 IC50 = 4370 nM T13260 CUY87L 54771788 IC50 = 5260 nM T13260 C3WVO7 54771789 IC50 = 3070 nM T13260 CYM98K 54771790 IC50 = 7880 nM T13260 CV5S9D 54771791 IC50 = 10700 nM T13260 C2G6DW 54771792 IC50 = 6090 nM T13260 CHOT94 54771793 IC50 = 3910 nM T13260 CA49SQ 54771794 IC50 = 9160 nM T13260 CN2ES5 54772014 IC50 = 15480 nM T13260 C38PQF 54772015 IC50 = 5620 nM T13260 C3Q9YI 54772016 IC50 = 4170 nM T13260 C76QVG 54772017 IC50 = 2340 nM T13260 C5KI4U 54772018 IC50 = 11570 nM T13260 CR1YL2 54772019 IC50 = 7470 nM T13260 C1OQ4B 54772020 IC50 = 9530 nM T13260 CL7XJ4 54772021 IC50 = 7980 nM T13260 C06PFH 56598207 IC50 = 10500 nM T13260 CL4KT8 56610874 Ki = 8.2 nM T13260 C78MXU 56612673 Ki = 8.2 nM T13260 CV1ZO2 56632357 Ki = 90 nM T13260 C4N0WL 56645363 IC50 = 1021 nM T13260 C57NSZ 56645568 IC50 = 1268 nM T13260 C6PUX9 56645570 IC50 = 4513 nM T13260 CM94ZH 56664989 IC50 = 2780 nM T13260 CMU51H 56681975 IC50 = 2270 nM T13260 C7G5IR 56835177 Ki = 790 nM T13260 C5US1Z 56835178 Ki = 60 nM T13260 C3IZU1 56835179 Ki = 50 nM T13260 CRGX16 56837844 IC50 > 50000 nM T13260 C7M1OX 56837845 IC50 > 50000 nM T13260 CHCM56 56837846 IC50 > 50000 nM T13260 CX19AT 57327815 IC50 = 93 nM T13260 C0I2DY 57327816 IC50 = 59 nM T13260 CY58ZD 57330086 IC50 > 5000 nM T13260 C1C0FZ 57384102 Ki = 0.06 nM T13260 CLJ8A1 57384103 Ki = 0.65 nM T13260 C6I3AN 57390179 IC50 > 50000 nM T13260 C1ZB3N 57390180 IC50 > 50000 nM T13260 CH19RM 57390181 IC50 > 50000 nM T13260 CG2J7F 57390275 IC50 = 64500 nM T13260 C0VRP8 57391308 Ki = 12560 nM T13260 C3BKO8 57391309 Ki = 1482 nM T13260 CW3P7T 57391581 Ki = 100 nM T13260 CI1R4S 57391583 Ki = 250 nM T13260 CB02XQ 57391954 IC50 > 50000 nM T13260 C94BSM 57392056 IC50 = 63200 nM T13260 CJA4L1 57393085 Ki = 1722 nM T13260 CS6V8A 57393681 IC50 > 50000 nM T13260 CPN7Q2 57393682 IC50 > 50000 nM T13260 CV4S6C 57393683 IC50 > 50000 nM T13260 CR5I9O 57393684 IC50 > 50000 nM T13260 C5VDL7 57395400 IC50 > 50000 nM T13260 CC53MX 57395527 IC50 = 47300 nM T13260 CV08LN 57395659 IC50 = 986 nM T13260 CI6Q5O 57395660 IC50 = 304 nM T13260 CQ06KW 57395661 IC50 = 229 nM T13260 C48VIY 57396573 Ki = 5321 nM T13260 C2NML8 57396574 Ki = 8.2 nM T13260 C83ZIP 57396575 Ki = 82.54 nM T13260 C2F1TI 57397238 IC50 > 50000 nM T13260 C4O5DT 57397345 IC50 = 68100 nM T13260 CBL9Z1 57397346 IC50 = 58600 nM T13260 CXP68J 57397347 IC50 = 72000 nM T13260 C5VLB1 57398353 Ki = 35.12 nM T13260 C4DE6B 57398582 Ki = 1000 nM T13260 CW2J6Z 57398927 IC50 > 50000 nM T13260 CP65RI 57398928 IC50 > 50000 nM T13260 CHB0A3 57398929 IC50 > 50000 nM T13260 C81RCO 57398930 IC50 > 50000 nM T13260 CD4BN7 57400011 Ki = 285.1 nM T13260 CJT2G9 57400012 Ki = 100 nM T13260 CJZX60 57400626 IC50 > 50000 nM T13260 CV8KD9 57400627 IC50 > 50000 nM T13260 C3G4RJ 57400766 IC50 = 44800 nM T13260 C2WJ7Y 57400842 IC50 = 57400 nM T13260 C5OYK8 57400879 IC50 = 114 nM T13260 CHVG47 57401821 Ki = 15000 nM T13260 C1MF0V 57402418 IC50 > 50000 nM T13260 CQ9C3L 57402419 IC50 = 26500 nM T13260 CUD85V 57402656 IC50 = 523 nM T13260 CD2U9L 57403526 Ki = 1160 nM T13260 CFI0L8 57403527 Ki = 3.17 nM T13260 C10SAL 57403795 Ki = 79.43 nM T13260 CRL10W 57413872 Ki = 86 nM T13260 C04MZQ 57520593 IC50 = 17000 nM T13260 CX8Q7H 57520594 IC50 = 5800 nM T13260 CYHS09 57679076 IC50 >= 200000 nM T13260 C7OK1X 57775654 IC50 = 4490 nM T13260 CQ0M7J 58215635 IC50 = 3400 nM T13260 C34JIZ 58255359 IC50 = 2130 nM T13260 C2TUJ7 58255382 IC50 = 228 nM T13260 C3DPC0 58255407 IC50 = 43 nM T13260 C9DK1X 58255415 IC50 = 488 nM T13260 CTI0D7 58255435 IC50 = 880 nM T13260 CRQ70M 58255438 IC50 > 500 nM T13260 CLQ65O 58255479 IC50 > 5000 nM T13260 CP6RA9 58255482 IC50 = 3073 nM T13260 CJX70M 58255566 IC50 = 105 nM T13260 CW71EO 58255581 IC50 = 447 nM T13260 C6XPA7 59356082 IC50 = 24000 nM T13260 CX2US1 59356084 IC50 = 35000 nM T13260 CD31PM 59356085 IC50 = 99000 nM T13260 CVRT12 59356087 IC50 = 41000 nM T13260 CLP2O3 60151424 IC50 = 6200 nM T13260 C9M4QI 60156307 IC50 = 112.3 nM T13260 CZ1WU8 60166590 IC50 = 169.3 nM T13260 CB7N8A 60195126 IC50 = 17 nM T13260 CE18JH 60202715 Ki = 48 nM T13260 CX4N0I 62707515 IC50 = 48 nM T13260 C0G3LA 66559847 IC50 = 49 nM T13260 C4RSI6 66559935 IC50 = 162 nM T13260 CDX7I8 66559936 IC50 = 22 nM T13260 CF9EQ5 66559939 IC50 = 2901 nM T13260 CQN6D3 66559940 IC50 = 394 nM T13260 CN4H8G 66559941 IC50 = 954 nM T13260 CTP6Q4 66559942 IC50 = 275 nM T13260 C9EGW2 66575742 IC50 > 10000 nM T13260 CMXA10 66575743 IC50 > 10000 nM T13260 CKWB91 66575744 IC50 > 10000 nM T13260 C7I3MW 66575745 IC50 > 10000 nM T13260 CPN17S 66575746 IC50 > 10000 nM T13260 CG0ZA7 66575747 IC50 > 10000 nM T13260 C6HF0U 66575748 IC50 > 10000 nM T13260 CDI93T 66575817 IC50 > 10000 nM T13260 CBP6I7 66576773 IC50 > 10000 nM T13260 C4NYB0 66576930 IC50 > 10000 nM T13260 C3LP5H 66576931 IC50 > 10000 nM T13260 CE03WG 66576932 IC50 > 10000 nM T13260 C9XYA1 67205290 Ki = 700 nM T13260 CO8IZ3 67854245 IC50 = 590 nM T13260 C2F5TS 68037237 Ki = 442 nM T13260 C97FZU 68561433 IC50 = 31 nM T13260 CK05PZ 68668617 Ki = 7 nM T13260 CC75HS 69198620 IC50 = 160000 nM T13260 CI6U5W 69649421 IC50 = 160 nM T13260 CZN04V 69828765 Ki = 45 nM T13260 CSUX85 70178310 Ki = 55 nM T13260 CBM80I 70354859 Ki = 77 nM T13260 COGQ93 70680979 IC50 = 30000 nM T13260 C96QKR 70683101 IC50 = 61000 nM T13260 CBNF56 70689398 IC50 = 20000 nM T13260 CPNR72 70689399 IC50 = 32000 nM T13260 CCG0U6 70691503 IC50 = 18000 nM T13260 CKE71B 70691504 IC50 = 11000 nM T13260 CA36IC 70695715 IC50 = 29000 nM T13260 CHEJ23 70748349 IC50 = 20900 nM T13260 C1VMF2 70977969 IC50 > 10000 nM T13260 CUV23H 71449132 Ki = 22 nM T13260 C37CSD 71450101 IC50 = 181.1 nM T13260 C7EDZ9 71452741 Ki = 753 nM T13260 CFKO73 71453732 IC50 = 2180 nM T13260 CI6B9U 71454429 IC50 > 50000 nM T13260 C70TUP 71455138 IC50 = 11 nM T13260 CH70RK 71456229 IC50 = 11000 nM T13260 CFG4L5 71456934 IC50 = 35 nM T13260 C8NPL7 71457257 IC50 = 83 nM T13260 CJCY84 71457258 IC50 = 20 nM T13260 C1KY3Q 71458062 Ki = 86 nM T13260 CK5TV7 71461661 Ki = 206 nM T13260 CI16NC 71520311 IC50 = 32 nM T13260 CE9A6B 71520312 IC50 = 246 nM T13260 C03VKJ 71520313 IC50 > 5000 nM T13260 C5J7DI 71520314 IC50 = 3340 nM T13260 CE0N5C 71520315 IC50 > 5000 nM T13260 C4Z6YP 71520316 IC50 = 565 nM T13260 CC8Z6L 71520431 IC50 > 5000 nM T13260 C1DK9P 71520432 IC50 = 1500 nM T13260 C9NOQ1 71521632 IC50 = 2130 nM T13260 C0OTA2 71521716 IC50 = 3660 nM T13260 CVLE07 71521717 IC50 > 5000 nM T13260 CJKX84 71521718 IC50 = 1350 nM T13260 CZ5P9U 71521719 IC50 = 140 nM T13260 C1YCB0 71521720 IC50 = 889 nM T13260 CE57PM 71521721 IC50 = 74 nM T13260 C0O2SA 71521798 IC50 = 81 nM T13260 CMEC10 71521799 IC50 = 59 nM T13260 CR9O5T 71521800 IC50 = 273 nM T13260 C0JBI3 71521801 IC50 = 74 nM T13260 CE7Z4I 71521802 IC50 = 116 nM T13260 CW2AG4 71521803 IC50 = 19 nM T13260 C6ID7K 71521804 IC50 = 55 nM T13260 CPZ5S8 71535400 IC50 = 790 nM T13260 CCRS95 71535683 IC50 = 2200 nM T13260 C9V7KW 71568307 IC50 = 9.01 nM T13260 CZGA56 71568308 IC50 = 148.93 nM T13260 C0E3WP 71568309 IC50 = 77.36 nM T13260 C3IX0R 71568310 IC50 = 4.93 nM T13260 C1B6UY 71568311 IC50 = 16.58 nM T13260 CF6DO2 71568312 IC50 = 21.39 nM T13260 CNBX98 71568313 IC50 = 164.01 nM T13260 CLD9N8 71568314 IC50 = 138.72 nM T13260 C7YVC9 71568442 IC50 = 56.83 nM T13260 C2ZS4G 71568443 IC50 = 27.01 nM T13260 C2BD6R 71568444 IC50 = 6.23 nM T13260 C03WJE 71568445 IC50 = 48.93 nM T13260 CXH93O 71568446 IC50 = 25.56 nM T13260 C0N6UG 71568447 IC50 = 46.92 nM T13260 C3PZG5 71568448 IC50 = 57.43 nM T13260 CPI06S 71568584 IC50 = 111.09 nM T13260 CL4YR2 71568585 IC50 = 203.34 nM T13260 C7ZCL4 71568586 IC50 = 235.33 nM T13260 CTQ79Z 71568587 IC50 = 217.43 nM T13260 C58SMB 71574941 IC50 = 480 nM T13260 CC09FQ 71574942 IC50 = 460 nM T13260 CA2T5L 71574943 IC50 = 300 nM T13260 C9MFZ7 71574944 IC50 = 1100 nM T13260 CW73OE 71574945 IC50 = 1973 nM T13260 C70NHJ 71574946 IC50 = 400 nM T13260 CLH83S 71574947 IC50 = 837 nM T13260 CF71AB 71575030 IC50 = 575 nM T13260 CCG1S5 71575031 IC50 = 565 nM T13260 CH9WE7 71575032 IC50 = 260 nM T13260 CO4ZQ7 71575033 IC50 = 170 nM T13260 CT86GV 71575034 IC50 = 6393 nM T13260 CHC8L4 71614085 IC50 = 0.2 nM T13260 CKPV51 71621803 IC50 > 100000 nM T13260 CG72JK 71681355 IC50 = 9257 nM T13260 C56LUJ 71716957 IC50 = 11160 nM T13260 CJE01S 71745100 IC50 > 10000 nM T13260 C54KVE 71748876 IC50 = 670 nM T13260 CT5Q9N 71812321 IC50 = 750 nM T13260 CBL42N 71812322 IC50 = 450 nM T13260 C9IOA1 71812324 Ki = 45 nM T13260 CX0WV5 71817943 IC50 > 2000 nM T13260 CN1LU6 71817944 IC50 > 2000 nM T13260 CGV4U3 71817945 IC50 > 2000 nM T13260 CJ4L5G 71818086 IC50 > 2000 nM T13260 COXA51 71818087 IC50 > 2000 nM T13260 CP1A3M 71818088 IC50 > 2000 nM T13260 CPJ42T 71818089 IC50 > 2000 nM T13260 CAP03I 71818090 IC50 > 2000 nM T13260 CO23PK 71818091 IC50 > 2000 nM T13260 CL4X6A 71818092 IC50 > 2000 nM T13260 CL8GK5 71818093 IC50 > 2000 nM T13260 C4ZVG0 71818094 IC50 > 2000 nM T13260 CH2GR0 71818232 IC50 > 2000 nM T13260 C0VGQ9 71818233 IC50 > 2000 nM T13260 C5QRF2 71818234 IC50 > 2000 nM T13260 C09VHD 72194216 IC50 = 5500 nM T13260 C4POE7 72546693 Ki = 80 nM T13260 CKI39Q 72546694 Ki = 20 nM T13260 C2SE6Q 72546935 Ki = 111 nM T13260 C49MBW 72546936 Ki = 160 nM T13260 CJCU54 72546937 Ki = 70 nM T13260 CN1Z5U 72546938 Ki = 20 nM T13260 CD6I2S 72546939 Ki = 330 nM T13260 CKE4O3 72546940 Ki = 170 nM T13260 CW5H8C 72546941 Ki = 820 nM T13260 C74PHD 72547200 Ki = 200 nM T13260 CDC4P8 72547201 Ki = 130 nM T13260 CZNW37 72547202 Ki = 841 nM T13260 CFLU42 72547203 Ki = 110 nM T13260 C76AZT 72547204 Ki = 90 nM T13260 C1IP7G 72547205 Ki = 237 nM T13260 C62CNP 72547206 Ki = 350 nM T13260 CG0LT8 72547452 Ki = 647 nM T13260 CU76NM 72703468 IC50 > 10000 nM T13260 C9PRT7 72703681 IC50 > 10000 nM T13260 CCG7R3 72703685 IC50 = 5.3 nM T13260 CU27CK 72703887 IC50 > 10000 nM T13260 CFR2V8 72703888 IC50 > 10000 nM T13260 CAU4Z0 72703889 IC50 = 3.1 nM T13260 C56KEC 72703890 IC50 = 13.3 nM T13260 CB7PR0 72704087 IC50 = 1472 nM T13260 C5SNU6 72708597 IC50 = 3200 nM T13260 CSB7R2 73055580 IC50 = 15000 nM T13260 CG37VI 73055876 IC50 = 20000 nM T13260 CU5DC1 73055877 IC50 = 190000 nM T13260 C5M7RH 73055879 IC50 = 2500 nM T13260 C53JKM 73055880 IC50 = 67100 nM T13260 CR8V7S 73055881 IC50 = 800 nM T13260 C72LFY 73346265 IC50 = 2700 nM T13260 C5F2VZ 73347760 IC50 = 3400 nM T13260 C5QTA7 73349312 IC50 = 3400 nM T13260 CPU7N5 73350879 IC50 = 12500 nM T13260 CT1J5B 73350882 IC50 = 12500 nM T13260 C9Y5FN 73353441 IC50 = 9257 nM T13260 CT9SN8 73353827 IC50 = 4600 nM T13260 CD13BV 73353828 IC50 = 8000 nM T13260 CGWY15 73355361 IC50 = 1800 nM T13260 C1YT7X 73355362 IC50 = 9400 nM T13260 CKEY08 73355363 IC50 = 7900 nM T13260 CGF87Z 73355403 IC50 = 3900 nM T13260 C0OY5P 73356914 IC50 = 1300 nM T13260 CX12ML 73356915 IC50 = 2900 nM T13260 C0UQ3M 73356955 IC50 = 29100 nM T13260 CKG8J2 73357190 IC50 = 590 nM T13260 C9WY3B 73386689 IC50 = 45 nM T13260 CK4NQ1 76186646 IC50 = 0.9 nM T13260 CM52SI 76308995 IC50 = 11900 nM T13260 CS80JY 76310075 IC50 = 50 nM T13260 CB1V2S 76311295 IC50 = 10700 nM T13260 C7XH3E 76314886 IC50 = 80 nM T13260 CPU3T6 76317295 IC50 = 1100 nM T13260 CAM49B 76318503 IC50 = 90 nM T13260 CFJ8G5 76322165 IC50 = 40 nM T13260 C7KEG3 76322166 IC50 = 150 nM T13260 CHBR20 76325787 IC50 = 1010 nM T13260 CXD53T 76327865 IC50 = 160 nM T13260 CS8D4U 76328231 IC50 = 3000 nM T13260 C3F0JZ 76329384 IC50 > 300000 nM T13260 C3JID2 76331906 IC50 = 650 nM T13260 C1YJW0 77846787 IC50 = 790 nM T13260 CV73PD 77846790 IC50 = 10000 nM T13260 C0DIH7 77846872 IC50 = 10000 nM T13260 COI25M 77846873 IC50 = 1000 nM T13260 CJI8R0 77846875 IC50 = 3800 nM T13260 CZK4J1 77846962 IC50 = 2800 nM T13260 CEK89G 77846963 IC50 = 10000 nM T13260 C5BA8Z 77846964 IC50 = 1240 nM T13260 C4D6XJ 77847803 IC50 = 1600 nM T13260 CF7O4Q 77847804 IC50 = 1200 nM T13260 CEC49D 85863219 IC50 = 1610 nM T13260 CZ5PM0 86277538 IC50 = 0.42 nM T13260 CHV8R6 86307678 IC50 = 620 nM T13260 C3X6MJ 86792466 IC50 = 21700 nM T13260 CL30TR 89471870 IC50 = 2300 nM T13260 C3BUS8 89471889 IC50 = 420 nM T13260 CI7HY8 89471890 IC50 = 120 nM T13260 CX0M7B 89961716 IC50 = 21 nM T13260 CR5D6Y 89961785 IC50 > 10000 nM T13260 C89TEU 89968659 IC50 > 10000 nM T13260 CY5IC7 90252834 IC50 = 4600 nM T13260 C84NVA 90252850 IC50 = 6300 nM T13260 CBY46O 90252851 IC50 = 5400 nM T13260 CNVA50 90252852 IC50 = 6200 nM T13260 C89BFG 90333640 IC50 = 1820 nM T13260 CJ8NI5 90655716 Ki = 57 nM T13260 COF02L 90655717 Ki = 62 nM T13260 CO9K2W 90655718 Ki = 31 nM T13260 CX8L7D 90655719 Ki = 69 nM T13260 CHD21I 90666137 IC50 = 14.4 nM T13260 C4A7JU 90677206 IC50 = 12500 nM T13260 C3T5BI 90677209 IC50 = 12500 nM T13260 CV96EW 90677213 IC50 = 12500 nM T13260 C3Y8AQ 90677215 IC50 = 12500 nM T13260 C6PJL5 90677216 IC50 = 12500 nM T13260 CFI3J8 90677218 IC50 = 12500 nM T13260 CQ91ZO 90677219 IC50 = 12500 nM T13260 CQS8C9 91664365 IC50 = 1000 nM T13260 CM9U7B 91758284 Ki = 20 nM T13260 CLB2E7 91827654 IC50 > 30000 nM T13260 C0KDB6 91983064 Ki = 32 nM T13260 CYL1S3 97191385 IC50 = 5100 nM T13260 CXRB41 101152219 IC50 > 10000 nM T13260 C3P9ZY 101199629 IC50 = 41 nM T13260 CL3UQ9 101354484 Ki = 10 nM T13260 C26AKT 101354485 Ki = 14 nM T13260 CZXS85 101354486 Ki = 81 nM T13260 CWXT16 101378163 Ki = 45 nM T13260 C8VZC7 101378164 Ki = 45 nM T13260 C4G5MB 101378165 Ki = 670 nM T13260 C5HLB7 101378166 Ki = 670 nM T13260 C0TOW6 101433013 Ki = 8.2 nM T13260 CLI59T 101579737 IC50 = 160 nM T13260 C18UTF 101587707 Ki = 150 nM T13260 C2SUC3 101587708 Ki = 1180 nM T13260 CI0N8C 101592374 Ki = 24.1 nM T13260 CV87DF 101592375 Ki = 24.1 nM T13260 C1ZN6O 101592376 Ki = 24.1 nM T13260 C5WGQ7 101620856 Ki = 5000 nM T13260 CC01NA 101650066 Ki = 12 nM T13260 CE9T0K 101650068 Ki = 12 nM T13260 CUDV46 101650069 Ki = 12 nM T13260 CBN09G 101651130 Ki = 2 nM T13260 C9CZN6 101668720 Ki = 11100 nM T13260 C9TID7 101701780 Ki = 5000 nM T13260 C0RN1M 101927481 Ki = 25 nM T13260 C9E7GV 102068512 Ki = 7 nM T13260 C63RAU 102068514 Ki = 7 nM T13260 C8YJK2 102068516 Ki = 7 nM T13260 C57AZV 102068518 Ki = 7 nM T13260 C4J1SX 102279741 Ki = 95 nM T13260 CE90MX 102346108 IC50 = 6870 nM T13260 CED87Z 102439715 Ki = 5000 nM T13260 C0DYC5 102532604 Ki = 5000 nM T13260 C9KZ5G 102533756 Ki = 16 nM T13260 CB1Z8U 102533759 Ki = 16 nM T13260 CMO84S 110730849 IC50 = 490 nM T13260 CJ9Z0S 118496546 IC50 = 6900 nM T13260 C2BMT8 118708021 IC50 = 34400 nM T13260 C8NES2 118711691 Ki = 630.96 nM T13260 CKT4A8 118711692 Ki = 707.95 nM T13260 COD91Y 118711693 Ki = 707.95 nM T13260 CGJ93V 118711694 Ki = 25.12 nM T13260 C0WLI2 118711695 Ki = 354.81 nM T13260 CXDE52 118711696 Ki = 144.54 nM T13260 CAW5K3 118723935 IC50 = 549 nM T13260 CK8UL1 118723936 IC50 = 387 nM T13260 CIW7O0 118723937 IC50 = 477 nM T13260 C42CEZ 118723938 IC50 = 584 nM T13260 CJQ63E 118723939 IC50 = 639 nM T13260 CCXN71 118723940 IC50 = 445 nM T13260 CS78BD 118723941 IC50 = 349 nM T13260 C9W3QX 118723942 IC50 = 17464 nM T13260 COJ2K8 118723943 IC50 = 5855 nM T13260 CZ23UL 118723944 IC50 = 3708 nM T13260 CIWU64 118723945 IC50 = 4566 nM T13260 CZI6A0 118723946 IC50 = 8299 nM T13260 COB46M 118723947 IC50 = 31813 nM T13260 CJ1HP9 118728223 Ki = 10000 nM T13260 CZR62N 118730170 IC50 = 810 nM T13260 CDHI10 118733086 IC50 > 10000 nM T13260 C18PWB 118733087 IC50 > 10000 nM T13260 C8WJ2Y 118733088 IC50 > 10000 nM T13260 C31ZXP 118733089 IC50 > 10000 nM T13260 CHR84E 118733090 IC50 > 10000 nM T13260 CAQ72M 118733091 IC50 > 10000 nM T13260 CIV1Z5 118733092 IC50 > 10000 nM T13260 CU3Y9W 118733093 IC50 > 10000 nM T13260 CF49NU 118733094 IC50 > 10000 nM T13260 CK73VU 118733095 IC50 > 10000 nM T13260 CR1WU5 118733096 IC50 > 10000 nM T13260 C5C4FZ 118735165 IC50 = 447 nM T13260 C1ZLM6 118735166 IC50 = 146 nM T13260 CQXM57 118735167 IC50 = 75 nM T13260 C0RYM4 118735168 IC50 = 137 nM T13260 C0DCB9 118735169 IC50 = 2425 nM T13260 CG4QF3 118735170 IC50 = 1894 nM T13260 CD3IY5 118735171 IC50 = 4993 nM T13260 C2VJU4 118735179 IC50 = 2090 nM T13260 CXWH51 118735180 IC50 = 165 nM T13260 C3YUS9 118735181 IC50 = 1546 nM T13260 CZET62 118735186 IC50 = 128 nM T13260 CZ8U2C 118735187 IC50 = 157 nM T13260 COJ81W 118735362 IC50 = 1020 nM T13260 C8VFT2 118735363 IC50 = 1320 nM T13260 CZE92I 118735364 IC50 = 53.1 nM T13260 CFB1G7 118735365 IC50 = 48.1 nM T13260 CX4V1E 118735366 IC50 = 6290 nM T13260 CW60ZD 118735367 IC50 = 337 nM T13260 C6ULM1 118735368 IC50 = 143 nM T13260 CE50LC 118735369 IC50 = 261 nM T13260 CMCW85 118735370 IC50 = 328 nM T13260 C6Y2NQ 118735371 IC50 = 1930 nM T13260 CVEQ39 118735372 IC50 = 48.9 nM T13260 C4LK0C 118735373 IC50 = 16.9 nM T13260 C93CNO 118735374 IC50 = 174 nM T13260 C4YR6E 118735375 IC50 = 715 nM T13260 CS3ZJ8 118735376 IC50 = 699 nM T13260 CV83KA 118735377 IC50 = 493 nM T13260 C0BP6M 118735378 IC50 = 30500 nM T13260 CG9RB4 118735379 IC50 = 1240 nM T13260 CGT60X 118735380 IC50 = 7340 nM T13260 CY6L8W 118735381 IC50 = 491 nM T13260 C3NB6I 122181247 IC50 = 12500 nM T13260 CYCG69 122181248 IC50 = 200 nM T13260 CME27L 122181249 IC50 = 1800 nM T13260 C0KHC3 122191579 IC50 = 0.26 nM T13260 CO7E3N 122191580 IC50 = 0.42 nM T13260 CML6C5 122191581 IC50 = 5.2 nM T13260 CYC63O 122191582 IC50 = 2.7 nM T13260 CP7S0B 122191583 IC50 = 2.3 nM T13260 C61IRT 122191584 IC50 = 4 nM T13260 CYJ32S 122191585 IC50 = 2.3 nM T13260 CAQ5S2 122191586 IC50 = 3.5 nM T13260 C03SBU 122191587 IC50 = 4.2 nM T13260 CLG6J4 122191588 IC50 = 5 nM T13260 CI42KY 122191589 IC50 = 20.7 nM T13260 C9GQP6 122191591 IC50 = 3.4 nM T13260 C0WN2U 122191592 IC50 = 5.5 nM T13260 C0WI6K 122191772 IC50 = 29 nM T13260 C5C2EM 122192355 IC50 = 250 nM T13260 C4HIF8 122192356 IC50 = 220 nM T13260 C0SJU6 122192359 IC50 = 100 nM T13260 C3T9CZ 122192360 IC50 = 41 nM T13260 C58OCL 122192361 IC50 = 0.1 nM T13260 C15NCI 122439267 IC50 = 10000 nM T13260 CX4T7L 122439274 IC50 = 10000 nM T13260 C3YG1J 122443028 IC50 > 19952.62 nM T13260 CW3K8X 122462796 IC50 > 19952.62 nM T13260 C80OLS 122462854 IC50 > 31622.78 nM T13260 CR4YC2 124012328 Ki = 38 nM T13260 C10TQU 124351848 Ki = 1 nM T13260 CCX94N 124351849 Ki = 75 nM T13260 C36AXJ 127025738 Ki = 100 nM T13260 CM2NC0 127025739 Ki = 100 nM T13260 CW5AZ0 127025740 Ki = 100 nM T13260 CY9Q8T 127025741 Ki = 100 nM T13260 C0X8HP 127026020 Ki = 24.1 nM T13260 C4LWG3 127026653 IC50 = 120500 nM T13260 C3ZQ5Y 127026654 IC50 = 1889 nM T13260 CZDU19 127026655 IC50 = 18570 nM T13260 CIT8S3 127026966 IC50 = 1820 nM T13260 CJTB10 127026967 IC50 = 1820 nM T13260 C2ZFR8 127027572 IC50 = 7900 nM T13260 CV1BD6 127027573 IC50 = 3100 nM T13260 C1L9TB 127027959 IC50 = 26000 nM T13260 CPX6K3 127028274 Ki = 100 nM T13260 CQO36B 127028499 IC50 = 5000 nM T13260 CCR07G 127028593 IC50 = 1820 nM T13260 CH6PU4 127028608 Ki = 100 nM T13260 C9WIB4 127028609 Ki = 100 nM T13260 CN42BR 127028817 IC50 > 10000 nM T13260 CIE4Q7 127028911 IC50 = 1820 nM T13260 C49IME 127031799 IC50 = 6100 nM T13260 CGEO60 127035149 IC50 = 245 nM T13260 CJ30BZ 127035150 IC50 = 236 nM T13260 C3MN9I 127035661 Ki = 5 nM T13260 CX3TB1 127035807 Ki = 5 nM T13260 CE6T8A 127035808 Ki = 5 nM T13260 C7JNM3 127036045 Ki = 75000 nM T13260 CS72ZI 127036174 Ki = 100 nM T13260 C9AFT8 127036253 IC50 = 6400 nM T13260 CQS2U0 127036843 IC50 = 2800 nM T13260 C7SM8Y 127037253 Ki = 31 nM T13260 CW08IP 127037254 IC50 = 1700 nM T13260 CXWJ74 127037557 Ki = 36 nM T13260 CK5N0X 127037559 Ki = 10000 nM T13260 CMQD16 127037560 Ki = 10000 nM T13260 CI6S7D 127037561 Ki = 10000 nM T13260 CTE51A 127047976 IC50 = 110 nM T13260 C1IBC5 127048009 IC50 = 530 nM T13260 CWE96C 127048149 IC50 = 12310 nM T13260 CDX0L1 127048499 IC50 = 51 nM T13260 CWD0J9 127048833 IC50 = 7 nM T13260 C9OEW2 127048838 IC50 = 46 nM T13260 CCJ3F0 127048839 IC50 = 6 nM T13260 CQ10PX 127048840 IC50 = 42 nM T13260 CWAH54 127048841 IC50 = 48 nM T13260 CD2O0K 127049168 IC50 = 129 nM T13260 C7ZHU6 127049169 IC50 = 48 nM T13260 CQN95D 127049828 IC50 = 36 nM T13260 C20LNJ 127050749 IC50 = 43 nM T13260 CH6E4C 127050950 IC50 = 168 nM T13260 CQ8PA9 127050951 IC50 = 512 nM T13260 C4Q6RA 127050952 IC50 = 800 nM T13260 C92CDW 127051351 IC50 = 14 nM T13260 CCR94D 127051352 IC50 = 13 nM T13260 CPL7A6 127051353 IC50 = 54 nM T13260 C7T2JR 127051680 IC50 = 339 nM T13260 CEJ1B8 127051681 IC50 = 131 nM T13260 CW3B0L 127051682 IC50 = 79 nM T13260 CE04JD 127052583 IC50 = 16 nM T13260 C48EUT 127052584 IC50 = 45 nM T13260 CT73HY 127052585 IC50 = 21 nM T13260 CL4ZK7 127052586 IC50 = 59 nM T13260 C1EI2R 127052880 IC50 = 22 nM T13260 CU9FI0 127052881 IC50 = 14 nM T13260 C01SHM 127052902 IC50 = 53 nM T13260 C09AZE 127052903 IC50 = 24 nM T13260 CH85FP 127052904 IC50 = 14 nM T13260 CYVM52 127052905 IC50 = 9 nM T13260 C12WOQ 129137247 IC50 = 62.2 nM T13260 C4O3QV 129137260 IC50 = 177.1 nM T13260 CJB4M3 129137266 IC50 = 230 nM T13260 CWVE96 129137276 IC50 = 13.4 nM T13260 CJ1N2M 129137280 IC50 = 220.8 nM T13260 CH42QX 129137285 IC50 = 8.8 nM T13260 CEH4N6 129750903 IC50 = 2600 nM T13260 CD7BX2 132601756 IC50 = 57.54 nM T13260 C5XSM4 132601757 IC50 = 12.11 nM T13260 CC2X1M 132601758 IC50 = 9.016 nM T13260 C8U1VZ 132601759 IC50 = 17.38 nM T13260 CH3V9Q 134139925 IC50 = 7700 nM T13260 CZV71F 134140768 IC50 = 6070 nM T13260 CVS3Q5 134142034 IC50 = 9724 nM T13260 CK4GS1 134142054 IC50 = 4660 nM T13260 C4B3MJ 134142750 IC50 = 9520 nM T13260 C2PT7N 134146686 IC50 = 12530 nM T13260 CK1BE9 134155077 IC50 = 286.9 nM T13260 C8QEA7 134155257 IC50 = 5089 nM T13260 C2BK3Z 134155779 IC50 = 645.3 nM T13260 C6G1CH 135185858 IC50 = 6445 nM T13260 CVR24H 135461648 IC50 = 29800 nM T13260 COWK61 135926058 IC50 > 50000 nM T13260 C7MP6W 135967555 Ki = 2548 nM T13260 CAV9U3 136219390 IC50 = 11.4 nM T13260 C59TUZ 136239410 IC50 > 10000 nM T13260 CH0O1B 136239411 IC50 > 10000 nM T13260 C52CVP 136239516 IC50 = 4152 nM T13260 CC7LY3 136239517 IC50 = 454 nM T13260 CSQR53 136239518 IC50 = 2112 nM T13260 C1N2WP 136244527 IC50 = 6195 nM T13260 C2V0IM 136244612 IC50 = 6 nM T13260 CLU5W1 136244613 IC50 = 922 nM T13260 C5LFY4 136245940 IC50 > 10000 nM T13260 CF07BL 136245941 IC50 > 10000 nM T13260 CYIF59 136245971 IC50 > 10000 nM T13260 CM6GS7 137632939 IC50 = 8900 nM T13260 CD7J1Z 137635610 IC50 = 5670 nM T13260 C4FYB7 137650013 IC50 = 9670 nM T13260 C2OC5D 137660208 IC50 = 6700 nM T13260 C3UK1Z 137660483 IC50 > 10000 nM T13260 C6VX2G 137662301 IC50 = 30.3 nM T13260 CEG7C9 140993853 IC50 = 1092.68 nM T13260 CY9QN0 145949171 IC50 = 2700 nM T13260 C0R6GF 145949298 IC50 = 237.6 nM T13260 C51BOX 145949540 IC50 = 700 nM T13260 C8T1HG 145949588 IC50 = 677.4 nM T13260 CBR4W8 145950208 IC50 = 2700 nM T13260 CVIW14 145950556 IC50 = 2800 nM T13260 C3L5IO 145950622 IC50 = 2300 nM T13260 C2EN9P 145950803 IC50 = 2500 nM T13260 CH80BF 145951156 IC50 = 32.3 nM T13260 CE8S3P 145951478 IC50 = 11900 nM T13260 CF2JT9 145951520 IC50 = 51.2 nM T13260 CD9G1O 145951806 IC50 = 2635 nM T13260 CL7V8M 145952266 IC50 = 11200 nM T13260 C9J0MP 145952426 IC50 = 1058 nM T13260 C4RX0H 145952545 IC50 = 276.8 nM T13260 CAD1R5 145953186 IC50 = 82.9 nM T13260 CGTW16 145953426 IC50 = 9800 nM T13260 C3PG4W 145953645 IC50 = 9800 nM T13260 CCF34U 145954042 IC50 = 8300 nM T13260 C8AR7H 145954077 IC50 = 5500 nM T13260 C5J7MO 145954302 IC50 = 4400 nM T13260 C6LU3T 145954433 IC50 = 7600 nM T13260 CRZ51Q 145954497 IC50 = 217.4 nM T13260 CEU5V2 145955100 IC50 = 4200 nM T13260 CGH62B 145955360 IC50 = 3900 nM T13260 CV49CR 145955375 IC50 = 11900 nM T13260 CYZ7R9 145955426 IC50 = 1400 nM T13260 C04FSJ 145955438 IC50 = 4600 nM T13260 CV5CZ7 145955551 IC50 = 207.5 nM T13260 CO3P9B 145955618 IC50 = 1300 nM T13260 CPS1E4 145956015 IC50 = 14.1 nM T13260 CCVP89 145956394 IC50 = 108.7 nM T13260 CR79QW 145956423 IC50 = 3400 nM T13260 CH8KZ4 145956588 IC50 = 260.8 nM T13260 CF4X3A 145956605 IC50 = 5400 nM T13260 CP65IV 145957520 IC50 = 8800 nM T13260 C7VQ6H 145958289 IC50 = 3500 nM T13260 CW8K2X 145958349 IC50 = 196.5 nM T13260 C8COZ7 145958369 IC50 = 4000 nM T13260 CC7UM6 145958531 IC50 = 36.1 nM T13260 C7TS3W 145958716 IC50 = 7772 nM T13260 C1FBC3 145958737 IC50 = 58.3 nM T13260 C0X5WO 145958928 IC50 = 96.9 nM T13260 C5IEV3 145958952 IC50 = 800 nM T13260 CTGM23 145959211 IC50 = 2300 nM T13260 CV1N0L 145959349 IC50 = 3800 nM T13260 C62HPO 145959622 IC50 = 2800 nM T13260 C4NYX7 145959688 IC50 = 210.6 nM T13260 CCW9R3 145959703 IC50 = 4100 nM T13260 C90VNG 145960023 IC50 = 3200 nM T13260 C7HA8N 145960331 IC50 = 3500 nM T13260 CK71RV 145963932 IC50 > 31622.78 nM T13260 C79FGQ 145965325 IC50 > 31622.78 nM T13260 CI56TJ 145967693 IC50 = 935.46 nM T13260 CKWV62 145967722 IC50 = 3591.14 nM T13260 C7XT0Z 145967929 IC50 = 3482.15 nM T13260 CHA9G8 145967940 IC50 = 3045.68 nM T13260 C0HP1U 145968036 IC50 = 2600.71 nM T13260 C5BM1L 145968186 IC50 = 999.74 nM T13260 C8XB7E 145968768 IC50 = 3253.28 nM T13260 C4JM2H 145968847 IC50 = 5715.79 nM T13260 C74IZW 145969198 IC50 = 3187.68 nM T13260 CNV0K1 145969871 IC50 = 1181.36 nM T13260 C4MQL6 145970012 IC50 = 1984.4 nM T13260 CDZV35 145970043 IC50 = 176.82 nM T13260 CEKI13 145970456 IC50 = 3321.79 nM T13260 C2Q1CO 145970604 IC50 = 1804.56 nM T13260 CW7XA4 145970723 IC50 = 3565.19 nM T13260 CE6P4U 145971254 IC50 = 1700 nM T13260 CGBW36 145972890 IC50 = 15300 nM T13260 CR50XP 145974563 IC50 = 54.4 nM T13260 CTB32X 145987737 IC50 = 3000.88 nM T13260 CJQ23A 145988166 IC50 = 3345.23 nM T13260 CAS5W8 145988425 IC50 = 3409.25 nM T13260 CZBY26 145988625 IC50 = 1703.22 nM T13260 C8I5JY 155511774 IC50 = 3200 nM T13260 C8ZYW2 155512683 Ki = 100 nM T13260 CWL61G 155513859 IC50 = 2750 nM T13260 COUZ40 155515111 Ki = 8 nM T13260 CQ0RX1 155519734 IC50 = 3300 nM T13260 CN8R0W 155521581 IC50 = 405 nM T13260 CS79RV 155522275 Ki = 24 nM T13260 CX9CY6 155523438 Ki = 97 nM T13260 C42DVB 155524075 Ki = 450 nM T13260 C7DX4M 155524253 IC50 = 110 nM T13260 CZCD39 155524316 Ki = 180 nM T13260 CO73MH 155528129 IC50 = 175 nM T13260 C9KHR3 155528792 IC50 = 210 nM T13260 C3PKZ1 155531378 IC50 = 0.2 nM T13260 CE2F1S 155532984 Ki = 81 nM T13260 C65EOC 155533109 Ki = 74 nM T13260 C2YTO1 155533392 IC50 = 520 nM T13260 C57SRY 155539404 IC50 = 105 nM T13260 CA01UF 155542148 IC50 = 210 nM T13260 C05WZC 155544203 Ki = 79 nM T13260 C1CJ3W 155544206 IC50 = 43.55 nM T13260 CZ48QO 155544544 IC50 = 660 nM T13260 C8NOR7 155548567 IC50 = 39.77 nM T13260 CO2G9W 155552576 IC50 = 73.17 nM T13260 C5CKA6 155553716 IC50 = 90.73 nM T13260 CAK73M 155557092 IC50 = 430 nM T13260 CA2H5K 155557102 IC50 = 17.42 nM T13260 C04ZVY 155557805 IC50 > 12500 nM T13260 CAY1Z7 155558257 IC50 = 14.52 nM T13260 CH3N8S 155558347 IC50 = 280 nM T13260 CJX17H 155558789 Ki = 57 nM T13260 CO6W0R 155559106 Ki = 125 nM T13260 C47PER 155559543 IC50 = 19.66 nM T13260 CH3IK5 155559681 IC50 = 8720 nM T13260 C3SWX8 155559867 IC50 = 58.85 nM T13260 CXT67R 155559873 IC50 = 560 nM T13260 CQU6N2 155562191 Ki = 290 nM T13260 C20AJK 155564333 IC50 = 55 nM T13260 CZ1OQ8 155569008 IC50 = 30.19 nM T13260 CH20CY 3114838 IC50 = 441 nM T13260 D00BVP 11847320 IC50 = 79.43 nM T13260 D00EMF 3644637 IC50 > 100000 nM T13260 D00HVZ 5271544 IC50 = 1860 nM T13260 D00RIX 5280443 IC50 = 1000 nM T13260 D00TWK 185914 IC50 > 50000 nM T13260 D00VUO 6539777 IC50 = 6360 nM T13260 D00ZPJ 408350 Ki = 25.5 nM T13260 D01IJX 10537337 IC50 = 3560 nM T13260 D01JZO 2779191 IC50 = 70 nM T13260 D01KKU 5281894 IC50 = 30.5 nM T13260 D01LOU 2238 IC50 = 40 nM T13260 D01MPK 12331302 Ki = 1750 nM T13260 D01REI 46901610 IC50 = 2440 nM T13260 D01SUE 6539759 IC50 = 2040 nM T13260 D01SZX 46867545 IC50 = 150 nM T13260 D01UYI 5281607 IC50 = 1 nM T13260 D02ALK 11514074 IC50 = 2700 nM T13260 D02BGR 9949648 IC50 = 13000 nM T13260 D02BWQ 6539818 IC50 = 2800 nM T13260 D02BXS 46901445 IC50 = 24560 nM T13260 D02CSU 6539786 IC50 = 12735030.81 nM T13260 D02LTV 10019821 IC50 = 110 nM T13260 D02LWB 6540046 IC50 > 36000 nM T13260 D02NAG 6539765 IC50 = 4260 nM T13260 D02QSH 339914 Ki = 1.9 nM T13260 D02SIT 9926623 IC50 = 74 nM T13260 D02XHH 6540043 IC50 = 100 nM T13260 D02XTS 6539811 IC50 = 3630 nM T13260 D03EXD 49864181 IC50 = 3070 nM T13260 D03FBI 49798900 IC50 = 8510 nM T13260 D03KLN 11413434 IC50 = 129 nM T13260 D03LOG 5280450 IC50 = 48000 nM T13260 D03MKT 6539788 IC50 = 1550 nM T13260 D03TRM 6540032 IC50 = 955 nM T13260 D03VRC 2989557 IC50 = 338.84 nM T13260 D04CLL 6539775 IC50 = 4720 nM T13260 D04DZZ 11646165 IC50 = 910 nM T13260 D04ELJ 6539766 IC50 = 4050 nM T13260 D04HVL 364705 IC50 = 2790 nM T13260 D04IBH 11616637 IC50 = 9107 nM T13260 D04IJE 256445 IC50 = 2741574.17 nM T13260 D04ISG 11680597 IC50 > 2000 nM T13260 D04LWL 97252 IC50 > 115600 nM T13260 D04QPK 6539783 IC50 = 1810 nM T13260 D04REX 6539808 IC50 = 790 nM T13260 D04TBB 10354739 IC50 = 2 nM T13260 D04VRY 11847169 IC50 = 467.74 nM T13260 D04WJN 10588478 IC50 = 389.05 nM T13260 D04ZGF 10561174 IC50 = 500 nM T13260 D05FFY 14231155 IC50 = 15 nM T13260 D05HBF 5353357 IC50 = 8.7 nM T13260 D05HRP 13596072 Ki = 800 nM T13260 D05IWY 5464078 IC50 = 4970 nM T13260 D05MQE 6539785 IC50 = 230 nM T13260 D05PXK 11847171 IC50 = 1800 nM T13260 D05QPR 12229388 IC50 = 880 nM T13260 D05YCI 42618032 IC50 = 18470 nM T13260 D05YJR 5495926 IC50 = 5200 nM T13260 D05YNW 6539790 IC50 = 6700 nM T13260 D05ZPO 1890 IC50 = 3800 nM T13260 D06AZC 135494055 IC50 = 1400 nM T13260 D06DDT 5315502 IC50 = 30000 nM T13260 D06FHE 44341253 IC50 = 205 nM T13260 D06GIV 337660 IC50 = 3100 nM T13260 D06HFV 6539805 IC50 = 7447319.74 nM T13260 D06HJB 14355826 IC50 = 55 nM T13260 D06PRC 5281650 IC50 = 20700 nM T13260 D06UQR 15306616 IC50 = 14800 nM T13260 D06WPP 11847170 IC50 = 4073.8 nM T13260 D07CTI 10853186 IC50 = 977.24 nM T13260 D07FGX 6116651 IC50 = 3300 nM T13260 D07IQG 10473365 IC50 = 933.25 nM T13260 D07JKK 11760063 IC50 = 1 nM T13260 D07LUJ 64945 IC50 = 14 ug.mL-1 T13260 D07PHT 324288 Ki = 6.5 nM T13260 D07PHV 10546089 IC50 = 89 nM T13260 D07PYC 6539760 IC50 = 3550 nM T13260 D07SOM 11847316 IC50 = 71 nM T13260 D07TIJ 3828439 IC50 = 2818.38 nM T13260 D07TUX 11230598 IC50 = 31622.78 nM T13260 D07UVN 6440384 IC50 = 3080 nM T13260 D07ZCD 6539804 IC50 = 1710 nM T13260 D07ZYL 6539797 IC50 = 3720 nM T13260 D08ARY 339906 Ki = 5.6 nM T13260 D08AZK 6539767 IC50 = 7830 nM T13260 D08EZA 11847317 IC50 = 45 nM T13260 D08FAB 11845485 IC50 > 2000 nM T13260 D08FHU 42618033 IC50 = 2720 nM T13260 D08FOJ 9898204 IC50 = 4300 nM T13260 D08HPU 6540052 IC50 = 1787 nM T13260 D08IIW 46887422 IC50 = 40 nM T13260 D08ISK 42618030 IC50 > 91290 nM T13260 D08KLN 13580711 IC50 = 3210 nM T13260 D08PKR 10845522 IC50 = 3060 nM T13260 D08PNF 6539770 IC50 = 5570 nM T13260 D08TKB 46889432 IC50 = 389.2 nM T13260 D08UQH 53600 IC50 = 190 nM T13260 D08ZTZ 11529133 IC50 = 1805 nM T13260 D09CPC 13728862 IC50 > 5000 nM T13260 D09DRS 42618031 IC50 = 960 nM T13260 D09HEA 1236449 IC50 = 1096.48 nM T13260 D09HGK 6539796 IC50 = 3960 nM T13260 D09HOE 6539789 IC50 = 800 nM T13260 D09HQH 13308 Ki = 260 nM T13260 D09MQF 15696376 IC50 = 900 nM T13260 D09MYQ 261365 Ki = 266 nM T13260 D09OPA 44593508 IC50 = 3400 nM T13260 D09QDY 6540033 IC50 = 130 nM T13260 D09TUB 11099375 IC50 > 308300 nM T13260 D09VPA 6539794 IC50 = 3400 nM T13260 D09VQM 442428 IC50 = 5000 nM T13260 D09XKH 10356745 IC50 = 2200 nM T13260 D09YXV 6539769 IC50 = 4310 nM T13260 D09ZHX 11847318 IC50 = 436.52 nM T13260 D09ZIW 10143276 IC50 = 7100 nM T13260 D0A0JL 2052 IC50 = 70600 nM T13260 D0A2FO 2825024 IC50 = 8000 nM T13260 D0A2GB 13660221 IC50 = 1300 nM T13260 D0A4EA 445639 IC50 = 32700 nM T13260 D0A4XA 25093379 IC50 > 50000 nM T13260 D0A7PA 49799639 IC50 = 11140 nM T13260 D0AH1B 6539782 IC50 = 12618275.35 nM T13260 D0AM2Z 13660216 IC50 = 11000 nM T13260 D0AW7Q 46867544 IC50 = 7900 nM T13260 D0AY4E 6539780 IC50 = 3930 nM T13260 D0B5MZ 13660218 IC50 = 2300 nM T13260 D0B8PE 10355761 IC50 = 3500 nM T13260 D0BH2T 10107266 IC50 > 40 ug.mL-1 T13260 D0C3XU 46887018 IC50 = 7 nM T13260 D0C5SV 5280934 IC50 = 44200 nM T13260 D0C5ZP 16125122 IC50 = 2140 nM T13260 D0C8EO 6539806 IC50 = 4330 nM T13260 D0C8KC 1504717 IC50 = 960 nM T13260 D0CR6B 11847319 IC50 = 69 nM T13260 D0D0DR 10081625 IC50 = 310 nM T13260 D0D7GG 510040 IC50 = 950 nM T13260 D0D8GU 6539803 IC50 = 1280 nM T13260 D0D8YE 6540048 IC50 = 5700 nM T13260 D0D9FR 6539795 IC50 = 3962780.34 nM T13260 D0DJ3R 10585323 IC50 = 100 nM T13260 D0DO1T 9819080 Ki = 10.3 nM T13260 D0DY5G 443389 IC50 > 100000 nM T13260 D0E2RV 360578 IC50 = 1700 nM T13260 D0E3IK 11680642 IC50 = 2510 nM T13260 D0E5FV 5318585 IC50 = 100 nM T13260 D0E9WX 6540042 IC50 = 27 nM T13260 D0F4MF 49799640 IC50 = 980 nM T13260 D0F4WQ 46867547 IC50 = 5.59 nM T13260 D0F5AC 46867542 IC50 = 17 nM T13260 D0F5YU 6539793 IC50 = 1990 nM T13260 D0F8IB 25256842 IC50 = 16500 nM T13260 D0F9MQ 11493409 IC50 = 2670 nM T13260 D0G2JV 49799657 IC50 = 2280 nM T13260 D0G6QL 23644748 IC50 = 2800 nM T13260 D0GL0L 11232117 IC50 = 3981.07 nM T13260 D0H1LK 161760 IC50 = 10200 nM T13260 D0HC9U 46867416 IC50 = 53 nM T13260 D0HD9P 444899 IC50 = 28200 nM T13260 D0HR9S 388623 Ki = 15.1 nM T13260 D0I1SI 49799655 IC50 = 760 nM T13260 D0I1YH 46901446 IC50 = 663 nM T13260 D0I2UE 46867543 IC50 = 3.98 nM T13260 D0I5NW 6540047 IC50 = 4073 nM T13260 D0I5PY 23585406 IC50 = 210 nM T13260 D0I7GE 11790 Ki = 20 nM T13260 D0J2WW 6539801 IC50 = 770 nM T13260 D0J3PK 11779089 IC50 = 41 nM T13260 D0J4VR 46191176 IC50 = 5000 nM T13260 D0J8FS 5377857 IC50 = 8330 nM T13260 D0JE1I 9815923 IC50 = 680 nM T13260 D0K2SE 10703161 IC50 = 6400 nM T13260 D0K3CE 6539800 IC50 = 280 nM T13260 D0K4PY 114829 IC50 = 2100 nM T13260 D0K5GG 49799652 IC50 = 3570 nM T13260 D0K5JU 46867417 IC50 = 1900 nM T13260 D0K5KG 6540050 IC50 = 6045 nM T13260 D0K8QD 63059 IC50 = 24880 nM T13260 D0L1JF 6539791 IC50 = 180 nM T13260 D0L3AJ 5324988 IC50 = 2020 nM T13260 D0L9BT 10823163 IC50 = 3700 nM T13260 D0M0FE 3317166 IC50 = 160 nM T13260 D0M2IB 9904788 Ki = 4 nM T13260 D0M4CX 356713 Ki = 385 nM T13260 D0M5EW 11276192 IC50 = 2089.3 nM T13260 D0M7FS 6539764 IC50 = 2490 nM T13260 D0M8RO 6128 Ki = 20 nM T13260 D0MA9G 6540051 IC50 = 1507 nM T13260 D0N1GH 11601068 IC50 > 36000 nM T13260 D0N1PQ 11506923 IC50 = 586 nM T13260 D0N5GZ 12229395 IC50 = 24500 nM T13260 D0N7QV 11819989 IC50 = 0.7 nM T13260 D0N9PY 6539773 IC50 = 7080 nM T13260 D0NB8V 49799650 IC50 = 16420 nM T13260 D0NH6T 14218027 IC50 = 400 nM T13260 D0NX0M 6540049 IC50 = 814 nM T13260 D0O0BL 44394887 IC50 = 430 nM T13260 D0O1ZM 13660225 IC50 = 1500 nM T13260 D0O4YS 42618026 IC50 > 98490 nM T13260 D0O6ZM 14256024 IC50 = 670 nM T13260 D0OY1J 11401873 IC50 = 676.08 nM T13260 D0P3ND 46887506 IC50 = 160 nM T13260 D0P5ZV 261861 IC50 = 9800 nM T13260 D0PU5V 10750911 IC50 = 1380 nM T13260 D0Q0BK 46901611 IC50 = 1670 nM T13260 D0Q3JZ 6539774 IC50 = 7680 nM T13260 D0Q6XB 5844100 IC50 = 7470 nM T13260 D0Q8UZ 18785180 IC50 = 590 nM T13260 D0QL1V 508445 IC50 = 1200 nM T13260 D0R0TE 11557864 IC50 = 6638 nM T13260 D0R2YN 5994480 IC50 = 15500 nM T13260 D0R4FM 122850 IC50 > 40 ug.mL-1 T13260 D0R4WW 44265823 Ki = 10.3 nM T13260 D0RJ6S 11558270 IC50 > 36000 nM T13260 D0S0EP 585819 IC50 = 28.18 nM T13260 D0S0OV 10267149 IC50 = 91 nM T13260 D0S0RK 10680 IC50 = 8 nM T13260 D0S1AY 269167 IC50 = 26800 nM T13260 D0S7VY 49798801 IC50 = 2940 nM T13260 D0S8MJ 337743 IC50 = 2100 nM T13260 D0S9YX 5280373 IC50 = 10.2 nM T13260 D0SY2M 5281708 Ki = 100000 nM T13260 D0SY6C 5282073 IC50 = 2 nM T13260 D0T0CK 49799648 IC50 = 14510 nM T13260 D0T3ED 44580826 Ki = 33.4 nM T13260 D0T3PW 5281672 IC50 = 10000 nM T13260 D0T5NO 15306617 IC50 = 100 nM T13260 D0TM4K 6539817 IC50 = 3680 nM T13260 D0U4BB 10748 IC50 > 10000 nM T13260 D0U6IT 6539807 IC50 = 4830 nM T13260 D0U6NJ 11311402 IC50 = 758.58 nM T13260 D0U7RR 6539768 IC50 = 7370 nM T13260 D0U8JC 9862769 IC50 = 4600 nM T13260 D0U9QB 73440 IC50 = 15 nM T13260 D0UI8Q 10566470 IC50 = 2089.3 nM T13260 D0V0DB 46887421 IC50 = 20 nM T13260 D0V1UY 133966 IC50 = 3 nM T13260 D0V3MV 46867546 IC50 = 11.45 nM T13260 D0V3YH 6539784 IC50 = 130 nM T13260 D0V8CR 6539763 IC50 = 2540 nM T13260 D0V8SM 10659706 IC50 = 1096.48 nM T13260 D0W3LG 9866908 IC50 = 9700 nM T13260 D0W3LM 10265122 IC50 = 3700 nM T13260 D0W4IB 23644623 Ki = 680 nM T13260 D0W7GU 5377410 IC50 = 1820 nM T13260 D0W7JA 5273567 IC50 = 35300 nM T13260 D0W9PF 13472 Ki = 43 nM T13260 D0W9ZC 46867540 IC50 = 16.5 nM T13260 D0WK9Q 14256034 IC50 = 2760 nM T13260 D0WN9P 46901444 IC50 = 2830 nM T13260 D0X0IH 77918 IC50 = 150 nM T13260 D0X1QS 6540053 IC50 = 3551 nM T13260 D0X8UK 10751574 IC50 = 350 nM T13260 D0XQ6T 42618029 IC50 = 5760 nM T13260 D0XS6T 53602 IC50 = 1840 nM T13260 D0Y0CT 6539819 IC50 = 4060 nM T13260 D0Y0EK 620596 IC50 = 3400 nM T13260 D0Y0QI 10774864 IC50 = 170 nM T13260 D0Y4TE 340000 Ki = 13.1 nM T13260 D0Y5KX 46901443 IC50 = 24500 nM T13260 D0Y7HG 5281616 Ki = 100000 nM T13260 D0Y7RB 6539781 IC50 = 4600 nM T13260 D0Y8XJ 5497182 IC50 = 16800 nM T13260 D0Y9HD 361928 Ki = 52.7 nM T13260 D0YD9J 6539792 IC50 = 5432503.31 nM T13260 D0YS2F 6539776 IC50 = 9740 nM T13260 D0Z1OI 124662 Ki = 1000 nM T13260 D0Z4GR 4594970 IC50 = 100 nM T13260 D0Z7EL 5280647 IC50 = 11000 nM T93509 D00MXN 25019940 Ki = 0.024 nM T93509 D0G5ME 11319053 Ki = 0.78 nM T93509 D0L5GH 6918509 Ki = 0.014 nM T93509 CXZA43 457930 Ki = 7300 nM T93509 C6W7AM 9847811 Ki = 2700 nM T93509 CANV26 10030220 Ki = 710 nM T93509 CH2NR6 11178760 Ki = 1700 nM T93509 C1LX9V 11397043 Ki = 1800 nM T93509 C8GB7A 11419496 Ki = 1900 nM T93509 CQT6I4 16728074 Ki = 16000 nM T93509 C5RC3J 44563430 IC50 >= 1000 nM T93509 C2BKH7 44563440 EC50 = 0.05 nM T93509 CQ1VU2 57392038 Ki = 26000 nM T93509 CF8R4H 57392039 Ki > 100000 nM T93509 C9T7IA 57393753 Ki = 8000 nM T93509 C6UID4 57393754 Ki = 5200 nM T93509 C1O0EL 57393755 Ki > 100000 nM T93509 C6B2JK 57395477 Ki = 14000 nM T93509 CD91MC 57395478 Ki = 45000 nM T93509 CV87FO 57397325 Ki > 100000 nM T93509 CK6L0F 57400721 Ki = 8 nM T93509 C6GF8M 57402496 Ki > 100000 nM T93509 CL85VH 57402497 IC50 > 10000 nM T93509 CPYG07 73345650 IC50 = 0.85 nM T93509 CH9LP4 73345651 IC50 = 3.45 nM T93509 CJ2V8U 73347156 IC50 = 29.73 nM T93509 C4DWG3 73347157 IC50 = 79.34 nM T93509 C8F9IO 73353230 IC50 = 4.15 nM T93509 CC5Q0Y 73354735 Ki = 0.73 nM T93509 CH7GY0 73354736 Ki = 3.3 nM T93509 C3LV6M 73356281 IC50 = 1.31 nM T93509 C3WJM4 127026899 IC50 = 130 nM T93509 CAJ24S 127026900 IC50 = 13 nM T93509 C7ZF6X 127026901 IC50 = 170 nM T93509 C6TRP3 127027478 IC50 = 15 nM T93509 C63EQW 127027479 IC50 = 19 nM T93509 C5VS7T 127027480 IC50 = 77 nM T93509 C26QAE 127027481 IC50 = 12 nM T93509 C9TR7O 127027482 IC50 = 22 nM T93509 C8DPY7 127027501 IC50 = 190 nM T93509 C1MW5C 127027502 IC50 = 460 nM T93509 CEK1B2 127027503 IC50 = 9.8 nM T93509 C9N5SC 127027797 IC50 = 44 nM T93509 C23NCY 127027803 IC50 = 33 nM T93509 C6JT4M 127027804 IC50 = 130 nM T93509 CXNT13 127027805 IC50 = 130 nM T93509 CI4Z3K 127027806 IC50 = 8.9 nM T93509 CZD67W 127027807 IC50 = 99 nM T93509 CR8GD0 127027810 IC50 = 110 nM T93509 CJH92D 127027811 IC50 = 44 nM T93509 C1BFU9 127027812 IC50 = 120 nM T93509 C0JIC7 127027814 IC50 = 350 nM T93509 CWS56B 127027815 IC50 = 4.3 nM T93509 CH0S6M 127027816 IC50 = 12 nM T93509 CQ3CR8 127027821 IC50 = 140 nM T93509 C0UGB6 127027822 IC50 = 97 nM T93509 CQ56CX 127027823 IC50 = 150 nM T93509 CT95NM 127027824 IC50 = 41 nM T93509 C3IJR5 127028113 IC50 = 46 nM T93509 CBJ5A4 127028116 IC50 = 7 nM T93509 C8SCZ7 127028121 IC50 = 34 nM T93509 CW1D3C 127028122 IC50 = 2.9 nM T93509 CDU86M 127028128 IC50 = 14 nM T93509 C1VEB4 127028129 IC50 = 0.23 nM T93509 CD70TW 127028130 IC50 = 0.11 nM T93509 C86NMZ 127028438 IC50 = 170 nM T93509 CHO8T2 127028443 IC50 = 92 nM T93509 C4Z1ND 127028444 IC50 = 120 nM T93509 CHM0F8 127028769 IC50 = 240 nM T93509 CM25XZ 127028770 IC50 = 54 nM T93509 C4NR9D 127028771 IC50 = 1.1 nM T93509 CTO2K3 127028772 IC50 = 19 nM T93509 CJ4IZ2 127028773 IC50 = 16 nM T93509 CPE3B1 127028774 IC50 = 24 nM T93509 CQ9R3C 127028775 IC50 = 430 nM T93509 D05LMD 16134896 Ki = 3.19 nM T93509 D0I2KW 44406785 IC50 = 740 nM T93509 D0U4BO 44563409 IC50 = 0.64 nM T08446 D0ED7U 60648 IC50 = 1670000 nM T08446 D08ESA 198693 IC50 = 300000 nM T08446 D0C9XA 119 IC50 = 2000 nM T08446 CJ9V4G 40598 IC50 = 290000 nM T08446 CXSD61 155246 IC50 = 3000 nM T08446 CHV0G9 639062 IC50 > 1000000 nM T08446 C97FYX 702501 IC50 = 100000 nM T08446 C8X9TQ 1069892 IC50 = 2884.03 nM T08446 C1A0UL 1502074 IC50 = 7943.28 nM T08446 C3DR8J 1502075 IC50 = 3981.07 nM T08446 C9EI4M 1530639 IC50 > 1000000 nM T08446 CU23IC 4531494 IC50 = 208000 nM T08446 CG1ZF6 5311322 Ki = 1600 nM T08446 CN2C7Q 6604883 IC50 = 630000 nM T08446 C4A6SU 8181355 IC50 = 180000 nM T08446 CQ64IH 9797818 IC50 = 7210000 nM T08446 C31HNE 9884272 Ki = 42000 nM T08446 CY2IS7 9888224 IC50 = 39000 nM T08446 CTZ5Q7 9983570 IC50 = 2660000 nM T08446 C75BDY 10031163 IC50 = 201000 nM T08446 CZ4PO2 10050339 IC50 = 1270000 nM T08446 CP2WF1 10072112 IC50 = 27000 nM T08446 CG1A4H 10073933 IC50 = 151000 nM T08446 C4S1CO 10096504 IC50 = 382000 nM T08446 C0XI3N 10252046 IC50 = 920000 nM T08446 CXJR61 10252950 IC50 = 655000 nM T08446 CC8V4E 10412575 IC50 = 109000 nM T08446 CZ8FQ2 10481573 IC50 = 88000 nM T08446 CU40KP 11743493 IC50 = 435000 nM T08446 CH6GX1 13314232 IC50 = 91000 nM T08446 C6VK4E 17173775 IC50 > 1000000 nM T08446 CE92MX 17174058 IC50 > 1000000 nM T08446 C3OQD7 17250318 IC50 = 170000 nM T08446 CME93B 43345728 IC50 > 1000000 nM T08446 C5JUW9 47058964 IC50 > 1000000 nM T08446 CLIK30 50941729 IC50 > 100000 nM T08446 CQ4XJ7 55285849 IC50 = 5480 nM T08446 CY9O8W 55285850 IC50 = 5480 nM T08446 C8UTR2 67642717 IC50 = 7300 nM T08446 C6ME5H 70684991 IC50 = 335000 nM T08446 C79CYX 70689234 IC50 = 2900000 nM T08446 CD9EV5 70691307 IC50 = 809000 nM T08446 CJ7P8C 70691309 IC50 = 436000 nM T08446 C53QGB 118711599 IC50 = 590 nM T08446 CO18BS 137635197 IC50 = 8000 nM T08446 CQL64H 137637846 IC50 > 1000000 nM T08446 CZ73DV 137638595 IC50 > 100000 nM T08446 CARI53 137638617 IC50 > 100000 nM T08446 CUM2T0 137638836 IC50 > 100000 nM T08446 C3PY5G 137638838 IC50 > 50000 nM T08446 CP7OV5 137639241 IC50 > 100000 nM T08446 C21IZT 137639281 IC50 > 1000000 nM T08446 CP24OX 137642163 IC50 > 100000 nM T08446 CK2VU3 137650102 IC50 > 1000000 nM T08446 C52PYO 137650910 IC50 > 1000000 nM T08446 CS6FX4 137651374 IC50 > 1000000 nM T08446 CPLJ94 137651669 IC50 > 1000000 nM T08446 CN04QK 137652511 IC50 > 1000000 nM T08446 CGC1Z4 137654858 IC50 > 50000 nM T08446 CADN74 137657292 IC50 > 100000 nM T08446 C4NK1W 137658990 IC50 > 50000 nM T08446 CPI4S8 137659917 IC50 > 50000 nM T08446 CI7S8H 155516242 IC50 > 100000 nM T08446 C4U8QT 155524561 IC50 > 100000 nM T08446 CJ4OV6 155530359 IC50 > 100000 nM T08446 C4RL9X 155535776 IC50 > 100000 nM T08446 CL2Q6G 155567178 IC50 > 100000 nM T08446 D02ANG 5216267 IC50 = 47400 nM T08446 D03IWW 6575389 IC50 = 6410000 nM T08446 D08YGM 92409 IC50 = 7210000 nM T08446 D0D2EF 1796510 IC50 = 2310000 nM T08446 D0H7WK 10458835 IC50 = 71700 nM T08446 D0P3KI 9888030 IC50 = 5100 nM T08446 D0RF2M 4498 IC50 = 2370000 nM T08446 D0V5OY 16725912 Ki = 15000 nM T08446 D0V7RG 3532 IC50 = 1870000 nM T97537 CQ5T2C 2837573 Ki = 7700 nM T97537 CIBH72 3834735 Ki > 100000 nM T97537 CA1ZC4 4188970 Ki = 5000 nM T97537 C4EBQ6 8823441 IC50 = 1100 nM T97537 CT45FK 24828324 Ki = 147.91 nM T97537 C1WKD6 24828325 Ki = 20.42 nM T97537 CJ6RS7 24828326 Ki = 5754.4 nM T97537 C98VUW 24828598 Ki = 5370.32 nM T97537 CW64AC 24828600 Ki = 144.54 nM T97537 CFP01R 24828743 Ki = 100 nM T97537 C9LUM1 24828881 Ki = 27.54 nM T97537 CER36P 24828882 Ki = 2137.96 nM T97537 C0VL7B 24890303 Ki = 10715.19 nM T97537 CJ6G0Y 42601512 Ki = 480 nM T97537 CL2A3I 42610322 Ki = 20 nM T97537 C12CDQ 44254309 Ki = 3019.95 nM T97537 C8EI1G 44254310 Ki = 8511.38 nM T97537 CD3L0N 44254402 Ki = 794.33 nM T97537 CHT0Z1 44254404 Ki = 2454.71 nM T97537 CW7LB9 44254495 Ki = 2041.74 nM T97537 C5FDC2 44254496 Ki = 2951.21 nM T97537 CE40ON 44277843 Ki = 52 nM T97537 CID3S9 44450222 Ki = 177.83 nM T97537 CCJ39L 44450246 Ki = 1071.52 nM T97537 CX05EH 44450286 Ki = 173.78 nM T97537 C87BVH 44450320 Ki = 165.96 nM T97537 C98XEN 44450334 Ki = 1318.26 nM T97537 CD7UO5 44450345 Ki = 630.96 nM T97537 CH02ZM 44450376 Ki = 81.28 nM T97537 CD85RG 44450377 Ki = 109.65 nM T97537 CZ4H7R 44560401 Ki = 1200 nM T97537 C70AIZ 44560402 Ki = 12000 nM T97537 C63VWA 44560403 Ki = 7400 nM T97537 CRX2G5 44560404 Ki = 2500 nM T97537 CA4IF6 44560405 Ki = 1400 nM T97537 C57LTE 44560406 Ki = 3700 nM T97537 C2F3TI 44560407 Ki = 3100 nM T97537 CC3GY2 44560408 Ki = 1300 nM T97537 C9YE7J 44560409 Ki = 1300 nM T97537 C1OEW5 44560410 Ki = 1800 nM T97537 CU4G1S 44560411 Ki = 1000 nM T97537 C2Y0OT 44560412 Ki = 97000 nM T97537 CG7BQ8 44560457 Ki = 16000 nM T97537 C1RK3C 44560557 Ki = 35000 nM T97537 C42VEQ 44560558 Ki = 76000 nM T97537 CMLG10 46882676 Ki = 4786.3 nM T97537 CTO1Q8 46882677 Ki = 3981.07 nM T97537 CP9WB0 49840768 Ki = 282 nM T97537 C51YRX 49840770 Ki = 54.8 nM T97537 CJ3Z7V 49840772 Ki = 1752 nM T97537 CS3I8G 49840774 Ki = 3.3 nM T97537 C3IT5V 49840844 Ki = 242 nM T97537 CYBW37 49840846 Ki = 18.5 nM T97537 CFEC23 49840848 Ki = 93.7 nM T97537 C64XMG 49840850 Ki = 5.2 nM T97537 CNU1Q7 49840921 Ki = 34.9 nM T97537 CQ90FE 52941108 Ki = 5506 nM T97537 CU4HK1 52943524 Ki = 196 nM T97537 C9HRG4 52946764 Ki = 22.5 nM T97537 C89EGH 52947188 Ki = 9.3 nM T97537 CU58OG 53257413 Ki = 4.1 nM T97537 C6XY5R 53259047 Ki = 50 nM T97537 C7AXD8 53259048 Ki = 41.1 nM T97537 CX51OK 53259216 Ki = 697 nM T97537 CBS92H 53259217 Ki = 351 nM T97537 C8RZW7 53259219 Ki = 5845 nM T97537 C4KZ7R 53259403 Ki = 4011 nM T97537 CA0Q2E 53259404 Ki = 12000 nM T97537 C6FU2G 53259405 Ki = 10800 nM T97537 CLSC37 53261358 Ki = 25 nM T97537 CXMC12 53261359 Ki = 64.2 nM T97537 C3Q4ZR 53261360 Ki = 193 nM T97537 CGF98A 54585162 Ki = 30.4 nM T97537 CG46AV 71817662 IC50 = 38300 nM T97537 C7P2UD 71817806 IC50 = 3900 nM T97537 CW85UH 71817807 IC50 > 100000 nM T97537 CO8K1H 71817808 IC50 = 46000 nM T97537 CMQN63 71817809 IC50 = 10300 nM T97537 CPNL07 71817811 IC50 = 9600 nM T97537 C1N7QD 71817963 IC50 = 2800 nM T97537 CMBJ36 71817964 IC50 = 1300 nM T97537 CK2T9X 71817965 IC50 = 16300 nM T97537 CE7VJ4 71817966 IC50 > 100000 nM T97537 C74CNV 72193911 IC50 = 30 nM T97537 C8ZGB7 118734158 IC50 = 10000 nM T97537 C0T8FC 118734159 IC50 = 10700 nM T97537 CU5F3O 118734160 IC50 = 57000 nM T97537 CB67XZ 118734161 IC50 = 10900 nM T97537 CJ19XY 118734162 IC50 = 2100 nM T97537 C67EIN 118734163 IC50 = 12000 nM T97537 C5HV4G 118734165 IC50 = 7200 nM T97537 CB7W1N 118734166 IC50 = 14600 nM T97537 CVQ9B5 118734167 IC50 = 34000 nM T97537 CTE28S 118734169 IC50 > 100000 nM T97537 C3VMB4 118734170 IC50 = 3800 nM T97537 C5B3AO 118734171 IC50 = 4800 nM T97537 CR02XN 118734172 IC50 = 10700 nM T97537 CYQ61P 118734173 IC50 = 5700 nM T97537 CG1NJ3 118734176 IC50 = 4100 nM T97537 CTL4C9 118734177 IC50 > 100000 nM T97537 CWK18R 118734179 IC50 = 12000 nM T97537 CED26H 118734180 IC50 > 100000 nM T97537 C24VOF 118734181 IC50 = 22000 nM T97537 C3KJR9 118734182 IC50 > 100000 nM T97537 CMWH70 118734252 IC50 = 7100 nM T97537 CS1R6T 118734253 IC50 > 100000 nM T97537 CK3NV4 118734254 IC50 = 933 nM T97537 C4VK6O 118734255 IC50 = 4400 nM T97537 C7AH4D 118734256 IC50 = 1300 nM T97537 CZ04FM 118734257 IC50 > 100000 nM T97537 CZ97HL 118734258 IC50 = 1200 nM T97537 C1DKP8 118734259 IC50 = 105 nM T97537 CET0D8 118734260 IC50 = 296 nM T97537 C4N7KF 118734261 IC50 = 31000 nM T97537 C2M4UZ 118734262 IC50 = 3300 nM T97537 C3PL1T 118734263 IC50 = 966 nM T97537 C3OS1H 118734264 IC50 = 655 nM T97537 C9NWC0 118734265 IC50 = 31000 nM T97537 C3PW9J 118734266 IC50 = 1700 nM T97537 CX0OA9 118734267 IC50 = 8300 nM T97537 CU8I4F 118734268 IC50 = 3300 nM T97537 CI6S8L 118734269 IC50 = 39600 nM T97537 C6IB5P 118734270 IC50 > 100000 nM T97537 CUGM56 118734271 IC50 = 9900 nM T97537 CH2LO8 118734272 IC50 = 22500 nM T97537 CI9RT3 118734273 IC50 > 100000 nM T97537 CK32TS 118734274 IC50 = 2500 nM T97537 CT5F3Q 118734275 IC50 = 20600 nM T97537 C3KLH4 118734276 IC50 = 14400 nM T97537 CPUI84 118734277 IC50 = 20200 nM T97537 C96PKA 118734278 IC50 = 1300 nM T97537 C4AL9Z 118734279 IC50 = 2400 nM T97537 C71TGN 118734280 IC50 = 4700 nM T97537 C8V9EB 118734281 IC50 = 2900 nM T97537 CIZ3Q6 118734282 IC50 = 3700 nM T97537 CJ64ZC 118734283 IC50 = 3800 nM T97537 C1K7AN 118734284 IC50 = 1300 nM T97537 C6XY9M 118734285 IC50 = 70000 nM T97537 CY8X0V 118734286 IC50 = 3400 nM T97537 CO4F3Y 118734287 IC50 = 5200 nM T97537 C9CN6S 118734288 IC50 = 3700 nM T97537 CI3R0S 118734289 IC50 > 100000 nM T97537 CN7SR4 118734290 IC50 = 3900 nM T97537 C57ZSG 118734291 IC50 > 100000 nM T97537 CKST54 118734292 IC50 = 3600 nM T97537 C9XDY5 118734293 IC50 = 438 nM T97537 C01PYL 118734294 IC50 = 1700 nM T97537 CO6PR7 118734295 IC50 = 35700 nM T97537 C4ZPC8 118734296 IC50 = 2200 nM T97537 CJ40TN 118734297 IC50 = 7600 nM T97537 CA9X0N 118734298 IC50 = 4900 nM T97537 C7FMV5 126456392 Ki = 18 nM T97537 C8QO7V 135554374 IC50 = 28000 nM T97537 CXLS30 137633011 IC50 = 381 nM T97537 CMC5E8 137634250 IC50 = 18 nM T97537 CER06G 137637900 IC50 = 577 nM T97537 C97XKO 137638141 IC50 = 16 nM T97537 CMTG53 137639983 IC50 = 1754 nM T97537 CH6DQ2 137640549 IC50 = 281 nM T97537 C9SWV7 137640590 IC50 = 46 nM T97537 CG0ED2 137641900 IC50 = 14 nM T97537 C3SP9K 137642894 IC50 = 317 nM T97537 C1U3ZM 137642974 IC50 = 1800 nM T97537 CYN9Z5 137646376 IC50 = 41 nM T97537 CDU93R 137646849 IC50 = 13 nM T97537 C96EWT 137647165 IC50 = 32 nM T97537 CJM57W 137648545 IC50 = 13 nM T97537 CC9T7O 137650040 IC50 = 9 nM T97537 CN9F2A 137650752 IC50 = 185 nM T97537 CB9VI7 137652734 IC50 = 102 nM T97537 CSM3V5 137653412 IC50 = 221 nM T97537 CVI87E 137654495 IC50 = 21 nM T97537 C8DV5C 137655020 IC50 = 4024 nM T97537 C2RIG6 137655030 IC50 = 4 nM T97537 CMT56C 137655972 IC50 = 434 nM T97537 C13POW 137656080 IC50 = 561 nM T97537 CCTK37 137657323 IC50 = 34 nM T97537 C4VS2D 137658289 IC50 = 20 nM T97537 CKHE71 137659752 IC50 = 10 nM T97537 C0ID7T 137660529 IC50 = 2 nM T97537 C8E6UD 137661774 IC50 = 29 nM T97537 CV2U0Z 137662110 IC50 = 41 nM T97537 D02MNM 71817810 IC50 = 6000 nM T97537 D04DTE 53259050 Ki = 1.8 nM T97537 D0L3PY 123814 Ki = 7 nM T88415 COQ0J9 9846486 IC50 = 3500 nM T88415 CSH73Q 43230121 IC50 = 5000 nM T88415 C09TSQ 145978898 IC50 = 100 nM T88415 CFX8E2 145979186 IC50 > 100000 nM T88415 CS9M7U 145990033 IC50 = 800 nM T88415 CS2HG5 145991728 IC50 = 100 nM T88415 C4K2YT 145992615 IC50 > 10000 nM T40488 D05VZE 119031 IC50 = 10000 nM T40488 D03BOZ 3342298 IC50 = 0.54 nM T40488 CN6E3U 2366268 IC50 = 83000 nM T40488 CR7T3J 10009978 Ki > 2000 nM T40488 C1LCH3 10016964 IC50 = 62000 nM T40488 CR5H6E 10163627 IC50 = 1600 nM T40488 CK0P3F 10186536 IC50 > 10000 nM T40488 C4K1MJ 10208262 IC50 = 4600 nM T40488 CBM0Y4 10252411 Ki < 100 nM T40488 CY08WJ 10322755 Ki = 1650 nM T40488 CFKA79 10395015 Ki > 2000 nM T40488 C5WV1N 10439082 Ki > 2000 nM T40488 C8C5AV 11294179 IC50 > 10000 nM T40488 CO8QT0 11753905 Ki = 240 nM T40488 C8YWV5 11778852 IC50 = 53000 nM T40488 C02BWA 11967143 Ki > 2000 nM T40488 CQS0F5 16719301 IC50 = 55 nM T40488 C75XDI 16730519 IC50 = 2400 nM T40488 C1MCG7 22004293 Ki = 335 nM T40488 CAQ9Z1 25022681 Ki > 5346 nM T40488 CHQG04 44576676 Ki = 23000 nM T40488 CR65DO 44576708 Ki = 1600 nM T40488 C2QFY7 44576710 Ki = 4570 nM T40488 CU2IP7 44576753 Ki = 22000 nM T40488 C93LDF 44576807 Ki = 372000 nM T40488 CJ41MB 44576851 Ki = 337000 nM T40488 CU2SX3 51355576 Ki > 10000 nM T40488 C6Y2EV 53374826 IC50 > 100000 nM T40488 C1PHI6 57708731 IC50 = 820 nM T40488 CF2Z7W 57708783 IC50 = 140 nM T40488 C9KV2W 57708792 IC50 = 460 nM T40488 CE36GP 57708799 IC50 = 270 nM T40488 C23QGY 57708843 IC50 > 1000 nM T40488 C2J5CW 57708880 IC50 > 1000 nM T40488 C1K6AP 57708886 IC50 = 30 nM T40488 C61NKZ 72720906 IC50 = 21 nM T40488 C7XWM5 72948626 IC50 = 17 nM T40488 CR70EY 72948808 IC50 = 12 nM T40488 C2WV4D 72948991 IC50 = 7810 nM T40488 CA76TR 72948995 IC50 = 18 nM T40488 CZ95GN 72949172 IC50 = 16 nM T40488 CSH7A5 90033597 IC50 = 11400 nM T40488 CYZP25 91824169 IC50 > 10000 nM T40488 C0M3QS 118179775 IC50 = 42 nM T40488 C0XML2 118179776 IC50 = 62 nM T40488 C0W3NG 118179777 IC50 = 435 nM T40488 CX9YG0 118179779 IC50 = 7 nM T40488 CW1TU9 118179786 IC50 = 54 nM T40488 CRG2W5 118179799 IC50 = 189 nM T40488 CH35NR 118179800 IC50 = 9 nM T40488 CK54UB 118179801 IC50 = 739 nM T40488 CP8QO0 118179807 IC50 = 13 nM T40488 CT4G5D 118179817 IC50 = 68 nM T40488 CIU02H 118179819 IC50 = 4 nM T40488 CD9TG2 118179830 IC50 = 103 nM T40488 CN72KV 118179833 IC50 = 184 nM T40488 CZ01AH 118179837 IC50 = 713 nM T40488 C6TR4O 118179845 IC50 = 25400 nM T40488 C5TZ1D 118179847 IC50 = 14 nM T40488 CVWR97 118179850 IC50 = 20700 nM T40488 CT8U1K 118179865 IC50 = 8700 nM T40488 CR64FW 118179867 IC50 = 84 nM T40488 CIXQ34 118179870 IC50 = 3 nM T40488 C27XIK 118225133 IC50 > 10000 nM T40488 C58KIN 118233723 IC50 > 10000 nM T40488 CU6ES2 118233724 IC50 > 10000 nM T40488 C8ET1Z 118233725 IC50 > 10000 nM T40488 C9P0LC 118233726 IC50 > 10000 nM T40488 C8SIM0 118233727 IC50 > 10000 nM T40488 CQTE52 118233728 IC50 > 10000 nM T40488 CEVI64 118233730 IC50 > 10000 nM T40488 C08CPE 118233731 IC50 > 10000 nM T40488 C8Q5XC 118233733 IC50 > 10000 nM T40488 CZQO42 118233734 IC50 > 10000 nM T40488 CCDG68 118233743 IC50 > 10000 nM T40488 C25TYU 118233744 IC50 > 10000 nM T40488 CL5UV6 118233745 IC50 > 10000 nM T40488 C8XWB9 118233746 IC50 > 10000 nM T40488 CC7K9R 118233747 IC50 > 10000 nM T40488 CGA7J1 118233748 IC50 > 10000 nM T40488 CVIG81 118233749 IC50 > 10000 nM T40488 CTU81Y 118233750 IC50 > 10000 nM T40488 CCA6W2 118233751 IC50 > 10000 nM T40488 C60QIZ 118233752 IC50 > 10000 nM T40488 CS5G9T 118233753 IC50 > 10000 nM T40488 CGKD16 118734983 IC50 = 32 nM T40488 C84NEC 118734984 IC50 = 89 nM T40488 CX7H5Q 118734985 IC50 = 17 nM T40488 CNF86U 121493953 Ki = 1.4 nM T40488 CH1GT7 123144081 IC50 > 10000 nM T40488 CKNI84 127050262 IC50 = 8400 nM T40488 CN9D7G 134155756 IC50 = 6300 nM T40488 CHV2U1 135438561 IC50 = 160 nM T40488 C6GR3K 135567051 IC50 = 140 nM T40488 CYH23I 136054468 IC50 = 220 nM T40488 CZ8DW1 136054472 IC50 = 34 nM T40488 C9H0DL 136054473 IC50 = 460 nM T40488 CX7MI0 136054475 IC50 = 64 nM T40488 CA5JR6 136054481 IC50 = 240 nM T40488 CO2VU9 136054484 IC50 < 10 nM T40488 CV47JN 136054485 IC50 = 6.2 nM T40488 CZ48WO 136054487 IC50 = 150 nM T40488 CR9CY5 136054490 IC50 < 10 nM T40488 C8FGT0 136054495 IC50 = 930 nM T40488 CGH39U 136054498 IC50 < 10 nM T40488 C2TO7Y 136054508 IC50 = 640 nM T40488 CG70BZ 136054516 IC50 = 0.35 nM T40488 CSM57W 136054520 IC50 = 2.6 nM T40488 CIEW62 136380958 IC50 = 2.4 nM T40488 C9HS7J 137287436 IC50 = 0.3 nM T40488 CAZ87R 137631621 IC50 = 676.08 nM T40488 C0R5ZT 137635841 IC50 = 436.52 nM T40488 CU5G8I 137636679 IC50 = 635 nM T40488 C1RID9 137636861 IC50 = 2050 nM T40488 CNM8J4 137638970 IC50 = 29.51 nM T40488 C7Y0FB 137642170 IC50 = 1210 nM T40488 CDOQ29 137644394 IC50 = 1698.24 nM T40488 C04KVQ 137647395 IC50 = 705 nM T40488 CHI2E1 137648744 IC50 = 112.2 nM T40488 C1U2QR 137651063 IC50 = 141.25 nM T40488 C5Y8RP 137654086 IC50 = 7380 nM T40488 CRD46H 137658344 IC50 = 347 nM T40488 C3ER5O 137658673 IC50 = 506 nM T40488 CEQ8I9 137659945 IC50 = 588.84 nM T40488 CHO70T 137660954 IC50 = 751 nM T40488 C1IF6L 137661809 IC50 = 131 nM T40488 CYFQ54 144883303 IC50 > 10000 nM T40488 CA2EI4 144883305 IC50 > 10000 nM T40488 CX80ML 144883318 IC50 > 10000 nM T40488 CQYH92 145949456 IC50 > 10000 nM T40488 C2SM0T 145950300 IC50 > 10000 nM T40488 C85BXD 145951133 IC50 > 10000 nM T40488 C6JP8O 145955500 IC50 > 10000 nM T40488 CXT3I5 145958912 IC50 > 10000 nM T40488 CQN59P 145959729 IC50 > 10000 nM T40488 CX6R5D 145959924 IC50 > 10000 nM T40488 C0K4JW 145972664 IC50 > 10000 nM T40488 CF64GH 155518335 Ki = 983 nM T40488 D03AMR 9849669 Ki = 190 nM T40488 D04VPH 45376872 IC50 = 16000 nM T40488 D07SPC 24857837 Ki = 356 nM T40488 D0B3UN 44580458 Ki = 149 nM T40488 D0OR6O 91623362 IC50 = 12 nM T40488 D0Y5IQ 44255320 IC50 = 5000 nM T10877 D04AIT 5280445 IC50 = 8200 nM T10877 D0K8KX 5280343 IC50 = 37900 nM T10877 D0E3LP 5113032 IC50 > 100000 nM T10877 D0U3EP 445154 IC50 > 100000 nM T10877 CU12QE 1203 IC50 > 100000 nM T10877 CEM9Q1 128853 IC50 = 14600 nM T10877 CNMW58 159287 IC50 = 17000 nM T10877 CAB1I4 440832 IC50 = 16300 nM T10877 CT2S6P 441667 IC50 = 6300 nM T10877 CG5OR9 441697 IC50 = 14200 nM T10877 CHE81U 441701 IC50 = 6000 nM T10877 CXB75J 441773 IC50 = 20900 nM T10877 CXG1I8 441774 IC50 = 39200 nM T10877 CLY6K3 661302 IC50 > 100000 nM T10877 CJ0T4E 3612016 IC50 > 100000 nM T10877 CY9C4T 5281680 IC50 = 48600 nM T10877 C4KG0A 5403988 IC50 = 296000 nM T10877 CKC79O 10053069 IC50 = 276000 nM T10877 C5J6HV 11170346 IC50 = 158000 nM T10877 CU7Y3S 12309895 IC50 = 70300 nM T10877 C5VH6T 14842007 IC50 = 32100 nM T10877 C4DQJ9 24285123 IC50 = 120000 nM T10877 C36ILR 44532635 IC50 = 1210 nM T10877 CLX72I 59474759 IC50 > 30000 nM T10877 C5GB8X 91827499 IC50 = 76 nM T10877 C64QCZ 91827500 IC50 = 7200 nM T10877 CM01EG 101886781 IC50 = 27000 nM T10877 CWC1Q3 101886782 IC50 = 6400 nM T10877 C5G1LT 101886783 IC50 = 33000 nM T10877 CDT01C 101886784 IC50 = 3300 nM T10877 CQUF15 118736849 IC50 = 58 nM T10877 C5KPU3 118736852 Ki = 14 nM T10877 CG7I6Z 118736853 IC50 = 52 nM T10877 CDR8M7 118736855 IC50 = 3.9 nM T10877 C3M6IP 118736856 Ki = 0.3 nM T10877 CZSB48 118736857 Ki = 0.7 nM T10877 CIE3W9 118736858 IC50 = 54 nM T10877 CH26AO 118736859 IC50 = 3.8 nM T10877 CAQM69 118736860 IC50 = 13 nM T10877 CEL48B 118736861 Ki = 0.45 nM T10877 C7JQ3Y 118736862 IC50 = 14 nM T10877 C6MZ9V 118736863 IC50 = 10773 nM T10877 C0U5DA 118736864 IC50 = 498 nM T10877 CZVT62 118736865 IC50 = 959 nM T10877 CE21BJ 118736866 IC50 = 1960 nM T10877 C30BIV 118736867 IC50 = 11400 nM T10877 CC10IV 118736868 IC50 = 3350 nM T10877 CXO8F1 118736869 IC50 = 2300 nM T10877 CAYX13 118736870 IC50 = 23400 nM T10877 CDW94Q 118736871 IC50 > 30200 nM T10877 CY4LA6 118736872 IC50 = 4710 nM T10877 CTCH72 118736873 IC50 = 1160 nM T10877 C3ARY5 118736874 IC50 = 1590 nM T10877 CW4O7N 118736875 IC50 = 263 nM T10877 CL51QY 118736876 IC50 = 206 nM T10877 CKMD80 118736877 IC50 = 28 nM T10877 CY93JQ 118736878 IC50 = 26 nM T10877 C73EMV 118736879 IC50 = 64 nM T10877 C1B2JZ 118736880 IC50 = 53 nM T10877 C5KGR7 118736881 IC50 = 42 nM T10877 CVM02C 118736882 IC50 = 245 nM T10877 CCH64S 118736883 IC50 = 50 nM T10877 CB6S3J 118736884 IC50 = 3.4 nM T10877 C2SWZ4 118736886 IC50 = 4.8 nM T10877 CXEC56 118736887 IC50 = 5.3 nM T10877 C9LJ0B 118736888 IC50 = 298 nM T10877 C06HDY 118736889 IC50 = 840 nM T10877 CT8G1K 118736890 IC50 = 1200 nM T10877 CUN41C 118736891 IC50 = 1320 nM T10877 CGJW47 118736892 IC50 = 700 nM T10877 CAU39P 118736893 IC50 = 3610 nM T10877 CT5A7R 118736894 IC50 = 2330 nM T10877 C1YMX6 118736895 IC50 = 970 nM T10877 C0RD2H 118736896 IC50 = 4680 nM T10877 CO70TW 118736897 IC50 = 1230 nM T10877 C8HC3W 118736898 IC50 = 1160 nM T10877 CK2LV7 118736899 IC50 = 12800 nM T10877 CXQ37E 118736900 IC50 = 2150 nM T10877 CRT50V 118736901 IC50 = 700 nM T10877 CPAE18 118736902 IC50 = 970 nM T10877 CUPZ76 118736903 IC50 = 2690 nM T10877 CA87UE 118736904 IC50 = 560 nM T10877 CS59UX 118736905 IC50 = 840 nM T10877 CL7CR9 118736906 IC50 = 460 nM T10877 CT0EM6 118736907 IC50 = 1460 nM T10877 C3AJ1K 118736908 IC50 = 12300 nM T10877 CXJQ24 118736909 IC50 = 3940 nM T10877 CL0OQ1 118736910 IC50 = 950 nM T10877 C8TWX1 118736911 IC50 = 7830 nM T10877 C4OW8Z 118736912 IC50 = 1930 nM T10877 C6W4EN 118736913 IC50 = 281 nM T10877 C4FY6U 118736914 IC50 = 132 nM T10877 C6M7KH 118736915 IC50 = 1680 nM T10877 C3U9ZQ 118736916 IC50 = 1060 nM T10877 CN3DE6 118736989 IC50 = 1030 nM T10877 C3A5TU 118736990 IC50 > 30200 nM T10877 C7USD5 118736991 IC50 > 30200 nM T10877 CH1XL4 118736992 IC50 = 149 nM T10877 C2U9HL 118736993 IC50 = 1220 nM T10877 CI24RE 118736994 IC50 = 117 nM T10877 CDC8E7 118736995 IC50 = 140 nM T10877 CND2U1 118736996 IC50 = 49 nM T10877 C1BGP6 118736997 IC50 = 142 nM T10877 CMO4B9 118736998 IC50 = 406 nM T10877 C0Y4VE 118736999 IC50 = 78 nM T10877 CDV30H 118737000 IC50 = 971 nM T10877 C0XI5O 118737001 IC50 = 92 nM T10877 CQD48J 122185943 IC50 > 30000 nM T10877 C6Y2MI 122185944 IC50 = 22000 nM T10877 CR9G7S 122185945 IC50 = 22000 nM T10877 CD64IJ 122185946 IC50 = 3300 nM T10877 CE9OP1 122185947 IC50 > 30000 nM T10877 CBEL62 122185948 IC50 > 30000 nM T10877 CYM8D4 122185949 IC50 = 19000 nM T10877 CE1ZO9 122185950 IC50 > 30000 nM T10877 CE6VJ3 122185951 IC50 > 30000 nM T10877 CX76QZ 122185952 IC50 = 17000 nM T10877 CZ8N9B 122185953 IC50 = 25000 nM T10877 CHE12L 122185954 IC50 = 3300 nM T10877 CL94EM 122185955 IC50 = 2300 nM T10877 CJ17HX 122185956 IC50 > 30000 nM T10877 CI01XG 122185957 IC50 = 18000 nM T10877 CR9AX0 122185958 IC50 = 620 nM T10877 C79BPI 122185959 IC50 > 30000 nM T10877 CZL15G 122185960 IC50 = 4500 nM T10877 CJOV10 122185961 IC50 > 30000 nM T10877 CY2W1Z 122185962 IC50 = 11000 nM T10877 CEV6S8 122185963 IC50 = 990 nM T10877 CM9A0O 122185964 IC50 > 30000 nM T10877 C6D9YZ 122185965 IC50 = 15000 nM T10877 C9CA8T 122185966 IC50 > 30000 nM T10877 C9KAB4 122185967 IC50 > 30000 nM T10877 CLJ1R3 122185968 IC50 = 16000 nM T10877 C6OA7C 122185969 IC50 = 4000 nM T10877 CH16FN 122185970 IC50 = 9600 nM T10877 C8V0WI 122185971 IC50 = 24000 nM T10877 C1FB8D 122185972 IC50 = 6200 nM T10877 CX89LW 122185973 IC50 = 780 nM T10877 CK0UN1 122185974 IC50 = 1200 nM T10877 CQ1WJ8 122185975 IC50 = 510 nM T10877 CKD43Z 122185976 IC50 = 150 nM T10877 CV73WF 122185977 IC50 = 4700 nM T10877 CS7YJ2 122185978 IC50 = 170 nM T10877 CEIT53 122185979 IC50 = 3600 nM T10877 C3ZNU8 122185980 IC50 = 130 nM T10877 CN5P3Q 122185981 IC50 = 280 nM T10877 CIU0M2 122185982 IC50 = 8500 nM T10877 C13TYI 122185983 IC50 = 7300 nM T10877 CSZ0K1 122185984 IC50 > 30000 nM T10877 C8OL5C 122185985 IC50 = 2100 nM T10877 CU47TS 122185986 IC50 = 4900 nM T10877 CVUP84 122185987 IC50 > 30000 nM T10877 CM47OU 122185988 IC50 = 11000 nM T10877 C1DVY8 122185989 IC50 > 30000 nM T10877 CI01VG 122185990 IC50 > 30000 nM T10877 C0M9EL 122185991 IC50 > 30000 nM T10877 CM4S0B 122185992 IC50 > 30000 nM T10877 CO2R4W 122185993 IC50 = 6600 nM T10877 CN4B2Y 122185994 IC50 = 2700 nM T10877 C8WPN3 122185995 IC50 > 30000 nM T10877 CUG8B4 122185996 IC50 > 30000 nM T10877 COYI82 122185997 IC50 > 30000 nM T10877 CSC4B7 122185998 IC50 > 30000 nM T10877 CSOI57 122185999 IC50 = 24000 nM T10877 CGAB47 122186000 IC50 > 10000 nM T10877 CB2H6L 122186001 IC50 > 30000 nM T10877 CZ3R6F 122186002 IC50 > 30000 nM T10877 C6DN9H 122186003 IC50 > 30000 nM T10877 CD0QV5 122186004 IC50 > 30000 nM T10877 CEHN13 122186005 IC50 > 30000 nM T10877 CKFD41 122186006 IC50 > 30000 nM T10877 CU87NS 122186007 IC50 > 30000 nM T10877 CSZ5T7 122186008 IC50 > 30000 nM T10877 C5DU6F 122186009 IC50 > 30000 nM T10877 CQB19L 122186010 IC50 = 9200 nM T10877 C46EGM 135900947 IC50 = 430000 nM T10877 C61OBZ 135949782 IC50 = 103000 nM T10877 C6MF7P 136124133 IC50 = 109000 nM T10877 C0E3AH 136198640 IC50 = 14000 nM T10877 CACG84 136198641 IC50 = 26000 nM T10877 C4Z1WR 137442659 IC50 = 1900 nM T10877 CN09RB 137442681 IC50 = 450 nM T10877 C9G6IA 137442708 IC50 = 630 nM T10877 C9PUZ4 137442715 IC50 = 620 nM T10877 C7DP2S 137442862 IC50 = 92 nM T10877 CW8LT6 137442987 IC50 = 2300 nM T10877 CK26ZH 145967624 IC50 = 7.8 nM T10877 C0YGC8 145967690 IC50 = 1600 nM T10877 CV90MY 145967850 IC50 = 110 nM T10877 C0KJD1 145967861 IC50 = 21 nM T10877 COYK91 145968096 IC50 = 370 nM T10877 CC4P8J 145968138 IC50 = 72 nM T10877 CIW3B1 145968359 IC50 = 3400 nM T10877 C6F4SD 145968563 IC50 = 4100 nM T10877 COA4B0 145968763 IC50 = 170 nM T10877 CX4GA2 145968779 IC50 = 310 nM T10877 C9YRW1 145968807 IC50 = 1900 nM T10877 C4D1JT 145968829 IC50 = 8000 nM T10877 C9SV6Y 145969196 IC50 = 17 nM T10877 CS70GC 145969309 IC50 = 82 nM T10877 CNH7O5 145969326 IC50 = 51 nM T10877 CHZ7N3 145969706 IC50 = 42 nM T10877 CN56YO 145969928 IC50 = 330 nM T10877 C4CDN0 145969972 IC50 = 83 nM T10877 C1I3TK 145970025 IC50 = 6800 nM T10877 C6A0HJ 145970175 IC50 = 140 nM T10877 CJC43R 145970183 IC50 = 5500 nM T10877 CMKZ95 145970214 IC50 = 4200 nM T10877 CB2NU1 145970392 IC50 = 1600 nM T10877 CJR21T 145970400 IC50 = 410 nM T10877 CQ82EI 145970446 IC50 = 4300 nM T10877 CORE90 145970461 IC50 = 230 nM T10877 C4GR7E 145970630 IC50 = 71 nM T10877 CB4RP9 145970636 IC50 = 160 nM T10877 C3LD1Y 145970800 IC50 = 20 nM T10877 C7N2ZY 145970856 IC50 = 45 nM T10877 CUSO84 145970885 IC50 = 110 nM T10877 CKDZ10 145971093 IC50 = 19000 nM T10877 CW6ER8 145987053 IC50 = 4 nM T10877 CYT73F 145987735 IC50 = 2500 nM T10877 D07NAY 5281692 IC50 = 37900 nM T10877 D0E1QP 4262314 IC50 > 100000 nM T10877 D0O0VZ 667639 IC50 > 100000 nM T10877 D0T3PW 5281672 IC50 = 24800 nM T10877 D0V3PG 128861 IC50 = 21800 nM T69912 D0T9TJ 3034010 IC50 = 50 nM T69912 D05GZD 9918381 IC50 = 0.2512 nM T69912 D0CW8S 71657619 IC50 > 10000 nM T69912 D09NBM 10417440 Ki = 0.03 nM T69912 D0L5UO 9939609 IC50 = 0.035 nM T69912 CN1K3D 5699 IC50 > 100000 nM T69912 CZI2U1 6491 IC50 > 1000000 nM T69912 CYFU26 130606 IC50 > 100000 nM T69912 CZ3R1F 669158 IC50 = 1000000 nM T69912 C2KRB1 973435 IC50 = 44000 nM T69912 CMN1P8 1217803 IC50 = 3431 nM T69912 C2F7OG 2412772 IC50 = 1000000 nM T69912 C9VZ3F 3638243 IC50 > 100000 nM T69912 C1FHP8 4811752 IC50 = 14000 nM T69912 CG0F8O 9808838 IC50 = 1 nM T69912 CC5Y0A 9809899 IC50 = 533 nM T69912 C4TB5Y 9831072 IC50 = 0.6 nM T69912 C4VH8G 9840384 IC50 = 850 nM T69912 CB0EP8 9850883 IC50 = 26 nM T69912 C4R6CU 9851531 IC50 = 20 nM T69912 C89RJZ 9852438 IC50 = 0.5 nM T69912 CTJO81 9893629 IC50 = 85 nM T69912 C9FWY2 9895919 IC50 = 2 nM T69912 C6MD8O 9917136 IC50 = 8 nM T69912 C19SKN 9917325 IC50 = 0.7 nM T69912 CX23UG 9917667 IC50 = 9 nM T69912 CMBO57 9917750 IC50 = 0.4 nM T69912 CSB71L 9938151 IC50 = 18 nM T69912 CFH61N 9938577 IC50 = 26 nM T69912 CMN74S 9938642 IC50 = 12 nM T69912 CGL13H 9939495 IC50 = 0.4 nM T69912 C2EF8Q 9939518 IC50 = 2 nM T69912 CQEN19 9959703 IC50 = 24 nM T69912 C8C0HB 9961561 IC50 = 1 nM T69912 CSW8T3 9961700 IC50 = 0.3 nM T69912 C8X7KP 9961715 IC50 = 9 nM T69912 C1DB0X 10055750 IC50 = 0.17 nM T69912 C1TY3F 10122289 IC50 = 0.25 nM T69912 C0KOC5 10122452 IC50 = 3 nM T69912 C1LSI8 10122657 IC50 = 0.1 nM T69912 CJ4R2U 10168216 IC50 = 0.4 nM T69912 CAK3E1 10189993 IC50 = 0.8 nM T69912 CPG87K 10189998 IC50 = 38 nM T69912 CG65NB 10190629 IC50 = 1 nM T69912 CIK7C8 10211722 IC50 = 1.5 nM T69912 CA4EF3 10211894 IC50 = 2 nM T69912 CFQ5L2 10232552 IC50 = 5 nM T69912 CB72SI 10233112 IC50 = 1 nM T69912 C9UIX5 10233517 IC50 = 0.8 nM T69912 C61ZEV 10282620 IC50 = 1 nM T69912 CQV98P 10305047 IC50 = 0.5 nM T69912 COAR34 10305066 IC50 = 19 nM T69912 CZA96C 10305422 IC50 = 0.8 nM T69912 C7W2NF 10305573 IC50 = 1 nM T69912 C8OPC6 10305637 IC50 = 6 nM T69912 C03CJA 10320992 IC50 = 64 nM T69912 C0JB9D 10394633 IC50 = 0.7 nM T69912 CD3MH2 10411777 IC50 = 54 nM T69912 CU78FP 11521655 IC50 = 25000 nM T69912 CZRT87 11543912 IC50 = 38000 nM T69912 CJW8M7 11564757 IC50 = 26000 nM T69912 C09ASJ 11764593 IC50 = 0.2 nM T69912 CU0Y2Z 12051594 IC50 = 2 nM T69912 C6O8ID 14490158 IC50 = 1000000 nM T69912 CS5CV2 16126765 IC50 = 120 nM T69912 CGN9S6 17899989 IC50 = 640 nM T69912 CK14ET 17899991 IC50 = 210 nM T69912 C8C4LK 18470089 IC50 = 110 nM T69912 C0EU2T 18470090 IC50 = 0.3 nM T69912 C63DZQ 18470117 IC50 = 19 nM T69912 C7FV0Y 18470125 IC50 = 850 nM T69912 CRS63W 18470138 IC50 = 90 nM T69912 CJ0Q9T 18470140 IC50 = 17000 nM T69912 CFI50Y 18470152 IC50 = 34 nM T69912 C1WJ5A 18470163 IC50 = 1000 nM T69912 CZJ25E 18470168 IC50 = 19 nM T69912 CK47RM 18470169 IC50 = 200 nM T69912 C69SCV 18470191 IC50 = 4 nM T69912 C38OXW 18470208 IC50 = 1400 nM T69912 C68IDK 18470209 IC50 = 1000 nM T69912 CYF0B8 18470218 IC50 = 4400 nM T69912 C24HOS 18470241 IC50 = 2 nM T69912 C1Q8NP 18470244 IC50 = 11 nM T69912 CIEQ59 18470251 IC50 = 780 nM T69912 CE69PL 18470253 IC50 = 210 nM T69912 CP5S1M 18470258 IC50 = 650 nM T69912 C1NLE8 18470267 Ki = 41 nM T69912 CA38TG 18470272 IC50 = 430 nM T69912 C9Z0PI 18470273 IC50 = 660 nM T69912 CUTF18 18470282 IC50 = 12000 nM T69912 C9BRG5 18470283 IC50 = 250 nM T69912 CBZ1V0 18470296 IC50 = 12600 nM T69912 CT10SU 18470303 IC50 = 19 nM T69912 CJ35LB 18470304 IC50 = 4400 nM T69912 CV2Q4O 18470306 IC50 = 150 nM T69912 C2EGW7 18470314 IC50 = 16 nM T69912 C6CVW9 18470315 IC50 = 7 nM T69912 CR6S2P 18470316 IC50 = 1300 nM T69912 CT1G0Z 18470322 IC50 = 285 nM T69912 CU3QI1 18470341 IC50 = 960 nM T69912 CEIF53 18470354 IC50 = 450 nM T69912 CS93WA 18470361 IC50 = 2900 nM T69912 C0BE4O 18470368 IC50 = 110 nM T69912 CLS52M 18470371 IC50 = 1000 nM T69912 C8HNR6 18470375 IC50 = 450 nM T69912 C7VK9N 18470385 IC50 = 300 nM T69912 CX6EC7 18470390 IC50 = 250 nM T69912 C45GTM 18470395 IC50 = 0.1 nM T69912 C2EL5G 18470399 IC50 = 55000 nM T69912 C60DVF 18470400 IC50 = 1200 nM T69912 CXW4D9 18470406 IC50 = 200 nM T69912 C07FGB 18470420 IC50 = 330 nM T69912 CPE8J7 18470422 IC50 = 5700 nM T69912 CE1Y8Q 18470432 IC50 = 1400 nM T69912 CL0GA7 18470436 IC50 = 1200 nM T69912 CUA07V 18470440 IC50 = 1100 nM T69912 C0TQ3E 18470452 IC50 = 1100 nM T69912 C5GC2U 18470455 IC50 = 1 nM T69912 CHN74T 18470468 IC50 = 70 nM T69912 C15KXN 18470470 IC50 = 2 nM T69912 CLGR76 18470474 IC50 = 2300 nM T69912 C14IMQ 18470482 IC50 = 630 nM T69912 CR50VA 18470483 IC50 = 1100 nM T69912 C78SLA 18470487 IC50 = 39 nM T69912 CDY3G7 18470494 IC50 = 230 nM T69912 CMFK89 18470498 IC50 = 36 nM T69912 CPI0Y6 18470516 IC50 = 250 nM T69912 CV47NE 18470522 IC50 = 110 nM T69912 C0FYD2 18470524 IC50 = 1100 nM T69912 CG18YS 18470527 IC50 = 7 nM T69912 CI9JK7 18470549 IC50 = 14000 nM T69912 C8Y9TC 18470552 IC50 = 140 nM T69912 CE83XT 18470555 IC50 = 3300 nM T69912 CJY4G6 18470556 IC50 = 1100 nM T69912 COIL12 18470582 IC50 = 2850 nM T69912 C1QV9I 18470585 IC50 = 990 nM T69912 CB95IU 18470590 IC50 = 0.4 nM T69912 CD2G1X 18470595 IC50 = 780 nM T69912 CH63UY 18540820 IC50 = 1 nM T69912 CRC64I 18768423 IC50 = 52.4 nM T69912 CY4AF7 21936103 IC50 = 0.1 nM T69912 C4VY5P 21936114 IC50 = 4 nM T69912 CMS86P 21936124 IC50 = 0.5 nM T69912 CDT3Y6 21936140 IC50 = 0.3 nM T69912 COEI56 21936146 IC50 = 5 nM T69912 C9C3JG 21936169 IC50 = 1 nM T69912 CN5ZP0 21936176 IC50 = 1 nM T69912 C4P8MH 21936183 IC50 = 0.2 nM T69912 C8U3FQ 21936197 IC50 = 8 nM T69912 C9PUJ0 21936206 IC50 = 15 nM T69912 CMR0P1 21936209 IC50 = 5 nM T69912 CB1W0U 21936229 IC50 = 4 nM T69912 CM8NF3 21936243 IC50 = 0.8 nM T69912 CV49NU 21936282 IC50 = 0.6 nM T69912 C6JX0D 21936319 IC50 = 0.2 nM T69912 CCU98M 21936326 IC50 = 3 nM T69912 CB5M3Q 21936345 IC50 = 0.2 nM T69912 CV8QT9 21936398 IC50 = 0.2 nM T69912 C0B2MU 21936403 IC50 = 4 nM T69912 CA4X5J 21936407 IC50 = 5 nM T69912 CEC2B6 22294074 IC50 = 0.5 nM T69912 C2BJY9 23395723 IC50 = 1 nM T69912 CW7FL6 23395729 IC50 = 0.6 nM T69912 C3CZL1 23395731 IC50 = 2.7 nM T69912 C02MBF 23395732 IC50 = 17 nM T69912 CDH5N2 23395748 IC50 = 8 nM T69912 C6Y9DO 23395749 IC50 = 4 nM T69912 CH3RP0 23395766 IC50 = 2 nM T69912 C0G8KF 23395772 IC50 = 0.7 nM T69912 C79IXE 23395774 IC50 = 0.12 nM T69912 CMQ2X3 23395778 IC50 = 1 nM T69912 CH7S9G 23395784 IC50 = 1.6 nM T69912 CXP67J 23395785 IC50 = 0.6 nM T69912 CFN51M 23395786 IC50 = 4.5 nM T69912 CVM86Y 23395788 IC50 = 1.4 nM T69912 C32CYB 23395790 IC50 = 0.8 nM T69912 C8A9OF 23395792 IC50 = 2 nM T69912 C4PL8S 23395794 IC50 = 5 nM T69912 CL2CM7 23395795 IC50 = 1 nM T69912 CW9G8Y 23395798 IC50 = 5 nM T69912 CE1J3W 23395801 IC50 = 0.7 nM T69912 CNDH71 23395803 IC50 = 0.2 nM T69912 CV9H3P 23395804 IC50 = 0.12 nM T69912 CH0G9B 23395805 IC50 = 0.2 nM T69912 CUXA85 23395806 IC50 = 0.35 nM T69912 C01DHS 23395807 IC50 = 0.5 nM T69912 CU2J0M 23395808 IC50 = 0.2 nM T69912 CET9J2 23395809 IC50 = 1.5 nM T69912 C73WNR 44266749 IC50 = 50 nM T69912 C4XW9G 44266800 IC50 = 3 nM T69912 C6OWG4 44300071 IC50 = 34 nM T69912 CKU80A 44300072 IC50 = 21 nM T69912 CLU67B 44300088 IC50 = 97 nM T69912 CD41MI 44300109 IC50 = 140 nM T69912 C6LK3F 44300123 IC50 = 66 nM T69912 C4CG6Q 44300126 IC50 = 1280 nM T69912 C1HYF9 44300132 IC50 = 460 nM T69912 CJE5Y8 44300187 IC50 = 39 nM T69912 CZ6M8X 44300263 IC50 = 350 nM T69912 CHR95L 44300266 IC50 = 260 nM T69912 C72MUZ 44300268 IC50 = 51 nM T69912 CZS4T9 44300303 IC50 = 44 nM T69912 CKNC02 44300306 IC50 = 70 nM T69912 C3WJC0 44300307 IC50 = 29 nM T69912 CUB07K 44300374 IC50 = 3 nM T69912 CD02LG 44300390 IC50 = 410 nM T69912 CQ7M6U 44300414 IC50 = 89 nM T69912 C3FAV2 44300418 IC50 = 6700 nM T69912 CX56UK 44300444 IC50 = 530 nM T69912 C8HPB9 44300446 IC50 = 720 nM T69912 C34HVB 44300478 IC50 = 130 nM T69912 C01MXK 44300573 IC50 = 10 nM T69912 CI2EA3 44300574 IC50 = 69 nM T69912 CK4D5X 44300578 IC50 = 5 nM T69912 CG5HW3 44300752 IC50 = 120 nM T69912 CXQI32 44300753 IC50 = 176 nM T69912 C4ZDS7 44319598 IC50 = 235 nM T69912 CVYP89 44319686 IC50 = 12 nM T69912 CFJD61 44319860 IC50 = 350 nM T69912 CH1TP7 44319861 IC50 = 300 nM T69912 CUV80P 44319972 IC50 = 250 nM T69912 COD96J 44319974 IC50 = 25 nM T69912 CJBU28 44319998 IC50 = 260 nM T69912 CCU1J0 44320037 IC50 = 3 nM T69912 C9UZM1 44320070 IC50 = 15 nM T69912 CL2A8D 44367433 IC50 = 1.6 nM T69912 C0BM7X 44367434 IC50 = 0.5 nM T69912 C0CNE9 44367483 IC50 = 1.6 nM T69912 C8HM0C 44367519 IC50 = 0.2 nM T69912 CGS4E6 44367542 IC50 = 1.7 nM T69912 C04WGR 44367559 IC50 = 5 nM T69912 C0Q9NA 44367560 IC50 = 2.6 nM T69912 CG7AQ0 44367583 IC50 = 0.9 nM T69912 CVB27E 44367645 IC50 = 194 nM T69912 CNK0A7 44367647 IC50 = 5 nM T69912 CQ6S3B 44367648 IC50 = 24 nM T69912 CP2GU1 53299144 IC50 > 100000 nM T69912 CCR5A9 56927662 IC50 = 59 nM T69912 CAG1J5 56927666 IC50 = 23 nM T69912 C6GKE8 56950525 IC50 = 16 nM T69912 C21HQB 57336782 IC50 = 3.4 nM T69912 C5WQ8S 57392555 IC50 = 96 nM T69912 CITS38 57394279 IC50 = 170 nM T69912 CR8GA1 57396026 IC50 = 31 nM T69912 CKN4Q7 57396027 IC50 = 55 nM T69912 C83CEW 57397828 IC50 = 64 nM T69912 CX65FQ 57397830 IC50 = 92 nM T69912 C89RKP 57397831 IC50 = 56 nM T69912 CN5L8A 57397832 IC50 = 91 nM T69912 CMBI04 57397833 IC50 = 2900 nM T69912 CK2C8H 57401254 IC50 = 61 nM T69912 CN9TM3 57401255 IC50 = 130 nM T69912 C4PC1W 57402997 IC50 = 4100 nM T69912 CF23GK 57402999 IC50 = 48 nM T69912 C5SE6Y 57403000 IC50 = 360 nM T69912 CLQ5P8 59900388 IC50 = 1 nM T69912 CL0FU7 63334771 IC50 = 100000 nM T69912 C59VAN 71181474 IC50 = 0.55 nM T69912 C13KJW 71181477 IC50 = 0.23 nM T69912 CI1Y9Z 71181626 IC50 = 1.6 nM T69912 CPXJ23 71181632 IC50 = 0.96 nM T69912 CML2I0 71181668 IC50 = 0.24 nM T69912 CU8YK1 71181747 IC50 = 1.72 nM T69912 C9B7MX 71181764 IC50 = 0.91 nM T69912 CO7K5M 71181859 IC50 = 0.46 nM T69912 C1FGZ5 71181861 IC50 = 0.81 nM T69912 CBG0P3 71181874 IC50 = 0.89 nM T69912 CO0W1H 71476859 IC50 = 0.14 nM T69912 CJPF24 71486715 IC50 = 0.86 nM T69912 C9DA6W 71562486 IC50 = 14000 nM T69912 C40WLD 71562487 IC50 = 230 nM T69912 C0N4SW 71562488 IC50 = 55 nM T69912 CS41XO 71562489 IC50 = 38 nM T69912 CB8E0O 71562597 IC50 = 370 nM T69912 CU02DS 71562598 IC50 = 86000 nM T69912 CX62RJ 71562599 IC50 = 820 nM T69912 CH5GA2 71562600 IC50 = 29000 nM T69912 C2XRB6 71562601 IC50 = 32 nM T69912 CL0KT3 71562602 IC50 = 9700 nM T69912 C6N7RZ 71562603 IC50 = 100 nM T69912 CT64JI 71562727 IC50 = 150 nM T69912 C8AOX0 71562728 IC50 = 150 nM T69912 CRX2Q4 71562729 IC50 = 16 nM T69912 CMWV34 71562730 IC50 = 70 nM T69912 CU4Z2Q 71562731 IC50 = 87 nM T69912 CJU1L8 71562732 IC50 = 44 nM T69912 CQ4AN0 71562733 IC50 = 240 nM T69912 CN15BR 71562848 IC50 = 3000 nM T69912 CY37JA 71562849 IC50 = 41000 nM T69912 C7APK1 71562850 IC50 = 31 nM T69912 CA1C8N 71562851 IC50 = 26 nM T69912 C4OBN3 71562852 IC50 = 13 nM T69912 C6PQG5 71562853 IC50 = 14 nM T69912 C50DMA 71562854 IC50 = 39 nM T69912 CCK65O 71562973 IC50 = 49 nM T69912 CUW2X3 71562974 IC50 = 52 nM T69912 CU2K4F 71562975 IC50 = 120 nM T69912 C1YI9V 71562976 IC50 = 250 nM T69912 C80IKC 71562977 IC50 = 450 nM T69912 CZEX42 71562978 IC50 = 100 nM T69912 C0TQ5W 71562979 IC50 = 39 nM T69912 CO8XE5 71563093 IC50 = 26 nM T69912 C71VWC 71563094 IC50 = 4 nM T69912 C42RMU 71563095 IC50 = 55 nM T69912 CQ39RC 71563096 IC50 = 28 nM T69912 CJU20T 71563097 IC50 = 3 nM T69912 CDJ92S 71563098 IC50 = 3 nM T69912 CUO97N 71563099 IC50 = 80 nM T69912 CC3LF8 71563229 IC50 = 22 nM T69912 C6G8OV 71614098 IC50 = 0.67 nM T69912 CPQ5H2 71614498 IC50 = 0.95 nM T69912 CYO64A 71656315 IC50 > 1000 nM T69912 C50OAM 71656796 IC50 = 210 nM T69912 C2TO5C 71656797 IC50 > 10000 nM T69912 CN89IX 71656798 IC50 = 93 nM T69912 C49OFR 71656799 IC50 = 26 nM T69912 C92YGU 71657082 IC50 = 5000 nM T69912 CV5PM2 71657185 IC50 = 10000 nM T69912 CPT0H5 71657290 IC50 = 10000 nM T69912 CM2ZB8 71657292 IC50 = 810 nM T69912 CBSW63 71657395 IC50 > 10000 nM T69912 CVUD47 71657398 IC50 > 10000 nM T69912 CV24SL 71716432 IC50 = 4 nM T69912 CTH15K 71717661 IC50 = 23 nM T69912 C1AYH2 71718263 IC50 = 32 nM T69912 CTPL54 71718264 IC50 > 100000 nM T69912 CS7WK3 74889411 IC50 > 100 nM T69912 C2KHF7 89677087 IC50 = 1400 nM T69912 CXT5C7 89682527 IC50 = 1500 nM T69912 CPF01Q 89682653 IC50 = 580 nM T69912 CY7PD2 89682704 IC50 = 930 nM T69912 CNU8L7 89682719 IC50 = 1800 nM T69912 C2JS9A 119057479 IC50 = 500000 nM T69912 CZL6P8 119057480 IC50 = 230 nM T69912 C1S6CA 119057481 IC50 = 2000 nM T69912 CV8MY3 119057482 IC50 = 1700 nM T69912 CGN2X5 119057483 IC50 = 230 nM T69912 CW6T2I 121005813 IC50 = 1.7 nM T69912 CL70DK 121448333 IC50 = 8.3 nM T69912 C3N6DK 121448334 IC50 = 1.8 nM T69912 CM4S9R 121448337 IC50 = 4.2 nM T69912 C9U7WD 121448368 IC50 = 1.6 nM T69912 CI86GD 121448372 IC50 = 1.9 nM T69912 C1A5GV 121448374 IC50 = 2.2 nM T69912 CKM5Z4 121448380 IC50 = 2.7 nM T69912 CW0V2U 121448402 IC50 = 4 nM T69912 CG9H1O 121448406 IC50 = 3.7 nM T69912 CRE5L4 121448411 IC50 = 2.2 nM T69912 CF65PJ 121448417 IC50 = 2.6 nM T69912 CX1LF9 121448418 IC50 = 8 nM T69912 C3OBQ9 121448429 IC50 = 4.6 nM T69912 CJ4F7G 121448430 IC50 = 1.2 nM T69912 CZM7L3 121448431 IC50 = 3.5 nM T69912 CSCG90 121448433 IC50 = 1.8 nM T69912 C8TVD7 121448459 IC50 = 1.1 nM T69912 COU74T 121448460 IC50 = 3.9 nM T69912 CIW92J 122196130 IC50 = 11.1 nM T69912 CY4XR8 122196132 IC50 = 10.6 nM T69912 CIY90U 122196137 IC50 = 19.3 nM T69912 C5AFS0 122196138 IC50 = 16 nM T69912 C32FMN 122196204 IC50 = 13.4 nM T69912 CJGP91 122196205 IC50 = 16.9 nM T69912 CKA4Y1 122196208 IC50 = 3.7 nM T69912 CCWJ26 122196209 IC50 = 2.9 nM T69912 C9WZI8 122196212 IC50 = 2.3 nM T69912 CEL90A 122196214 IC50 = 6.5 nM T69912 CQBA39 122196215 IC50 = 10.9 nM T69912 CI3CW8 122196216 IC50 = 6.3 nM T69912 C7JU5Q 122530045 IC50 = 6300 nM T69912 C5BW4Z 122707116 IC50 = 15000 nM T69912 CX92RI 122707117 IC50 = 1600 nM T69912 C23EKP 122707118 IC50 = 1000 nM T69912 CU95PT 122707120 IC50 = 32 nM T69912 CK05FL 127050954 IC50 = 3.6 nM T69912 C8TUI5 127050955 IC50 = 2.4 nM T69912 C7DA4S 127050956 IC50 = 18 nM T69912 C01RCH 127050977 IC50 = 30000 nM T69912 CJW7D2 127051244 IC50 = 560 nM T69912 C1GSK5 127053040 IC50 = 180 nM T69912 CRC6Z1 127053472 IC50 = 1.1 nM T69912 CU0D3S 130346049 IC50 = 1400 nM T69912 CH7EL8 132427687 IC50 = 14 nM T69912 CW74SC 134133758 IC50 = 75 nM T69912 CM5R6E 134135433 IC50 = 10000 nM T69912 CYXB84 134136689 IC50 = 39000 nM T69912 CM98WH 134137624 IC50 = 7900 nM T69912 C1SP0U 134138704 IC50 = 620 nM T69912 CJG9M7 134140857 IC50 = 1500 nM T69912 CP3HL5 134143019 IC50 = 860 nM T69912 CFQ13X 134144083 IC50 = 2700 nM T69912 C1GZ9U 134145078 IC50 = 2000 nM T69912 CUV5B0 134145387 IC50 = 5400 nM T69912 CSN0D4 134146496 IC50 = 1900 nM T69912 C5YD1G 134147073 IC50 = 6200 nM T69912 C8WF9X 134147739 IC50 = 20000 nM T69912 C69BXV 134148543 IC50 = 160 nM T69912 CCE7M2 134150004 IC50 = 0.3981 nM T69912 C36ZHN 134150110 IC50 = 11000 nM T69912 CXV2M9 134150242 IC50 = 4300 nM T69912 C58MQS 134152799 IC50 = 110 nM T69912 C8MA0Z 134153116 IC50 = 980 nM T69912 CZGB70 134154962 IC50 = 160 nM T69912 CA85UF 134155224 IC50 = 86 nM T69912 C16NSU 134155260 IC50 = 660 nM T69912 CHL74N 134156788 IC50 = 10000 nM T69912 CEW49V 134157408 IC50 = 72 nM T69912 C3SVZ5 134693749 IC50 = 355 nM T69912 C3DE5Y 134693750 IC50 = 5 nM T69912 CZ3F5D 135239539 IC50 = 844 nM T69912 C0U9TO 137546866 IC50 = 430 nM T69912 CH4MR3 137633945 IC50 = 902 nM T69912 CTD75A 137633962 IC50 = 9 nM T69912 CRCU09 137634263 IC50 = 236 nM T69912 CH05MV 137636050 IC50 = 613 nM T69912 CG3K6U 137637253 IC50 = 12 nM T69912 CMNT10 137638920 IC50 = 23 nM T69912 CK70BJ 137641309 IC50 = 42 nM T69912 C6LIG7 137642017 IC50 = 222 nM T69912 CZ3F7X 137642755 IC50 = 2477 nM T69912 CJP45C 137643198 IC50 = 924 nM T69912 CS4W0J 137643921 IC50 = 13 nM T69912 CA50JV 137645485 IC50 = 1027 nM T69912 C4F5GR 137647910 IC50 = 322 nM T69912 CFL68S 137649687 IC50 = 1070 nM T69912 CL61YI 137651817 IC50 = 152 nM T69912 CX3AJ9 137652098 IC50 = 17 nM T69912 CJ73YS 137654141 IC50 = 65 nM T69912 CSR0J2 137655061 IC50 = 57 nM T69912 CGBL78 137655982 IC50 = 232 nM T69912 CTU98S 137658155 IC50 = 100 nM T69912 C9X3WS 137658880 IC50 = 1915 nM T69912 CLVM39 137660910 IC50 = 45 nM T69912 C4JV2G 137661511 IC50 = 1418 nM T69912 CO67DI 137661556 IC50 = 45 nM T69912 CEQ7G4 155510849 IC50 > 10000 nM T69912 C9CD3Q 155511585 IC50 = 430 nM T69912 C25OAR 155512542 IC50 = 2000 nM T69912 CI2WL8 155513853 IC50 > 1000 nM T69912 CBG4Q8 155521008 IC50 > 1000 nM T69912 CL6Z1R 155526799 IC50 = 750 nM T69912 CW7N6K 155533489 IC50 = 1000 nM T69912 CQ67EK 155543660 IC50 = 1800 nM T69912 C8XZ7V 155545255 IC50 = 330 nM T69912 C9WGK1 155547201 IC50 = 1300 nM T69912 CH78YM 155549832 IC50 > 1000 nM T69912 C4U9WO 155550747 IC50 = 10000 nM T69912 D05LXG 5063 IC50 = 11000 nM T69912 D09QHC 7370 IC50 > 1000000 nM T69912 D0A1SO 11206881 IC50 = 3800 nM T69912 D0D7AS 11701397 IC50 = 11200 nM T69912 D0FO2B 1923 IC50 > 100000 nM T69912 D0JI8S 11470979 IC50 = 2000 nM T69912 D0WW7A 9939109 IC50 = 8 nM T69912 D0X6UV 11368513 IC50 = 4400 nM T89826 D04AIT 5280445 IC50 = 20000 nM T89826 D07EXH 359 IC50 > 200000 nM T89826 D07MGA 72281 IC50 = 8300 nM T89826 D0J9ZR 4477 IC50 = 40000 nM T89826 D0K8KX 5280343 IC50 = 8100 nM T89826 C5H9TY 14697 IC50 = 207000 nM T89826 C3I7VB 102678 IC50 = 24500 nM T89826 CL5Y4J 159516 Ki = 3100 nM T89826 CV0B7W 442027 IC50 = 49600 nM T89826 C1E2FR 442048 IC50 = 283500 nM T89826 CZ3MD8 647122 IC50 = 16100 nM T89826 C2C8QU 948801 Ki = 27500 nM T89826 CXA4P6 1265413 IC50 = 90720 nM T89826 CUD4A1 1328543 IC50 = 58350 nM T89826 C3ZP4U 2131972 Ki = 9110 nM T89826 CA1N3H 2131982 Ki = 9930 nM T89826 CKL8B2 2219105 IC50 = 29900 nM T89826 CN43XQ 2806068 IC50 = 160 nM T89826 C5J6MO 2849659 IC50 = 28800 nM T89826 CN3P7A 2911959 IC50 = 74500 nM T89826 CZDG23 2947583 IC50 = 186000 nM T89826 CBIP72 2986413 IC50 = 76700 nM T89826 CCU3P7 3635406 IC50 = 2200 nM T89826 CZF0R5 4004950 IC50 = 500 nM T89826 C3AN7C 4117477 IC50 = 1180 nM T89826 CS2WB7 4236803 IC50 = 29800 nM T89826 C0AW3N 4378077 IC50 = 13860 nM T89826 CO3Y0T 4614896 IC50 = 9910 nM T89826 CY68ZT 4788586 IC50 = 940 nM T89826 CTR4Q1 5320532 IC50 = 13300 nM T89826 CVG47I 5958938 IC50 = 10500 nM T89826 CD8ZT2 6026688 IC50 > 50000 nM T89826 C3LZX9 8027611 IC50 = 12660 nM T89826 CJ4C5K 9180583 IC50 = 10800 nM T89826 CYQ8Z4 9882716 IC50 > 50000 nM T89826 C8K2NO 10062715 IC50 = 800000 nM T89826 C49CMU 10411574 IC50 = 21700 nM T89826 C6GN2F 11642725 IC50 = 870000 nM T89826 CHYP53 12310492 IC50 = 233400 nM T89826 C65EOH 15949840 IC50 = 7500 nM T89826 C9V8EM 15956553 IC50 = 300000 nM T89826 C3WYR4 16061499 IC50 = 2000 nM T89826 CTO43V 16085283 Ki = 116000 nM T89826 CU35DQ 21582568 IC50 = 220800 nM T89826 CN45FL 23427055 IC50 = 164700 nM T89826 CK3AF8 25256829 IC50 = 5400 nM T89826 C2SZ7L 42624533 IC50 = 14000 nM T89826 CYP8V1 44404067 IC50 > 50000 nM T89826 CD20PF 44433696 IC50 = 80000 nM T89826 CI4P2V 44433697 IC50 = 10000 nM T89826 CW7B0J 44433698 IC50 = 15000 nM T89826 C8DWL3 44433699 IC50 = 200000 nM T89826 C0ZPE2 44517748 IC50 = 2700 nM T89826 C0OH2T 44584893 IC50 = 5400 nM T89826 C0NZ5E 44584944 IC50 = 7300 nM T89826 CT70DZ 44590821 IC50 = 22500 nM T89826 C0SW2K 45266425 IC50 = 2500 nM T89826 C5WBP2 45266482 IC50 = 3800 nM T89826 CA4K8F 45266488 IC50 = 6600 nM T89826 C3BHZ4 45268445 IC50 > 50000 nM T89826 CC05NI 45268452 IC50 = 15400 nM T89826 C6QD9E 45269292 IC50 > 50000 nM T89826 CY7RV4 45269761 Ki = 21000 nM T89826 CO80TH 45269762 Ki = 297000 nM T89826 CU34ZK 45269763 Ki = 584000 nM T89826 C9P3LZ 45269764 Ki = 478000 nM T89826 CXS19V 45269765 Ki = 45200 nM T89826 C3DY4T 45270971 IC50 > 50000 nM T89826 CR4WA8 45270979 IC50 = 20900 nM T89826 CM78GO 45271412 Ki = 462000 nM T89826 CC90BU 45271826 IC50 = 5200 nM T89826 C0B6KX 45271831 IC50 = 9300 nM T89826 CN85IQ 45271832 IC50 = 8100 nM T89826 C7IF2O 45272299 Ki = 363000 nM T89826 CZRV73 45272304 Ki = 34100 nM T89826 CGV14L 45272305 Ki = 112000 nM T89826 CVTL97 45272306 Ki = 2200 nM T89826 CAM89I 45273174 Ki = 135000 nM T89826 CZT67B 45273179 Ki = 614000 nM T89826 CHF4M5 45273180 Ki = 49300 nM T89826 CND1R3 45273184 Ki = 159000 nM T89826 C0V5WT 45273625 IC50 > 50000 nM T89826 C6OE7V 46784066 IC50 = 28300 nM T89826 C6LH5I 46881919 Ki = 800 nM T89826 CI2FO1 49870840 IC50 = 5500 nM T89826 CF2D0I 49870841 IC50 = 8400 nM T89826 CM52SZ 49870842 IC50 = 6800 nM T89826 C8Q2CZ 50885062 IC50 > 50000 nM T89826 CJ6KV7 52941131 IC50 = 13900 nM T89826 C8M2QD 52943127 IC50 = 24300 nM T89826 CQ84MD 52945913 IC50 = 12000 nM T89826 CJ1LG2 52945915 IC50 = 42000 nM T89826 CZ35DX 52945977 IC50 = 128900 nM T89826 CAB1Y3 52946772 IC50 = 163200 nM T89826 CO4R1B 52947200 IC50 = 18000 nM T89826 CC4X1O 52948928 IC50 = 137700 nM T89826 CMG4U7 52949213 IC50 = 10800 nM T89826 C0X5BL 58589722 IC50 = 76740 nM T89826 CY3CL6 71544384 IC50 = 610 nM T89826 CV3P2U 71544385 IC50 = 230 nM T89826 CJS60O 71571220 IC50 = 49000 nM T89826 C1AY0M 71571221 IC50 = 49000 nM T89826 CY21XB 71571222 IC50 = 4600 nM T89826 C1DX9H 71571223 IC50 = 39000 nM T89826 CKE2C3 73056463 IC50 > 100000 nM T89826 C9S8ZH 73056464 IC50 > 100000 nM T89826 CK9OI0 73056465 IC50 = 31710 nM T89826 C4D8LK 73056466 IC50 = 32080 nM T89826 CRY86G 73056467 IC50 = 34910 nM T89826 C3VS4F 73056760 IC50 = 10070 nM T89826 CYH1F4 73056761 IC50 = 51330 nM T89826 C2CRZ8 73056762 IC50 = 2250 nM T89826 CD4YR3 73056763 IC50 = 11830 nM T89826 C3P2OZ 73056764 IC50 = 67200 nM T89826 C1H8PX 73056765 IC50 = 82910 nM T89826 C8JO7B 73056766 IC50 = 13860 nM T89826 CCYE63 73057087 IC50 = 5520 nM T89826 C54JWM 73057088 IC50 = 39870 nM T89826 C8RBU6 73057089 IC50 = 1040 nM T89826 CEBH65 73057090 IC50 = 1690 nM T89826 C8M2DX 73057091 IC50 = 17820 nM T89826 CQ42AZ 73057092 IC50 = 2820 nM T89826 CPLJ64 73057388 IC50 = 4700 nM T89826 CIN5V0 76320984 IC50 = 4300 nM T89826 C05AYV 102341658 IC50 = 16400 nM T89826 C8S3CR 102341659 IC50 = 37500 nM T89826 C2G9CP 127043455 IC50 = 20200 nM T89826 CVZ4I3 127043641 IC50 = 6000 nM T89826 C7BST4 127043642 IC50 = 5800 nM T89826 CGO01F 127043643 IC50 > 50000 nM T89826 C2TU5A 127043644 IC50 = 6400 nM T89826 C0Y9IT 127043645 IC50 = 41200 nM T89826 CF3B1Z 127045220 IC50 = 11700 nM T89826 CIXJ94 127045221 IC50 = 8600 nM T89826 CQ1CT5 127045222 IC50 = 18700 nM T89826 CKRX04 127045227 IC50 = 30700 nM T89826 CDZ2E1 127045228 IC50 > 50000 nM T89826 CG3E9B 127045229 IC50 = 6700 nM T89826 CG6VR3 127045386 IC50 = 15700 nM T89826 CK9JE3 127045387 IC50 > 50000 nM T89826 CY1E4Z 127045392 IC50 > 50000 nM T89826 CK5PA4 127045393 IC50 = 44700 nM T89826 C34TWD 127045394 IC50 > 50000 nM T89826 C97MQC 127048409 IC50 = 20000 nM T89826 C41VRM 127048410 IC50 = 7500 nM T89826 CZ0B1R 127052510 IC50 = 10000 nM T89826 CRW05E 127052511 IC50 > 50000 nM T89826 CC3TX0 127052512 Ki = 72000 nM T89826 CIQ1U9 127052513 Ki = 41000 nM T89826 CI13JZ 135452883 IC50 = 10000 nM T89826 CG1KW5 135470831 IC50 = 77090 nM T89826 CH4Q6A 145964401 IC50 = 5500 nM T89826 CHU61S 145964420 IC50 = 42100 nM T89826 C6YCA8 145964710 IC50 = 28800 nM T89826 CV6F7L 145966788 IC50 = 2100 nM T89826 CBWX17 145967285 IC50 = 4300 nM T89826 COR9X3 145972736 IC50 = 3900 nM T89826 CQ0M2X 145972809 IC50 = 4100 nM T89826 CF95RZ 145972878 IC50 = 3200 nM T89826 CXI0D1 145975081 IC50 = 6300 nM T89826 CG84ZR 145975487 IC50 = 5100 nM T89826 C91FOT 145976006 IC50 = 5200 nM T89826 C3F4UH 145978039 IC50 = 8800 nM T89826 CL7FB0 2919450 IC50 = 62790 nM T89826 D00RIX 5280443 IC50 = 280800 nM T89826 D01XMM 4117383 IC50 = 4450 nM T89826 D08MZY 145937 Ki = 8200 nM T89826 D08UYP 3008868 Ki = 2400 nM T89826 D09BUG 10207 IC50 = 132000 nM T89826 D0L7AT 10480940 Ki = 19300 nM T89826 D0S0BN 130976 Ki = 10600 nM T89826 D0SY2M 5281708 IC50 = 105000 nM T89826 D0UQ6U 10569 IC50 = 189100 nM T89826 D0WA9S 10429214 IC50 = 146500 nM T90961 C3VRO9 44557921 IC50 > 10000 nM T90961 C67OJG 44588117 Ki = 4400 nM T90961 C4YWO9 134812845 Ki = 17 nM T90961 CG15PY 134812846 Ki > 100000 nM T90961 C9O8CQ 137348448 Ki = 13 nM T90961 C63TGO 137349551 Ki = 17 nM T90961 C6I5ME 137349552 Ki = 19 nM T90961 CRC8D2 155489850 Ki = 95000 nM T90961 CG8J5X 155518911 Ki = 27 nM T90961 CAN08J 155534113 Ki = 36 nM T90961 C16JRL 155535406 Ki = 74 nM T90961 C3XR8O 155536206 Ki = 51 nM T90961 CX68YN 155541385 Ki > 100000 nM T90961 CWU67H 155543077 Ki = 59 nM T90961 CD8K3O 155543384 Ki = 42 nM T90961 CUTW39 155546618 Ki = 20 nM T90961 C4E0HB 155546757 Ki = 120 nM T90961 C49UVQ 155547733 Ki = 17 nM T90961 CI2J4O 155551330 Ki = 37 nM T90961 CP2K8O 155554487 Ki = 30 nM T90961 CS8MC1 155562025 Ki = 33 nM T90961 C8UW4P 155562878 Ki = 17 nM T90961 CDP94M 155569521 Ki = 53 nM T88806 D0BN9X 60947 IC50 > 300000 nM T88806 D01TJY 53340771 IC50 = 7.7 nM T88806 D09ZXO 176873 IC50 = 13.2 nM T88806 D0Q5LF 9961766 IC50 > 100000 nM T88806 D08LIG 153986 IC50 > 3 nM T88806 D0P8JX 177831 IC50 > 5 nM T88806 C7CL3Y 107775 IC50 = 2200 nM T88806 CE19HD 132605 IC50 = 27000 nM T88806 CDOC86 303776 IC50 > 1000 nM T88806 C4U0BM 1878893 IC50 > 20000 nM T88806 C2E9ZX 3080994 IC50 = 1546000 nM T88806 C42AWQ 3797164 IC50 = 20500 nM T88806 CI51MD 9807891 IC50 > 500000 nM T88806 C68UYS 9808123 IC50 = 64 nM T88806 CK6A0I 9808598 IC50 > 500000 nM T88806 CB8GP1 9828375 IC50 = 26 nM T88806 CJ9HV0 9828819 IC50 = 20 nM T88806 C1OP9I 9828979 EC50 > 100000 nM T88806 C87ADQ 9830626 IC50 = 421 nM T88806 C13KPA 9848051 Ki < 10000 nM T88806 C04PAT 9849697 IC50 > 500000 nM T88806 CTM7V0 9851337 IC50 = 316 nM T88806 C2XD7P 9851886 IC50 > 100000 nM T88806 CN1R0K 9852055 IC50 > 500000 nM T88806 CR38MP 9853559 IC50 = 2200 nM T88806 C6E3OL 9863046 IC50 > 100000 nM T88806 C2ZAK6 9870468 IC50 > 800000 nM T88806 CHC56Q 9870640 IC50 = 640 nM T88806 C5EJN9 9884317 IC50 > 20000 nM T88806 CV4T6H 9885053 IC50 = 7800 nM T88806 CME97S 9894966 IC50 = 930 nM T88806 C04INH 9895205 IC50 > 100000 nM T88806 CNX29T 9907082 IC50 = 70000 nM T88806 C9QN4D 9919094 IC50 = 1100000 nM T88806 CF4J2Z 9923982 IC50 = 15000 nM T88806 CUBV32 9924032 IC50 > 20000 nM T88806 CCPD70 9927009 IC50 = 180000 nM T88806 CDU79H 9957105 IC50 = 95 nM T88806 C2R7TW 10069591 IC50 > 500000 nM T88806 C71AIN 10077862 IC50 > 30000 nM T88806 CO8D9C 10196873 IC50 = 133 nM T88806 C7U5CM 10336795 IC50 = 8000 nM T88806 C0IA8K 10455265 IC50 > 450000 nM T88806 CTZC60 10461016 IC50 > 100000 nM T88806 CY1JM2 11024622 IC50 = 1300000 nM T88806 CZO3H7 11399588 IC50 = 3.7 nM T88806 CX9G5B 11534748 IC50 = 25 nM T88806 CFZ2O9 11613998 IC50 = 1.6 nM T88806 CD87UQ 11627754 IC50 = 286 nM T88806 CXA2U4 11671832 IC50 = 670 nM T88806 CWU71P 11699824 IC50 = 15 nM T88806 CGU84F 11721315 IC50 = 1.7 nM T88806 C2ONX6 11721442 IC50 = 6 nM T88806 CT4D1K 11799915 IC50 > 100000 nM T88806 CS24BW 11973730 IC50 > 10000 nM T88806 CZTJ02 12795460 EC50 = 1031 nM T88806 CW41XZ 16663331 IC50 > 10000 nM T88806 CDUC32 16665100 IC50 = 2.5 nM T88806 CTGC60 16678135 IC50 = 2.3 nM T88806 C4T7ZE 16724119 IC50 = 1500 nM T88806 CU8YQ3 16756502 IC50 = 1.1 nM T88806 C9LF8T 16756503 IC50 = 445 nM T88806 CJUK37 16756504 IC50 = 155 nM T88806 C0KW3V 16756505 IC50 = 3.5 nM T88806 C04JOX 16756621 IC50 = 0.54 nM T88806 C4CU7T 16756622 IC50 = 0.55 nM T88806 CFH96E 16756623 IC50 = 0.8 nM T88806 CXK79J 16756847 IC50 = 231 nM T88806 CB15RX 16756849 IC50 = 86 nM T88806 CM18ZN 16756955 IC50 = 1.4 nM T88806 CL38IU 16756956 IC50 = 0.9 nM T88806 CW5P8L 16756957 IC50 = 0.55 nM T88806 CX6AR9 23627460 IC50 = 2 nM T88806 CAVY89 23636144 IC50 > 10000 nM T88806 C1VUH4 23636254 IC50 > 10000 nM T88806 C6LR7V 23636255 IC50 > 10000 nM T88806 C5MSF6 23636502 IC50 > 10000 nM T88806 CYND24 23729562 IC50 > 20000 nM T88806 C96PUZ 23729563 IC50 > 20000 nM T88806 CZ17YE 23731146 IC50 = 3900 nM T88806 CHXT18 23731243 IC50 = 4300 nM T88806 CEA9Z8 23731244 IC50 = 1200 nM T88806 CNK5O6 23731245 IC50 > 20000 nM T88806 C6W9OS 23731246 IC50 = 20000 nM T88806 C79OBD 24864541 IC50 = 82 nM T88806 CR72IF 24864718 IC50 = 11 nM T88806 CFRX87 24864719 IC50 = 710 nM T88806 C9L0QD 24864721 IC50 < 1 nM T88806 CXH2G0 24864898 IC50 < 1 nM T88806 CF23RY 24865076 IC50 = 8 nM T88806 CO3I0M 24865264 IC50 = 69 nM T88806 CPD30N 24865443 IC50 = 480 nM T88806 C17IUE 24865620 IC50 = 8 nM T88806 C7TPO5 24865624 IC50 = 2 nM T88806 C5DVB6 24865625 IC50 = 3 nM T88806 C5DYT6 24865999 IC50 = 24 nM T88806 C5JB3F 24866187 IC50 = 220 nM T88806 C8G2FE 24866358 IC50 = 2 nM T88806 C6I1OF 24866515 IC50 < 1 nM T88806 CZ7QL8 24866516 IC50 = 90 nM T88806 CNCH18 24866519 IC50 = 3 nM T88806 CY6WR2 24872066 IC50 = 2.1 nM T88806 CUM4E3 24872070 IC50 = 2 nM T88806 CG09DH 24872646 IC50 = 1.6 nM T88806 CRS65Q 24873110 IC50 = 2.2 nM T88806 C0HZ7E 24873345 IC50 = 2.7 nM T88806 C28KAH 24873465 IC50 = 43 nM T88806 C1PB6T 25025343 IC50 = 12 nM T88806 CDA2B9 25025730 IC50 = 130 nM T88806 CD2L7Z 25025937 IC50 < 1 nM T88806 C43TCR 25183860 IC50 = 5 nM T88806 CR92LD 25184415 IC50 = 7 nM T88806 C3J7GQ 28510125 IC50 = 136 nM T88806 CLX6T9 28510811 IC50 > 1000 nM T88806 C2SLU4 44286634 IC50 = 3100000 nM T88806 C7B6FS 44286652 IC50 = 65000 nM T88806 C47DUX 44320508 IC50 = 1000000 nM T88806 CX46NY 44343237 IC50 = 6100 nM T88806 C08QPE 44350169 IC50 = 3000 nM T88806 CELV48 44350342 IC50 = 0.18 nM T88806 CP4R1A 44350344 IC50 = 230 nM T88806 C14OBS 44350379 IC50 = 2700 nM T88806 CDE56C 44350392 IC50 = 18 nM T88806 C0W9CT 44350404 IC50 = 1500 nM T88806 CEP6G1 44350415 IC50 = 0.39 nM T88806 CR83VC 44350419 IC50 = 670 nM T88806 CX3MK8 44350425 IC50 = 4700 nM T88806 C4U0XW 44350427 IC50 = 310 nM T88806 CJ47ZT 44350428 IC50 = 13 nM T88806 CX09AV 44350435 IC50 = 1800 nM T88806 CX28UF 44350441 IC50 = 170 nM T88806 C7J9NH 44350447 IC50 = 21 nM T88806 CH6UX8 44350448 IC50 = 14 nM T88806 C4C2PF 44350449 IC50 = 39 nM T88806 CP4TD3 44350450 IC50 = 1.4 nM T88806 CR51ID 44378699 IC50 = 6000 nM T88806 CAO29R 44378701 IC50 = 100 nM T88806 CWP41H 44378720 IC50 = 4300 nM T88806 C2U6ZA 44378747 IC50 = 2100 nM T88806 CT9H2B 44378748 IC50 = 4500 nM T88806 CNS75M 44378858 IC50 = 830 nM T88806 CENU52 44378961 IC50 = 4300 nM T88806 C3UQT1 44378995 IC50 = 1560 nM T88806 CHC7N5 44379066 IC50 = 1200 nM T88806 CVYB52 44393453 IC50 > 20000 nM T88806 CAD12L 44393517 IC50 > 1000 nM T88806 C6G7RF 44436701 IC50 > 1000000 nM T88806 CZ1L9O 44436703 IC50 > 1000000 nM T88806 C7CAJ3 44436705 IC50 > 1000000 nM T88806 CR6XE2 44436707 IC50 = 18 nM T88806 CYOC34 44436708 IC50 > 1000000 nM T88806 CSF3V2 44436709 IC50 > 1000000 nM T88806 C67VHW 44436710 IC50 > 1000000 nM T88806 CBW09N 44436711 IC50 > 1000000 nM T88806 CRNQ31 44436712 IC50 > 1000000 nM T88806 C1YMJ2 44436713 IC50 = 170 nM T88806 CF4UR2 44436714 IC50 > 1000000 nM T88806 C52DMG 44436715 IC50 > 1000000 nM T88806 CLU84X 44436716 IC50 = 35100 nM T88806 CRO80K 44436717 IC50 = 57 nM T88806 CVGW76 44549110 IC50 = 0.3 nM T88806 CWL7J1 44549224 IC50 = 0.7 nM T88806 CO8EM6 44550577 IC50 = 0.1 nM T88806 CX1C4T 44552445 IC50 = 151.6 nM T88806 CCFW92 44605870 IC50 = 220 nM T88806 CM9VI1 44626482 IC50 = 1300 nM T88806 CBO95I 44626483 IC50 > 100000 nM T88806 CS36GK 44627949 IC50 = 520 nM T88806 CX6LM3 44628051 IC50 = 24 nM T88806 CVTO84 44628052 IC50 = 4700 nM T88806 CJQ37N 44628053 IC50 > 100000 nM T88806 CV4P3J 44628054 IC50 > 100000 nM T88806 CTU9W0 44628055 IC50 > 100000 nM T88806 C89ZFA 46224777 IC50 = 0.92 nM T88806 C5X1NZ 46224858 IC50 = 0.9 nM T88806 CDG6B1 46224859 IC50 = 351 nM T88806 CKM2X1 46224860 IC50 = 70 nM T88806 CL39GY 46224861 IC50 = 234 nM T88806 C56PVC 46226894 IC50 = 1.6 nM T88806 CVXH79 46226896 IC50 = 1.6 nM T88806 CBKZ57 46226897 IC50 = 1.5 nM T88806 C30JXH 46226899 IC50 = 13 nM T88806 C2WHK1 46226900 IC50 = 46 nM T88806 C5H9YT 46226901 IC50 = 65 nM T88806 CV8W7P 46226902 IC50 = 887 nM T88806 C83EWD 46226903 IC50 = 79 nM T88806 CRVU54 46226904 IC50 = 87 nM T88806 CE85AX 46226905 IC50 = 6.1 nM T88806 CP7U9T 50907449 IC50 = 19 nM T88806 CK7ZI0 56838719 IC50 = 1050 nM T88806 CG2NY0 57819421 IC50 = 466 nM T88806 CEG3V7 59665282 IC50 = 5900 nM T88806 C5MA9U 59665328 IC50 < 41 nM T88806 CR71ZG 59665343 IC50 = 150 nM T88806 CJ84CU 59665347 IC50 = 83 nM T88806 CTP16I 59665394 IC50 = 76 nM T88806 C5DJB3 59665402 IC50 = 140 nM T88806 C60EVZ 59665407 IC50 = 3 nM T88806 C4UH8X 59665418 IC50 = 6 nM T88806 C5RDW1 59665480 IC50 < 1 nM T88806 CSRE10 59665495 IC50 = 49 nM T88806 C1C0UT 68898764 IC50 = 21 nM T88806 CN93KB 68898863 IC50 = 39 nM T88806 CD10PM 68899361 IC50 = 9 nM T88806 CBF0K8 68899684 IC50 = 1900 nM T88806 C9LB1Y 68900219 IC50 = 1 nM T88806 C74UPO 68900657 IC50 = 9 nM T88806 CD4N6F 68901257 IC50 = 180 nM T88806 CK8UT9 68901290 IC50 = 110 nM T88806 CF4BZ9 68901306 IC50 = 1 nM T88806 CI0AL7 69244056 IC50 = 4 nM T88806 C31IUF 69863577 IC50 = 2807 nM T88806 CPF6S0 70681588 IC50 = 890 nM T88806 CQ4G2O 70683715 IC50 = 5 nM T88806 CVCJ03 70687988 IC50 = 2200 nM T88806 CX73MA 70689988 IC50 = 130 nM T88806 C92FXR 70690012 IC50 = 150 nM T88806 CPA07E 70694227 IC50 = 360 nM T88806 C8NZ7A 70694228 IC50 = 1 nM T88806 CM2AD4 70696326 IC50 < 1 nM T88806 C48NIF 70696327 IC50 = 970 nM T88806 CGMR28 71450831 IC50 = 1200 nM T88806 C8EM7Y 71550913 IC50 = 126.5 nM T88806 CY1MD5 71574157 IC50 = 7.3 nM T88806 C02ZBI 71574158 IC50 = 111 nM T88806 C16JKI 71574159 IC50 = 7 nM T88806 CU95LC 71574160 IC50 = 94 nM T88806 COJ8Y4 71574161 IC50 = 8.7 nM T88806 C5SG9H 71574261 IC50 = 115 nM T88806 C3C9QK 71574262 IC50 = 92 nM T88806 CTZU49 71574263 IC50 = 11 nM T88806 C4HB7F 71574264 IC50 = 39 nM T88806 C3S9QJ 71574355 IC50 = 72 nM T88806 C8V4UB 71574356 IC50 = 5.5 nM T88806 CX0SQ1 71574452 IC50 = 8.7 nM T88806 C1QE0K 71716365 IC50 = 197 nM T88806 CFYM81 71720633 IC50 = 27 nM T88806 CA9K6E 72204688 IC50 = 19 nM T88806 CLC7R0 72204689 IC50 = 9800 nM T88806 CCW43J 72204873 IC50 = 2100 nM T88806 CQ6TF8 72204875 IC50 = 9800 nM T88806 CC49AN 72204878 IC50 > 100000 nM T88806 C0N3SX 72205060 IC50 = 170 nM T88806 CZ2P8U 73345565 IC50 = 6600 nM T88806 CQAE56 73345568 IC50 > 10000 nM T88806 CU1VZ5 73345570 IC50 = 6400 nM T88806 CPT7S8 73345576 IC50 > 10000 nM T88806 C4P3JC 73346588 IC50 = 3650 nM T88806 CZ6Y9R 73347081 IC50 = 4190 nM T88806 CZ35TD 73347085 IC50 = 440 nM T88806 CGM9F7 73347087 IC50 = 7720 nM T88806 C89ENA 73347090 IC50 = 6800 nM T88806 CN1A2D 73347092 IC50 = 5190 nM T88806 CO9L2V 73348591 IC50 = 6240 nM T88806 C43LWV 73348592 IC50 = 1810 nM T88806 CM37AE 73348593 IC50 = 7200 nM T88806 C5BQ6R 73349139 IC50 = 57 nM T88806 CQ5D7B 73350175 IC50 = 870 nM T88806 CJEH13 73350177 IC50 = 6800 nM T88806 C20AJB 73350179 IC50 = 10000 nM T88806 C19PJE 73350181 IC50 = 4790 nM T88806 C2F3YZ 73351673 IC50 = 9200 nM T88806 CJA25I 73351674 IC50 = 2300 nM T88806 C6NCQ1 73351675 IC50 = 440 nM T88806 C46ULG 73351676 IC50 = 10000 nM T88806 C8B6NV 73351677 IC50 = 5100 nM T88806 CIYV49 73351678 IC50 = 1500 nM T88806 C20FGN 73353141 IC50 = 8700 nM T88806 CP6AJ3 73353143 IC50 = 8500 nM T88806 CUPR57 73353147 IC50 = 1200 nM T88806 C83RAM 73353150 IC50 = 8200 nM T88806 CAJ27W 73354663 IC50 = 7720 nM T88806 CT4A5S 73354664 IC50 = 4700 nM T88806 C6XTP9 73354667 IC50 > 10000 nM T88806 CZ1BL4 73354668 IC50 = 1230 nM T88806 C4EJK0 73356213 IC50 = 980 nM T88806 CH8G5C 73356216 IC50 > 10000 nM T88806 CPG36Q 73356217 IC50 = 6000 nM T88806 CD1S3N 73356221 IC50 = 840 nM T88806 C5ALQ2 76285468 IC50 = 74 nM T88806 CI07FE 90645591 IC50 = 66000 nM T88806 C8N6OE 90654504 IC50 = 108 nM T88806 C8TWH9 90654505 IC50 > 10000 nM T88806 CDVB75 90654506 IC50 > 10000 nM T88806 C5HG9N 90654507 IC50 = 64.2 nM T88806 CLCN89 117977916 IC50 = 63 nM T88806 CJO3B6 117978172 IC50 > 10000 nM T88806 C7ANO1 118709464 IC50 = 0.39 nM T88806 CY1IS6 118718872 IC50 = 10000 nM T88806 CV7DK0 122181680 IC50 > 1000 nM T88806 CWY3V2 122181682 IC50 > 1000 nM T88806 CRG07Q 124155531 IC50 > 10000 nM T88806 C69XPN 124163720 IC50 > 10000 nM T88806 C4R3BT 124163838 IC50 = 3200 nM T88806 CS2QR4 124163840 IC50 = 3200 nM T88806 C93HFX 127025140 IC50 = 15 nM T88806 CEU4X3 127025441 IC50 = 26 nM T88806 CTX71B 127025442 IC50 = 1500 nM T88806 C21ACR 133633869 IC50 > 1000 nM T88806 CPU86F 135438774 IC50 > 20000 nM T88806 C3JVT0 136152923 IC50 > 20000 nM T88806 C85WBP 137634338 IC50 = 95.8 nM T88806 C4IX7Z 137649002 IC50 = 30.7 nM T88806 C6NVW5 137652892 IC50 = 101.3 nM T88806 C0X8ER 145949722 IC50 = 20 nM T88806 C2MO7K 145951845 IC50 = 13 nM T88806 CG80FB 145951878 IC50 = 48 nM T88806 C1P0NL 145952828 IC50 = 22 nM T88806 CJA7N9 145953608 IC50 = 41 nM T88806 CZ4SK6 145954275 IC50 = 18 nM T88806 CTA08K 145956036 IC50 = 76 nM T88806 CY5I1O 145956101 IC50 = 45 nM T88806 C8RAG3 145956154 IC50 = 36 nM T88806 CCB51L 145956802 IC50 = 40 nM T88806 CTS5R3 145959048 IC50 = 28 nM T88806 CQ4ET5 145959752 IC50 = 31 nM T88806 CO0W4J 145961652 IC50 = 22 nM T88806 C23HZY 145971531 IC50 = 22 nM T88806 C75GFR 154734316 IC50 = 158 nM T88806 CR9DN2 154734318 EC50 = 9.9 nM T88806 C8ZUJ5 154734319 IC50 = 41.5 nM T88806 C17RZG 155515221 IC50 = 547 nM T88806 CHT1J6 155515540 IC50 = 72.9 nM T88806 CQ5C4M 155516533 IC50 = 689 nM T88806 CQNC74 155517321 IC50 > 10000 nM T88806 CRIA18 155519034 IC50 > 10000 nM T88806 C3S2YZ 155519712 IC50 = 563 nM T88806 CZY8F6 155520344 IC50 = 325 nM T88806 C9HB1M 155526953 IC50 = 5669 nM T88806 C2GJ5V 155527654 IC50 = 835 nM T88806 CQ1G0D 155528127 IC50 = 419 nM T88806 C2GSD7 155528224 IC50 = 3660 nM T88806 CPIL79 155528977 IC50 = 2722 nM T88806 C58JIQ 155530986 IC50 = 1.92 nM T88806 CJZU81 155532583 IC50 = 9287 nM T88806 C9T6SE 155533508 IC50 = 983 nM T88806 CJ7O2X 155534687 IC50 > 1000 nM T88806 C6TCP5 155546837 IC50 = 409 nM T88806 C6D2SM 155550380 IC50 > 10000 nM T88806 CWF98D 155552156 IC50 > 1000 nM T88806 CC64PJ 155561080 IC50 = 8029 nM T88806 C80PGY 155563043 IC50 = 5944 nM T88806 CEF3T8 155563936 IC50 = 38.4 nM T88806 C0SZJ1 155564443 IC50 = 1110 nM T88806 C98UME 155566748 IC50 = 2161 nM T88806 CY8S2L 155569251 IC50 = 11.9 nM T88806 C9NH4F 155569254 IC50 = 154 nM T88806 CZ9D2V 90645090 EC50 = 12 nM T88806 CWA6N4 90645092 EC50 = 763 nM T88806 CA8W7Q 90645094 EC50 = 365 nM T88806 D01AXA 11764797 IC50 = 259000 nM T88806 D06LUT 44379110 IC50 = 3440 nM T88806 D07WDB 104802 IC50 = 830000 nM T88806 D0A0KS 9851104 IC50 = 34700 nM T88806 D0B4JU 15409414 IC50 = 740 nM T20251 D00FGR 3599 IC50 > 100000 nM T20251 D00JAU 3749 IC50 = 194984.46 nM T20251 D00JVR 2267 IC50 = 100 nM T20251 D00KHM 16362 IC50 = 3.02 nM T20251 D00PEH 135449332 IC50 = 630.96 nM T20251 D00SBN 4746 IC50 = 7762.47 nM T20251 D00STL 644241 IC50 = 125.89 nM T20251 D00UVA 11556711 IC50 = 92100 nM T20251 D00UYE 4058 IC50 = 323.59 nM T20251 D00YLW 3033818 IC50 = 6025.6 nM T20251 D01AXB 60835 IC50 = 10000 nM T20251 D01AZG 5073 IC50 = 148 nM T20251 D01FGR 3100 IC50 = 2570.4 nM T20251 D01KPV 3348 IC50 = 21379.62 nM T20251 D01UTL 2995 IC50 = 1380.38 nM T20251 D01ZII 2726 IC50 = 1470 nM T20251 D01ZSO 4235 IC50 = 79432.82 nM T20251 D02EYG 10096344 IC50 > 30000 nM T20251 D02KOF 3948 IC50 = 2398832.92 nM T20251 D02MLW 60753 IC50 = 20 nM T20251 D02YIZ 12560 IC50 = 39 nM T20251 D03CJL 3168 IC50 = 32.2 nM T20251 D03CQE 5379 IC50 = 128824.96 nM T20251 D03DAP 3356 IC50 = 3890.45 nM T20251 D03DIG 5284371 IC50 = 301995.17 nM T20251 D03FLC 3878 IC50 = 251188.64 nM T20251 D03HFG 5324346 IC50 = 3100 nM T20251 D03IGH 213039 IC50 = 100000 nM T20251 D03MIR 3157 IC50 = 588.84 nM T20251 D03NHW 4583 IC50 = 1412537.54 nM T20251 D03QWT 73303 IC50 = 5011872.34 nM T20251 D04AAN 4078 IC50 = 320 nM T20251 D04CRN 54841 IC50 = 2100 nM T20251 D04FVU 6337614 IC50 = 1995.26 nM T20251 D04JCN 47811 IC50 = 120.23 nM T20251 D04JEE 4946 IC50 = 2828 nM T20251 D04LVK 57379345 IC50 = 1250 nM T20251 D04MSM 2554 IC50 = 104712.85 nM T20251 D04OSE 4485 IC50 = 50118.72 nM T20251 D04XGT 31593 IC50 > 100000 nM T20251 D04XPW 446220 IC50 = 4.4 nM T20251 D05CPV 208898 IC50 = 3000 nM T20251 D05EAM 4735 IC50 = 18800 nM T20251 D05LYX 3488 IC50 = 74000 nM T20251 D05MQK 110635 IC50 = 79432.82 nM T20251 D05OFX 219078 IC50 = 50118723.36 nM T20251 D05PIZ 15130 IC50 = 2187.76 nM T20251 D05SBO 46220502 IC50 = 10900 nM T20251 D05XGO 11154555 IC50 = 20720 nM T20251 D06ABF 3957 IC50 = 169.82 nM T20251 D06BCB 443955 IC50 = 39 nM T20251 D06GKN 2099 IC50 = 3235.94 nM T20251 D06MAJ 65906 IC50 = 350 nM T20251 D06MQM 6437380 IC50 = 8100 nM T20251 D06PZN 119584 IC50 = 4800 nM T20251 D06ZUK 3696 IC50 = 3388.44 nM T20251 D07KSG 2733526 IC50 = 1584.89 nM T20251 D07MVK 37393 IC50 = 40 nM T20251 D08CDI 208908 IC50 = 630957.34 nM T20251 D08JZS 4992 IC50 = 1100 nM T20251 D08VXO 6834 IC50 = 891.25 nM T20251 D08YIN 1727 IC50 = 4400000 nM T20251 D09EGZ 2719 IC50 = 2500 nM T20251 D09GOS 2812 IC50 = 3019.95 nM T20251 D09HNR 3002190 IC50 = 40000 nM T20251 D09KTS 24821094 Ki = 1100 nM T20251 D09MWJ 2092 IC50 = 125892.54 nM T20251 D09OJQ 4095 IC50 = 9772.37 nM T20251 D09QUQ 92253 IC50 = 20892.96 nM T20251 D09SGV 25154714 IC50 = 29200 nM T20251 D0AO5H 5578 IC50 = 239883.29 nM T20251 D0AR3J 439501 IC50 = 5800 nM T20251 D0AV3G 3151 IC50 = 162 nM T20251 D0B3UJ 115237 IC50 = 1000 nM T20251 D0B5LF 448042 Ki = 79432.82 nM T20251 D0B7NG 2725 IC50 = 1100 nM T20251 D0BD8D 6917698 IC50 = 12 nM T20251 D0BP9C 193962 IC50 = 25118.86 nM T20251 D0BZ7W 443879 IC50 = 125.89 nM T20251 D0C3SW 53465279 IC50 > 30000 nM T20251 D0C9SY 135400189 IC50 = 79432.82 nM T20251 D0CL9S 159269 IC50 = 5011872.34 nM T20251 D0CS2F 3955 IC50 = 33 nM T20251 D0D1AL 3559 IC50 = 10 nM T20251 D0D7KC 5488548 IC50 = 63095734.45 nM T20251 D0D9FV 4601 IC50 = 851.14 nM T20251 D0DK8V 2678 IC50 = 30199.52 nM T20251 D0DV3O 3241 IC50 = 100000 nM T20251 D0E1WI 3345 IC50 = 1819.7 nM T20251 D0E4DW 1775 IC50 = 100000 nM T20251 D0E6XR 3062316 IC50 = 15848.93 nM T20251 D0E7PQ 5311 IC50 > 30000 nM T20251 D0F0YZ 4737 IC50 = 22800000 nM T20251 D0G9YH 2179 IC50 = 208.93 nM T20251 D0GQ7K 4046 IC50 = 2600 nM T20251 D0GV8J 135565082 IC50 > 100000 nM T20251 D0H0KB 5070 IC50 > 25000 nM T20251 D0H3HM 60795 Ki = 598 nM T20251 D0H7AV 4820 IC50 = 20417.38 nM T20251 D0H7KF 5002 IC50 = 5754.4 nM T20251 D0I0DL 3689 IC50 = 100 nM T20251 D0I1FQ 54671008 IC50 > 50000 nM T20251 D0J0BU 10275777 Ki = 1800 nM T20251 D0J2KV 4932 IC50 = 440 nM T20251 D0JL2K 72474 IC50 = 50000 nM T20251 D0K3QS 6442177 IC50 = 15848931.92 nM T20251 D0K6GZ 60464 IC50 = 21700 nM T20251 D0K7WK 4595 IC50 = 812.83 nM T20251 D0L0ZF 5663 IC50 = 1096.48 nM T20251 D0L4YD 154059 IC50 = 251.19 nM T20251 D0L5WM 2157 IC50 = 10000 nM T20251 D0L7VL 3926 IC50 = 15.85 nM T20251 D0M4YC 3114 IC50 = 91201.08 nM T20251 D0N3VR 71616 IC50 > 40000 nM T20251 D0NJ3V 4680 IC50 = 7244.36 nM T20251 D0NR6S 3002977 IC50 = 79432.82 nM T20251 D0NS6H 3152 IC50 = 1995.26 nM T20251 D0NW3X 71329 IC50 = 5 nM T20251 D0O1WX 2764 IC50 > 30000 nM T20251 D0O3FG 125017 IC50 = 251188.64 nM T20251 D0O3OS 104850 IC50 = 4800 nM T20251 D0O8GK 71496458 IC50 = 16200 nM T20251 D0OB1J 39186 IC50 = 17300 nM T20251 D0P9RF 5401 IC50 = 17782.79 nM T20251 D0Q5UQ 214348 IC50 = 3981071.71 nM T20251 D0Q9EV 11965427 IC50 > 20000 nM T20251 D0R0FE 2520 IC50 = 10 nM T20251 D0R0MW 5329102 IC50 = 500 nM T20251 D0R1JV 60854 IC50 = 120.23 nM T20251 D0R1RS 3715 IC50 = 301995.17 nM T20251 D0RM9Q 68778 IC50 = 851.14 nM T20251 D0S5CU 4499 IC50 = 23000 nM T20251 D0T6WN 6451164 IC50 = 500 nM T20251 D0T8GD 89594 IC50 = 245470.89 nM T20251 D0T8XB 44513473 IC50 > 500000 nM T20251 D0TR5X 3386 IC50 = 10 nM T20251 D0U0VU 5312125 IC50 = 7943.28 nM T20251 D0U1OE 5452 IC50 = 33.2 nM T20251 D0U2JP 4369359 IC50 = 501187.23 nM T20251 D0U2OO 2477 IC50 = 3981.07 nM T20251 D0U3SY 49806720 IC50 > 30000 nM T20251 D0U5FS 3396 IC50 = 2300 nM T20251 D0U5GB 92727 IC50 = 8511.38 nM T20251 D0U5SI 4913 IC50 = 138038.43 nM T20251 D0V4QS 135398745 IC50 = 181.97 nM T20251 D0V8HJ 11671467 IC50 > 1000 nM T20251 D0W8WB 2353 IC50 = 3100 nM T20251 D0W9LX 2585 IC50 = 350 nM T20251 D0WE3O 5288826 IC50 = 1000000 nM T20251 D0WO8W 4062 IC50 = 154881.66 nM T20251 D0WV3U 4893 IC50 = 1584.89 nM T20251 D0X0RI 4178 IC50 = 10000 nM T20251 D0X4RN 3676 IC50 = 263026.8 nM T20251 D0X5ZI 6918493 IC50 = 501187.23 nM T20251 D0Y4JJ 2351 IC50 = 33 nM T20251 D0Y4QG 5388906 IC50 = 0.2 ug.mL-1 T20251 D0Y5AM 444031 IC50 = 79.43 nM T20251 D0Y5DO 2771 IC50 = 3981.07 nM T20251 D0Y5UG 2160 IC50 = 3280 nM T20251 D0Y7RW 4763 IC50 = 3019951.72 nM T20251 D0Z1RV 135398737 IC50 = 191 nM T20251 D0Z1UA 71301 IC50 = 316.23 nM T20251 D0Z1ZM 84029 IC50 = 33113.11 nM T20251 D0Z7ZM 135398744 IC50 = 3300 nM T20251 D00AUX 25230266 IC50 > 20000 nM T20251 D00BUR 216327 IC50 > 1000 nM T20251 D00DRL 44137946 IC50 > 30000 nM T20251 D00FHR 9865515 IC50 > 30000 nM T20251 D00IFR 58423153 IC50 > 30000 nM T20251 D00NZL 11955855 IC50 = 28100 nM T20251 D00RYA 16750271 IC50 > 10000 nM T20251 D00SWQ 10429242 IC50 > 100000 nM T20251 D00WDY 53477157 IC50 = 1400 nM T20251 D00XKB 57406537 IC50 = 2800 nM T20251 D01HLO 58438464 IC50 = 6900 nM T20251 D01NUR 118169620 IC50 = 69000 nM T20251 D01QSO 16654980 IC50 > 30000 nM T20251 D01UBY 46208367 IC50 > 50000 nM T20251 D01UUD 9948102 IC50 = 1700 nM T20251 D01ZAQ 25227436 IC50 > 100000 nM T20251 D02AIN 122678117 IC50 > 33000 nM T20251 D02AYL 456199 IC50 > 30000 nM T20251 D02DTQ 24745335 Ki = 3467.37 nM T20251 D02QWY 24785538 IC50 > 10000 nM T20251 D02WFN 46207733 IC50 = 60000 nM T20251 D03GNI 2166 IC50 = 3900 nM T20251 D03ISJ 135564632 IC50 > 30000 nM T20251 D03KHO 52934180 IC50 = 141000 nM T20251 D03KKR 3547 Ki = 25118.86 nM T20251 D03QAO 25008769 IC50 = 233000 nM T20251 D03QHC 49856296 IC50 = 13400 nM T20251 D03QIE 47953 IC50 = 44668.36 nM T20251 D03RIO 24743758 IC50 = 460 nM T20251 D04COD 25101874 IC50 = 588 ug.mL-1 T20251 D04JZH 11659955 IC50 = 30000 nM T20251 D04LOR 51030730 IC50 = 1900 nM T20251 D04LSD 9818903 Ki = 400 nM T20251 D04OSA 46202416 IC50 = 4800 nM T20251 D04QKU 11438771 IC50 = 7100 nM T20251 D04WUA 219101 IC50 = 10000 nM T20251 D05EXN 58298316 IC50 = 33000 nM T20251 D05LPW 25022354 IC50 = 79600 nM T20251 D05LRD 59286554 IC50 > 30000 nM T20251 D05UYQ 15984937 IC50 = 15848.93 nM T20251 D06DMQ 59472121 IC50 = 3000 nM T20251 D06ENM 66553195 IC50 = 6200 nM T20251 D06EPO 11192346 IC50 = 20000 nM T20251 D06TQR 76287260 IC50 = 26800 nM T20251 D06WHY 16747683 IC50 = 3200 nM T20251 D07EHV 44814409 IC50 = 12000 nM T20251 D07HPJ 11476171 IC50 = 130 nM T20251 D07HZG 11516136 IC50 = 126000 nM T20251 D07LWK 9811357 IC50 = 10000 nM T20251 D08AAV 46893585 IC50 > 100000 nM T20251 D08AOZ 86582336 IC50 = 5500 nM T20251 D08HOM 46207586 IC50 = 1000 nM T20251 D08QGT 17755052 IC50 = 64000 nM T20251 D08UUL 46700756 IC50 = 20000 nM T20251 D09NAW 60195662 Ki > 15857 nM T20251 D09OTX 89741565 IC50 = 1800 nM T20251 D09RVI 23649154 IC50 = 794.33 nM T20251 D0A3CL 49801838 IC50 = 22000 nM T20251 D0A7ZK 56944144 IC50 = 6100 nM T20251 D0B3FV 6445533 IC50 = 10300 nM T20251 D0B5HF 44476893 IC50 > 100000 nM T20251 D0C9UF 155805 IC50 = 1 nM T20251 D0CE6C 135565042 IC50 = 6300 nM T20251 D0DH5X 44472635 IC50 > 30000 nM T20251 D0E0JO 117857370 EC50 > 33000 nM T20251 D0EQ9T 24771368 IC50 > 10000 nM T20251 D0EY0A 42636350 IC50 > 32000 nM T20251 D0F0JJ 11560787 IC50 = 1200 nM T20251 D0F6YM 3035000 IC50 = 20000 nM T20251 D0F7PZ 53316710 IC50 = 12000 nM T20251 D0FD6D 11751922 IC50 = 20000 nM T20251 D0G6QV 208952 IC50 = 34860 nM T20251 D0H9DA 54761306 IC50 = 166000 nM T20251 D0HS5V 11234052 IC50 = 18000 nM T20251 D0HZ2E 5311271 Ki = 1100 nM T20251 D0I2XM 3038500 IC50 = 220 nM T20251 D0I3LO 91933883 IC50 > 10000 nM T20251 D0I3TU 45268455 Ki > 39000 nM T20251 D0I4PW 60164925 IC50 > 30000 nM T20251 D0IZ8X 90111638 IC50 > 10000 nM T20251 D0JU5X 400769 IC50 > 200000 nM T20251 D0K4FP 44548240 IC50 > 33000 nM T20251 D0K4HW 135409468 IC50 = 4466.84 nM T20251 D0K9IF 71666749 IC50 > 30000 nM T20251 D0L9KH 44623998 IC50 > 30000 nM T20251 D0L9QM 59568713 IC50 = 22000 nM T20251 D0LI1C 44469321 IC50 = 30440 nM T20251 D0LQ3L 77108121 IC50 = 195000 nM T20251 D0M3XR 46209133 IC50 = 39000 nM T20251 D0M4TJ 44219292 IC50 > 30000 nM T20251 D0M7CB 9919680 IC50 = 65700 nM T20251 D0M8FD 4261 IC50 > 30000 nM T20251 D0M8OC 16061509 IC50 > 10000 nM T20251 D0M9RQ 11697697 IC50 = 10000 nM T20251 D0MR0B 54766013 IC50 = 31040 nM T20251 D0N6NM 71721648 IC50 > 10000 nM T20251 D0N8QK 24743471 Ki = 8830 nM T20251 D0NU8J 117947097 IC50 > 50000 nM T20251 D0O0BM 44156901 IC50 = 8500 nM T20251 D0O1IM 58298318 IC50 > 33000 nM T20251 D0O1ZI 25006684 IC50 > 100000 nM T20251 D0O8BS 16039797 IC50 > 100000 nM T20251 D0O9XN 11691484 IC50 = 13000 nM T20251 D0OW9L 11973780 IC50 > 10000 nM T20251 D0P5CM 56945146 IC50 = 12589.25 nM T20251 D0PM5U 135564890 IC50 > 40000 nM T20251 D0PM7Q 11152667 IC50 = 15000 nM T20251 D0PW4N 6851740 IC50 = 4810 nM T20251 D0Q7RE 16007391 IC50 > 30000 nM T20251 D0QX8X 71479709 Ki = 3100 nM T20251 D0R0LB 91668194 IC50 > 100000 nM T20251 D0R2OU 25070031 IC50 = 13800 nM T20251 D0R3VK 42642654 IC50 = 4400 nM T20251 D0R8IU 24946280 IC50 > 100000 nM T20251 D0R9IU 44462758 IC50 = 8600 nM T20251 D0R9KG 11604525 IC50 = 11000 nM T20251 D0S1XX 134821691 IC50 > 80000 nM T20251 D0S5IR 86294073 IC50 > 30000 nM T20251 D0SG7B 49831257 IC50 = 85000 nM T20251 D0T0PN 9821217 Ki = 1800 nM T20251 D0T4QA 90456533 IC50 > 10000 nM T20251 D0U4FF 10437018 IC50 = 4000 nM T20251 D0U7KH 86567195 IC50 > 30000 nM T20251 D0U8QH 59239165 IC50 > 100000 nM T20251 D0V2YJ 11655511 IC50 = 20500 nM T20251 D0VI4N 90409366 IC50 > 10000 nM T20251 D0W8XT 60663 Ki = 190 nM T20251 D0XD4I 118502708 IC50 > 33000 nM T20251 D0XT0W 66555680 IC50 = 6900 nM T20251 D0XT6W 6918638 IC50 > 30000 nM T20251 D0Y3ZP 23480 IC50 = 500 nM T20251 D0Y5NA 118435360 IC50 = 9900 nM T20251 D0Y7NA 49871007 IC50 = 4500 nM T20251 D0Z2UQ 25262792 IC50 = 47500 nM T20251 D08IMD 16755780 IC50 = 23000 nM T20251 D0E2FZ 10149311 IC50 > 30000 nM T20251 D0HM5J 118253852 IC50 > 33000 nM T20251 D0IY0R 11591505 IC50 = 23600 nM T20251 D0X5OV 42609962 IC50 > 30000 nM T20251 D01KIJ 72545600 IC50 >= 18500 nM T20251 D02NRD 9865421 IC50 > 10000 nM T20251 D03GTM 118485599 IC50 = 69 nM T20251 D04MAZ 71731606 IC50 = 100000 nM T20251 D0AF0O 54670056 IC50 = 590 nM T20251 D0CV8T 874670 IC50 > 10000 nM T20251 D0D3GL 137662068 IC50 = 15000 nM T20251 D0D4OW 57338826 Ki > 100000 nM T20251 D0F8KE 71059525 Ki = 41.3 nM T20251 D0HG2S 86294663 IC50 = 67000 nM T20251 D0J1LK 118485649 IC50 = 490 nM T20251 D0LU9X 74221950 IC50 = 19000 nM T20251 D0NG8Q 75203906 IC50 = 20900 nM T20251 D0PJ8X 71562840 IC50 = 61700 nM T20251 D0PO8N 117881270 IC50 > 33000 nM T20251 D0V8FC 60169096 IC50 = 25000 nM T20251 D0WS3T 72706254 IC50 = 2700 nM T20251 D0YN2T 86302836 IC50 > 10000 nM T20251 D00PDG 44454750 IC50 = 800 nM T20251 D00PXQ 60785 Ki = 200 nM T20251 D02NGR 9934294 IC50 = 670 nM T20251 D03KWN 11373432 IC50 > 100000 nM T20251 D03OFO 9851380 IC50 = 6000 nM T20251 D04BQR 4342 IC50 = 100000 nM T20251 D06BPG 4528 IC50 > 27000 nM T20251 D06TGE 11226090 IC50 = 14200 nM T20251 D06VXY 9845214 IC50 = 420 nM T20251 D07BUO 25067561 IC50 = 19000 nM T20251 D07GIB 11614352 IC50 = 11000 nM T20251 D07KIJ 10008367 IC50 = 13000 nM T20251 D08AWI 11430856 Ki > 2000 nM T20251 D08SOF 5405 IC50 = 22 nM T20251 D09EVZ 507806 IC50 > 80000 nM T20251 D09RGW 11753159 IC50 > 15848.93 nM T20251 D09XHI 9879103 IC50 = 6350 nM T20251 D0A1NU 16049769 Ki > 45100 nM T20251 D0AQ3H 11505444 IC50 > 10000 nM T20251 D0B4TT 17747460 IC50 = 50.12 nM T20251 D0B7SP 11292933 Ki = 12589.25 nM T20251 D0E2PX 3087190 IC50 = 18.1 nM T20251 D0E3SD 9838729 IC50 > 33000 nM T20251 D0E6OA 65941 IC50 = 251.19 nM T20251 D0G1RH 6918446 IC50 = 194 nM T20251 D0H9GQ 9795276 IC50 = 10000 nM T20251 D0I5UU 123618 IC50 = 27.54 nM T20251 D0J0AE 10052040 IC50 > 3000 nM T20251 D0J9UI 9807238 Ki > 10000 nM T20251 D0K1VK 25262965 IC50 = 30400 nM T20251 D0N8NK 11641563 IC50 = 40000 nM T20251 D0OS6O 60149 IC50 ~ 3 nM T20251 D0Q3ES 11705608 IC50 = 3000 nM T20251 D0W7IR 9887884 IC50 = 32000 nM T20251 D0Y2HR 2247 IC50 = 0.9 nM T20251 D0Y6SN 5311096 IC50 = 630.96 nM T20251 D0Z0CH 3033962 IC50 = 5 nM T20251 C9H6CG 1287 IC50 = 6025.6 nM T20251 CXUC05 2215 IC50 = 2398.83 nM T20251 CCNZ53 2340 IC50 = 3981071.71 nM T20251 CPJ0C2 2747 IC50 = 8800 nM T20251 CZUI83 2769 IC50 = 6.457 nM T20251 CCW9O8 2825 IC50 = 1202.26 nM T20251 CYO1K2 2826 IC50 = 7244.36 nM T20251 C2AXN5 3148 IC50 = 12022.64 nM T20251 CDR20M 3185 IC50 = 1.2 nM T20251 C0H8GR 3191 IC50 = 331.13 nM T20251 C2XP5J 3255 IC50 = 72443.6 nM T20251 CY4WG9 3793 IC50 > 40000 nM T20251 C9LCD8 3823 IC50 = 1905.46 nM T20251 CP4RM6 4486 IC50 = 10000 nM T20251 C5ZC4S 5977 IC50 = 4365158.32 nM T20251 CP1QC0 9801 IC50 = 65 nM T20251 CBHG51 9822 IC50 > 10000 nM T20251 CZXE86 15330 IC50 = 2754.23 nM T20251 CN0WP7 15630 IC50 < 10000 nM T20251 CKCT41 28292 IC50 = 50118.72 nM T20251 CA12TG 38911 IC50 > 40000 nM T20251 C6GN7M 40692 Ki = 1900 nM T20251 CI93MP 51106 IC50 = 9100 nM T20251 C8ODZ3 56069 IC50 > 25000 nM T20251 CV4S2E 62969 IC50 = 200 nM T20251 CP8F7B 64143 IC50 = 12589.25 nM T20251 CD9TC8 64737 IC50 = 22000 nM T20251 C92TML 65014 IC50 > 100000 nM T20251 C97NOS 68634 IC50 = 2100 nM T20251 C1O4FS 73400 IC50 = 16000 nM T20251 CU1H3J 83952 IC50 = 316227.77 nM T20251 C7SXL6 87152 IC50 > 25000 nM T20251 C36LYP 104904 IC50 = 416869.38 nM T20251 C09TNA 107927 IC50 = 40000 nM T20251 CL4IR8 115159 IC50 = 50118.72 nM T20251 CR91WU 117964 IC50 = 84000 nM T20251 CZ48UK 117965 IC50 = 13000 nM T20251 CJ1XF0 119478 IC50 = 169824.37 nM T20251 CEP43C 122068 IC50 = 9500 nM T20251 C6SRK5 123942 IC50 = 1047.13 nM T20251 CMN95P 127718 IC50 = 20.89 nM T20251 CM01FR 128820 IC50 = 44000 nM T20251 CU0C6S 131698 IC50 = 491.4 nM T20251 CIG7L1 160023 IC50 = 8 nM T20251 CGSA42 163906 IC50 = 6100 nM T20251 CDB9P5 170922 IC50 < 10000 nM T20251 C7AV9Z 175533 Ki = 0.4 nM T20251 CLY60V 187063 IC50 = 6606.93 nM T20251 C97DNP 194450 IC50 = 4.3 nM T20251 CI2WO8 219099 IC50 = 120.23 nM T20251 C2V5FA 398712 IC50 = 5000 nM T20251 CLD6J9 441074 IC50 = 323.59 nM T20251 C1Z4HP 441362 IC50 = 5623.41 nM T20251 CQ0XH2 467825 IC50 = 10370 nM T20251 CKC8U4 507751 IC50 > 80000 nM T20251 CPXL01 507783 IC50 > 80000 nM T20251 CM40AT 507791 IC50 > 80000 nM T20251 CFY12E 516173 Ki > 10000 nM T20251 CNCR59 516203 Ki = 30000 nM T20251 C9MVL1 516212 Ki = 16000 nM T20251 CJUT37 516217 Ki = 5700 nM T20251 CRG4W0 516223 Ki = 3800 nM T20251 C2WHI5 516226 Ki = 22000 nM T20251 C9UOI0 516233 Ki = 8100 nM T20251 C67BKT 516235 Ki = 3000 nM T20251 CWTN29 516239 Ki > 10000 nM T20251 C6L1BX 516246 Ki = 3400 nM T20251 C4MQR0 516247 Ki = 5600 nM T20251 C1LB4X 516254 Ki = 37000 nM T20251 CQ52IA 516260 Ki = 14000 nM T20251 C65AZI 516264 Ki = 1000 nM T20251 COA04U 516275 Ki = 3500 nM T20251 C59YWP 516276 Ki = 9600 nM T20251 C9XU6R 516280 Ki = 6000 nM T20251 CHN28A 516284 Ki = 11000 nM T20251 CBYO78 516292 Ki = 2100 nM T20251 C4XN2D 516293 Ki = 2300 nM T20251 CUAO78 516314 Ki = 400 nM T20251 CF2J7U 592280 IC50 = 169824.37 nM T20251 C4TY8B 607867 IC50 = 74 nM T20251 C8WX7B 621620 IC50 = 109647.82 nM T20251 C2M9UC 656771 IC50 = 20 nM T20251 CP7U6Y 667468 IC50 = 6456.54 nM T20251 CN5CJ7 688803 IC50 = 99300 nM T20251 CZN6S9 743974 IC50 > 50118.72 nM T20251 CSMB29 759456 IC50 = 12400 nM T20251 C3LM4S 821286 IC50 > 100000 nM T20251 C90NZF 853261 IC50 > 10000 nM T20251 C79YAJ 1034176 IC50 = 1350 nM T20251 CT2VP9 1471775 IC50 > 32000 nM T20251 CK0JI9 1548955 IC50 = 181.97 nM T20251 C8JLO0 2243267 IC50 = 6300 nM T20251 CTZ4R5 2730286 IC50 = 1500 nM T20251 CD28JA 2735964 IC50 = 10000 nM T20251 CHTM19 2747356 Ki = 1538 nM T20251 C2J9ML 2781852 IC50 > 10000 nM T20251 CORX94 2804997 IC50 > 26302.68 nM T20251 CMRX81 2811640 IC50 > 10000 nM T20251 C9LDS2 2971413 Ki = 5418 nM T20251 C0F4YK 2980278 Ki > 40000 nM T20251 C14NBG 3008866 IC50 > 80000 nM T20251 CUY7J9 3008902 IC50 = 550 nM T20251 CE3Q4V 3008904 IC50 = 1300 nM T20251 CZ1V8Q 3008913 IC50 = 670 nM T20251 C1IS9G 3008917 IC50 = 150 nM T20251 CZV0O6 3008927 IC50 = 570 nM T20251 C8KY7B 3008930 IC50 = 1200 nM T20251 CSED31 3011729 IC50 = 13000 nM T20251 C3U7EZ 3035784 IC50 = 100 nM T20251 C2YQ0B 3082684 IC50 = 14000 nM T20251 CS5F1I 3083481 Ki = 1200 nM T20251 C3HJK8 3525815 IC50 = 2500 nM T20251 C8KN4J 3876755 IC50 > 10000 nM T20251 CO23EI 3959338 IC50 = 27300 nM T20251 C0TV9U 4227718 IC50 > 10000 nM T20251 C9INQ8 4390854 IC50 > 33000 nM T20251 CWE45H 4497898 IC50 = 27000 nM T20251 CO2SY7 4630909 Ki = 870 nM T20251 CE1CP8 4663848 IC50 = 33113.11 nM T20251 C3JHM8 4687521 IC50 = 100000 nM T20251 C16EGI 4961254 IC50 > 10000 nM T20251 CJP1K5 4987129 IC50 > 14790 nM T20251 CZ32RC 5230270 IC50 = 1445.44 nM T20251 CLNI10 5281408 IC50 = 773000 nM T20251 CJB7T6 5288494 IC50 > 33000 nM T20251 CW38FP 5311047 IC50 < 1000 nM T20251 C8EG4K 5326625 IC50 = 8100 nM T20251 C1OZS6 5436342 IC50 > 100000 nM T20251 C3Q2XB 5495793 IC50 > 80000 nM T20251 C0ZAM9 5495818 IC50 > 80000 nM T20251 C6SON9 5837004 IC50 = 36307.81 nM T20251 C95DOH 6098167 IC50 = 12000 nM T20251 CPV72R 6102824 IC50 = 3500 nM T20251 CGL87W 6483572 IC50 = 10500 nM T20251 CO9NP6 6890860 IC50 = 43620 nM T20251 CFTO93 6918704 IC50 = 710 nM T20251 CU68IK 7141881 IC50 > 10000 nM T20251 CZAN92 7472794 IC50 > 25000 nM T20251 C5J8HN 8902499 IC50 = 12700 nM T20251 CL9O2G 9390285 IC50 = 30000 nM T20251 C9IFX8 9390560 IC50 = 13000 nM T20251 CJ07ZA 9800555 IC50 = 32000 nM T20251 C5Z2KM 9805944 IC50 = 245 nM T20251 C2H4ZK 9806118 IC50 = 24 nM T20251 C1W2VB 9814248 IC50 = 5230 nM T20251 CAD92E 9815159 IC50 = 900 nM T20251 CTR6H5 9817349 IC50 = 1995.26 nM T20251 CJS5L9 9819317 IC50 > 30000 nM T20251 C71XRT 9821510 IC50 = 7199.99 nM T20251 CE6NF9 9823363 IC50 = 3100 nM T20251 CEL3C9 9824630 IC50 = 480 nM T20251 C0PQT8 9824969 IC50 = 39800 nM T20251 CZV60D 9825288 Ki = 26400 nM T20251 C97VAE 9825776 Ki = 22700 nM T20251 C8EC9B 9828617 IC50 = 2511.89 nM T20251 CWM26G 9830364 IC50 = 25118.86 nM T20251 C1FQ5A 9835490 IC50 = 8290 nM T20251 C0E7YV 9836903 IC50 > 30000 nM T20251 CU0HE4 9839392 Ki = 18 nM T20251 C30IAQ 9840150 IC50 = 5300 nM T20251 CXE1Y8 9842436 IC50 = 3200 nM T20251 CG3U7J 9843049 IC50 = 1100 nM T20251 CA6N0H 9843867 IC50 = 4700 nM T20251 C7VSU2 9845018 IC50 = 440 nM T20251 CT4E5Z 9846543 IC50 = 210 nM T20251 CKD2H4 9848990 IC50 = 7585.78 nM T20251 C9XY6D 9849838 Ki = 1180 nM T20251 CH57DZ 9850318 IC50 = 1413 nM T20251 CF72XZ 9860561 IC50 = 1600 nM T20251 CRBW42 9861124 IC50 = 5570 nM T20251 C3EX7S 9862272 IC50 = 204 nM T20251 CGC0F7 9864462 IC50 = 2760 nM T20251 CXZ6Q7 9866918 IC50 = 8200 nM T20251 CAOK24 9867098 IC50 = 80 nM T20251 CN9YD5 9868131 IC50 = 3000 nM T20251 C7T3VS 9870145 IC50 = 70 nM T20251 CK7FJ6 9870185 IC50 = 6309.57 nM T20251 CR0EG2 9879772 IC50 = 692 nM T20251 CQJ5X2 9879974 IC50 = 1240 nM T20251 CPS24V 9880847 IC50 = 27460 nM T20251 CS6FN7 9883254 IC50 > 100000 nM T20251 C9IR5L 9884379 IC50 = 90 nM T20251 C2TV9M 9884543 IC50 = 1100 nM T20251 CZ8C7G 9885279 Ki = 6800 nM T20251 C64EOU 9885465 Ki = 1000 nM T20251 CO84WK 9885754 Ki = 62000 nM T20251 C9I8ZU 9887120 IC50 = 10000 nM T20251 CUF35J 9887834 IC50 = 12600 nM T20251 C85BQG 9890458 IC50 = 14000 nM T20251 C2P3GS 9899500 IC50 = 2500 nM T20251 CE28TW 9900179 IC50 = 3020 nM T20251 C2Z9BL 9908431 Ki = 560 nM T20251 CYZ5N4 9909089 EC50 = 7.943 nM T20251 CHB5G9 9909904 IC50 = 199.53 nM T20251 CVJ7I8 9910573 IC50 = 176 nM T20251 C4B2QY 9913339 IC50 = 25000 nM T20251 CF4VO1 9914506 IC50 = 25118.86 nM T20251 CIW81R 9923839 IC50 = 3400 nM T20251 CQF2X8 9925089 IC50 = 974 nM T20251 C10VOI 9930235 IC50 = 3600 nM T20251 CANK40 9931593 IC50 = 10000 nM T20251 C1F4WB 9932192 IC50 = 6960 nM T20251 C9FZO7 9932679 IC50 = 10499.99 nM T20251 C5HQM7 9932974 IC50 = 150 nM T20251 C6RF9U 9933928 IC50 = 1000 nM T20251 CDY39E 9934161 IC50 > 5000 nM T20251 COP96L 9936388 IC50 = 1600 nM T20251 CV5X7E 9938284 Ki = 1000 nM T20251 CS58EO 9944019 IC50 = 3850 nM T20251 CX3ZK9 9946374 IC50 = 1190 nM T20251 CZ4X5D 9946965 IC50 = 101 nM T20251 CV1T2W 9947009 IC50 = 1620 nM T20251 CH6IJ8 9947172 IC50 = 1120 nM T20251 C8T1HO 9948670 Ki = 1300 nM T20251 CLR78W 9952894 Ki = 35000 nM T20251 CKF9X1 9953268 Ki = 1300 nM T20251 CMI58L 9956563 IC50 = 1.7 nM T20251 CJ6BV9 9959777 IC50 = 36 nM T20251 C1NPJ7 9965169 IC50 = 7390 nM T20251 CT7BR0 9965311 IC50 > 1000 nM T20251 C3KTF6 9965610 IC50 = 4670 nM T20251 C6CXJ3 9966330 IC50 = 4560 nM T20251 C0ORJ4 9966331 IC50 = 1310 nM T20251 C49MPX 9966437 IC50 = 3390 nM T20251 CJ2DK6 9966438 IC50 = 1480 nM T20251 C7ZK5J 9966516 IC50 > 10000 nM T20251 CC35UV 9966603 IC50 = 6830 nM T20251 CPX92V 9979309 Ki = 794.33 nM T20251 C7TPF5 9983233 Ki = 445 nM T20251 CGO70N 9983801 IC50 = 82 nM T20251 CJOV70 9983904 IC50 = 54000 nM T20251 CGEJ24 9985625 IC50 = 5100 nM T20251 CRYX90 9986337 IC50 = 9000 nM T20251 C7OAK1 9986346 IC50 = 25.12 nM T20251 CD86AJ 10000396 Ki = 85000 nM T20251 CUQF40 10003657 IC50 = 6309.57 nM T20251 CQL12P 10004545 IC50 > 5000 nM T20251 CGY63T 10004877 IC50 = 85000 nM T20251 CZW1M7 10005242 IC50 > 31622.78 nM T20251 C4Y8TH 10006938 IC50 = 14000 nM T20251 CE7IB5 10007642 IC50 = 11000 nM T20251 CCO68X 10008352 IC50 = 100 nM T20251 CUN7T8 10019811 Ki = 10000 nM T20251 C3NPS8 10025899 Ki = 1750 nM T20251 CA06TQ 10028888 IC50 = 6600 nM T20251 CI3Q9B 10030247 IC50 = 130 nM T20251 CWD3B7 10030344 IC50 = 400 nM T20251 C6V8MF 10032207 IC50 = 8300 nM T20251 C1WH8Q 10042344 IC50 > 10000 nM T20251 C90AVX 10044868 Ki = 51000 nM T20251 C04HZE 10046270 IC50 > 10 nM T20251 CA42DO 10047196 IC50 = 3000 nM T20251 C02OIU 10047339 IC50 = 2250 nM T20251 C73QBA 10047509 IC50 > 10 nM T20251 CR6NW9 10054055 IC50 = 5400 nM T20251 CH5SZ3 10073306 IC50 = 70000 nM T20251 CF7OC8 10073954 IC50 = 21000 nM T20251 CRQL64 10075375 Ki = 120 nM T20251 CR01QE 10076802 IC50 = 1800 nM T20251 C2BG6C 10085660 IC50 > 10000 nM T20251 C8G1PU 10087576 Ki = 2900 nM T20251 CH14BN 10089061 Ki = 480 nM T20251 CR17PA 10093856 IC50 = 2200 nM T20251 CS5K6Q 10095195 IC50 = 2000 nM T20251 C83ZDL 10096130 Ki = 2800 nM T20251 CTN9C2 10097082 IC50 = 3000 nM T20251 C9D5FP 10099787 Ki = 730 nM T20251 C3L9IN 10110435 IC50 = 34000 nM T20251 CBUX03 10113183 IC50 = 8950 nM T20251 CFY9M8 10115569 IC50 = 23000 nM T20251 CVK61T 10116047 IC50 = 26000 nM T20251 CD9EV1 10126599 Ki = 3600 nM T20251 C1WYS8 10127169 Ki = 46 nM T20251 C6N2TK 10131545 IC50 = 2150 nM T20251 CVZ3S9 10132138 IC50 = 10100 nM T20251 C26HWK 10132572 IC50 = 1310 nM T20251 CV67NU 10136016 IC50 = 16700 nM T20251 C09XVI 10144709 IC50 = 54 nM T20251 CLBD08 10144909 Ki = 850 nM T20251 CQM6E2 10149720 Ki = 20000 nM T20251 CLW3J6 10151756 IC50 = 5011.87 nM T20251 CB6V1X 10162604 Ki = 58400 nM T20251 C7JP1A 10163439 Ki = 610 nM T20251 C75JIV 10167216 Ki = 38100 nM T20251 CSHY89 10172243 Ki = 39000 nM T20251 CQ6JH8 10173083 Ki = 15000 nM T20251 CR80BV 10175126 IC50 > 30000 nM T20251 CW0OK6 10178465 IC50 = 6100 nM T20251 C85DYP 10183035 IC50 = 13600 nM T20251 C5K2GS 10185181 Ki = 200 nM T20251 C3DM7B 10186910 IC50 = 12200 nM T20251 CW98JD 10187118 IC50 = 400 nM T20251 C73LXY 10188021 Ki = 11 nM T20251 CK7UT9 10188786 Ki = 290 nM T20251 CLJ02H 10194468 Ki = 240 nM T20251 COV97M 10199905 IC50 = 18600 nM T20251 CCE6H8 10203632 IC50 = 36600 nM T20251 CO51ZR 10205659 Ki = 420 nM T20251 CISE26 10206059 IC50 = 89400 nM T20251 C51SKM 10209082 Ki = 25 nM T20251 CK72XG 10209108 Ki = 490 nM T20251 CCG65P 10210026 Ki = 1200 nM T20251 CT2N1Z 10222208 Ki = 840 nM T20251 C18FMW 10237542 Ki = 320 nM T20251 CQGN38 10237827 Ki = 29 nM T20251 C2PLB1 10239891 IC50 > 30000 nM T20251 C8PJ1V 10248119 IC50 > 10000 nM T20251 CZ90LD 10250452 IC50 = 4600 nM T20251 C24QZK 10256734 IC50 = 4000 nM T20251 CXJ2O5 10256826 IC50 = 2000 nM T20251 C3OE5Z 10257392 IC50 = 2100 nM T20251 C67GCK 10258336 Ki = 43 nM T20251 CF2M9O 10268223 IC50 = 234 nM T20251 CGRQ23 10274114 IC50 = 2700 nM T20251 CHY71P 10274246 IC50 = 960 nM T20251 CM6SE7 10280445 IC50 = 4400 nM T20251 CMNH04 10286136 IC50 = 3300 nM T20251 CUQC81 10287415 Ki = 9400 nM T20251 C9K0SA 10288761 IC50 = 5000 nM T20251 CT89LX 10297708 IC50 = 4000 nM T20251 CV10CU 10297977 Ki = 100 nM T20251 C90DYG 10297996 IC50 = 50100 nM T20251 C1AP6H 10298858 Ki = 2100 nM T20251 CAX9W2 10302405 Ki = 34 nM T20251 C1W5ZD 10308681 Ki = 8050 nM T20251 C3M1VR 10309552 Ki = 225 nM T20251 CZ18PL 10316203 IC50 = 7500 nM T20251 C26EKI 10316979 IC50 = 31000 nM T20251 CF1S8U 10320144 IC50 = 86000 nM T20251 C03ZKG 10324551 IC50 = 5000 nM T20251 CBA2C6 10325032 IC50 = 224 nM T20251 CLKX29 10335984 Ki = 4500 nM T20251 CEZ95L 10342016 Ki = 52000 nM T20251 C5MH7Y 10343434 IC50 = 300 nM T20251 CW50TU 10345610 IC50 = 35200 nM T20251 CIYQ04 10358984 Ki = 6300 nM T20251 CGQN51 10359235 IC50 > 30000 nM T20251 CT6Y9I 10365686 IC50 = 38000 nM T20251 CFH29X 10367570 IC50 = 300 nM T20251 CDA5F7 10369999 IC50 = 6200 nM T20251 C2KO8V 10388264 IC50 = 29000 nM T20251 CP7CH6 10389946 IC50 = 38000 nM T20251 C3H9SB 10390717 IC50 = 19700 nM T20251 CJQV19 10391684 IC50 > 80000 nM T20251 CM9R2K 10391877 IC50 = 1200 nM T20251 CCZ17H 10392978 IC50 = 844 nM T20251 C9WC5D 10393066 IC50 > 8900 nM T20251 CU6X7E 10393880 IC50 = 130 nM T20251 C59QRY 10393962 Ki = 950 nM T20251 C76WZF 10401439 Ki = 11000 nM T20251 CG1T4B 10405623 IC50 = 2700 nM T20251 C6EJ8D 10410012 IC50 = 6.2 nM T20251 C56SLV 10412648 IC50 = 38 nM T20251 CV60SK 10413034 IC50 > 30000 nM T20251 CBN4H0 10415698 IC50 = 1300 nM T20251 CW80YU 10415870 Ki = 710 nM T20251 CUZE30 10416011 IC50 = 100 nM T20251 C6GXW2 10426299 Ki = 1200 nM T20251 C6KR8Z 10428027 Ki = 5100 nM T20251 CS7FG5 10429706 IC50 = 2570.4 nM T20251 C5ZXU8 10433753 IC50 = 25000 nM T20251 C5GQF1 10436125 IC50 = 22700 nM T20251 CWCA76 10439426 IC50 = 76000 nM T20251 C80TCL 10450279 Ki = 5000 nM T20251 CQ4C7Y 10450926 IC50 = 28600 nM T20251 CHW2U1 10451701 IC50 > 33000 nM T20251 C1T7QW 10456093 IC50 = 11000 nM T20251 CVSP85 10456367 IC50 = 29000 nM T20251 C8DWH6 10456892 IC50 = 30700 nM T20251 C38VGA 10457264 IC50 = 2000 nM T20251 C10NHR 10457710 IC50 = 2000 nM T20251 CMDU71 10460463 IC50 = 100 nM T20251 CWFK56 10461282 IC50 = 660 nM T20251 CGXY36 10482372 IC50 = 18100 nM T20251 CEW7C9 10482996 IC50 = 400 nM T20251 C7YPV6 10483558 IC50 = 250 nM T20251 CB52TQ 10495305 Ki = 3000 nM T20251 CPG8U3 10495787 Ki = 1500 nM T20251 C7W9LB 10498834 IC50 = 400 nM T20251 CI0PU7 10518508 IC50 = 10.96 nM T20251 CUQ03E 10520440 Ki = 1600 nM T20251 C2B9PT 10522146 Ki = 930 nM T20251 CV57XZ 10546579 Ki = 110 nM T20251 CMK39Q 10553487 IC50 > 10000 nM T20251 C8E1UH 10570940 IC50 = 3000 nM T20251 CKYT25 10597785 IC50 = 8800 nM T20251 C74NSJ 10615016 Ki = 7000 nM T20251 CQ75TL 10640054 Ki = 1400 nM T20251 C8C2GN 10640055 Ki = 2100 nM T20251 CY9A6G 10689687 IC50 = 790 nM T20251 CG0M4S 10697284 IC50 = 2400 nM T20251 COQ25N 10697363 IC50 = 100 nM T20251 C49IUL 10708935 Ki > 1100 nM T20251 C52SWI 10711404 Ki > 7000 nM T20251 C7PDA6 10713670 Ki = 500 nM T20251 C18ZBG 10758132 Ki = 238 nM T20251 CDK53W 10763704 IC50 = 1000 nM T20251 CFH1Q4 10805130 Ki = 2500 nM T20251 CDOH18 10851309 Ki = 8200 nM T20251 C0VQ3C 10853014 Ki = 5400 nM T20251 CV6ZN3 10861900 Ki = 710 nM T20251 C9QUV7 10863652 Ki = 25000 nM T20251 CX3RT7 10874250 IC50 = 180 nM T20251 C6KW8J 10884405 IC50 = 4300 nM T20251 C4QZ2E 10895064 IC50 = 5800 nM T20251 CLI84D 10895869 IC50 = 9900 nM T20251 C5L2FR 10896860 IC50 = 110 nM T20251 CZFJ03 10899797 IC50 > 60000 nM T20251 CAB0O8 10906012 IC50 = 2700 nM T20251 CDR7G5 10925892 Ki = 69 nM T20251 C9OI8S 10927262 Ki = 1900 nM T20251 CD10XK 10928028 IC50 = 4700 nM T20251 CR8NL2 10950878 IC50 = 870 nM T20251 C4PK7X 10971209 Ki = 570 nM T20251 C6HI0W 10971692 IC50 = 8399.99 nM T20251 C0BUR1 10991521 Ki = 110 nM T20251 CE6XI4 10993905 IC50 = 190 nM T20251 C3WI1P 11004853 IC50 = 4400 nM T20251 CH2A4Z 11016041 IC50 = 4900 nM T20251 C0A7DI 11017241 Ki = 39000 nM T20251 C1N5EF 11026589 IC50 = 9099.99 nM T20251 CG9JC8 11036563 Ki = 4000 nM T20251 C5P8RW 11048955 Ki = 22400 nM T20251 C0EWV4 11056631 Ki = 47 nM T20251 CEPM03 11068867 IC50 = 5870 nM T20251 C56YON 11069321 IC50 = 77 nM T20251 CKBM74 11070099 IC50 = 220 nM T20251 CG2WF1 11111531 Ki = 251 nM T20251 CHX96W 11133309 Ki = 7143 nM T20251 C0VBZ4 11144668 IC50 = 11999.99 nM T20251 CLU8C6 11145028 IC50 = 10000 nM T20251 C7HM0O 11152739 IC50 = 9200 nM T20251 C4NAJ5 11154544 IC50 = 1600 nM T20251 C76YFB 11155030 IC50 = 3300 nM T20251 C3X0AC 11155482 IC50 = 65000 nM T20251 C9AT4X 11163693 IC50 > 20000 nM T20251 CDY8S7 11165745 IC50 = 1650 nM T20251 CK67YW 11166256 Ki > 150000 nM T20251 C6FX8E 11166272 IC50 = 7700 nM T20251 C7OEX0 11174494 IC50 = 17200 nM T20251 CI7L1C 11176908 IC50 = 10000 nM T20251 C1QWM8 11178027 IC50 = 27000 nM T20251 CPEV03 11178961 IC50 = 466 nM T20251 C3TW2O 11187225 IC50 = 2700 nM T20251 C6EWJ9 11188910 IC50 = 13000 nM T20251 C3CAP9 11189372 IC50 = 1000 nM T20251 CUBX19 11189444 IC50 = 1300 nM T20251 CAN73X 11189693 IC50 = 730 nM T20251 CDOC09 11199458 IC50 = 33500 nM T20251 CE6HS7 11200189 IC50 = 56700 nM T20251 CC25EY 11200344 IC50 = 9900 nM T20251 CP6UL9 11200377 IC50 = 9800 nM T20251 CIAE47 11211122 IC50 = 44113 nM T20251 CS5ET8 11212373 IC50 = 1800 nM T20251 CY57AG 11212679 Ki = 794.33 nM T20251 CQ1E8L 11213136 IC50 = 1000 nM T20251 C20HPU 11220991 IC50 = 2300 nM T20251 C5TAN7 11223519 IC50 = 15000 nM T20251 C1VM2S 11225043 IC50 = 200 nM T20251 C0FSV9 11225074 IC50 = 1400 nM T20251 CP9Z1V 11225445 IC50 = 440 nM T20251 CHC3F8 11226573 IC50 = 820 nM T20251 CU75LJ 11227168 IC50 = 26000 nM T20251 CA39QR 11227406 IC50 = 400 nM T20251 C6D3UR 11237434 IC50 = 17900 nM T20251 CC62PB 11238080 IC50 = 52 nM T20251 CTS6F4 11238521 IC50 = 460 nM T20251 C8J5KI 11238580 IC50 = 750 nM T20251 CP8EW3 11245596 IC50 > 10000 nM T20251 C8TD3U 11247946 IC50 = 900 nM T20251 CX43IH 11248146 IC50 = 700 nM T20251 CW1O5V 11256620 IC50 = 220 nM T20251 CP0C2Q 11257803 IC50 > 11000 nM T20251 CZ98EU 11259253 IC50 = 3.6 nM T20251 C7XI0R 11260032 IC50 = 794.33 nM T20251 C92CYH 11265950 Ki > 3000 nM T20251 CRZ3V0 11269310 IC50 = 11784 nM T20251 C2U7OP 11270012 IC50 = 1800 nM T20251 C3N1MF 11270500 IC50 > 24000 nM T20251 C26HWL 11270869 IC50 = 560 nM T20251 CRDU42 11271947 IC50 = 12000 nM T20251 CL0DP6 11272440 IC50 = 501.19 nM T20251 CK36XS 11273324 IC50 = 83.18 nM T20251 CZ8DU0 11273379 IC50 = 10000 nM T20251 C53DQM 11273508 IC50 = 100 nM T20251 COV2U9 11281200 IC50 = 1700 nM T20251 C83KDF 11281738 Ki > 150000 nM T20251 C8CS5F 11282651 IC50 = 6900 nM T20251 CP27SY 11283686 IC50 = 1300 nM T20251 C9X0TH 11291017 IC50 = 15000 nM T20251 CNE3Z7 11296572 IC50 = 700 nM T20251 CV1LG4 11301893 IC50 = 1100 nM T20251 C9BLC7 11304596 Ki = 1995.26 nM T20251 CIMB79 11305766 IC50 = 199.53 nM T20251 C9L0IK 11313056 IC50 = 300000 nM T20251 C30MLR 11313946 IC50 > 31600 nM T20251 CNT19Q 11315446 IC50 = 11000 nM T20251 CVB45M 11315811 IC50 = 24000 nM T20251 C8S4FU 11317045 IC50 = 600 nM T20251 C5DBK1 11326750 IC50 > 50000 nM T20251 CWT28O 11328029 IC50 = 11.5 nM T20251 CP8Y7T 11328449 IC50 = 1800 nM T20251 C5M3ZN 11329138 IC50 = 6100 nM T20251 CQ1CG9 11330529 IC50 = 30000 nM T20251 CIT2Y7 11330837 IC50 > 30000 nM T20251 C7O0ER 11337925 IC50 = 5094 nM T20251 CKZ20A 11353843 IC50 = 9000 nM T20251 CX6C2M 11353855 IC50 = 28000 nM T20251 C0PUK5 11360073 IC50 = 20500 nM T20251 C9L7AT 11364901 IC50 = 40 nM T20251 CZ82WH 11365166 IC50 > 30000 nM T20251 C4BZ1C 11372427 IC50 = 20000 nM T20251 COH57K 11373894 Ki = 1000 nM T20251 C25ZCN 11374110 IC50 > 30000 nM T20251 C36OES 11374857 IC50 = 3.6 nM T20251 CWO2A7 11382160 IC50 = 62000 nM T20251 C2E8MJ 11382472 IC50 = 11989 nM T20251 CEKP86 11383454 IC50 = 501.19 nM T20251 CO1I8H 11384634 Ki = 885 nM T20251 CL1W3C 11387497 IC50 = 100 nM T20251 CE2M9F 11387511 IC50 = 13000 nM T20251 CCK08I 11388055 IC50 = 650 nM T20251 C53ANS 11393281 IC50 > 30000 nM T20251 C9AOM3 11397017 IC50 = 470 nM T20251 CF4OX6 11397149 Ki = 316.23 nM T20251 C7M3XJ 11397742 IC50 = 22600 nM T20251 C82ERW 11397777 IC50 = 350 nM T20251 CQE92F 11406708 IC50 = 21079 nM T20251 CE5ZK6 11409228 IC50 > 30000 nM T20251 CMW42X 11416123 IC50 > 20000 nM T20251 C6I0YP 11416924 IC50 = 3000 nM T20251 C6BE9Q 11417954 IC50 = 78000 nM T20251 CFX98O 11418182 Ki = 5561 nM T20251 C2N0AG 11421712 IC50 > 30000 nM T20251 CML2H3 11428837 IC50 = 7900 nM T20251 CREQ51 11429654 IC50 > 30000 nM T20251 C1YV6P 11442292 IC50 > 100000 nM T20251 CKU8Y3 11442383 IC50 = 18000 nM T20251 CG58SO 11444350 IC50 = 6309.57 nM T20251 CC9D4O 11444936 IC50 = 100 nM T20251 C07VBT 11445050 IC50 = 1900 nM T20251 CY7HT3 11452117 IC50 = 766 nM T20251 CQTM82 11452706 Ki > 150000 nM T20251 CE42DM 11453673 Ki = 1000 nM T20251 CP1WH5 11461365 Ki = 1100 nM T20251 CF6DQ2 11462727 IC50 = 40000 nM T20251 CKU5J7 11464405 IC50 = 4 nM T20251 C39QNY 11464915 IC50 = 500 nM T20251 CO95HP 11474838 IC50 = 19750 nM T20251 C3GMQ1 11477018 IC50 = 794.33 nM T20251 CH6X2L 11478011 IC50 = 6400 nM T20251 CRJ90F 11478858 IC50 = 870 nM T20251 C69PFD 11484605 IC50 > 30000 nM T20251 C8BY4A 11489501 IC50 = 501.19 nM T20251 CA8KE0 11492902 Ki > 20000 nM T20251 C1O9XD 11493620 IC50 = 240 nM T20251 CV41ER 11494867 IC50 = 2400 nM T20251 CXW96U 11495012 IC50 = 18000 nM T20251 CMQ86R 11495432 IC50 = 2530 nM T20251 C7H9AB 11495849 IC50 > 100000 nM T20251 CPX26I 11496746 IC50 = 50118.72 nM T20251 C5Z7GQ 11497411 IC50 = 251.19 nM T20251 CL17QT 11497455 IC50 > 10000 nM T20251 C9YU1O 11497679 IC50 = 1000 nM T20251 CQT5U8 11497680 IC50 = 1995.26 nM T20251 C9JD4N 11497924 IC50 = 1000 nM T20251 C69AMJ 11500781 IC50 = 910 nM T20251 C3B0LO 11501191 IC50 = 760 nM T20251 C6HM0U 11501983 IC50 > 10000 nM T20251 CZIE58 11502008 IC50 = 8.1 nM T20251 CI62OX 11502343 IC50 = 1800 nM T20251 CPO8S1 11502381 IC50 = 7900 nM T20251 CGB8M5 11502401 Ki = 30 nM T20251 C2TVA0 11502638 IC50 = 3800 nM T20251 C3ME1U 11502912 IC50 = 20000 nM T20251 C3ROH5 11504077 IC50 = 2511.89 nM T20251 COD9Z2 11504477 IC50 = 1300 nM T20251 CFSH67 11504490 IC50 = 10000 nM T20251 C10FVQ 11505089 IC50 = 800 nM T20251 C97WGN 11505187 IC50 = 7700 nM T20251 CHX56T 11508058 IC50 = 20200 nM T20251 CLPO39 11508317 Ki = 1100 nM T20251 CH75CA 11508844 IC50 = 4000 nM T20251 C7G4VM 11508924 IC50 = 12000 nM T20251 CV4IZ7 11509189 IC50 = 3036 nM T20251 CCP2Z0 11510399 IC50 = 1370 nM T20251 C72BCW 11510887 IC50 = 13.5 nM T20251 C1LCD7 11510932 IC50 = 560 nM T20251 CF45XR 11511026 Ki = 10 nM T20251 COT4H9 11511117 IC50 = 10000 nM T20251 CE62TB 11511267 IC50 = 1500 nM T20251 C2T8YD 11511361 IC50 > 10000 nM T20251 CP8B7T 11511719 IC50 > 10000 nM T20251 C9DE5V 11511776 IC50 = 490 nM T20251 CDQ18N 11515125 IC50 > 5000 nM T20251 CP9RB7 11515387 Ki > 3000 nM T20251 C23DKS 11516307 Ki = 160 nM T20251 CO0T6Q 11516310 Ki = 910 nM T20251 CS24AX 11516386 IC50 = 2800 nM T20251 CNM42D 11516387 IC50 = 5000 nM T20251 C6X1AJ 11516392 Ki = 710 nM T20251 CZ4OM7 11516508 IC50 = 1730 nM T20251 CVNP35 11517292 IC50 > 3200 nM T20251 C20FMG 11517340 IC50 = 10000 nM T20251 CPQN50 11517341 IC50 = 10000 nM T20251 CTA7M3 11517739 IC50 = 4600 nM T20251 CG3BZ9 11517980 IC50 = 137000 nM T20251 CW68BJ 11518143 IC50 = 14500 nM T20251 CLGO54 11518300 IC50 = 9190 nM T20251 C1KL7T 11518341 IC50 = 4000 nM T20251 CZ3D5Y 11518933 IC50 > 10000 nM T20251 C0WU7G 11518972 IC50 = 125.89 nM T20251 CM4B3J 11519133 IC50 = 6309.57 nM T20251 C08JSL 11519134 IC50 = 5011.87 nM T20251 CY47AQ 11519784 IC50 > 10000 nM T20251 C04RCG 11519858 IC50 = 7943.28 nM T20251 CM09RF 11524148 Ki = 690 nM T20251 CL09JW 11524225 IC50 = 2000 nM T20251 CBRO68 11524900 Ki = 4100 nM T20251 CU7B8I 11525190 IC50 = 110000 nM T20251 CR83WI 11525569 IC50 = 2500 nM T20251 CTNX29 11526451 IC50 = 1000 nM T20251 CR9NA7 11526531 IC50 = 1000 nM T20251 C0O3XD 11527019 IC50 = 58500 nM T20251 CEX8Y5 11527102 IC50 > 10000 nM T20251 CNL15V 11527195 IC50 = 10000 nM T20251 C0BF5R 11527661 IC50 > 30 nM T20251 C75FPD 11529874 Ki = 2840 nM T20251 C0BC6Y 11530223 Ki > 5000 nM T20251 C7NO5X 11531213 Ki = 1000 nM T20251 CZ93HX 11531536 Ki = 710 nM T20251 C94AGK 11531634 Ki = 5000 nM T20251 CS7Q6G 11532065 Ki = 70 nM T20251 CDX19H 11532153 Ki = 42 nM T20251 C89JTB 11532924 IC50 = 1800 nM T20251 C4W2IN 11533195 IC50 = 23900 nM T20251 CFU5V9 11533398 Ki = 800 nM T20251 CJF92G 11533429 IC50 = 3981.07 nM T20251 C2EQ1U 11533448 IC50 = 3981.07 nM T20251 C4LOQ9 11533473 IC50 = 1258.93 nM T20251 CZW9U3 11534726 IC50 = 1995.26 nM T20251 CR53ZL 11537871 IC50 = 18000 nM T20251 C29LCK 11537876 IC50 > 63000 nM T20251 C7R3HN 11538251 Ki = 2200 nM T20251 C8GZ1I 11539020 IC50 = 10000 nM T20251 CIR9M2 11539598 Ki = 16 nM T20251 CSN91H 11539722 IC50 = 6309.57 nM T20251 CJGL17 11539751 IC50 = 19054.61 nM T20251 C0J9NF 11539823 Ki = 3800 nM T20251 CIJ51X 11539903 IC50 = 38000 nM T20251 C0X6CJ 11540474 IC50 = 5011.87 nM T20251 CFS7T8 11540675 IC50 = 17100 nM T20251 CBR9K8 11541314 IC50 > 100000 nM T20251 C8P5GF 11541506 Ki > 10000 nM T20251 CY0JX9 11541985 IC50 = 8428 nM T20251 C5JEZ9 11544171 IC50 < 31622.78 nM T20251 C9UG2V 11544758 Ki > 40000 nM T20251 CS0B4G 11544795 IC50 = 940 nM T20251 CX0DJ3 11545423 Ki = 8252 nM T20251 CF52ZB 11545686 IC50 = 5940 nM T20251 CGE5W7 11546121 Ki = 2800 nM T20251 CFNG56 11546387 Ki = 430 nM T20251 CHT8D7 11547260 IC50 > 30000 nM T20251 CD14OF 11547466 IC50 = 1000 nM T20251 C61LDE 11548217 IC50 = 630.96 nM T20251 CKZ9B0 11548239 IC50 = 158.49 nM T20251 CPA7K8 11548755 IC50 = 251.19 nM T20251 C34JAV 11551351 Ki > 5000 nM T20251 C3DG8U 11552010 IC50 = 340 nM T20251 CCLR26 11552773 IC50 = 19000 nM T20251 CKGI84 11553070 IC50 = 2100 nM T20251 CH0E4A 11553554 Ki = 3100 nM T20251 CKT1O8 11554040 Ki = 2600 nM T20251 CA16WP 11554165 IC50 > 90000 nM T20251 CZD24Q 11554412 IC50 = 47400 nM T20251 CMC79Y 11554762 Ki = 4200 nM T20251 C0VMG7 11555265 IC50 = 251.19 nM T20251 C64NID 11555572 IC50 = 16000 nM T20251 C3Y4GR 11555971 IC50 = 5011.87 nM T20251 CNWU65 11556070 IC50 = 1750 nM T20251 C3RMI1 11559300 IC50 = 5030 nM T20251 C5WKO2 11559625 IC50 > 10 nM T20251 CXR53E 11561126 IC50 = 30 nM T20251 CX1VD8 11562113 IC50 = 1258.93 nM T20251 C0JU9T 11562199 IC50 = 5011.87 nM T20251 CD9SM0 11562361 IC50 > 10000 nM T20251 CQ8CJ9 11562662 IC50 = 10000 nM T20251 C7B4YX 11563243 Ki > 10000 nM T20251 C1VF0P 11566266 IC50 = 1080 nM T20251 CDP9Z0 11566316 IC50 > 20000 nM T20251 C8C1VW 11566318 IC50 > 18700 nM T20251 CCQ8O9 11567495 IC50 = 4300 nM T20251 CZMB92 11567596 IC50 = 2900 nM T20251 CP7W6H 11567952 IC50 = 4300 nM T20251 CJ3FH6 11568363 IC50 = 80 nM T20251 C52PDV 11568714 IC50 = 3162.28 nM T20251 CMFZ35 11568741 IC50 = 10000 nM T20251 CNV08X 11569158 IC50 = 14000 nM T20251 C0J3VR 11569300 IC50 = 2.5 nM T20251 CU6EY8 11569996 IC50 = 1000 nM T20251 CB59HM 11570626 IC50 > 10000 nM T20251 CZD62R 11572546 Ki = 8000 nM T20251 C18BAJ 11572597 IC50 = 27700 nM T20251 C12VCK 11573765 IC50 = 20000 nM T20251 CMX60P 11573849 IC50 > 6870 nM T20251 C3UQL8 11573971 IC50 = 3500 nM T20251 C86YFM 11575878 IC50 < 25118.86 nM T20251 CFC7D3 11576079 IC50 = 9000 nM T20251 CTVX46 11576269 IC50 > 10000 nM T20251 CASH81 11576387 IC50 = 1258.93 nM T20251 C8JW7U 11577059 IC50 = 11000 nM T20251 C8YLD3 11577158 IC50 = 3162.28 nM T20251 CN87ZF 11577588 IC50 = 1550 nM T20251 CR8E2F 11578028 IC50 = 3162.28 nM T20251 CXP2M0 11580426 Ki > 5000 nM T20251 CW7G3X 11580427 Ki > 5 nM T20251 C7I5KM 11581252 Ki = 5200 nM T20251 CE0U8J 11581337 IC50 = 2900 nM T20251 CN1I8D 11581636 IC50 = 6300 nM T20251 CZ28HJ 11581919 IC50 = 6600 nM T20251 CICM46 11582059 Ki = 1600 nM T20251 CVIP95 11582321 IC50 = 2000 nM T20251 C2DG4A 11582651 IC50 = 930 nM T20251 CM0H2R 11583049 IC50 = 6.2 nM T20251 CZ6C8H 11583193 IC50 = 51100 nM T20251 CP53LK 11583743 IC50 > 10000 nM T20251 CP07QN 11583835 IC50 = 450 nM T20251 C0HFP7 11584185 IC50 = 398.11 nM T20251 C6D1MA 11584660 IC50 = 1995.26 nM T20251 CU4J2W 11584694 IC50 = 31.62 nM T20251 CN5DQ9 11585034 IC50 = 2511.89 nM T20251 C73UHS 11585248 IC50 = 1584.89 nM T20251 CR78YS 11585375 IC50 < 1200 nM T20251 CY3A4K 11587772 IC50 = 2270 nM T20251 C5JBF8 11589054 IC50 < 25118.86 nM T20251 COE14C 11589812 IC50 = 6080 nM T20251 CA2KX0 11590078 IC50 > 10000 nM T20251 C7A3OZ 11590444 IC50 < 31622.78 nM T20251 CC75MD 11590828 IC50 = 3981.07 nM T20251 CK4E6V 11591222 IC50 = 12000 nM T20251 CYX50J 11591601 IC50 = 1000 nM T20251 CIUL60 11591633 IC50 = 251.19 nM T20251 CD6Y3F 11592099 IC50 = 11000 nM T20251 C47TZG 11595633 IC50 = 14000 nM T20251 C1A3PZ 11595635 IC50 = 31600 nM T20251 CMAF85 11596311 IC50 = 9.8 nM T20251 COS24N 11596426 IC50 = 8100 nM T20251 C5NRD9 11596521 Ki = 390 nM T20251 CAU85E 11597758 IC50 = 2400 nM T20251 C3LO6F 11597868 IC50 = 7079.46 nM T20251 CH0OD8 11598084 IC50 < 300 nM T20251 C1TOP5 11598123 IC50 = 2511.89 nM T20251 C6KVY0 11598137 IC50 = 9600 nM T20251 CP56DO 11599295 IC50 > 10000 nM T20251 CKI9D5 11599973 IC50 > 31600 nM T20251 CY72UC 11602409 IC50 > 1500 nM T20251 C1GL6E 11602780 IC50 = 3698.63 nM T20251 C7T3WI 11603194 Ki = 480 nM T20251 CRDU82 11603367 IC50 = 11600 nM T20251 C8GVH9 11603554 IC50 = 22387.21 nM T20251 C04ORX 11603648 Ki = 5000 nM T20251 CPXV24 11603996 IC50 > 100000 nM T20251 CH4AE5 11604196 Ki = 6400 nM T20251 C3V9LT 11604824 IC50 = 70000 nM T20251 COI0G2 11605470 Ki = 89 nM T20251 C9DI6R 11606176 IC50 = 19952.62 nM T20251 CO1A5Z 11606378 IC50 = 2511.89 nM T20251 CL04ZJ 11606435 IC50 = 1000 nM T20251 CJC5N8 11606456 IC50 = 3981.07 nM T20251 C83DCU 11609760 IC50 = 2800 nM T20251 C6HLN8 11610150 IC50 = 2810 nM T20251 CC5R1Q 11610423 Ki = 200 nM T20251 CAU61Q 11610483 IC50 = 3550 nM T20251 CD2PU0 11610816 IC50 > 10000 nM T20251 CTF7J8 11611218 IC50 > 30000 nM T20251 COW93C 11611844 IC50 > 63000 nM T20251 C1WI4H 11611859 IC50 = 6100 nM T20251 CZ4B9T 11612643 IC50 = 7500 nM T20251 C6LUG4 11612700 IC50 > 10000 nM T20251 CT16JP 11613587 IC50 = 199.53 nM T20251 CQL5S8 11613750 IC50 = 16000 nM T20251 CN91SZ 11613873 IC50 = 2511.89 nM T20251 C3FQP1 11614515 IC50 = 2100 nM T20251 C8JAM4 11616357 Ki = 12000 nM T20251 CD28IH 11618024 IC50 = 5600 nM T20251 CA5W9R 11618060 EC50 = 9000 nM T20251 C36OSA 11618702 IC50 = 1100 nM T20251 C1GB6K 11618861 Ki = 1500 nM T20251 CA6X1R 11619076 IC50 < 25118.86 nM T20251 CG1RP5 11619850 IC50 = 1.4 nM T20251 CJ73BI 11619909 IC50 = 10000 nM T20251 CKB59U 11620847 IC50 = 3981.07 nM T20251 CXY07A 11621352 IC50 = 251.19 nM T20251 C79OMR 11623756 Ki > 5 nM T20251 C1KD4Z 11623823 IC50 = 40200 nM T20251 CSB9O5 11623845 Ki > 5000 nM T20251 CD2H3T 11624832 IC50 = 18000 nM T20251 C9WMX4 11624970 IC50 = 500 nM T20251 CX1M6Z 11625277 IC50 = 1800 nM T20251 C34OQC 11626062 IC50 = 1000 nM T20251 C6EGB7 11626833 IC50 = 54000 nM T20251 C7C8FX 11626984 Ki = 42 nM T20251 CIO53A 11627085 IC50 > 31600 nM T20251 C3CP2G 11627368 IC50 > 3200 nM T20251 C9FSA8 11627847 IC50 = 1995.26 nM T20251 C51IBH 11627879 IC50 = 5011.87 nM T20251 CEK0Z8 11628328 IC50 > 31600 nM T20251 CE8W1Z 11628452 IC50 = 501.19 nM T20251 CFJN71 11628631 IC50 = 100 nM T20251 C95RDI 11631662 IC50 > 30000 nM T20251 C0G6PN 11632103 IC50 > 10000 nM T20251 CPV49C 11632254 IC50 = 1000 nM T20251 CNS5P7 11632418 IC50 = 1600 nM T20251 C9HCM6 11632711 Ki = 340 nM T20251 CK34LS 11632737 IC50 = 16600 nM T20251 C7H0AV 11633028 Ki = 1500 nM T20251 C1R2BZ 11633045 IC50 = 12600 nM T20251 CWE63G 11633344 IC50 < 25118.86 nM T20251 CD83GL 11634069 IC50 = 36000 nM T20251 CJBR83 11634073 IC50 = 17000 nM T20251 COB0P4 11634166 Ki = 5100 nM T20251 CO68YB 11634336 IC50 = 31000 nM T20251 CYL45U 11634544 IC50 > 10000 nM T20251 C52ZKM 11634651 IC50 > 10000 nM T20251 C75FNR 11634886 IC50 = 1730 nM T20251 CDE1G8 11635187 IC50 > 31600 nM T20251 C8Y9AL 11635230 IC50 > 31600 nM T20251 CUN3R9 11635332 IC50 > 31600 nM T20251 C23XSL 11638166 Ki = 1800 nM T20251 CCE90V 11638319 IC50 > 60000 nM T20251 CQ1U9W 11638962 IC50 = 7570 nM T20251 COLF16 11639342 IC50 = 213000 nM T20251 CR5QB1 11640354 Ki = 930 nM T20251 CIMW51 11640376 Ki = 3800 nM T20251 CY3IN5 11640515 IC50 = 8300 nM T20251 CMNV51 11640588 Ki = 400 nM T20251 CI2KZ1 11641036 IC50 = 170 nM T20251 CWHK19 11641315 IC50 = 11000 nM T20251 C0XC2N 11641596 IC50 = 3981.07 nM T20251 C25KGE 11641641 IC50 = 251.19 nM T20251 C8DXS0 11642163 IC50 = 794.33 nM T20251 CSE96X 11645396 Ki = 3000 nM T20251 CDP23M 11645473 IC50 = 6400 nM T20251 C0M9NX 11646364 Ki = 2100 nM T20251 CW42YV 11646372 IC50 = 7400 nM T20251 CLR3P8 11646541 IC50 = 10000 nM T20251 C24DVX 11647025 Ki = 2600 nM T20251 C9IOM8 11647276 IC50 = 1300 nM T20251 CJQK24 11647458 IC50 = 34600 nM T20251 C6Y4HR 11647548 IC50 > 30000 nM T20251 CPO25R 11647576 IC50 = 4000 nM T20251 C83VLD 11648483 Ki = 1200 nM T20251 CYQB50 11648990 IC50 = 794.33 nM T20251 C0WAT8 11649549 IC50 = 42000 nM T20251 CXG1B4 11649741 IC50 > 100000 nM T20251 CZPG34 11650178 IC50 > 10000 nM T20251 CM5PG0 11653478 Ki = 10000 nM T20251 CEXK54 11653686 IC50 = 15190 nM T20251 C8I7UT 11654412 IC50 = 9 nM T20251 C2R9QT 11654739 Ki = 300 nM T20251 CGU87J 11654962 IC50 = 6300 nM T20251 C0EF3I 11655513 IC50 = 36900 nM T20251 CPH9X5 11655664 IC50 = 4100 nM T20251 CX7FR8 11655728 IC50 > 10000 nM T20251 C48HCV 11656243 IC50 = 2511.89 nM T20251 CVY3H4 11656753 IC50 = 5610 nM T20251 CPE83G 11656848 IC50 = 1258.93 nM T20251 CT14BC 11657494 IC50 = 251.19 nM T20251 CH3N1I 11659592 IC50 = 490 nM T20251 CF92SM 11659664 IC50 = 24700 nM T20251 CC36GP 11660512 Ki = 10000 nM T20251 CR92TH 11660563 IC50 = 3450 nM T20251 CN6Y7D 11661294 IC50 = 7900 nM T20251 C4G9CM 11661358 IC50 > 10000 nM T20251 CMC02O 11661752 Ki = 8700 nM T20251 CXPC31 11662060 IC50 > 100000 nM T20251 CEL15N 11662194 IC50 > 63095.73 nM T20251 C1F9VA 11662657 IC50 = 15600 nM T20251 CKP76R 11662966 IC50 = 10000 nM T20251 CT2AZ4 11663315 Ki = 380 nM T20251 CBU0L8 11663504 IC50 = 5011.87 nM T20251 C69RQX 11663526 IC50 = 2511.89 nM T20251 C3SJO5 11663578 IC50 = 794.33 nM T20251 C1PB0O 11663999 IC50 = 1258.93 nM T20251 C16UWH 11664328 IC50 = 5011.87 nM T20251 CO15KF 11664409 IC50 > 10000 nM T20251 CG3W2T 11666681 Ki = 31000 nM T20251 CPW3A8 11667985 IC50 = 6600 nM T20251 CJSN27 11668594 IC50 = 3000 nM T20251 C64GUF 11668827 Ki = 7900 nM T20251 CFEQ23 11669001 Ki = 5100 nM T20251 C5SJ9K 11669355 Ki = 700 nM T20251 CNE2K5 11669953 IC50 = 25118.86 nM T20251 CU9P5O 11670029 Ki = 900 nM T20251 CPVR45 11670647 IC50 = 794.33 nM T20251 CE6A2S 11671079 IC50 = 780 nM T20251 CX1GS0 11672017 IC50 = 1220 nM T20251 CON70D 11672049 IC50 = 7900 nM T20251 CT3BP5 11674529 IC50 > 10000 nM T20251 CD9XU6 11675152 IC50 < 25118.86 nM T20251 C7A0WS 11675333 IC50 > 10000 nM T20251 C0V7SU 11675388 IC50 = 5235 nM T20251 C29PWK 11675645 IC50 = 1300 nM T20251 CXB59V 11676220 IC50 = 1.7 nM T20251 CX04MA 11676364 IC50 > 150000 nM T20251 CFQP90 11676381 Ki = 62 nM T20251 C3US8X 11676399 Ki = 720 nM T20251 CY5UB8 11676600 Ki = 260 nM T20251 C6GVU2 11676790 IC50 = 31600 nM T20251 CWQ3M4 11677768 IC50 = 1584.89 nM T20251 C6C4BJ 11678080 IC50 = 1995.26 nM T20251 C34RDZ 11678857 Ki = 364 nM T20251 C7JVX2 11681378 Ki > 5000 nM T20251 C7T9ES 11681588 IC50 = 27000 nM T20251 C8RA5V 11682068 IC50 > 10000 nM T20251 C2JSO8 11683474 IC50 < 31622.78 nM T20251 CEHG64 11683903 IC50 = 15.9 nM T20251 CI6JR2 11684405 IC50 = 6300 nM T20251 C1ZD6V 11685267 IC50 = 1258.93 nM T20251 C9K3EO 11688027 IC50 > 60000 nM T20251 CY36RI 11688223 IC50 = 220 nM T20251 CD1O9I 11688761 IC50 > 1000 nM T20251 C87TCD 11689687 IC50 = 1700 nM T20251 C6S2GN 11689802 IC50 = 400 nM T20251 CR91QA 11690139 IC50 = 5000 nM T20251 CRXO13 11690171 Ki = 1200 nM T20251 CG13YQ 11691697 IC50 = 1258.93 nM T20251 CE1KI3 11692214 IC50 = 501.19 nM T20251 CKX65Z 11692293 IC50 = 66000 nM T20251 CGM36K 11692376 IC50 = 1584.89 nM T20251 C7Z0SX 11695591 IC50 = 2300 nM T20251 CFGR63 11695646 IC50 = 15000 nM T20251 CP3G0Q 11695811 IC50 = 1800 nM T20251 CLT3Z7 11695929 EC50 = 5000 nM T20251 CWX2F0 11696319 IC50 = 940 nM T20251 C8QIH0 11696657 IC50 = 2000 nM T20251 CDV58J 11696813 Ki = 930 nM T20251 CX7MT8 11697412 Ki = 500 nM T20251 C8K3OV 11698389 Ki = 150 nM T20251 CT5J9M 11699340 IC50 = 1584.89 nM T20251 CFCB20 11699532 IC50 = 316.23 nM T20251 C4DJ1V 11699804 IC50 > 10000 nM T20251 CBDC74 11702114 IC50 = 590 nM T20251 CQ5P2F 11702115 IC50 = 890 nM T20251 CXFK83 11702578 Ki > 5000 nM T20251 CZ9SY1 11702625 IC50 = 75000 nM T20251 C5UEI7 11703527 Ki = 320 nM T20251 C9SX7H 11704191 Ki = 13000 nM T20251 C3XDB2 11704592 IC50 = 4100 nM T20251 CTZ61B 11704809 IC50 > 95000 nM T20251 CGD80W 11705119 IC50 = 5011.87 nM T20251 CH5B6O 11705343 IC50 = 32000 nM T20251 C2E8BF 11705395 Ki = 30 nM T20251 CLK68A 11705570 IC50 = 1995.26 nM T20251 CPC67X 11705929 IC50 = 501.19 nM T20251 CG2LE3 11706442 IC50 = 3800 nM T20251 CE1FU8 11706443 IC50 = 2300 nM T20251 C04VLB 11706579 Ki > 10000 nM T20251 CG0B5Q 11706981 IC50 = 3300 nM T20251 C3M8DW 11709098 IC50 = 16200 nM T20251 CXMH25 11710453 Ki = 2000 nM T20251 C4M9AU 11710505 IC50 = 2950 nM T20251 CK1FB9 11710573 IC50 < 25118.86 nM T20251 C12EZH 11710694 Ki = 10000 nM T20251 C5FZ1J 11710873 Ki = 3000 nM T20251 C6CM7S 11711078 IC50 = 7900 nM T20251 CIZQ65 11711452 IC50 = 5280 nM T20251 CIUV17 11711973 IC50 = 800 nM T20251 CN8FE3 11712044 IC50 = 15848.93 nM T20251 C9WI7N 11712071 IC50 = 8317.64 nM T20251 CLY3T0 11712237 IC50 = 8000 nM T20251 C5RZ3S 11712530 Ki = 200 nM T20251 CL3H6E 11712583 IC50 = 1200 nM T20251 CHK5I2 11712756 IC50 = 1584.89 nM T20251 C8V9XO 11712898 IC50 = 560 nM T20251 CWQ67V 11713742 IC50 = 9180 nM T20251 C1XYK2 11717025 IC50 = 17000 nM T20251 CI1C4Z 11718272 Ki = 400 nM T20251 C74DRE 11719291 IC50 = 85500 nM T20251 C9R0FW 11719590 IC50 > 10000 nM T20251 CO29BN 11719912 IC50 = 3080 nM T20251 CD9A0J 11720104 IC50 > 10000 nM T20251 C3FP8J 11720191 IC50 = 5600 nM T20251 CX9VH0 11720815 IC50 = 1000 nM T20251 CXUM63 11720838 IC50 = 794.33 nM T20251 C37DMH 11721190 IC50 = 794.33 nM T20251 CIH38K 11723422 Ki = 10000 nM T20251 CP7EV6 11731453 Ki = 21000 nM T20251 CB8N9K 11732098 IC50 = 11000.01 nM T20251 CA7FS4 11732896 IC50 = 2600 nM T20251 CT23IZ 11742071 IC50 = 6.918 nM T20251 CM95SZ 11744578 Ki = 530 nM T20251 CG0YB2 11751828 IC50 = 390 nM T20251 C4L9EC 11752457 IC50 = 24000 nM T20251 C41OBD 11756414 IC50 = 4000 nM T20251 CKW9D4 11756884 IC50 = 17000 nM T20251 C58DMZ 11757696 IC50 = 3200 nM T20251 CZ8E3X 11771731 IC50 < 1000 nM T20251 C7JD4S 11775505 IC50 = 10.5 nM T20251 C5QGC3 11775544 IC50 = 3162.28 nM T20251 CHS9Q3 11785237 IC50 = 5000 nM T20251 CD13QV 11786769 IC50 = 2800 nM T20251 COB43E 11825520 Ki = 150 nM T20251 CG6Q1B 11842628 IC50 = 19700 nM T20251 CD0F5T 11842667 IC50 = 15135.61 nM T20251 CBC08P 11846124 IC50 > 100000 nM T20251 C5LIW2 11846126 IC50 > 100000 nM T20251 CAD8P9 11848624 IC50 < 100 nM T20251 CCT5G7 11848677 IC50 = 3500 nM T20251 CL6B5X 11848835 IC50 = 430 nM T20251 C3UQT0 11853349 IC50 = 2000 nM T20251 C8VK4D 11853588 IC50 = 13000 nM T20251 CYLO43 11854292 Ki = 1900 nM T20251 C1YD8G 11857777 IC50 = 954992586 nM T20251 CXLW54 11948707 Ki > 10000 nM T20251 CP79ZF 11949710 IC50 = 3900 nM T20251 CQSU51 11950826 IC50 = 14125.38 nM T20251 C85VJZ 11950827 IC50 = 1905.46 nM T20251 CQVX45 11950828 IC50 = 208.93 nM T20251 C0WVX4 11951000 IC50 = 8511.38 nM T20251 C0HT7M 11951722 IC50 = 28000 nM T20251 CTR9Z0 11951723 IC50 = 14200 nM T20251 C4EVI9 11951724 IC50 > 30000 nM T20251 CFYK69 11951728 IC50 = 2700 nM T20251 C5M9VQ 11951901 IC50 > 31600 nM T20251 C0GLF5 11952264 IC50 = 11600 nM T20251 CJLB31 11952265 IC50 = 7700 nM T20251 C4JE5Y 11952437 IC50 = 4100 nM T20251 CS3FO8 11952438 IC50 = 6700 nM T20251 CB0LK9 11952439 IC50 = 2400 nM T20251 CK13QD 11953409 IC50 = 6000 nM T20251 C8SZH2 11965686 IC50 = 1995.26 nM T20251 C38ACD 11973711 Ki = 107 nM T20251 CA54WB 11973799 IC50 = 5.4 nM T20251 C09SBY 11973800 IC50 = 21.2 nM T20251 C4G3JS 11973801 IC50 = 14.7 nM T20251 CJ51DI 11973802 IC50 = 47.7 nM T20251 C68TIS 11974129 IC50 = 63.7 nM T20251 CU3J7M 11974130 IC50 = 7.4 nM T20251 CN38YH 11974131 IC50 = 5 nM T20251 C5W7EA 11974229 IC50 = 5.6 nM T20251 C3C2EN 11974230 IC50 = 12.2 nM T20251 CAN81B 11974231 IC50 = 10.4 nM T20251 CNCP71 11974346 IC50 = 20.3 nM T20251 C7W6UZ 11975326 IC50 = 6.7 nM T20251 C3EU8T 11975438 IC50 = 19.9 nM T20251 CN5W3V 11978858 Ki = 10000 nM T20251 C1O8ZJ 11983278 Ki > 9000 nM T20251 CHC85I 11983362 IC50 = 34000 nM T20251 CZ9FS3 11990142 Ki > 9000 nM T20251 C0KM5I 11992827 IC50 = 4500 nM T20251 C56OSH 11995342 IC50 = 21877.62 nM T20251 C0SMQ3 11995420 IC50 = 135000 nM T20251 C9KSG8 11995421 IC50 = 16000 nM T20251 CEYB03 11995422 IC50 > 30000 nM T20251 C58BPD 11995424 IC50 = 21000 nM T20251 CTYE90 11995521 IC50 = 10000 nM T20251 C0DE5H 11995522 IC50 = 76000 nM T20251 CR4YS2 11996303 IC50 = 794.33 nM T20251 C7D1AY 11996304 IC50 = 1258.93 nM T20251 C1A2IB 12001199 IC50 = 1584.89 nM T20251 CNO57E 12001832 IC50 > 50118.72 nM T20251 C1QBK8 12094039 IC50 = 9800 nM T20251 C4CE8D 12111141 Ki = 4000 nM T20251 C5P6ND 12429371 IC50 = 1608 nM T20251 CZ1V4O 12896968 IC50 = 1120 nM T20251 CCS5B1 12951762 IC50 = 506 nM T20251 C7BE0Q 12991318 IC50 = 31600 nM T20251 CM6IO1 14645090 Ki = 24 nM T20251 CIJA82 14645095 Ki = 1.6 nM T20251 C3S8RY 14793784 IC50 = 163.9 nM T20251 C0TO1Z 14921509 IC50 = 17 nM T20251 C0I8GC 14985965 IC50 = 190 nM T20251 CE78SG 15006442 IC50 = 10 nM T20251 C8BF2P 15254720 IC50 = 199.53 nM T20251 C60TVD 15392306 Ki = 3900 nM T20251 C9ZO7G 15604796 IC50 = 19300 nM T20251 CCDX50 15940498 IC50 > 50000 nM T20251 C8JIP7 15940801 IC50 = 16000 nM T20251 CBE59I 15940927 Ki = 5800 nM T20251 CTH2A9 15941083 IC50 = 8400 nM T20251 CF30UM 15941086 IC50 = 10800 nM T20251 CM10PF 15941255 IC50 = 300 nM T20251 CHFW18 15942650 IC50 = 35000 nM T20251 CB8H6M 15947119 IC50 = 250 nM T20251 CPD3V1 15949508 IC50 = 4800 nM T20251 CLD0M2 15949839 IC50 = 33000 nM T20251 CUS3W4 15950258 IC50 = 25000 nM T20251 CM63YP 15950387 IC50 = 14000 nM T20251 C9KJ6D 15950538 IC50 > 80000 nM T20251 C4S7AB 15950540 IC50 > 80000 nM T20251 C3U1VO 15950542 IC50 > 80000 nM T20251 CKX8M6 15950615 IC50 > 80000 nM T20251 C2ZYA6 15951338 IC50 = 39000 nM T20251 C1Q8IV 15951410 IC50 = 23000 nM T20251 C8IJ0O 15952316 IC50 = 1300 nM T20251 CWZM24 15953526 IC50 = 13400 nM T20251 CSA02I 15979148 IC50 = 2778 nM T20251 CBE54Y 15979149 IC50 = 5312 nM T20251 C9QO8U 15979276 IC50 > 10000 nM T20251 C3W8ZL 15981007 IC50 = 290 nM T20251 C8VYW0 15981180 IC50 = 10100 nM T20251 CE4VG5 15981891 IC50 = 24300 nM T20251 C3L4HO 15981894 IC50 = 14800 nM T20251 CB76UT 15981895 IC50 = 49100 nM T20251 C5UOH2 15982018 IC50 = 20000 nM T20251 CI1SK2 15982019 IC50 > 100000 nM T20251 CXD9I3 15982149 IC50 = 50700 nM T20251 CX3M7T 15982150 IC50 > 100000 nM T20251 CP3N4C 15982151 IC50 = 42000 nM T20251 CS9N5F 15982407 IC50 = 40000 nM T20251 CAB1P3 15982533 IC50 = 19000 nM T20251 CD34SB 15982534 IC50 = 35000 nM T20251 CG50BK 15983304 IC50 = 44000 nM T20251 C5OY3I 15983430 IC50 = 29000 nM T20251 CBE59Y 15983549 IC50 = 13000 nM T20251 C6YAJ0 15983550 IC50 = 12900 nM T20251 CUX86I 15983552 IC50 = 6000 nM T20251 CO02BA 15983553 IC50 = 9000 nM T20251 C9TO6J 15983677 IC50 = 3000 nM T20251 CIV82J 15983679 IC50 = 41000 nM T20251 C30OTX 15983680 IC50 = 1400 nM T20251 CT2G7E 15983809 IC50 = 2800 nM T20251 C0GMT8 15983810 IC50 > 100000 nM T20251 CPR25X 15986917 IC50 < 31622.78 nM T20251 CRBP36 15987008 IC50 = 6309.57 nM T20251 C5KW3L 15987108 IC50 = 9332.54 nM T20251 CF6S2D 15987282 IC50 < 63095.73 nM T20251 CXU15Z 15987451 IC50 = 7943.28 nM T20251 C6V3WY 15987452 IC50 < 15848.93 nM T20251 C0HKS9 16004748 IC50 > 10000 nM T20251 CV0YA4 16005493 IC50 = 8410 nM T20251 CG8KR9 16005860 IC50 = 4114 nM T20251 C70KBE 16006079 IC50 = 2220 nM T20251 CCL59Z 16007088 IC50 = 1900 nM T20251 CG5A7W 16013152 IC50 > 30000 nM T20251 CBMF65 16013184 IC50 > 30000 nM T20251 C6V4TG 16013186 IC50 > 30000 nM T20251 CUB5X2 16038385 IC50 > 63095.73 nM T20251 C8AB4L 16039796 IC50 = 18000 nM T20251 CA7QW1 16039834 IC50 = 40000 nM T20251 CPCZ62 16040329 IC50 = 19000 nM T20251 C20CRP 16040587 IC50 > 31622.78 nM T20251 CH8K6G 16040671 IC50 = 31622.78 nM T20251 C8ZP3G 16041292 IC50 > 25118.86 nM T20251 CDU1L0 16041411 IC50 > 30000 nM T20251 CGM4N8 16041594 IC50 > 40000 nM T20251 C1V9EY 16041612 IC50 > 10000 nM T20251 CX9W7Q 16043220 IC50 = 690 nM T20251 CJ78MO 16045297 Ki = 31622.78 nM T20251 CB64EN 16049818 IC50 > 30000 nM T20251 CU27FI 16049886 IC50 = 156666.67 nM T20251 CZC7L2 16049887 IC50 = 115000 nM T20251 CQ9U1Y 16051921 IC50 = 2400 nM T20251 CS8NZ0 16059780 Ki = 6200 nM T20251 C6V4HS 16059786 IC50 = 440 nM T20251 CC2YJ8 16062553 IC50 > 10000 nM T20251 C1LH5T 16062816 IC50 > 10000 nM T20251 C7UCS5 16064456 Ki > 20000 nM T20251 CEZI54 16064872 IC50 = 37153.52 nM T20251 C0V9RI 16064896 Ki > 20000 nM T20251 CM1V6L 16064897 Ki > 20000 nM T20251 C96FEP 16065425 IC50 = 20892.96 nM T20251 CVCJ16 16065428 IC50 = 7762.47 nM T20251 C6MC0Z 16065567 IC50 = 30199.52 nM T20251 CPN9H5 16065569 IC50 = 16595.87 nM T20251 CL1M3W 16065704 IC50 = 16595.87 nM T20251 CF3UG1 16066664 IC50 = 1100 nM T20251 C30UFT 16066811 Ki > 30000 nM T20251 CI1EC9 16068009 Ki = 17000 nM T20251 C3ZKJ5 16068120 Ki = 4400 nM T20251 CPLU48 16068121 Ki = 3800 nM T20251 C9S6QP 16068233 Ki = 13000 nM T20251 CB9Z0L 16068234 Ki = 2600 nM T20251 CW4U7H 16068235 Ki > 20000 nM T20251 CT4JA5 16068236 Ki > 20000 nM T20251 C8SQ5I 16068237 Ki = 6300 nM T20251 CVT0E7 16070046 Ki = 30000 nM T20251 CZ47FJ 16071018 IC50 = 12589.25 nM T20251 CQ06FD 16071731 IC50 = 28000 nM T20251 C3LK2C 16072132 IC50 = 8100 nM T20251 CBM80K 16091080 IC50 = 5319 nM T20251 CX5KI3 16105788 Ki > 10000 nM T20251 CKPQ93 16112836 IC50 = 1584.89 nM T20251 CZC0H1 16116961 IC50 = 25000 nM T20251 CYV05C 16123136 IC50 = 1000 nM T20251 C8C2IW 16123138 IC50 = 100 nM T20251 C7YF8I 16123140 IC50 = 1258.93 nM T20251 C91DQN 16123241 IC50 = 1584.89 nM T20251 CQG7P8 16123247 IC50 = 1258.93 nM T20251 CA6D4S 16123347 IC50 = 1258.93 nM T20251 CBH5P4 16123349 IC50 = 794.33 nM T20251 CPN48R 16123353 IC50 = 1995.26 nM T20251 CK7H2W 16123462 IC50 = 1258.93 nM T20251 C5MY2Q 16123464 IC50 = 10000 nM T20251 CNQ6J2 16123467 IC50 = 3162.28 nM T20251 CWU6P3 16123945 IC50 = 25118.86 nM T20251 CZF23I 16124479 Ki > 100000 nM T20251 C9G8TZ 16124598 IC50 > 31622.78 nM T20251 CYI7J5 16126731 Ki = 16 nM T20251 CTRP20 16190907 IC50 = 15500 nM T20251 CK8Z9L 16220221 IC50 = 2750 nM T20251 CFI8G2 16220223 IC50 = 5300 nM T20251 CTU7J0 16220225 IC50 > 10000 nM T20251 C0ZUH7 16220280 IC50 = 1800 nM T20251 C39SIQ 16220281 IC50 > 10000 nM T20251 C0JA4Q 16220791 IC50 = 5190 nM T20251 CWIT69 16220793 IC50 = 450 nM T20251 CI84RL 16220795 IC50 = 790 nM T20251 C3W1LK 16220874 IC50 = 2590 nM T20251 CUNW89 16220876 IC50 = 3590 nM T20251 C1VUC5 16220877 IC50 = 2500 nM T20251 CN91VO 16220879 IC50 = 3390 nM T20251 CVQ9T5 16220880 IC50 = 4800 nM T20251 C1U9XM