Drug Information
| Drug General Information | Top | |||
|---|---|---|---|---|
| Drug ID |
D0T1MP
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| Former ID |
DIB004073
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| Drug Name |
Lurosetron
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| Synonyms |
Lurosetron mesylate; GR-87442; GR-87442N
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| Drug Type |
Small molecular drug
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| Indication | Vomiting [ICD-11: MD90; ICD-10: R11; ICD-9: 787] | Discontinued in Phase 2 | [1] | |
| Company |
Glaxo Wellcome plc
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| Structure |
 |
Download2D MOL |
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| Formula |
C17H17FN4O
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| Canonical SMILES |
CC1=C(N=CN1)CN2CCC3=C(C2=O)C4=C(N3C)C(=CC=C4)F
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| InChI |
1S/C17H17FN4O/c1-10-13(20-9-19-10)8-22-7-6-14-15(17(22)23)11-4-3-5-12(18)16(11)21(14)2/h3-5,9H,6-8H2,1-2H3,(H,19,20)
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| InChIKey |
NUMKWGDDRWJQMY-UHFFFAOYSA-N
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| CAS Number |
CAS 128486-54-4
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| PubChem Compound ID | ||||
| Target and Pathway | Top | |||
|---|---|---|---|---|
| Target(s) | 5-HT 3 receptor (5HT3R) | Target Info | Modulator | [2] |
| References | Top | |||
|---|---|---|---|---|
| REF 1 | Trusted, scientifically sound profiles of drug programs, clinical trials, safety reports, and company deals, written by scientists. Springer. 2015. Adis Insight (drug id 800002948) | |||
| REF 2 | US patent application no. 7,932,267, Use of α-glucosidase inhibitors to treat alphavirus infections. | |||
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