Patent(s) and the Corresponding Patented Drug(s) |
Top |
World Intellectual Property Organization (WIPO) |
Patent ID |
WO2007019083 |
Title |
Pyrimidine Compounds As Serotonin Receptor Modulators. |
Abstract |
Certain pyrimidine-containing compounds are serotonin receptor modulators useful in the treatment of serotonin-mediated diseases. |
Applicant(s) |
Janssen Pharmaceutica Nv |
Representative Drug(s) |
D00YGY |
Drug Info
|
Ki = 30 nM |
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[1] |
2
|
D0B7NS
|
Drug Info
|
Ki = 70 nM
|
[1] |
3
|
D0P9VX
|
Drug Info
|
Ki = 250 nM
|
[1] |
4
|
D0N2VA
|
Drug Info
|
Ki = 900 nM
|
[1] |
5
|
D0SE9K
|
Drug Info
|
Ki = 1185 nM
|
[1] |
6
|
D08DJY
|
Drug Info
|
Ki = 2200 nM
|
[1] |
7
|
D0U9UH
|
Drug Info
|
Ki = 2250 nM
|
[1] |
Patent ID |
WO2010058858 |
Title |
Novel Pyrazole-3-Carboxamide Derivative Having 5-Ht2B Receptor Antagonist Activity. |
Abstract |
Disclosed is a compound represented by general formula (I) or a pharmaceutically acceptable salt thereof, which is useful as a selective antagonist of a 5-HT2B receptor.The compound and salt are useful for treatment or prevention of various diseases and conditions associated with a 5-HT2B receptor. |
Applicant(s) |
Raqualia Pharma Inc |
Representative Drug(s) |
D0D3BL |
Drug Info
|
N.A. |
[1] |
Patent ID |
WO2003091250 |
Title |
[1,4]Diazepino[6,7,1-Ij]Quinoline Derivatives As Anti Psychotic and Antiobesity Agents. |
Abstract |
Compounds of formula 1 or a pharmaceutically acceptable salt thereof are provided: I where R1 through R7 are defined herein. The compounds of formula I are 5HT2c agonists or partial agonists, and are useful for treating a variety of disorders. |
Applicant(s) |
RAMAMOORTHY, Sivaramakrishnan, P et al |
Representative Drug(s) |
D01LVT |
Drug Info
|
N.A. |
[1] |
United States Patent and Trademark Office (USPTO) |
Patent ID |
US8618288 |
Title |
Pyrimidine Compounds As Serotonin Receptor Modulators. |
Applicant(s) |
Janssen Pharmaceutica Nv |
Representative Drug(s) |
D00YGY |
Drug Info
|
Ki = 30 nM |
Click to Show More |
[1] |
2
|
D0B7NS
|
Drug Info
|
Ki = 70 nM
|
[1] |
3
|
D0P9VX
|
Drug Info
|
Ki = 250 nM
|
[1] |
4
|
D0N2VA
|
Drug Info
|
Ki = 900 nM
|
[1] |
5
|
D0SE9K
|
Drug Info
|
Ki = 1185 nM
|
[1] |
6
|
D08DJY
|
Drug Info
|
Ki = 2200 nM
|
[1] |
7
|
D0U9UH
|
Drug Info
|
Ki = 2250 nM
|
[1] |