Drug Information

Drug General Information
Drug ID
D0C2JS
Former ID
DIB019656
Drug Name
CPI-203
Synonyms
CPI203; CPI 203
Drug Type
Small molecular drug
Indication Discovery agent Investigative [542527]
Structure
Download
2D MOL
Formula
C19H18ClN5OS
InChI
InChI=1S/C19H18ClN5OS/c1-9-10(2)27-19-16(9)17(12-4-6-13(20)7-5-12)22-14(8-15(21)26)18-24-23-11(3)25(18)19/h4-7,14H,8H2,1-3H3,(H2,21,26)/t14-/m0/s1
InChIKey
QECMENZMDBOLDR-AWEZNQCLSA-N
PubChem Compound ID
71291068
PubChem Substance ID
172842964, 187051815, 198043960, 209266411, 210275381, 210281029, 239729098, 249714958, 249896068, 252158782, 252211774, 252451473, 252471207
Target and Pathway
Target(s) Bromodomain-containing protein 4 Target Info Inhibitor [531875]
WikiPathways Chemical Compounds to monitor Proteins
References
Ref 542527(http://www.guidetopharmacology.org/) Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 7513).
Ref 531875BRD4 is an atypical kinase that phosphorylates serine2 of the RNA polymerase II carboxy-terminal domain. Proc Natl Acad Sci U S A. 2012 May 1;109(18):6927-32.

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