Drug General Information
Drug ID D08FKE
Drug Name Aminoglycosides Drug Info
Drug Resistance Mutations
Target Name Bacterial 16S/23S rRNA (cytidine-2'-O)-methyltransferase (TlyA)
Gene Name tlyA
Uniprot ID TLYA_MYCTU
Species Mycobacterium tuberculosis
Reference Sequence MARRARVDAELVRRGLARSRQQAAELIGAGKVRIDGLPAVKPATAVSDTTALTVVTDSER
AWVSRGAHKLVGALEAFAIAVAGRRCLDAGASTGGFTEVLLDRGAAHVVAADVGYGQLAW
SLRNDPRVVVLERTNARGLTPEAIGGRVDLVVADLSFISLATVLPALVGCASRDADIVPL
VKPQFEVGKGQVGPGGVVHDPQLRARSVLAVARRAQELGWHSVGVKASPLPGPSGNVEYF
LWLRTQTDRALSAKGLEDAVHRAISEGP [Mycobacterium tuberculosis]
Targeted Disease Tuberculosis
Drug Resistance Mutations
Mutation info Missense: A91E [556229]
Mutation info Missense: L150P [556229]
Mutation info Missense: N236K [556229]
Mutation info Missense: R14W [556229]
References
Ref 1572605The ChEMBL database in 2017.
Ref 556229The comprehensive antibiotic resistance database. Antimicrob Agents Chemother. 2013 Jul;57(7):3348-57. doi: 10.1128/AAC.00419-13. Epub 2013 May 6.

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