| Target Validation Information | |||||
|---|---|---|---|---|---|
| Target ID | T75570 | ||||
| Target Name | Proto-oncogene tyrosine-protein kinase Yes | ||||
| Target Type | Clinical Trial |
||||
| Drug Potency against Target | TG-100435 | Drug Info | Ki = 12.9 nM | [528527] | |
| References | |||||
| Ref 528527 | Bioorg Med Chem Lett. 2007 Feb 1;17(3):602-8. Epub 2006 Nov 7.Discovery of [7-(2,6-dichlorophenyl)-5-methylbenzo [1,2,4]triazin-3-yl]-[4-(2-pyrrolidin-1-ylethoxy)phenyl]amine--a potent, orally active Src kinase inhibitor with anti-tumor activity in preclinical assays. | ||||
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