Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T58674 | Target Info | |||
| Target Name | APJ endogenous ligand (Apelin) | ||||
| Synonyms |
Apelin13; APEL
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| Target Type | Literature-reported Target | ||||
| Gene Name | APLN | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 1 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
5-[4-[[(5S)-6-[[(2S)-3-(1-Benzyl-3-methylimidazol-1-ium-4-yl)-1-[(1-methylpiperidin-4-yl)amino]-1-oxopropan-2-yl]amino]-5-[[2-(2-imino-3-methyl-1,3-thiazol-4-yl)acetyl]amino]-6-oxohexyl]amino]butylsulfamoyl]-2-[3-(diethylamino)-6-diethylazaniumylidenexanthen-9-yl]benzenesulfonate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234456; BDBM50009564
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| Activity |
Ki ~ 100000 nM
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[1] | |||
| References | Top | ||||
|---|---|---|---|---|---|
| REF 1 | Structure-activity relationship studies toward the discovery of selective apelin receptor agonists. J Med Chem. 2014 Apr 10;57(7):2908-19. | ||||
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