Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T67162 | Target Info | |||
| Target Name | Dopamine D2 receptor (D2R) | ||||
| Synonyms |
Dopamine receptor 2; D(2) dopamine receptor
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| Target Type | Successful Target | ||||
| Gene Name | DRD2 | ||||
| Biochemical Class | GPCR rhodopsin | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 74 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
Procaterol
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|
Approved | Compound Info | ||
| Synonyms |
Meptin; Procaterolo; Procaterolum; Procaterol Monohydrochloride; Procaterolo [DCIT]; Procaterolum [Latin]; Meptin (TN); OPC-2009; Procaterol (INN); Procaterol [INN:BAN]; Procaterolum [INN-Latin]; (R*,S*)-(+-)-8-Hydroxy-5-(1-hydroxy-2-((1-methylethyl)amino)butyl)-2(1H)-quinolinone; 5-[1-hydroxy-2-(propan-2-ylamino)butyl]quinoline-2,8-diol; 8-Hydroxy-5-(1-hydroxy-2-((1-methylethyl)amino)butyl)-2(1H)-quinolinone; 8-hydroxy-5-[1-hydroxy-2-(propan-2-ylamino)butyl]-1H-quinolin-2-one
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| Activity |
Ki = 86000 nM
|
[1] | |||
| Compound Name |
Armodafinil
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Approved | Compound Info | ||
| Synonyms |
Nuvigil; 112111-43-0; (R)-Modafinil; (R)-(-)-Modafinil; CEP-10953; UNII-V63XWA605I; CRL 40982; CEP 10953; V63XWA605I; CHEMBL1201192; CHEBI:77590; 2-[(R)-(Diphenylmethyl)sulfinyl]acetamide; (-)-2-((R)-(Diphenylmethyl)sulfinyl)acetamide; (-)-2-[(r)-(diphenylmethyl)sulfinyl]acetamide; Armodafinil [USAN:INN]; armodafinilo; armodafinilum; l-Modafinil; Nuvigil (TN); (-)-(R)-modafinil; Armodafinil (USAN/INN); SCHEMBL34489; ZINC6156; ACE037; Armodafinil, > YFGHCGITMMYXAQ-LJQANCHMSA-N
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| Activity |
Ki ~ 100000 nM
|
[2] | |||
| Compound Name |
L-745,870
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Phase 2 | Compound Info | ||
| Synonyms |
158985-00-3; L-745870; UNII-J3OLN3XSX7; J3OLN3XSX7; L-745,870; CHEMBL267014; L 745,870; 3-((4-(4-Chlorophenyl)piperazin-1-yl)methyl)-1H-pyrrolo[2,3-b]pyridine; 3-(4-[4-Chlorophenyl]piperazin-1-yl)-methyl-1H-pyrrolo[2,3-b]pyridine trihydrochloride; 3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-1H-pyrrolo(2,3-b)pyridine; 3-[[4-(4-chlorophenyl)piperazin-1-yl]methyl]-1H-pyrrolo[2,3-b]pyridine; CPMPP-3; Tocris-1002; Lopac-L-131; Biomol-NT_000049; AC1NSK75; L745870; Lopac0_000791; GTPL3303; BPBio1_001299; SCHEMBL1059886; CHEBI:92099
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| Activity |
Ki = 53703.18 nM
|
[3] | |||
| Compound Name |
ABT-724
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Discontinued in Phase 2 | Compound Info | ||
| Synonyms |
2-[4-(2-Pyridyl)piperazin-1-ylmethyl]-1H-benzimidazole maleate
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| Activity |
Ki = 51000 nM
|
[4] | |||
| Compound Name |
Ebalzotan
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Discontinued in Phase 1 | Compound Info | ||
| Synonyms |
NAE-086
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| Activity |
Ki ~ 50000 nM
|
[5] | |||
| Compound Name |
ZM-241385
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Terminated | Compound Info | ||
| Synonyms |
ZM241385; 139180-30-6; ZM 241385; ZM-241385; CHEMBL113142; 4-(2-(7-Amino-2-(2-furyl)(1,2,4)triazolo(2,3-a)(1,3,5)triazin-5-ylamino)ethyl)phenol; 4-(2-[7-Amino-2-(2-furyl)[1,2,4]triazolo[2,3-a][1,3,5]triazin-5-ylamino]ethyl)phenol; 4-(2-(7-Amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-ylamino)ethyl)phenol; 4-{2-[(7-Amino-2-Furan-2-Yl[1,2,4]triazolo[1,5-A][1,3,5]triazin-5-Yl)amino]ethyl}phenol; 4-[2-[[7-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl]amino]ethyl]phenol
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| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
N-(4-Propylaminobutyl)-4-biphenylcarboxamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL444128; N-(4-Propylaminobutyl)-4-biphenylcarboxamide
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| Activity |
Ki ~ 100000 nM
|
[7] | |||
| Compound Name |
ADS-103253
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Investigative | Compound Info | ||
| Synonyms |
ADS-103253; CHEMBL216228; SCHEMBL6507329; BDBM50200788
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| Activity |
IC50 ~ 100000 nM
|
[8] | |||
| Compound Name |
tyramine
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Investigative | Compound Info | ||
| Synonyms |
Tyramine; 4-(2-Aminoethyl)phenol; 51-67-2; 4-Hydroxyphenethylamine; p-Tyramine; 2-(4-Hydroxyphenyl)ethylamine; Uteramine; Tyramin; Tyrosamine; Tocosine; 4-Hydroxyphenylethylamine; Systogene; Phenol, 4-(2-aminoethyl)-; p-Hydroxyphenethylamine; Tenosin-wirkstoff; p-Hydroxyphenylethylamine; p-(2-Aminoethyl)phenol; 2-(p-Hydroxyphenyl)ethylamine; Phenethylamine, p-hydroxy-; p-beta-Aminoethylphenol; Phenol, p-(2-aminoethyl)-; Benzeneethanamine, 4-hydroxy-; Tyramine base; beta-Hydroxyphenylethylamine; NSC 249188; p-tyramine; [3H]tyramine
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| Activity |
Ki = 160000 nM
|
[9] | |||
| Compound Name |
(11R)-5-Methyl-6,11-dioxo-N-(2-thiophen-2-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234545; SCHEMBL17837157; BDBM50003075; NCGC00250207-01
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| Activity |
Ki ~ 50000 nM
|
[10] | |||
| Compound Name |
6-Chloro-3-(4-(3-(2-chloro-4-fluorophenyl)-1,2,4-oxadiazol-5-yl)piperidin-1-yl)quinoline
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL468176; BDBM50261729
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| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
(R)-3-[Isopropyl(propyl)amino]-3,4-dihydro-2H-1-benzopyran-5-carboxamide
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|
Investigative | Compound Info | ||
| Synonyms |
NAE-111; SCHEMBL8823635; CHEMBL3085216; BDBM85827; (3R)-3-[propan-2-yl(propyl)amino]-3,4-dihydro-2H-chromene-5-carboxamide
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| Activity |
Ki ~ 50000 nM
|
[5] | |||
| Compound Name |
Pyrazolo[1,5-a]pyridine,2-[[4-[4-(2-fluoroethoxy)phenyl]-1-piperazinyl]methyl]-
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL272853; BDBM50373496; ZINC29133960; Pyrazolo[1,5-a]pyridine, 2-[[4-[4-(2-fluoroethoxy)phenyl]-1-piperazinyl]methyl]-
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| Activity |
Ki = 50000 nM
|
[12] | |||
| Compound Name |
(S)-N-Isopropyl-3-[isopropyl(propyl)amino]-3,4-dihydro-2H-1-benzopyran-5-carboxamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2111582
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| Activity |
Ki ~ 50000 nM
|
[5] | |||
| Compound Name |
(2S,3S,4S,5R,6R)-2-(Fluoromethyl)-6-[4-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]triazol-1-yl]oxane-3,4,5-triol
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2443003; BDBM50442753
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| Activity |
Ki = 51000 nM
|
[13] | |||
| Compound Name |
4-[4-(4-Chlorophenyl)piperazine-1-ylmethyl]pyrazolo[1,5-a]pyridine-3-methanol
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL328925; BDBM50102716; {4-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-pyrazolo[1,5-a]pyridin-3-yl}-methanol
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| Activity |
Ki = 53000 nM
|
[14] | |||
| Compound Name |
Dipropyl-(R)-4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyridin-5-yl-amine
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL197159; BDBM50172509; ZINC13672663
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|
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| Activity |
Ki = 53000 nM
|
[15] | |||
| Compound Name |
3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-2,7-dimethylimidazo[1,2-c]pyrimidine
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL561262; BDBM50295933
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| Activity |
Ki = 53000 nM
|
[16] | |||
| Compound Name |
1,2,3,4-Tetrahydroisoquinoline-6-carbonitrile
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|
Investigative | Compound Info | ||
| Synonyms |
6-ISOQUINOLINECARBONITRILE, 1,2,3,4-TETRAHYDRO-; CHEMBL4076796; SCHEMBL1638541; DTXSID10437121; 8464AA; ANW-75169; BDBM50267215; ZINC35571313; AKOS006276440; AB16298; AM803297; SC-95468; 6-cyano-1,2,3,4-tetrahydro-isoquinoline; DB-013752; FT-0648423; 1,2,3,4-tetrahydro-isoquinolin-6-carbonitrile; 398T341; J-503766; 1,2,3,4-TETRAHYDRO-6-ISOQUINOLINECARBONITRILE; 1,2,3,4-TETRAHYDROISOQUINOLINE-6-CARBONITRILE98%
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| Activity |
Ki = 53800 nM
|
[17] | |||
| Compound Name |
(E)-Tert-butyl 6-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyleneamino)indoline-1-carboxylate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL240021; BDBM50206176
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| Activity |
Ki = 54000 nM
|
[18] | |||
| Compound Name |
Benzo[b]thiophen-3-yl(4-fluoro-4-(((5-methylpyridin-2-yl)methylamino)methyl)piperidin-1-yl)methanone
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1259241; SCHEMBL3976254; BDBM50328637
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|
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| Activity |
Ki = 54000 nM
|
[19] | |||
| Compound Name |
2-[4-(4-Fluorophenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyrimidine
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL425064; BDBM50189836
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| Activity |
Ki = 55000 nM
|
[20] | |||
| Compound Name |
3-[4-(4-Chlorophenyl)piperazinomethyl]-4-(hydroxymethyl)pyrazolo[1,5-a]pyridine
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL160396; BDBM50109951; {3-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-pyrazolo[1,5-a]pyridin-4-yl}-methanol
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| Activity |
Ki = 56000 nM
|
[21] | |||
| Compound Name |
(-)-Govadine
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1950491
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| Activity |
EC50 = 56000 nM
|
[22] | |||
| Compound Name |
3-{[4-(4-Chlorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL554692; BDBM50295938
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| Activity |
Ki = 57000 nM
|
[16] | |||
| Compound Name |
3-[9-[3-[(4-Methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecan-3-yl]benzonitrile
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL4076086; BDBM50250805
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| Activity |
Ki = 57101 nM
|
[23] | |||
| Compound Name |
2-Methyl-3-[4-(4-chlorophenyl)piperazinomethyl]-7-cyanopyrazolo[1,5-a]pyridine
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL160932; BDBM50109945; 3-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-2-methyl-pyrazolo[1,5-a]pyridine-7-carbonitrile
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| Activity |
Ki = 58000 nM
|
[21] | |||
| Compound Name |
((R)-7-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL335971; SCHEMBL2702018; BDBM50054080; ZINC13759800; (2R)-7-methoxy-N-propyl-1,2,3,4-tetrahydronaphthalen-2-amine
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| Activity |
Ki = 58882 nM
|
[24] | |||
| Compound Name |
(E)-N-Benzyl-N''-(3-hydroxy-2,3-dihydro-1H-inden-5-yl)-N-methylformamidine
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL392888; SCHEMBL8308123; BDBM50206167
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|
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| Activity |
Ki = 59000 nM
|
[18] | |||
| Compound Name |
2-{5-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-pyrrol-2-ylmethylene}-malononitrile
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL303538; BDBM50079646; 4-(4-Chloro-phenyl)-1-[5-(2,2-dicyano-vinyl)-1H-pyrrol-2-ylmethyl]-piperazin-1-ium; 5-(2,2-Dicyanovinyl)-2-[[4-(4-chlorophenyl)piperazine-1-yl]methyl]-1H-pyrrole
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| Activity |
Ki = 59000 nM
|
[25] | |||
| Compound Name |
7-(2-Methoxyphenyl)-2-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-2,7-diazaspiro[3.4]octane
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL4089290; BDBM50250811
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| Activity |
Ki = 60152 nM
|
[23] | |||
| Compound Name |
2-[4-(4-Fluorophenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyrazine
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL377542; BDBM50189838
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| Activity |
Ki = 64000 nM
|
[20] | |||
| Compound Name |
1-(1-Benzyl-4-piperidinyl)-1H-pyrrole-3-carbaldehyde
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL422959; BDBM50082172; 1-(1-Benzyl-piperidin-4-yl)-1H-pyrrole-3-carbaldehyde
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| Activity |
Ki = 65000 nM
|
[26] | |||
| Compound Name |
[(1S,2R,5S,6S,7S)-3-Benzyl-2-methyl-7-pyrrolidin-1-yl-3-azabicyclo[3.2.0]heptan-6-yl]methanol
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2062854; BDBM50389443
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| Activity |
Ki = 66000 nM
|
[27] | |||
| Compound Name |
3-[[4-[4-(2-Fluoroethoxy)phenyl]piperazin-1-yl]methyl]pyrazolo[1,5-a]pyridine
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL272873; BDBM50373493
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| Activity |
Ki = 66000 nM
|
[12] | |||
| Compound Name |
7-[4-(4-Chlorophenyl)piperazine-1-ylmethyl]pyrazolo[1,5-a]pyridine
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL88937; BDBM50102715; 7-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-pyrazolo[1,5-a]pyridine
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| Activity |
Ki = 67000 nM
|
[14] | |||
| Compound Name |
4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(2''-methoxyphenyl)piperazine
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL516334; SCHEMBL4317685; BDBM50275163
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| Activity |
Ki = 67000 nM
|
[28] | |||
| Compound Name |
(4-Bromothiophen-2-yl)(4-fluoro-4-(((5-methylpyridin-2-yl)methylamino)methyl)piperidin-1-yl)methanone
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1259071; SCHEMBL3982351; BDBM50328628
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| Activity |
Ki = 73000 nM
|
[19] | |||
| Compound Name |
N-[4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl]-5-phenyl-1,2,4-oxadiazol-3-amine;hydrochloride
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL3739820; BDBM50500112
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| Activity |
Ki = 79630 nM
|
[29] | |||
| Compound Name |
9-[3-[(4-Methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3-pyridin-2-yl-3,9-diazaspiro[5.5]undecane
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL4076527; BDBM50250806
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| Activity |
Ki = 83671 nM
|
[23] | |||
| Compound Name |
4-[4-(Pyrazolo[1,5-a]pyridin-3-ylmethyl)piperazin-1-yl]phenol
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL407818; BDBM50373489
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| Activity |
Ki = 87000 nM
|
[12] | |||
| Compound Name |
3-(2,3,4,9-Tetrahydro-1H-pyrido[3,4-b]indol-1-yl)phenol
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL392401; Oprea1_477691; SCHEMBL3568230; BDBM50206182; STL525287; AKOS022219509; MCULE-7408578401; 3-(2,3,4,9-tetrahydro-1H-beta-carbolin-1-yl)phenol
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| Activity |
Ki = 88000 nM
|
[18] | |||
| Compound Name |
4-(2-Piperazin-1-ylethyl)-1,3-dihydroindol-2-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL3394274; BDBM50059802
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| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
4-[2-(1,4-Diazepan-4-ium-1-yl)ethyl]-1,3-dihydroindol-2-one;2,2,2-trifluoroacetate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL3394275; BDBM50059801
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| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
2-[[(2R)-2-Phenethylmorpholino]methyl]-1H-benzoimidazole
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL3335537; BDBM50027074
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|
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| Activity |
Ki ~ 100000 nM
|
[30] | |||
| Compound Name |
Tert-butyl 4-[2-(2-oxo-1,3-dihydroindol-4-yl)ethyl]piperazine-1-carboxylate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL3394272; BDBM50059805
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| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
5-Propylamino-4,5,6,7-tetrahydro-pyrazolo[1,5-a]pyridine-3-carboxylic acid methyl ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL383805; BDBM50172510
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| Activity |
Ki ~ 100000 nM
|
[31] | |||
| Compound Name |
5-N-[2-[4-[(4-Chloro-6-morpholin-4-yl-1,3,5-triazin-2-yl)oxy]phenyl]ethyl]-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL3394261; BDBM50059853
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| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
Methyl 12-[4-[4-[2-[[7-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl]amino]ethyl]phenoxy]butanoylamino]dodecanoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL3394260; BDBM50059872
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| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
4-[2-[[7-Amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl]-propylamino]ethyl]-1,3-dihydroindol-2-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL3394263; BDBM50059840
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| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
(E)-N-((6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methylene)-3,4a,9,9a-tetrahydro-2H-indeno[1,2-b][1,4]dithiin-6-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL240024; BDBM50206162
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[18] | |||
| Compound Name |
4-(1H-Benzimidazol-2-ylmethyl)-2-(2-phenylethyl)morpholine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3335535; SCHEMBL8926632; BDBM50027072; MCULE-2416114663; L013202
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[32] | |||
| Compound Name |
3-(4-Allylmorpholin-2-yl)phenol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL398480; BDBM50226036
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[33] | |||
| Compound Name |
N-(Propan-2-yl)-1H-indole-2-carboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4073520; N-Isopropyl-1H-indole-2-carboxamide; 1H-Indole-2-carboxamide, N-(1-methylethyl)-; ACMC-20m9h5; SCHEMBL13753384; CTK0G4080; DTXSID60546575; BDBM50267203; AKOS008953205; MCULE-2614608477; N-propan-2-yl-1H-indole-2-carboxamide
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[17] | |||
| Compound Name |
(E)-N-((6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methylene)-2,3,4a,5,6,10b-hexahydronaphtho[1,2-b][1,4]dithiin-9-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL241282; BDBM50206184
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[18] | |||
| Compound Name |
4-[2-[4-[[7-Amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl]amino]piperidin-1-yl]ethyl]-1,3-dihydroindol-2-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3394271; BDBM50059806
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
(2S)-4-(1H-Benzimidazol-2-ylmethyl)-2-(2-phenylethyl)morpholine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3335536; BDBM50027077
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[32] | |||
| Compound Name |
[1-[2-(2-Oxo-1,3-dihydroindol-4-yl)ethyl]piperidin-4-yl] N-tert-butylcarbamate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3394269; BDBM50059808
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
4-[2-[4-[7-Amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl]piperazin-1-yl]ethyl]-1,3-dihydroindol-2-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3394276; BDBM50059799
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
Dopamine hydrochloride
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
3-Hydroxytyramine hydrochloride; Dopamine HCl; 4-(2-aminoethyl)benzene-1,2-diol hydrochloride; intropin; Dopastat; Revivan; 1,2-Benzenediol, 4-(2-aminoethyl)-, hydrochloride; 3,4-Dihydroxyphenethylamine hydrochloride; Dynatra; Dopamine.HCl; 2-(3,4-Dihydroxyphenyl)ethylamine hydrochloride; (Dopamine HCl); ASL 279; 4-(2-Aminoethyl)pyrocatechol hydrochloride; m-Hydroxytyramine hydrochloride; Dopamine (hydrochloride); UNII-7L3E358N9L; 4-(2-aminoethyl)benzene-1,2-diol;hydrochloride; 3-Hydroxytyramine, Hydrochloride; ASL-279; P 498; MFCD00012898; MLS000069419; 7L3E358N9L; NSC-169105; Cardiosteril; SMR000059081; Dopamine chloride; Dopamine Fresenius; 62-31-7 (HCl); 51-61-6 (free base); 3-hydroxytyraminium chloride; Abbodop; Inotropin; Rascordin; Tensamin; 4-(2-Aminoethyl)-1,2-benzenediol hydrochloride; Pyrocatechol, 4-(2-aminoethyl)-, hydrochloride; 3-Hydroxytyramine hydrochloride, 99%; NSC169105; EINECS 200-527-8; NSC 169105; 4-(2-aminoethyl)benzene-1,2-diol, chloride; SR-01000075366; 3,4-Dihydroxyphenethylamine, HCl; Actopamin (TN); Dopamine HCl salt; Intropin (TN); 4-(2-Aminoethyl)-1-2-benzenediol; Dopamine hydrochloride in dextrose 5%; Dopamine hydrochloride and dextrose 5%; 3-Hydroxytyramine HCl; Dopamine hydrochloride [USAN:USP:JAN]; PubChem22727; 3-Hydroxytyramine, HCl; Opera_ID_218; dopamine hydrogen chloride; DSSTox_CID_550; ACMC-1B1TV; Intropin [as hydrochloride]; Dopamini hydrochloridum,(S); CHEMBL1557; DSSTox_RID_75655; DSSTox_GSID_20550; SCHEMBL40951; KSC353A3H; MLS001074180; SPECTRUM1500263; SGCUT00110; DTXSID7020550; CTK2F3033; HY-B0451A; Dopamine hydrochloride (Inotropin); HMS1920I18; KUC104380C; Pharmakon1600-01500263; BCP06611; KS-00000JK7; to_000060; Dopamine hydrochloride (JP17/USP); Tox21_201018; Tox21_500586; CCG-40211; NSC756749; s2529; SBB003668; AKOS008056421; 1, 4-(2-aminoethyl)-, hydrochloride; KS-5304; KSC-10-159; LP00586; MCULE-8844188424; NC00545; NSC-756749; 3,4-dihydoxyphenethylamine hydrochloride; NCGC00093965-01; NCGC00093965-02; NCGC00093965-03; NCGC00093965-04; NCGC00258571-01; NCGC00261271-01; 3,4-dihydroxyphenylethylaminehydrochloride; AC-12190; AK142758; SC-16285; AB0013398; DB-023081; 3,4-dihydroxyphenyl-ethylamine hydrochloride; A0305; AM20080715; EU-0100586; FT-0603260; FT-0667775; FT-0695562; SW199608-2; W0031; D00633; H 8502; J10150; M-7455; 2-(3,4-dihydroxyphenyl)ethyl-1-13c-amine hcl; 4-(2-aminoethyl)benzene-1,2-diol,hydrochloride; 2-(3,4-dihydroxyphenyl)-ethylamine hydrochloride; Dopamine hydrochloride, puriss., >=98.5% (AT); SR-01000075366-1; SR-01000075366-8; Q27268491; F0001-1648; Z262221794; 963AD780-3E96-47B5-9044-7E59F6C84D67
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[34] | |||
| Compound Name |
2-[5-(4-Phenylpiperazinomethyl)-1H-pyrrole-2-ylmethylene]malononitrile
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL293956; BDBM50079642; 2-[5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-ylmethylene]-malononitrile
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[25] | |||
| Compound Name |
Tert-butyl 4-[2-(2-oxo-1,3-dihydroindol-4-yl)ethyl]-1,4-diazepane-1-carboxylate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3394273; BDBM50059804
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
3-(4-Fluorophenyl)-9-methyl-1-oxa-9-azaspiro[5.5]undec-2-en-4-one;hydrochloride
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL544055
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[35] | |||
| Compound Name |
4-[2-(4-Aminopiperidin-1-yl)ethyl]-1,3-dihydroindol-2-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3394270; BDBM50059807
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
2-[3-[4-(4-Methoxyphenyl)piperazin-1-yl]propyl]-4,5-dihydro-3H-2-benzazepin-1-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL476642
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[36] | |||
| Compound Name |
4-[2-[4-[7-Amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl]-1,4-diazepan-1-ium-1-yl]ethyl]-1,3-dihydroindol-2-one;2,2,2-trifluoroacetate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3394277; BDBM50059798
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
9-Methyl-3-phenyl-1-oxa-9-azaspiro[5.5]undec-2-en-4-one;hydrochloride
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL539518
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[35] | |||
| Compound Name |
N-(Cyclopropylmethyl)-1H-indole-2-carboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4092619; SCHEMBL6885051; BDBM50267204; AKOS009156341; MCULE-8383290655
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[17] | |||
| Compound Name |
3-(4-Methoxyphenyl)-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4100699; BDBM50250809
Click to Show/Hide
|
||||
| Activity |
Ki = 104847 nM
|
[23] | |||
| Compound Name |
1-(4-Fluorophenyl)-6-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-1,6-diazaspiro[3.3]heptane
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4098399; BDBM50250800
Click to Show/Hide
|
||||
| Activity |
Ki ~ 109574 nM
|
[23] | |||
| Compound Name |
3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(3,4-dihydroisoquinoline)
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL485720; BDBM50275251
Click to Show/Hide
|
||||
| Activity |
Ki = 114000 nM
|
[28] | |||
| Compound Name |
1-(2-Methoxyphenyl)-6-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-1,6-diazaspiro[3.3]heptane
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL4079642; BDBM50250801
Click to Show/Hide
|
||||
| Activity |
Ki = 114945 nM
|
[23] | |||
| Compound Name |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(N-methyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL487960; BDBM50275220
Click to Show/Hide
|
||||
| Activity |
Ki = 178000 nM
|
[28] | |||
| Compound Name |
6-Methoxy-1-(1-methyl-4-nitro-1H-pyrrol-2-yl)-4,9-dihydro-3H-pyrido[3,4-b]indole
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL241099; BDBM50206185
Click to Show/Hide
|
||||
| Activity |
Ki = 200000 nM
|
[18] | |||
| Click to Show/Hide the Information of All Poor Binders | |||||
| Non Binders of This Target (in total, 35 non binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
SKF 38393
Click to Show/Hide
|
Terminated | Compound Info | ||
| Synonyms |
SKF-38393; F-38393; 67287-49-4; F 38393; SKF38393; BRN 1543419; CHEMBL286080; 1-phenyl-2,3,4,5-tetrahydro-1h-3-benzazepine-7,8-diol; 2,3,4,5-Tetrahydro-1-phenyl-1H-3-benzazepine-7,8-diol; 1H-3-Benzazepine-7,8-diol, 2,3,4,5-tetrahydro-1-phenyl-; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; SKF-38,393; SK-38393; C16H17NO2; 5-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine-7,8-diol; 1-Phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol
Click to Show/Hide
|
||||
| Activity |
Ki = 720000 nM
|
[37] | |||
| Compound Name |
3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3''-chlorophenyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL458792; SCHEMBL4179477; BDBM50275099; 1-(3-chlorophenyl)-4-[3-[2-[2-(3-methoxyphenyl)ethyl]phenoxy]propyl]piperazine
Click to Show/Hide
|
||||
| Activity |
Ki = 298000 nM
|
[28] | |||
| Compound Name |
(E)-6-((6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyleneamino)-2,3-dihydro-1H-inden-1-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL391192; SCHEMBL8313860; BDBM50206192
Click to Show/Hide
|
||||
| Activity |
Ki > 300000 nM
|
[18] | |||
| Compound Name |
(E)-6-((3,4-Dihydroisoquinolin-2(1H)-yl)methyleneamino)-2,3-dihydro-1H-inden-1-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL442093; SCHEMBL5826269; BDBM50206171; 6-(3,4-dihydro-1H-isoquinolin-2-ylmethylideneamino)-2,3-dihydro-1H-inden-1-ol
Click to Show/Hide
|
||||
| Activity |
Ki > 300000 nM
|
[18] | |||
| Compound Name |
1-Phenyl-2,3,4,9-tetrahydro-1H-beta-carboline
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole; 1-Phenyl-tetrahydrocarboline; CHEMBL241083; CMLDBU00002587; CMLD2_000054; Oprea1_201098; Oprea1_407648; SCHEMBL274149; DTXSID40276762; ALBB-008773; BDBM50206179; STK505562; AKOS000558803; AKOS016050245; CCG-102255; MCULE-6546088378; NCGC00017826-02; AS-66675; FT-0673838; R4816; 1,2,3,4-Tetrahydro-1-phenyl-beta-carboline; 1-Phenyl-1,2,3,4-tetrahydro-beta-carboline; 1-Phenyl-2,3,4,9-tetrahydro-1H-b-carboline; SR-05000001242; 1-Phenyl-2,3,4,9-tetrahydro-1H-beta-carboline #; SR-05000001242-1; 1-PHENYL-1H,2H,3H,4H,9H-PYRIDO[3,4-B]INDOLE; 1H-Pyrido[3,4-b]indole, 2,3,4,9-tetrahydro-1-phenyl-
Click to Show/Hide
|
||||
| Activity |
Ki > 300000 nM
|
[18] | |||
| Compound Name |
2{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(2''-methoxyphenyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL514286; SCHEMBL4186798; BDBM50275137
Click to Show/Hide
|
||||
| Activity |
Ki = 427000 nM
|
[28] | |||
| Compound Name |
1-[3-[2-[2-(3-Methoxyphenyl)ethyl]phenoxy]propyl]-4-methylpiperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL518931; SCHEMBL4180271; BDBM50275221; 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3''-methyl)piperazine
Click to Show/Hide
|
||||
| Activity |
Ki = 565000 nM
|
[28] | |||
| Compound Name |
1-(1-Propylpiperidin-4-yl)benzimidazole
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2207492; BDBM50401409
Click to Show/Hide
|
||||
| Activity |
IC50 > 580000 nM
|
[38] | |||
| Compound Name |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(2''-pyrimidil)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL456674; BDBM50275195
Click to Show/Hide
|
||||
| Activity |
Ki = 629000 nM
|
[28] | |||
| Compound Name |
3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(4''-fluorophenyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL457921; SCHEMBL4176822; BDBM50275166
Click to Show/Hide
|
||||
| Activity |
Ki = 655000 nM
|
[28] | |||
| Compound Name |
(4As,5R,10bR)-5-phenyl-1,2,3,4,4a,5,6,10b-octahydrobenzo[h]isoquinoline-7,8-diol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1224527; BDBM50325822; trans-(5R)-5-phenyl-1,2,3,4,4a,5,6,10b-octahydrobenzo[h]isoquinoline-7,8-diol
Click to Show/Hide
|
||||
| Activity |
Ki = 750000 nM
|
[39] | |||
| Compound Name |
6,9-Dichloro-3-methyl-5-phenyl-1,2,4,5-tetrahydro-3-benzazepine-7,8-diol;hydrochloride
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL544118
Click to Show/Hide
|
||||
| Activity |
Ki = 810000 nM
|
[40] | |||
| Compound Name |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(4''-fluorophenyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL514098; BDBM50275194
Click to Show/Hide
|
||||
| Activity |
Ki = 847000 nM
|
[28] | |||
| Compound Name |
4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(2''-pyrimidyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL487760; BDBM50275218
Click to Show/Hide
|
||||
| Activity |
Ki = 854000 nM
|
[28] | |||
| Compound Name |
2{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(4''-fluorophenyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL458992; SCHEMBL4172184; BDBM50275165
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(3''-trifluoromethyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL457891; SCHEMBL4183345; BDBM50275102
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-(3,4-dihydroisoquinoline)
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL521025; BDBM50275250
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(3''-trifluoromethylphenyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL459158; SCHEMBL4179806; BDBM50275136
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
6,7-Dimethoxy-2-[2-[2-[2-(3-methoxyphenyl)ethyl]phenoxy]ethyl]-3,4-dihydro-1H-isoquinoline
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL486336; BDBM50275283; 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-(6,7-dimethoxy-3,4-dihydroisoquinoline)
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
6,7-Dimethoxy-2-[4-[2-[2-(3-methoxyphenyl)ethyl]phenoxy]butyl]-3,4-dihydro-1H-isoquinoline
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL485727; BDBM50275285; 4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-(6,7-dimethoxy-3,4-dihydroisoquinoline)
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(N-methyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL486534; BDBM50275248
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(3''-trifluoromethylphenyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL457889; SCHEMBL4168989; BDBM50275100
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
6,7-Dimethoxy-2-[3-[2-[2-(3-methoxyphenyl)ethyl]phenoxy]propyl]-3,4-dihydro-1H-isoquinoline
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL486337; BDBM50275284; 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(6,7-dimethoxy-3,4-dihydroisoquinoline)
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(3''-chlorophenyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL515853; SCHEMBL4181085; BDBM50275061
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(3''-chlorophenyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL457890; BDBM50275101
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(2''-pyrimidyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL487761; BDBM50275219
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
6,7-Dimethoxy-2-[5-[2-[2-(3-methoxyphenyl)ethyl]phenoxy]pentyl]-3,4-dihydro-1H-isoquinoline
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL519547; BDBM50275324; 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(6,7-dimethoxy-3,4-dihydroisoquinoline)
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(N-methyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL485719; BDBM50275249
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(2''-methoxyphenyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL458991; BDBM50275164
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-(3,4-dihydroisoquinoline)
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL485918; BDBM50275252
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-(3,4-dihydroisoquinoline)
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL519228; BDBM50275282
Click to Show/Hide
|
||||
| Activity |
Ki > 1000000 nM
|
[28] | |||
| Compound Name |
4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(4''-fluorophenyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL456673; SCHEMBL4182261; BDBM50275193
Click to Show/Hide
|
||||
| Activity |
Ki = 1324000 nM
|
[28] | |||
| Compound Name |
3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3''-trifluoromethylphenyl)piperazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL457899; SCHEMBL4186793; BDBM50275135
Click to Show/Hide
|
||||
| Activity |
Ki = 1412000 nM
|
[28] | |||
| Compound Name |
trans-4-Tert-Butoxy-N-(4-{2-[4-(2,3-dihydro-benzofuran-4-yl)-piperidin-1-yl]-ethyl}-cyclohexyl)-benzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL9933882; SCHEMBL9934198; CHEMBL3695441; BDBM138484; US8877778, 88
Click to Show/Hide
|
||||
| Activity |
Ki > 10000000 nM
|
[41] | |||
| Compound Name |
4-Tert-butyl-N-[4-[2-[4-(2,3-dihydro-1-benzofuran-4-yl)piperidin-1-yl]ethyl]cyclohexyl]benzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL9933529; SCHEMBL9933531; CHEMBL3695424; BDBM138467; US8877778, 71
Click to Show/Hide
|
||||
| Activity |
Ki > 10000000 nM
|
[41] | |||
| Click to Show/Hide the Information of All Non Binders | |||||
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