Target Validation Information
TTD ID T40016
Target Name Glucocorticoid receptor (NR3C1)
Type of Target
Drug Potency against Target GW685698X Drug Info IC50 = 69000 nM [2]
BAY 86-5044 Drug Info IC50 = 16 nM [1]
REF 1 Synthesis and biological activity of a novel, highly potent progesterone receptor antagonist. J Med Chem. 2000 Dec 28;43(26):5010-6.
REF 2 Structure-activity relationships of selective GABA uptake inhibitors. Curr Top Med Chem. 2006;6(17):1861-82.

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