Target Information
Target General Infomation | |||||
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Target ID |
T99665
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Former ID |
TTDI03210
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Target Name |
GABAA receptor rho1 subunit
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Gene Name |
GABRR1
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Synonyms |
GABRR1
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Target Type |
Research
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UniProt ID | |||||
Sequence |
MLAVPNMRFGIFLLWWGWVLATESRMHWPGREVHEMSKKGRPQRQRREVHEDAHKQVSPI
LRRSPDITKSPLTKSEQLLRIDDHDFSMRPGFGGPAIPVGVDVQVESLDSISEVDMDFTM TLYLRHYWKDERLSFPSTNNLSMTFDGRLVKKIWVPDMFFVHSKRSFIHDTTTDNVMLRV QPDGKVLYSLRVTVTAMCNMDFSRFPLDTQTCSLEIESYAYTEDDLMLYWKKGNDSLKTD ERISLSQFLIQEFHTTTKLAFYSSTGWYNRLYINFTLRRHIFFFLLQTYFPATLMVMLSW VSFWIDRRAVPARVPLGITTVLTMSTIITGVNASMPRVSYIKAVDIYLWVSFVFVFLSVL EYAAVNYLTTVQERKEQKLREKLPCTSGLPPPRTAMLDGNYSDGEVNDLDNYMPENGEKP DRMMVQLTLASERSSPQRKSQRSSYVSMRIDTHAIDKYSRIIFPAAYILFNLIYWSIFS |
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Agonist | (+/-)-cis-2-CAMP | Drug Info | [1] | ||
5-Me-IAA | Drug Info | [1] | |||
CACA | Drug Info | [2] | |||
Antagonist | aza-THIP | Drug Info | [1] | ||
cis-3-ACPBPA | Drug Info | [1] | |||
isonipecotic acid | Drug Info | [1] | |||
piperidine-4-sulphonic acid | Drug Info | [1] | |||
TPMPA | Drug Info | [1] | |||
trans-3-ACPBPA | Drug Info | [1] | |||
Blocker (channel blocker) | TBPS | Drug Info | [1] | ||
References | |||||
REF 1 | (http://www.guidetopharmacology.org/) Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Target id: 420). | ||||
REF 2 | Characterization of bicuculline/baclofen-insensitive (rho-like) gamma-aminobutyric acid receptors expressed in Xenopus oocytes. II. Pharmacology of gamma-aminobutyric acidA and gamma-aminobutyric acidB receptor agonists and antagonists. Mol Pharmacol. 1993 Apr;43(4):609-25. |
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