Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T91180 | Target Info | |||
| Target Name | Solute carrier family 15 member 1 (SLC15A1) | ||||
| Synonyms |
PEPT1; Oligopeptide transporter, small intestine isoform; Intestinal H(+)/peptide cotransporter
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| Target Type | Literature-reported Target | ||||
| Gene Name | SLC15A1 | ||||
| Biochemical Class | Proton-dependent oligopeptide transporter | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 81 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
H-Phe-Phe-NH2
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL108438; 15893-46-6; Phe-phe-amide; Phenylalanylphenylalanylamide; L-Phe-L-phe-amide; H-Phe-Phe-NH2; L-Phenylalanine-L-phenylalanylamide; L-Phe-L-Phe-NH2; AC1L38WX; XXPXQEQOAZMUDD-HOTGVXAUSA-N; L-Phenylalaninamide, L-phenylalanyl-; BDBM50188489; (S)-2-Amino-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-phenyl-propionamide
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| Activity |
IC50 = 80000 nM
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[1] | |||
| Compound Name |
Trp-val
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Investigative | Compound Info | ||
| Synonyms |
H-Trp-Val-OH; L-Valine, L-tryptophyl-; tryptophanyl-valine; CHEMBL39159; L-Tryptophyl-L-Valine; L-Trp-L-Val; L-Trp-L-Val-OH; L-Tryptophanyl-L-valine; SCHEMBL9822472; CTK0J9867; ZINC2384982; BDBM50188526; MFCD00037958; Q27144987; (S)-2-[(S)-2-Amino-3-(1H-indol-3-yl)-propionylamino]-3-methyl-butyric acid
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| Activity |
EC50 = 50000 nM
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[1] | |||
| Compound Name |
Val-phe
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Investigative | Compound Info | ||
| Synonyms |
H-VAL-PHE-OH; L-valyl-L-phenylalanine; CHEMBL8486; N-Valylphenylalanine; L-Phenylalanine, L-valyl-; L-Val-L-Phe-OH; SCHEMBL7335375; ZINC1605725; BDBM50142287; MFCD00020423; AKOS010421061; CS-7910; DS-012099; HY-107378; ST50410826; Q27145075; (S)-2-((S)-2-Amino-3-methyl-butyrylamino)-3-phenyl-propionic acid; (2S)-2-((2S)-2-amino-3-methylbutanoylamino)-3-phenylpropanoic acid
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| Activity |
Ki = 50000 nM
|
[2] | |||
| Compound Name |
4-Methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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Investigative | Compound Info | ||
| Synonyms |
GSK137647A; GSK 137647; GSK-137647A; N-mesityl-4-methoxybenzenesulfonamide; CHEMBL3311308; MFCD02007969; 4-methoxy-N-(2,4,6-trimethylphenyl)-benzenesulfonamide; CBMicro_012617; Oprea1_349531; Oprea1_545891; SCHEMBL19357604; KS-00000TIW; AOB2991; ZINC184126; BCP17136; EX-A1097; GSK 137647A; SMSF0014079; BDBM50044849; STK899558; AKOS003261220; CB15818; CS-5549; GSK-137647; MCULE-5583867808; N-mesityl-4-methoxy-1-benzenesulfonamide; NCGC00387253-02; NCGC00387253-05; AK240703; AS-16737; HY-19995; BIM-0012523.P001; FFA4 (GPR120) agonist GSK137647A; B7793; EU-0076636; FT-0700296; S0001; ST50719559; GSK137647A, >=98% (HPLC); A14542; AJ-292/14925630; SR-01000478738; J-690285; SR-01000478738-1; [(4-methoxyphenyl)sulfonyl](2,4,6-trimethylphenyl)amine; 4-methoxy-N-(2,4,6-trimethylphenyl)benzene-1-sulfonamide; 4-Methoxy-N-(2,4,6-triMethylphenyl)benzenesulfonaMide, 97%
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| Activity |
EC50 ~ 50118.72 nM
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[3] | |||
| Compound Name |
Val-pro
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Investigative | Compound Info | ||
| Synonyms |
L-valyl-L-proline; L-Proline, L-valyl-; valyl-proline; CHEMBL439762; N-Valyl-L-proline; L-Valine-L-proline; L-Val-L-Pro; L-Val-L-Pro-OH; L-Proline, L-L-valyl-; SCHEMBL1647354; CTK1A3700; BCP30415; ZINC4899618; BDBM50348866; AKOS010419473; Pro-Val; L-Valyl-L-proline; Val-pro; Valylproline; Q27143865
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| Activity |
Ki = 60000 nM
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[4] | |||
| Compound Name |
Ala-Tyr
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Investigative | Compound Info | ||
| Synonyms |
L-Alanyl-L-tyrosine; H-Ala-Tyr-OH; Alanyltyrosine; (S)-2-((S)-2-Aminopropanamido)-3-(4-hydroxyphenyl)propanoic acid; L-Tyrosine, L-alanyl-; CHEMBL94016; MFCD00038164; (2S)-2-[[(2S)-2-aminopropanoyl]amino]-3-(4-hydroxyphenyl)propanoic acid; L-Tyrosine, N-L-alanyl-; N-L-Alanyl-L-tyrosine; Ala-Tyr-OH; EINECS 221-305-7; L-Alanyl-L-tyrisine; L-Ala-L-Tyr; L-Ala-L-Tyr-OH; SCHEMBL2493049; CTK1C3463; DTXSID00184677; KS-000012KO; ZINC2390894; 7056AH; ANW-26929; BDBM50188523; AKOS010368061; AKOS015840021; AC-31995; AS-10477; A1263; K-7319; 061A889; J-018040; Q27140488; (S)-2-((S)-2-Amino-propionylamino)-3-(4-hydroxy-phenyl)-propionic acid
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| Activity |
EC50 = 60000 nM
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[1] | |||
| Compound Name |
(2S)-1-(L-Ala-)Piperidine-2-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2371146; AKOS015606809
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| Activity |
Ki = 60000 nM
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[2] | |||
| Compound Name |
Tyrosyltyrosine
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Investigative | Compound Info | ||
| Synonyms |
Tyr-tyr; L-Tyrosyl-L-tyrosine; H-TYR-TYR-OH; Peptide tyrosine-tyrosine; CHEMBL95286; Tyrosyl-Tyrosine; L-Tyrosine, L-tyrosyl-, monomer; di-L-tyrosine; L-Tyr-L-Tyr; L-Tyr-L-Tyr-OH; H-L-Tyr-L-Tyr-OH; N-L-tyrosyl-L-tyrosine; L-Tyrosine, L-tyrosyl-; L-Tyrosine, N-L-tyrosyl-; SCHEMBL1574161; CTK0I0569; L-Tyrosine, L-tyrosyl-, mononer; ZINC2004481; BDBM50081840; MFCD00063044; Q27130548; Melanin synthesized from Tyr-Tyr substrate catalyzed by tyrosinase for 40 hrs
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| Activity |
EC50 = 60000 nM
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[1] | |||
| Compound Name |
L-Alanyl-L-alanine
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Investigative | Compound Info | ||
| Synonyms |
Ala-ala; H-Ala-Ala-OH; N-L-Alanyl-L-alanine; Dialanine; (S)-2-((S)-2-Aminopropanamido)propanoic acid; Alanyl-alanine; UNII-MY4X7L3WAM; (2S)-2-[[(2S)-2-aminopropanoyl]amino]propanoic acid; Alanylalanine; Ala-Ala-OH; MY4X7L3WAM; CHEMBL17697; MFCD00008075; L-Ala-L-Ala; Alanine, N-L-alanyl-, L-; Di-L-Alanine; .alpha.-Alanylalanine; (2S)-2-{[(2S)-2-aminopropanoyl]amino}propanoic acid; Alanine dipeptide; EINECS 217-751-7; Ala-Ala-OH HCl; l-Alanine N-l-alanyl; L-Alanine, L-alanyl-; bmse000403; (2S)-2-[(2S)-2-aminopropanamido]propanoic acid; SCHEMBL159553; D-Alanine, D-alanyl-, rel-; CTK0H9986; D-Alanyl-D-alanine, (+/-)-; DTXSID00173127; KS-00000Y9Q; ZINC1575493; BDBM50016695; N-(2-Aminopropanoyl)alanine. (L)-; AKOS010420276; AKOS015840020; AS-56749; K-5742; 948A318; A813755; (S)-2-((S)-2-Amino-propionylamino)-propionic acid; Q27140163; (2S)-2-[[(2S)-2-azanylpropanoyl]amino]propanoic acid; DF49DD8A-D390-4F75-8C8A-3A07EF07DD48; (2S)-2-[[(2S)-2-amino-1-oxopropyl]amino]propanoic acid; UNII-37AOH3N58S component DEFJQIDDEAULHB-IMJSIDKUSA-N; UNII-3EE68A29TN component DEFJQIDDEAULHB-IMJSIDKUSA-N; L-Alanyl-L-alanine, United States Pharmacopeia (USP) Reference Standard
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| Activity |
IC50 = 63000 nM
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[5] | |||
| Compound Name |
2-(3-Amino-2-oxo-4-phenyl-butyl)-succinic acid 4-benzyl ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL189777; BDBM50152062
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| Activity |
Ki = 68000 nM
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[6] | |||
| Compound Name |
Glycyl-L-leucine
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Investigative | Compound Info | ||
| Synonyms |
Gly-Leu; N-Glycyl-L-leucine; Glycylleucine; (S)-2-(2-Aminoacetamido)-4-methylpentanoic acid; Glycyl-leucine; L-Leucine, glycyl-; H-Gly-Leu-OH; UNII-8L97V505GU; CHEMBL56119; 8L97V505GU; MFCD00008127; Gly-L-Leu; Leucine, glycyl-; GLY-DL-LEU; Leucine, N-glycyl-, L-; Glycinyl-l-leucine; EINECS 212-785-9; Gly-Leu-OH; NSC 83257; Gly-L-Leu-OH; N-(Aminoacetyl)leucine #; C02155; SCHEMBL65869; (2S)-2-[(2-aminoacetyl)amino]-4-methylpentanoic acid; L-Leucine, N-glycyl- (9CI); CTK2F5157; DTXSID601017040; KS-00000M0Q; Leucine, N-glycyl-, L- (8CI); ZINC1529368; ANW-38407; BDBM50188492; KM2452; s6054; AKOS016843131; CS-W016793; HY-W016077; BP-24275; DS-16202; DB-038199; G0181; 69G192; 2-(2-Amino-acetylamino)-4-methyl-pentanoic acid; (S)-2-(2-Amino-acetylamino)-4-methyl-pentanoic acid; Q27140595
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| Activity |
IC50 = 70000 nM
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[1] | |||
| Compound Name |
Alanylphenylalanine
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Investigative | Compound Info | ||
| Synonyms |
Ala-phe; L-Alanyl-L-phenylalanine; H-Ala-Phe-OH; (S)-2-((S)-2-Aminopropanamido)-3-phenylpropanoic acid; Ala-Phe-OH; L-Ala-L-Phe; Phenylalanine, alanyl-; CHEMBL57338; MFCD00066031; (2S)-2-[[(2S)-2-aminopropanoyl]amino]-3-phenylpropanoic acid; NSC 89630; 2-(2-Amino-propionylamino)-3-phenyl-propionic acid; L-Phenylalanine,L-alanyl-; SCHEMBL893240; CTK0I2079; ZINC1575524; 3227AB; BDBM50188503; AKOS010420856; CS-W012877; HY-W012161; L-Phenylalanine, N-L-alanyl- (9CI); VC31009; AS-57743; K-7320; 061A903; Q27144123; 2-(2-Amino-propionylamino)-3-phenyl-propionic acid anion; (S)-2-((S)-2-Amino-propionylamino)-3-phenyl-propionic acid; (2S)-2-[(2S)-2-AMINOPROPANAMIDO]-3-PHENYLPROPANOIC ACID
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| Activity |
IC50 = 70000 nM
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[1] | |||
| Compound Name |
Phe-ala
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Investigative | Compound Info | ||
| Synonyms |
Phenylalanylalanine; H-PHE-ALA-OH; L-Phenylalanyl-L-alanine; (S)-2-((S)-2-Amino-3-phenylpropanamido)propanoic acid; CHEMBL429950; MFCD00037229; Phe-Ala-OH; L-Phe-L-Ala; N-phenylalanyl-alanine; L-Alanine, N-L-phenylalanyl-; SCHEMBL1711543; DTXSID20192411; (2S)-2-[[(2S)-2-amino-3-phenylpropanoyl]amino]propanoic acid; ZINC1605731; 7217AH; BDBM50139892; AKOS010420277; CS-W010318; HY-W009602; Q27142042; (S)-2-((S)-2-Amino-3-phenyl-propionylamino)-propionic acid; (S,S)2-(2-phenyl-1-trimethylammonioethylcarboxamido)propanoate
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| Activity |
IC50 = 70000 nM
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[1] | |||
| Compound Name |
H-Ala-Abu-OH
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2371145; ZINC2556516; MFCD00237699; AKOS006275478; (2S)-2-[[(2S)-2-aminopropanoyl]amino]butanoic acid
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| Activity |
Ki = 70000 nM
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[4] | |||
| Compound Name |
Val-val
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Investigative | Compound Info | ||
| Synonyms |
L-Valyl-L-valine; H-VAL-VAL-OH; CHEMBL54552; (2S)-2-[[(2S)-2-AMINO-3-METHYL-BUTANOYL]AMINO]-3-METHYL-BUTANOIC ACID,; L-Valine, L-valyl-; L-Valine, N-L-valyl-; Val-Val-OH; L-Val-L-Val; H-L-Val-L-Val-OH; SCHEMBL4582286; CTK1C4952; DTXSID40959967; ZINC1848346; BDBM50188521; MFCD00026463; AKOS010421666; MCULE-8571520026; SC-13750; N-(2-Amino-1-hydroxy-3-methylbutylidene)valine; Q27143934; (2S)-2-[[(2S)-2-AMINO-3-METHYL-BUTANOYL]AMINO]-3-M; (S)-2-((S)-2-Amino-3-methyl-butyrylamino)-3-methyl-butyric acid; (2S)-2-[[(2S)-2-amino-3-methyl-butanoyl]amino]-3-methyl-butanoic acid
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| Activity |
EC50 = 70000 nM
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[1] | |||
| Compound Name |
Ala-asp
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Investigative | Compound Info | ||
| Synonyms |
H-Ala-Asp-OH; l-alanyl-l-aspartic acid; Alanylaspartic acid; L-Aspartic acid, N-L-alanyl-; CHEMBL380047; Alanyl-Aspartic acid; L-Ala-L-Asp; N-Alanylaspartic acid; 2-[(2-ammoniopropanoyl)amino]succinate; SCHEMBL8648570; (2S)-2-[[(2S)-2-aminopropanoyl]amino]butanedioic acid; CTK8D8706; ZINC1731782; BDBM50188504; MFCD00038165; (S)-2-((S)-2-aminopropanamido)succinic acid; 727H655; Q27144119
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| Activity |
Ki = 78000 nM
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[7] | |||
| Compound Name |
Trp-tyr
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Investigative | Compound Info | ||
| Synonyms |
H-Trp-Tyr-OH; Tryptophyl-tyrosine; Tryptophyltyrosine; l-tryptophyl-l-tyrosine; CHEMBL39179; L-Tyrosine, L-tryptophyl-; Tryptophanyl-tyrosine; L-Trp-L-Tyr; L-Trp-L-Tyr-OH; L-Tryptophanyl-L-tyrosine; N-L-Tryptophyl-L-tyrosine; L-Tyrosine, N-L-tryptophyl-; SCHEMBL11835619; DTXSID90941418; ZINC2384987; BDBM50188524; MFCD00037962; J-012702; Q27144988; N-[2-Amino-1-hydroxy-3-(1H-indol-3-yl)propylidene]tyrosine
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| Activity |
IC50 = 80000 nM
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[1] | |||
| Compound Name |
Leu-Leu
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Investigative | Compound Info | ||
| Synonyms |
H-LEU-LEU-OH; N-L-Leucyl-L-leucine; l-Leucyl-l-leucine; (S)-2-((S)-2-Amino-4-methylpentanamido)-4-methylpentanoic acid; Leucylleucine; CHEMBL54933; (2S)-2-[[(2S)-2-amino-4-methylpentanoyl]amino]-4-methylpentanoic acid; LL dipeptide; Leucine, leucyl-; EINECS 221-976-6; L-Leu-L-Leu; L-Leu-L-Leu-OH; H-L-Leu-L-Leu-OH; SCHEMBL235250; CTK1A2273; KS-00000GDW; DTXSID00186696; ZINC1532219; BDBM50188496; MFCD00065185; AKOS010420853; DS-14566; K-7628; Q27140613; 2-(2-Amino-4-methyl-pentanoylamino)-4-methyl-pentanoic acid; (S)-2-((S)-2-Amino-4-methyl-pentanoylamino)-4-methyl-pentanoic acid
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| Activity |
EC50 = 80000 nM
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[1] | |||
| Compound Name |
L-Alanyl-L-tryptophan
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Investigative | Compound Info | ||
| Synonyms |
Ala-Trp; L-Tryptophan, L-alanyl-; (S)-2-((S)-2-Aminopropanamido)-3-(1H-indol-3-yl)propanoic acid; CHEMBL91792; N-L-Alanyl-L-tryptophan; (2S)-2-[[(2S)-2-aminopropanoyl]amino]-3-(1H-indol-3-yl)propanoic acid; Alanyl-Tryptophan; Ala-Trp-OH; L-Ala-L-Trp; L-Ala-L-Trp-OH; L-Tryptophan, N-L-alanyl-; SCHEMBL2488765; CTK0H6326; N-(2-Aminopropanoyl)tryptophan #; KS-000014TB; ZINC1638001; 7295AH; Ala-Trp, >=99.0% (TLC); ANW-22024; BDBM50188485; MFCD00037948; AKOS010367580; AKOS015853838; A1262; 305A752; J-009993; Q27144124; (S)-2-((S)-2-Amino-propionylamino)-3-(1H-indol-3-yl)-propionic acid
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| Activity |
EC50 = 80000 nM
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[1] | |||
| Compound Name |
(S)-2-[(S)-2-Amino-3-(4-benzyloxy-phenyl)-propionylamino]-propionic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL190728; BDBM50169157; ZINC13531470
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| Activity |
Ki = 90000 nM
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[2] | |||
| Compound Name |
2-Amino-N-((S)-2-amino-hexanoyl)-propionamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL190327; BDBM50169212
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| Activity |
Ki = 90000 nM
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[2] | |||
| Compound Name |
3-Amino-N-((S)-1-carboxy-ethyl)-succinamic acid (S)-benzyl ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL189273; BDBM50169221
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| Activity |
Ki = 90000 nM
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[2] | |||
| Compound Name |
L-Alanyl-L-norleucine
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Investigative | Compound Info | ||
| Synonyms |
H-ALA-NLE-OH; CHEMBL1814488; L-Norleucine, L-alanyl-; L-Norleucine,L-alanyl-; 2-[(2-ammoniopropanoyl)amino]hexanoate; SCHEMBL15757005; CTK6D4144; ZINC1575566; BDBM50350462; AKOS024337852; ST50553914; (S)-2-((S)-2-aminopropanamido)hexanoic acid; (2S)-2-((2S)-2-aminopropanoylamino)hexanoic acid; (S)-2-[[(S)-2-Aminopropanoyl]amino]hexanoic acid
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| Activity |
Ki = 90000 nM
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[4] | |||
| Compound Name |
Tyr-Ala
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Investigative | Compound Info | ||
| Synonyms |
H-TYR-ALA-OH; L-Alanine, L-tyrosyl-; Tyrosyl-Alanine; L-tyrosyl-L-alanine; CHEMBL316103; (S)-2-((S)-2-Amino-3-(4-hydroxyphenyl)propanamido)propanoic acid; (2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoic acid; L-Alanine, L-tyrosyl-, monomer; Tyr-Ala-OH; L-Tyr-L-Ala; SCHEMBL238988; CTK2H7022; ZINC2566273; BDBM50169129; MFCD00020398; AKOS010420474; Melanin synthesized from Tyr-Ala substrate catalyzed by tyrosinase for 40 hrs; Q27144989; (S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionic acid
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| Activity |
Ki = 90000 nM
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[2] | |||
| Compound Name |
Tyr-Phe
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Investigative | Compound Info | ||
| Synonyms |
H-Tyr-Phe-OH; Tyrosyl-Phenylalanine; tyrosylphenylalanine; L-tyrosyl-L-phenylalanine; CHEMBL447844; (S)-2-((S)-2-Amino-3-(4-hydroxyphenyl)propanamido)-3-phenylpropanoic acid; L-Tyr-L-Phe; L-Tyr-L-Phe-OH; SCHEMBL8695556; ZINC2384820; BDBM50169178; MFCD00037255; Q27145062; (S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-phenyl-propionic acid
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| Activity |
Ki = 90000 nM
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[4] | |||
| Compound Name |
(S)-2-((S)-2-Amino-3-methylbutanamido)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
H-VAL-ALA-OH; Val-Ala; L-valyl-L-alanine; Valyl-Alanine; L-Val-L-Ala; (2S)-2-[[(2S)-2-amino-3-methylbutanoyl]amino]propanoic acid; Alanine, N-L-valyl-; Val-Ala-OH; L-Alanine,l-valyl-; L-Val-L-Ala-OH; L-Alanine, L-valyl-; H-Val-Ala-OH, AldrichCPR; CHEMBL55523; SCHEMBL1711406; CTK1A1804; KS-00000GEK; DTXSID60426328; ZINC1578617; ANW-73087; MFCD00020397; AKOS010420475; CS-W007035; DS-4133; HY-W007035; K-6982; J-016790; Q27145065
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| Activity |
Ki = 90000 nM
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[4] | |||
| Compound Name |
(S)-2-((S)-2-Amino-3-benzyloxy-propionylamino)-propionic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL191493; BDBM50169225
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| Activity |
Ki = 90000 nM
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[2] | |||
| Compound Name |
[(2R,3S,4R)-5-(2-Bromo-5,6-dichlorobenzimidazol-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2S)-2-amino-3-(4-ethoxyphenyl)propanoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL608788; BDBM50370614
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| Activity |
IC50 = 96000 nM
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[8] | |||
| Compound Name |
Val-pro-pro
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Investigative | Compound Info | ||
| Synonyms |
L-valyl-L-prolyl-L-proline; H-val-pro-pro-oh; valyl-prolyl-proline; UNII-2U1R84870F; CHEMBL190414; 2U1R84870F; L-Proline, L-valyl-L-prolyl-; L-Proline, 1-(1-L-valyl-L-prolyl)-; L-Val-L-Pro-L-Pro; L-Val-L-Pro-L-Pro-OH; V-P-P; SCHEMBL1644894; BDBM50169128; MFCD08458654; ZINC13646338; HY-114161; CS-0077520; X5324; Q27143860
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| Activity |
Ki = 100000 nM
|
[2] | |||
| Compound Name |
Gln-Gln
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Investigative | Compound Info | ||
| Synonyms |
H-Gln-Gln-OH; Glutaminyl-Glutamine; L-GLUTAMINYL-L-GLUTAMINE; glutaminylglutamine; CHEMBL438960; QQ dipeptide; Q-Q Dipeptide; L-Gln-L-Gln; H-L-Gln-L-Gln-OH; Glutamine Glutamine dipeptide; Glutamine-Glutamine dipeptide; SCHEMBL19375; CTK7D3094; ZINC2391099; BDBM50188528; MFCD00038689; Q27144168; (2S)-5-amino-2-[[(2S)-2,5-diamino-5-oxopentanoyl]amino]-5-oxopentanoic acid
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| Activity |
EC50 = 100000 nM
|
[1] | |||
| Compound Name |
Leu-Pro-Arg
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL361278; Leucyl-prolyl-arginine; L-Leucyl-L-prolyl-L-arginine; BDBM50169215
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| Activity |
Ki = 100000 nM
|
[2] | |||
| Compound Name |
Trp-Ala
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Investigative | Compound Info | ||
| Synonyms |
H-TRP-ALA-OH; CHEMBL188866; tryptophyl-alanine; L-tryptophyl-L-alanine; Tryptophanyl-alanine; L-Trp-L-Ala; L-Trp-L-Ala-OH; L-Tryptophanyl-L-alanine; L-Alanine, L-tryptophyl-; SCHEMBL1617917; CTK1A7723; ZINC1638007; BDBM50169160; MFCD00037965; AKOS010420472; Q27144060; (S)-2-[(S)-2-Amino-3-(1H-indol-3-yl)-propionylamino]-propionic acid
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| Activity |
EC50 = 100000 nM
|
[1] | |||
| Compound Name |
Val-trp
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Investigative | Compound Info | ||
| Synonyms |
L-Valyl-L-tryptophan; N-Valyltryptophan; L-Tryptophan, L-valyl-; H-VAL-TRP-OH; UNII-3G64B4AFQN; valyltryptophan; 3G64B4AFQN; CHEMBL91777; (S)-2-((S)-2-Amino-3-methylbutanamido)-3-(1H-indol-3-yl)propanoic acid; N-L-Valyl-L-tryptophan; L-Val-L-Trp-OH; Spectrum2_001488; Spectrum3_001812; L-Tryptophan, N-L-valyl-; BSPBio_003423; SCHEMBL150533; SPECTRUM1502210; SPBio_001475; CTK1A2687; KBio3_002926; DTXSID40947460; ZINC2047221; BDBM50038066; CCG-39170; MFCD00037947; AKOS015914032; (2S)-2-[[(2S)-2-amino-3-methylbutanoyl]amino]-3-(1H-indol-3-yl)propanoic acid; AS-57858; 587H379; N-(2-Amino-1-hydroxy-3-methylbutylidene)tryptophan; BRD-K46272620-001-02-2; Q27164569; (2S)-2-[(2S)-2-AMINO-3-METHYLBUTANAMIDO]-3-(1H-INDOL-3-YL)PROPANOIC ACID; (S)-2-((S)-2-Amino-3-methyl-butyrylamino)-3-(1H-indol-3-yl)-propionic acid; 2-((S)-2-Amino-3-methyl-butyrylamino)-3-(S)-1H-indol-3-yl-propionic acid
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| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Trimethionine
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Investigative | Compound Info | ||
| Synonyms |
Met-met-met; H-Met-Met-Met-OH; L-METHIONYL-L-METHIONYL-L-METHIONINE; CHEMBL190272; Methionyl-methionyl-methionyl; C15H29N3O4S3; Methionyl-methionyl-methionine; CTK7B5604; DTXSID90162823; ZINC4899465; 7147AA; BDBM50169153; MFCD00038231; AKOS015913861; L-Methionine, N-(N-L-methionyl-L-methionyl)-
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||||
| Activity |
Ki = 100000 nM
|
[2] | |||
| Compound Name |
Tyrosyl-tryptophan
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Investigative | Compound Info | ||
| Synonyms |
H-TYR-TRP-OH; Tyr-Trp; L-tyrosyl-L-tryptophan; CHEMBL210851; L-Tyr-L-Trp; L-Tyr-L-Trp-OH; SCHEMBL9852041; CTK7J9109; ZINC2575132; BDBM50188527; MFCD00083832; Q27145063
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||||
| Activity |
IC50 = 100000 nM
|
[1] | |||
| Compound Name |
Val-Tyr
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Investigative | Compound Info | ||
| Synonyms |
H-VAL-TYR-OH; valyl-tyrosine; L-valyl-L-tyrosine; (S)-2-((S)-2-Amino-3-methylbutanamido)-3-(4-hydroxyphenyl)propanoic acid; CHEMBL90069; L-Val-L-Tyr; L-Val-L-Tyr-OH; L-Tyrosine, L-valyl-; Ang(3-4); SCHEMBL4273366; CTK1C0945; KS-00000YA8; ZINC2384776; BDBM50169147; MFCD00037182; AKOS010408835; CS-W010054; HY-W009338; AS-56393; Q27143866; (S)-2-((S)-2-Amino-3-methyl-butyrylamino)-3-(4-hydroxy-phenyl)-propionic acid
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| Activity |
Ki = 100000 nM
|
[2] | |||
| Compound Name |
Ala-phe-leu
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL191472; Alanyl-phenylalanyl-leucine; CTK0J3102; DTXSID50461066; L-Alanyl-L-phenylalanyl-L-leucine; BDBM50169170; L-Leucine, L-alanyl-L-phenylalanyl-; (2S)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoic acid; (S)-2-[(S)-2-((S)-2-Amino-propionylamino)-3-phenyl-propionylamino]-4-methyl-pentanoic acid
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| Activity |
Ki = 100000 nM
|
[2] | |||
| Compound Name |
Leu-Ala-Arg
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL190897; Leucyl-alanyl-arginine; L-Leucyl-L-alanyl-L-arginine; SCHEMBL9450543; BDBM50169169; (S)-2-[(S)-2-((S)-2-Amino-4-methyl-pentanoylamino)-propionylamino]-5-guanidino-pentanoic acid
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| Activity |
Ki = 100000 nM
|
[9] | |||
| Compound Name |
Aspartyllysine
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Investigative | Compound Info | ||
| Synonyms |
H-ASP-LYS-OH; Asp-lys; L-Aspartyl-L-lysine; Alpha-Aspartyl-lysine; CHEMBL66839; Aspartyl-Lysine; alpha-Asp-Lys; alpha-aspartyllysine; L-alpha-Asp-L-Lys; L-Asp-L-Lys; L-alpha-aspartyl-L-lysine; N2-L-a-aspartyl-L-Lysine; L-Lysine, L-alpha-aspartyl-; N2-L-alpha-aspartyl-L-Lysine; SCHEMBL1308762; ZINC2390911; BDBM50169217; MFCD00038206; Q27144147; (S)-6-amino-2-((S)-2-amino-3-carboxypropanamido)hexanoic acid; (2S)-6-amino-2-[[(2S)-2-amino-3-carboxypropanoyl]amino]hexanoic acid; (S)-6-Amino-2-((S)-2-amino-3-carboxy-propionylamino)-hexanoic acid; 6-Amino-2-(2-amino-3-carboxy-propionylamino)-hexanoic acid (AspLys)
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| Activity |
Ki = 108000 nM
|
[7] | |||
| Compound Name |
H-Phe-phe-OH
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Investigative | Compound Info | ||
| Synonyms |
L-Phe-L-Phe; Phe-Phe; (S)-2-((S)-2-Amino-3-phenylpropanamido)-3-phenylpropanoic acid; L-Phenylalanyl-L-phenylalanine; Phenylalanyl-phenylalanine; CHEMBL55868; (2S)-2-[[(2S)-2-amino-3-phenylpropanoyl]amino]-3-phenylpropanoic acid; MFCD00063154; (2S)-2-{[(2S)-2-amino-3-phenylpropanoyl]amino}-3-phenylpropanoic acid; L-Phe-L-Phe-OH; H-L-Phe-L-Phe-OH; N-Phenylalanylphenylalanine; SCHEMBL825577; KS-00000GE8; ZINC1605264; (2S)-2-[(2S)-2-amino-3-phenylpropanamido]-3-phenylpropanoic acid; BDBM50169134; s6093; 2-(2-Amino-3-phenyl-propionylamino)-3-phenyl-propionic acid; AKOS015919869; CS-W007970; HY-W007970; AS-18242; BR-28439; W4912; S-2406; Q27140102; (2S)-2-[[(2S)-2-amino-3-phenyl-propanoyl]amino]-3-phenyl-propanoic acid; (S)-2-((S)-2-Amino-3-phenyl-propionylamino)-3-phenyl-propionic acid; I(S)-2-((S)-2-Amino-3-phenyl-propionylaIImino)-3-phenyl-propionic acid
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| Activity |
Ki = 110000 nM
|
[2] | |||
| Compound Name |
Leucylproline
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Investigative | Compound Info | ||
| Synonyms |
Leu-pro; l-leucyl-l-proline; L-Proline, L-leucyl-; CHEMBL189210; leucyl-proline; H-Leu-Pro-OH; L-Leu-L-Pro; L-Leu-L-Pro-OH; L-Proline, 1-L-leucyl-; SCHEMBL3052903; CTK2F5692; DTXSID30214012; ZINC4556774; (2S)-1-[(2S)-2-amino-4-methylpentanoyl]pyrrolidine-2-carboxylic acid; BDBM50169151; AKOS010419273; Q27141752; (S)-1-((S)-2-Amino-4-methyl-pentanoyl)-pyrrolidine-2-carboxylic acid
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| Activity |
Ki = 110000 nM
|
[4] | |||
| Compound Name |
Phe-gly
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Investigative | Compound Info | ||
| Synonyms |
H-PHE-GLY-OH; l-Phenylalanyl-glycine; CHEMBL417979; L-Phenylalanylglycine; Phe-Gly hydrate; L-Phe-Gly; L-Phe-Gly-OH; (S)-Phenylalanylglycine; Glycine, N-phenylalanyl-; N-(L-phenylalanyl)glycine; SCHEMBL1329817; CTK7D1065; ZINC1569733; 7220AH; BDBM50139894; KM1459; MFCD00021728; (2-Amino-3-phenyl-propionylamino)-acetic acid; (S)-2-(2-amino-3-phenylpropanamido)acetic acid; ((S)-2-Amino-3-phenyl-propionylamino)-acetic acid; ((S)-3-Amino-2-oxo-4-phenyl-butylamino)-acetic acid; {[(2S)-2-Amino-3-phenylpropanoyl]amino}acetic acid; Q27142685
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| Activity |
EC50 = 110000 nM
|
[1] | |||
| Compound Name |
H-Ala-Phe-Pro-OH
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL187898; alanyl-phenylalanyl-proline; SCHEMBL7259790; ZINC2560943; BDBM50169193; MFCD00237746; (2S)-1-[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-3-phenylpropanoyl]pyrrolidine-2-carboxylic acid; (2S)-1-[(2S)-2-[[(2S)-2-azaniumylpropanoyl]amino]-3-phenylpropanoyl]pyrrolidine-2-carboxylate; (S)-1-[(S)-2-((S)-2-Amino-propionylamino)-3-phenyl-propionyl]-pyrrolidine-2-carboxylic acid
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| Activity |
Ki = 110000 nM
|
[2] | |||
| Compound Name |
(S)-2-{(2S,3R)-2-[((S)-2-Amino-4-methyl-pentanoyl)-methyl-amino]-3-hydroxy-butyrylamino}-4-methyl-pentanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL188159; BDBM50169201
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||||
| Activity |
Ki = 110000 nM
|
[2] | |||
| Compound Name |
Ala-Lys
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Investigative | Compound Info | ||
| Synonyms |
L-Alanyl-L-lysine; L-Lysine, L-alanyl-; CHEMBL191057; alanyl-lysine; Ala-Lys-OH; L-Ala-L-Lys; SCHEMBL1711244; CTK2A8639; DTXSID30426799; ZINC2522662; BDBM50169125; 6-Amino-2-(2-amino-propionylamino)-hexanoic acid; (S)-6-Amino-2-((S)-2-amino-propionylamino)-hexanoic acid; (2S)-6-amino-2-[[(2S)-2-aminopropanoyl]amino]hexanoic acid
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| Activity |
Ki = 117000 nM
|
[7] | |||
| Compound Name |
(2S)-2-[[(2S)-2-Aminopropanoyl]amino]-3-(4-benzylphenyl)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2371152
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| Activity |
Ki = 120000 nM
|
[4] | |||
| Compound Name |
Ile-tyr
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Investigative | Compound Info | ||
| Synonyms |
H-Ile-Tyr-OH; L-ISOLEUCYL-L-TYROSINE; Ile-Tyr-OH; CHEMBL91090; Isoleucyl-Tyrosine; (S)-2-((2S,3S)-2-Amino-3-methylpentanamido)-3-(4-hydroxyphenyl)propanoic acid; L-Ile-L-Tyr; SCHEMBL4261778; CTK6B1461; ZINC4899517; 7185AH; BDBM50038069; MFCD00063032; AKOS010406606; Q27144616
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| Activity |
Ki = 120000 nM
|
[2] | |||
| Compound Name |
Glycyl-L-tyrosine
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Investigative | Compound Info | ||
| Synonyms |
Gly-Tyr; N-Glycyl-L-tyrosine; H-Gly-Tyr-OH; Glycyltyrosine; glycyl-tyrosine; L-Tyrosine, glycyl-; Gly-Tyr-OH; (S)-2-(2-Aminoacetamido)-3-(4-hydroxyphenyl)propanoic acid; UNII-A226496H4O; CHEMBL53400; A226496H4O; L-Tyrosine, glycyl-, monomer; (2S)-2-[(2-aminoacetyl)amino]-3-(4-hydroxyphenyl)propanoic acid; MFCD00008126; n-glycyltyrosine; GY dipeptide; G-Y Dipeptide; EINECS 211-525-1; Gly-L-Tyr; NSC 83260; Gly-L-Tyr-OH; L-Glycyl-L-Tyrosine; NSC 118362; PubChem13027; Glycine Tyrosine dipeptide; Glycine-Tyrosine dipeptide; Glycyl-L-tyrosine 2-hydrate; SCHEMBL479126; CTK2F3209; KS-00000GCF; L-Tyrosine, N-glycyl- (9CI); (2S)-2-(2-aminoacetamido)-3-(4-hydroxyphenyl)propanoic acid; BCP24671; ZINC1730678; BDBM50188508; KM0964; STL466189; AKOS010366204; AC-6976; MCULE-8379516554; DS-13668; G0145; ST50320046; G-6370; 658G797; Q27140599; (2S)-2-(2-aminoacetylamino)-3-(4-hydroxyphenyl)propanoic acid; 2-(2-Amino-acetylamino)-3-(4-hydroxy-phenyl)-propionic acid; (S)-2-(2-Amino-acetylamino)-3-(4-hydroxy-phenyl)-propionic acid
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| Activity |
IC50 = 120000 nM
|
[1] | |||
| Compound Name |
DL-Alanyl-DL-alanine
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Investigative | Compound Info | ||
| Synonyms |
2-(2-aminopropanamido)propanoic acid; Alanylalanine; DL-Ala-DL-Ala; N-DL-Alanyl-DL-alanine; Alanine, alanyl-; 2-(2-aminopropanoylamino)propanoic acid; DL-Alanine, N-DL-alanyl-; L-Alanine, N-L-alanyl-; CHEMBL52461; 2-[(2-ammoniopropanoyl)amino]propanoate; Di-L-Alanine; .alpha.-Alanylalanine; D-Alaninyl-D-alanine; Alanine, N-L-alanyl-, L-; (2R)-2-[[(2R)-2-aminopropanoyl]amino]propanoic acid; alanine-alanine; Alanine, N-DL-alanyl-, DL-; NSC-203792; EINECS 220-687-2; NSC 89654; (2S)-2-(2-aminopropanoylamino)propanoic acid; ACMC-209mbp; ACMC-1AVL4; DL-Ala-DL-Ala, 98%; SCHEMBL159552; N-(2-Aminopropanoyl)alanine #; CTK8B1378; DTXSID30862471; ALBB-023612; KS-00000Y9W; NSC89598; NSC89654; 7505AF; ANW-26445; BDBM50085124; DL-Alanine, N-DL-alanyl- (9CI); MFCD00064407; NSC-89598; NSC-89654; NSC186898; NSC203792; AKOS009159418; MCULE-1972648882; NSC-186898; VC30862; VC31008; ST092688; 2-(2-amino-propanoylamino)-propionic acid; 2-(2-Amino-propionylamino)-propionic acid; DB-040990; DB-044872; DB-047430; DB-049041; DB-057297; FT-0625420; FT-0633100; FT-0633339; FT-0633930; FT-0634973; FT-0693019; R1907; 867A201; J-017187
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| Activity |
Ki = 120000 nM
|
[4] | |||
| Compound Name |
L-Leucyl-L-alanine
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Investigative | Compound Info | ||
| Synonyms |
Leu-ala; Leucyl-alanine; H-Leu-Ala-OH; (S)-2-((S)-2-Amino-4-methylpentanamido)propanoic acid; L-Leucyl-L-alanine hydrate; L-Alanine, L-leucyl-; Alanine, N-L-leucyl-, L-; L-?Leucyl-?L-?alanine; CHEMBL541207; L-Alanine, N-L-leucyl-; l-leu-l-ala; Leu-Ala hydrate; Alanine, leucyl-; EINECS 230-737-5; Leu-Ala-OH; L-Levcyl-L-alanine; NSC 89180; L-Leu-L-Ala-OH; Spectrum2_001499; Spectrum3_001934; L-Leucyl-L-alanineHydrate; BSPBio_003534; SCHEMBL259116; SPECTRUM1502207; SPBio_001517; CTK1H0940; KBio3_002789; DTXSID60884368; L-Alanine, N-L-leucyl- (9CI); ZINC1569727; ANW-60563; BDBM50407466; CCG-39171; KM1530; MFCD00002641; s6153; Leucyl-Alanine; AIF; CE0; CorrDec; AKOS010366053; KS-0000150N; N-(2-Amino-4-methylpentanoyl)alanine #; NCGC00178004-01; HY-128434; CS-0099269; L0126; ST50307162; X5370; Q27140609; (2S)-2-((2S)-2-amino-4-methylpentanoylamino)propanoic acid
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| Activity |
Ki = 120000 nM
|
[4] | |||
| Compound Name |
[(2R,3S,4R,5R)-5-(2-Bromo-5,6-dichlorobenzimidazol-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2S)-2-amino-3-methylpentanoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1791442; BDBM50370616
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| Activity |
IC50 = 121000 nM
|
[8] | |||
| Compound Name |
Glycyl-L-phenylalanine
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Investigative | Compound Info | ||
| Synonyms |
Gly-Phe; Glycyl-phenylalanine; (S)-2-(2-Aminoacetamido)-3-phenylpropanoic acid; H-Gly-Phe-OH; N-Glycyl-3-phenylalanine; CHEMBL299889; Gly-L-Phe; (2S)-2-(2-aminoacetylamino)-3-phenylpropanoic acid; MFCD00065110; Gly-Phe-OH; Gly-L-Phe-OH; 2-(2-Amino-acetylamino)-3-phenyl-propionic acid; SCHEMBL232699; (2S)-2-[(2-aminoacetyl)amino]-3-phenylpropanoic acid; CTK7E1879; ZINC1569529; EINECS 222-027-9; ANW-13819; BDBM50188491; SBB058635; AKOS010366203; AKOS015855060; Gly-Phe, puriss., >=99.0% (NT); DB-002743; G0136; ST50320047; K-0041; 321G037; (S)-2-(2-Amino-acetylamino)-3-phenyl-propionic acid; Q27144236; 784F522A-C4BB-4849-AC2F-13E036818073; (glycyldehydrophenylalanine)2-(2-Amino-acetylamino)-3-phenyl-propionic acid
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| Activity |
EC50 = 130000 nM
|
[1] | |||
| Compound Name |
Ser-Pro
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Investigative | Compound Info | ||
| Synonyms |
H-Ser-Pro-OH; L-Proline, L-seryl-; seryl-proline; (S)-1-((S)-2-Amino-3-hydroxypropanoyl)pyrrolidine-2-carboxylic acid; L-seryl-L-proline; L-serinyl-L-proline; 1-Serylproline; L-Ser-L-Pro; CHEMBL2371153; CTK1A1655; DTXSID90402478; ZINC4899432; MFCD00037333; (2S)-1-[(2S)-2-amino-3-hydroxypropanoyl]pyrrolidine-2-carboxylic acid; Q27144929
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||||
| Activity |
Ki = 130000 nM
|
[4] | |||
| Compound Name |
(2S)-1-[(2S)-2-Amino-3-(1H-indol-2-yl)propanoyl]pyrrolidine-2-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2371155
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||||
| Activity |
Ki = 130000 nM
|
[4] | |||
| Compound Name |
Glycyl-L-proline
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Investigative | Compound Info | ||
| Synonyms |
gly-pro; H-Gly-Pro-OH; N-glycylproline; L-Proline, glycyl-; Glycyl-proline; (S)-1-(2-aminoacetyl)pyrrolidine-2-carboxylic acid; N-Glycyl-L-proline; Glycyl proline; UNII-BJZ69WB3VD; GP-OH; BJZ69WB3VD; CHEMBL80548; Gly-L-Pro; 1-(Aminoacetyl)proline; L-Proline, 1-glycyl- (9CI); Proline, 1-glycyl-, L-; gly pro; Proline, 1-glycyl-, L- (8CI); EINECS 211-880-2; NSC 97929; Gly-L-Pro-OH; GLY-PRO-OH; 1-(2-Amino-acetyl)-pyrrolidine-2-carboxylic acid; (S)-1-(2-Amino-acetyl)-pyrrolidine-2-carboxylic acid; SCHEMBL155067; (2S)-1-(2-aminoacetyl)pyrrolidine-2-carboxylic acid; CTK2H7181; DTXSID701016976; ZINC1637972; ANW-35899; BDBM50169189; MFCD00020840; s6133; AKOS010366353; AKOS015855091; AB01296; CS-W017603; HY-W016887; DS-16203; AB0012963; G0137; X-3940; (2S)-1-(aminoacetyl)pyrrolidine-2-carboxylic acid; J-521416; Q27139057; 2F533D4C-20F0-4B6A-891A-3E2D5D51562C; UNII-1TA6DL3YKT component KZNQNBZMBZJQJO-YFKPBYRVSA-N
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||||
| Activity |
EC50 = 130000 nM
|
[1] | |||
| Compound Name |
Phe-Pro
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Investigative | Compound Info | ||
| Synonyms |
L-phenylalanyl-L-proline; Phenylalanylproline; H-Phe-Pro-OH; (S)-1-((S)-2-Amino-3-phenylpropanoyl)pyrrolidine-2-carboxylic acid; CHEMBL1807686; Phenylalanyl-proline; Phe-Pro-OH; L-Phe-L-Pro; L-Proline, L-phenylalanyl-; SCHEMBL3726264; CTK2G7446; (1R)-1-L-Phenylalanyl-L-proline; (1S)-1-L-Phenylalanyl-L-proline; KS-00000Y9Y; ZINC2392313; (2S)-1-[(2S)-2-amino-3-phenylpropanoyl]pyrrolidine-2-carboxylic acid; BDBM50348852; MFCD00020833; AKOS010419073; AS-72048; H-D-PHE-PRO-OH TRIFLUOROACETATE SALT; Q27144877
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||||
| Activity |
Ki = 130000 nM
|
[4] | |||
| Compound Name |
H-Ser-ser-OH
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Investigative | Compound Info | ||
| Synonyms |
Ser-Ser; L-seryl-L-serine; CHEMBL379810; seryl-serine; Seryl-serin; Ser-Ser-OH; L-Ser-L-Ser; L-Serine, L-seryl-; H-L-Ser-L-Ser-OH; SCHEMBL4958339; CTK5C3628; ZINC2556659; BDBM50188515; MFCD00191021; AKOS006275761; Q27143825
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||||
| Activity |
IC50 = 130000 nM
|
[1] | |||
| Compound Name |
5-Amino-6-methyl-4-oxo-heptanoic acid benzyl ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL189248; BDBM50152063
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|
||||
| Activity |
Ki = 133000 nM
|
[6] | |||
| Compound Name |
Ala-Ser
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Investigative | Compound Info | ||
| Synonyms |
H-Ala-Ser-OH; L-alanyl-L-serine; Ala-Ser-OH; CHEMBL190179; (S)-2-((S)-2-aminopropanamido)-3-hydroxypropanoic acid; L-Serine, L-alanyl-; Alanylserin; N-alanylserine; L-Ala-L-Ser; Serine, alanyl- (9CI); SCHEMBL7123863; CTK1C4649; ZINC1575549; 7055AH; BDBM50169132; MFCD00066028; AKOS010408397; MCULE-4947152314; 303A411; J-018982; Q27140486; (S)-2-((S)-2-Amino-propionylamino)-3-hydroxy-propionic acid
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||||
| Activity |
Ki = 140000 nM
|
[2] | |||
| Compound Name |
Lysylvaline
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Investigative | Compound Info | ||
| Synonyms |
lys-val; H-Lys-Val-OH; L-Valine, L-lysyl-; L-lysyl-L-valine; UNII-ZB4A1U383X; CHEMBL208094; ZB4A1U383X; Lysyl-valin; L-Lys-L-Val; SCHEMBL22612668; CTK1A4971; ZINC1572038; BDBM50188531; Q27141916; (2S)-2-[[(2S)-2,6-diaminohexanoyl]amino]-3-methylbutanoic acid
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||||
| Activity |
EC50 = 140000 nM
|
[1] | |||
| Compound Name |
Ser-Ala
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Investigative | Compound Info | ||
| Synonyms |
H-SER-ALA-OH; L-seryl-L-alanine; CHEMBL192867; (2S)-2-[[(2S)-2-amino-3-hydroxypropanoyl]amino]propanoic acid; seryl-alanine; N-Serylalanine; Serinyl-Alanine; L-Ser-L-Ala; L-Alanine, L-seryl-; SCHEMBL5841680; CTK2F2187; DTXSID20426566; ZINC2384800; 7240AH; BDBM50169164; MFCD00037228; AKOS006275350; Q27144912; (S)-2-((S)-2-Amino-3-hydroxy-propionylamino)-propionic acid
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||||
| Activity |
Ki = 140000 nM
|
[2] | |||
| Compound Name |
Glu-Pro
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Investigative | Compound Info | ||
| Synonyms |
glutamylproline; L-Glutamyl-L-Proline; L-Proline, L-alpha-glutamyl-; EP dipeptide; Glutamyl-Proline; E-P Dipeptide; L-Glu-L-Pro; Glutamate Proline dipeptide; Glutamate-Proline dipeptide; L-alpha-glutamyl-L-proline; CHEMBL2372590; SCHEMBL10779357; Q27140588
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||||
| Activity |
Ki = 140000 nM
|
[4] | |||
| Compound Name |
Phe-Leu-Leu
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL190933; Phenylalanyl-leucyl-leucine; L-Phenylalanyl-L-leucyl-L-leucine; BDBM50169116; (S)-2-[(S)-2-((S)-2-Amino-3-phenyl-propionylamino)-4-methyl-pentanoylamino]-4-methyl-pentanoic acid
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||||
| Activity |
Ki = 140000 nM
|
[2] | |||
| Compound Name |
Val-Ala-Leu
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL189887; Valyl-alanyl-leucine; L-Valyl-L-alanyl-L-leucine; BDBM50169188; ZINC13646344; (S)-2-[(S)-2-((S)-2-Amino-3-methyl-butyrylamino)-propionylamino]-4-methyl-pentanoic acid; (2S)-2-[[(2S)-2-[[(2S)-2-amino-3-methylbutanoyl]amino]propanoyl]amino]-4-methylpentanoic acid
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||||
| Activity |
Ki = 140000 nM
|
[2] | |||
| Compound Name |
Ala-Gly
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Investigative | Compound Info | ||
| Synonyms |
Glycine, L-alanyl-; L-Alanyl-glycine; CHEMBL94250; 2-[[(2S)-2-aminopropanoyl]amino]acetic acid; (S)-2-(2-Aminopropanamido)acetic acid; DL-ALA-GLY; alanyl-glycine; Glycine, alanyl-; Ala-Gly-OH; L-Ala-Gly; SCHEMBL483863; CTK0I2966; ZINC1888744; BDBM50169210; MFCD00065107; (3-Amino-propionylamino)-acetic acid; AKOS010367582; AS-55965; ((S)-2-Amino-propionylamino)-acetic acid; Q27144089
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||||
| Activity |
Ki = 140000 nM
|
[4] | |||
| Compound Name |
(2S)-2-{[(2S)-2-Aminohexanoyl]amino}propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2371154; ZINC4761004; AKOS024337871
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|
||||
| Activity |
Ki = 140000 nM
|
[4] | |||
| Compound Name |
[(2R,3S,4R)-5-(2-Bromo-5,6-dichlorobenzimidazol-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2S)-2-amino-3-(4-chlorophenyl)propanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL607948; BDBM50370613
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||||
| Activity |
IC50 = 142000 nM
|
[8] | |||
| Compound Name |
L-Alanyl-L-proline
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|
Investigative | Compound Info | ||
| Synonyms |
Alanylproline; ALA-PRO; (S)-1-((S)-2-Aminopropanoyl)pyrrolidine-2-carboxylic acid; Ala-Pro hydrate; L-Proline, L-alanyl-; (2S)-1-[(2S)-2-aminopropanoyl]pyrrolidine-2-carboxylic acid; H-Ala-Pro-OH; L-Ala-L-Pro; UNII-C6G5K79L0O; C6G5K79L0O; CHEMBL414828; 1-L-Alanyl-L-proline; alanyl-l-proline; Ala-Pro-OH; EINECS 236-795-8; L-Ala-Pro; NSC 97932; H-Ala-Pro-OH;; PubChem13023; 1-(2-Amino-propionyl)-pyrrolidine-2-carboxylic acid; (S)-alanyl-(S)-proline; SCHEMBL152403; CTK0H4927; KS-00000LZM; ACT05223; ZINC4521128; ANW-19722; BDBM50020390; MFCD00037332; AKOS010419072; AKOS015853859; EBD2203488; DS-16120; SC-95335; AB0017308; DB-000289; 485A591; H-Ala-Pro-OH inverted exclamation mark currencyH2O; Q27140485
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||||
| Activity |
Ki = 150000 nM
|
[4] | |||
| Compound Name |
H-Ala-pro-leu-OH
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Investigative | Compound Info | ||
| Synonyms |
Ala-Pro-Leu; CHEMBL188505; Alanyl-prolyl-leucine; L-Alanyl-L-prolyl-L-leucine; SCHEMBL11090289; BDBM50169121; (2S)-2-[[(2S)-1-[(2S)-2-aminopropanoyl]pyrrolidine-2-carbonyl]amino]-4-methylpentanoic acid; (S)-2-{[(S)-1-((S)-2-Amino-propionyl)-pyrrolidine-2-carbonyl]-amino}-4-methyl-pentanoic acid
Click to Show/Hide
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||||
| Activity |
Ki = 150000 nM
|
[2] | |||
| Compound Name |
(2S)-2-[[(2S)-2-Amino-3-(1H-indol-2-yl)propanoyl]amino]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2371156
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||||
| Activity |
Ki = 160000 nM
|
[4] | |||
| Compound Name |
L-Proline, L-norleucyl-
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Investigative | Compound Info | ||
| Synonyms |
SCHEMBL556799; CHEMBL2371158
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||||
| Activity |
Ki = 160000 nM
|
[4] | |||
| Compound Name |
Tyr-pro
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Investigative | Compound Info | ||
| Synonyms |
L-Tyrosyl-L-proline; CHEMBL1807689; (2S)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carboxylic Acid; YP dipeptide; Y-P Dipeptide; Tyrosine Proline dipeptide; Tyrosyl-prolin; H-Tyr-Pro-OH; L-Tyr-L-Pro-OH; b-Casomorphin (1-2); L-Proline, L-tyrosyl-; SCHEMBL5336562; CTK1G3867; DTXSID20430840; ZINC4899652; 7272AB; BDBM50348856; MFCD00236912; AKOS010419272; (2S)-1-[(2S)-2-azaniumyl-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carboxylate
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|
||||
| Activity |
Ki = 160000 nM
|
[4] | |||
| Compound Name |
[(2R,3S,4R)-5-(2-Bromo-5,6-dichlorobenzimidazol-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2S)-2-amino-3-methylbutanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL607668; BDBM50370608
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||||
| Activity |
IC50 = 166000 nM
|
[8] | |||
| Compound Name |
Ser-Pro-Ile
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL427343; Seryl-prolyl-isoleucine; L-Seryl-L-prolyl-L-isoleucine; BDBM50169140
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||||
| Activity |
Ki = 170000 nM
|
[2] | |||
| Compound Name |
H-Trp-Trp-Trp-OH
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Investigative | Compound Info | ||
| Synonyms |
Trp-Trp-Trp; CHEMBL434535; SCHEMBL9868128; CTK1E8396; DTXSID80658740; Tryptophanyl-tryptophanyl-tryptophan; ZINC5411474; BDBM50169218; MFCD00238208; L-Tryptophyl-L-tryptophyl-L-tryptophan; L-Tryptophan, L-tryptophyl-L-tryptophyl-; L-Tryptophanyl-L-tryptophanyl-L-tryptophan
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||||
| Activity |
Ki = 170000 nM
|
[2] | |||
| Compound Name |
Ala-Ala-Ala
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Investigative | Compound Info | ||
| Synonyms |
H-Ala-Ala-Ala-OH; Alanyl-alanyl-alanine; L-alanyl-L-alanyl-L-alanine; Tri-L-alanine; L-Ala-L-Ala-L-Ala; (S)-2-((S)-2-((S)-2-Aminopropanamido)propanamido)propanoic acid; CHEMBL189368; (2S)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]propanoyl]amino]propanoic acid; Trialanine; alanylalanylalanine; N-L-Alanyl-N-L-alanyl-L-alanine; EINECS 227-538-0; Alanine, alanylalanyl-; A-A-A; SCHEMBL1674747; CTK0E9843; ZINC4533743; BDBM50169192; MFCD00025557; 874A908; Q27140430; (S)-2-[(S)-2-((S)-2-Amino-propionylamino)-propionylamino]-propionic acid
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||||
| Activity |
Ki = 180000 nM
|
[2] | |||
| Compound Name |
(2R)-1-[(2S)-2,6-Diaminohexanoyl]pyrrolidine-2-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL209032; BDBM50188517
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|
||||
| Activity |
EC50 = 190000 nM
|
[1] | |||
| Compound Name |
His-Trp
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Investigative | Compound Info | ||
| Synonyms |
histidyltryptophan; L-histidyl-L-tryptophan; CHEMBL209765; H-His-Trp-OH; Histidinyl-Tryptophan; Histidyl-tryptophan; L-His-L-Trp; SCHEMBL7046020; SCHEMBL21641789; BDBM50188497; MFCD00037949; Q27144371
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||||
| Activity |
EC50 = 190000 nM
|
[1] | |||
| Compound Name |
Ile-Val-Tyr
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL188747; isoleucyl-valyl-tyrosine; L-Ile-L-Val-L-Tyr-OH; L-Isoleucyl-L-valyl-L-tyrosine; CTK0E7828; DTXSID30459289; L-Tyrosine, L-isoleucyl-L-valyl-; BDBM50169207
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||||
| Activity |
Ki = 200000 nM
|
[2] | |||
| Compound Name |
H-Glu-Phe-Tyr-OH
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Investigative | Compound Info | ||
| Synonyms |
Glu-Phe-Tyr; CHEMBL363341; Glutamyl-phenylalanyl-tyrosine; BDBM50169202; L-Glutamyl-L-phenylalanyl-L-tyrosine; MFCD00237883; ZINC13646347
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||||
| Activity |
Ki = 200000 nM
|
[2] | |||
| Compound Name |
Cysteinylglycine
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Investigative | Compound Info | ||
| Synonyms |
Cys-Gly; L-Cysteinylglycine; Glycine, L-cysteinyl-; L-Cysteinyl-glycine; cysteinyl-glycine; N-L-cysteinylglycine; H-Cys-Gly-OH; UNII-384644SZ9T; CHEMBL371579; (R)-2-(2-Amino-3-mercaptopropanamido)acetic acid; Glycine, N-cysteinyl; 384644SZ9T; cysteine-glycine; CCRIS 2905; L-cysteinylglycine zwitterion; BRN 1724689; Glycine, N-L-cysteinyl-; 2-[[(2R)-2-amino-3-sulfanylpropanoyl]amino]acetic acid; N-cysteinyl Glycine; N-Cysteinyl-Glycine; N-L-cysteinyl-Glycine; 4-04-00-03158 (Beilstein Handbook Reference); SCHEMBL213626; CTK0H6652; DTXSID10864877; ZINC4095652; BDBM50169213; MFCD00055567; AKOS006272654; HY-113110; CS-0059601; C01419; Q27106297; 1F802DB1-4F4D-4B9F-9C68-CA4998E23132
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|
||||
| Activity |
Ki = 200000 nM
|
[2] | |||
| Click to Show/Hide the Information of All Poor Binders | |||||
| Non Binders of This Target (in total, 204 non binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
Cyclacillin
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|
Approved | Compound Info | ||
| Synonyms |
Aminocyclohexylpenicillin; Bastcillin; Calthor; Ciclacilina; Ciclacillin; Ciclacilline; Ciclacillinum; Ciclacillum; Citosarin; Cyclapen; Noblicil; Orfilina; Peamezin; Syngacillin; Ultracillin; Vastcillin; Vipicil; Wyvital; Aminocyclohexyl penicillin; Cyclacillin [USAN]; AC 98; WY 4508; WY4508; C-12104; Ciclacilina [INN-Spanish]; Ciclacilline [INN-French]; Ciclacillinum [INN-Latin]; Cyclacillin (USAN); Cyclapen (TN); Cyclapen-W; Vastcillin (TN); Wy-4508; Ciclacillin (JP15/INN); Cyclapen-W (TN); (1-Aminocyclohexyl)penicillin; (2S,5R,6R)-6-[(1-aminocyclohexanecarbonyl)amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-{[(1-aminocyclohexyl)carbonyl]amino}-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; 4-Thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid, 6-(1-aminocyclohexanecarboxamido)-3,3-dimethyl-7-oxo-(8CI); 6-(1-Aminocyclohexanecarboxamido)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid; 6-(1-Aminocyclohexanecarboxamido)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; 6-(1-Aminocyclohexanecarboxamido)penicillanic acid; 6-(1-Aminocyclohexylcarboxamido)penicillanic acid; 6beta-(1-aminocyclohexanecarboxamido)-2,2-dimethylpenam-3alpha-carboxylic acid
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|
||||
| Activity |
IC50 = 350000 nM
|
[10] | |||
| Compound Name |
Valaciclovir
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|
Approved | Compound Info | ||
| Synonyms |
Talavir; VACV; ValACV; Valacyclovir; Virval; Zelitrex; Valaciclovir Hcl; Valacyclover Hydrochloric; Valacyclover Hydrochloride; BW256U87; TBB067866; Acyclovir-valine; BW-256U; Valaciclovir (INN); Valaciclovir [INN:BAN]; Valaciclovir, Valtrex; Valtrex (TN); Zelitrex (TN); Valacyclovir, (L)-isomer; L-Valine ester with 9-((2-hydroxyethoxy)methyl)guanine; L-Valine, 2-((2-amino-1,6-dihydro-6-oxo-9H-purin-9-yl)methoxy)ethyl ester; L-valine, 2-[(2-amino-1,6-dihydro-6-oxo-9 H-purin-9-yl)methoxy]ethyl ester, monohydrochloride; 2-[(2-amino-6-oxo-1,6-dihydro-9H-purin-9-yl)methoxy]ethyl L-valinate; 2-[(2-amino-6-oxo-3H-purin-9-yl)methoxy]ethyl (2S)-2-amino-3-methylbutanoate; 2-{[(2-amino-6-oxo-1,6-dihydro-9H-purin-9-yl)methyl]oxy}ethyl L-valinate
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|
||||
| Activity |
IC50 = 400000 nM
|
[11] | |||
| Compound Name |
Aminolevulinic acid hci
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|
Approved | Compound Info | ||
| Synonyms |
Aminolevulinic acid; 5-Aminolevulinic acid; 5-Amino-4-oxopentanoic acid; 106-60-5; 5-Aminolevulinate; delta-aminolevulinic acid; Pentanoic acid, 5-amino-4-oxo-; Aladerm; 5-Amino-4-oxovaleric acid; Kerastick; Ameluz; Aminolevulinate; 5-ALA; delta-ALA; 5-Amino-4-oxopentanoate; 5-amino-levulinate; 5-amino-levulinic acid; 5-amino-4-oxo-pentanoic acid; CCRIS 8958; UNII-88755TAZ87; EINECS 203-414-1; Levulinic acid, 5-amino-; CHEMBL601; 4-oxo-5-amino-pentanoic acid; CHEBI:17549; ZGXJTSGNIOSYLO-UHFFFAOYSA-N; 88755TAZ87; Levulan (TN)
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|
||||
| Activity |
Ki = 790000 nM
|
[4] | |||
| Compound Name |
Cefadroxil
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|
Approved | Compound Info | ||
| Synonyms |
CDX; Cefadroxilo; Cefadroxilum; Cephadroxil; Sumacef; Cefadroxil anhydrous; S 578; BL-S 578; BL-S578; Cefadroxil (JP15); Cefadroxilo [INN-Spanish]; Cefadroxilum [INN-Latin]; Curisafe (TN); D-Cefadroxil; S-578; Sumacef (TN); MJF-11567-3; (6R,7R)-7-((R)-2-Amino-2-(p-hydroxyphenyl)acetamido)-3-methyl-8-oxo-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid; (6R,7R)-7-[[(2R)-2-amino-2-(4-hydroxyphenyl)acetyl]amino]-3-methyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-{[(2R)-2-amino-2-(4-hydroxyphenyl)acetyl]amino}-3-methyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 7beta-{[(2R)-2-amino-2-(4-hydroxyphenyl)acetyl]amino}-3,4-didehydrocepham-4-carboxylic acid
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|
||||
| Activity |
IC50 = 870000 nM
|
[10] | |||
| Compound Name |
Cefixime
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|
Approved | Compound Info | ||
| Synonyms |
CFIX; Cefixima; Cefiximum; Denvar; Necopen; Tricef; CL-284635; FK-027; FR-17027; Ofex (TN); Suprax (TN); Cefixime (JP15/USP/INN); (6R,7R)-7-({(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-[(carboxymethoxy)imino]acetyl}amino)-3-ethenyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-(carboxymethyloxyimino)acetyl]amino]-3-ethenyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-{[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-{[(carboxymethyl)oxy]imino}acetyl]amino}-3-ethenyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6r,7r)-7-[-2-(2-amino-thiazol-4-yl)-2-carboxymethoxyimino-acetylamino]-8-oxo-3-vinyl-5-thia-1-aza-b; 7beta-{(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-[(carboxymethoxy)imino]acetamido}-3-ethenyl-3,4-didehydrocepham-4-carboxylic acid
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|
||||
| Activity |
Ki = 1310000 nM
|
[12] | |||
| Compound Name |
Cloxacillin
Click to Show/Hide
|
Approved | Compound Info | ||
| Synonyms |
Chloroxacillin; Clossacillina; Cloxacilina; Cloxacilline; Cloxacillinum; MCIPC; Orbenin; Syntarpen; Tegopen; Clossacillina [DCIT]; Cloxacillin sodium; Methocillin S; BRL 1621; Cloxacilina [INN-Spanish]; Cloxacillin (INN); Cloxacillin [INN:BAN]; Cloxacilline [INN-French]; Cloxacillinum [INN-Latin]; Cloxapen (TN); Cloxapen (sodium monohydrate); Methylchlorphenylisoxazoryl-penicillin; Novo-Cloxin; Nu-Cloxi; Orbenin (TN); Tegopen (sodium monohydrate); BRL-1621 (sodium monohydrate); P-25 (sodium monohydrate); [3-(O-CHLOROPHENYL)-5-METHYL-4-ISOXAZOLYL]PENICILLIN; (2S,5R,6R)-6-({[3-(2-chlorophenyl)-5-methylisoxazol-4-yl]carbonyl}amino)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-[[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (3-(o-Chlorophenyl)-5-methyl-4-isoxazolyl)penicillin; 6-(((3-(2-Chlorophenyl)-5-methyl-4-isoxazolyl)carbonyl)amino)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid; 6-(3-(o-Chlorophenyl)-5-methyl-4-isoxazolecarboxamido)penicillanic acid
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| Activity |
Ki = 2500000 nM
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[2] | |||
| Compound Name |
Flucloxacillin
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Approved | Compound Info | ||
| Synonyms |
FLOXACILLIN; Floxapen; Fluclox; Flucloxacilina; Flucloxacilline; Flucloxacillinum; Fluorochloroxacillin; MFIPC; Floxacillin [USAN]; Flucloxacillin sodium; BRL 2039; Flopen (TN); Floxacillin (USAN); Floxapen (TN); Flucloxacilina [INN-Spanish]; Flucloxacillin (INN); Flucloxacillin-Sodium; Flucloxacilline [INN-French]; Flucloxacillinum [INN-Latin]; Rel-(2R,6S)-6-({[3-(2-chloro-6-fluorophenyl)-5-methylisoxazol-4-yl]carbonyl}amino)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylato; (2S,5R,6R)-6-({[3-(2-chloro-6-fluorophenyl)-5-methyl-1,2-oxazol-4-yl]carbonyl}amino)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-({[3-(2-chloro-6-fluorophenyl)-5-methylisoxazol-4-yl]carbonyl}amino)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-[[3-(2-chloro-6-fluorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; 3-(2-Chloro-6-fluorophenyl)-5-methyl-4-isoxazolylpenicillin; 4-Thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid, 6-(((3-(2-chloro-6-fluorophenyl)-5-methyl-4-isoxazolyl)carbonyl)amino)-3,3-dimethyl-7-oxo-, (2S(2alpha,5alpha,6beta)); 6beta-[3-(2-chloro-6-fluorophenyl)-5-methyl-1,2-oxazole-4-carboxamido]-2,2-dimethylpenam-3alpha-carboxylic acid
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| Activity |
Ki = 3200000 nM
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[2] | |||
| Compound Name |
Enalapril
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Approved | Compound Info | ||
| Synonyms |
Vasotec; Enalapril (INN); Enalapril (TN); N-{(1S)-1-[(ethyloxy)carbonyl]-3-phenylpropyl}-L-alanyl-L-proline; N-[(2S)-1-ethoxy-1-oxo-4-phenylbutan-2-yl]-L-alanyl-L-proline; (2S)-1-[(2S)-2-[[(2S)-1-ethoxy-1-oxo-4-phenylbutan-2-yl]amino]propanoyl]pyrrolidine-2-carboxylic acid
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| Activity |
IC50 = 4500000 nM
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[13] | |||
| Compound Name |
Cephalexin
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Approved | Compound Info | ||
| Synonyms |
Adcadina; Ades[prex; Alcephin; Alexin; Alsporin; Ambal; Aristosporin; Azabort; Bactopenor; Beliam; Biocef; CEX; Carnosporin; Cefablan; Cefacet; Cefadal; Cefadin; Cefadina; Cefalekey; Cefaleksin; Cefalessina; Cefalexgobens; Cefalexin; Cefalexina; Cefalexine; Cefalexinum; Cefalin; Cefalival; Cefaloto; Cefaseptin; Cefax; Ceffanex; Cefibacter; Ceflax; Ceforal; Cefovit; Celexin; Cepastar; Cepexin; Cephacillin; Cephalexine; Cephalexinum; Cephalobene; Cephanasten; Cephaxin; Cephin; Cepol; Ceporex; Ceporexin; Ceporexine; Check; Cophalexin; Domucef; Doriman; Durantel; Efemida; Erocetin; Factagard; Felexin; Fexin; Ibilex; Ibrexin; Inphalex; Karilexina; Kefalospes; Keflet; Keflex; Kefolan; Keforal; Keftab; Kekrinal; Kidolex; Lafarine; Larixin; Lenocef; Lexibiotico; Loisine; Lonflex; Lopilexin; Losporal; Madlexin; Maksipor; Mamalexin; Mamlexin; Medolexin; Medoxine; Neokef; Neolexina; Noveol; Novolexin; Nufex; Oracef; Oriphex; Oroxin; Ortisporina; Ospexin; Palitrex; Pectril; Prindex; Pyassan; Rilexine; Roceph; Rogevil; Sanaxin; Sartosona; Sencephalin; Sepexin; Servicef; Servispor; Sialexin; Sinthecillin; Sintolexyn; Sporicef; Sporidex; Syncl; Syncle; Synecl; Tepaxin; Theratrex; Tokiolexin; Uphalexin; Viosporine; Voxxim; Winlex; Zabytrex; Zozarine; Cefalessina [DCIT]; Cefalexin Scand Pharm; Cefalexin Sodium; Cefalexin generics; Cefalexin hydrate; Cefalexin monohydrate; Cefalexina Northia; Cefalexina Richet; Cephalex von ct; Cephalexin hydrate; Cephalexin monohydrate; Ceporex Forte; Durantel DS; Henina Oral; Panixine Disperdose; Roceph Distab; Lilly 66873; S 6437; SQ 20248; Cefa-iskia; Cefalexin (JP15); Cefalexin.H2O; Cefalexina [INN-Spanish]; Cefalexine [INN-French]; Cefalexinum [INN-Latin]; Cephalexin(USP); Cephalexin (anhydrous); Cephalexin 1-hydrate; Cephalexin 1-wasser; Cephalexin [USAN:BAN]; Cephalexin.H2O; Ceporexin-E; Cusisporina-Cefalox; Ed A-Ceph; KS-1134; Keflex (TN); Keftab (TN); L-Keflex; Panixine disperdose (TN); Sporidex (TN); Cephalexin, (6R-(6alpha,7beta))-Isomer; 7-(D-2-Amino-2-phenylacetamido)-3-methyl-delta (sup 3)-cephem-4-carboxylic acid; 7-(D-2-Amino-2-phenylacetamido)-3-methyl-delta3-cephem-4-carboxylic acid; 7-(D-alpha-Aminophenylacetamido)desacetoxycephalosporanic acid
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| Activity |
IC50 = 5200000 nM
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[5] | |||
| Compound Name |
Dicloxacillin
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Approved | Compound Info | ||
| Synonyms |
Dichloroxacillin; Diclossacillina; Dicloxaciclin; Dicloxacilin; Dicloxacilina; Dicloxacilline; Dicloxacillinum; Dicloxacycline; Dycill; Dynapen; Maclicine; Methyldichlorophenylisoxazolylpenicillin; Pathocil; Diclossacillina [DCIT]; Dicloxacillin sodium; BRL 1702; Diclocil (TN); Dicloxacilina [INN-Spanish]; Dicloxacilline [INN-French]; Dicloxacillinum [INN-Latin]; R-13423; Dicloxacillin (USAN/INN); Dicloxacillin [USAN:INN:BAN]; Dicloxacillin, Monosodium Salt, Mono-Hydrate; (2S,5R,6R)-6-({[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]carbonyl}amino)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-({[3-(2,6-dichlorophenyl)-5-methylisoxazol-4-yl]carbonyl}amino)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-[[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; 3-(2,6-Dichlorophenyl)-5-methyl-4-isoxazolylpenicillin; 6-(3-(2,6-Dichlorophenyl)-5-methyl-4-isoxazolecarboxamido)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid; 6-(3-(2,6-Dichlorophenyl)-5-methyl-4-isoxazolecarboxamido)penicillanic acid; 6beta-{[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]carboxamido}-2,2-dimethylpenam-3alpha-carboxylic acid
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| Activity |
Ki = 7200000 nM
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[2] | |||
| Compound Name |
Cefamandole
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Approved | Compound Info | ||
| Synonyms |
Cefadole; Cefamandolum; Cefamandole (USAN/INN); (6R,7R)-7-(R)-Mandelamido-3-(((1-methyl-1H-tetrazol-5-yl)thio)methyl)-8-oxo-5-thia-1-azabicyclo(4.2.0)oct-2-ene-carboxylic acid; (6R,7R)-7-[[(2R)-2-hydroxy-2-phenylacetyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-{[(2R)-2-hydroxy-2-phenylacetyl]amino}-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-{[(2R)-2-hydroxy-2-phenylacetyl]amino}-3-{[(1-methyl-1H-tetrazol-5-yl)thio]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 7beta-[(2R)-2-hydroxy-2-phenylacetamido]-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}ceph-3-em-4-carboxylic acid
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| Activity |
Ki = 8100000 nM
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[2] | |||
| Compound Name |
Cefaclor
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Approved | Compound Info | ||
| Synonyms |
Alenfral; Alfacet; Alfatil; CCL; Ceclor; Cefaclorum; Distaclor; Kefolor; Panacef; Panoral; Alfatil Kapseln; Cefaclor anhydrous; Cefaclor hydrate; Cefaclor monohydrate; Dystaclor MR; Kefolor Suspension; Muco Panoral; Lilly 99638 hydrate; Alenfral (TN); Ceclor (TN); Cefaclor (JP15); Cefaclor (USP); Distaclor (TN); Keflor (TN); L-Kefral; Raniclor (TN); S-6472; Cefaclor-1-wasser; Cefaclor [USAN:INN:BAN:JAN]; Ceclor, Distaclor, Keflor, Raniclor, Cefaclor; (6R,7R)-7-((R)-2-Amino-2-phenylacetamido)-3-chloro-8-oxo-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid monohydrate; (6R,7R)-7-[[(2R)-2-amino-2-phenylacetyl]amino]-3-chloro-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-[[(2R)-2-amino-2-phenylacetyl]amino]-3-chloro-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid hydrate; (6R,7R)-7-{[(2R)-2-amino-2-phenylacetyl]amino}-3-chloro-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 3-Chloro-7-D-(2-phenylglycinamido)-3-cephem-4-carboxylic acid; 3-Chloro-7-D-(2-phenylglycinamido)-3-cephem-4-carboxylic acid monohydrate; 7-(2-Amino-2-phenyl-acetylamino)-3-chloro-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 7beta-{[(2R)-2-amino-2-phenylacetyl]amino}-3-chloro-3,4-didehydrocepham-4-carboxylic acid
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| Activity |
IC50 = 8200000 nM
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[13] | |||
| Compound Name |
Cefradine
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Approved | Compound Info | ||
| Synonyms |
Anspor; Cefradin; Cefradina; Cefradinum; Cephradin; Cephradine; Eskacef; Sefril; Velosef; CEPHRADINE SODIUM; SKF D 39304; SQ 11436; VELOSEF 125; VELOSEF 250; VELOSEF 500; Anspor (TN); Cefradina [INN-Spanish]; Cefradinum [INN-Latin]; Cephradine (USP); Cephradine (anhydrous); Cephradine [USAN:BAN]; SQ-11436; SQ-22022; Velosef (TN); Cefradine (JAN/INN); SK&F D-39304; SK-D-39304; (6R,7R)-7-((R)-2-Amino-2-(1,4-cyclohexadien-1-yl)acetamido)-3-methyl-8-oxo-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid; (6R,7R)-7-[[(2R)-2-amino-2-cyclohexa-1,4-dien-1-ylacetyl]amino]-3-methyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-{[(2R)-2-amino-2-cyclohexa-1,4-dien-1-ylacetyl]amino}-3-methyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 7-(D-2-Amino-2-(1,4-cyclohexadien-1-yl)acetamido)-3-methyl-8-oxo-5-thia-1-azabicyclo(4.2.0)-oct-2-ene-2-caboxylic acid; 7-(D-2-Amino-2-(1,4-cyclohexadienyl)acetamide)desacetoxycephalosporanicacid; 7beta-[(2R)-2-(cyclohexa-1,4-dienyl)-2-phenylacetamido]-3-methyl-3,4-didehydrocepham-4-carboxylic acid
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| Activity |
Ki = 9800000 nM
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[2] | |||
| Compound Name |
Cephapirin
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Approved | Compound Info | ||
| Synonyms |
CEPR; Cefa; Cefadyl; Cefapirin; Cefapirina; Cefapirine; Cefapirinum; Cefaprin; Cephapirine; Metricure; CEPHAPIRIN SODIUM; Cefaprinsodium; Cephapirin Monosodium Salt; ANTIBIOTIC BL-P1322; BL-P 1322; Cefa-ak; Cefadyl (TN); Cefapirin (BAN); Cefapirin [INN:BAN]; Cefapirina [INN-Spanish]; Cefapirine [INN-French]; Cefapirinum [INN-Latin]; Metricure (TN); (6R,7R)-3-(Acetoxymethyl)-8-oxo-7-(2-(4-pyridylthio)acetamido)-5-thia-1-azabicyclo(4.2.0)oct-2-en-2-carbonsaeure; (6R,7R)-3-(acetyloxymethyl)-8-oxo-7-[(2-pyridin-4-ylsulfanylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-3-[(acetyloxy)methyl]-8-oxo-7-{[(pyridin-4-ylthio)acetyl]amino}-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-3-acetoxymethyl-7-[(pyridin-4-ylsulfanyl)acetamido]-3,4-didehydrocepham-4-carboxylic acid; 3-(Hydroxymethyl)-8-oxo-7-(2-(4-pyridylthio)acetamidol-5-thia-1-azabicyclo(4.2.0)oct-2-en-2carbonsaeure acetat; 5-Thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid, 3-(hydroxymethyl)-8-oxo-7-(2-(4-pyridylthio)acetamido)-, acetate (ester); 7-(2-(4-Pyridylthio)acetamido)cephalosporanic acid
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| Activity |
Ki > 10000000 nM
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[2] | |||
| Compound Name |
Cefalotin
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Approved | Compound Info | ||
| Synonyms |
Cefalothin; Cefalotina; Cefalotine; Cefalotinum; Cemastin; Cephalothinum; Cephalotin; Coaxin; Cefalotina fabra; Cephalothin Monosodium Salt; Averon-1; Cefalotin (BAN); Cefalotina [INN-Spanish]; Cefalotina fabra (TN); Cefalotine [INN-French]; Cefalotinum [INN-Latin]; Keflin (TN); (6R,7R)-3-(acetyloxymethyl)-8-oxo-7-[(2-thiophen-2-ylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-3-[(acetyloxy)methyl]-8-oxo-7-[(2-thienylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 3-(Acetoxymethyl)-8-oxo-7-(2-(2-thienyl)acetamido)-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid; 3-(Hydroxymethyl)-8-oxo-7-(2-(2-thienyl)acetamido)-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid acetate; 3-ACETOXYMETHYL-8-OXO-7-(2-THIOPHEN-2-YL-ACETYLAMINO)-5-THIA-1-AZA-BICYCLO[4.2.0]OCT-2-ENE-2-CARBOXYLIC ACID; 3-Acetoxymethyl-7-(2-thienylacetamido)-3-cephem-4-carboxylic acid; 5-Thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid, 3-(hydroxymethyl)-8-oxo-7-(2-(2-thienyl)acetamido)-, acetate (ester); 6R-trans-3-((Acetyloxy)methyl)-8-oxo-7-((2-thienylacetyl)amino)-5-thia-1-azabicyclo(4.2.0)-oct-2-ene-2-carboxylic acid; 7-(2-(2-Thienyl)acetylamido)cephalosporanic acid; 7-(2-Thienylacetamido)cephalosporanic acid; 7-(Thiophene-2-acetamido)cephalosporanic acid; 7-(Thiophene-2-acetamido)cephalosporin; 7beta-(thiophen-2-ylacetamido)-3-acetoxymethyl-3,4-didehydrocepham-4-carboxylic acid
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| Activity |
Ki > 10000000 nM
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[2] | |||
| Compound Name |
Amoxicillin
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Approved | Compound Info | ||
| Synonyms |
AMPC; Actimoxi; Amoclen; Amolin; Amopen; Amopenixin; Amoxi; Amoxibiotic; Amoxicaps; Amoxicilina; Amoxicillanyl; Amoxicilline; Amoxicillinum; Amoxiden; Amoxil; Amoxivet; Amoxycillin; Anemolin; Aspenil; Biomox; Bristamox; Cemoxin; Clamoxyl; Delacillin; DisperMox; Efpenix; Flemoxin; Hiconcil; Histocillin; Hydroxyampicillin; Ibiamox; Imacillin; Lamoxy; Larotid; Moxacin; Moxal; Moxatag; Ospamox; Pamoxicillin; Piramox; Polymox; Robamox; Sumox; Tolodina; Trimox; Unicillin; Utimox; Vetramox; Wymox; AMOXICILLIN CRYSTALLINE; AMOXICILLIN PEDIATRIC; Amoxicillin anhydrous; Amoxicilline [INN]; Amoxycillin Trihydrate; Metafarma capsules; Metifarma capsules; Sawamox PM; BLP 1410; AMK (TN); Actimoxi (TN); Alphamox (TN); Amoksibos (TN); Amoksiklav (TN); Amoxi-Mast; Amoxibiotic (TN); Amoxicilina (TN); Amoxicilina [INN-Spanish]; Amoxicillin (INN); Amoxicillin (TN); Amoxicillin (anhydrous); Amoxicilline [INN-French]; Amoxicillinum [INN-Latin]; Amoxiclav (TN); Amoxidal (TN); Amoxil (TN); Amoxin (TN); Apo-Amoxi; Augmentin (TN); BL-P 1410; BRL-2333; Bactox (TN); Betalaktam (TN); Cilamox (TN); Clamoxyl (TN); Curam (TN); D-Amoxicillin; Dedoxil (TN); Dispermox (TN); Duomox (TN); Enhancin (TN); Geramox (TN); Gimalxina (TN); Hiconcil (TN); Isimoxin (TN); Klavox (TN); Lamoxy (TN); Moxatag (TN); Moxilen (TN); Moxypen (TN); Moxyvit (TN); Nobactam (TN); Novamoxin (TN); Ospamox (TN); P-Hydroxyampicillin; Pamoxicillin (TN); Panamox (TN); Panklav (TN); Polymox (TN); Ro 10-8756; Samthongcillin (TN); Sandoz (TN); Senox (TN); Sinacilin (TN); Tolodina (TN); Trimox (TN); Wymox (TN); Yucla (TN); Zerrsox (TN); Zimox (TN); Apo-Amoxi (TN); Alpha-Amino-p-hydroxybenzylpenicillin; D-2-Amino-2-(4-hydroxyphenyl)acetamidopenicillanic acid; D-(-)-alpha-Amino-p-hydroxybenzylpenicillin; (-)-6-(2-Amino-2-(P-hydroxyphenyl)acetamido)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo-(3.2.0)heptane-2-carboxylic acid; (2S,5R,6R)-6-[[(2R)-2-amino-2-(4-hydroxyphenyl)acetyl]amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-{[(2R)-2-amino-2-(4-hydroxyphenyl)acetyl]amino}-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; 4-Thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid, 6-(2-amino-2-(p-hydroxyphenyl)acetamido)-3,3-dimethyl-7-oxo-, D-(8CI); 6-(D-(-)-alpha-Amino-p-hydroxyphenylacetamido)penicillanic acid; 6-(D-(-)-p-Hydroxy-alpha-aminobenzyl)penicillin; 6-(p-Hydroxy-alpha-aminophenylacetamido)penicillanic acid; 6beta-[(2R)-2-amino-2-(4-hydroxyphenyl)acetamido]-2,2-dimethylpenam-3alpha-carbonyl; 6beta-[(2R)-2-amino-2-(4-hydroxyphenyl)acetamido]-2,2-dimethylpenam-3alpha-carboxylic acid
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| Activity |
Ki > 10000000 nM
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[14] | |||
| Compound Name |
Ampicillin
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Approved | Compound Info | ||
| Synonyms |
ABPC; Acillin; Adobacillin; Alpen; Amblosin; Amcill; Amfipen; Aminobenzylpenicillin; Ampen; Ampichel; Ampicil; Ampicilina; Ampicillanyl; Ampicillina; Ampicilline; Ampicillinum; Ampicin; Ampifarm; Ampikel; Ampimed; Ampipenin; Ampiscel; Ampisyn; Ampivax; Ampivet; Amplacilina; Amplin; Amplipenyl; Amplisom; Amplital; Austrapen; Binotal; Bonapicillin; Britacil; Campicillin; Cimex; Copharcilin; Delcillin; Deripen; Divercillin; Doktacillin; Duphacillin; Grampenil; Guicitrina; Guicitrine; Lifeampil; Morepen; Norobrittin; Nuvapen; Omnipen; Orbicilina; Penbristol; Penbritin; Penbrock; Penicline; Penimic; Pensyn; Pentrex; Pentrexl; Pentrexyl; Polycillin; Ponecil; Princillin; Principen; QIDamp; Racenacillin; Rosampline;Roscillin; Semicillin; Servicillin; Sumipanto; Supen; Synpenin; Texcillin; Tokiocillin; Tolomol; Totacillin; Totalciclina; Totapen; Trifacilina; Ukapen; Ultrabion; Ultrabron; Vampen; Viccillin; Wypicil; Amfipen V; Amipenix S; Ampicillin A; Ampicillin Anhydrous; Ampicillin Base; Ampicillin acid; Ampicillin anhydrate; Ampicillina [DCIT]; Anhydrous ampicillin; Olin Kid; Pen A; Pen A Oral; Pen Ampil;Penbritin paediatric; Penbritin syrup; Pfizerpen A; Semicillin R; Viccillin S; AY 6108; BA 7305; BRL 1341; Bayer 5427; HI 63; P 50; Principen 125; Principen 250; Principen 500; SQ 17382; AB-PC; AB-PCSol; AY-6108; Ambidrin (TN); Ampi-Co; Ampi-Tab; Ampi-bol; Ampicilina [INN-Spanish]; Ampicilline [INN-French]; Ampicillinum [INN-Latin]; Ampipenin, nt3; Ampy-Penyl; Anhydrous ampicillin (JP15); BRL-1341; D-Ampicillin; D-Cillin; KS-R1; Novo-ampicillin; OMNIPEN (AMPICILLIN); Omnipen (TN); Omnipen-N; P-50; Penbritin-S; Penicillin, Aminobenzyl; Pfizerpen-A; Polycillin-N; Polyflex (Veterinary); Ro-Ampen; SK-Ampicillin; Totacillin (sodium); Totacillin-N; WY-5103; Ampicillin (USP/INN); AMPICILLIN (SEE ALSO AMPICILLIN TRIHYDRATE 7177-48-2); Ampicillin [USAN:BAN:INN:JAN]; Ampicillin [USAN:INN:BAN:JAN];D-(-)-Ampicillin; D-(-)-alpha-Aminobenzylpenicillin; D-(-)-alpha-Aminopenicillin; D-(-)-6-(alpha-Aminophenylacetamido)penicillanic acid; 6-(D(-)-alpha-Aminophenylacetamido)penicillanic acid; 6beta-[(2R)-2-amino-2-phenylacetamido]-2,2-dimethylpenam-3alpha-carbonyl; 6beta-[(2R)-2-amino-2-phenylacetamido]-2,2-dimethylpenam-3alpha-carboxylic acid
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| Activity |
IC50 = 10000000 nM
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[5] | |||
| Compound Name |
Oxacillin
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Approved | Compound Info | ||
| Synonyms |
Bactocill; Ossacillina; Oxacilina; Oxacilline; Oxacillinum; Oxazocillin; Oxazocilline; Prostaphlin; Prostaphlyn; OXACILLIN SODIUM; Ossacillina [DCIT]; Sodium oxacillin; Bactocill (TN); MPI-penicillin; MPi-PC; Oxacilina (TN); Oxacilina [INN-Spanish]; Oxacillin (INN); Oxacillin [INN:BAN]; Oxacilline [INN-French]; Oxacillinum [INN-Latin]; Penicillin, Methylphenylisoxazolyl; Oxacillin, Monosodium Salt, Anhydrous; (2S,5R,6R)-3,3-dimethyl-6-[(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)amino]-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-3,3-dimethyl-6-{[(5-methyl-3-phenylisoxazol-4-yl)carbonyl]amino}-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (5-methyl-3-phenyl-4-isoxazolyl)penicillin; 2,2-dimethyl-6beta-(5-methyl-3-phenyl-1,2-oxazole-4-carboxamido)penam-3alpha-carboxylic acid; 5-Methyl-3-phenyl-4-isoxazolyl-penicillin; 6beta-(5-methyl-3-phenylisoxazol-4-yl)penicillanic acid
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| Activity |
Ki = 12000000 nM
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[2] | |||
| Compound Name |
Latamoxef
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Approved | Compound Info | ||
| Synonyms |
Festamoxin; LMOX; Lamoxactam; Latamoxefum; Moxalactam; Disodium Moxalactam; Lilly 127935; Ly127935; Sid 734787; Latamoxef (INN); Latamoxef [INN:BAN]; Latamoxefum [INN-Latin]; Oxa-cephem; S-6059; (6R,7R)-7-[[3-hydroxy-2-(4-hydroxyphenyl)-3-oxopropanoyl]amino]-7-methoxy-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-oxa-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-{[carboxy(4-hydroxyphenyl)acetyl]amino}-7-(methyloxy)-3-{[(1-methyl-1H-tetrazol-5-yl)thio]methyl}-8-oxo-5-oxa-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-{[carboxy(4-hydroxyphenyl)acetyl]amino}-7-methoxy-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-8-oxo-5-oxa-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R-(6alpha,7alpha,7(S*)))-7-((Carboxy(4-hydroxyphenyl)acetyl)amino)-7-methoxy-3-(((1-methyl-1H-tetrazol-5-yl)thio)methyl)-8-oxo-5-oxa-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid; 1-Oxacephalosporin; 7b-[2-carboxy-2-(4-hydroxyphenyl)acetamido]-7a-methoxy-3-[[(1-methyl-1h-tetrazol-5-yl)thio]methyl]-1-oxa-1-dethia-3-cephem-4-carboxylic acid; 7beta-(2-Carboxy-2-(4-hydroxyphenyl)acetamido)-7alpha-methoxy-3-(((1-methyl-1H-tetrazol-5-yl)thio)methyl)-1-oxa-1-dethia-3-cephem-4-carboxylic acid
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| Activity |
Ki = 12000000 nM
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[2] | |||
| Compound Name |
Penicillin V
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Approved | Compound Info | ||
| Synonyms |
Apocillin; Apopen; Beromycin; Calcipen; Fenacilin; Fenospen; Fenossimetilpenicillina; Fenoximetilpenicilina; Fenoxymethylpenicillin; Fenoxypen; Meropenin; Oracillin; Oratren; Ospen; PNV; PVA; Phenocillin; Phenomycilline; Phenopenicillin; Phenoximethylpenicillinum; Phenoxomethylpenicillanyl; Phenoxomethylpenicillin; Phenoxymethylpenicillanyl; Phenoxymethylpenicillin; Phenoxymethylpenicilline; Phenoxymethylpenicillinum; Robicillin; Rocilin; Stabicillin; Vebecillin; Vegacillin; Acipen V; Compocillin V; Crystapen V; Distaquaine V; Eskacillian V; Eskacillin V; Fenossimetilpenicillina [DCIT]; Penicillin V [USAN]; Penicillin phenoxymethyl; Phenoxymethyl penicillin; Phenoxymethylenepenicillinic acid; Phenoxymethylpenicillinic acid; Phenoxymethylpenicillinic acid potassium salt; Acipen-v; Beromycin, Penicillin; Berromycin, Penicillin; Fenoximetilpenicilina [INN-Spanish]; Pen-Oral; Pen-V; Pen-vee; Penicillin V (USP); Penicillin, Phenoxymethyl; Phenoxymethylpenicillin (INN); Phenoxymethylpenicilline [INN-French]; Phenoxymethylpenicillinum [INN-Latin]; V-Cil; V-Cillin; V-Cylina; V-Cyline; V-Tablopen; P-Mega-Tablinen; V-Cillin (TN); (2S,5R,6R)-3,3-DIMETHYL-7-OXO-6-(2-PHENOXYACETAMIDO)-4-THIA-1-AZABICYCLO(3.2.0)HEPTANE-2-CARBOXYLIC ACID; (2S,5R,6R)-3,3-Dimethyl-7-oxo-6-(2-phenoxyacetamido)-4-thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid; (2S,5R,6R)-3,3-Dimethyl-7-oxo-6-[(phenoxyacetyl)amino]-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-3,3-dimethyl-7-oxo-6-[(2-phenoxyacetyl)amino]-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-3,3-dimethyl-7-oxo-6-{[(phenyloxy)acetyl]amino}-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; 2,2-dimethyl-6beta-[(phenoxyacetyl)amino]penam-3alpha-carbonyl; 2,2-dimethyl-6beta-[(phenoxyacetyl)amino]penam-3alpha-carboxylic acid; 3,3-Dimethyl-7-oxo-6-((phenyloxyacetyl)amino)-4-thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid; 3,3-dimethyl-6beta-[(phenoxyacetyl)amino]penam-2alpha-carboxylic acid (PIN); 6-Phenoxyacetamidopenicillanic acid
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| Activity |
Ki = 21000000 nM
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[2] | |||
| Compound Name |
Cefmetazole
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Approved | Compound Info | ||
| Synonyms |
CMZ; Cefmetazolo; Cefmetazolum; Cefmetazole Monosodium Salt; CS 1170; SKF 83088; U 72791; CS-1170; Cefmetazole [USAN:INN]; Cefmetazolo [INN-Spanish]; Cefmetazolum [INN-Latin]; U-72791A; Cefmetazole (USP/INN); (6R,7S)-7-(2-((Cyanomethyl)thio)acetamido)-7-methoxy-3-(((1-methyl-1H-tetrazol-5-yl)thio)methyl)-8-oxo-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid; (6R,7S)-7-(2-((Cyanomethyl)thio)acetamido)-7-methoxy-3-(((1-methyl-1H-tetrazol-5-yl)thiomethyl)-8-oxo-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid, sodium salt; (6R,7S)-7-({[(cyanomethyl)sulfanyl]acetyl}amino)-7-methoxy-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7S)-7-({[(cyanomethyl)thio]acetyl}amino)-7-(methyloxy)-3-{[(1-methyl-1H-tetrazol-5-yl)thio]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7S)-7-[[2-(cyanomethylsulfanyl)acetyl]amino]-7-methoxy-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 6beta-{[(cyanomethyl)sulfanyl]acetamido}-6alpha-methoxy-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}ceph-3-em-4-carboxylic acid
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| Activity |
Ki = 28000000 nM
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[2] | |||
| Compound Name |
Piperacillin
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Approved | Compound Info | ||
| Synonyms |
PIPC; Peperacillin; Peracin; Pipercillin; Pipracil; Pipril; PIPERACILLIN SODIUM; Piperacillin Monosodium Salt; Piperacillin anhydrous; Cl-227193; Peracin (TN); Piperacillin (INN); Piperacillin (anhydrous); Pipracil, Piper; T-1220; Zobactin (TN); (2S,5R,6R)-6-[[(2R)-2-[(4-ethyl-2,3-dioxopiperazine-1-carbonyl)amino]-2-phenylacetyl]amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-{[(2R)-2-{[(4-ethyl-2,3-dioxopiperazin-1-yl)carbonyl]amino}-2-phenylacetyl]amino}-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S-(2alpha,5alpha,6beta(S*)))-6-(((((4-Ethyl-2,3-dioxopiperazin-1-yl)carbonyl)amino)phenylacetyl)amino)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid; 4-ethyl-2,3-dioxopiperazine carbonyl ampicillin; 6-(D-(-)-alpha-(4-Ethyl-2,3-dioxo-1-piperazinecarboxamido)phenylacetamido)penicillanicacid; 6beta-{(2R)-2-[(4-ethyl-2,3-dioxopiperazin-1-yl)carboxamido]-2-phenylacetamido}-2,2-dimethylpenam-3alpha-carboxylic acid
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| Activity |
Ki > 30000000 nM
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[2] | |||
| Compound Name |
Ceftriaxone
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Approved | Compound Info | ||
| Synonyms |
Biotrakson; CTRX; Cefatriaxone; Ceftriaxon; Ceftriaxona; Ceftriaxonum; Ceftriazone; Longacef; Longaceph; Rocefin; Rocephin; Rocephine; CEFTRIAXONE SODIUM; Ceftriaxone intravenous; Ro 139904; Ceftriaxona [INN-Spanish]; Ceftriaxone (INN); Ceftriaxone (TN); Ceftriaxone [USAN:JAN]; Ceftriaxone, Disodium Salt; Ceftriaxonum [INN-Latin]; DRG-0071; Ro13-9904; Rocephin (TN); Ceftriaxone, Disodium Salt, Hemiheptahydrate; Ro-13-9904; (6R,7R)-7-(2-(2-Amino-4-thiazolyl)glyoxylamido)-8-oxo-3-(((1,2,5,6-tetrahydro-2-methyl-5,6-dioxo-as-triazin-3-yl)thio)methyl)-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid, 7(sup 2)-(Z)-(O-methyloxime), sesquaterhydrate; (6R,7R)-7-({(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-[(methyloxy)imino]acetyl}amino)-3-{[(6-hydroxy-2-methyl-5-oxo-2,5-dihydro-1,2,4-triazin-3-yl)thio]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-methoxyiminoacetyl]amino]-3-[(2-methyl-5,6-dioxo-1H-1,2,4-triazin-3-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-{[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-(methoxyimino)acetyl]amino}-3-{[(2-methyl-5,6-dioxo-1,2,5,6-tetrahydro-1,2,4-triazin-3-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 7beta-{[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-(methoxyimino)acetyl]amino}-3-{[(2-methyl-5,6-dioxo-1,2,5,6-tetrahydro-1,2,4-triazin-3-yl)sulfanyl]methyl}-3,4-didehydrocepham-4-carboxylic acid
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| Activity |
Ki > 30000000 nM
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[2] | |||
| Compound Name |
Cefazolin
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Approved | Compound Info | ||
| Synonyms |
CEZ; Cefamezin; Cefamezine; Cefazolina; Cefazoline; Cefazolinum; Cephamezine; Cephazolidin; Cephazolin; Cephazoline; Elzogram; Cephazolin Sodium; Ancef (TN); Cefacidal (TN); Cefamezin (TN); Cefazolin (USP); Cefazolin [USAN:INN]; Cefazolin(usp); Cefazolina [INN-Spanish]; Cefazoline [INN-French]; Cefazolinum [INN-Latin]; Cefrina (TN); Elzogram (TN); Faxilen (TN); Gramaxin (TN); Kefazol (TN); Kefol (TN); Kefzol (TN); Kefzolan (TN); Kezolin (TN); Novaporin (TN); Zolicef (TN); (6R, 7R)-3-[[(5-Methyl-1,3,4-thiadiazol-2-yl)thio]methyl]-8-oxo-7-[[1H-tetrazol-1-yl)acetyl]amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-3-(((5-Methyl-1,3,4-thiadiazol-2-yl)thio)methyl)-8-oxo-7-(2-(1H-tetrazol-1-yl)acetamido)-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid; (6R,7R)-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-7-[[2-(tetrazol-1-yl)acetyl]amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-3-{[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-8-oxo-7-[(1H-tetrazol-1-ylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-3-{[(5-methyl-1,3,4-thiadiazol-2-yl)thio]methyl}-8-oxo-7-[(1H-tetrazol-1-ylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R-trans)-3-(((5-Methyl-1,3,4-thiadiazol-2-yl)thio)methyl)-8-oxo-7-(((1H-tetrazol-1-yl)acetyl)-amino)-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid; 3-{[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-7beta-[(1H-tetrazol-1-ylacetyl)amino]-3,4-didehydrocepham-4-carboxylic acid; 7-(1-(1H-)-Tetrazolylacetamido)-3-(2-(5-methyl-1,3,4-thiadiazolyl)thiomethyl)delta3-cephem-4-carboxylic acid
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| Activity |
Ki > 30000000 nM
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[2] | |||
| Compound Name |
Cefepime
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Approved | Compound Info | ||
| Synonyms |
Axepim; CFPM; Cefepima; Cefepimum; Cepimax; Cepimex; Maxcef; Maxipime; Cefepima [Spanish]; Cefepimum [Latin]; BMY 28142; Axepim (TN); BMY-28142; Cefepime [USAN:INN]; Cepimax (TN); Cepimex (TN); Maxcef (TN); Maxipime (TN); Cefepime (USAN/INN); (6R,7R)-7-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-methoxyiminoacetyl]amino]-3-[(1-methylpyrrolidin-1-ium-1-yl)methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate; (6R,7R)-7-{[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-(methoxyimino)acetyl]amino}-3-[(1-methylpyrrolidinium-1-yl)methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate; 1-(((6R,7R)-7-(2-(2-Amino-4-thiazolyl)glyoxylamido)-2-carboxy-8-oxo-5-thia-1-azabicyclo(4.2.0)oct-2-en-3-yl)methyl)-1-methylpyrrolidinium hydroxide, inner salt, 7(sup 2)-(Z)-(O-methyloxime); 7beta-[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-(methoxyimino)acetamido]-3-[(1-methylpyrrolidinium-1-yl)methyl]-3,4-didehydrocepham-4-carboxylate
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| Activity |
Ki > 30000000 nM
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[2] | |||
| Compound Name |
Cefpodoxime
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Approved | Compound Info | ||
| Synonyms |
CPDX; Cefpodoxima; Cefpodoximum; Epoxim; Cefpodoxim acid; Cefpodoxima [Spanish]; Cefpodoximum [Latin]; RU 51807; Cefpodoxime (INN); Cefpodoxime [INN:BAN]; Epoxim (TN); Vantin (TN); (6R,7R)-7-({(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-[(methyloxy)imino]acetyl}amino)-3-[(methyloxy)methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-[[(2E)-2-(2-amino-1,3-thiazol-4-yl)-2-methoxyiminoacetyl]amino]-3-(methoxymethyl)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-methoxyiminoacetyl]amino]-3-(methoxymethyl)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 7-{[(2-amino-1,3-thiazol-4-yl)(methoxyimino)acetyl]amino}-3-(methoxymethyl)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
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| Activity |
Ki > 30000000 nM
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[2] | |||
| Compound Name |
Levodopa
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Approved | Compound Info | ||
| Synonyms |
Levodopa (optimized formulation, Parkinson's disease); More effective levodopa (Parkinson's disease), Orion; Levodopa (optimized formulation, Parkinson's disease), Orion
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| Activity |
IC50 = 141200000 nM
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[13] | |||
| Compound Name |
Methyldopa
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Approved | Compound Info | ||
| Synonyms |
AMD; Aldometil; Aldomin; Alphamethyldopa; Baypresol; Becanta; Dopamet; Dopamethyperpax; Dopatec; Dopegit; Dopegyt; Dopergit; Grospisk; Hyperpax; Hypolag; Medomet; Medopa; Medopal; Medopren; Methoplain; Methyldopum; Metildopa; Novomedopa; Presinol; Presolisin; Sedometil; Sembrina; Alpha medopa; Methyl dopa; Methyldopa anhydrous; Aldoril D30; Aldoril D50; Bayer 1440 L; LT00847269; MK 351; Aldomet (TN); Aldoril (TN); Alpha-Methyl dopa; Alpha-Methyldihydroxyphenylalanine; Alpha-Methyldopa; Apo-Methyldopa; Dopamet (TN); Dopegyt (TN); L-Methyl Dopa; L-Methyldopa; METHYL DOPA (SEE ALSO METHYL DOPA SESQUIHYDRATE); MK-351; Methyldopa (INN); Methyldopa (anhydrous); Methyldopum [INN-Latin]; Metildopa [INN-Spanish]; Mk. b51; Nr.C 2294; Nu-Medopa; Alpha-Methyldopa (VAN); L-alpha-Methyl DOPA; L-alpha-Methyldopa; Methyl-L-dopa; Aldoril, Dopamet, Dopegyt, Methyldopa; L-(alpha-Md); Methyldopa (L,-); Alpha-Methyl-L-3,4-dihydroxyphenylalanine; L-alpha-Methyl-3,4-dihydroxyphenylalanine; L-3-(3,4-Dihydroxyphenyl)-2-methylalanine; Levo-3-(3,4-Dihydroxyphenyl)-2-methylalanine; Alpha-Methyl-beta-(3,4-dihydroxyphenyl)-L-alanine; L(-)-beta-(3,4-Dihydroxyphenyl)-alpha-methylalanine; L-2-Amino-2-methyl-3-(3,4-dihydroxyphenyl)propionic acid; L-(-)-3-(3,4-Dihydroxyphenyl)-2-methylalanine; L-(-)-alpha-Methyl-beta-(3,4-dihydroxyphenyl)alanine; (-)-3-(3,4-Dihydroxyphenyl)-2-Methyl-L-Alanine Sesqui-Hydrate; (2S)-2-amino-3-(3,4-dihydroxyphenyl)-2-methylpropanoic acid; (S)-(-)-alpha-Methyldopa; 3-(3,4-DIHYDROXYPHENYL)-2-METHYL-L-ALANINE; 3-Hydroxy-.alpha.-methyl-L-tyrosine; 3-Hydroxy-alpha-methyl-L-tyrosine
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| Activity |
IC50 = 151600000 nM
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[13] | |||
| Compound Name |
Benzylpenicillin
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Phase 3 | Compound Info | ||
| Synonyms |
penicillin g; Benzylpenicillinic acid; Free penicillin II; Pencillin G; 61-33-6; Benzylpenicillin G; Bencilpenicilina; Benzylpenicillinum; Benzyl penicillin; Free penicillin G; Dropcillin; Pharmacillin; Gelacillin; Liquacillin; Benzopenicillin; Cilopen; Pradupen; Benzylpenicilline; Specilline G; Cilloral; Cosmopen; Ursopen; Galofak; Free benzylpenicillin; Compocillin G; Phenylacetamidopenicillanic acid; 6-(2-Phenylacetamido)penicillanic acid; Pfizerpen; Benzyl-6-aminopenicillinic acid
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| Activity |
Ki > 30000000 nM
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[2] | |||
| Compound Name |
Cephaloridine
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Withdrawn from market | Compound Info | ||
| Synonyms |
cephaloridine; cefaloridine; Cefaloridin; Cephaloridin; Cephaloridinum; Cepaloridin; Cefalorizin; Cephalomycine; Cefaloridinum; Cepalorin; Cefaloridina; Loridine; Ceflorin; 50-59-9; Kefloridin; Glaxoridin; Ceporin; Vioviantine; Intrasporin; Sefacin; Keflordin; Deflorin; Cilifor; Ceporan; Sasperin; Faredina; Ceporine; Keflodin; Verolgin; Lloncefal; Kefspor; Ampligram; Betaine cephaloridine; CHEBI:3537; UNII-LVZ1VC61HB; Cefaloridinum [INN-Latin]; Cefaloridina [INN-Spanish]; N-(7-(2'-Thienylacetamidoceph-3-ylmethyl))-pyridinium-2-carboxylate; SCH
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| Activity |
Ki > 30000000 nM
|
[14] | |||
| Compound Name |
N-(N-Glycyl-L-leucyl)glycine
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Investigative | Compound Info | ||
| Synonyms |
gly-leu-gly; H-GLY-LEU-GLY-OH; Glycyl-L-leucinyl-glycine; GLYCYL-L-LEUCYL-GLYCINE; CHEMBL209341; 2-[[(2S)-2-[(2-aminoacetyl)amino]-4-methylpentanoyl]amino]acetic acid; Glycine, glycyl-L-leucyl-; Glycine, N-(N-glycyl-L-leucyl)-; Glycylleucylglycin; EINECS 219-925-8; Glycyl-leucyl-glycine; Gly-L-Leu-Gly-OH; CTK7E1874; ZINC2384921; BDBM50188482; MFCD00037776; ((2-[(Aminoacetyl)amino]-4-methylpentanoyl)amino)acetic acid #
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||||
| Activity |
EC50 = 210000 nM
|
[1] | |||
| Compound Name |
H-Val-Val-Val-OH
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Investigative | Compound Info | ||
| Synonyms |
Val-Val-Val; CHEMBL380174; valyl-valyl-valin; valyl-valyl-valine; l-valyl-l-valyl-l-valine; SCHEMBL7344595; ZINC2561148; BDBM50188506; MFCD00238287; CCG-208120; BS-16358; BRD-K04431258-001-01-5; Q27216090
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||||
| Activity |
EC50 = 210000 nM
|
[1] | |||
| Compound Name |
2-[[(2S)-2-Amino-4-hydroxy-5-[(5-methyl-2,4-dioxopyrimidin-1-yl)methoxy]-5-oxopentanoyl]-methylamino]acetic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2074601; BDBM50420184
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| Activity |
Ki = 210000 nM
|
[15] | |||
| Compound Name |
Glycine, L-phenylalanyl-N-methyl-
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Investigative | Compound Info | ||
| Synonyms |
phenylalanylsarcosine; CHEMBL2371159; SCHEMBL11357126
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||||
| Activity |
Ki = 210000 nM
|
[4] | |||
| Compound Name |
[(2R,3S,4R)-5-(2-Bromo-5,6-dichlorobenzimidazol-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2S)-2-amino-3-phenylpropanoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL608238; BDBM50370612
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||||
| Activity |
IC50 = 218000 nM
|
[8] | |||
| Compound Name |
Ac-Phe-di-iodo-Tyr
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL378713; BDBM50188509
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||||
| Activity |
IC50 = 230000 nM
|
[1] | |||
| Compound Name |
H-Trp-Gly-Tyr-OH
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Investigative | Compound Info | ||
| Synonyms |
Trp-Gly-Tyr; CHEMBL364928; Tryptophanyl-glycyl-tyrosine; CTK0E8540; L-Tryptophanyl-glycyl-L-tyrosine; DTXSID40436268; ZINC2561119; BDBM50169115; MFCD00238200; L-Tyrosine, N-(N-L-tryptophylglycyl)-
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||||
| Activity |
Ki = 240000 nM
|
[2] | |||
| Compound Name |
Tyr-Gly
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Investigative | Compound Info | ||
| Synonyms |
H-TYR-GLY-OH; Tyrosyl-Glycine; L-Tyrosylglycine; Glycine, L-tyrosyl-; L-TYROSYL-GLYCINE; (S)-2-(2-Amino-3-(4-hydroxyphenyl)propanamido)acetic acid; UNII-QJH0S8U69Z; QJH0S8U69Z; CHEMBL89956; MFCD00037779; L-Tyr-Gly; Tyr-Gly-OH; L-Tyr-Gly-OH; TYR-GLY CRYSTALLINE; SCHEMBL4407092; CTK2F6911; ZINC2575475; 7253AH; BDBM50188519; KM1087; Human beta-endorphin(1-2) component of imreg-1; Q27145056; UNII-VMX0XQ62KT component HPYDSVWYXXKHRD-VIFPVBQESA-N; [(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-acetic acid
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||||
| Activity |
EC50 = 240000 nM
|
[1] | |||
| Compound Name |
Glycine, L-alanyl-N-methyl-
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Investigative | Compound Info | ||
| Synonyms |
N-(L-Alanyl)-N-methylglycine; CHEMBL2371157; SCHEMBL10908256; 2-[[(2S)-2-aminopropanoyl]-methylamino]acetic acid
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||||
| Activity |
Ki = 250000 nM
|
[4] | |||
| Compound Name |
Tyr-Pro-Ile
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Investigative | Compound Info | ||
| Synonyms |
L-Isoleucine, N-(1-L-tyrosyl-L-prolyl)-; Tyrosyl-prolyl-isoleucine; CHEMBL2371839; CTK0C0420; L-Tyrosyl-L-prolyl-L-isoleucine
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||||
| Activity |
Ki = 250000 nM
|
[2] | |||
| Compound Name |
Pro-leu
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Investigative | Compound Info | ||
| Synonyms |
H-Pro-Leu-OH; L-prolyl-L-leucine; L-Leucine, L-prolyl-; CHEMBL293494; (S)-4-Methyl-2-((S)-pyrrolidine-2-carboxamido)pentanoic acid; Prolyl-leucine; L-Pro-L-Leu; L-Pro-L-Leu-OH; SCHEMBL6373762; ZINC4040320; BDBM50188501; MFCD00037871; STL527240; AKOS010421057; MCULE-4010644832; Q27144902; 4-Methyl-2-[(pyrrolidine-2-carbonyl)-amino]-pentanoic acid; (S)-4-Methyl-2-[((S)-pyrrolidine-2-carbonyl)-amino]-pentanoic acid
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||||
| Activity |
EC50 = 250000 nM
|
[1] | |||
| Compound Name |
Trp-Trp
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Investigative | Compound Info | ||
| Synonyms |
H-TRP-TRP-OH; l-tryptophyl-l-tryptophan; N-L-Tryptophyl-L-tryptophan; L-Tryptophan, N-L-tryptophyl-; CHEMBL286852; Tryptophyl-Tryptophan; L-Tryptophan, L-tryptophyl-; L-Trp-L-Trp; tryptophanyl-tryptophan; L-Trp-L-Trp-OH; H-L-Trp-L-Trp-OH; L-Tryptophanyl-L-tryptophan; SCHEMBL5583839; CTK1A3898; ZINC1557161; BDBM50188479; MFCD00037959; Q27144986; 2-[2-Amino-3-(1H-indol-3-yl)-propionylamino]-3-(1H-indol-3-yl)-propionic acid
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||||
| Activity |
IC50 = 250000 nM
|
[1] | |||
| Compound Name |
Glutamylalanine
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Investigative | Compound Info | ||
| Synonyms |
Glu-ala; H-GLU-ALA-OH; glutamyl-alanine; n-l-alpha-glutamyl-L-alanine; alpha-glutamylalanine; L-Glutamyl-L-alanine; CHEMBL90074; a-Glutamylalanine; alpha-Glu-Ala; L-alpha-Glu-L-Ala; L-Glu-L-Ala; a-L-Glutamyl-L-alanine; L-Alanine,l-a-glutamyl-; L-alpha-glutamyl-L-alanine; alpha-L-Glutamyl-L-alanine; SCHEMBL751142; L-alpha-Glutamyl-L-amino acid; ZINC1576200; BDBM50169155; MFCD00037233; Q27144175; (S)-4-Amino-4-((S)-1-carboxy-ethylcarbamoyl)-butyric acid; (4S)-4-amino-5-[[(1S)-1-carboxyethyl]amino]-5-oxopentanoic acid
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||||
| Activity |
Ki = 250000 nM
|
[2] | |||
| Compound Name |
(3S)-3-Amino-4-[[(2R,3S,4R)-5-(2-bromo-5,6-dichlorobenzimidazol-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy]-4-oxobutanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL610518; BDBM50370611
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||||
| Activity |
IC50 = 260000 nM
|
[8] | |||
| Compound Name |
Tryptophylglycine
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Investigative | Compound Info | ||
| Synonyms |
Trp-gly; (S)-2-(2-Amino-3-(1H-indol-3-yl)propanamido)acetic acid; H-TRP-GLY-OH; l-tryptophylglycine; Glycine, L-tryptophyl-; UNII-GLE75A3004; N-L-Tryptophylglycine; CHEMBL327588; Tryptophyl-Glycine; GLE75A3004; Glycine, N-L-tryptophyl-; Tryptophanylglycine; Tryptophylglycine,l; Tryptophylglycine, L-; 2-[[(2S)-2-amino-3-(1H-indol-3-yl)propanoyl]amino]acetic acid; Tryptophanyl-glycine; L-Trp-Gly; Trp-Gly-OH; NSC 97945; L-Tryptophanyl-glycine; SCHEMBL8699875; CTK2H8443; TNP00242; ZINC2384992; 1433AC; A0H155; BDBM50188498; MFCD00037967; AKOS010405232; NCGC00017311-01; DS-14684; Q27144980; [(S)-2-Amino-3-(1H-indol-3-yl)-propionylamino]-acetic acid
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||||
| Activity |
EC50 = 260000 nM
|
[1] | |||
| Compound Name |
Glycine, N-L-arginyl-
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Investigative | Compound Info | ||
| Synonyms |
Arg-Gly; Glycine, L-arginyl-; L-Arginyl glycine; CHEMBL382777; 2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]acetic acid; arginylglycine; N-Arginylglycine; L-Arginyl-glycine; N-L-Arginylglycine; SCHEMBL2117673; CTK1A3739; DTXSID10178885; ZINC2545093; BDBM50188522; AKOS015910638; Glycine,l-arginyl-,dihydrochloride(9ci); (S)-2-(2-Amino-5-guanidinopentanamido)acetic acid; N-[N5-[Amino(iminio)methyl]-L-ornithyl]glycine anion
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||||
| Activity |
EC50 = 270000 nM
|
[1] | |||
| Compound Name |
Isoleucyl-prolyl-proline
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Investigative | Compound Info | ||
| Synonyms |
H-ILE-PRO-PRO-OH; Ile-Pro-Pro; l-isoleucyl-l-prolyl-l-proline; CHEMBL190994; isoleucine-proline-proline; L-Proline, L-isoleucyl-L-prolyl-; IPP-OH; L-Ile-L-Pro-L-Pro-OH; SCHEMBL1646849; L-Proline,L-isoleucyl-L-prolyl-; BDBM50169149; ZINC13646353; HY-114424; CS-0085280
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||||
| Activity |
Ki = 280000 nM
|
[2] | |||
| Compound Name |
2-[[(2S)-2-Amino-5-[2-[(2-amino-6-oxo-1H-purin-9-yl)methoxy]ethoxy]-5-oxopentanoyl]-methylamino]acetic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1823468
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||||
| Activity |
Ki = 280000 nM
|
[15] | |||
| Compound Name |
Histidylglycine
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Investigative | Compound Info | ||
| Synonyms |
His-Gly; L-His-Gly; (S)-2-(2-Amino-3-(1H-imidazol-4-yl)propanamido)acetic acid; l-histidylglycine; H-HIS-GLY-OH; CHEMBL90452; Histidinyl-Glycine; Glycine, L-histidyl-; histidyl-glycine; L-Histidyl-glycine; His-Gly-OH; L-His-Gly-OH; Glycine, N-L-histidyl-; SCHEMBL483855; CTK1A2385; ZINC2384936; 4404AH; BDBM50188486; MFCD00037863; AKOS016014021; AS-56395; Q27144253; 2-[(2S)-2-amino-3-(1H-imidazol-5-yl)propanamido]acetic acid; [(S)-2-Amino-3-(3H-imidazol-4-yl)-propionylamino]-acetic acid
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||||
| Activity |
EC50 = 280000 nM
|
[1] | |||
| Compound Name |
Glycyl-leucyl-phenylalanine
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Investigative | Compound Info | ||
| Synonyms |
H-Gly-Leu-Phe-OH; GLY-LEU-PHE; CHEMBL209670; L-Gly-L-leu-L-phe; Gly-L-Leu-L-Phe-OH; SCHEMBL4281374; Glycyl-L-leucyl-L-phenylalanine; DTXSID60908255; ZINC2522593; BDBM50188525; MFCD00057838; L-Phenylalanine, N-(N-glycyl-L-leucyl)-
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||||
| Activity |
EC50 = 280000 nM
|
[1] | |||
| Compound Name |
[(2R,3S,4R)-5-(2-Bromo-5,6-dichlorobenzimidazol-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2R)-2-amino-3-phenylpropanoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL609379; BDBM50370604
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||||
| Activity |
IC50 = 282000 nM
|
[8] | |||
| Compound Name |
2-Amino-N-(3-phenylphenyl)propanamide
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Investigative | Compound Info | ||
| Synonyms |
SCHEMBL1750966; CHEMBL1161365
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||||
| Activity |
Ki = 290000 nM
|
[4] | |||
| Compound Name |
1-(2-Ammoniopropanethioyl)pyrrolidine-2-carboxylate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL347510; BDBM50137011
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||||
| Activity |
Ki = 300000 nM
|
[16] | |||
| Compound Name |
[(2R,3S,4R)-5-(2-Bromo-5,6-dichlorobenzimidazol-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2S)-2-amino-3-(4-methoxyphenyl)propanoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL607680; BDBM50370606
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||||
| Activity |
IC50 = 300000 nM
|
[8] | |||
| Compound Name |
H-Leu-arg-pro-OH
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Investigative | Compound Info | ||
| Synonyms |
Leucylarginylproline; CHEMBL188695; SCHEMBL9616909; CTK6A4188; HY-P0143; ZINC4899610; BDBM50169168; MFCD00190940; CS-6486; Z-L-LEUCYL-L-ARGINYL-L-PROLINE
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||||
| Activity |
Ki = 300000 nM
|
[2] | |||
| Compound Name |
Asp-Val
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Investigative | Compound Info | ||
| Synonyms |
H-Asp-Val-OH; Aspartyl-Valine; l-aspartyl-l-valine; CHEMBL441685; L-Valine, L-alpha-aspartyl-; alpha-aspartylvaline; L-alpha-Asp-L-Val; L-Asp-L-Val; L-alpha-aspartyl-L-valine; N-L-alpha-Aspartyl-L-valine; SCHEMBL3785072; ZINC2384839; BDBM50188511; MFCD00037285; Q27144150; (2S)-2-[[(2S)-2-amino-3-carboxypropanoyl]amino]-3-methylbutanoic acid; (S)-3-amino-4-((S)-1-carboxy-2-methylpropylamino)-4-oxobutanoic acid
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||||
| Activity |
IC50 = 310000 nM
|
[1] | |||
| Compound Name |
Glu-lys
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Investigative | Compound Info | ||
| Synonyms |
H-Glu-Lys-OH; glutamyl-lysine; L-alpha-glutamyl-L-Lysine; CHEMBL190361; Glutamyllysine; L-Glu-L-Lys; L-Glutamyl-L-Lysine; N2-a-glutamyl-lysine; L-Glu-L-Lys-OH; N2-L-a-Glutamyllysine; N2-L-a-glutamyl-Lysine; N2-alpha-glutamyl-lysine; N2-L-alpha-Glutamyllysine; N2-L-alpha-glutamyl-Lysine; L-Lysine, L-alpha-glutamyl-; SCHEMBL170727; ZINC2516165; BDBM50169173; MFCD00056129; Q27140603; (S)-6-Amino-2-((S)-2-amino-4-carboxy-butyrylamino)-hexanoic acid; (2S)-6-amino-2-[[(2S)-2-amino-4-carboxybutanoyl]amino]hexanoic acid
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||||
| Activity |
EC50 = 310000 nM
|
[1] | |||
| Compound Name |
3-[(2-Ammoniopropanoyl)amino]benzoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL152123
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||||
| Activity |
Ki = 310000 nM
|
[4] | |||
| Compound Name |
Alanine glutamate
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Investigative | Compound Info | ||
| Synonyms |
H-Ala-Glu-OH; l-alanyl-l-glutamic acid; Ala-Glu-OH; UNII-8D40GXI4MA; alanylglutamic acid; alanyl-glutamic acid; L-Alanyl-L-glutamate; 8D40GXI4MA; Alanylglutamate; ALA-GLU; L-Ala-L-Glu; (2S)-2-[[(2S)-2-aminopropanoyl]amino]pentanedioic acid; (2S)-2-{[(2S)-2-Aminopropanoyl]amino}pentanedioic acid; AlaGlu; Glutamic acid, alanyl-; L-Alanyl-L-glutaminsaeure; 2-[(2-ammoniopropanoyl)amino]pentanedioate; SCHEMBL2490631; L-Glutamic acid, N-L-alanyl-; CHEMBL2074938; CTK3C9161; DTXSID70927376; ZINC2242980; 7043AH; MFCD00025556; AKOS010407205; C20958; K-4133; N-(2-Amino-1-hydroxypropylidene)glutamic acid; (S)-2-((S)-2-aminopropanamido)pentanedioic acid; L-Glutamic acid, compd., with L-alanine (1:1); Q27131168
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||||
| Activity |
Ki = 320000 nM
|
[4] | |||
| Compound Name |
Lys-gly
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Investigative | Compound Info | ||
| Synonyms |
lysylglycine; CHEMBL91561; L-lysylglycine; L-Lysyl-glycine; L-Lys-Gly; Lys-Gly-OH; Glycine, L-lysyl-; Glycine, N-L-lysyl-; SCHEMBL345265; CTK2G8826; DTXSID80427433; ZINC2579078; BDBM50188483; ((S)-2,6-Diamino-hexanoylamino)-acetic acid; Q27141913
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||||
| Activity |
EC50 = 320000 nM
|
[1] | |||
| Compound Name |
Aspartylalanine
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Investigative | Compound Info | ||
| Synonyms |
Asp-Ala; alpha-Asp-ala; alpha-Aspartylalanine; Aspartyl-Alanine; CHEMBL17503; H-Asp-Ala-OH; L-Aspartyl-L-Alanine; Asp-Ala-OH; L-Asp-L-Ala; L-Alanine,l-a-aspartyl-; L-alpha-aspartyl-L-alanine; N-L-alpha-Aspartyl-L-alanine; SCHEMBL3341838; DTXSID10928569; ZINC2123927; BDBM50169166; MFCD00037231; MCULE-9587398290; 3-Amino-N-((S)-1-carboxy-ethyl)-succinamic acid; Q27144144; (S)-3-Amino-N-((S)-1-carboxy-ethyl)-succinamic acid; 3-Amino-4-[(1-carboxyethyl)imino]-4-hydroxybutanoic acid; (3S)-3-amino-4-[[(1S)-1-carboxyethyl]amino]-4-oxobutanoic acid; (S)-3-Amino-4-(((S)-1-carboxyethyl)amino)-4-oxobutanoic acid
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||||
| Activity |
Ki = 320000 nM
|
[2] | |||
| Compound Name |
Glycyltryptophan
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Investigative | Compound Info | ||
| Synonyms |
Glycyl-L-tryptophan; H-Gly-Trp-OH; GLY-TRP; alpha-Glycyltryptophan; N-Glycyltryptophan; UNII-35BKX0QF16; Clycyl-L-tryptophan; Gly-Trp-OH; L-Tryptophan, glycyl-; 35BKX0QF16; CHEMBL299759; (2S)-2-[(2-aminoacetyl)amino]-3-(1H-indol-3-yl)propanoic acid; l-Glycyltryptophan; EINECS 219-235-7; Gly-L-Trp; Gly-L-Trp-OH; NSC 118371; N-Glycyl-l-tryptophan; Glycyl-L-tryptophanHydrate; Nalpha-glycyl-L-tryptophan; 2-(2-Amino-acetylamino)-3-(1H-indol-3-yl)-propionic acid; Tryptophan, N-glycyl-, l-; N.alpha.-Glycyl-l-tryptophan; SCHEMBL1407979; CTK1A2113; L-Tryptophan, N-glycyl- (9CI); N-(Aminoacetyl)tryptophan, (L)-; KS-000016HA; ZINC1708201; 7025AH; BDBM50188499; Tryptophan, N-(aminomethylcarbonyl)-; AS-56406; G0144; Q27144244; (S)-2-(2-aminoacetamido)-3-(1H-indol-3-yl)propanoic acid; (S)-2-(2-Amino-acetylamino)-3-(1H-indol-3-yl)-propionic acid; 2-((S)-2-Amino-acetylamino)-3-(1H-indol-3-yl)-propionic acid
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||||
| Activity |
EC50 = 330000 nM
|
[1] | |||
| Compound Name |
Ala-His
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Investigative | Compound Info | ||
| Synonyms |
H-Ala-His-OH; L-alanyl-L-histidine; N-L-Alanyl-L-histidine; alanyl-histidine; CHEMBL1221620; (2S)-2-[[(2S)-2-aminopropanoyl]amino]-3-(1H-imidazol-5-yl)propanoic acid; L-Histidine, L-alanyl-; Ala-His-OH; L-Ala-L-His; SCHEMBL308989; CTK1C5043; DTXSID201016440; ZINC5115824; BDBM50348857; MFCD00037853; AKOS010421081; AKOS015893950; W-106836; Q27144099; (S)-2-((S)-2-aminopropanamido)-3-(1H-imidazol-4-yl)propanoic acid; (S)-2-((S)-2-Aminopropanamido)-3-(1H-imidazol-5-yl)propanoic acid
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||||
| Activity |
Ki = 330000 nM
|
[4] | |||
| Compound Name |
(S)-3-((S)-2,6-Diamino-hexanoylamino)-4-oxo-butyric acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL188696; BDBM50169142
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||||
| Activity |
Ki = 330000 nM
|
[2] | |||
| Compound Name |
2-Amino-N-(4-chlorophenyl)propanamide
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Investigative | Compound Info | ||
| Synonyms |
N-(4-chlorophenyl)alaninamide; 2-Amino-N-(4-chloro-phenyl)-propionamide; CHEMBL1161355; CTK6A3149; STK185380; AKOS000167831; AKOS016049871; MCULE-5775564877; EN300-39560; 2-amino-N-(4-chloro-phenyl)-propionamide, AldrichCPR
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||||
| Activity |
Ki = 330000 nM
|
[4] | |||
| Compound Name |
L-Lysyl-L-alanine
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Investigative | Compound Info | ||
| Synonyms |
lysyl-alanine; LYS-ALA; H-Lys-Ala-OH; CHEMBL93178; L-Lys-L-Ala-OH; L-Alanine, L-lysyl-; Epitope ID:143649; SCHEMBL1641741; CTK0H2100; DTXSID20426662; ZINC2390920; BDBM50169138; (S)-2-((S)-2,6-Diaminohexanamido)propanoic acid; Q27131473; (S)-2-((S)-2,6-Diamino-hexanoylamino)-propionic acid; (2S)-2-[[(2S)-2,6-diaminohexanoyl]amino]propanoic acid
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| Activity |
Ki = 340000 nM
|
[2] | |||
| Compound Name |
Ceftibuten
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Investigative | Compound Info | ||
| Synonyms |
Cedax; Ceftibuteno; Ceftibutenum; Ceftibutene; Sch 39720; cis-ceftibuten; UNII-IW71N46B4Y; Cephem; cis-Ceftibutin; Sch-39720; Ceftibuten hydrate; 7432-S; Antibiotic 7432S; Cephalosporin 7432-S; IW71N46B4Y; 97519-39-6 (free); Isocef; MFCD00864918; Ceftibutene [INN-French]; Ceftibutenum [INN-Latin]; Ceftibuteno [INN-Spanish]; Ceftibuten [USAN:INN:BAN]; S 7432; Ceprifran; Ceftem; Keimax; NCGC00095137-01; Ceftibuten, 95%; Ceftibuten (USAN/INN); Spectrum5_001558; CHEMBL1605; DSSTox_CID_25925; DSSTox_RID_81227; DSSTox_GSID_45925; SCHEMBL37054; ACHN383; BSPBio_002733; SPECTRUM1505207; ACHN-383; DTXSID4045925; HMS1922L17; HMS2093K18; HMS3715P10; Pharmakon1600-01505207; HY-B0698; ZINC3871967; Tox21_111446; BDBM50370586; CC0255; CCG-39440; NSC758925; AKOS005146205; AKOS015854930; DB01415; NSC-758925; NCGC00178501-01; NCGC00178501-04; SC-27736; SBI-0206740.P001; C08117; D00922; AB01563048_01; 519C396; Ceftibuten, Antibiotic for Culture Media Use Only; Q419521; SR-05000001989; SR-05000001989-1
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| Activity |
Ki = 340000 nM
|
[2] | |||
| Compound Name |
2-Amino-N-(4-methylphenyl)propanamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1161352; SCHEMBL10975281; AKOS000189524
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| Activity |
Ki = 340000 nM
|
[4] | |||
| Compound Name |
[(2R,3S,4R)-5-(2-Bromo-5,6-dichlorobenzimidazol-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2R)-2-amino-3-methylbutanoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL609093; BDBM50370607
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| Activity |
IC50 = 342000 nM
|
[8] | |||
| Compound Name |
Tyr-gly-gly
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Investigative | Compound Info | ||
| Synonyms |
tyrosyl-glycyl-glycine; l-tyrosylglycylglycine; Tyrosylglycylglycine; L-Tyr-Gly-Gly-OH; Glycine, N-(N-L-tyrosylglycyl)-; UNII-DS6B3J0V03; CHEMBL191422; DS6B3J0V03; H-TYR-GLY-GLY-OH; (S)-2-(2-(2-Amino-3-(4-hydroxyphenyl)propanamido)acetamido)acetic acid; Tgg tripeptide; Ygg tripeptide; L-Tyr-Gly-Gly; L-Tyrosyl-glycyl-glycine; IMREG-1; SCHEMBL4405069; ZINC2575477; 1055AB; BDBM50169197; MFCD00037786; TYR-GLY-GLY CRYSTALLINE 99%; AKOS010407461; Q27145057; UNII-VMX0XQ62KT component HIINQLBHPIQYHN-JTQLQIEISA-N; {2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-acetylamino}-acetic acid
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| Activity |
Ki = 350000 nM
|
[2] | |||
| Compound Name |
Glycyl-L-aspartic acid
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Investigative | Compound Info | ||
| Synonyms |
GLY-ASP; (S)-2-(2-Aminoacetamido)succinic acid; H-Gly-Asp-OH; Aspartic acid, glycyl-; Glycylaspartic acid; N-Glycyl-L-aspartic acid; CHEMBL91392; L-Aspartic acid, N-glycyl-; N-(Aminoacetyl)aspartic acid #; (2S)-2-(2-aminoacetamido)butanedioic acid; Gly-Asp-OH; Gly-L-Asp; glycyl-aspartic acid; 2-[(ammonioacetyl)amino]succinate; Gly-L-Asp-OH; (2S)-2-[(2-aminoacetyl)amino]butanedioic acid; Gly-Asp, >=99.0%; SCHEMBL3207709; CTK2H6985; KS-00000YLG; ZINC1708196; EINECS 225-140-1; BDBM50188493; MFCD00025585; AKOS015855053; AKOS015893977; NSC 118367; AS-63212; (S)-2-(2-Amino-acetylamino)-succinic acid; G0121; K-0071; Q27144120
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| Activity |
Ki = 350000 nM
|
[4] | |||
| Compound Name |
His-his
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Investigative | Compound Info | ||
| Synonyms |
H-His-His-OH; histidyl-histidine; L-histidyl-L-histidine; N'alpha-Histidylhistidine; CHEMBL377872; His-His-OH; L-His-L-His; H-L-His-L-His-OH; SCHEMBL2958250; SCHEMBL21828671; ZINC1605452; BDBM50188500; Q27144364
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| Activity |
EC50 = 370000 nM
|
[1] | |||
| Compound Name |
Glycyl-DL-alanine
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Investigative | Compound Info | ||
| Synonyms |
Glycylalanine; 2-[(2-aminoacetyl)amino]propanoic acid; 2-(2-aminoacetamido)propanoic acid; DL-Alanine, N-glycyl-; DL-glycylalanine; L-Alanine, N-glycyl-; N-Glycyl-L-alanine; Glycine-.alpha.-alanine; 2-[(ammonioacetyl)amino]propanoate; Glycine-alanine dipeptide; N-Glycyl-DL-alanine; H-Gly-DL-Ala-OH; Alanine, N-glycyl-, L-; GLY-DL-ALA; Glcylalanine; NSC-522445; EINECS 213-144-6; ACMC-209ipy; ACMC-1CPCL; N-(Aminoacetyl)alanine #; NCIOpen2_001044; CHEMBL56351; SCHEMBL783990; CTK4F1183; DTXSID60919063; ALBB-031714; NSC83246; 7315AF; ANW-39874; MFCD00025587; NSC-83246; NSC522445; STL524949; 2-(2-aminoacetylamino)propanoic acid; AKOS009157380; MCULE-2027405418; 2-[(2-azaniumylacetyl)amino]propanoate; N-(2-Amino-1-hydroxyethylidene)alanine; DB-049039; DB-055237; DB-057321; FT-0632815; FT-0633106; FT-0634971; G0112; ST50409393; Q27258751
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| Activity |
Ki = 380000 nM
|
[4] | |||
| Compound Name |
Glu-Gly
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Investigative | Compound Info | ||
| Synonyms |
H-Glu-Gly-OH; glutamylglycine; Glu-Gly-OH; Glycine, L-alpha-glutamyl-; CHEMBL421361; alpha-glutamylglycine; (4S)-4-amino-5-(carboxymethylamino)-5-oxopentanoic acid; glutamyl glycine; glutamyl-glycine; EG dipeptide; E-G Dipeptide; alpha-L-Glu-Gly; L-Glutamyl-glycine; L-Glu-Gly; L-Glutamyl-L-Glycine; L-alpha-glutamylglycine; Glutamate Glycine dipeptide; Glutamate-Glycine dipeptide; SCHEMBL6045489; ZINC1731776; 7152AH; BDBM50188507; MFCD00037311; AS-57857; K-4407; 4-Amino-4-(carboxymethyl-carbamoyl)-butyric acid; (S)-4-Amino-4-(carboxymethyl-carbamoyl)-butyric acid; Q27140585; (4S)-4-amino-4-[(carboxymethyl)carbamoyl]butanoic acid; (S)-4-amino-5-(carboxymethylamino)-5-oxopentanoic acid; (4S)-4-Amino-5-[(carboxymethyl)amino]-5-oxopentanoic acid
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| Activity |
IC50 = 390000 nM
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[1] | |||
| Compound Name |
(S)-2-Amino-3-methylbutanoic benzoic anhydride
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL592658; SCHEMBL6483049; BDBM50308747
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| Activity |
IC50 = 390000 nM
|
[17] | |||
| Compound Name |
Leucyl-glycyl-glycine
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Investigative | Compound Info | ||
| Synonyms |
Leu-Gly-Gly; l-leucylglycylglycine; L-Leucyl-glycyl-glycine; H-Leu-Gly-Gly-OH; N-(N-L-Leucylglycyl)glycine; Leucylglycylglycine; CHEMBL297722; (S)-2-(2-(2-Amino-4-methylpentanamido)acetamido)acetic acid; MFCD00065942; 2-[[2-[[(2S)-2-amino-4-methylpentanoyl]amino]acetyl]amino]acetic acid; Glycine,L-leucylglycyl-; EINECS 214-698-1; L-Leu-Gly-Gly; L-Leu-Gly-Gly-OH; NSC 118380; Glycine, leucylglycyl-; SCHEMBL1036014; CTK1D7669; ZINC1708209; ANW-17230; BDBM50169136; AKOS010367266; AKOS015853931; 187L504; Q27144715; 0962ABF0-21F5-4144-B541-32E255DFA0CA; [2-(2-Amino-4-methyl-pentanoylamino)-acetylamino]-acetic acid; [2-((S)-2-Amino-4-methyl-pentanoylamino)-acetylamino]-acetic acid
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| Activity |
Ki = 390000 nM
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[2] | |||
| Compound Name |
Gly-his
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Investigative | Compound Info | ||
| Synonyms |
Glycyl-L-histidine; H-Gly-His-OH; L-Histidine, glycyl-; Glycylhistidine; CHEMBL93127; (S)-2-(2-Aminoacetamido)-3-(1H-imidazol-4-yl)propanoic acid; Gly-L-His; Gly-L-His-OH; SCHEMBL483799; CTK1A1128; (2S)-2-(2-aminoacetamido)-3-(1H-imidazol-4-yl)propanoic acid; ZINC4533503; BDBM50169199; MFCD00167467; AS-57332; Q27140597; 2-(2-Amino-acetylamino)-3-(3H-imidazol-4-yl)-propionic acid; (S)-2-(2-Amino-acetylamino)-3-(3H-imidazol-4-yl)-propionic acid
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| Activity |
EC50 = 400000 nM
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[1] | |||
| Compound Name |
[(2S,3R)-3-Amino-2-hydroxy-4-phenylbutyryl]-L-leucine
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Investigative | Compound Info | ||
| Synonyms |
Bestatin;Ubenimex; NSC265489; NSC-265489; SCHEMBL8191715; CHEMBL1161364; CTK5A9162; WLN: 1Y1&1YVQMVYQYZ1R; HMS3370B12; HMS3394A03; HMS3748C21; L-Leucine, [S-(R*,S*)]-; SBB066073; AKOS015894858; MCULE-5470002097; (8S,2R)-DIAMINONONANEDIOIC ACID; AK162414; NCI60_002133; SC-13323; FT-0630708; N-((2S,3R)-3-AMINO-2-HYDROXY-4-PHENYLBUTYRYL)-L-LE; 2-(3-amino-2-hydroxy-4-phenylbutanoylamino)-4-methylpentanoic acid; L-Leucine,N-[(2S,3R)-3-amino-2-hydroxy-1-oxo-4-phenylbutyl]-
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| Activity |
Ki = 400000 nM
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[4] | |||
| Compound Name |
Asp-Asp
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Investigative | Compound Info | ||
| Synonyms |
H-ASP-ASP-OH; (S)-2-((S)-2-Amino-3-carboxypropanamido)succinic acid; CHEMBL17171; Aspartyl-aspartic Acid; Asp-Asp-OH; L-Asp-L-Asp; NH2-Asp-Asp-COOH; alpha-aspartylaspartic acid; L-Aspartyl-L-aspartic acid; SCHEMBL434560; L-alpha-aspartyl-L-aspartic acid; ZINC1575288; BDBM50169127; MFCD00055820; 2-(2-Amino-3-carboxy-propionylamino)-succinic acid; Q27140532; (S)-2-((S)-2-Amino-3-carboxy-propionylamino)-succinic acid
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| Activity |
Ki = 410000 nM
|
[2] | |||
| Compound Name |
2-Amino-N-(3-methylphenyl)propanamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1161354; SCHEMBL12812735; AKOS000183588; AKOS016049746
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| Activity |
Ki = 410000 nM
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[4] | |||
| Compound Name |
3-Amino-4-oxo-heptanedioic acid 1-benzyl ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL434541; BDBM50152065
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| Activity |
Ki = 417000 nM
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[6] | |||
| Compound Name |
Gln-Glu
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Investigative | Compound Info | ||
| Synonyms |
H-GLN-GLU-OH; L-glutaminyl-L-glutamic acid; glutaminylglutamic acid; CHEMBL210850; QE dipeptide; Glutaminylglutamate; Q-E Dipeptide; L-Gln-L-Glu; Glutaminyl-glutaminsaure; glutaminyl-glutamic acid; L-Glutaminyl-L-Glutamate; Glutamine Glutamate dipeptide; Glutamine-Glutamate dipeptide; SCHEMBL435320; ZINC2560992; BDBM50188514; MFCD00237870; Q27144170; (2S)-2-[[(2S)-2,5-diamino-5-oxopentanoyl]amino]pentanedioic acid
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| Activity |
EC50 = 420000 nM
|
[1] | |||
| Compound Name |
(3R)-3-Amino-4-[[(2R,3S,4R)-5-(2-bromo-5,6-dichlorobenzimidazol-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy]-4-oxobutanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL607962; BDBM50370615
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| Activity |
IC50 = 421000 nM
|
[8] | |||
| Compound Name |
Asp-gly
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Investigative | Compound Info | ||
| Synonyms |
(S)-3-Amino-4-((carboxymethyl)amino)-4-oxobutanoic acid; H-ASP-GLY-OH; L-alpha-aspartylglycine; aspartyl-glycine; UNII-69Y3FAP7XY; 69Y3FAP7XY; CHEMBL421171; (3S)-3-amino-4-(carboxymethylamino)-4-oxobutanoic acid; L-Aspartylglycine; alpha-aspartylglycine; H-Asp(gly)-OH; Glycine, L-alpha-aspartyl-; L-Aspartyl-glycine; CMX-1152; L-Asp-Gly; H-Asp-Glp-OH; L-Asp-Gly-OH; NSC 186907; Glycine, N-L-alpha-aspartyl-; SCHEMBL2581218; CTK8C2557; ZINC2384840; 4856AB; ANW-68588; BDBM50188502; MFCD00037287; AKOS006275621; (S)-3-Amino-N-carboxymethyl-succinamic acid; Q27140535; (3S)-3-amino-3-[(carboxymethyl)carbamoyl]propanoic acid; (S)-3-amino-4-(carboxymethylamino)-4-oxobutanoic acid
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| Activity |
EC50 = 440000 nM
|
[1] | |||
| Compound Name |
(2S,3S,4R,5R)-2-(2-Bromo-5,6-dichloro-benzimidazol-1-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2093921; SCHEMBL7635326; BDBM50422694; 2-Bromo-5,6-dichloro-1-(.alpha.-D-lyxofuranosyl)benzimidazole; 1-(alpha-D-Lyxofuranosyl)-2-bromo-5,6-dichloro-1H-benzimidazole; (2S,3S,4R,5R)-2-(2-bromo-5,6-dichlorobenzimidazol-1-yl)-5-(hydroxymethyl)oxolane-3,4-diol
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| Activity |
IC50 = 447000 nM
|
[8] | |||
| Compound Name |
2-Amino-N-(3-chlorophenyl)propanamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1161361; AKOS000182342
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| Activity |
Ki = 460000 nM
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[4] | |||
| Compound Name |
Asp-Trp
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Investigative | Compound Info | ||
| Synonyms |
H-Asp-Trp-OH; Aspartyl-Tryptophan; CHEMBL210490; aspartyltryptophan; L-Aspartyl-L-Tryptophan; L-alpha-Asp-L-Trp; L-Asp-L-Trp; alpha-aspartyltryptophan; L-alpha-aspartyl-L-tryptophan; SCHEMBL7422711; ZINC2560972; BDBM50188490; MFCD00237825; Q27144149; (S)-3-amino-4-((S)-1-carboxy-2-(1H-indol-3-yl)ethylamino)-4-oxobutanoic acid
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| Activity |
EC50 = 470000 nM
|
[1] | |||
| Compound Name |
[(2R,3S,4R)-5-(2-Bromo-5,6-dichlorobenzimidazol-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2S)-2,6-diaminohexanoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL607956; BDBM50370605
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| Activity |
IC50 = 477000 nM
|
[8] | |||
| Compound Name |
Glycylglycine
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Investigative | Compound Info | ||
| Synonyms |
Diglycine; N-GLYCYLGLYCINE; Gly-Gly; Glycine, glycyl-; Glycyl-glycine; Glycine dipeptide; 2-(2-Aminoacetamido)Acetic Acid; Glycine, N-glycyl-; H-Gly-Gly-OH; Gly-Gly-OH; 2-(Aminoacetamido)acetic acid; 2-[(2-aminoacetyl)amino]acetic acid; alpha-Glycylglycine; MFCD00008130; [(Aminoacetyl)amino]acetic acid; UNII-10525P22U0; CHEMBL292467; Glycylglycine, 99+%; 10525P22U0; glycylglycine zwitterion; ((aminoacetyl)amino)acetic acid; 2-(2-aminoacetylamino)acetic acid; Glycyl Glycine; Glycylgycine; EINECS 209-127-8; H-Gly-Gly; Glycylglycine, DL-; NSC 49346; .alpha.-Glycylglycine; n-GLYCYL- Glycine; PubChem14973; ACMC-1AWKP; AI3-62521; Glycylglycine (GLYGLY); Gly-Gly, 98%; B-GLYGLY250; SCHEMBL14934; KSC492E0P; CTK3J2207; DTXSID90862194; Gly-Gly, >=99% (titration); [(Aminoacetyl)amino]acetic acid #; HY-D0889; NSC49346; ZINC5112515; ANW-32355; BBL018705; BDBM50169222; NSC-49346; s4810; SBB067231; STL194277; AKOS001045997; CCG-231053; MCULE-1239116894; KS-000002A7; Gly-Gly, BioXtra, >=99.0% (NT); AK-46058; AS-14771; Gly-Gly, BioUltra, >=99.5% (NT); SC-17448; ST099026; SY018005; Gly-Gly, Vetec(TM) reagent grade, 99%; AB0006830; DB-002742; CS-0015211; FT-0626788; G0124; T7982; C02037; G-6000; G-6001; Glycylglycine, 0.2M buffer solution, pH 8.0; Glycylglycine, 0.2M buffer solution, pH 8.5; 556G503; Q665455; F2191-0195; 2,3,6,2',3',4',6'-Hepta-O-acetyl-a-D-lactosyl bromide; 33903968-DDB2-47F2-9B6C-7C232D1962DA; Dyglycine, United States Pharmacopeia (USP) Reference Standard; Gly-Gly, BioPerformance Certified, cell culture tested, >=99%
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| Activity |
EC50 = 480000 nM
|
[1] | |||
| Compound Name |
Histidylalanine
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Investigative | Compound Info | ||
| Synonyms |
His-ala; L-His-ala; l-histidyl-l-alanine; Histidinoalanine; (S)-2-((S)-2-Amino-3-(1H-imidazol-4-yl)propanamido)propanoic acid; H-His-Ala-OH; N-(2-Amino-2-carboxyethyl)histidine; Histidinylalanine; histidyl-alanine; (2S)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]propanoic acid; His-Ala-OH; L-His-L-Ala; NSC 522632; L-Alanine, L-histidyl-; SCHEMBL5077779; CHEMBL2371149; CTK0H9808; ZINC1605278; MFCD00055955; Q27144247; 1H-Imidazole-1,4-dipropanoic acid, alpha,alpha'-diamino-, (S-(R*,R*))-
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| Activity |
Ki = 480000 nM
|
[4] | |||
| Compound Name |
Glycyl-L-alanine
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Investigative | Compound Info | ||
| Synonyms |
Gly-ala; H-Gly-Ala-OH; N-Glycylalanine; Glycylalanine; (S)-2-(2-Aminoacetamido)propanoic acid; L-glycylalanine; UNII-2M7GF488BL; CHEMBL91241; 2M7GF488BL; N-Glycyl-L-alanine; Gly-L-Ala; Alanine, N-glycyl-, L-; Glycylalanine, L-; Glycine-.alpha.-alanine; Glycine-alanine dipeptide; glycyl-alanine; GlyAla; gly ala; Alanine, glycyl-; EINECS 223-019-8; Gly-Ala-OH; Gly-L-Ala-OH; (2S)-2-[(2-aminoacetyl)amino]propanoic acid; N-(Aminoacetyl)alanine, L-; SCHEMBL564562; CTK1C3318; KS-000015SB; ZINC1730665; 7020AH; ANW-28532; BDBM50188530; Gly-Ala, >=99.0% (NT); MFCD00065112; NSC 83246; AKOS010397041; AKOS015855052; MCULE-7578084271; AS-48944; G0113; (S)-2-(2-Amino-acetylamino)-propionic acid; K-8203; Q27144182; UNII-44L9158R9G component VPZXBVLAVMBEQI-VKHMYHEASA-N
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| Activity |
EC50 = 520000 nM
|
[1] | |||
| Compound Name |
Lysylglutamic acid
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Investigative | Compound Info | ||
| Synonyms |
H-LYS-GLU-OH; Lys-Glu; Peptide vilon; UNII-H34V7IM5ML; L-LYSYL-L-GLUTAMIC ACID; H34V7IM5ML; CHEMBL365790; (S)-2-((S)-2,6-Diaminohexanamido)pentanedioic acid; Lysyl-Glutamate; (2S)-2-[[(2S)-2,6-diaminohexanoyl]amino]pentanedioic Acid; (2S)-2-{[(2S)-2,6-Diaminohexanoyl]amino}pentanedioic acid; CCRIS 8868; Lysyl-glutaminsaure; Lysyl-glutamic acid; L-Lys-L-Glu; L-Glutamic acid,L-lysyl-; N-L-Lysyl-L-glutamic acid; SCHEMBL1973948; CTK7E7756; DTXSID50196442; ZINC2390919; 7202AH; BDBM50169126; MFCD00038215; Q27144733; (S)-2-((S)-2,6-Diamino-hexanoylamino)-pentanedioic acid
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| Activity |
EC50 = 530000 nM
|
[1] | |||
| Compound Name |
[(2R,3S,4R)-5-(2-Bromo-5,6-dichlorobenzimidazol-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2S)-pyrrolidine-2-carboxylate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL608509; BDBM50370610
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||||
| Activity |
IC50 = 537000 nM
|
[8] | |||
| Compound Name |
Glycylsarcosine
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Investigative | Compound Info | ||
| Synonyms |
Glycyl-sarcosine; Gly-Sar; H-Gly-Sar-OH; 2-(2-amino-N-methylacetamido)acetic acid; N-Glycylsarcosine; Gly-Sarcosin; 2-[(2-aminoacetyl)-methylamino]acetic acid; UNII-2JE8SG6VDT; 2JE8SG6VDT; CHEMBL175737; MFCD00038193; N-glycyl-Sar-OH; EINECS 249-875-2; Gly-Sar-OH; [3H]GlySar; NSC 206288; glycyl-N-methylglycine; [3H]-GlySar; tritiated glycylsarcosine; N-glycyl-N-methylglycine; ACMC-209hb7; Glycine, N-glycyl-N-methyl-; SCHEMBL510835; GTPL4659; GTPL9505; CTK8B1399; DTXSID50183953; KS-000012VZ; ZINC1742265; 7028AH; ANW-26705; BDBM50188516; NSC206288; [(ammonioacetyl)(methyl)amino]acetate; AKOS009157522; NSC-206288; [(Aminoacetyl)(methyl)amino]acetic acid; AS-56734; [(Aminoacetyl)(methyl)amino]acetic acid #; FT-0760838; G0138; [(2-Amino-acetyl)-methyl-amino]-acetic acid; K-7194; J-017657
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||||
| Activity |
EC50 = 540000 nM
|
[1] | |||
| Compound Name |
Glycylglycylglycine
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Investigative | Compound Info | ||
| Synonyms |
Triglycine; Glycyl-glycyl-glycine; H-Gly-Gly-Gly-OH; Gly-Gly-Gly; Diglycylglycine; N-(N-Glycylglycyl)glycine; Glycine, glycylglycyl-; 2-(2-(2-Aminoacetamido)acetamido)acetic acid; GlyGlyGly; UNII-CVK73ZDQ8B; 2-[[2-[(2-aminoacetyl)amino]acetyl]amino]acetic acid; MFCD00036223; Gly-Gly-Gly-OH; CVK73ZDQ8B; CHEMBL54278; Glycine, N-(N-glycylglycyl)-; Glycine, N-(N-glycylglycyl)- (8CI)(9CI); [2-(2-Amino-acetylamino)-acetylamino]-acetic acid; Glycylpeptide; Triglycine (van); NSC46707; EINECS 209-122-0; NSC 46707; Maybridge1_006812; (Gly)3; ACMC-209lo4; Glycylglycylglycine, 98+%; SCHEMBL98565; N-(N-GLYCYLGLYCYL)-Glycine; CTK1H1133; HMS560N14; DTXSID80204140; ZINC1678871; ANW-32354; BDBM50188484; NSC-46707; SBB071512; AKOS005207234; DS-7430; MCULE-8930278374; AK161962; SC-15976; SY025319; FT-0690006; G0126; Gly-Gly-Gly, BioUltra, >=99.0% (NT); (([(Aminoacetyl)amino]acetyl)amino)acetic acid; K-9925; (([(Aminoacetyl)amino]acetyl)amino)acetic acid #; 2-[2-(2-aminoacetylamino)acetylamino]acetic acid; 556G332; Q27132936; Triglycine, United States Pharmacopeia (USP) Reference Standard; 2-[[2-[(2-Aminoacetyl)amino]acetyl]amino]acetic Acid (Triglycine)
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||||
| Activity |
EC50 = 580000 nM
|
[1] | |||
| Compound Name |
(S)-2-((S)-2-Amino-3-(2,5,7-tri-tert-butyl-1H-indol-3-yl)propanamido)-5-guanidinopentanamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL365705; TbtR-NH2; BDBM50341599
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||||
| Activity |
IC50 = 600000 nM
|
[18] | |||
| Compound Name |
Glu-glu
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Investigative | Compound Info | ||
| Synonyms |
Glutamyl-glutamic acid; H-GLU-GLU-OH; L-Glutamyl-L-glutamic acid; Glu(Glu); L-Glutamic acid, L-a-glutamyl-; (S)-2-((S)-2-Amino-4-carboxybutanamido)pentanedioic acid; CHEMBL318315; L-alpha-Glutamyl-L-glutamic acid; L-glutamyl-L-glutamate; glutamylglutamic acid; glutamylglutamate; EE dipeptide; E-E Dipeptide; Glu-Glu-OH; L-Glu-L-Glu; glutamyl glutamic acid; H-L-Glu-L-Glu-OH; alpha-glutamylglutamic acid; Glutamate Glutamate dipeptide; Glutamate-Glutamate dipeptide; SCHEMBL435318; ZINC1529201; BDBM50102260; MFCD00037309; VA50422; AS-60181; C01425; 2-(2-Amino-4-carboxy-butyrylamino)-pentanedioic acid; Q27106747; (2S)-2-[(2S)-2-amino-4-carboxybutanamido]pentanedioic acid
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|
||||
| Activity |
IC50 = 620000 nM
|
[1] | |||
| Compound Name |
(2S,3S)-2-Amino-3-methylpentanoic benzoic anhydride
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL604252; BDBM50308748
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||||
| Activity |
IC50 = 630000 nM
|
[17] | |||
| Compound Name |
L-Isoleucine[3-[(Aminoiminomethyl)amino]phenyl]methyl Ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL589585; BDBM50308745
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||||
| Activity |
IC50 = 630000 nM
|
[17] | |||
| Compound Name |
Glycyl-L-glutamic acid
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
Gly-Glu; N-Glycylglutamic acid; N-Glycyl-L-glutamic acid; (S)-2-(2-Aminoacetamido)pentanedioic acid; CHEMBL314532; (2S)-2-[(2-aminoacetyl)amino]pentanedioic acid; EINECS 231-019-4; Gly-L-Glu; Glycyl-glutamic acid; Gly-L-Glu-OH; H-Gly-Glu-OH; NSC 203441; L-Glutamic acid,glycyl-; (2S)-2-(2-aminoacetamido)pentanedioic acid; SCHEMBL709721; N-(Aminoacetyl)glutamic acid #; CTK5D9394; ZINC2567986; ANW-36435; BDBM50188529; MFCD00008128; AKOS010408430; AKOS015855061; AS-64954; 2-(2-Amino-acetylamino)-pentanedioic acid; G0123; ST50319374; (2S)-2-(2-aminoacetylamino)pentanedioic acid; KS-00001781; Q27144115
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|
||||
| Activity |
IC50 = 650000 nM
|
[1] | |||
| Compound Name |
L-Valine[3-[(Aminoiminomethyl)amino]phenyl]methyl Ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL590321; BDBM50308744
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||||
| Activity |
IC50 = 650000 nM
|
[17] | |||
| Compound Name |
Lys-trp
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Investigative | Compound Info | ||
| Synonyms |
H-LYS-TRP-OH; LYSYL-TRYPTOPHAN; L-lysyl-L-tryptophan; CHEMBL169360; L-Lys-L-Trp; SCHEMBL1939435; CTK7E7754; ZINC2384979; BDBM50001946; Q27144746; 2-(6-Amino-2-aminomethyl-hexanoylamino)-3-(1H-indol-3-yl)-propionic acid
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||||
| Activity |
IC50 = 660000 nM
|
[1] | |||
| Compound Name |
Pro-Pro
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL371194; L-prolyl-L-proline; L-Proline, L-prolyl-; prolyl-proline; L-Pro-L-Pro; L-Pro-L-Pro-OH; SCHEMBL825679; ZINC4899613; BDBM50169141; AKOS010419474; Q27143817; (S)-1-((S)-Pyrrolidine-2-carbonyl)pyrrolidine-2-carboxylic acid; i(S)-1-((S)-Pyrrolidine-2-carbonyl)-pyrroliidine-2-carboxylic acid
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||||
| Activity |
EC50 = 700000 nM
|
[1] | |||
| Compound Name |
Prolyl-tyrosine
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Investigative | Compound Info | ||
| Synonyms |
H-Pro-Tyr-OH; Pro-tyr; L-prolyl-L-tyrosine; L-Tyrosine, L-prolyl-; N-L-prolyl-L-tyrosine; prolyltyrosine; L-Prolyl-L-tyrosine monohydrate; (2S)-3-(4-hydroxyphenyl)-2-[[(2S)-pyrrolidine-2-carbonyl]amino]propanoic acid; L-Pro-L-Tyr; L-Tyrosine, N-L-prolyl-; H-Pro-Tyr-OH, AldrichCPR; CHEMBL298979; SCHEMBL6367397; CTK0H5203; DTXSID30173493; ZINC4899447; 7237AH; MFCD00037870; AKOS010408836; Q27144910
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||||
| Activity |
Ki = 730000 nM
|
[4] | |||
| Compound Name |
Gly-lys
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Investigative | Compound Info | ||
| Synonyms |
Glycyl-L-lysine; Glycyllysine; Glycyl-Lysine; L-Lysine, glycyl-; CHEMBL420061; Glycinyl-L-lysine; Gly-L-Lys; Gly-Lys-OH; L-Lysine, N2-glycyl-; SCHEMBL1455499; CTK3I7347; DTXSID50244215; BDBM50188513; ZINC71755677; (S)-6-Amino-2-(2-amino-acetylamino)-hexanoic acid; Q27144235
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||||
| Activity |
EC50 = 750000 nM
|
[1] | |||
| Compound Name |
Phe-Ala-NH2
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL210616; L-Alaninamide, L-phenylalanyl-; BDBM50188495; (2S)-2-amino-N-[(2S)-1-amino-1-oxopropan-2-yl]-3-phenylpropanamide
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||||
| Activity |
EC50 = 850000 nM
|
[1] | |||
| Compound Name |
Methyl 2-(2-aminopropanoylamino)benzoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1161359
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||||
| Activity |
Ki = 890000 nM
|
[4] | |||
| Compound Name |
5-Amino-4-oxo-6-phenyl-hexanoic acid benzyl ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL187172; BDBM50152066
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||||
| Activity |
Ki = 905000 nM
|
[6] | |||
| Compound Name |
Alanyl ornithine
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Investigative | Compound Info | ||
| Synonyms |
L-Ornithine, L-alanyl-; UNII-ZR4JSN38SV; ZR4JSN38SV; (S)-5-amino-2-((S)-2-aminopropanamido)pentanoic acid; Dipeptide ao-a; Alanyl ornithine [INCI]; alanylornithine; CHEMBL2371842; Q27295860; (2S)-5-amino-2-[[(2S)-2-aminopropanoyl]amino]pentanoic acid
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||||
| Activity |
Ki = 970000 nM
|
[2] | |||
| Compound Name |
Methyl 4-(2-aminopropanoylamino)benzoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1161368; AKOS009132452
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||||
| Activity |
Ki = 1100000 nM
|
[4] | |||
| Compound Name |
Thr-Lys-Tyr
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Investigative | Compound Info | ||
| Synonyms |
H-THR-LYS-TYR-OH; CHEMBL363832; Threonyl-lysyl-tyrosine; L-Threonyl-L-lysyl-L-tyrosine; ZINC4899469; BDBM50169162; MFCD00038590
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||||
| Activity |
Ki = 1100000 nM
|
[2] | |||
| Compound Name |
Alanine, N-L-alanyl-2-methyl-
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Investigative | Compound Info | ||
| Synonyms |
SCHEMBL1979304; CHEMBL2371160; AKOS010518183
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||||
| Activity |
Ki = 1200000 nM
|
[4] | |||
| Compound Name |
2-[(2-Ammoniopropanoyl)amino]ethanesulfonate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL154626; SCHEMBL8460853
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||||
| Activity |
Ki = 1200000 nM
|
[4] | |||
| Compound Name |
(S)-2-[(S)-2-Amino-3-(4-phenoxy-phenyl)-propionylamino]-propionic acid
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL190668; BDBM50169144
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|
||||
| Activity |
Ki = 1400000 nM
|
[2] | |||
| Compound Name |
2-[[(2R)-2-Amino-3-(4-phenylmethoxyphenyl)propanoyl]amino]propanoic acid
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2111209; BDBM50409776
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||||
| Activity |
Ki = 1400000 nM
|
[4] | |||
| Compound Name |
2-[(2-Amino-6-oxo-3H-purin-9-yl)methoxy]ethyl 2-aminoacetate
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
UNII-T3FT9SC1UC; T3FT9SC1UC; CHEMBL1194823; Glycine, 2-((2-amino-1,6-dihydro-6-oxo-9H-purin-9-yl)methoxy)ethyl ester; Glycine, 2-[(2-amino-1,6-dihydro-6-oxo-9H-purin-9-yl)methoxy]ethyl ester; 2'-O-Glycyl acyclovir; Acyclovir 2'-O-glycyl ester; GLYCYL ESTER OF ACYCLOVIR; DTXSID401004770; 9-(2-glycyloxyethoxy-methyl)guanine; BDBM50391005; 2-[(2-amino-6-oxo-1H-purin-9-yl)methoxy]ethyl 2-aminoacetate; 2-Amino-9-[[2-(glycyloxy)ethoxy]methyl]-1H-purine-6(9H)-one; 2-[(6-Hydroxy-2-imino-2,3-dihydro-9H-purin-9-yl)methoxy]ethyl glycinate
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||||
| Activity |
IC50 = 1400000 nM
|
[11] | |||
| Compound Name |
Cyclohexanecarboxylic acid ((S)-2-amino-propionyl)-amide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL190085; BDBM50169179
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||||
| Activity |
Ki = 1500000 nM
|
[2] | |||
| Compound Name |
2-Amino-N-cyclohexylpropanamide
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Investigative | Compound Info | ||
| Synonyms |
2-Amino-N-cyclohexyl-DL-propanamide; SCHEMBL5220274; CHEMBL1161363; 2-amino-N-cyclohexyl-propionamide; KM2392; AKOS000188663; AKOS017263138
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||||
| Activity |
Ki = 1500000 nM
|
[4] | |||
| Compound Name |
Pro-Ser
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Investigative | Compound Info | ||
| Synonyms |
H-Pro-Ser-OH; CHEMBL209083; L-prolyl-L-serine; prolylserine; prolyl-serine; L-Pro-L-Ser; (2S)-3-hydroxy-2-[[(2S)-pyrrolidine-2-carbonyl]amino]propanoic acid; L-Serine, L-prolyl-; L-Serine, N-L-prolyl-; CTK2H3274; DTXSID70428595; ZINC4899564; BDBM50188510; MFCD00083811; AKOS010408212; Q27143819
Click to Show/Hide
|
||||
| Activity |
EC50 = 1600000 nM
|
[1] | |||
| Compound Name |
Sar-pro-OH
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Investigative | Compound Info | ||
| Synonyms |
1-Sarcosyl-L-proline; L-Proline, N-methylglycyl-; SCHEMBL7364621; CHEMBL2371139; ZINC4899479; MFCD00038855; AKOS010419670; (2S)-1-[2-(methylamino)acetyl]pyrrolidine-2-carboxylic acid
Click to Show/Hide
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||||
| Activity |
Ki = 1600000 nM
|
[4] | |||
| Compound Name |
N-Methyl-L-alanyl-L-alanine
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2371151; SCHEMBL13165106; CTK2E1272; DTXSID30817981; ZINC13531511; L-Alanine, N-(N-methyl-L-alanyl)-
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||||
| Activity |
Ki = 1800000 nM
|
[4] | |||
| Compound Name |
L-Prolyl-L-phenylalanine
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|
Investigative | Compound Info | ||
| Synonyms |
H-Pro-Phe-OH; Pro-Phe; L-Pro-L-Phe; Prolyl-phenylalanine; L-Pro-L-Phe-OH; (S)-3-Phenyl-2-((S)-pyrrolidine-2-carboxamido)Propanoic acid; CHEMBL52922; SCHEMBL601567; ZINC4038394; MFCD00037869; STL527311; AKOS010421062; MCULE-8228255768; Q27144906
Click to Show/Hide
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||||
| Activity |
Ki = 1900000 nM
|
[4] | |||
| Compound Name |
d-Alanyl-l-alanine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
H-D-Ala-Ala-OH; L-Alanine, D-alanyl-; N-ALANYLALANINE; UNII-C7641UJG3Q; C7641UJG3Q; CHEMBL1814491; (2S)-2-[[(2R)-2-aminopropanoyl]amino]propanoic acid; (S)-2-((R)-2-Aminopropanamido)propanoic acid; d-alanylalanine; NSC-203792; D-Ala-Ala-OHHCl; D-Ala-L-Ala-OH; D-Ala-Ala-OH HCl; N-D-Alanyl-L-alanine; H-D-Ala-Ala-OH HCl; SCHEMBL574263; CTK0I2831; DTXSID901016946; ZINC1575494; 7092AH; BDBM50350475; MFCD00066039; AKOS017430148; UNII-3CUV6EVI23 component DEFJQIDDEAULHB-DMTCNVIQSA-N; UNII-3EE68A29TN component DEFJQIDDEAULHB-DMTCNVIQSA-N
Click to Show/Hide
|
||||
| Activity |
Ki = 2000000 nM
|
[4] | |||
| Compound Name |
(2S)-6-Amino-2-[[(2S)-3-phenyl-2-[[(2S)-pyrrolidine-2-carbonyl]amino]propanoyl]amino]hexanoic Acid
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
Pro-Phe-Lys; CHEMBL426809; H-Pro-Phe-Lys-OH; Prolyl-phenylalanyl-lysine; L-Prolyl-L-phenylalanyl-L-lysine; ZINC4899895; BDBM50169183; (S)-6-Amino-2-{(S)-3-phenyl-2-[((S)-pyrrolidine-2-carbonyl)-amino]-propionylamino}-hexanoic acid
Click to Show/Hide
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||||
| Activity |
Ki = 2000000 nM
|
[2] | |||
| Compound Name |
3-(3-Aminopropyl)-6-methylpiperazine-2,5-dione
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1161346
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||||
| Activity |
Ki = 2300000 nM
|
[4] | |||
| Compound Name |
L-Phenylalanine[3-[(Aminoiminomethyl)amino]phenyl]methyl Ester
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL603829; BDBM50308746
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|
||||
| Activity |
IC50 = 2330000 nM
|
[17] | |||
| Compound Name |
Prolylarginine
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Investigative | Compound Info | ||
| Synonyms |
Pro-arg; L-prolyl-L-arginine; prolyl-arginine; L-Arginine, L-prolyl-; CHEMBL190549; H-Pro-Arg-OH; H-Pro-Arg; L-Pro-L-Arg; L-Arginine, N2-L-prolyl-; SCHEMBL8759341; CTK1A3223; DTXSID30178887; ZINC4899789; BDBM50169180; Q27143816; (S)-5-Guanidino-2-((S)-pyrrolidine-2-carboxamido)pentanoic acid; (S)-5-Guanidino-2-[((S)-pyrrolidine-2-carbonyl)-amino]-pentanoic acid
Click to Show/Hide
|
||||
| Activity |
Ki = 2500000 nM
|
[2] | |||
| Compound Name |
(2S)-2-Amino-N-[(2S)-1-[[(2S)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-5-(diaminomethylideneamino)pentanamide
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL41644; BDBM50341600
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||||
| Activity |
IC50 = 2700000 nM
|
[18] | |||
| Compound Name |
3-(2-Aminopropanoylamino)propanoic acid
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL186269; 3-[(2-ammoniopropanoyl)amino]propanoate; SCHEMBL7290638; DTXSID80967243; N-(2-aminopropanoyl)-beta-alanine; BDBM50169204; AKOS010404015; 3-(2-Amino-propionylamino)-propionic acid; FT-0695784; FT-0695787; N-(2-Amino-1-hydroxypropylidene)-beta-alanine
Click to Show/Hide
|
||||
| Activity |
Ki = 2700000 nM
|
[2] | |||
| Compound Name |
2-(2-Azaniumylpropanoylamino)benzoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL157386; 2-[(2-ammoniopropanoyl)amino]benzoate; BDBM50136990
Click to Show/Hide
|
||||
| Activity |
Ki = 2800000 nM
|
[4] | |||
| Compound Name |
2-Amino-N-phenylpropanamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
2-Amino-N-phenyl-DL-propanamide; Propanamide, 2-amino-N-phenyl-, (R)-; NSC194596; ACMC-20mbnm; SCHEMBL4741417; CHEMBL1161345; AKOS000183934; AKOS017263117; MCULE-5365959341; NSC-194596; K-0268; H-193/10
Click to Show/Hide
|
||||
| Activity |
Ki = 2900000 nM
|
[4] | |||
| Compound Name |
((S)-2-Amino-propionyl)-phenyl-carbamic acid
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL190126; BDBM50169191
Click to Show/Hide
|
||||
| Activity |
Ki = 2900000 nM
|
[2] | |||
| Compound Name |
[3-(Hydroxymethyl)phenyl]guanidine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL590071; SCHEMBL1186272; 3-(hydroxymethyl)phenylguanidine; BDBM50308743; 1-(3-(hydroxymethyl)phenyl)guanidine; 2-[3-(hydroxymethyl)phenyl]guanidine; 1-(3-(hydroxymethyl)phenyl)-guanidine
Click to Show/Hide
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||||
| Activity |
IC50 > 3000000 nM
|
[17] | |||
| Compound Name |
[(2S)-2-Amino-3-phenylpropanoyl] benzoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL592659; SCHEMBL2638485; BDBM50308749; (S)-2-amino-3-phenylpropanoic benzoic anhydride
Click to Show/Hide
|
||||
| Activity |
IC50 > 3000000 nM
|
[17] | |||
| Compound Name |
((S)-2-Amino-propionyl)-(3-fluoro-phenyl)-carbamic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL190809; BDBM50169214
Click to Show/Hide
|
||||
| Activity |
Ki = 3100000 nM
|
[2] | |||
| Compound Name |
2-Amino-N-(2,3,4,5,6-pentafluorophenyl)propanamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1161360
Click to Show/Hide
|
||||
| Activity |
Ki = 3100000 nM
|
[4] | |||
| Compound Name |
Alanyl-D-alanine
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
H-ALA-D-ALA-OH; D-Alanine, L-alanyl-; l-alanyl-d-alanine; Ala-D-Ala-OH; (2R)-2-[[(2S)-2-aminopropanoyl]amino]propanoic acid; CHEMBL1814487; UNII-A8235021UP; A8235021UP; L-Ala-D-Ala-OH; N-L-Alanyl-D-alanine; SCHEMBL380600; CTK1C3694; DTXSID201016945; ZINC1575495; 7042AH; BDBM50350461; MFCD00066040; AKOS010842226; NSC 186898; (R)-2-((S)-2-Aminopropanamido)propanoic acid; K-8204; Q27896855; UNII-3CUV6EVI23 component DEFJQIDDEAULHB-IUYQGCFVSA-N; UNII-3EE68A29TN component DEFJQIDDEAULHB-IUYQGCFVSA-N
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||||
| Activity |
Ki = 4200000 nM
|
[2] | |||
| Compound Name |
(R)-1-[(S)-1-((S)-2-Amino-3-methyl-butyryl)-pyrrolidine-2-carbonyl]-pyrrolidine-2-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL362955; BDBM50169171; ZINC13646355
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||||
| Activity |
Ki = 4300000 nM
|
[2] | |||
| Compound Name |
H-Ala-beta-Ala-OH
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL189696; Ala-beta-Ala; L-Alanine-; A-alanine; 3-[[(2S)-2-aminopropanoyl]amino]propanoic acid; N-L-Alanyl-beta-alanine; L-Alanyl-.beta.-alanine; SCHEMBL7290633; ZINC2390897; BDBM50169124; (S)-3-(2-aminopropanamido)propanoic acid; 3-((S)-2-Amino-propionylamino)-propionic acid; 788A020
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||||
| Activity |
Ki = 4800000 nM
|
[2] | |||
| Compound Name |
2-(3-Aminopropanoylamino)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL154156; 2-[(3-ammoniopropanoyl)amino]propanoate; NSC186897; .beta.-Alanyl-L-alanine; SCHEMBL434916; NSC-186897; 2-(3-azaniumylpropanoylamino)propanoate; DB-048598; FT-0639182
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||||
| Activity |
Ki = 4800000 nM
|
[4] | |||
| Compound Name |
1-D-Alanyl-L-proline
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Investigative | Compound Info | ||
| Synonyms |
H-D-Ala-Pro-OH; L-Proline, D-alanyl-; UNII-X5CGA70XLT; X5CGA70XLT; CHEMBL425551; (S)-1-((R)-2-Aminopropanoyl)pyrrolidine-2-carboxylic acid; (2S)-1-[(2R)-2-aminopropanoyl]pyrrolidine-2-carboxylic acid; d-Alanyl-l-prolin; EINECS 262-783-7; D-Ala-Pro-OH HCl; L-Proline, 1-D-alanyl-; SCHEMBL2115246; CTK2F7420; DTXSID00210369; ZINC1637975; BDBM50169181; AKOS010842269; Q27896445; (2S)-1-[(2R)-2-azaniumylpropanoyl]pyrrolidine-2-carboxylate; i(S)-1-((R)-2-Amino-propionyl)-pyrrolidine-2-carboxylic acid
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||||
| Activity |
Ki = 4900000 nM
|
[4] | |||
| Compound Name |
Cefuroxime
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Investigative | Compound Info | ||
| Synonyms |
Cephuroxime; Cefuroximo; Cefuroxim; Cefuroximum; Zinacef Danmark; Zinacef; Cefuroximum [INN-Latin]; Cefuroximo [INN-Spanish]; UNII-O1R9FJ93ED; Biofuroksym; Cefuril; O1R9FJ93ED; Q63409033; Cefuroxime [USAN:INN:BAN]; C16H16N4O8S; EINECS 259-560-1; BRN 5783190; Cefuroximine; Cefuroxime [USAN:BAN:INN]; Cefuroxime (TN); Cefuroxime (USAN/INN); Prestwick3_000720; CHEMBL1436; BSPBio_000939; BIDD:GT0619; BPBio1_001033; SCHEMBL1821942; HY-B1256A; ZINC3830485; BDBM50422689; MFCD00864889; AKOS015962849; AC-4539; DB01112; KS-5162; AB0010602; CS-0013520; EN300-53016; C06894; Cefuroxime, VETRANAL(TM), analytical standard; D00262; 268C752; A830563; Cefuroxime, Antibiotic for Culture Media Use Only; W-105575; BRD-K02733959-236-02-8; BRD-K02733959-236-07-7
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||||
| Activity |
Ki > 5000000 nM
|
[14] | |||
| Compound Name |
Pro-Asp
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Investigative | Compound Info | ||
| Synonyms |
H-Pro-Asp-OH; L-prolyl-L-aspartic acid; CHEMBL190704; (2S)-2-[[(2S)-pyrrolidine-2-carbonyl]amino]butanedioic acid; Prolyl-Aspartate; l-pro l-asp; prolyl-aspartic acid; L-Pro-L-Asp; L-Aspartic acid, L-prolyl-; CTK3C9100; ZINC4029831; BDBM50169195; MFCD00057886; STL527058; AKOS030494433; MCULE-3726564210; AS-56431; Q27144883; (S)-2-[((S)-Pyrrolidine-2-carbonyl)-amino]-succinic acid
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||||
| Activity |
EC50 > 5000000 nM
|
[1] | |||
| Compound Name |
Prolylglutamic acid
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Investigative | Compound Info | ||
| Synonyms |
Pro-glu; L-Prolyl-L-glutamic acid; CHEMBL190027; Prolyl-Glutamate; H-Pro-Glu-OH; pro glu; Prolyl-glutamic acid; L-Pro-L-Glu; N-L-Prolyl-L-glutamic acid; L-Glutamic acid, L-prolyl-; SCHEMBL5408968; L-Glutamic acid, N-L-prolyl-; CTK5C6473; DTXSID70987011; C10H16N2O5; ZINC3776573; BDBM50169114; MFCD00037872; STL527174; AKOS010408434; MCULE-1644415057; AS-58357; N-[Hydroxy(pyrrolidin-2-yl)methylidene]glutamic acid; Q27144887; (2S)-2-{[(2S)-pyrrolidin-2-yl]formamido}pentanedioic acid
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||||
| Activity |
EC50 > 5000000 nM
|
[1] | |||
| Compound Name |
3-(4-Aminobutyl)-6-methylpiperazine-2,5-dione
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1161356
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||||
| Activity |
Ki = 5400000 nM
|
[4] | |||
| Compound Name |
L-Alaninamide, L-alpha-aspartyl-
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL191532; SCHEMBL1083057; BDBM50169167; (S)-3-Amino-N-((S)-1-carbamoyl-ethyl)-succinamic acid; (3S)-3-amino-4-[[(2S)-1-amino-1-oxopropan-2-yl]amino]-4-oxobutanoic acid
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||||
| Activity |
Ki = 5400000 nM
|
[2] | |||
| Compound Name |
Z-Ala-ala-OH
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Investigative | Compound Info | ||
| Synonyms |
N-Cbz-L-alanyl-L-alanine; L-Alanine, N-[(phenylmethoxy)carbonyl]-L-alanyl-; (2S)-2-[[(2S)-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoic acid; benzyloxycarbonylalanyl alanine; (S)-2-((S)-2-(((Benzyloxy)carbonyl)amino)propanamido)propanoic acid; SCHEMBL3358693; CHEMBL2372591; N-carbobenzoxy-L-alanyl-L-alanine; ZINC2384803; MFCD00037234; N-benzyloxycarbonyl-L-alanyl-L-alanine; AS-17921; V3595; K-5022; J-009679; N-[N-[(Phenylmethoxy)carbonyl]-L-alanyl]-L-alanine; L-Alanine, N-[N-[(phenylmethoxy)carbonyl]-L-alanyl]-
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||||
| Activity |
Ki = 5600000 nM
|
[4] | |||
| Compound Name |
3-Methyl-1-oxo-1-piperidin-1-ylpentan-2-aminium
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL93507; SCHEMBL6824150; BDBM50118936; AKOS000171918; 2-Amino-3-methyl-1-piperidin-1-yl-pentan-1-one
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||||
| Activity |
Ki = 5620000 nM
|
[4] | |||
| Compound Name |
2-Amino-3-methyl-1-thiazolidin-3-yl-pentan-1-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL357606; SCHEMBL356202; BDBM50135043; PS32/98; 3-methyl-1-oxo-1-(1,3-thiazolidin-3-yl)pentan-2-aminium
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||||
| Activity |
Ki = 6300000 nM
|
[4] | |||
| Compound Name |
L-Alaninamide, L-lysyl-
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL191212; BDBM50169206; (S)-2,6-Diamino-hexanoic acid ((S)-1-carbamoyl-ethyl)-amide; (2S)-2,6-diamino-N-[(2S)-1-amino-1-oxopropan-2-yl]hexanamide
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||||
| Activity |
Ki = 6400000 nM
|
[2] | |||
| Compound Name |
Methyl 3-(2-aminopropanoylamino)benzoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1161351; AKOS010503499
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||||
| Activity |
Ki = 6900000 nM
|
[4] | |||
| Compound Name |
H-D-Phe-Ala-OH
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Investigative | Compound Info | ||
| Synonyms |
D-phenylalanyl-L-alanine; d-phenyl-alanyl-l-alanine; L-Alanine, D-phenylalanyl-; CHEMBL2371838; SCHEMBL11113147; ZINC1605729; MFCD00672389; AKOS017461598
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||||
| Activity |
Ki = 7000000 nM
|
[2] | |||
| Compound Name |
L-Lysine, N2-D-alanyl-
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL364484; ZINC3014479; BDBM50169175; (S)-6-Amino-2-((R)-2-amino-propionylamino)-hexanoic acid; (2S)-6-amino-2-[[(2R)-2-aminopropanoyl]amino]hexanoic acid
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||||
| Activity |
Ki = 7000000 nM
|
[2] | |||
| Compound Name |
Lys-Arg
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Investigative | Compound Info | ||
| Synonyms |
Lysyl-Arginine; H-Lys-Arg-OH; L-lysyl-L-arginine; CHEMBL380183; L-Arginine, L-lysyl-; L-Lys-L-Arg; SCHEMBL288962; CTK0J9659; DTXSID00567683; ZINC5180993; BDBM50188532; L-Lysyl-N~5~-(diaminomethylidene)-L-ornithine; Q27144728
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||||
| Activity |
IC50 = 7200000 nM
|
[1] | |||
| Compound Name |
beta-Alanylglycine
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Investigative | Compound Info | ||
| Synonyms |
H-BETA-ALA-GLY-OH; beta-Ala-Gly; beta-Alanyl glycine; CHEMBL157332; [(3-ammoniopropanoyl)amino]acetate; H-b-Ala-Gly-OH; 2-(3-aminopropanoylamino)acetic acid; betaAla-Gly-OH; beta-alanyl-glycine; NSC89652; Glycine, b-alanyl-; .beta.-Alanylglycine; SCHEMBL2476159; CTK4F8423; DTXSID30181230; 2-(3-aminopropanamido)acetic acid; ZINC1575546; MFCD00025611; NSC-89652; [(3-aminopropanoyl)amino]acetic acid; MCULE-9256160395; DB-047007; FT-0634436; Q27144152
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||||
| Activity |
Ki = 7300000 nM
|
[4] | |||
| Compound Name |
Arg-arg
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Investigative | Compound Info | ||
| Synonyms |
Arginylarginine; L-arginyl-L-arginine; H-Arg-Arg-OH; CHEMBL296756; Arginyl-L-arginine; Arginyl-arginin; L-Arg-L-Arg; L-Arginine, L-arginyl-; L-Arginine, N2-L-arginyl-; SCHEMBL288599; CTK0H1982; DTXSID60165745; ZINC5706877; BDBM50188488; Q27144127; (S)-2-((S)-2-Amino-5-guanidinopentanamido)-5-guanidinopentanoic acid; 2-((S)-2-Amino-5-guanidino-1-oxo-pentylamino)-5-guanidino-pentanoic acid
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||||
| Activity |
IC50 = 7310000 nM
|
[1] | |||
| Compound Name |
2-Amino-N-(2-chlorophenyl)propanamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1161347; AKOS000186128
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||||
| Activity |
Ki = 7800000 nM
|
[4] | |||
| Compound Name |
(S)-2-[(S)-2-(2-Amino-propionylamino)-propionylamino]-propionic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL364278; BDBM50169224
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||||
| Activity |
Ki = 7900000 nM
|
[2] | |||
| Compound Name |
Arg-Lys
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Investigative | Compound Info | ||
| Synonyms |
L-Lysine, L-arginyl-; Arginyllysine; Arginyl-Lysine; H-Arg-Lys-OH; CHEMBL380024; L-arginyl-L-lysine; L-Arg-L-Lys; L-Arg-L-Lys-OH; SCHEMBL1067832; CTK1D5369; DTXSID80423793; ZINC4899463; BDBM50188520; HY-126487; CS-0104925; Q27144132
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||||
| Activity |
IC50 = 8110000 nM
|
[1] | |||
| Compound Name |
(3S)-3-Amino-4-oxo-4-[[(2R)-1-oxo-1-phenylmethoxypropan-2-yl]amino]butanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2372648; ZINC29400559
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||||
| Activity |
Ki = 8300000 nM
|
[4] | |||
| Compound Name |
H-Ala-Ala-D-Ala-OH
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL189476; CTK7F3243; L-ALANYL-ALANYL-D-ALANINE; ZINC2572099; BDBM50169135; (R)-2-((S)-2-((S)-2-aminopropanamido)propanamido)propanoic acid; (R)-2-[(S)-2-((S)-2-Amino-propionylamino)-propionylamino]-propionic acid
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||||
| Activity |
Ki = 8300000 nM
|
[2] | |||
| Compound Name |
4-[(2-Ammoniopropanoyl)amino]benzoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL157008; SCHEMBL5192071
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||||
| Activity |
Ki = 9100000 nM
|
[4] | |||
| Compound Name |
Tyr-Tyr-NH2
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL208922; BDBM50188494; ZINC53274750; (2S)-2-amino-N-[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-3-(4-hydroxyphenyl)propanamide
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||||
| Activity |
IC50 = 9110000 nM
|
[1] | |||
| Compound Name |
Pro-ala
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Investigative | Compound Info | ||
| Synonyms |
H-PRO-ALA-OH; L-prolyl-L-alanine; L-Alanine, L-prolyl-; Prolyl-Alanine; (S)-2-((S)-Pyrrolidine-2-carboxamido)propanoic acid; L-Pro-L-Ala; L-Pro-L-Ala-OH; CHEMBL293555; SCHEMBL2841482; CTK2F6866; ZINC4038298; 7228AH; KM0831; MFCD00037875; STL527372; AKOS010420673; MCULE-5153866058; Q27144880
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||||
| Activity |
Ki = 9500000 nM
|
[4] | |||
| Compound Name |
7-Aminocephalosporanic acid
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Investigative | Compound Info | ||
| Synonyms |
7-ACA; 7-Aminocephalosporinic acid; 7-ACS; 7beta-Aminocephalosporanic acid; UNII-9XI67897RG; (7R)-7-aminocephalosporanic acid; MFCD00005177; (7R)-7-Aminocephalosporanate; Cephalosporanic acid, 7-amino; 9XI67897RG; DSSTox_CID_25342; DSSTox_RID_80810; DSSTox_GSID_45342; 7-Aminocephalosporanic acid, 95-102%; CHEMBL1615585; NCGC00016552-01; Prestwick_714; EINECS 213-485-0; PubChem24166; Prestwick0_000424; Prestwick1_000424; Prestwick2_000424; Prestwick3_000424; 7-Aminocephalosporans??ure; Epitope ID:120362; EC 213-485-0; 7-amino cephalosporanic acid; SCHEMBL78638; BSPBio_000408; SPBio_002347; BPBio1_000450; 7beta-amino-cephalosporanic acid; DTXSID9045342; 7-Aminocephalosporanic Acid,(S); 7-beta-aminocephalosporanic acid;; 7-Aminocephalosporanic acid, 98%; HMS1569E10; HMS2096E10; HMS3713E10; (7R)-7-amino-cephalosporanic acid; BCP22888; EBD18443; HY-B1434; ZINC3861379; 7-AMINO-CEPHALOSPORANIC ACID; Tox21_110490; s2530; AKOS015951379; Tox21_110490_1; ACN-039962; CCG-220424; CS-4823; SMP2_000203; NCGC00179570-01; NCGC00179570-03; NCGC00263474-01; AC-24181; AS-15727; (6R,7R)-3-(acetoxymethyl)-7-amino-8-; AB0017588; B1652; oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-; C07756; J10226; M-1429; 3-Acetoxymethyl-7-amino-3-cephem-4-carbons??ure; 957A686; Q4642864; BRD-K65377893-001-01-7; 3-Acetoxymethyl-7beta-aminoceph-3-em-4-carboxylic acid; 7beta-amino-3-acetoxymethyl-3-cephem-4-carboxylic acid; (6R,7R)-3-acetoxymethyl-7-aminoceph-3-em-4-carboxylic acid; 3-acetoxymethyl-7beta-amino-3,4-didehydrocepham-4-carboxylic acid; 7-Aminocephalosporanic acid, Antibiotic for Culture Media Use Only
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||||
| Activity |
Ki > 10000000 nM
|
[14] | |||
| Compound Name |
Cefoxitin
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Investigative | Compound Info | ||
| Synonyms |
Mefoxin; CEPHOXITIN; Cefoxitina; Cefoxitine; Cefoxitinum; Rephoxitin; Mefoxitin; ceftoxitin; UNII-6OEV9DX57Y; Cenomycin; CHEMBL996; 6OEV9DX57Y; DSSTox_CID_2764; DSSTox_RID_76721; DSSTox_GSID_22764; MK-306; NCGC00183034-01; Cefoxotin; MK306; MFCD00072014; Spectrum_001399; Cefoxitin (USAN/INN); Prestwick0_000832; Prestwick1_000832; Prestwick2_000832; Prestwick3_000832; Spectrum2_000676; Spectrum3_001491; Spectrum4_000153; Spectrum5_001145; Epitope ID:116201; C06887; SCHEMBL15971; BSPBio_000783; BSPBio_003101; KBioGR_000626; KBioSS_001879; DivK1c_000576; SPBio_000771; SPBio_002704; BPBio1_000863; DTXSID1022764; GTPL10937; KBio1_000576; KBio2_001879; KBio2_004447; KBio2_007015; KBio3_002601; J01DC01; NINDS_000576; BCP09061; ZINC3830449; Tox21_113009; BDBM50335563; s5951; AKOS022185232; Tox21_113009_1; DB01331; DS-5384; IDI1_000576; NCGC00093351-06; AK118716; SC-65784; SBI-0051927.P002; AB0072765; D02345; 607C660; A822898; Q2353907
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||||
| Activity |
Ki = 10000000 nM
|
[2] | |||
| Compound Name |
Ceftazidime
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Investigative | Compound Info | ||
| Synonyms |
Tazidime; Pentacef; Tazicef; Ceptaz; Fortaz; ceftazidima; ceftazidimum; Fortum; Ceftazidime anhydrous; GR 20263; Tazidime In Plastic Container; Ceftazidime (INN); Fortaz (TN); SN 401; LY 139381; C22H22N6O7S2; GR-20263; LY-139381; Ceftazidime (TN); Ceptaz (TN); SCHEMBL36849; BIDD:GT0734; CHEMBL44354; DTXSID5022770; J01DD07; HMS2090M13; HY-B0593; BDBM50420259; AKOS015951273; CCG-269983; DB00438; NCGC00179584-05; CEFTAZIDIME (ARGININE FORMULATION); AB00513848; C06889; D07654; AB00513848-02; Cefprozil, Antibiotic for Culture Media Use Only; Q-200811
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||||
| Activity |
Ki > 10000000 nM
|
[14] | |||
| Compound Name |
Lysyllysine
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Investigative | Compound Info | ||
| Synonyms |
Lys-lys; L-Lysyl-L-lysine; Lysyl-Lysine; L-Lys-L-lys; H-Lys-Lys-OH; UNII-96TER1JROC; 96TER1JROC; CHEMBL379332; Dilysine; L-Lys-L-Lys-OH; L-Lysine, L-lysyl-; H-L-Lys-L-Lys-OH; L-Lysine, N(2)-L-lysyl-; SCHEMBL1070057; CTK0H8106; DTXSID00927364; ZINC2043137; BDBM50188512; N~2~-(2,6-Diamino-1-hydroxyhexylidene)lysine; Q27144740; UNII-96TER1JROC component NVGBPTNZLWRQSY-UWVGGRQHSA-N
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||||
| Activity |
IC50 = 10900000 nM
|
[1] | |||
| Compound Name |
1-(3-Thiazolidinyl)-2-amino-1-propanone
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1161341
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|
||||
| Activity |
Ki = 11000000 nM
|
[4] | |||
| Compound Name |
Metampicillin
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Investigative | Compound Info | ||
| Synonyms |
METHAMPICILLIN; UNII-G0H6U7VSTK; Magnipen; G0H6U7VSTK; METAMPICILLIN SODIUM; 6beta-[(2R)-2-(methylideneamino)-2-phenylacetamido]penicillanic acid; metampilene; Metampicillinum; Celinmicina; Elatocilline; Metampicilina; Metampicillina; Metampicilline; Pangocilin; Relyothenate; Blomopen; Bonopen; Filorex; Metambac; Micinovo; Probiotic; Ruticina; Rutizina; Sedomycin; Suvipen; Viderpen; Viderpin; Vioplex; Teonicon Trofen; Italcina kapseln; Suvipen ampullen; Rastomycin K; Meta-Alvar; Metiskia ampullen; Micinovo ampullen; Rutizina ampullen; Tampilen ampullen; Fedacilina kapseln; Metabacter ampullen; Metampicillina [DCIT]; Metampicilina [Spanish]; Metampicilline [French]; Metampicillinum [Latin]; Metampicillin [INN:DCF]; Metampicilina [INN-Spanish]; Metampicillinum [INN-Latin]; EINECS 229-365-6; Metampicillin (INN); (alpha-(Methyleneamino)benzyl)penicillin; CB 28020; D-(-)-alpha-Methyleneaminobenzylpenicillin; Prestwick0_000235; Prestwick1_000235; Prestwick2_000235; Prestwick3_000235; Epitope ID:141487; SCHEMBL34032; BSPBio_000309; SPBio_002230; BPBio1_000341; CHEMBL1908324; DTXSID5048479; ZINC3874216; BDBM50370588; DB13836; D07234; BRD-K83350436-236-03-4
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||||
| Activity |
Ki = 12700000 nM
|
[14] | |||
| Compound Name |
2-Amino-1-(piperidin-1-yl)propan-1-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
2-Amino-1-piperidin-1-yl-propan-1-one; 2-amino-1-piperidin-1-ylpropan-1-one; 1-methyl-2-oxo-2-piperidin-1-ylethylamine; 2-amino-1-piperidylpropan-1-one; SCHEMBL856280; CHEMBL1161340; CTK6A3026; 2-amino-1-piperidino-1-propanone; HMS1704C18; ALBB-007443; 9981AE; SBB002500; STK504546; AKOS000194671; AKOS016042350; MCULE-4421899149; Propan-1-one, 2-amino-1-piperidin-1-yl-; ST4094285; (1-methyl-2-oxo-2-piperidin-1-ylethyl)amine; EN300-45227; W-8379; Z44548922; (1-methyl-2-oxo-2-piperidin-1-ylethyl)amine(SALTDATA; F2147-1562
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||||
| Activity |
Ki = 12900000 nM
|
[4] | |||
| Compound Name |
H-D-Tyr-val-gly-OH
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL187443; D-Tyr-Val-Gly; d-tyrosylvalyl glycine; SCHEMBL7588275; ZINC2597013; BDBM50169158; MFCD00063349; 2-[[(2S)-2-[[(2R)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylbutanoyl]amino]acetic acid; {(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-butyrylamino}-acetic acid
Click to Show/Hide
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||||
| Activity |
Ki = 14000000 nM
|
[2] | |||
| Compound Name |
Tyrosyl-alanyl-glycine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
H-TYR-D-ALA-GLY-OH; CHEMBL190254; Tag peptide; SCHEMBL9724057; DTXSID20219793; ZINC2391106; BDBM50169185; MFCD00038703; Glycine, N-(N-L-tyrosyl-D-alanyl)-
Click to Show/Hide
|
||||
| Activity |
Ki = 14000000 nM
|
[2] | |||
| Compound Name |
2-Amino-N-benzylpropanamide
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL318725; 2-Amino-N-benzyl-DL-propanamide; 2-Amino-N-benzyl-propionamide; SCHEMBL6461987; BDBM50532874; KM3237; AKOS000172357; AKOS017263136; MCULE-6987327254; Propanamide, 2-amino-N-(phenylmethyl)-; H-193/12
Click to Show/Hide
|
||||
| Activity |
Ki = 14100000 nM
|
[4] | |||
| Compound Name |
7-[[(2S)-2-Azido-2-phenylacetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1161744
Click to Show/Hide
|
||||
| Activity |
Ki = 15000000 nM
|
[2] | |||
| Compound Name |
1-L-Alanyl-D-proline
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
UNII-1B9JC6P4Q5; 1B9JC6P4Q5; CHEMBL327608; l-alanyl-d-proline; H-Ala-Pro-OH; D-Proline, L-alanyl-; EINECS 262-343-4; SCHEMBL8316371; CTK5B1971; DTXSID20209452; (2R)-1-[(2S)-2-aminopropanoyl]pyrrolidine-2-carboxylic acid; ZINC1637976; BDBM50169194; AKOS017336994; W-108277; Q27896661; 1-((S)-2-Amino-propionyl)-pyrrolidine-2-carboxylic acid; (S)-1-((S)-2-Amino-propionyl)-pyrrolidine-2-carboxylic acid
Click to Show/Hide
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||||
| Activity |
Ki = 15000000 nM
|
[2] | |||
| Compound Name |
H-Pro-gly-gly-OH
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
Pro-gly-gly; Prolyl-glycyl-glycine; CHEMBL190343; 2-[[2-[[(2S)-pyrrolidine-2-carbonyl]amino]acetyl]amino]acetic acid; l-prolylglycylglycine; Pro-Gly-Gly-OH; Prolyl-glycyl-glycin; NSC 97937; Glycine,L-prolylglycyl-; L-Prolyl-glycyl-glycine; Glycine, L-prolylglycyl-; SCHEMBL10788841; CTK8D8729; Glycine, N-(N-L-prolylglycyl)-; ZINC4899450; 7229AH; BDBM50169143; MFCD00037877; AKOS010407662; 561P253; (S)-2-(2-(pyrrolidine-2-carboxamido)acetamido)acetic acid; {2-[(Pyrrolidine-2-carbonyl)-amino]-acetylamino}-acetic acid
Click to Show/Hide
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||||
| Activity |
Ki = 16000000 nM
|
[2] | |||
| Compound Name |
Pro-Lys
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Investigative | Compound Info | ||
| Synonyms |
L-Prolyl-L-lysine; Prolyl-Lysine; CHEMBL377325; H-Pro-Lys-OH; L-Pro-L-Lys; H-Pro-Lys-OHacetatesalt; SCHEMBL18075734; ZINC8076544; BDBM50188505; Q27144903
Click to Show/Hide
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||||
| Activity |
IC50 > 16000000 nM
|
[1] | |||
| Compound Name |
L-Prolylglycine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
H-PRO-GLY-OH; Prolylglycine; Pro-Gly; Prolyl-glycine; UNII-42521I3FYC; CHEMBL59426; L-Prolylgycine; 42521I3FYC; L-Prolyl-glycine; Pro-Gly-OH; 2-[[(2S)-pyrrolidine-2-carbonyl]amino]acetic acid; MFCD00022391; Glycine,l-prolyl-; (S)-Prolylglycine; L-Pro-Gly; Glycine, L-prolyl-; L-Pro-Gly-OH; SCHEMBL620067; CS-WAA0142; HY-WAA0142; CTK1A3975; ZINC4899418; 7230AH; BDBM50188480; CS-W017602; Glycine, N-L-prolyl- (8CI)(9CI); AS-56392; (S)-2-(pyrrolidine-2-carboxamido)acetic acid; [(Pyrrolidine-2-carbonyl)-amino]-acetic acid; K-6726; [((S)-Pyrrolidine-2-carbonyl)-amino]-acetic acid; Q27893792; 654E0B74-C991-4228-B739-3A3AB574E291
Click to Show/Hide
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||||
| Activity |
IC50 > 16000000 nM
|
[1] | |||
| Compound Name |
2-Amino-N-(2-phenylphenyl)propanamide
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Investigative | Compound Info | ||
| Synonyms |
N-biphenyl-2-ylalaninamide; SCHEMBL1752021; CHEMBL1161339; HMS1598J09; STK181752; AKOS005411682; MCULE-1962624659; SR-01000286421; SR-01000286421-1
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||||
| Activity |
Ki = 16600000 nM
|
[4] | |||
| Compound Name |
H-Ala-D-Ala-Ala-OH
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
H-Ala-D-Ala-L-Ala; CHEMBL361880; l-alanyl d-alanyl l-alanine; SCHEMBL12227547; ZINC2539572; BDBM50169209; MFCD00066037; (S)-2-((R)-2-((S)-2-aminopropanamido)propanamido)propanoic acid; (S)-2-[(R)-2-((S)-2-Amino-1-oxo-propylamino)-propionylamino]-propionic acid
Click to Show/Hide
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||||
| Activity |
Ki = 17000000 nM
|
[2] | |||
| Compound Name |
5-Aminovaleric acid
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Investigative | Compound Info | ||
| Synonyms |
5-Aminopentanoic acid; H-5-Ava-OH; delta-Aminovaleric acid; Homopiperidinic acid; 5-amino-pentanoic acid; Pentanoic acid, 5-amino-; Valeric acid, 5-amino-; delta-Amino-n-valeric acid; 5-aminopentanoate; 5-AMINO-N-VALERIC ACID; 5-Aminopentanoicacid; 5-aminovalerate; 5-ammoniopentanoate; MFCD00008232; .delta.-Aminovaleric acid; Delta-Aminovalerianic Acid; 5-Aminovaleric acid, 97%; .delta.-Amino-n-valeric acid; CHEMBL284116; Valeric acid, 5-amino- (8CI); Pentanoic acid, 5-amino- (9CI); delta-aminovalerate; delta-Amino-n-valerate; 5-Amino pentanoic acid; EINECS 211-544-5; NSC 58383; NSC 73123; DANVA; 5-amino valeric acid; 5-amino-valeric acid; PubChem18964; Spectrum_001627; ACMC-209nti; SpecPlus_000854; Spectrum2_001410; Spectrum3_001447; Spectrum4_001015; Spectrum5_001809; 5-AMINOVALERICACID; bmse000957; bmse000990; H-Ape(5)-OH; Lopac-194336; H2N(CH2)4COOH; NCIOpen2_000480; Valeric acid, (5-amino)-; Lopac0_000031; BSPBio_002913; KBioGR_001509; KBioSS_002107; DivK1c_006950; SCHEMBL190150; SPBio_001460; CTK3I9762; KBio1_001894; KBio2_002107; KBio2_004675; KBio2_007243; KBio3_002413; KS-00000UNB; DTXSID70216212; ACN-S002887; ACT10888; NSC58383; NSC73123; ZINC1532654; ANW-35140; BBL027702; BDBM50026409; LMFA01100040; NSC-58383; NSC-73123; SBB061559; STL257473; AKOS009140748; AM82459; CCG-204127; CS-W016594; HY-W015878; MCULE-4971679857; RS-1002; SDCCGSBI-0050020.P003; MLS-0412455; NCGC00014991-01; NCGC00014991-02; NCGC00014991-03; NCGC00014991-05; NCGC00162049-01; AK-78795; BP-13016; SC-10120; DB-054865; A0663; FT-0620031; ST45026838; C00431; M-3556; 660A888; Q11751639; F8889-6991; Z1262246173; F8D56633-B691-4612-9B69-981EF090A047
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||||
| Activity |
Ki = 17400000 nM
|
[4] | |||
| Compound Name |
H-Ala-D-Phe-Ala-OH
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2371837; ZINC2560936; (2S)-2-[[(2R)-2-[[(2S)-2-aminopropanoyl]amino]-3-phenylpropanoyl]amino]propanoic acid
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||||
| Activity |
Ki = 19000000 nM
|
[2] | |||
| Compound Name |
Cefodizime
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Investigative | Compound Info | ||
| Synonyms |
Cefodizima; Cefodizimum; UNII-Z31298J4HQ; HR 221 [AS SODIUM]; THR 221 [AS SODIUM]; Z31298J4HQ; S 77 1221 B [AS SODIUM]; THR-221; Cefodizime [INN:BAN]; Cefodizimum [INN-Latin]; Cefodizima [INN-Spanish]; Cefodizme; Diezime; Modivid; Timecef; Neucef; Cefodizime Acid; Cefodizime (INN); EC 700-301-3; HR-221 [As Sodium]; THR-221 [As Sodium]; SCHEMBL151101; CHEMBL2303613; DTXSID2022757; S-771221B [As Sodium]; EX-A1379; ZINC3871933; A0C261; BDBM50422690; HR-221; MFCD00864926; DB13470; HY-108402; CS-0028575; D07643; J-700161
Click to Show/Hide
|
||||
| Activity |
Ki = 22000000 nM
|
[2] | |||
| Compound Name |
D-Leucylglycylglycine
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
(R)-2-(2-(2-Amino-4-methylpentanamido)acetamido)acetic acid; D-Leucyl-glycyl-glycine; H-D-Leu-Gly-Gly-OH; CHEMBL1222388; 2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]acetic acid; (R)-2-(2-(2-Amino-4-methylpentanamido)-acetamido)acetic acid; N-(N-D-Leucylglycyl)glycine; Glycine, N-(N-D-leucylglycyl)-; EINECS 242-457-0; Glycine,D-leucylglycyl-; D-LEU-GLY-GLY; (([(2-Amino-4-methylpentanoyl)amino]acetyl)amino)acetic acid #; CTK4D9196; ZINC1575521; ANW-23273; BDBM50410267; MFCD00021740; 2-{2-[(2R)-2-Amino-4-methylpentanamido]acetamido}acetic acid; AKOS015854090; KS-0000138O; AS-70790; L0031; N-[(R)-2-Amino-4-methylpentanoyl]-Gly-Gly-OH; 625L224
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||||
| Activity |
Ki = 25000000 nM
|
[2] | |||
| Compound Name |
Oseltamivir phosphate
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Investigative | Compound Info | ||
| Synonyms |
Tamiflu; Oseltamivir (phosphate); UNII-4A3O49NGEZ; Ro 64-0796/002; GS 4104; 4A3O49NGEZ; GS4104; Oseltamir Phosphate; 204255-11-8 (phosphate); Osteltamivir phosphate; Oseltamivir phosphate, 98%; C16H28N2O4.H3PO4; SR-05000001499; MFCD08059548; Ebilfumin (TN); Oseltamivir phosphate [USAN:USP]; Tamiflu (TN); GS 4104 phosphate; SCHEMBL8730; cc-563; MLS006011559; CHEMBL1200340; DTXSID0044230; Oseltamivir phosphate (JAN/USP); BCPP000138; ACT03369; ABP000749; s2597; AKOS015896056; BCP9001033; CCG-230250; CS-0871; KS-1184; MCULE-3939535663; Oseltamivir phosphate, >=98% (HPLC); AC-25911; HY-17016; SMR004703323; AB0011433; GS-4104/002; Ro-64-0796-002; Ro-64-0796/002; C08093; D00900; J10429; W-5362; 255O118; SR-05000001960; J-013302; J-523838; SR-05000001499-2; SR-05000001960-1; Q27107588; Z1550675456; BENZOFURAN-3-YL-(3-BOC-AMINO-AZETIDIN-1-YL)-ACETICACID; Oseltamivir phosphate, United States Pharmacopeia (USP) Reference Standard
Click to Show/Hide
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||||
| Activity |
IC50 = 27400000 nM
|
[19] | |||
| Compound Name |
Cefsulodin sodium salt
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL3351077; BDBM50282169; SDCCGSBI-0050247.P002
Click to Show/Hide
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||||
| Activity |
Ki > 30000000 nM
|
[14] | |||
| Compound Name |
Cefpirome
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
Cefpiroma; Cefpiromum; Cefrom; HR 810; UNII-S72Q2F09HY; cefpirome sulfate; S72Q2F09HY; Cefpiromum [Latin]; Cefpiroma [Spanish]; Cefpirome [INN:BAN]; HR-810; cefpirome sulphate; NCGC00181339-01; C22H22N6O5S2; Cerfpirome; Broact; Keiten; Cefpirome (INN); Cefir (TN); HR-810 FREE BASE; SCHEMBL49406; cc-319; MLS006010792; CHEMBL65794; DTXSID2048244; SCHEMBL22207951; AKOS016013926; DB13682; SMR004701476; C11199; D07649
Click to Show/Hide
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||||
| Activity |
Ki > 30000000 nM
|
[2] | |||
| Compound Name |
Acetylalanylalanine
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Investigative | Compound Info | ||
| Synonyms |
AC-ALA-ALA-OH; (2S)-2-[[(2S)-2-acetamidopropanoyl]amino]propanoic acid; Ac-D-Ala-D-ala; Acetyl-ala-ala; N-acetylalanylalanine; N-Acetyl-Ala-Ala-OH; Alanine, N-acetylalanyl-; Acetyl-D-alanyl-D-alanine; Ac-Ala-Ala-OH, AldrichCPR; SCHEMBL291483; CHEMBL2372592; CTK2C7754; DTXSID40173808; ZINC2572098; MFCD00080977; D-Alanine, N-(N-acetyl-D-alanyl)-; (S)-2-((S)-2-acetamidopropanamido)propanoic acid
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||||
| Activity |
Ki > 30000000 nM
|
[4] | |||
| Compound Name |
D-Alanyl-D-alanine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
D-ALA-D-ALA; (R)-2-((R)-2-Aminopropanamido)propanoic acid; H-D-Ala-D-Ala-OH; D-Alanine, D-alanyl-; D-Ala-D-Ala-OH; UNII-1BVK9QMW8G; 1BVK9QMW8G; (D-Ala)2; Alanylalanine; CHEMBL299420; D-Alaninyl-D-alanine; (2R)-2-[[(2R)-2-aminopropanoyl]amino]propanoic acid; AA dipeptide; A-A Dipeptide; Dialanine, D,D-; Alanine Alanine dipeptide; Alanine-Alanine dipeptide; Epitope ID:141113; SCHEMBL476353; CTK3I8002; DTXSID601016947; KS-00000Y9O; ZINC1532807; BDBM50022571; KM3090; MFCD00066038; AKOS016843636; AS-57348; SC-90279; C00993; (2R)-2-[(2R)-2-aminopropanamido]propanoic acid; 923A160; Q27101980; UNII-37AOH3N58S component DEFJQIDDEAULHB-QWWZWVQMSA-N; UNII-3EE68A29TN component DEFJQIDDEAULHB-QWWZWVQMSA-N
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||||
| Activity |
Ki > 30000000 nM
|
[2] | |||
| Compound Name |
Cefotaxime
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Investigative | Compound Info | ||
| Synonyms |
Cephotaxime; Cefotaxime acid; E-cefotaxime; UNII-N2GI8B1GK7; Cefotaximum; Cefotaxima; N2GI8B1GK7; Omnatax; Taxim; HR 756; Cefotaxime [INN:BAN]; RU 24756; Cefotaximum [INN-Latin]; Cefotaxima [INN-Spanish]; Cefotaxime (INN); EINECS 264-299-1; Cefotaxim Hikma (TN); RU 24662; Prestwick2_000139; Prestwick3_000139; Claforan (*Sodium salt*); CHEMBL1730; Lopac0_000278; BSPBio_000218; BPBio1_000240; SCHEMBL3731931; DTXSID6022761; HY-A0088A; HMS2090M11; ZINC3830437; AC-217; BDBM50482777; MFCD00864971; s4720; AKOS015951267; DB00493; SDCCGSBI-0050266.P002; AS-12690; clo[4.2.0]oct-2-ene-2-carboxylic acid; CS-0013515; C06885; D07647; J90010; 527C526; BRD-K78364995-236-03-5; Q27262497; Di- poundg-chlorotetrakis[2,4-dimethyl-6-(2-quinolinyl-KN)phenyl-KC]di-iridium
Click to Show/Hide
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||||
| Activity |
Ki > 30000000 nM
|
[2] | |||
| Compound Name |
D-Lysine, N2-D-alanyl-
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL190049; ZINC3014483; BDBM50169146; (R)-6-Amino-2-((R)-2-amino-propionylamino)-hexanoic acid
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||||
| Activity |
Ki > 30000000 nM
|
[2] | |||
| Compound Name |
3-(3-Aminopropanoylamino)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
H-BETA-ALA-BETA-ALA-OH; beta-Alanine, N-beta-alanyl-; beta-Alanyl-beta-alanine; 3-(3-aminopropanamido)propanoic acid; CHEMBL153975; 3-[(3-ammoniopropanoyl)amino]propanoate; NSC97926; beta-Ala-beta-Ala-OH; b-Alanine,N-b-alanyl-; .beta.-Ala-.beta.-Ala; N-(beta-Alanyl)-beta-alanine; SCHEMBL2897506; CTK1A5862; DTXSID00294760; N-(3-aminopropanoyl)-beta-alanine; ZINC1637971; 7080AH; MFCD00038199; NSC-97926; STL522404; AKOS010403808; MCULE-9840310477; AM803512; AS-39424; FT-0694084; K-6124
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||||
| Activity |
Ki > 30000000 nM
|
[4] | |||
| Compound Name |
D-Proline, D-alanyl-
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL365196; D-alanyl-D-proline; D-Proline, 1-D-alanyl-; SCHEMBL9164453; CTK0D2278; ZINC1637977; BDBM50169137; AKOS017337085; (R)-1-((R)-2-Aminopropanoyl)pyrrolidine-2-carboxylic acid; (R)-1-((R)-2-Amino-propionyl)-pyrrolidine-2-carboxylic acid
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|
||||
| Activity |
Ki > 30000000 nM
|
[2] | |||
| Compound Name |
L-Alanyl-D-lysine
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2096813; D-Lysine, L-alanyl-; ZINC3014482; BDBM50410266
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||||
| Activity |
Ki > 30000000 nM
|
[2] | |||
| Compound Name |
Boc-ala-ala-OH
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|
Investigative | Compound Info | ||
| Synonyms |
L-Alanine, N-[(1,1-dimethylethoxy)carbonyl]-L-alanyl-; Boc-L-Ala-L-ala; L-Alanine,N-[(1,1-dimethylethoxy)carbonyl]-L-alanyl-; boc-alanyl-alanine; Boc-(Ala)2-OH; Boc-Ala-Ala-OH, AldrichCPR; SCHEMBL6891888; CHEMBL2371142; CTK4F9468; KS-00000FSI; ZINC1576305; 6260AH; MFCD00038564; AKOS027340118; (tert-Butoxycarbonyl)-L-alanyl-L-alanine; DS-12425; SC-91700; N-tert-butyloxycarbonyl-L-alanyl-L-alanine; CS-0097837; K-6962; (S)-2-((S)-2-(tert-butoxycarbonylamino)propanamido)propanoic acid
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||||
| Activity |
Ki > 30000000 nM
|
[4] | |||
| Compound Name |
6-Aminopenicillanic acid
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Investigative | Compound Info | ||
| Synonyms |
6-Apa; Penicin; Penin; Aminopenicillanic acid; 6-Aps; Phenacyl 6-aminopenicillinate; 6-Aminopenicillamine acid; (+)-6-Aminopenicillanic acid; UNII-QR0C4R7XVN; 6-aminopenicillanate; AI3-52557; MFCD00005176; QR0C4R7XVN; 6beta-aminopenicillanic acid; CHEMBL1236749; 6-amino-2,2-dimethylpenam-3alpha-carboxylic acid; SR-01000640154-1; 6-Aminopenicillanic acid, 96%; 6-Aminopenicillanicacid; EINECS 208-993-4; NSC 50071; NCGC00160198-01; amino penicillanic acid; 6-amino-penicillanic acid; 6-aminopenici llanic acid; bmse000312; Epitope ID:117703; EC 208-993-4; Sulbactam Impurity B (Amoxicillin Impurity A); DSSTox_CID_26097; DSSTox_RID_81336; DSSTox_GSID_46097; SCHEMBL66332; Amoxicillin Related Compound A; DTXSID7046097; 09070_FLUKA; 6-aminopenicillinic acid (6-APA); BCP13375; STR03060; ZINC3860188; Tox21_111749; BDBM50420257; CCG-50809; s5035; (+)-6-Aminopenicillanic acid, 96%; AKOS015907713; CS-W014265; EBD2197937; HY-W013549; KS-5277; MCULE-7780131013; VZ30646; AC-11282; BR-26116; SC-19462; A0800; C02954; M-5489; (+)-6-Aminopenicillanic acid, analytical standard; Q2823234; W-105586; 6beta-amino-2,2-dimethylpenam-3alpha-carboxylic acid; Z1741972222; (3S,5R,6R)-6-amino-2,2-dimethylpenam-3-carboxylic acid; (3S, 5R, 6R)-6-amino-2,2-dimethylpenam-3-carboxylic acid; Flucloxacillin impurity C, European Pharmacopoeia (EP) Reference Standard
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||||
| Activity |
Ki > 30000000 nM
|
[14] | |||
| Compound Name |
{Methyl[(methylammonio)acetyl]amino}acetate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL346341; BDBM50136974
Click to Show/Hide
|
||||
| Activity |
Ki = 32000000 nM
|
[4] | |||
| Compound Name |
(2S)-2-[[(2S,5S)-5-Amino-2-(benzoyloxymethyl)-4-oxo-6-phenylhexanoyl]amino]-2-cyclohexylacetic acid;2,2,2-trifluoroacetic acid
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1807354
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|
||||
| Activity |
Ki = 46773514.13 nM
|
[20] | |||
| Compound Name |
(2S)-2-[[(2S)-2-[[(2S)-2-Amino-3-phenylpropanoyl]amino]-3-benzoyloxypropanoyl]amino]pentanoic acid;2,2,2-trifluoroacetic acid
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1807356
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|
||||
| Activity |
Ki = 123026877.1 nM
|
[20] | |||
| Compound Name |
(2S)-2-[[(2S)-2-[[(2S)-2-Amino-3-phenylpropanoyl]amino]-3-benzoyloxypropanoyl]amino]-2-cyclohexylacetic acid;2,2,2-trifluoroacetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1807357
Click to Show/Hide
|
||||
| Activity |
Ki = 245470891.6 nM
|
[20] | |||
| Compound Name |
(2S)-2-[[(2S,5S)-5-Amino-2-(benzoyloxymethyl)-4-oxo-6-phenylhexanoyl]amino]pentanoic acid;2,2,2-trifluoroacetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1807353
Click to Show/Hide
|
||||
| Activity |
Ki = 251188643.2 nM
|
[20] | |||
| Compound Name |
Phe-Ser-Ala
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1807351; Phenylalanyl-seryl-alanine; L-Phenylalanyl-L-seryl-L-alanine; BDBM50418931; (2S)-2-[[(2S)-2-[[(2S)-2-amino-3-phenylpropanoyl]amino]-3-hydroxypropanoyl]amino]propanoic acid
Click to Show/Hide
|
||||
| Activity |
Ki = 257039578.3 nM
|
[20] | |||
| Compound Name |
(2S)-2-[[(2S,5S)-5-Amino-2-(benzoyloxymethyl)-4-oxo-6-phenylhexanoyl]amino]propanoic acid;2,2,2-trifluoroacetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1807352
Click to Show/Hide
|
||||
| Activity |
Ki = 323593656.9 nM
|
[20] | |||
| Click to Show/Hide the Information of All Non Binders | |||||
| References | Top | ||||
|---|---|---|---|---|---|
| REF 1 | Human PEPT1 pharmacophore distinguishes between dipeptide transport and binding. J Med Chem. 2006 Jun 15;49(12):3636-44. | ||||
| REF 2 | Three-dimensional quantitative structure-activity relationship analyses of beta-lactam antibiotics and tripeptides as substrates of the mammalian H+/peptide cotransporter PEPT1. J Med Chem. 2005 Jun 30;48(13):4410-9. | ||||
| REF 3 | Identification of diarylsulfonamides as agonists of the free fatty acid receptor 4 (FFA4/GPR120). Bioorg Med Chem Lett. 2014 Jul 15;24(14):3100-3. | ||||
| REF 4 | Three-dimensional quantitative structure-activity relationship analyses of peptide substrates of the mammalian H+/peptide cotransporter PEPT1. J Med Chem. 2003 Dec 18;46(26):5725-34. | ||||
| REF 5 | Human dipeptide transporter, hPEPT1, stably transfected into Chinese hamster ovary cells. Pharm Res. 1996 Nov;13(11):1631-4. | ||||
| REF 6 | Dipeptidomimetic ketomethylene isosteres as pro-moieties for drug transport via the human intestinal di-/tripeptide transporter hPEPT1: design, synthesis, stability, and biological investigations. J Med Chem. 2004 Sep 9;47(19):4755-65. | ||||
| REF 7 | Proton/peptide cotransporter (PEPT 2) from human kidney: functional characterization and chromosomal localization. Biochim Biophys Acta. 1995 Nov 22;1240(1):1-4. | ||||
| REF 8 | Amino acid ester prodrugs of the antiviral agent 2-bromo-5,6-dichloro-1-(beta-D-ribofuranosyl)benzimidazole as potential substrates of hPEPT1 transporter. J Med Chem. 2005 Feb 24;48(4):1274-7. | ||||
| REF 9 | Structural requirements for the substrates of the H+/peptide cotransporter PEPT2 determined by three-dimensional quantitative structure-activity relationship analysis. J Med Chem. 2006 Jul 13;49(14):4286-96. | ||||
| REF 10 | Differential recognition of beta -lactam antibiotics by intestinal and renal peptide transporters, PEPT 1 and PEPT 2. J Biol Chem. 1995 Oct 27;270(43):25672-7. | ||||
| REF 11 | 5'-Amino acid esters of antiviral nucleosides, acyclovir, and AZT are absorbed by the intestinal PEPT1 peptide transporter. Pharm Res. 1998 Aug;15(8):1154-9. | ||||
| REF 12 | Transport characteristics of differently charged cephalosporin antibiotics in oocytes expressing the cloned intestinal peptide transporter PepT1 and in human intestinal Caco-2 cells. J Pharmacol Exp Ther. 1996 May;277(2):831-9. | ||||
| REF 13 | CHO/hPEPT1 cells overexpressing the human peptide transporter (hPEPT1) as an alternative in vitro model for peptidomimetic drugs. J Pharm Sci. 1999 Mar;88(3):347-50. | ||||
| REF 14 | Interaction of 31 beta-lactam antibiotics with the H+/peptide symporter PEPT2: analysis of affinity constants and comparison with PEPT1. Eur J Pharm Biopharm. 2005 Jan;59(1):17-24. | ||||
| REF 15 | Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism. J Control Release. 2003 Jan 17;86(2-3):279-92. | ||||
| REF 16 | Evidence for the absolute conformational specificity of the intestinal H+/peptide symporter, PEPT1. J Biol Chem. 1998 Feb 13;273(7):3861-4. | ||||
| REF 17 | Enhancing the intestinal absorption of molecules containing the polar guanidino functionality: a double-targeted prodrug approach. J Med Chem. 2010 Jan 28;53(2):624-32. | ||||
| REF 18 | In vitro characterization of human peptide transporter hPEPT1 interactions and passive permeation studies of short cationic antimicrobial peptides. J Med Chem. 2011 Apr 14;54(7):2422-32. | ||||
| REF 19 | Species-dependent uptake of glycylsarcosine but not oseltamivir in Pichia pastoris expressing the rat, mouse, and human intestinal peptide transporter PEPT1. Drug Metab Dispos. 2012 Jul;40(7):1328-35. | ||||
| REF 20 | The tandem chain extension aldol reaction used for synthesis of ketomethylene tripeptidomimetics targeting hPEPT1. Bioorg Med Chem Lett. 2011 Aug 1;21(15):4597-601. | ||||
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