Target Pair Drug Name
5HT1b --- SERT 3-(3,4-Diacetyl-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester Drug Info
5LOX --- HRH1 1-(4-{4-[2-(4-{13-chloro-4-azatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-ylidene}piperidin-1-yl)ethoxy]phenyl}but-3-yn-1-yl)-1-hydroxyurea Drug Info
ADRA1A --- HRH1 DROPERIDOL Drug Info
ADRA1A --- HRH1 CHEMBL2068762 Drug Info
ADRA1A --- HRH1 2-({(2R)-1-[4-(4-{[3-(Hexahydro-1H-azepin-1-yl)propyl]oxy}phenyl)butyl]-2-pyrrolidinyl}methyl)-4-[(4-hydroxyphenyl)methyl]-1(2H)-phthalazinone Drug Info
CABL --- Ckit PD-0173956 Drug Info
CABL --- MCSF Sunitinib Drug Info
CAI --- CAIX Zonisamide Drug Info
Aurora --- VEGFR N-(4-(benzo[d]thiazol-2-yl)phenyl)-4-(4-methylpiperazin-1-yl)pyrimidin-2-amine Drug Info
AuroraA --- STK1 N-(6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl)-3-((4-(methylsulfonyl)piperazin-1-yl)methyl)isothiazol-5-amine Drug Info
AuroraA --- STK1 N-(3-(1H-pyrazol-4-yl)-6-(trifluoromethyl)imidazo[1,2-a]pyrazin-8-yl)-3-methylisothiazol-5-amine Drug Info
AuroraA --- STK1 N-(3-(1-methyl-1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl)-3-(piperidin-4-yl)isothiazol-5-amine Drug Info
AuroraA --- STK1 (Z)-5-(Indolin-1-ylsulfonyl)-3-{[3-(3-morpholino-3-oxopropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-2-yl]methylene}indolin-2-one Drug Info
AuroraA --- STK1 N-(6-(ethylthio)-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl)-3-methylisothiazol-5-amine Drug Info
AuroraA --- STK1 2-(2-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinazolin-4-yl]amino}-1,3-thiazol-5-yl)-N-(3-methylbutyl)acetamide Drug Info
AuroraA --- STK1 5-(6-methoxy-7-(3-morpholinopropoxy)quinazolin-4-ylamino)-N-phenylthiophene-2-carboxamide Drug Info
AuroraA --- STK1 3-(8-oxa-5-azaspiro[3.5]nonan-5-ylmethyl)-N-(6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl)isothiazol-5-amine Drug Info
B1R --- B2R D-Arg-Arg-Pro-Hyp-Gly-Thi-Ser-Pro(4-0-n-Propyl)-pro(2,3-dihexyl)-arg Drug Info
Beta PDGFR --- CD135 CHEMBL1940272 Drug Info
BNOS --- Hepatocyte NOS 2-Ethyl-1-(4-hydroxy-phenyl)-isothiourea; hydriodide Drug Info
BNOS --- Hepatocyte NOS 4-chloro-2-((isopropyl(piperidin-4-yl)amino)methyl)benzonitrile Drug Info
BNOS --- Hepatocyte NOS 2-((azepan-4-yl(methyl)amino)methyl)-4-chlorobenzonitrile Drug Info
BNOS --- Hepatocyte NOS 6-Isopropyl-4-methyl-pyridin-2-ylamine Drug Info
BNOS --- Hepatocyte NOS Hexahydro-cyclopenta[c]pyrrol-(1Z)-ylideneamine Drug Info
BNOS --- Hepatocyte NOS 5-Butyl-4-methyl-pyrrolidin-(2E)-ylideneamine; hydrochloride Drug Info
BNOS --- Hepatocyte NOS SID56462977 Drug Info
BNOS --- Hepatocyte NOS (3aR,9bS)-8-Chloro-7-[2-(3-chloro-benzylamino)-ethyl]-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-ylamine Drug Info
BNOS --- Hepatocyte NOS SID11113814 Drug Info
BNOS --- Hepatocyte NOS 6-{4-[2-(4-Dimethylamino-piperidin-1-yl)-ethoxy]-naphthalen-1-yl}-pyridin-2-ylamine Drug Info
5HT1a --- SERT 1-phenyl-3-(4-(pyrimidin-2-yl)piperazin-1-yl)propan-1-ol Drug Info
5HT1a --- SERT [2-(5-Fluoro-2-methoxy-phenoxy)-ethyl]-[2-(1H-indol-3-yl)-ethyl]-amine Drug Info
5HT1a --- SERT (S)-1-(1H-Indol-4-yloxy)-3-[4-(4-isopropoxy-benzo[b]thiophen-2-yl)-piperidin-1-yl]-propan-2-ol Drug Info
5HT1b --- SERT N-[3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)propyl]-N-methylamine Drug Info
AChE --- NMDA SID124882535 Drug Info
ADRA1A --- HRH1 N-((cis)-4-(4-(dimethylamino)-5-methylpyrimidin-2-ylamino)cyclohexyl)-3-methylbenzamide Drug Info
ADRA1A --- HRH1 7-[3-(4-Benzhydryl-piperidin-1-yl)-propyl]-1,3-dimethyl-3,7-dihydro-purine-2,6-dione; compound with (E)-but-2-enedioic acid Drug Info
ADRA1A --- HRH1 2,8-dimethyl-5-phenethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole Drug Info
CABL --- Ckit Sunitinib Drug Info
CABL --- TEK WYE-130600 Drug Info
Aurora --- GSK 4-[4-(3-Hydroxy-adamantan-1-ylamino)-5-nitro-pyrimidin-2-ylamino]-benzoic acid Drug Info
AuroraA --- CDK4 N-4-4-methylpiperazin-1-yl-phenyl-7-3-methylsulfonyl-phenyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine Drug Info
AuroraA --- STK1 PHA-680632 Drug Info
AuroraA --- STK1 1-phenyl-3-(5-(2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl)thiazol-2-yl)urea Drug Info
AuroraA --- STK1 N-(3-fluorophenyl)-2-{2-[(7-{3-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]propoxy}-6-methoxyquinazolin-4-yl)amino]-1,3-thiazol-5-yl}acetamide Drug Info
AuroraA --- STK1 2-[3-(4-{[(Phenylamino)carbonyl]amino}phenyl)-4-(1H-pyrrolo-[2,3-b]pyridin-4-yl)-1H-pyrazol-1-yl]acetamide Drug Info
AuroraA --- STK1 1-(4-((5-(6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-ylamino)isothiazol-3-yl)methyl)piperazin-1-yl)ethanone Drug Info
AuroraA --- STK1 5-Ethyl-7,7-dimethyl-2-(5-methyl-1H-pyrazol-3-yl)-6-oxo-1Himidazo[4,5-f]indole Drug Info
AuroraA --- STK1 CHEMBL424899 Drug Info
AuroraA --- STK1 N-(4-(4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidin-2-ylthio)phenyl)acetamide Drug Info
CDK1 --- Cyclin E Purvalanol A Drug Info

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