Multi-target agents
Target Pair | Drug Name | |
---|---|---|
5HT1a --- SERT | [3-(5-Fluoro-1H-indol-3-yl)-propyl]-[2-(5-fluoro-2-methoxy-phenoxy)-ethyl]-amine | Drug Info |
5HT1a --- SERT | [2-(1H-Benzoimidazol-4-yloxy)-ethyl]-[3-(5-fluoro-1H-indol-3-yl)-propyl]-amine | Drug Info |
5HT1b --- SERT | 4'-Carbamimidoyl-2'-methyl-biphenyl-4-carboxylic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide | Drug Info |
AChE --- COX | SID11111897 | Drug Info |
ADRA1A --- HRH1 | 4-[(4-Methylphenyl)methyl]-2-{[(2R)-1-methyl-2-pyrrolidinyl]methyl}-1(2H)-phthalazinone | Drug Info |
ADRA1A --- HRH1 | SID26749206 | Drug Info |
ADRA1A --- HRH1 | OLANZAPINE_2-HYDROXYMETHYL METABOLITE | Drug Info |
CABL --- Ckit | AZD0530 | Drug Info |
CABL --- STK1 | VX-680 | Drug Info |
Aurora --- GSK | 4-(3-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-ylamino)benzoic acid | Drug Info |
AuroraA --- CD135 | N1-3-[5-(2-Methyl-6-[(3-morpholinopropyl)amino]-4-pyrimidinylamino)-1H-3-pyrazolyl]phenyl-1-benzenesulfonamide | Drug Info |
AuroraA --- STK1 | N-{4-[1-(3-Hydroxypropyl)-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}-N'-phenylurea | Drug Info |
AuroraA --- STK1 | (Z)-N-Methyl-3-(4-oxo-2-{[2-oxo-5-(phenylsulfonamido)-indolin-3-ylidene]methyl}-4,5,6,7-tetrahydro-1H-indol-3-yl)-propanamide | Drug Info |
AuroraA --- STK1 | (R)-4-(4-methylpiperazin-1-yl)-N-(5-(2-phenylpropanoyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)benzamide | Drug Info |
AuroraA --- STK1 | tert-butyl 4-(4-(5-methyl-1H-pyrazol-3-ylamino)quinazolin-2-ylthio)phenylcarbamate | Drug Info |
AuroraA --- STK1 | (S)-4-(2-amino-6-(3-amino-1H-indazol-6-yl)pyrimidin-4-yl)-N-phenylmorpholine-2-carboxamide | Drug Info |
AuroraA --- STK1 | Deuterated 6-Methyl-3-(1H-pyrazol-4-tl)-N-[3-[[(3,3,3-trifluoropropyl)amino]methyl-(d2)]-5-isothiazolyl]imidazo[1,2-a]pyrazin-8-amine Hydrochloride | Drug Info |
AuroraA --- STK1 | 3-((2,2-dimethylpiperidin-1-yl)methyl)-N-(6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl)isothiazol-5-amine | Drug Info |
AuroraA --- STK1 | 4-methyl-N-(3-(2-(5-(methylsulfonamido)-6-(pyrrolidin-1-yl)-1H-indazol-3-yl)vinyl)phenyl)piperazine-1-carboxamide | Drug Info |
CDK1 --- Cyclin E | R-roscovitine | Drug Info |
Beta PDGFR --- Ckit | 4-[6-Methoxy-7-(2-pyrrolidin-1-yl-ethoxy)-quinazolin-4-yl]-piperazine-1-carbothioic acid (furan-2-ylmethyl)-amide | Drug Info |
BNOS --- Hepatocyte NOS | 2-(2-(1H-imidazol-1-yl)-6-methylpyrimidin-4-yl)-N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)pyrrolidine-1-carboxamide | Drug Info |
BNOS --- Hepatocyte NOS | 6-{7-[2-(4-Methyl-piperazin-1-yl)-ethoxy]-indan-4-yl}-pyridin-2-ylamine | Drug Info |
BNOS --- Hepatocyte NOS | 2-Amino-3-(2-guanidino-phenyl)-propionic acid | Drug Info |
BNOS --- Hepatocyte NOS | 5,6-Dimethyl-pyridin-2-ylamine | Drug Info |
BNOS --- Hepatocyte NOS | SID124880731 | Drug Info |
BNOS --- Hepatocyte NOS | 5-Imino-3-methyl-2-pentyl-pyrrolidinium; chloride | Drug Info |
BNOS --- Hepatocyte NOS | N-(3-Aminomethyl-phenyl)-furan-2-carboxamidine | Drug Info |
BNOS --- Hepatocyte NOS | N1-(3-(1H-imidazol-1-yl)-1,2,4-thiadiazol-5-yl)-N3-(benzo[d][1,3]dioxol-5-ylmethyl)-N1-(thiophen-2-ylmethyl)propane-1,3-diamine | Drug Info |
BNOS --- Hepatocyte NOS | 3-Methyl-pyridin-2-ylamine | Drug Info |
CAI --- CAIX | SID144212941 | Drug Info |
5HT1a --- SERT | (S)-1-(1H-Indol-4-yloxy)-3-[4-(7-methoxy-benzo[b]thiophen-2-yl)-piperidin-1-yl]-propan-2-ol | Drug Info |
5HT1a --- SERT | 3-(4-(2-methoxyphenyl)piperazin-1-yl)-1-phenylpropan-1-one | Drug Info |
5HT1a --- SERT | (S)-1-(1H-Indol-4-yloxy)-3-[4-(6-methoxy-3-methyl-benzo[b]thiophen-2-yl)-piperidin-1-yl]-propan-2-ol | Drug Info |
5HT1a --- SERT | 6-{1-[2-(Quinolin-5-yloxy)-ethyl]-pyrrolidin-3-ylmethoxy}-4H-benzo[1,4]oxazin-3-one | Drug Info |
5LOX --- HRH1 | 1-{4-[4-(2-{4-[bis(4-fluorophenyl)methyl]piperazin-1-yl}ethoxy)phenyl]but-3-yn-1-yl}-1-hydroxyurea | Drug Info |
ADRA1A --- HRH1 | (R)-4-(3,4-Difluoro-phenyl)-1,2-dimethyl-6-oxo-1,4,5,6-tetrahydro-pyridine-3-carboxylic acid {3-[4-(2-cyano-4-fluoro-phenyl)-piperidin-1-yl]-propyl}-amide | Drug Info |
ADRA1A --- HRH1 | N-((cis)-4-(4-(dimethylamino)-6-methylpyrimidin-2-ylamino)cyclohexyl)-3,5-bis(trifluoromethyl)benzamide | Drug Info |
ADRA1A --- HRH1 | 4-(3,4-Difluoro-phenyl)-5-methyl-2-oxo-oxazolidine-3-carboxylic acid {3-[4-(4-fluoro-phenyl)-piperidin-1-yl]-propyl}-amide | Drug Info |
ADRA1A --- HRH1 | trans-1-benzyl-3-dimethylamino-6-phenylpiperidine | Drug Info |
CABL --- FGFR1 | ENMD-2076 | Drug Info |
CAI --- CAIX | Estradiol 3,17-O,O-bis-sulfamate | Drug Info |
Aurora --- VEGFR | 6-methoxy-2-(4-(2-(pyridin-3-yl)vinyl)-1H-pyrazol-3-yl)-1H-benzo[d]imidazole | Drug Info |
AuroraA --- CDK4 | 2-3-7-cyclohexyl-7H-pyrrolo[2,3-d]pyrimidin-2-ylamino-phenyl-acetic acid | Drug Info |
AuroraA --- STK1 | CHEMBL385049 | Drug Info |
AuroraA --- STK1 | N-(2-(2-(1H-benzo[d]imidazol-2-ylamino)thiazol-5-yl)ethyl)thieno[3,2-d]pyrimidin-4-amine | Drug Info |
AuroraA --- STK1 | (3S,6R)-1-[2-Amino-6-(3-amino-1H-indazol-6-yl)-4-pyrimidinyl]-N-cyclohexyl-6-methyl-3-piperidinecarboxamide | Drug Info |
AuroraA --- STK1 | (Z)-3-(2-{[5-(N,N-Dimethylsulfamoyl)-2-oxoindolin-3-ylidene]-methyl}-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)propanoic Acid | Drug Info |
AuroraA --- STK1 | 4-(5-Methyl-1H-pyrazol-3-ylamino)-2-(4-nitrobenzyl)-2Hphthalazin-1-one | Drug Info |
AuroraA --- STK1 | N-2-fluorophenyl-2-3-7-3-4-hydroxymethyl-piperidin-1-yl-propoxy-6-methoxyquinazolin-4-ylamino-1H-pyrazol-5-yl-acetamide | Drug Info |
Pagination
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