Target Information
Target General Infomation | |||||
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Target ID |
T51487
|
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Former ID |
TTDS00403
|
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Target Name |
Gamma-aminobutyric acid receptor subunit alpha-1
|
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Gene Name |
GABRA1
|
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Synonyms |
GABA(A) receptor subunit alpha-1; GABRA1
|
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Target Type |
Successful
|
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Disease | Anxiety disorder [ICD9: 300, 311; ICD10: F32, F40-F42] | ||||
Anesthesia [ICD9: 338; ICD10: R20.0] | |||||
Depression [ICD9: 311; ICD10: F30-F39] | |||||
Epilepsy; Anxiety disorder [ICD9: 300, 345; ICD10: F40-F42, G40] | |||||
Epilepsy [ICD10: G40] | |||||
Epileptic seizures [ICD9: 345.9, 780.3; ICD10: G40, P90, R56] | |||||
Headache; Anxiety disorder [ICD9:339, 784.0, 300, 311; ICD10: G43-G44, R51, F32, F40-F42] | |||||
Inflammation [ICD10: E08-E13, E10.2, E11, E11.2, E13.2, I73.9, I80-I82, N00-N29, G89] | |||||
Insomnia [ICD9: 307.41, 307.42, 327.0, 780.51, 780.52; ICD10: F51.0, G47.0] | |||||
Insomnia; Anxiety disorder [ICD9:307.41, 307.42, 327.0, 780.51, 780.52, 300, 311; ICD10: F51.0, G47.0, F32, F40-F42] | |||||
Intractable insomnia [ICD10: G47] | |||||
Intractable chronic pain; Cystitis [ICD9:338, 780; ICD10: R52, G89, N30] | |||||
Insomnia; Epilepsy [ICD9:307.41, 307.42, 327.0, 780.51, 780.52; ICD10: F51.0, G47.0, G40] | |||||
Muscle spasm [ICD10: M62.838] | |||||
Premenstrual syndrome [ICD10: N94.3] | |||||
Respiratory distress syndrome [ICD9: 518.5, 518.82; ICD10: J80] | |||||
Sleep maintenance insomnia [ICD9: 307.41, 307.42, 327.0, 780.51, 780.52; ICD10: F51.0, G47.0] | |||||
Function |
Component of the heteropentameric receptor for GABA, the major inhibitory neurotransmitter in the vertebrate brain. Functions also as histamine receptor and mediates cellular responses to histamine. Functions as receptor for diazepines and various anesthetics, such as pentobarbital; these are bound at a separate allosteric effector binding site. Functions as ligand- gated chloride channel (By similarity).
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BioChemical Class |
Ligand-gated ion channel
|
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Target Validation |
T51487
|
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UniProt ID | |||||
Sequence |
MRKSPGLSDCLWAWILLLSTLTGRSYGQPSLQDELKDNTTVFTRILDRLLDGYDNRLRPG
LGERVTEVKTDIFVTSFGPVSDHDMEYTIDVFFRQSWKDERLKFKGPMTVLRLNNLMASK IWTPDTFFHNGKKSVAHNMTMPNKLLRITEDGTLLYTMRLTVRAECPMHLEDFPMDAHAC PLKFGSYAYTRAEVVYEWTREPARSVVVAEDGSRLNQYDLLGQTVDSGIVQSSTGEYVVM TTHFHLKRKIGYFVIQTYLPCIMTVILSQVSFWLNRESVPARTVFGVTTVLTMTTLSISA RNSLPKVAYATAMDWFIAVCYAFVFSALIEFATVNYFTKRGYAWDGKSVVPEKPKKVKDP LIKKNNTYAPTATSYTPNLARGDPGLATIAKSATIEPKEVKPETKPPEPKKTFNSVSKID RLSRIAFPLLFGIFNLVYWATYLNREPQLKAPTPHQ |
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Drugs and Mode of Action | |||||
Drug(s) | Amobarbital | Drug Info | Approved | Insomnia; Anxiety disorder | [550722], [551871] |
Barbital | Drug Info | Approved | Insomnia | [536555] | |
Barbituric acid | Drug Info | Approved | Depression | [536555] | |
Butabarbital | Drug Info | Approved | Insomnia | [538357], [542144] | |
Butalbital | Drug Info | Approved | Headache; Anxiety disorder | [538316], [542145], [551871] | |
Butethal | Drug Info | Approved | Insomnia | [550763] | |
Clobazam | Drug Info | Approved | Epilepsy; Anxiety disorder | [542156], [550702] | |
Ethanol | Drug Info | Approved | Intractable chronic pain; Cystitis | [537292], [539450], [551871] | |
Ethchlorvynol | Drug Info | Approved | Insomnia | [538355], [542191] | |
Hexobarbital | Drug Info | Approved | Anesthesia | [550698] | |
Meprobamate | Drug Info | Approved | Anxiety disorder | [538193], [542240] | |
Methohexital | Drug Info | Approved | Anesthesia | [538449], [542249] | |
Methoxyflurane | Drug Info | Approved | Anesthesia | [542250], [550732] | |
Methylphenobarbital | Drug Info | Approved | Anxiety disorder | [550692] | |
Methyprylon | Drug Info | Approved | Insomnia | [536255], [542254] | |
Nitrazepam | Drug Info | Approved | Insomnia; Epilepsy | [550758], [551871] | |
Pentobarbital | Drug Info | Approved | Insomnia; Anxiety disorder | [538348], [540880], [551871] | |
Picrotoxin | Drug Info | Approved | Respiratory distress syndrome | [540650], [550699] | |
Primidone | Drug Info | Approved | Epilepsy | [538190], [540777] | |
Secobarbital | Drug Info | Approved | Intractable insomnia | [551871] | |
THIOCOLCHICOSIDE | Drug Info | Approved | Muscle spasm | [551871] | |
Zaleplon | Drug Info | Approved | Insomnia | [467682], [538325] | |
Zolpidem | Drug Info | Approved | Insomnia | [467685], [551871] | |
ZK-93423 | Drug Info | Phase 3 | Epileptic seizures | [467683], [533661] | |
ALLOPREGNANOLONE | Drug Info | Phase 2 | Discovery agent | [467451], [524035] | |
Zolpidem | Drug Info | Phase 1 | Sleep maintenance insomnia | [531325] | |
ELTANOLONE | Drug Info | Discontinued in Phase 3 | Premenstrual syndrome | [546011] | |
U-78875 | Drug Info | Discontinued in Phase 1 | Anxiety disorder | [544810] | |
CGS-9896 | Drug Info | Terminated | Discovery agent | [544687] | |
Divaplon | Drug Info | Terminated | Discovery agent | [544692] | |
Inhibitor | (2-Amino-4,5-dihydro-thiazol-4-yl)-acetic acid | Drug Info | [551228] | ||
(2E,4S)-4-ammoniopent-2-enoate | Drug Info | [533514] | |||
(4R)-4-ammoniopentanoate | Drug Info | [533514] | |||
(4S)-4-ammoniopentanoate | Drug Info | [533514] | |||
(6-Benzylamino-9H-beta-carbolin-3-yl)-methanol | Drug Info | [533414] | |||
(9-Benzyl-9H-purin-6-yl)-cyclopropyl-amine | Drug Info | [533033] | |||
(9H-beta-Carbolin-3-yl)-carbamic acid ethyl ester | Drug Info | [533400] | |||
(9H-beta-Carbolin-3-yl)-ethyl-amine | Drug Info | [533400] | |||
(9H-beta-Carbolin-3-yl)-methanol | Drug Info | [533414] | |||
(beta-CCE)9H-beta-Carboline-3-carboxylic acid | Drug Info | [526738] | |||
1,1-Dimethyl-5-oxa-spiro[2.4]heptan-4-one | Drug Info | [533975] | |||
1,3-Diphenyl-1H-chromeno[4,3-c]pyrazol-4-one | Drug Info | [533354] | |||
1-(4-chlorophenyl)-4-phenyl-1H-imidazole | Drug Info | [528080] | |||
1-(9H-beta-Carbolin-3-yl)-butan-1-one | Drug Info | [526755] | |||
1-(9H-beta-Carbolin-3-yl)-ethanone | Drug Info | [533414] | |||
1-Methyl-5-oxa-spiro[2.4]heptan-4-one | Drug Info | [533975] | |||
2-(1H-Indol-3-yl)-2-oxo-N-phenethyl-acetamide | Drug Info | [526738] | |||
2-(3-Bromo-phenyl)-6-nitro-chromen-4-one | Drug Info | [551323] | |||
2-(3-Bromo-phenyl)-chromen-4-one | Drug Info | [551323] | |||
2-(3-Chloro-phenyl)-chromen-4-one | Drug Info | [551323] | |||
2-(4-Chloro-phenyl)-3H-imidazo[4,5-c]quinoline | Drug Info | [534155] | |||
2-(4-chlorophenyl)-5-phenyl-4-isoxazolin-3-one | Drug Info | [528080] | |||
2-(9-Benzyl-9H-purin-6-ylamino)-ethanol | Drug Info | [533033] | |||
2-Furan-2-yl-6H-pyrazolo[1,5-c]quinazolin-5-one | Drug Info | [534157] | |||
2-Isoxazol-3-yl-3H-imidazo[4,5-c]quinoline | Drug Info | [534155] | |||
2-Isoxazol-5-yl-3H-imidazo[4,5-c]quinoline | Drug Info | [534155] | |||
2-Oxa-spiro[4.4]nonan-1-one | Drug Info | [533975] | |||
2-p-Tolyl-6H-pyrazolo[1,5-c]quinazolin-5-one | Drug Info | [534157] | |||
2-Phenyl-3H-imidazo[4,5-c]quinoline | Drug Info | [534155] | |||
2-Phenyl-5,6-dihydro-pyrazolo[1,5-c]quinazoline | Drug Info | [534157] | |||
2-Phenyl-6H-pyrazolo[1,5-c]quinazolin-5-one | Drug Info | [534157] | |||
2-Pyridin-2-yl-6H-pyrazolo[1,5-c]quinazolin-5-one | Drug Info | [534157] | |||
2-Thiophen-2-yl-3H-imidazo[4,5-c]quinoline | Drug Info | [534155] | |||
3,3-Diethyl-dihydro-furan-2-one | Drug Info | [533975] | |||
3,3-Diisopropyl-dihydro-furan-2-one | Drug Info | [533975] | |||
3-(2,2-Dimethyl-propoxy)-9H-beta-carboline | Drug Info | [526755] | |||
3-(3-Methyl-butoxy)-9H-beta-carboline | Drug Info | [526755] | |||
3-(benzyloxy)-9H-pyrido[3,4-b]indole | Drug Info | [531188] | |||
3-(hexa-1,3-dienyloxy)-9H-pyrido[3,4-b]indole | Drug Info | [531188] | |||
3-(isopentyloxy)-9H-pyrido[3,4-b]indole | Drug Info | [531188] | |||
3-amino-3-demethoxythiocolchicine | Drug Info | [528408] | |||
3-Butoxy-9H-beta-carboline | Drug Info | [526755] | |||
3-butoxy-9H-pyrido[3,4-b]indole | Drug Info | [531188] | |||
3-butoxycarbonyl-4-quinolone | Drug Info | [528134] | |||
3-butoxycarbonyl-6-ethyl-4-quinolone | Drug Info | [528134] | |||
3-butylaminocarbonyl-6-ethyl-4-quinolone | Drug Info | [528134] | |||
3-carboxy-6-ethyl-4-quinolone | Drug Info | [528134] | |||
3-Chloro-9H-beta-carboline | Drug Info | [533363] | |||
3-cyclopentoxycarbonyl-6-ethyl-4-quinolone | Drug Info | [528134] | |||
3-demethoxy-3-D-lyxopyranosylaminothiocolchicine | Drug Info | [528408] | |||
3-demethoxy-3-D-mannopyranosylaminothiocolchicine | Drug Info | [528408] | |||
3-demethoxy-3-D-xylopyranosylaminothiocolchicine | Drug Info | [528408] | |||
3-demethoxy-3-L-fucopyranosylaminothiocolchicine | Drug Info | [528408] | |||
3-demethoxy-3D-glucopyranosylaminothiocolchicine | Drug Info | [528408] | |||
3-Ethoxy-9H-beta-carboline | Drug Info | [533363] | |||
3-ethoxy-9H-pyrido[3,4-b]indole | Drug Info | [531188] | |||
3-ethoxycarbonyl-4-quinolone | Drug Info | [528134] | |||
3-ethoxycarbonyl-6-ethyl-2-methyl-4-quinolone | Drug Info | [528134] | |||
3-ethoxycarbonyl-6-propyl-4-quinolone | Drug Info | [528134] | |||
3-Ethyl-3-isopropyl-dihydro-furan-2-one | Drug Info | [533975] | |||
3-Ethyl-3-methyl-dihydro-furan-2-one | Drug Info | [533975] | |||
3-Isobutoxy-9H-beta-carboline | Drug Info | [526755] | |||
3-isobutoxy-9H-pyrido[3,4-b]indole | Drug Info | [531188] | |||
3-Isopropoxy-9H-beta-carboline | Drug Info | [526755] | |||
3-Isopropyl-3-methyl-dihydro-furan-2-one | Drug Info | [533975] | |||
3-Isothiocyanato-9H-beta-carboline | Drug Info | [531518] | |||
3-Methoxy-9H-beta-carboline | Drug Info | [533363] | |||
3-Methoxycarbonyl-2-methyl-9H-beta-carbolin-2-ium | Drug Info | [551248] | |||
3-Methyl-1-phenyl-1H-chromeno[4,3-c]pyrazol-4-one | Drug Info | [533354] | |||
3-Methyl-2-phenyl-2H-chromeno[4,3-c]pyrazol-4-one | Drug Info | [533354] | |||
3-Methyl-9H-beta-carboline | Drug Info | [533745] | |||
3-Nitro-9H-beta-carboline | Drug Info | [533363] | |||
3-Propoxy-9H-beta-carboline | Drug Info | [533363] | |||
3-propoxy-9H-pyrido[3,4-b]indole | Drug Info | [531188] | |||
3-sec-Butoxy-9H-beta-carboline | Drug Info | [526755] | |||
3-tert-Butyl-3-ethyl-dihydro-furan-2-one | Drug Info | [533975] | |||
4-(2-aminoethyl)-1,2,5-oxadiazol-3-ol | Drug Info | [528295] | |||
4-(4-chlorophenyl)-1-pyrid-2-yl-pyrazole | Drug Info | [528080] | |||
4-(biphenyl-3-yl)-5-(piperidin-4-yl)isoxazol-3-ol | Drug Info | [530818] | |||
4-benzyl-5-(4-piperidyl)isothiazol-3-ol | Drug Info | [528034] | |||
4-Benzyl-5-piperidin-4-yl-isoxazol-3-ol | Drug Info | [527382] | |||
4-Methoxymethyl-3,6-dipropoxy-9H-beta-carboline | Drug Info | [534660] | |||
4-Methyl-5-(4-piperidyl)isothiazol-3-ol | Drug Info | [528034] | |||
4-Naphthalen-1-yl-5-piperidin-4-yl-isoxazol-3-ol | Drug Info | [527382] | |||
4-Naphthalen-2-yl-5-piperidin-4-yl-isoxazol-3-ol | Drug Info | [527382] | |||
4-Phenyl-5-piperidin-4-yl-isoxazol-3-ol | Drug Info | [527382] | |||
5-(4-piperidyl)-4-propylisothiazol-3-ol | Drug Info | [528034] | |||
5-(piperidin-4-yl)isothiazol-3-ol | Drug Info | [528034] | |||
5-(piperidin-4-yl)isoxazol-3-ol | Drug Info | [527382] | |||
5-[(1R)-1-ammonioethyl]isoxazol-3-olate | Drug Info | [533514] | |||
5-[(1S)-1-ammonioethyl]isoxazol-3-olate | Drug Info | [533514] | |||
6,6-Dimethyl-2-oxa-spiro[4.4]nonan-1-one | Drug Info | [533975] | |||
6,9-Dimethyl-2-oxa-spiro[4.4]nonan-1-one | Drug Info | [533975] | |||
6-benzyl-3-ethoxycarbonyl-4-quinolone | Drug Info | [528134] | |||
6-benzyl-3-propoxycarbonyl-4-quinolone | Drug Info | [528134] | |||
6-benzyl-3-propylaminocarbonyl-4-quinolone | Drug Info | [528134] | |||
6-Bromo-2-(2-nitro-phenyl)-chromen-4-one | Drug Info | [551336] | |||
6-Bromo-2-(3-bromo-phenyl)-chromen-4-one | Drug Info | [551323] | |||
6-Bromo-2-(3-nitro-phenyl)-chromen-4-one | Drug Info | [551336] | |||
6-Bromo-2-(4-nitro-phenyl)-chromen-4-one | Drug Info | [551336] | |||
6-Bromo-2-phenyl-chromen-4-one | Drug Info | [551323] | |||
6-bromo-3-ethoxycarbonyl-2-methyl-4-quinolone | Drug Info | [528134] | |||
6-bromo-3-ethoxycarbonyl-4-quinolone | Drug Info | [528134] | |||
6-Chloro-2-(3-nitro-phenyl)-chromen-4-one | Drug Info | [551323] | |||
6-Chloro-2-phenyl-chromen-4-one | Drug Info | [551323] | |||
6-ethyl-3-(2-ethylbutoxycarbonyl)-4-quinolone | Drug Info | [528134] | |||
6-ethyl-3-(2-methylbutoxycarbonyl)-4-quinolone | Drug Info | [528134] | |||
6-ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone | Drug Info | [528134] | |||
6-ethyl-3-(3-pentoxycarbonyl)-4-quinolone | Drug Info | [528134] | |||
6-ethyl-3-i-propoxycarbonyl-4-quinolone | Drug Info | [528134] | |||
6-ethyl-3-pentoxycarbonyl-4-quinolone | Drug Info | [528134] | |||
6-ethyl-3-propoxycarbonyl-4-quinolone | Drug Info | [528134] | |||
6-ethyl-3-propylaminocarbonyl-4-quinolone | Drug Info | [528134] | |||
6-Fluoro-2-(3-nitro-phenyl)-chromen-4-one | Drug Info | [551323] | |||
6-Methyl-2-oxa-spiro[4.4]nonan-1-one | Drug Info | [533975] | |||
6-Nitro-2-(3-nitro-phenyl)-chromen-4-one | Drug Info | [551290] | |||
6-Nitro-2-(4-nitro-phenyl)-chromen-4-one | Drug Info | [551290] | |||
6-Nitro-2-phenyl-chromen-4-one | Drug Info | [551323] | |||
7,12-Dihydro-5,7,12-triaza-indeno[1,2-a]fluorene | Drug Info | [533412] | |||
7,12-Dihydro-7,12-diaza-indeno[1,2-a]fluorene | Drug Info | [533363] | |||
9H-beta-Carbolin-3-ol | Drug Info | [533363] | |||
9H-beta-Carbolin-6-ylamine | Drug Info | [533414] | |||
9H-beta-Carboline-3-carboxylic acid butyl ester | Drug Info | [533546] | |||
9H-beta-Carboline-3-carboxylic acid ethyl ester | Drug Info | [533546] | |||
9H-beta-Carboline-3-carboxylic acid propyl ester | Drug Info | [533546] | |||
ALLOPREGNANOLONE | Drug Info | [527511] | |||
AMENTOFLAVONE | Drug Info | [526653] | |||
Barbituric acid derivative | Drug Info | [551407] | |||
Benzyl-(9H-beta-carbolin-6-yl)-amine | Drug Info | [533363] | |||
Beta-Carboline-3-carboxylic acid t-butyl ester | Drug Info | [531188] | |||
BETA-CCM | Drug Info | [533763] | |||
CGP-27492 | Drug Info | [533678] | |||
CGS-13767 | Drug Info | [529466] | |||
CGS-8216 | Drug Info | [529466] | |||
CGS-9895 | Drug Info | [533348] | |||
CGS-9896 | Drug Info | [528080] | |||
CI-218872 | Drug Info | [533745] | |||
Divaplon | Drug Info | [533379] | |||
ELTANOLONE | Drug Info | [527511] | |||
Ethyl 6-iodo-9H-pyrido[3,4-b]indole-3-carboxylate | Drug Info | [531188] | |||
Ethyl 9H-pyrido[3,4-b]indole-3-carboxylate | Drug Info | [531188] | |||
GABAZINE | Drug Info | [528034] | |||
GAMMA-AMINO-BUTANOIC ACID | Drug Info | [528408] | |||
GNF-PF-3645 | Drug Info | [528134] | |||
GNF-PF-4421 | Drug Info | [528134] | |||
Isoquinoline-3-carboxylic acid methyl ester | Drug Info | [533363] | |||
L-655708 | Drug Info | [527005] | |||
N-(9H-beta-Carbolin-3-yl)-acetamide | Drug Info | [533400] | |||
N-(9H-beta-Carbolin-3-yl)-formamide | Drug Info | [533400] | |||
N-(p-methylbenzyl)-5-nitroindol-3-ylglyoxylamide | Drug Info | [528709] | |||
N-Benzyl-2-(1H-indol-3-yl)-2-oxo-acetamide | Drug Info | [528709] | |||
N-benzyl-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide | Drug Info | [528709] | |||
N-butyl-2-(1H-indol-3-yl)-2-oxoacetamide | Drug Info | [528709] | |||
N-butyl-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide | Drug Info | [528709] | |||
N-Indan-1-yl-2-(1H-indol-3-yl)-2-oxo-acetamide | Drug Info | [526094] | |||
NORHARMANE | Drug Info | [533363] | |||
NSC-19028 | Drug Info | [551323] | |||
NSC-73613 | Drug Info | [551323] | |||
NSC-93394 | Drug Info | [551323] | |||
Pyrrolidin-3-yl-acetic acid | Drug Info | [533396] | |||
Ridine-5-carboxylic acid ethyl ester | Drug Info | [533164] | |||
RIPAZEPAM | Drug Info | [533397] | |||
RO-054520 | Drug Info | [533368] | |||
RO-145974 | Drug Info | [534008] | |||
RO-145975 | Drug Info | [534008] | |||
RO-147437 | Drug Info | [534008] | |||
Ro-151310 | Drug Info | [534008] | |||
Ro-154513 | Drug Info | [534008] | |||
RO-194603 | Drug Info | [534008] | |||
Ro-4938581 | Drug Info | [530391] | |||
RWJ-16979 | Drug Info | [533762] | |||
RY-066 | Drug Info | [534718] | |||
Sec-butyl 9H-pyrido[3,4-b]indole-3-carboxylate | Drug Info | [531188] | |||
THIOCOLCHICOSIDE | Drug Info | [528408] | |||
U-78875 | Drug Info | [525465] | |||
U-89267 | Drug Info | [533912] | |||
ZK-93423 | Drug Info | [530319] | |||
Antagonist | Amobarbital | Drug Info | [536555], [537688] | ||
Barbital | Drug Info | [536555], [537688] | |||
Barbituric acid | Drug Info | [536555], [537688] | |||
Butabarbital | Drug Info | [535022], [536555], [537688] | |||
Butalbital | Drug Info | [536555] | |||
Butethal | Drug Info | [536555] | |||
Clobazam | Drug Info | [536555] | |||
Ethanol | Drug Info | [536555] | |||
Ethchlorvynol | Drug Info | [536555] | |||
Hexobarbital | Drug Info | [536555], [537688] | |||
Meprobamate | Drug Info | [536555] | |||
Methohexital | Drug Info | [536555] | |||
Methoxyflurane | Drug Info | [536555] | |||
Methylphenobarbital | Drug Info | [536555], [537688] | |||
Methyprylon | Drug Info | [536555] | |||
Nitrazepam | Drug Info | [536555] | |||
Pentobarbital | Drug Info | [536555], [537688] | |||
Picrotoxin | Drug Info | [536555] | |||
Primidone | Drug Info | [536555] | |||
Secobarbital | Drug Info | [536555], [537688] | |||
Modulator | Zaleplon | Drug Info | [556264] | ||
Zolpidem | Drug Info | ||||
Target Expression Profile (TEP) and Drug Resistance Mutation (DRM) | |||||
TEP | EXP Info | ||||
Pathways | |||||
KEGG Pathway | Neuroactive ligand-receptor interaction | ||||
Retrograde endocannabinoid signaling | |||||
GABAergic synapse | |||||
Morphine addiction | |||||
Nicotine addiction | |||||
Reactome | Ligand-gated ion channel transport | ||||
GABA A receptor activation | |||||
WikiPathways | SIDS Susceptibility Pathways | ||||
Neurotransmitter Receptor Binding And Downstream Transmission In The Postsynaptic Cell | |||||
Iron uptake and transport | |||||
References | |||||
Ref 467451 | (http://www.guidetopharmacology.org/) Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 4108). | ||||
Ref 467682 | (http://www.guidetopharmacology.org/) Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 4345). | ||||
Ref 467683 | (http://www.guidetopharmacology.org/) Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 4346). | ||||
Ref 467685 | (http://www.guidetopharmacology.org/) Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 4348). | ||||
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